General Information of the Compound
Compound ID
CP0104425
Compound Name
2,2,4-Trimethyl-5-[1-o-tolyl-meth-(Z)-ylidene]-2,5-dihydro-1H-6-oxa-1-aza-chrysene
    Show/Hide
Synonyms
5-(2-Methylbenzylidene)-2,2,4-trimethyl-1,2-dihydro-5H-1-aza-6-oxachrysene
BDBM50067684
CHEMBL302362
LG-120838
SCHEMBL4175160
SCHEMBL4175162
    Show/Hide
Structure
Formula
C27H25NO
Molecular Weight
379.503
Canonical SMILES
CC1=CC(C)(C)Nc2ccc3-c4ccccc4O\C(=C/c4ccccc4C)c3c12
    Show/Hide
InChI
InChI=1S/C27H25NO/c1-17-9-5-6-10-19(17)15-24-26-21(20-11-7-8-12-23(20)29-24)13-14-22-25(26)18(2)16-27(3,4)28-22/h5-16,28H,1-4H3/b24-15-
    Show/Hide
InChIKey
YXKBVHXOKVRRKO-IWIPYMOSSA-N
Physicochemical Property
logP
7.15992
Rotatable Bonds
1
Heavy Atom Count
29
Polar Areas
21.26
Hydrogen Bond Donor Count
1
Hydrogen Bond Acceptor Count
2
Complexity
29

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

    Show/Hide
Click to Show/Hide the External Link(s) of This Compound
PubChem ID
CID: 9951771
SID: 14927037
ChEMBL ID
CHEMBL302362
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT00894, Androgen receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000044 CV-1 Chlorocebus aethiops (Green monkey)  1
1
IC50 = 1062 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 Ki = 844 nM
Protein ID: PT00967, Glucocorticoid receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000044 CV-1 Chlorocebus aethiops (Green monkey)  1
1
IC50 = 1050 nM
   TI
   LI
   LO
   TS
CL000778 SF-12 Spodoptera frugiperda (Fall armyworm)  1
1
Ki = 564 nM
   TI
   LI
   LO
   TS
Protein ID: PT01154, Mineralocorticoid receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000044 CV-1 Chlorocebus aethiops (Green monkey)  1
1
IC50 < 20 nM
   TI
   LI
   LO
   TS
Protein ID: PT01172, Progesterone receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000044 CV-1 Chlorocebus aethiops (Green monkey)  1
1
EC50 = 5.7 nM
   TI
   LI
   LO
   TS
CL000078 T-47D Homo sapiens (Human)  1
1
EC50 = 28 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 Ki = 0.66 nM
Clinical Information about the Compound
Drug 1 ( LG-120838 )
Drug Name LG-120838
Target(s)
Mineralocorticoid receptor (MR)
Inhibitor
Androgen receptor messenger RNA (AR mRNA)
Inhibitor
Glucocorticoid receptor messenger RNA (GCR mRNA)
Inhibitor