Brief Information of the Cell Line and Protein
Cell Line ID: CL000079 , Expi293F
Category Transformed cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_D615
Protein ID: PT01279 , Adenosine receptor A3
Gene Name ADORA3
Organism Homo sapiens, Human
Protein Classification Membrane receptor
Uniprot ID P0DMS8
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000079  Protein ID: PT01279
 
Compound ID Compound Name Compound Formula
CP0001102
(2R,3R,4S,5R)-2-(6-amino-9H-purin-9-yl)-5-(hydroxymethyl)oxolane-3,4-diol
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C10H13N5O4
 2
1
Kd = 740 nM
   TI
   LI
   LO
   TS
2
Ki = 290 nM
   TI
   LI
   LO
   TS
CP0019682
2-(4-fluorophenyl)-3-(4-pyridinyl)pyrazolo-[1,5-a]pyridine
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C18H12FN3
 1
1
Kd = 740 nM
   TI
   LI
   LO
   TS
CP0547170
N-(3-chlorophenyl)-4-methylsulfonylbenzamide
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C14H12ClNO3S
 1
1
Kd = 18000 nM
   TI
   LI
   LO
   TS
CP0546740
3-methyl-1H-quinazoline-2,4-dione
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C9H8N2O2
 1
1
Kd = 18900 nM
   TI
   LI
   LO
   TS
CP0546737
5-(4-chlorophenyl)-1,2,4-thiadiazol-3-amine
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C8H6ClN3S
 1
1
Kd = 36500 nM
   TI
   LI
   LO
   TS
CP0547178
3-phenyl-1,2,4-thiadiazol-5-amine
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C8H7N3S
 1
1
Kd = 50700 nM
   TI
   LI
   LO
   TS
CP0546741
1-phenyl-3-pyridin-2-ylurea
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C12H11N3O
 1
1
Kd = 52000 nM
   TI
   LI
   LO
   TS
CP0562631
N-quinolin-2-ylfuran-2-carboxamide
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C14H10N2O2
 1
1
Kd = 56000 nM
   TI
   LI
   LO
   TS
CP0568019
3-phenyl-N-propan-2-yl-1H-pyrazole-5-carboxamide
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C13H15N3O
 1
1
Kd = 80000 nM
   TI
   LI
   LO
   TS
CP0543588
US8993552, 1F4 Compound 44
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C10H10N4O
 1
1
Kd = 101000 nM
   TI
   LI
   LO
   TS
CP0568020
BENZOGUANAMINE
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C9H9N5
 1
1
Kd = 104200 nM
   TI
   LI
   LO
   TS
CP0546728
3-phenyl-[1,2,4]triazolo[4,3-b]pyridazin-6-amine
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C11H9N5
 1
1
Kd = 160000 nM
   TI
   LI
   LO
   TS
CP0492321
2-(benzylamino)pyrido[1,2-a]pyrimidin-4-one
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C15H13N3O
 1
1
Kd = 200000 nM
   TI
   LI
   LO
   TS