| Compound ID |
Compound Name |
Compound Formula |
|
CP0108032
|
(S)-2-(2-Benzoyl-phenylamino)-3-{4-[2-(5-methyl-2-phenyl-oxazol-4-yl)-ethoxy]-phenyl}-propionic acid
Show/Hide
|
C34H30N2O5
|
2
|
| 1 |
EC50 = 0.3388 nM
|
|
|
| 2 |
EC50 = 0.34 nM
|
|
|
|
CP0468295
|
4-Isocyanato-benzoic acid 2-((2,4-bis-trifluoromethyl-benzyl)-{3-[3-(1-carboxy-1-methyl-ethoxy)-phenyl]-propyl}-amino)-ethyl ester
Show/Hide
|
C32H30F6N2O6
|
1
|
| 1 |
EC50 = 0.5 nM
|
|
|
|
CP0088667
|
2-((S)-1-carboxy-2-{4-[2-(5-methyl-2-phenyl-oxazol-4-yl)-ethoxy]-phenyl}-ethylamino)-benzoic acid methyl ester
Show/Hide
|
C29H28N2O6
|
3
|
| 1 |
EC50 = 0.631 nM
|
|
|
| 2 |
EC50 = 0.71 nM
|
|
|
| 3 |
IC50 < 10000 nM
|
|
|
|
CP0429811
|
4'-((2,3-dimethyl-5-(1-phenylpropylcarbamoyl)-1H-indol-1-yl)methyl)biphenyl-2-carboxylic acid
Show/Hide
|
C34H32N2O3
|
1
|
| 1 |
EC50 = 0.8 nM
|
|
|
|
CP0449515
|
(S)-3-{4-[2-(2-Cyclohexyl-5-methyl-oxazol-4-yl)-ethoxy]-phenyl}-2-methyl-2-phenoxy-propionic acid
Show/Hide
|
C28H33NO5
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0492739
|
4'-((2-methyl-3-(methylthio)-5-(1-phenylpropylcarbamoyl)-1H-indol-1-yl)methyl)biphenyl-2-carboxylic acid
Show/Hide
|
C34H32N2O3S
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0406324
|
3-(4-(2-(5-(3-fluorophenyl)-1,2,4-oxadiazol-3-yl)ethoxy)phenyl)-2-isopropoxypropanoic acid
Show/Hide
|
C22H23FN2O5
|
1
|
| 1 |
EC50 = 2 nM
|
|
|
|
CP0051825
|
3-(2-((isopropoxycarbonyl)methyl)-4-(2-(5-methyl-2-(4-phenoxyphenyl)oxazol-4-yl)ethoxy)phenyl)propanoic acid
Show/Hide
|
C32H34N2O7
|
1
|
| 1 |
EC50 = 2 nM
|
|
|
|
CP0132962
|
3-{4-[2-(2-biphenyl-4-yl-5-methyl-oxazol-4-yl)-ethoxy]-2-[(pyrazin-2-yloxycarbonylamino)-methyl]-phenyl}-propionic acid
Show/Hide
|
C33H30N4O6
|
1
|
| 1 |
EC50 = 2 nM
|
|
|
|
CP0447684
|
4'-((5-(2-phenylbutanamido)-2-propyl-1H-indol-1-yl)methyl)biphenyl-2-carboxylic acid
Show/Hide
|
C35H34N2O3
|
1
|
| 1 |
EC50 = 2 nM
|
|
|
|
CP0439850
|
2-[4-[[1-methyl-6-(1-phenylpropylcarbamoyl)-2-propylindol-3-yl]methyl]phenyl]benzoic acid
Show/Hide
|
C36H36N2O3
|
1
|
| 1 |
EC50 = 2 nM
|
|
|
|
CP0309669
|
(2S)-3-[4-[2-[1,3-benzoxazol-2-yl(methyl)amino]ethoxy]phenyl]-2-(2-benzoylanilino)propanoic acid
Show/Hide
|
C32H29N3O5
|
1
|
| 1 |
EC50 = 2.63 nM
|
|
|
|
CP0401328
|
3-(4-((5-(4-tert-butylphenyl)-1,2,4-oxadiazol-3-yl)methoxy)phenyl)-2-isopropoxypropanoic acid
Show/Hide
|
C25H30N2O5
|
1
|
| 1 |
EC50 = 3 nM
|
|
|
|
CP0152177
|
(S)-2-Methyl-3-{4-[2-(5-methyl-2-phenyl-oxazol-4-yl)-ethoxy]-phenyl}-2-phenoxy-propionic acid
Show/Hide
|
C28H27NO5
|
1
|
| 1 |
EC50 = 3 nM
|
|
|
|
CP0452274
|
4'-((3-(methylthio)-5-(2-phenylbutanamido)-2-propyl-1H-indol-1-yl)methyl)biphenyl-2-carboxylic acid
Show/Hide
|
C36H36N2O3S
|
1
|
| 1 |
EC50 = 3 nM
|
|
|
|
CP0675045
|
5-{4-[2-(5-Methyl-2-phenyl-oxazol-4-yl)-ethoxy]-benzyl}-thiazolidine-2,4-dione
Show/Hide
|
C22H20N2O4S
|
1
|
| 1 |
EC50 = 3.162 nM
|
|
|
|
CP0380581
|
(S)-2-Benzyl-3-(3-(((4-adamantan-1-yl)benzamido)-methyl)-4-propoxyphenyl)propanoic Acid
Show/Hide
|
C37H43NO4
|
1
|
| 1 |
EC50 = 3.6 nM
|
|
|
|
CP0377839
|
2-[3-(3-{(2,4-Bis-trifluoromethyl-benzyl)-[2-(4-trifluoromethyl-phenyl)-acetyl]-amino}-propyl)-phenoxy]-2-methyl-propionic acid
Show/Hide
|
C31H28F9NO4
|
1
|
| 1 |
EC50 = 4 nM
|
|
|
|
CP0114157
|
2-Isopropoxy-3-{4-[5-(4-isopropyl-phenyl)-[1,2,4]oxadiazol-3-ylmethoxy]-phenyl}-propionic acid
Show/Hide
|
C24H28N2O5
|
1
|
| 1 |
EC50 = 4 nM
|
|
|
|
CP0204433
|
3-(4-(2-(5-(3-chlorophenyl)-1,2,4-oxadiazol-3-yl)ethoxy)phenyl)-2-isopropoxypropanoic acid
Show/Hide
|
C22H23ClN2O5
|
1
|
| 1 |
EC50 = 4 nM
|
|
|
|
CP0051318
|
(R)-3-(4-(3-(2-benzoyl-4-ethylphenoxy)butoxy)-2-methylphenyl)propanoic acid
Show/Hide
|
C29H32O5
|
1
|
| 1 |
EC50 = 4 nM
|
|
|
|
CP0253618
|
3-(2-((isopropoxycarbonyl)methyl)-4-(2-(5-methyl-2-(4-(pyrimidin-2-yl)phenyl)oxazol-4-yl)ethoxy)phenyl)propanoic acid
Show/Hide
|
C30H32N4O6
|
1
|
| 1 |
EC50 = 4 nM
|
|
|
|
CP0259062
|
(S)-2-Methyl-3-{4-[2-(5-methyl-2-thiophen-2-yl-oxazol-4-yl)-ethoxy]-phenyl}-2-phenoxy-propionic acid
Show/Hide
|
C26H25NO5S
|
1
|
| 1 |
EC50 = 4 nM
|
|
|
|
CP0057743
|
(R)-3-{2-methyl-4-[3-(2-phenoxy-4-trifluoromethyl-phenoxy)-butoxy]-phenyl}-propionic acid
Show/Hide
|
C27H27F3O5
|
1
|
| 1 |
EC50 = 4 nM
|
|
|
|
CP0071093
|
3-(4-(2-(5-(3,5-bis(trifluoromethyl)phenyl)-1,2,4-oxadiazol-3-yl)ethoxy)phenyl)-2-isopropoxypropanoic acid
Show/Hide
|
C24H22F6N2O5
|
1
|
| 1 |
EC50 = 4 nM
|
|
|
|
CP0082065
|
(R)-3-{2-methyl-4-[3-(2-phenoxy-4-trifluoromethoxy-phenoxy)-butoxy]-phenyl}-propionic acid
Show/Hide
|
C27H27F3O6
|
1
|
| 1 |
EC50 = 5 nM
|
|
|
|
CP0311276
|
3-[4-[2-[1,3-benzoxazol-2-yl(methyl)amino]ethoxy]phenyl]-2-[(9,10-dioxoanthracen-1-yl)amino]propanoic acid
Show/Hide
|
C33H27N3O6
|
1
|
| 1 |
EC50 = 5.012 nM
|
|
|
|
CP0404578
|
2-(4-{2-[1-Cycloheptyl-3-(2,4-difluoro-phenyl)-ureido]-ethyl}-phenoxy)-2-methyl-propionic acid
Show/Hide
|
C26H32F2N2O4
|
1
|
| 1 |
EC50 = 6 nM
|
|
|
|
CP0233674
|
2-Isopropoxy-3-(4-{2-[5-(3-trifluoromethyl-phenyl)-[1,2,4]oxadiazol-3-yl]-ethoxy}-phenyl)-propionic acid
Show/Hide
|
C23H23F3N2O5
|
1
|
| 1 |
EC50 = 6 nM
|
|
|
|
CP0052679
|
3-{4-[2-(2-Biphenyl-3-yl-5-methyl-oxazol-4-yl)-ethoxy]-phenyl}-2-methyl-2-phenoxy-propionic acid
Show/Hide
|
C34H31NO5
|
1
|
| 1 |
EC50 = 6 nM
|
|
|
|
CP0210693
|
2-Methyl-3-{4-[2-(5-methyl-2-thiophen-2-yl-oxazol-4-yl)-ethoxy]-phenyl}-2-phenoxy-propionic acid
Show/Hide
|
C26H25NO5S
|
1
|
| 1 |
EC50 = 6 nM
|
|
|
|
CP0082061
|
2-{4-[3-(2-benzoyl-4-ethyl-phenoxy)-butoxy]-phenoxy}-2-methyl-propionic acid
Show/Hide
|
C29H32O6
|
1
|
| 1 |
EC50 = 6 nM
|
|
|
|
CP0118647
|
(S)-2-(2-Benzoyl-phenylamino)-3-{4-[2-(methyl-pyridin-2-yl-amino)-ethoxy]-phenyl}-propionic acid
Show/Hide
|
C30H29N3O4
|
1
|
| 1 |
EC50 = 6 nM
|
|
|
|
CP0432278
|
2-[4-[[6-(1-phenylpropylcarbamoyl)-2-propyl-1H-indol-3-yl]methyl]phenyl]benzoic acid
Show/Hide
|
C35H34N2O3
|
1
|
| 1 |
EC50 = 6 nM
|
|
|
|
CP0296394
|
3-(4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)-2-(((pyrazin-2-yloxy)carbonyl)methyl)phenyl)propanoic acid
Show/Hide
|
C27H26N4O6
|
1
|
| 1 |
EC50 = 7 nM
|
|
|
|
CP0052677
|
3-{4-[2-(2-Biphenyl-4-yl-5-methyl-oxazol-4-yl)-ethoxy]-phenyl}-2-methyl-2-phenoxy-propionic acid
Show/Hide
|
C34H31NO5
|
1
|
| 1 |
EC50 = 7 nM
|
|
|
|
CP0051709
|
3-(2-((isopropoxycarbonyl)methyl)-4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)phenyl)propanoic acid
Show/Hide
|
C26H30N2O6
|
1
|
| 1 |
EC50 = 8 nM
|
|
|
|
CP0152175
|
2-Methyl-3-{4-[2-(5-methyl-2-phenyl-oxazol-4-yl)-ethoxy]-phenyl}-2-phenoxy-propionic acid
Show/Hide
|
C28H27NO5
|
1
|
| 1 |
EC50 = 8 nM
|
|
|
|
CP0074936
|
(R)-3-{4-[3-(4-ethyl-2-phenoxy-phenoxy)-butoxy]-2-methyl-phenyl}-propionic acid
Show/Hide
|
C28H32O5
|
1
|
| 1 |
EC50 = 8 nM
|
|
|
|
CP0228655
|
3-{4-[2-(2-Cyclohexyl-5-methyl-oxazol-4-yl)-ethoxy]-phenyl}-2-methyl-2-phenoxy-propionic acid
Show/Hide
|
C28H33NO5
|
1
|
| 1 |
EC50 = 9 nM
|
|
|
|
CP0221733
|
3-{4-[3-(2-benzoyl-4-ethyl-phenoxy)-butoxy]-2-methyl-phenyl}-propionic acid
Show/Hide
|
C29H32O5
|
1
|
| 1 |
EC50 = 9 nM
|
|
|
|
CP0097650
|
(2S)-2-(2-benzoylanilino)-3-[4-[(6-hydroxy-2,5,7,8-tetramethyl-3,4-dihydrochromen-2-yl)methoxy]phenyl]propanoic acid
Show/Hide
|
C36H37NO6
|
1
|
| 1 |
EC50 = 9.12 nM
|
|
|
|
CP0035146
|
2-methyl-2-(2-methyl-4-(3-((2-methyl-4-(trifluoromethoxy)benzamido)methyl)phenoxy)phenoxy)propanoic acid
Show/Hide
|
C27H26F3NO6
|
1
|
| 1 |
EC50 = 10 nM
|
|
|
|
CP0378684
|
(S)-3-(3-((E)-1-(3-Chlorobenzyloxyimino)ethyl)phenyl)-2-ethoxypropanoicAcid
Show/Hide
|
C20H22ClNO4
|
1
|
| 1 |
EC50 = 10 nM
|
|
|
|
CP0678274
|
5-{4-[2-(Benzooxazol-2-yl-methyl-amino)-ethoxy]-benzyl}-thiazolidine-2,4-dione
Show/Hide
|
C20H19N3O4S
|
1
|
| 1 |
EC50 = 11.22 nM
|
|
|
|
CP0271168
|
2-Isopropoxy-3-{4-[2-(5-phenyl-[1,2,4]oxadiazol-3-yl)-ethoxy]-phenyl}-propionic acid
Show/Hide
|
C22H24N2O5
|
1
|
| 1 |
EC50 = 13 nM
|
|
|
|
CP0943391
|
N-(2-{4-[(2,4-dioxo-1,3-thiazolidin-5-yl)methyl]phenoxy}ethyl)-5-(1,2-dithiolan-3-yl)-N-methylpentanamide
Show/Hide
|
C21H28N2O4S3
|
1
|
| 1 |
EC50 = 15 nM
|
|
|
|
CP0231600
|
2-Isopropoxy-3-[4-(5-p-tolyl-[1,2,4]oxadiazol-3-ylmethoxy)-phenyl]-propionic acid
Show/Hide
|
C22H24N2O5
|
1
|
| 1 |
EC50 = 16 nM
|
|
|
|
CP0136124
|
2-(4-(3-((2-methoxy-4-(trifluoromethyl)benzamido)methyl)phenoxy)-2-methylphenoxy)-2-methylpropanoic acid
Show/Hide
|
C27H26F3NO6
|
1
|
| 1 |
EC50 = 16 nM
|
|
|
|
CP0320788
|
4'-((2-methyl-5-(1-phenylpropylcarbamoyl)-1H-indol-1-yl)methyl)biphenyl-2-carboxylic acid
Show/Hide
|
C33H30N2O3
|
1
|
| 1 |
EC50 = 17 nM
|
|
|
|
CP0145965
|
3-[4-[2-(2-biphenyl-4-yl-5-methyl-oxazol-4-yl)-ethoxy]-2-(isopropoxycarbonylamino-methyl)-phenyl]-propionic acid
Show/Hide
|
C32H34N2O6
|
1
|
| 1 |
EC50 = 19 nM
|
|
|
|
CP0114160
|
3-(4-((5-(4-chlorophenyl)-1,2,4-oxadiazol-3-yl)methoxy)phenyl)-2-isopropoxypropanoic acid
Show/Hide
|
C21H21ClN2O5
|
1
|
| 1 |
EC50 = 20 nM
|
|
|
|
CP0942098
|
4-({8-[(2-{4-[(2,4-dioxo-1,3-thiazolidin-5-yl)methyl]phenoxy}-ethyl)(methyl)amino]-3-mercapto-8-oxooctyl}thio)-4-oxobutanoic acid sodium salt
Show/Hide
|
C25H33N2NaO7S3
|
1
|
| 1 |
EC50 = 20 nM
|
|
|
|
CP0296984
|
2-(4-(3-fluoro-5-((2-fluoro-4-(trifluoromethyl)benzamido)methyl)phenoxy)-2-methylphenoxy)-2-methylpropanoic acid
Show/Hide
|
C26H22F5NO5
|
1
|
| 1 |
EC50 = 22 nM
|
|
|
|
CP0371730
|
4'-((2,3-dimethyl-5-(3-phenylpropylcarbamoyl)-1H-indol-1-yl)methyl)biphenyl-2-carboxylic acid
Show/Hide
|
C34H32N2O3
|
1
|
| 1 |
EC50 = 22 nM
|
|
|
|
CP0073187
|
(S)-3-{4-[2-(5-Methyl-2-phenyl-oxazol-4-yl)-ethoxy]-phenyl}-2-morpholin-4-yl-propionic acid
Show/Hide
|
C25H28N2O5
|
1
|
| 1 |
EC50 = 24 nM
|
|
|
|
CP0035136
|
3-(4-(3-((5-chloro-3-methyl-1H-indole-2-carboxamido)methyl)phenoxy)-2-methylphenyl)propanoic acid
Show/Hide
|
C27H25ClN2O4
|
1
|
| 1 |
EC50 = 24 nM
|
|
|
|
CP0035143
|
2-(4-(5-((2-fluoro-4-(trifluoromethyl)benzamido)methyl)-2-methylphenoxy)-2-methylphenoxy)-2-methylpropanoic acid
Show/Hide
|
C27H25F4NO5
|
1
|
| 1 |
EC50 = 24 nM
|
|
|
|
CP0216421
|
2-(4-(3-((2-fluoro-4-(trifluoromethyl)benzamido)methyl)phenoxy)-2-methylphenoxy)-2-methylpropanoic acid
Show/Hide
|
C26H23F4NO5
|
1
|
| 1 |
EC50 = 24 nM
|
|
|
|
CP0216422
|
2-methyl-2-(2-methyl-4-(3-((2-methyl-4-(trifluoromethyl)benzamido)methyl)phenoxy)phenoxy)propanoic acid
Show/Hide
|
C27H26F3NO5
|
1
|
| 1 |
EC50 = 24 nM
|
|
|
|
CP0342886
|
2-Isopropoxy-3-{4-[5-(4-trifluoromethyl-phenyl)-[1,2,4]oxadiazol-3-ylmethoxy]-phenyl}-propionic acid
Show/Hide
|
C22H21F3N2O5
|
1
|
| 1 |
EC50 = 25 nM
|
|
|
|
CP0367812
|
3-(4-(2-(5-(4-chlorophenyl)-1,2,4-oxadiazol-3-yl)ethoxy)phenyl)-2-isopropoxypropanoic acid
Show/Hide
|
C22H23ClN2O5
|
1
|
| 1 |
EC50 = 25 nM
|
|
|
|
CP0210104
|
2-(4-(3-((2,4-dimethylbenzamido)methyl)phenoxy)-2-methylphenoxy)-2-methylpropanoic acid
Show/Hide
|
C27H29NO5
|
1
|
| 1 |
EC50 = 25 nM
|
|
|
|
CP0221348
|
3-(4-(3-((5-chloro-1H-indole-2-carboxamido)methyl)phenoxy)-2-methylphenyl)propanoic acid
Show/Hide
|
C26H23ClN2O4
|
1
|
| 1 |
EC50 = 25 nM
|
|
|
|
CP0035145
|
2-(4-(3-((4-methoxy-2-methylbenzamido)methyl)phenoxy)-2-methylphenoxy)-2-methylpropanoic acid
Show/Hide
|
C27H29NO6
|
1
|
| 1 |
EC50 = 26 nM
|
|
|
|
CP0371991
|
(S)-3-(3-((E)-1-(2-Chlorobenzyloxyimino)ethyl)phenyl)-2-ethoxypropanoicAcid
Show/Hide
|
C20H22ClNO4
|
1
|
| 1 |
EC50 = 26 nM
|
|
|
|
CP0035108
|
2-(4-(3-((4-chloro-2-methylbenzamido)methyl)phenoxy)-2-methylphenoxy)-2-methylpropanoic acid
Show/Hide
|
C26H26ClNO5
|
1
|
| 1 |
EC50 = 28 nM
|
|
|
|
CP0075561
|
2-(4-(4-fluoro-3-((2-fluoro-4-(trifluoromethyl)benzamido)methyl)phenoxy)-2-methylphenoxy)-2-methylpropanoic acid
Show/Hide
|
C26H22F5NO5
|
1
|
| 1 |
EC50 = 28 nM
|
|
|
|
CP0417381
|
(S)-3-(3-((E)-1-(4-Chlorobenzyloxyimino)ethyl)phenyl)-2-ethoxypropanoicAcid
Show/Hide
|
C20H22ClNO4
|
1
|
| 1 |
EC50 = 28 nM
|
|
|
|
CP0162116
|
3-(2-((isopropoxycarbonyl)methyl)-4-(2-(5-methyl-2-morpholinothiazol-4-yl)ethoxy)phenyl)propanoic acid
Show/Hide
|
C24H33N3O6S
|
1
|
| 1 |
EC50 = 28 nM
|
|
|
|
CP0393546
|
(2R)-2-benzyl-3-[3-[[[4-(3-fluorophenyl)benzoyl]amino]methyl]-4-propoxyphenyl]propanoic acid
Show/Hide
|
C33H32FNO4
|
1
|
| 1 |
EC50 = 28.7 nM
|
|
|
|
CP0183251
|
3-[4-[2-[1,3-benzoxazol-2-yl(methyl)amino]ethoxy]phenyl]-2-[2-(2-phenylacetyl)anilino]propanoic acid
Show/Hide
|
C33H31N3O5
|
1
|
| 1 |
EC50 = 28.84 nM
|
|
|
|
CP0374481
|
2-[3-(3-{(2,4-Bis-trifluoromethyl-benzyl)-[2-(3,4-dichloro-phenoxy)-acetyl]-amino}-propyl)-phenoxy]-2-methyl-propionic acid
Show/Hide
|
C30H27Cl2F6NO5
|
1
|
| 1 |
EC50 = 30 nM
|
|
|
|
CP0005387
|
Avandamet
Show/Hide
|
C18H19N3O3S
|
7
|
| 1 |
EC50 = 30 nM
|
|
|
| 2 |
EC50 = 33 nM
|
|
|
| 3 |
EC50 = 43 nM
|
|
|
| 4 |
EC50 = 76 nM
|
|
|
| 5 |
EC50 = 89.13 nM
|
|
|
| 6 |
EC50 = 100 nM
|
|
|
| 7 |
EC50 = 308 nM
|
|
|
|
CP0114159
|
3-(4-((5-(4-bromophenyl)-1,2,4-oxadiazol-3-yl)methoxy)phenyl)-2-isopropoxypropanoic acid
Show/Hide
|
C21H21BrN2O5
|
1
|
| 1 |
EC50 = 32 nM
|
|
|
|
CP0204434
|
3-(4-((5-(3,5-bis(trifluoromethyl)phenyl)-1,2,4-oxadiazol-3-yl)methoxy)phenyl)-2-isopropoxypropanoic acid
Show/Hide
|
C23H20F6N2O5
|
1
|
| 1 |
EC50 = 32 nM
|
|
|
|
CP0035196
|
3-(4-(3-((5-bromo-1H-indole-2-carboxamido)methyl)phenoxy)-2-methylphenyl)propanoic acid
Show/Hide
|
C26H23BrN2O4
|
1
|
| 1 |
EC50 = 32 nM
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CP0380576
|
(2R)-2-benzyl-3-[4-propoxy-3-[[(4-pyrimidin-2-ylbenzoyl)amino]methyl]phenyl]propanoic acid
Show/Hide
|
C31H31N3O4
|
1
|
| 1 |
EC50 = 34.6 nM
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CP0453617
|
(S)-3-(3-((E)-1-(4-Bromobenzyloxyimino)ethyl)phenyl)-2-ethoxypropanoicAcid
Show/Hide
|
C20H22BrNO4
|
1
|
| 1 |
EC50 = 36 nM
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CP0035140
|
2-(4-(3-((2-fluoro-4-(trifluoromethyl)benzamido)methyl)-5-methylphenoxy)-2-methylphenoxy)-2-methylpropanoic acid
Show/Hide
|
C27H25F4NO5
|
1
|
| 1 |
EC50 = 37 nM
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|
|
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CP0886328
|
S,S'-{8-[(2-{4-[(2,4-dioxo-1,3-thiazolidin-5-yl)methyl]phenoxy}-ethyl)(methyl)amino]-8-oxooctane-1,3-diyl} Diethanethioate
Show/Hide
|
C25H34N2O6S3
|
1
|
| 1 |
EC50 = 39 nM
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CP0114153
|
3-(4-(2-(5-(4-fluorophenyl)-1,2,4-oxadiazol-3-yl)ethoxy)phenyl)-2-isopropoxypropanoic acid
Show/Hide
|
C22H23FN2O5
|
1
|
| 1 |
EC50 = 40 nM
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CP0371993
|
(S)-3-(3-((E)-1-(4-Iodobenzyloxyimino)ethyl)phenyl)-2-ethoxypropanoicAcid
Show/Hide
|
C20H22INO4
|
1
|
| 1 |
EC50 = 40 nM
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|
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CP0075559
|
2-methyl-2-(2-methyl-4-(3-((4-(trifluoromethyl)benzamido)methyl)phenoxy)phenoxy)propanoic acid
Show/Hide
|
C26H24F3NO5
|
1
|
| 1 |
EC50 = 42 nM
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CP0035142
|
2-(4-(3-((2-fluoro-4-(trifluoromethyl)benzamido)methyl)-4-methylphenoxy)-2-methylphenoxy)-2-methylpropanoic acid
Show/Hide
|
C27H25F4NO5
|
1
|
| 1 |
EC50 = 43 nM
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|
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CP0136122
|
2-(4-(3-((2-bromo-4-(trifluoromethyl)benzamido)methyl)phenoxy)-2-methylphenoxy)-2-methylpropanoic acid
Show/Hide
|
C26H23BrF3NO5
|
1
|
| 1 |
EC50 = 43 nM
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CP0075562
|
3-(4-(3-((5-chloro-1,3-dimethyl-1H-indole-2-carboxamido)methyl)phenoxy)-2-methylphenyl)propanoic acid
Show/Hide
|
C28H27ClN2O4
|
1
|
| 1 |
EC50 = 44 nM
|
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CP0441191
|
(S)-3-(3-((E)-1-(4-Trifluoromethylbenzyloxyimino)ethyl)phenyl)-2-ethoxypropanoic Acid
Show/Hide
|
C21H22F3NO4
|
1
|
| 1 |
EC50 = 46 nM
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CP0166832
|
3-{4-[3-(2-benzoyl-4-ethyl-phenoxy)-pentyloxy]-2-methyl-phenyl}-propionic acid
Show/Hide
|
C30H34O5
|
1
|
| 1 |
EC50 = 46 nM
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CP0429825
|
4'-((5-(benzylcarbamoyl)-2,3-dimethyl-1H-indol-1-yl)methyl)biphenyl-2-carboxylic acid
Show/Hide
|
C32H28N2O3
|
1
|
| 1 |
EC50 = 47 nM
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CP0035149
|
2-(4-(3-((2-chloro-4-(trifluoromethyl)benzamido)methyl)phenoxy)-2-methylphenoxy)-2-methylpropanoic acid
Show/Hide
|
C26H23ClF3NO5
|
1
|
| 1 |
EC50 = 49 nM
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|
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CP0380579
|
(2R)-2-benzyl-3-[3-[[[4-(2-fluorophenyl)benzoyl]amino]methyl]-4-propoxyphenyl]propanoic acid
Show/Hide
|
C33H32FNO4
|
1
|
| 1 |
EC50 = 49.5 nM
|
|
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CP0071095
|
2-Isopropoxy-3-[4-(5-m-tolyl-[1,2,4]oxadiazol-3-ylmethoxy)-phenyl]-propionic acid
Show/Hide
|
C22H24N2O5
|
1
|
| 1 |
EC50 = 50 nM
|
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CP0212898
|
(2S)-2-(2-benzoylanilino)-3-[4-[2-(5-ethylpyridin-2-yl)ethoxy]phenyl]propanoic acid
Show/Hide
|
C31H30N2O4
|
1
|
| 1 |
EC50 = 50.12 nM
|
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|
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CP0254225
|
(R)-3-{4-[3-(4-chloro-2-phenoxy-phenoxy)-butoxy]-2-methyl-phenyl}-propionic acid
Show/Hide
|
C26H27ClO5
|
1
|
| 1 |
EC50 = 52 nM
|
|
|
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CP0261716
|
2-(4-(3-((2-ethyl-4-(trifluoromethyl)benzamido)methyl)phenoxy)-2-methylphenoxy)-2-methylpropanoic acid
Show/Hide
|
C28H28F3NO5
|
1
|
| 1 |
EC50 = 57 nM
|
|
|
|
CP0917967
|
2,2'-[{8-[(2-{4-[(2,4-dDioxo-1,3-thiazolidin-5-yl)methyl]phenoxy}-ethyl)(methyl)amino]-8-oxooctane-1,3-diyl}bis(thio)]bis(2-oxoethanaminium) dichloride
Show/Hide
|
C25H38Cl2N4O6S3
|
1
|
| 1 |
EC50 = 60 nM
|
|
|
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CP0114158
|
2-Isopropoxy-3-{4-[5-(4-trifluoromethoxy-phenyl)-[1,2,4]oxadiazol-3-ylmethoxy]-phenyl}-propionic acid
Show/Hide
|
C22H21F3N2O6
|
1
|
| 1 |
EC50 = 63 nM
|
|
|
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CP0380580
|
(2R)-2-benzyl-3-[4-propoxy-3-[[(4-thiophen-2-ylbenzoyl)amino]methyl]phenyl]propanoic acid
Show/Hide
|
C31H31NO4S
|
1
|
| 1 |
EC50 = 65.2 nM
|
|
|
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CP0136164
|
3-(2-methyl-4-((R)-3-(2-(pyridin-2-yl)-4-(trifluoromethyl)phenoxy)butoxy)phenyl)propanoic acid
Show/Hide
|
C26H26F3NO4
|
1
|
| 1 |
EC50 = 67 nM
|
|
|
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CP0455980
|
(2R)-2-benzyl-3-[3-[[[4-(2-methylphenyl)benzoyl]amino]methyl]-4-propoxyphenyl]propanoic acid
Show/Hide
|
C34H35NO4
|
1
|
| 1 |
EC50 = 73.8 nM
|
|
|
|
CP0926762
|
N-(2-{4-[(2,4-dioxo-1,3-thiazolidin-5-yl)methyl]phenoxy}-ethyl)-6,8-dimercapto-N-methyloctanamide
Show/Hide
|
C21H30N2O4S3
|
1
|
| 1 |
EC50 = 75 nM
|
|
|
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CP0071096
|
2-Isopropoxy-3-[4-(5-phenyl-[1,2,4]oxadiazol-3-ylmethoxy)-phenyl]-propionic acid
Show/Hide
|
C21H22N2O5
|
1
|
| 1 |
EC50 = 79 nM
|
|
|
|
CP0938860
|
4,4'-[{8-[(2-{4-[(2,4-dioxo-1,3-thiazolidin-5-yl)methyl]phenoxy}-ethyl)(methyl)amino]-8-oxooctane-1,3-diyl}bis(thio)]bis(4-oxobutanoic acid) disodium salt
Show/Hide
|
C29H36N2Na2O10S3
|
1
|
| 1 |
EC50 = 80 nM
|
|
|
|
CP0421159
|
2-propyl-5-(1-propylbenzimidazol-2-yl)-3-[[4-[2-(2H-tetrazol-5-yl)phenyl]phenyl]methyl]pyrazolo[1,5-a]pyridine
Show/Hide
|
C34H32N8
|
1
|
| 1 |
EC50 = 80 nM
|
|
|
|
CP0463084
|
2-[3-(3-{(2-Cyclopropyl-3-[1,2,4]oxadiazol-3-yl-phenyl)-[2-(4-trifluoromethyl-phenyl)-acetyl]-amino}-propyl)-phenoxy]-2-methyl-propionic acid
Show/Hide
|
C33H32F3N3O5
|
1
|
| 1 |
EC50 = 81 nM
|
|
|
|
CP0376472
|
(2R)-2-benzyl-3-[3-[[(4-phenylbenzoyl)amino]methyl]-4-propoxyphenyl]propanoic acid
Show/Hide
|
C33H33NO4
|
1
|
| 1 |
EC50 = 85.9 nM
|
|
|
|
CP0439849
|
2-[4-[[1-methoxy-5-(1-phenylpropylcarbamoyl)-2-propylindol-3-yl]methyl]phenyl]benzoic acid
Show/Hide
|
C36H36N2O4
|
1
|
| 1 |
EC50 = 90 nM
|
|
|
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CP0085230
|
3-(4-((5-(3-fluorophenyl)-1,2,4-oxadiazol-3-yl)methoxy)phenyl)-2-isopropoxypropanoic acid
Show/Hide
|
C21H21FN2O5
|
1
|
| 1 |
EC50 = 100 nM
|
|
|
|
CP0231601
|
2-Isopropoxy-3-[4-(5-o-tolyl-[1,2,4]oxadiazol-3-ylmethoxy)-phenyl]-propionic acid
Show/Hide
|
C22H24N2O5
|
1
|
| 1 |
EC50 = 100 nM
|
|
|
|
CP0286632
|
3-(4-((5-(3,5-difluorophenyl)-1,2,4-oxadiazol-3-yl)methoxy)phenyl)-2-isopropoxypropanoic acid
Show/Hide
|
C21H20F2N2O5
|
1
|
| 1 |
EC50 = 100 nM
|
|
|
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CP0393242
|
2-methyl-2-(2-methyl-4-((4-methyl-2-(4-(trifluoromethyl)phenyl)thiazol-5-yl)methylselanyl)phenoxy)propanoic acid
Show/Hide
|
C23H22F3NO3SSe
|
1
|
| 1 |
EC50 = 100.2 nM
|
|
|
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CP0221700
|
(R)-3-{4-[3-(4-chloro-2-phenoxy-phenoxy)-butoxy]-2-ethyl-phenyl}-propionic acid
Show/Hide
|
C27H29ClO5
|
1
|
| 1 |
EC50 = 102 nM
|
|
|
|
CP0477434
|
(2R)-2-benzyl-3-[3-[[[4-(4-fluorophenyl)benzoyl]amino]methyl]-4-propoxyphenyl]propanoic acid
Show/Hide
|
C33H32FNO4
|
1
|
| 1 |
EC50 = 102.6 nM
|
|
|
|
CP0185360
|
3-[4-[2-[1,3-benzoxazol-2-yl(methyl)amino]ethoxy]phenyl]-2-(2-phenoxyanilino)propanoic acid
Show/Hide
|
C31H29N3O5
|
1
|
| 1 |
EC50 = 107.15 nM
|
|
|
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CP0112273
|
3-(2-ethyl-4-((R)-3-(2-(pyridin-2-yl)-4-(trifluoromethyl)phenoxy)butoxy)phenyl)propanoic acid
Show/Hide
|
C27H28F3NO4
|
1
|
| 1 |
EC50 = 111 nM
|
|
|
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CP0053319
|
2-(4-(3-(2-benzoyl-4-ethylphenoxy)propoxy)phenoxy)-2-methylpropanoic acid
Show/Hide
|
C28H30O6
|
1
|
| 1 |
EC50 = 112 nM
|
|
|
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CP0104572
|
3-(2-((benzyloxycarbonyl)methyl)-4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)phenyl)propanoic acid
Show/Hide
|
C30H30N2O6
|
1
|
| 1 |
EC50 = 115 nM
|
|
|
|
CP0075560
|
(R)-3-(4-(3-(1-(5-chloro-1,3-dimethyl-1H-indole-2-carboxamido)ethyl)-5-fluorophenoxy)-2-ethylphenyl)propanoic acid
Show/Hide
|
C30H30ClFN2O4
|
1
|
| 1 |
EC50 = 116 nM
|
|
|
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CP0371990
|
(S)-3-(3-((E)-1-Benzyloxyiminoethyl)phenyl)-2-ethoxypropanoic Acid
Show/Hide
|
C20H23NO4
|
1
|
| 1 |
EC50 = 121 nM
|
|
|
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CP0374172
|
(R)-2-Methyl-3-{4-[2-(5-methyl-2-thiophen-2-yl-oxazol-4-yl)-ethoxy]-phenyl}-2-phenoxy-propionic acid
Show/Hide
|
C26H25NO5S
|
1
|
| 1 |
EC50 = 121 nM
|
|
|
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CP0035144
|
2-methyl-2-(2-methyl-4-(3-((2-methylbenzamido)methyl)phenoxy)phenoxy)propanoic acid
Show/Hide
|
C26H27NO5
|
1
|
| 1 |
EC50 = 125 nM
|
|
|
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CP0430042
|
2-[4-[[5-(1-phenylpropylcarbamoyl)-2-propylindazol-3-yl]methyl]phenyl]benzoic acid
Show/Hide
|
C34H33N3O3
|
1
|
| 1 |
EC50 = 130 nM
|
|
|
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CP0051472
|
3-(4-(3-((5-chloro-1-methyl-1H-indole-2-carboxamido)methyl)phenoxy)-2-methylphenyl)propanoic acid
Show/Hide
|
C27H25ClN2O4
|
1
|
| 1 |
EC50 = 135 nM
|
|
|
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CP0151693
|
(S)-3-{4-[2-(5-Methyl-2-phenyl-oxazol-4-yl)-ethoxy]-phenyl}-2-piperidin-1-yl-propionic acid
Show/Hide
|
C26H30N2O4
|
1
|
| 1 |
EC50 = 138 nM
|
|
|
|
CP0371986
|
(S)-3-(3-((E)-1-(4-Fluorobenzyloxyimino)ethyl)phenyl)-2-ethoxypropanoicAcid
Show/Hide
|
C20H22FNO4
|
1
|
| 1 |
EC50 = 139 nM
|
|
|
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CP0035355
|
3-(4-((R)-3-(4-ethyl-2-(pyridin-3-yl)phenoxy)butoxy)-2-methylphenyl)propanoic acid
Show/Hide
|
C27H31NO4
|
1
|
| 1 |
EC50 = 140 nM
|
|
|
|
CP0444352
|
(2R)-3-(4-(3-((4-tert-butylbenzyl)carbamothioyloxy)-3-phenylpropyl)phenyl)-2-ethoxypropanoic acid
Show/Hide
|
C32H39NO4S
|
1
|
| 1 |
EC50 = 140 nM
|
|
|
|
CP0955609
|
4-({3-(acetylthio)-8-[(2-{4-[(2,4-dioxo-1,3-thiazolidin-5-yl)-methyl]phenoxy}ethyl)(methyl)amino]-8-oxooctyl}thio)-4-oxobutanoic acid sodium salt
Show/Hide
|
C27H35N2NaO8S3
|
1
|
| 1 |
EC50 = 150 nM
|
|
|
|
CP0261715
|
3-(4-(3-((7-bromo-1H-indole-2-carboxamido)methyl)phenoxy)-2-methylphenyl)propanoic acid
Show/Hide
|
C26H23BrN2O4
|
1
|
| 1 |
EC50 = 158 nM
|
|
|
|
CP0136386
|
alkynyl ether, 21
Show/Hide
|
C31H29F3O5S
|
1
|
| 1 |
EC50 = 160 nM
|
|
|
|
CP0373699
|
(2S)-3-(4-(3-((4-tert-butylbenzyl)carbamothioyloxy)-3-phenylpropyl)phenyl)-2-ethoxypropanoic acid
Show/Hide
|
C32H39NO4S
|
1
|
| 1 |
EC50 = 160 nM
|
|
|
|
CP0233673
|
2-Isopropoxy-3-(4-{2-[5-(2-trifluoromethyl-phenyl)-[1,2,4]oxadiazol-3-yl]-ethoxy}-phenyl)-propionic acid
Show/Hide
|
C23H23F3N2O5
|
2
|
| 1 |
EC50 = 160 nM
|
|
|
| 2 |
EC50 = 600 nM
|
|
|
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CP0215238
|
(R)-3-(4-(3-(1-(5-chloro-3-methylbenzo[b]thiophene-2-carboxamido)ethyl)-5-fluorophenoxy)-2-ethylphenyl)propanoic acid
Show/Hide
|
C29H27ClFNO4S
|
1
|
| 1 |
EC50 = 163 nM
|
|
|
|
CP0430855
|
4'-((2-methyl-6-(1-phenylpropylcarbamoyl)-1H-indol-1-yl)methyl)biphenyl-2-carboxylic acid
Show/Hide
|
C33H30N2O3
|
1
|
| 1 |
EC50 = 163 nM
|
|
|
|
CP0212814
|
3-[4-[2-[1,3-benzoxazol-2-yl(methyl)amino]ethoxy]phenyl]-2-[(2-benzoylphenyl)methylamino]propanoic acid
Show/Hide
|
C33H31N3O5
|
1
|
| 1 |
EC50 = 165.96 nM
|
|
|
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CP0035358
|
3-(2-ethyl-4-((R)-3-(4-ethyl-2-(pyridin-2-yl)phenoxy)butoxy)phenyl)propanoic acid
Show/Hide
|
C28H33NO4
|
1
|
| 1 |
EC50 = 167 nM
|
|
|
|
CP0448498
|
2-[3-(3-{(2-Cyclopropyl-3-[1,2,4]oxadiazol-3-yl-phenyl)-[2-(3,4-dichloro-phenoxy)-acetyl]-amino}-propyl)-phenoxy]-2-methyl-propionic acid
Show/Hide
|
C32H31Cl2N3O6
|
1
|
| 1 |
EC50 = 170 nM
|
|
|
|
CP0384607
|
(S)-3-(3-((E)-1-(4-Methoxybenzyloxyimino)ethyl)phenyl)-2-ethoxypropanoicAcid
Show/Hide
|
C21H25NO5
|
1
|
| 1 |
EC50 = 175 nM
|
|
|
|
CP0425898
|
N-(1-phenylpropyl)-2-propyl-3-[[4-[2-(2H-tetrazol-5-yl)phenyl]phenyl]methyl]pyrazolo[1,5-a]pyridine-5-carboxamide
Show/Hide
|
C34H33N7O
|
1
|
| 1 |
EC50 = 180 nM
|
|
|
|
CP0264567
|
3-(4-((R)-3-(4-ethyl-2-(pyridin-2-yl)phenoxy)butoxy)-2-methylphenyl)propanoic acid
Show/Hide
|
C27H31NO4
|
1
|
| 1 |
EC50 = 182 nM
|
|
|
|
CP0465587
|
(2R)-2-benzyl-3-[4-propoxy-3-[[(4-pyridin-2-ylbenzoyl)amino]methyl]phenyl]propanoic acid
Show/Hide
|
C32H32N2O4
|
1
|
| 1 |
EC50 = 186.1 nM
|
|
|
|
CP0889255
|
2-({3-(acetylthio)-8-[(2-{4-[(2,4-dioxo-1,3-thiazolidin-5-yl)-methyl]phenoxy}ethyl)(methyl)amino]-8-oxooctyl}thio)-2-oxoethanaminium chloride
Show/Hide
|
C25H36ClN3O6S3
|
1
|
| 1 |
EC50 = 195 nM
|
|
|
|
CP0397728
|
2-(4-{2-[3-(2,4-Difluoro-phenyl)-1-heptyl-ureido]-ethyl}-phenoxy)-2-methyl-propionic acid
Show/Hide
|
C26H34F2N2O4
|
1
|
| 1 |
EC50 = 200 nM
|
|
|
|
CP0367813
|
3-(4-((5-(4-fluorophenyl)-1,2,4-oxadiazol-3-yl)methoxy)phenyl)-2-isopropoxypropanoic acid
Show/Hide
|
C21H21FN2O5
|
1
|
| 1 |
EC50 = 200 nM
|
|
|
|
CP0502261
|
4'-((3-(methylthio)-6-(2-phenylbutanamido)-2-propyl-1H-indol-1-yl)methyl)biphenyl-2-carboxylic acid
Show/Hide
|
C36H36N2O3S
|
1
|
| 1 |
EC50 = 201 nM
|
|
|
|
CP0371989
|
(2(S)-2-Ethoxy-3-(3-(5-phenyl-4,5-dihydroisoxazole-3-yl)phenyl)propanoic Acid
Show/Hide
|
C20H21NO4
|
1
|
| 1 |
EC50 = 220 nM
|
|
|
|
CP0131907
|
3-{4-[3-(2-benzyl-4-ethyl-phenoxy)-butoxy]-2-methyl-phenyl}-propionic acid
Show/Hide
|
C29H34O4
|
1
|
| 1 |
EC50 = 228 nM
|
|
|
|
CP0383272
|
3-(4-((5-cyclohexyl-1,2,4-oxadiazol-3-yl)methoxy)phenyl)-2-isopropoxypropanoic acid
Show/Hide
|
C21H28N2O5
|
1
|
| 1 |
EC50 = 230 nM
|
|
|
|
CP0261714
|
3-(4-(3-((5,6-dichloro-1H-indole-2-carboxamido)methyl)phenoxy)-2-methylphenyl)propanoic acid
Show/Hide
|
C26H22Cl2N2O4
|
1
|
| 1 |
EC50 = 238 nM
|
|
|
|
CP0208139
|
(S)-3-{4-[2-(5-Methyl-2-phenyl-oxazol-4-yl)-ethoxy]-phenyl}-2-propylamino-propionic acid
Show/Hide
|
C24H28N2O4
|
1
|
| 1 |
EC50 = 240 nM
|
|
|
|
CP0432277
|
5-(1-butylbenzimidazol-2-yl)-2-propyl-3-[[4-[2-(2H-tetrazol-5-yl)phenyl]phenyl]methyl]indazole
Show/Hide
|
C35H34N8
|
1
|
| 1 |
EC50 = 250 nM
|
|
|
|
CP0437345
|
2-(4-((2-(3-fluoro-4-(trifluoromethyl)phenyl)-4-methylthiazol-5-yl)methylselanyl)-2-methylphenoxy)butanoic acid
Show/Hide
|
C23H21F4NO3SSe
|
1
|
| 1 |
EC50 = 270.6 nM
|
|
|
|
CP0384219
|
(S)-3-(3-((E)-1-(4-(tert-Butylbenzyloxyimino)ethyl)phenyl)-2-ethoxypropanoic Acid
Show/Hide
|
C24H31NO4
|
1
|
| 1 |
EC50 = 279 nM
|
|
|
|
CP0374670
|
2-(4-{2-[3-(4-Fluoro-phenyl)-1-heptyl-ureido]-ethyl}-phenoxy)-2-methyl-propionic acid
Show/Hide
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C26H35FN2O4
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1
|
| 1 |
EC50 = 280 nM
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CP0380009
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2-[4-[[2-propyl-5-(1-propylbenzimidazol-2-yl)pyrazolo[1,5-a]pyridin-3-yl]methyl]phenyl]benzoic acid
Show/Hide
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C34H32N4O2
|
1
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| 1 |
EC50 = 280 nM
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CP0406362
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2-{4-[2-(5-Methyl-2-phenyl-oxazol-4-yl)-ethoxy]-benzyl}-2-phenoxy-butyric acid
Show/Hide
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C29H29NO5
|
1
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| 1 |
EC50 = 285 nM
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CP0381217
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2-(4-((2-(3-fluoro-4-(trifluoromethyl)phenyl)-4-methylthiazol-5-yl)methylselanyl)-2-methylphenoxy)-2-methylpropanoic acid
Show/Hide
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C23H21F4NO3SSe
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1
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| 1 |
EC50 = 290.3 nM
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CP0086938
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alkynyl ether, 29
Show/Hide
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C31H29F3O5S
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1
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| 1 |
EC50 = 300 nM
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CP0441016
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2-methyl-2-[6-(5-methyl-2-phenyl-1,3-oxazol-4-yl)hexoxy]propanoic acid
Show/Hide
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C20H27NO4
|
1
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| 1 |
EC50 = 300 nM
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CP0496924
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2-methyl-5-[5-(5-methyl-2-phenyl-1,3-oxazol-4-yl)pentyl]-1,3-dioxane-2-carboxylic acid
Show/Hide
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C21H27NO5
|
1
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| 1 |
EC50 = 300 nM
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CP0405640
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(2S)-2-ethoxy-3-(4-(3-hydroxy-3-phenylpropyl)phenyl)propanoic acid
Show/Hide
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C20H24O4
|
1
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| 1 |
EC50 = 300 nM
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CP0051320
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3-(4-((R)-3-(4-chloro-2-(pyridin-2-yl)phenoxy)butoxy)-2-methylphenyl)propanoic acid
Show/Hide
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C25H26ClNO4
|
1
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| 1 |
EC50 = 304 nM
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CP0377750
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2-(3-{3-[(3,4-Bis-trifluoromethyl-benzoyl)-(2-cyclopropyl-3-[1,2,4]oxadiazol-3-yl-phenyl)-amino]-propyl}-phenoxy)-2-methyl-propionic acid
Show/Hide
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C33H29F6N3O5
|
1
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| 1 |
EC50 = 320 nM
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CP0380840
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2-(4-{2-[1-(4-Cyclohexyl-butyl)-3-(2-methoxy-phenyl)-ureido]-ethyl}-phenylsulfanyl)-2-methyl-propionic acid
Show/Hide
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C30H42N2O4S
|
1
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| 1 |
EC50 = 320 nM
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CP0417838
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4'-((2,3-dimethyl-5-(2-phenylbutanamido)-1H-indol-1-yl)methyl)biphenyl-2-carboxylic acid
Show/Hide
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C34H32N2O3
|
1
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| 1 |
EC50 = 338 nM
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CP0035141
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3-(2-methyl-4-(3-((2-methyl-4-(trifluoromethyl)benzamido)methyl)phenoxy)phenyl)propanoic acid
Show/Hide
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C26H24F3NO4
|
1
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| 1 |
EC50 = 345 nM
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CP0035138
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3-(4-(3-((6-chloro-1H-indole-2-carboxamido)methyl)phenoxy)-2-methylphenyl)propanoic acid
Show/Hide
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C26H23ClN2O4
|
1
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| 1 |
EC50 = 348 nM
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CP0444351
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(2R)-3-(4-(3-(benzylcarbamothioyloxy)-3-phenylpropyl)phenyl)-2-ethoxypropanoic acid
Show/Hide
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C28H31NO4S
|
1
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| 1 |
EC50 = 350 nM
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CP0437799
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2-[4-[[5-(1-phenylpropylcarbamoyl)-2-propyl-1H-indol-3-yl]methyl]phenyl]benzoic acid
Show/Hide
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C35H34N2O3
|
1
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| 1 |
EC50 = 350 nM
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CP0221734
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(R)-3-{4-[3-(4-chloro-2-phenoxy-phenoxy)-butoxy]-2-trifluoromethyl-phenyl}-propionic acid
Show/Hide
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C26H24ClF3O5
|
1
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| 1 |
EC50 = 355 nM
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CP0077439
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(R)-2-Methyl-3-{4-[2-(5-methyl-2-phenyl-oxazol-4-yl)-ethoxy]-phenyl}-2-phenoxy-propionic acid
Show/Hide
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C28H27NO5
|
1
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| 1 |
EC50 = 382 nM
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CP0353943
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(S)-3-{4-[2-(5-Methyl-2-phenyl-oxazol-4-yl)-ethoxy]-phenyl}-2-pyrrolidin-1-yl-propionic acid
Show/Hide
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C25H28N2O4
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1
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| 1 |
EC50 = 390 nM
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CP0208857
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alkynyl ether, 37
Show/Hide
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C28H32O5S
|
1
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| 1 |
EC50 = 390 nM
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CP0461864
|
3-{4-[2-(5-Methyl-2-phenyl-oxazol-4-yl)-ethoxy]-phenyl}-2-phenoxy-propionic acid
Show/Hide
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C27H25NO5
|
1
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| 1 |
EC50 = 390 nM
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CP0432279
|
2-[4-[[5-(1-phenylpropylcarbamoyl)-2-propylpyrazolo[1,5-a]pyridin-3-yl]methyl]phenyl]benzoic acid
Show/Hide
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C34H33N3O3
|
1
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| 1 |
EC50 = 390 nM
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CP0048240
|
BDBM50101974
Show/Hide
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C24H27NO5S
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2
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| 1 |
EC50 = 400 nM
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| 2 |
EC50 = 537.03 nM
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CP0057749
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(R)-3-{4-[3-(4-chloro-2-phenoxy-phenoxy)-butoxy]-2-fluoro-phenyl}-propionic acid
Show/Hide
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C25H24ClFO5
|
1
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| 1 |
EC50 = 402 nM
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CP0292262
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(S)-2-Dimethylamino-3-{4-[2-(5-methyl-2-phenyl-oxazol-4-yl)-ethoxy]-phenyl}-propionic acid
Show/Hide
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C23H26N2O4
|
1
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| 1 |
EC50 = 410 nM
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CP0356376
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2-[2-[hydroxy(phenyl)methyl]anilino]-3-[4-[2-[methyl(pyridin-2-yl)amino]ethoxy]phenyl]propanoic acid
Show/Hide
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C30H31N3O4
|
1
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| 1 |
EC50 = 446.68 nM
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CP0035147
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2-methyl-2-(2-methyl-4-(3-((2-phenoxy-4-(trifluoromethyl)benzamido)methyl)phenoxy)phenoxy)propanoic acid
Show/Hide
|
C32H28F3NO6
|
1
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| 1 |
EC50 = 479 nM
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CP0310008
|
3-[4-[2-[1,3-benzoxazol-2-yl(methyl)amino]ethoxy]phenyl]-2-[(9-oxofluoren-1-yl)amino]propanoic acid
Show/Hide
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C32H27N3O5
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1
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| 1 |
EC50 = 489.78 nM
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CP0795074
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(S)-3-(4-Benzyloxy-phenyl)-2-((Z)-1-methyl-3-oxo-3-phenyl-propenylamino)-propionamide
Show/Hide
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C26H26N2O3
|
1
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| 1 |
EC50 = 489.78 nM
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CP0145069
|
alkynyl ether, 33
Show/Hide
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C30H28F3NO5S
|
1
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| 1 |
EC50 = 490 nM
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CP0373620
|
(2S)-2-ethoxy-3-(4-(3-(phenethylcarbamothioyloxy)-3-phenylpropyl)phenyl)propanoic acid
Show/Hide
|
C29H33NO4S
|
1
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| 1 |
EC50 = 490 nM
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CP0201561
|
alkynyl ether, 36
Show/Hide
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C29H34O5S
|
1
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| 1 |
EC50 = 500 nM
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CP0382216
|
2-[1-benzyl-5-[3-[3-[(4-chlorophenyl)methoxy]phenoxy]propoxy]indol-3-yl]acetic acid
Show/Hide
|
C33H30ClNO5
|
1
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| 1 |
EC50 = 500 nM
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CP0156647
|
3-(4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)-2-((phenylmethylsulfonamido)methyl)phenyl)propanoic acid
Show/Hide
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C29H30N2O6S
|
1
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| 1 |
EC50 = 527 nM
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CP0041219
|
Actos
Show/Hide
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C19H20N2O3S
|
3
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| 1 |
EC50 = 550 nM
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| 2 |
EC50 = 580 nM
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| 3 |
EC50 = 588.84 nM
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CP0036483
|
alkynyl ether, 31
Show/Hide
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C30H29ClO5S
|
1
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| 1 |
EC50 = 560 nM
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CP0035354
|
(R)-3-(4-(3-(4-ethyl-2-(pyridin-4-yl)phenoxy)butoxy)-2-methylphenyl)propanoic acid
Show/Hide
|
C27H31NO4
|
1
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| 1 |
EC50 = 576 nM
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CP0400048
|
(2S)-3-(4-(3-(benzylcarbamothioyloxy)-3-phenylpropyl)phenyl)-2-ethoxypropanoic acid
Show/Hide
|
C28H31NO4S
|
1
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| 1 |
EC50 = 580 nM
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CP0042069
|
(S)-3-{4-[2-(5-Methyl-2-phenyl-oxazol-4-yl)-ethoxy]-phenyl}-2-(pyrimidin-2-ylamino)-propionic acid
Show/Hide
|
C25H24N4O4
|
1
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| 1 |
EC50 = 590 nM
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CP0442664
|
(S)-2-Ethoxy-3-(3-(5-(4-iodophenyl)-4,5-dihydroisoxazol-3-yl)phenyl)propanoic Acid
Show/Hide
|
C20H20INO4
|
1
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| 1 |
EC50 = 606 nM
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CP0086940
|
alkynyl ether, 32
Show/Hide
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C31H31ClO5S
|
1
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| 1 |
EC50 = 610 nM
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CP0167310
|
alkynyl ether, 26
Show/Hide
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C31H29F3O6S
|
1
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| 1 |
EC50 = 610 nM
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CP0108120
|
(2S)-2-(2-benzoylanilino)-3-[4-[(1-methylcyclohexyl)methoxy]phenyl]propanoic acid
Show/Hide
|
C30H33NO4
|
1
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| 1 |
EC50 = 616.6 nM
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CP0082985
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N-[(2S)-2-(2-benzoylanilino)-3-[4-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]propyl]butanamide
Show/Hide
|
C38H39N3O4
|
2
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| 1 |
EC50 = 630.96 nM
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| 2 |
IC50 = 2511.89 nM
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CP0167603
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N-[(2S)-2-(2-benzoylanilino)-3-[4-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]propyl]cyclopropanecarboxamide
Show/Hide
|
C38H37N3O4
|
2
|
| 1 |
EC50 = 630.96 nM
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| 2 |
IC50 = 2511.89 nM
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CP0380010
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2-[4-[[5-(1-butylbenzimidazol-2-yl)-2-propylindazol-3-yl]methyl]phenyl]benzoic acid
Show/Hide
|
C35H34N4O2
|
1
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| 1 |
EC50 = 640 nM
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CP0274937
|
(S)-3-{4-[3-(2-benzoyl-4-ethyl-phenoxy)-butoxy]2-methyl-phenyl}propionic acid
Show/Hide
|
C29H32O5
|
1
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| 1 |
EC50 = 674 nM
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CP0722969
|
(S)-3-(4-Benzyloxy-phenyl)-2-((Z)-1-methyl-3-oxo-3-phenyl-propenylamino)-propionic acid methyl ester
Show/Hide
|
C27H27NO4
|
1
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| 1 |
EC50 = 691.83 nM
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CP0274499
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3-(4-((R)-3-(4-ethyl-2-(oxazol-2-yl)phenoxy)butoxy)-2-methylphenyl)propanoic acid
Show/Hide
|
C25H29NO5
|
1
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| 1 |
EC50 = 696 nM
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CP0280556
|
alkynyl ether, 20
Show/Hide
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C30H27F3O5S
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1
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| 1 |
EC50 = 700 nM
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CP0064613
|
(2S)-2-ethoxy-3-(4-{2-[4-(methanesulfonyloxy)phenyl]ethoxy}phenyl)propanoic acid
Show/Hide
|
C20H24O7S
|
1
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| 1 |
EC50 = 704 nM
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CP0220511
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(S)-2-(2,5-Dimethyl-pyrrol-1-yl)-3-{4-[2-(5-methyl-2-phenyl-oxazol-4-yl)-ethoxy]-phenyl}-propionic acid
Show/Hide
|
C27H28N2O4
|
1
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| 1 |
EC50 = 710 nM
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CP0393545
|
(2R)-2-benzyl-3-[4-propoxy-3-[[(4-pyrazin-2-ylbenzoyl)amino]methyl]phenyl]propanoic acid
Show/Hide
|
C31H31N3O4
|
1
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| 1 |
EC50 = 713.9 nM
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CP0409327
|
2-methyl-2-[4-({[4-(trifluoromethyl)-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl]formamido}methyl)phenoxy]propanoic acid
Show/Hide
|
C23H18F6N2O4S
|
1
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| 1 |
EC50 = 730 nM
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CP0442663
|
(S)-2-Ethoxy-3-(3-(5-(4-bromophenyl)-4,5-dihydroisoxazol-3-yl)phenyl)propanoic Acid
Show/Hide
|
C20H20BrNO4
|
1
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| 1 |
EC50 = 740 nM
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CP0472124
|
(S)-2-Ethoxy-3-(3-(5-(4-chlorophenyl)-4,5-dihydroisoxazol-3-yl)phenyl)propanoic Acid
Show/Hide
|
C20H20ClNO4
|
1
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| 1 |
EC50 = 816 nM
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CP0035360
|
3-{4-[(R)-3-(5-ethyl-biphenyl-2-yloxy)-butoxy]-2-methyl-phenyl}-propionic acid
Show/Hide
|
C28H32O4
|
1
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| 1 |
EC50 = 836 nM
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CP0035191
|
3-(4-((R)-3-(4-ethyl-2-(thiazol-4-yl)phenoxy)butoxy)-2-methylphenyl)propanoic acid
Show/Hide
|
C25H29NO4S
|
1
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| 1 |
EC50 = 837 nM
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CP0380578
|
(2R)-2-benzyl-3-[4-propoxy-3-[[(4-pyridin-3-ylbenzoyl)amino]methyl]phenyl]propanoic acid
Show/Hide
|
C32H32N2O4
|
1
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| 1 |
EC50 = 844 nM
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CP0723695
|
2-(2-(hydrazono(phenyl)methyl)phenylamino)-3-(4-(2-(methyl(pyridin-2-yl)amino)ethoxy)phenyl)propanoic acid
Show/Hide
|
C30H31N5O3
|
1
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| 1 |
EC50 = 851.14 nM
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CP0372105
|
2-[4-({[2-(4-tert-butylphenyl)-4-methyl-1,3-thiazol-5-yl]formamido}methyl)phenoxy]-2-methylpropanoic acid
Show/Hide
|
C26H30N2O4S
|
1
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| 1 |
EC50 = 860 nM
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CP0447683
|
4'-((6-(1-phenylpropylcarbamoyl)-2-propyl-1H-benzo[d]imidazol-1-yl)methyl)biphenyl-2-carboxylic acid
Show/Hide
|
C34H33N3O3
|
1
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| 1 |
EC50 = 900 nM
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CP0687662
|
5-(2,4-Dioxo-thiazolidin-5-ylmethyl)-2-methoxy-N-(4-trifluoromethyl-benzyl)-benzamide
Show/Hide
|
C20H17F3N2O4S
|
1
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| 1 |
EC50 = 900 nM
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CP0459249
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2-[3-[2-[4-Isopropyl-2-[4-(trifluoromethyl)phenyl]-5-thiazolyl]ethyl]-5-methyl-1,2-benzisoxazol-6-yloxy]-2-methylpropionic acid
Show/Hide
|
C27H27F3N2O4S
|
1
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| 1 |
EC50 = 910 nM
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CP0200699
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3-[4-[2-[1,3-benzoxazol-2-yl(methyl)amino]ethoxy]phenyl]-2-(2-benzoylphenoxy)propanoic acid
Show/Hide
|
C32H28N2O6
|
1
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| 1 |
EC50 = 933.25 nM
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CP0274904
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3-{4-[3-(2-benzoyl-4-ethyl-phenoxy)-hexyloxy]-2-methyl-phenyl}-propionic acid
Show/Hide
|
C31H36O5
|
1
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| 1 |
EC50 = 968 nM
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CP0170396
|
2-{[4-(2-{[(2,4-difluorophenyl)carbamoyl](heptyl)amino}ethyl)phenyl]sulfanyl}-2-methylpropanoic acid
Show/Hide
|
C26H34F2N2O3S
|
1
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| 1 |
EC50 = 1000 nM
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CP0409243
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2-(4-{2-[3-(3-Cyano-phenyl)-1-(4-cyclohexyl-butyl)-ureido]-ethyl}-phenylsulfanyl)-2-methyl-propionic acid
Show/Hide
|
C30H39N3O3S
|
1
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| 1 |
EC50 = 1000 nM
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CP0515829
|
2-(4-{2-[1-(4-Cyclohexyl-butyl)-3-(3,5-dichloro-phenyl)-ureido]-ethyl}-phenylsulfanyl)-2-methyl-propionic acid
Show/Hide
|
C29H38Cl2N2O3S
|
1
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| 1 |
EC50 = 1000 nM
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CP0441017
|
2-methyl-5-[[3-[(5-methyl-2-phenyl-1,3-oxazol-4-yl)methyl]phenyl]methyl]-1,3-dioxane-2-carboxylic acid
Show/Hide
|
C24H25NO5
|
1
|
| 1 |
EC50 = 1000 nM
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CP0145159
|
N-[(2S)-2-(2-benzoylanilino)-3-[4-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]propyl]acetamide
Show/Hide
|
C36H35N3O4
|
2
|
| 1 |
EC50 = 1000 nM
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| 2 |
IC50 = 1584.89 nM
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CP0441380
|
2-[3-[2-[2-(4-tert-Butylphenyl)-5-isopropyl-4-oxazolyl]ethyl]-1,2-benzisoxazol-6-yloxy]-2-methylpropionic acid
Show/Hide
|
C29H34N2O5
|
1
|
| 1 |
EC50 = 1000 nM
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CP0347599
|
3-(4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)-2-((3-phenylpropanamido)methyl)phenyl)propanoic acid
Show/Hide
|
C31H32N2O5
|
1
|
| 1 |
EC50 = 1019 nM
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CP0444350
|
(2R)-2-ethoxy-3-(4-(3-(phenethylcarbamothioyloxy)-3-phenylpropyl)phenyl)propanoic acid
Show/Hide
|
C29H33NO4S
|
1
|
| 1 |
EC50 = 1050 nM
|
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CP0075564
|
2-(4-(3-((2,4-bis(trifluoromethyl)benzamido)methyl)phenoxy)-2-methylphenoxy)-2-methylpropanoic acid
Show/Hide
|
C27H23F6NO5
|
1
|
| 1 |
EC50 = 1058 nM
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CP0444353
|
(2S)-3-(4-(3-((cyclohexylmethyl)carbamothioyloxy)-3-phenylpropyl)phenyl)-2-ethoxypropanoic acid
Show/Hide
|
C28H37NO4S
|
1
|
| 1 |
EC50 = 1060 nM
|
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CP0035109
|
3-(4-(3-((4-chloro-1H-indole-2-carboxamido)methyl)phenoxy)-2-methylphenyl)propanoic acid
Show/Hide
|
C26H23ClN2O4
|
1
|
| 1 |
EC50 = 1088 nM
|
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CP0023801
|
2-(4-(2-(3-cyclohexyl-1-(4-cyclohexylbutyl)ureido)ethyl)phenylthio)-2-methylpropanoic acid
Show/Hide
|
C29H46N2O3S
|
1
|
| 1 |
EC50 = 1100 nM
|
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CP0423213
|
(S)-2-Ethoxy-3-(3-(5-(4-fluorophenyl)-4,5-dihydroisoxazol-3-yl)phenyl)propanoic Acid
Show/Hide
|
C20H20FNO4
|
1
|
| 1 |
EC50 = 1160 nM
|
|
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CP0460135
|
2-(4-{2-[1-(2-Biphenyl-4-yl-ethyl)-3-(2,4-dimethoxy-phenyl)-ureido]-ethyl}-phenylsulfanyl)-2-methyl-propionic acid
Show/Hide
|
C35H38N2O5S
|
1
|
| 1 |
EC50 = 1200 nM
|
|
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CP0386004
|
2-[1-benzyl-6-[3-[3-[(4-methylphenyl)methoxy]phenoxy]propoxy]indol-3-yl]acetic acid
Show/Hide
|
C34H33NO5
|
1
|
| 1 |
EC50 = 1300 nM
|
|
|
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CP0406631
|
2-(4-{2-[1-(2-Biphenyl-4-yl-ethyl)-3-(2,4,5-trimethyl-phenyl)-ureido]-ethyl}-phenylsulfanyl)-2-methyl-propionic acid
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C36H40N2O3S
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1
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| 1 |
EC50 = 1350 nM
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CP0208934
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3-[4-[2-[1,3-benzoxazol-2-yl(methyl)amino]ethoxy]phenyl]-2-(2-benzoylphenyl)sulfanylpropanoic acid
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C32H28N2O5S
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1
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| 1 |
EC50 = 1380.38 nM
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CP0036481
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alkynyl ether, 27
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C32H31F3O6S
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1
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| 1 |
EC50 = 1400 nM
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CP0434129
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(S)-3-(4-(3-(benzylcarbamothioyloxy)propyl)phenyl)-2-ethoxypropanoic acid
Show/Hide
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C22H27NO4S
|
1
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| 1 |
EC50 = 1400 nM
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CP0400047
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(2S)-3-(4-(3-(benzylcarbamoyloxy)-3-phenylpropyl)phenyl)-2-ethoxypropanoic acid
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C28H31NO5
|
1
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| 1 |
EC50 = 1420 nM
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CP0208859
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alkynyl ether, 35
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C29H34O6S
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1
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| 1 |
EC50 = 1500 nM
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CP0403631
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2-(4-{2-[1-(5-Cyclohexyl-pentyl)-3-(4-fluoro-phenyl)-ureido]-ethyl}-phenoxy)-2-methyl-propionic acid
Show/Hide
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C30H41FN2O4
|
1
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| 1 |
EC50 = 1600 nM
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CP0086937
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alkynyl ether, 28
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C34H28F3NO5S
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1
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| 1 |
EC50 = 1600 nM
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CP0374136
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(S)-3-(3-((E)-1-(4-Methanesulfonyloxybenzyloxyimino)ethyl)phenyl)-2-ethoxypropanoicacid
Show/Hide
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C21H25NO7S
|
1
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| 1 |
EC50 = 1610 nM
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CP0051319
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3-(4-((R)-3-(4-ethyl-2-(thiophen-3-yl)phenoxy)butoxy)-2-methylphenyl)propanoic acid
Show/Hide
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C26H30O4S
|
1
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| 1 |
EC50 = 1670 nM
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CP0393544
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(2R)-2-benzyl-3-[4-propoxy-3-[[(4-pyridin-4-ylbenzoyl)amino]methyl]phenyl]propanoic acid
Show/Hide
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C32H32N2O4
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1
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| 1 |
EC50 = 1688 nM
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CP0448920
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2-[5-[3-[3-[(4-methylphenyl)methoxy]phenoxy]propoxy]-1H-indol-3-yl]acetic acid
Show/Hide
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C27H27NO5
|
1
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| 1 |
EC50 = 1700 nM
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CP0200308
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2-Methyl-2-{4-[2-(5-methyl-2-phenyl-oxazol-4-yl)-ethoxy]-phenoxy}-3-phenyl-propionic acid
Show/Hide
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C28H27NO5
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1
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| 1 |
EC50 = 1776 nM
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CP0049835
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2-[2-(benzenesulfonyl)anilino]-3-[4-[2-[1,3-benzoxazol-2-yl(methyl)amino]ethoxy]phenyl]propanoic acid
Show/Hide
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C31H29N3O6S
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1
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| 1 |
EC50 = 1819.7 nM
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CP0374134
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(S)-2-Ethoxy-3-(3-(4,5-dihydro-5-phenethylisoxazol-3-yl)phenyl)propanoic Acid
Show/Hide
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C22H25NO4
|
1
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| 1 |
EC50 = 1850 nM
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CP0461586
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2-methyl-2-[4-(2-{4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl}ethyl)phenoxy]propanoic acid
Show/Hide
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C23H22F3NO3S
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1
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| 1 |
EC50 = 1870 nM
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CP0489798
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(R)-3-(3-((E)-1-Benzyloxyiminoethyl)phenyl)-2-ethoxypropanoicAcid
Show/Hide
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C20H23NO4
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1
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| 1 |
EC50 = 1890 nM
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CP0385975
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2-[1-benzyl-5-[2-[3-[(4-methoxyphenyl)methoxy]phenoxy]ethoxy]indol-3-yl]acetic acid
Show/Hide
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C33H31NO6
|
1
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| 1 |
EC50 = 1900 nM
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CP0145397
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3-(4-((R)-3-(4-ethyl-2-(oxazol-4-yl)phenoxy)butoxy)-2-methylphenyl)propanoic acid
Show/Hide
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C25H29NO5
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1
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| 1 |
EC50 = 1980 nM
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CP0035359
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3-(4-((R)-3-(4-ethyl-2-(thiophen-2-yl)phenoxy)butoxy)-2-methylphenyl)propanoic acid
Show/Hide
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C26H30O4S
|
1
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| 1 |
EC50 = 1990 nM
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CP0460136
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2-(4-{2-[1-(4-Cyclohexyl-butyl)-3-(4-methyl-3-nitro-phenyl)-ureido]-ethyl}-phenylsulfanyl)-2-methyl-propionic acid
Show/Hide
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C30H41N3O5S
|
1
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| 1 |
EC50 = 2000 nM
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CP0465322
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2-(4-{2-[1-(2-Biphenyl-4-yl-ethyl)-3-(3,5-dichloro-phenyl)-ureido]-ethyl}-phenylsulfanyl)-2-methyl-propionic acid
Show/Hide
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C33H32Cl2N2O3S
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1
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| 1 |
EC50 = 2000 nM
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CP0083167
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4'-((1,4'-dimethyl-2'-propyl(2,6'-bi-1H-benzimidazol)-1'-yl)methyl)-(1,1'-biphenyl)-2-carboxylic acid
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C33H30N4O2
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1
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| 1 |
EC50 = 2020 nM
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CP0167306
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alkynyl ether, 22
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C32H31F3O6S
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1
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| 1 |
EC50 = 2200 nM
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CP0035353
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3-(4-((R)-3-(4-ethyl-2-(thiazol-2-yl)phenoxy)butoxy)-2-methylphenyl)propanoic acid
Show/Hide
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C25H29NO4S
|
1
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| 1 |
EC50 = 2270 nM
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CP0145396
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3-(4-((R)-3-(4-ethyl-2-(furan-2-yl)phenoxy)butoxy)-2-methylphenyl)propanoic acid
Show/Hide
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C26H30O5
|
1
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| 1 |
EC50 = 2300 nM
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CP0381165
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2-(4-{2-[1-(2-Biphenyl-4-yl-ethyl)-3-cyclohexyl-ureido]-ethyl}-phenylsulfanyl)-2-methyl-propionic acid
Show/Hide
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C33H40N2O3S
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1
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| 1 |
EC50 = 2400 nM
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CP0451513
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2-{4-[2-(5-Methyl-2-phenyl-oxazol-4-yl)-ethoxy]-benzyl}-2-phenoxy-hexanoic acid
Show/Hide
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C31H33NO5
|
1
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| 1 |
EC50 = 2507 nM
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CP0208706
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(2S)-2-azaniumyl-3-(4-phenylmethoxyphenyl)propanoate
Show/Hide
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C16H17NO3
|
1
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| 1 |
EC50 = 2511.89 nM
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CP0043419
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(S)-2-Methanesulfonylamino-3-{4-[2-(5-methyl-2-phenyl-oxazol-4-yl)-ethoxy]-phenyl}-propionic acid
Show/Hide
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C22H24N2O6S
|
1
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| 1 |
EC50 = 2600 nM
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CP0459247
|
2-[3-[2-[2-(4-Butylphenyl)-5-isopropyl-4-oxazolyl]ethyl]-1,2-benzisoxazol-6-yloxy]-2-methylpropionic acid
Show/Hide
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C29H34N2O5
|
1
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| 1 |
EC50 = 2600 nM
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CP0880191
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4'-((5-(1-phenylpropylcarbamoyl)-2-propyl-1H-benzo[d]imidazol-1-yl)methyl)biphenyl-2-carboxylic acid
Show/Hide
|
C34H33N3O3
|
1
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| 1 |
EC50 = 2650 nM
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CP0104575
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3-(2-((3-benzylureido)methyl)-4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)phenyl)propanoic acid
Show/Hide
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C30H31N3O5
|
1
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| 1 |
EC50 = 2684 nM
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CP0442661
|
(S)-2-Ethoxy-3-(3-(5-(4-(tert-butylphenyl)-4,5-dihydroisoxazol-3-yl)phenyl)propanoic Acid
Show/Hide
|
C24H29NO4
|
1
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| 1 |
EC50 = 2730 nM
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CP0374137
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(S)-3-(3-((E)-1-(4-Hydroxybenzyloxyimino)ethyl)phenyl)-2-ethoxypropanoicAcid
Show/Hide
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C20H23NO5
|
1
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| 1 |
EC50 = 2940 nM
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CP0322303
|
alkynyl ether, 10
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C27H23F3O5S
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1
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| 1 |
EC50 = 3000 nM
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CP0372751
|
2-methyl-5-[[4-[(5-methyl-2-phenyl-1,3-oxazol-4-yl)methyl]phenyl]methyl]-1,3-dioxane-2-carboxylic acid
Show/Hide
|
C24H25NO5
|
1
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| 1 |
EC50 = 3000 nM
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CP0015504
|
2-(4-{2-[(4-chlorophenyl)formamido]ethyl}phenoxy)-2-methylpropanoic acid
Show/Hide
|
C19H20ClNO4
|
3
|
| 1 |
EC50 = 3000 nM
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| 2 |
EC50 = 60000 nM
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| 3 |
EC50 = 100000 nM
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CP0467731
|
5-[4-[2-(4-ethylphenyl)-5-methyl-1,3-oxazol-4-yl]butyl]-2-methyl-1,3-dioxane-2-carboxylic acid
Show/Hide
|
C22H29NO5
|
1
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| 1 |
EC50 = 3000 nM
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CP0504506
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2-methyl-5-[4-[2-(4-methylphenyl)-5-(trifluoromethyl)-1,3-oxazol-4-yl]butyl]-1,3-dioxane-2-carboxylic acid
Show/Hide
|
C21H24F3NO5
|
1
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| 1 |
EC50 = 3000 nM
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CP0376473
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(2R)-2-benzyl-3-[4-propoxy-3-[[(4-pyrimidin-5-ylbenzoyl)amino]methyl]phenyl]propanoic acid
Show/Hide
|
C31H31N3O4
|
1
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| 1 |
EC50 = 3095 nM
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CP0374135
|
(S)-2-Ethoxy-3-(3-(5-(4-methoxyphenyl)-4,5-dihydroisoxazol-3-yl)phenyl)propanoic Acid
Show/Hide
|
C21H23NO5
|
1
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| 1 |
EC50 = 3190 nM
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CP0371988
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(S)-2-Ethoxy-3-(3-(5-phenylisoxazole-3-yl)phenyl)propanoic Acid
Show/Hide
|
C20H19NO4
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1
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| 1 |
EC50 = 3290 nM
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CP0086936
|
alkynyl ether, 25
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C31H29F3O6S
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1
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| 1 |
EC50 = 3300 nM
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CP0405641
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(2S)-2-ethoxy-3-(4-(3-phenyl-3-(propylcarbamothioyloxy)propyl)phenyl)propanoic acid
Show/Hide
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C24H31NO4S
|
1
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| 1 |
EC50 = 3480 nM
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CP0236912
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(S)-2-Acetylamino-3-{4-[2-(5-methyl-2-phenyl-oxazol-4-yl)-ethoxy]-phenyl}-propionic acid
Show/Hide
|
C23H24N2O5
|
1
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| 1 |
EC50 = 3500 nM
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CP0403096
|
(2S)-3-(4-(3-(butylcarbamothioyloxy)-3-phenylpropyl)phenyl)-2-ethoxypropanoic acid
Show/Hide
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C25H33NO4S
|
1
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| 1 |
EC50 = 3600 nM
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CP0039118
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2-{2-methyl-4-[({4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl}methyl)sulfanyl]phenoxy}acetic acid
Show/Hide
|
C21H18F3NO3S2
|
4
|
| 1 |
EC50 = 4100 nM
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| 2 |
EC50 = 8900 nM
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| 3 |
EC50 > 1200 nM
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| 4 |
EC50 > 1500 nM
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CP0086939
|
alkynyl ether, 30
Show/Hide
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C31H29F3O5S
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1
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| 1 |
EC50 = 4500 nM
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CP0374566
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(2S)-2-ethoxy-3-(4-(3-phenyl-3-(phenylcarbamothioyloxy)propyl)phenyl)propanoic acid
Show/Hide
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C27H29NO4S
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1
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| 1 |
EC50 = 4580 nM
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CP0292417
|
alkynyl ether, 19
Show/Hide
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C29H25F3O5S
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1
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| 1 |
EC50 = 4900 nM
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CP0163089
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(S)-2-Methylamino-3-{4-[2-(5-methyl-2-phenyl-oxazol-4-yl)-ethoxy]-phenyl}-propionic acid
Show/Hide
|
C22H24N2O4
|
1
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| 1 |
EC50 = 5000 nM
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CP0113991
|
2-[(2E)-3,7-dimethylocta-2,6-dienyl]-5-[(E)-2-[3-(trifluoromethyl)phenyl]ethenyl]benzene-1,3-diol
Show/Hide
|
C25H27F3O2
|
1
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| 1 |
EC50 = 5000 nM
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CP0123476
|
AMORPHASTILBOL
Show/Hide
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C24H28O2
|
1
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| 1 |
EC50 = 5000 nM
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CP0125657
|
2-[(2E)-3,7-dimethylocta-2,6-dienyl]-5-[(E)-2-(furan-3-yl)ethenyl]benzene-1,3-diol
Show/Hide
|
C22H26O3
|
1
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| 1 |
EC50 = 5000 nM
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CP0502910
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2-[3-[2-[4-Isopropyl-2-[4-(trifluoromethyl)phenyl]-5-thiazolyl]ethyl]-1,2-benzisoxazol-6-yloxy]-2-methylpropionic acid
Show/Hide
|
C26H25F3N2O4S
|
1
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| 1 |
EC50 = 5100 nM
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CP0374565
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(2S)-2-ethoxy-3-(4-(3-(ethylcarbamothioyloxy)-3-phenylpropyl)phenyl)propanoic acid
Show/Hide
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C23H29NO4S
|
1
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| 1 |
EC50 = 5390 nM
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CP0568375
|
(E)-6-[2-[[3-[4-(furan-2-yl)phenyl]-5-methyl-1H-pyrazol-4-yl]methyl]phenoxy]-4-methylhex-4-enoic acid
Show/Hide
|
C28H28N2O4
|
1
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| 1 |
EC50 = 5530 nM
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CP0086935
|
alkynyl ether, 23
Show/Hide
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C30H27F3O6S
|
1
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| 1 |
EC50 = 5900 nM
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CP0482215
|
2-[3-[2-[2-(2-Chlorophenyl)-5-hexyl-4-oxazolyl]ethyl]-1,2-benzisoxazol-6-yloxy]-2-methylpropionic acid
Show/Hide
|
C28H31ClN2O5
|
1
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| 1 |
EC50 = 5900 nM
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CP0133914
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2-[(2E)-3,7-dimethylocta-2,6-dienyl]-5-[(E)-2-thiophen-3-ylethenyl]benzene-1,3-diol
Show/Hide
|
C22H26O2S
|
1
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| 1 |
EC50 = 6000 nM
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CP0415749
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(S)-3-(3-(5-Benzyl-4,5-dihydroisoxazol-3-yl)phenyl)-2-ethoxypropanoicAcid
Show/Hide
|
C21H23NO4
|
1
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| 1 |
EC50 = 6930 nM
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CP0155180
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5-[(E)-2-(3,5-difluorophenyl)ethenyl]-2-[(2E)-3,7-dimethylocta-2,6-dienyl]benzene-1,3-diol
Show/Hide
|
C24H26F2O2
|
1
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| 1 |
EC50 = 7000 nM
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CP0406598
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(2S)-3-(4-(2-(benzylcarbamothioyloxy)-2-phenylethoxy)phenyl)-2-ethoxypropanoic acid
Show/Hide
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C27H29NO5S
|
1
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| 1 |
EC50 = 7170 nM
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CP0364879
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2-[(2E)-3,7-dimethylocta-2,6-dienyl]-5-[(E)-2-(4-hydroxyphenyl)ethenyl]benzene-1,3-diol
Show/Hide
|
C24H28O3
|
1
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| 1 |
EC50 = 8000 nM
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CP0372747
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(2s,5s)-2-methyl-5-(4-(5-methyl-2-p-tolyloxazol-4-yl)butyl)-1,3-dioxane-2-carboxylic acid
Show/Hide
|
C21H27NO5
|
1
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| 1 |
EC50 = 9600 nM
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CP0518415
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2-(4-{2-[1-(2-Biphenyl-4-yl-ethyl)-3-(2-methoxy-5-methyl-phenyl)-ureido]-ethyl}-phenylsulfanyl)-2-methyl-propionic acid
Show/Hide
|
C35H38N2O4S
|
1
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| 1 |
EC50 = 10000 nM
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CP0039791
|
phenoxyacetic acid-ether, 13
Show/Hide
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C29H26F3NO6S
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1
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| 1 |
EC50 > 10000 nM
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CP0086886
|
phenoxyacetic acid-ether, 14
Show/Hide
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C30H26F3NO5S
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1
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| 1 |
EC50 > 10000 nM
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CP0086887
|
phenoxyacetic acid-ether, 16
Show/Hide
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C29H29F3O6S
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1
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| 1 |
EC50 > 10000 nM
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CP0086888
|
phenoxyacetic acid-ether, 18
Show/Hide
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C30H32F3NO5S
|
1
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| 1 |
EC50 > 10000 nM
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CP0128464
|
alkynyl ether, 24
Show/Hide
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C31H29F3O6S
|
1
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| 1 |
EC50 > 10000 nM
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CP0146580
|
phenoxyacetic acid-ether, 15
Show/Hide
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C30H26F3NO5S
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1
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| 1 |
EC50 > 10000 nM
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CP0194611
|
phenoxyacetic acid-ether, 12
Show/Hide
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C26H22F3NO5S
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1
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| 1 |
EC50 > 10000 nM
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CP0201564
|
phenoxyacetic acid-ether, 9
Show/Hide
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C28H29F3O6S
|
1
|
| 1 |
EC50 > 10000 nM
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CP0275263
|
phenoxyacetic acid-ether, 17
Show/Hide
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C30H32F3NO6S
|
1
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| 1 |
EC50 > 10000 nM
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CP0276403
|
phenoxyacetic acid-ether, 11
Show/Hide
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C27H27F3O6S
|
1
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| 1 |
EC50 > 10000 nM
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CP0942100
|
N-(2-{4-[(2,4-dioxa-1,3-thiazolidine-5-yl)methyl]phenoxy}-ethyl)-5-(1,2-dithiolan-3-yl)pentanamide
Show/Hide
|
C20H26N2O4S3
|
1
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| 1 |
EC50 = 10000 nM
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CP0268622
|
2-methyl-2-phenoxypropanoic acid, 25a
Show/Hide
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C23H21F3N2O4S
|
1
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| 1 |
EC50 > 10000 nM
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CP0409204
|
2-methyl-2-phenoxypropanoic acid, 25c
Show/Hide
|
C23H21F3N2O5S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
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CP0409323
|
2-[2-methyl-4-(2-{4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl}ethyl)phenoxy]acetic acid
Show/Hide
|
C22H20F3NO3S
|
1
|
| 1 |
EC50 = 10000 nM
|
|
|
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CP0409324
|
2-[4-({[2-(4-aminophenyl)-4-methyl-1,3-thiazol-5-yl]formamido}methyl)phenoxy]-2-methylpropanoic acid
Show/Hide
|
C22H23N3O4S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
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CP0409325
|
2-methyl-2-phenoxypropanoic acid, 25l
Show/Hide
|
C23H24N2O7S2
|
1
|
| 1 |
EC50 > 10000 nM
|
|
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CP0409326
|
2-[4-({[2-(4-methoxyphenyl)-4-methyl-1,3-thiazol-5-yl]formamido}methyl)phenoxy]-2-methylpropanoic acid
Show/Hide
|
C23H24N2O5S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
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CP0409331
|
2-[4-({[2-(4-fluorophenyl)-4-methyl-1,3-thiazol-5-yl]formamido}methyl)phenoxy]-2-methylpropanoic acid
Show/Hide
|
C22H21FN2O4S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
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CP0409332
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2-[4-({[2-(4-chlorophenyl)-4-methyl-1,3-thiazol-5-yl]formamido}methyl)phenoxy]-2-methylpropanoic acid
Show/Hide
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C22H21ClN2O4S
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1
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| 1 |
EC50 > 10000 nM
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CP0409333
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2-methyl-2-phenoxypropanoic acid, 34
Show/Hide
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C23H21F3N2O4S
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1
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| 1 |
EC50 > 10000 nM
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CP0442419
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2-methyl-2-[4-({[4-methyl-2-(4-nitrophenyl)-1,3-thiazol-5-yl]formamido}methyl)phenoxy]propanoic acid
Show/Hide
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C22H21N3O6S
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1
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| 1 |
EC50 > 10000 nM
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CP0442420
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2-[4-({[2-(4-hydroxyphenyl)-4-methyl-1,3-thiazol-5-yl]formamido}methyl)phenoxy]-2-methylpropanoic acid
Show/Hide
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C22H22N2O5S
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1
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| 1 |
EC50 > 10000 nM
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CP0442421
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2-methyl-2-phenoxypropanoic acid, 27
Show/Hide
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C24H23F3N2O4S
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1
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| 1 |
EC50 > 10000 nM
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CP0445955
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2-methyl-2-(4-{[({4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl}methyl)amino]methyl}phenoxy)propanoic acid
Show/Hide
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C23H23F3N2O3S
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1
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| 1 |
EC50 > 10000 nM
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CP0453688
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2-methyl-2-phenoxypropanoic acid, 37
Show/Hide
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C24H23F3N2O4S
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1
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| 1 |
EC50 > 10000 nM
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CP0503895
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2-methyl-2-[4-({4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazole-5-}amido)phenoxy]propanoic acid
Show/Hide
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C22H19F3N2O4S
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1
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| 1 |
EC50 > 10000 nM
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CP0847204
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2-methyl-2-[4-{[(5-methyl-2-[4-trifluoromethylphenyl]-thiazol-4-ylcarbonyl)amino]methyl}phenoxy]propionic acid
Show/Hide
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C17H20N2O4S
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1
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| 1 |
EC50 > 10000 nM
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CP0938856
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2-methyl-2-[4-{[(4-methyl-2-phenylthiazol-5-ylcarbonyl)amino]-methyl}phenoxy]propionic acid
Show/Hide
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C21H20N2O4S
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1
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| 1 |
EC50 > 10000 nM
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CP0394931
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5-[4-(5-methyl-2-phenyl-1,3-oxazol-4-yl)butyl]-2-(2-methylpropyl)-1,3-dioxane-2-carboxylic acid
Show/Hide
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C23H31NO5
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1
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| 1 |
EC50 = 10000 nM
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CP0516059
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2-ethyl-5-[4-(5-methyl-2-phenyl-1,3-oxazol-4-yl)butyl]-1,3-dioxane-2-carboxylic acid
Show/Hide
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C21H27NO5
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1
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| 1 |
EC50 = 10000 nM
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CP0486795
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5-[4-[5-ethyl-2-(4-methylphenyl)-1,3-oxazol-4-yl]butyl]-2-methyl-1,3-dioxane-2-carboxylic acid
Show/Hide
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C22H29NO5
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1
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| 1 |
EC50 = 10000 nM
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CP0375119
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2-[3-[2-[2-(2,6-Dichlorophenyl)-5-isopropyl-4-oxazolyl]ethyl]-1,2-benzisoxazol-6-yloxy]-2-methylpropionic acid
Show/Hide
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C25H24Cl2N2O5
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1
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| 1 |
EC50 > 10000 nM
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CP0376052
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2-(3-(2-(2-(2,4-dichlorophenyl)-5-isopropyloxazol-4-yl)ethyl)-5-methylbenzo[d]isoxazol-6-yloxy)acetic acid
Show/Hide
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C24H22Cl2N2O5
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1
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| 1 |
EC50 > 10000 nM
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CP0390776
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2-[3-[2-[5-Isopropyl-2-[2-(trifluoromethyl)phenyl]-4-oxazolyl]ethyl]-1,2-benzisoxazol-6-yloxy]-2-methylpropionic acid
Show/Hide
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C26H25F3N2O5
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1
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| 1 |
EC50 > 10000 nM
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CP0482214
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2-[3-[2-[5-tert-Butyl-2-(2-chlorophenyl)-4-oxazolyl]ethyl]-1,2-benzisoxazol-6-yloxy]-2-methylpropionic acid
Show/Hide
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C26H27ClN2O5
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1
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| 1 |
EC50 > 10000 nM
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CP0134379
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2-[2-methyl-4-[1-[4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl]-2-phenylethyl]sulfanylphenoxy]acetic acid
Show/Hide
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C28H24F3NO3S2
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1
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| 1 |
EC50 > 10000 nM
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CP0385347
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2-[2-methyl-4-[1-[4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl]butylsulfanyl]phenoxy]acetic acid
Show/Hide
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C24H24F3NO3S2
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1
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| 1 |
EC50 > 10000 nM
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CP0410205
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2-[2-methyl-4-[1-[4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl]-2-(4-nitrophenyl)ethyl]sulfanylphenoxy]acetic acid
Show/Hide
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C28H23F3N2O5S2
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1
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| 1 |
EC50 > 10000 nM
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CP0410206
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2-[4-[2-(4-methoxyphenyl)-1-[4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl]ethyl]sulfanyl-2-methylphenoxy]acetic acid
Show/Hide
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C29H26F3NO4S2
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1
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| 1 |
EC50 > 10000 nM
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CP0410207
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2-[4-[2-(2,6-dichlorophenyl)-1-[4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl]ethyl]sulfanyl-2-methylphenoxy]acetic acid
Show/Hide
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C28H22Cl2F3NO3S2
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1
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| 1 |
EC50 > 10000 nM
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CP0410209
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2-[4-[2-anthracen-9-yl-1-[4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl]ethyl]sulfanyl-2-methylphenoxy]acetic acid
Show/Hide
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C36H28F3NO3S2
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1
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| 1 |
EC50 > 10000 nM
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CP0410219
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2-[2-methyl-4-[1-[4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl]-2-(2,3,4,5,6-pentafluorophenyl)ethyl]sulfanylphenoxy]acetic acid
Show/Hide
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C28H19F8NO3S2
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1
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| 1 |
EC50 > 10000 nM
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CP0410222
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2-[2-methyl-4-[1-[4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl]-6-phenylhexyl]sulfanylphenoxy]acetic acid
Show/Hide
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C32H32F3NO3S2
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1
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| 1 |
EC50 > 10000 nM
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CP0410223
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2-[2-methyl-4-[1-[4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl]-8-phenyloctyl]sulfanylphenoxy]acetic acid
Show/Hide
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C34H36F3NO3S2
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1
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| 1 |
EC50 > 10000 nM
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CP0410224
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2-[2-methyl-4-[1-[4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl]-2-(3,4,5-trifluorophenyl)ethyl]sulfanylphenoxy]acetic acid
Show/Hide
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C28H21F6NO3S2
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1
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| 1 |
EC50 > 10000 nM
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CP0416092
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2-[2-methyl-4-[1-[4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl]propylsulfanyl]phenoxy]acetic acid
Show/Hide
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C23H22F3NO3S2
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1
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| 1 |
EC50 > 10000 nM
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CP0416093
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2-[2-methyl-4-[1-[4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl]pentylsulfanyl]phenoxy]acetic acid
Show/Hide
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C25H26F3NO3S2
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1
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| 1 |
EC50 > 10000 nM
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CP0416104
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2-[2-methyl-4-[1-[4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl]-5-phenylpentyl]sulfanylphenoxy]acetic acid
Show/Hide
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C31H30F3NO3S2
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1
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| 1 |
EC50 > 10000 nM
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CP0416105
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2-[4-[2-(2,5-difluorophenyl)-1-[4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl]ethyl]sulfanyl-2-methylphenoxy]acetic acid
Show/Hide
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C28H22F5NO3S2
|
1
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| 1 |
EC50 > 10000 nM
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CP0420883
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2-[2-methyl-4-[1-[4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl]-2-[4-(trifluoromethyl)phenyl]ethyl]sulfanylphenoxy]acetic acid
Show/Hide
|
C29H23F6NO3S2
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1
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| 1 |
EC50 > 10000 nM
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|
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CP0420884
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2-[2-methyl-4-[1-[4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl]-11-phenylundecyl]sulfanylphenoxy]acetic acid
Show/Hide
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C37H42F3NO3S2
|
1
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| 1 |
EC50 > 10000 nM
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CP0432336
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2-[4-[2-cyclopropyl-1-[4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl]ethyl]sulfanyl-2-methylphenoxy]acetic acid
Show/Hide
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C25H24F3NO3S2
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1
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| 1 |
EC50 > 10000 nM
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CP0432345
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2-[2-methyl-4-[1-[4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl]-4-phenylbutyl]sulfanylphenoxy]acetic acid
Show/Hide
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C30H28F3NO3S2
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1
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| 1 |
EC50 > 10000 nM
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CP0447734
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2-[4-[2-[2-fluoro-6-(trifluoromethyl)phenyl]-1-[4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl]ethyl]sulfanyl-2-methylphenoxy]acetic acid
Show/Hide
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C29H22F7NO3S2
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1
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| 1 |
EC50 > 10000 nM
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CP0447760
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2-[2-methyl-4-[1-[4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl]-2,2-diphenylethyl]sulfanylphenoxy]acetic acid
Show/Hide
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C34H28F3NO3S2
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1
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| 1 |
EC50 > 10000 nM
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CP0450700
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2-[4-[2-(2,6-difluorophenyl)-1-[4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl]ethyl]sulfanyl-2-methylphenoxy]acetic acid
Show/Hide
|
C28H22F5NO3S2
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1
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| 1 |
EC50 > 10000 nM
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CP0454766
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2-[2-methyl-4-[3-methyl-1-[4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl]butyl]sulfanylphenoxy]acetic acid
Show/Hide
|
C25H26F3NO3S2
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1
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| 1 |
EC50 > 10000 nM
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CP0454767
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2-[2-methyl-4-[1-[4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl]-2-(4-phenylphenyl)ethyl]sulfanylphenoxy]acetic acid
Show/Hide
|
C34H28F3NO3S2
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1
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| 1 |
EC50 > 10000 nM
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CP0454802
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2-[2-methyl-4-[1-[4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl]-3-phenylpropyl]sulfanylphenoxy]acetic acid
Show/Hide
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C29H26F3NO3S2
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1
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| 1 |
EC50 > 10000 nM
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CP0495380
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2-[2-methyl-4-[1-[4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl]-2-naphthalen-1-ylethyl]sulfanylphenoxy]acetic acid
Show/Hide
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C32H26F3NO3S2
|
1
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| 1 |
EC50 > 10000 nM
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CP0495382
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2-[4-[2-(2-chloro-6-fluorophenyl)-1-[4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl]ethyl]sulfanyl-2-methylphenoxy]acetic acid
Show/Hide
|
C28H22ClF4NO3S2
|
1
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| 1 |
EC50 > 10000 nM
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CP0548509
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2-[4-[2-(2,4-difluorophenyl)-1-[4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl]ethyl]sulfanyl-2-methylphenoxy]acetic acid
Show/Hide
|
C28H22F5NO3S2
|
1
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| 1 |
EC50 > 10000 nM
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CP0062441
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(E)-6-[2-[[[4-(furan-2-yl)benzoyl]-methylamino]methyl]phenoxy]-4-methylhex-4-enoic acid
Show/Hide
|
C26H27NO5
|
1
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| 1 |
EC50 > 10000 nM
|
|
|
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CP0365610
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2-[2-methyl-4-[2-phenyl-1-[4-[4-(trifluoromethyl)phenyl]phenyl]ethyl]sulfanylphenoxy]acetic acid
Show/Hide
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C30H25F3O3S
|
1
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| 1 |
EC50 > 10000 nM
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|
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CP0396626
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2-[4-[2-(2-chloro-6-fluorophenyl)-1-[4-(3,4,5-trifluorophenyl)phenyl]ethyl]sulfanyl-2-methylphenoxy]acetic acid
Show/Hide
|
C29H21ClF4O3S
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1
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| 1 |
EC50 > 10000 nM
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CP0396627
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2-[2-methyl-4-[1-[4-[3-(trifluoromethyl)phenyl]phenyl]-2-(3,4,5-trifluorophenyl)ethyl]sulfanylphenoxy]acetic acid
Show/Hide
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C30H22F6O3S
|
1
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| 1 |
EC50 > 10000 nM
|
|
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CP0396628
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2-[2-methyl-4-[2-phenyl-1-[4-(3,4,5-trifluorophenyl)phenyl]ethyl]sulfanylphenoxy]acetic acid
Show/Hide
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C29H23F3O3S
|
1
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| 1 |
EC50 > 10000 nM
|
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CP0396629
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2-[4-[2-(2,6-difluorophenyl)-1-[4-[3-(trifluoromethyl)phenyl]phenyl]ethyl]sulfanyl-2-methylphenoxy]acetic acid
Show/Hide
|
C30H23F5O3S
|
1
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| 1 |
EC50 > 10000 nM
|
|
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CP0396630
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2-[4-[2-(2,6-difluorophenyl)-1-[4-(4-fluorophenyl)phenyl]ethyl]sulfanyl-2-methylphenoxy]acetic acid
Show/Hide
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C29H23F3O3S
|
1
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| 1 |
EC50 > 10000 nM
|
|
|
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CP0404373
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2-[4-[2-(2-chloro-6-fluorophenyl)-1-[4-(4-fluorophenyl)phenyl]ethyl]sulfanyl-2-methylphenoxy]acetic acid
Show/Hide
|
C29H23ClF2O3S
|
1
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| 1 |
EC50 > 10000 nM
|
|
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CP0415611
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2-[4-[2-(2,6-difluorophenyl)-1-[4-(3,4,5-trifluorophenyl)phenyl]ethyl]sulfanyl-2-methylphenoxy]acetic acid
Show/Hide
|
C29H21F5O3S
|
1
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| 1 |
EC50 > 10000 nM
|
|
|
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CP0415613
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2-[4-[2-(2-chloro-6-fluorophenyl)-1-[4-[3-(trifluoromethyl)phenyl]phenyl]ethyl]sulfanyl-2-methylphenoxy]acetic acid
Show/Hide
|
C30H23ClF4O3S
|
1
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| 1 |
EC50 > 10000 nM
|
|
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CP0415614
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2-[4-[1-[4-(4-fluorophenyl)phenyl]-2-phenylethyl]sulfanyl-2-methylphenoxy]acetic acid
Show/Hide
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C29H25FO3S
|
1
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| 1 |
EC50 > 10000 nM
|
|
|
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CP0415615
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2-[4-[1-[4-(4-fluorophenyl)phenyl]-2-(3,4,5-trifluorophenyl)ethyl]sulfanyl-2-methylphenoxy]acetic acid
Show/Hide
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C29H22F4O3S
|
1
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| 1 |
EC50 > 10000 nM
|
|
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CP0415617
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2-[2-methyl-4-[2-phenyl-1-[4-[3-(trifluoromethyl)phenyl]phenyl]ethyl]sulfanylphenoxy]acetic acid
Show/Hide
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C30H25F3O3S
|
1
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| 1 |
EC50 > 10000 nM
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|
|
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CP0415618
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2-[4-[2-(2,6-dichlorophenyl)-1-[4-(3,4,5-trifluorophenyl)phenyl]ethyl]sulfanyl-2-methylphenoxy]acetic acid
Show/Hide
|
C29H21Cl2F3O3S
|
1
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| 1 |
EC50 > 10000 nM
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|
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CP0415619
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2-[4-[2-(2-chloro-6-fluorophenyl)-1-(4-phenylphenyl)ethyl]sulfanyl-2-methylphenoxy]acetic acid
Show/Hide
|
C29H24ClFO3S
|
1
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| 1 |
EC50 > 10000 nM
|
|
|
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CP0455775
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2-[2-methyl-4-[1-(4-phenylphenyl)-2-(3,4,5-trifluorophenyl)ethyl]sulfanylphenoxy]acetic acid
Show/Hide
|
C29H23F3O3S
|
1
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| 1 |
EC50 > 10000 nM
|
|
|
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CP0455776
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2-[2-methyl-4-[1-[6-[4-(trifluoromethyl)phenyl]pyridin-3-yl]-2-(3,4,5-trifluorophenyl)ethyl]sulfanylphenoxy]acetic acid
Show/Hide
|
C29H21F6NO3S
|
1
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| 1 |
EC50 > 10000 nM
|
|
|
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CP0466247
|
2-[2-methyl-4-[2-phenyl-1-[6-[4-(trifluoromethyl)phenyl]pyridin-3-yl]ethyl]sulfanylphenoxy]acetic acid
Show/Hide
|
C29H24F3NO3S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
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CP0471906
|
2-[4-[2-[2-fluoro-6-(trifluoromethyl)phenyl]-1-[4-[3-(trifluoromethyl)phenyl]phenyl]ethyl]sulfanyl-2-methylphenoxy]acetic acid
Show/Hide
|
C31H23F7O3S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
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CP0492681
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2-[4-[2-[2-fluoro-6-(trifluoromethyl)phenyl]-1-(4-phenylphenyl)ethyl]sulfanyl-2-methylphenoxy]acetic acid
Show/Hide
|
C30H24F4O3S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
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CP0549063
|
2-[4-[1-[4-(4-fluorophenyl)phenyl]-2-[2-fluoro-6-(trifluoromethyl)phenyl]ethyl]sulfanyl-2-methylphenoxy]acetic acid
Show/Hide
|
C30H23F5O3S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
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CP0421004
|
(3R)-3-methyl-6-[2-[[5-methyl-2-[4-(trifluoromethoxy)phenyl]imidazol-1-yl]methyl]phenoxy]hexanoic acid
Show/Hide
|
C25H27F3N2O4
|
1
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| 1 |
EC50 > 10000 nM
|
|
|
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CP0444762
|
(E)-6-[2-[[3-[4-(furan-2-yl)phenyl]-5-methyl-1,2-oxazol-4-yl]methyl]phenoxy]-4-methylhex-4-enoic acid
Show/Hide
|
C28H27NO5
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
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CP0444890
|
(E)-6-[2-[[3-[4-(furan-2-yl)phenyl]-5-methylimidazol-4-yl]methyl]phenoxy]-4-methylhex-4-enoic acid
Show/Hide
|
C28H28N2O4
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
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CP0444891
|
(3R)-6-[2-[[2-(4-chloro-3-fluorophenyl)-5-methylimidazol-1-yl]methyl]phenoxy]-3-methylhexanoic acid
Show/Hide
|
C24H26ClFN2O3
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
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CP0444892
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6-[2-[[2-[4-(furan-2-yl)phenyl]-5-methylimidazol-1-yl]methyl]phenoxy]hexanoic acid
Show/Hide
|
C27H28N2O4
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
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CP0444893
|
(E)-6-[2-[[2-[4-(furan-2-yl)phenyl]-5-methylimidazol-1-yl]methyl]phenoxy]-4-methylhex-4-enoic acid
Show/Hide
|
C28H28N2O4
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
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CP0451331
|
US10399958, Compound 2e
Show/Hide
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C25H25F3N2O4
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
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CP0451332
|
6-[2-[[2-[4-(furan-2-yl)phenyl]-5-methylimidazol-1-yl]methyl]phenoxy]-2,2-dimethylhexanoic acid
Show/Hide
|
C29H32N2O4
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0527649
|
(3R)-6-[2-[[2-[4-(difluoromethoxy)phenyl]-5-methylimidazol-1-yl]methyl]phenoxy]-3-methylhexanoic acid
Show/Hide
|
C25H28F2N2O4
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0527650
|
(E)-6-[2-[[5-[4-(furan-2-yl)phenyl]-3-methylimidazol-4-yl]methyl]phenoxy]-4-methylhex-4-enoic acid
Show/Hide
|
C28H28N2O4
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
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CP0527651
|
(3R)-3-methyl-6-[2-[[5-methyl-2-(4-methylphenyl)imidazol-1-yl]methyl]phenoxy]hexanoic acid
Show/Hide
|
C25H30N2O3
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0527652
|
(3R)-6-[2-[[2-(4-chlorophenyl)-5-methylimidazol-1-yl]methyl]phenoxy]-3-methylhexanoic acid
Show/Hide
|
C24H27ClN2O3
|
1
|
| 1 |
EC50 > 10000 nM
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|
|
|
CP0549452
|
(3R)-6-[2-[[2-(4-fluorophenyl)-5-methylimidazol-1-yl]methyl]phenoxy]-3-methylhexanoic acid
Show/Hide
|
C24H27FN2O3
|
1
|
| 1 |
EC50 > 10000 nM
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|
|
|
CP0549453
|
(E)-6-[2-[[4-[4-(furan-2-yl)phenyl]-2-methyl-1,3-thiazol-5-yl]methyl]phenoxy]-4-methylhex-4-enoic acid
Show/Hide
|
C28H27NO4S
|
1
|
| 1 |
EC50 > 10000 nM
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|
|
|
CP0549476
|
(3R)-6-[2-[[2-[4-(furan-2-yl)phenyl]-5-methylimidazol-1-yl]methyl]phenoxy]-3-methylhexanoic acid
Show/Hide
|
C28H30N2O4
|
1
|
| 1 |
EC50 > 10000 nM
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|
|
|
CP0557787
|
(E)-6-[2-[[3-[4-(furan-2-yl)phenyl]-5-methyltriazol-4-yl]methyl]phenoxy]-4-methylhex-4-enoic acid
Show/Hide
|
C27H27N3O4
|
1
|
| 1 |
EC50 > 10000 nM
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|
|
|
CP0450935
|
2-[4-[3-[4-[(3-methoxyphenyl)methyl]-1-[(4-methylphenyl)methyl]-5-oxo-1,2,4-triazol-3-yl]propyl]phenoxy]-2-methylpropanoic acid
Show/Hide
|
C31H35N3O5
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0450936
|
2-[4-[3-[4-[(4-chlorophenyl)methyl]-1-[(4-methylphenyl)methyl]-5-oxo-1,2,4-triazol-3-yl]propyl]phenoxy]-2-methylpropanoic acid
Show/Hide
|
C30H32ClN3O4
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0450937
|
2-[4-[3-[1-[(4-ethenylphenyl)methyl]-4-[(4-methylphenyl)methyl]-5-oxo-1,2,4-triazol-3-yl]propyl]phenoxy]-2-methylpropanoic acid
Show/Hide
|
C32H35N3O4
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0450938
|
2-[4-[3-[4-[(4-methoxyphenyl)methyl]-1-[(4-methylphenyl)methyl]-5-oxo-1,2,4-triazol-3-yl]propyl]phenoxy]-2-methylpropanoic acid
Show/Hide
|
C31H35N3O5
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0538367
|
2-[4-[3-[1,4-bis[(4-methylphenyl)methyl]-5-oxo-1,2,4-triazol-3-yl]propyl]phenoxy]-2-methylpropanoic acid
Show/Hide
|
C31H35N3O4
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0538368
|
2-methyl-2-[4-[3-[1-[(4-methylphenyl)methyl]-5-oxo-4-[(3,4,5-trimethoxyphenyl)methyl]-1,2,4-triazol-3-yl]propyl]phenoxy]propanoic acid
Show/Hide
|
C33H39N3O7
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0551890
|
2-[4-[3-[4-benzyl-1-[(4-methylphenyl)methyl]-5-oxo-1,2,4-triazol-3-yl]propyl]phenoxy]-2-methylpropanoic acid
Show/Hide
|
C30H33N3O4
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0568641
|
2-[4-[3-[4-[(4-fluorophenyl)methyl]-1-[(4-methylphenyl)methyl]-5-oxo-1,2,4-triazol-3-yl]propyl]phenoxy]-2-methylpropanoic acid
Show/Hide
|
C30H32FN3O4
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0777387
|
(S)-2-(2-Benzoyl-cyclohex-1-enylamino)-3-(4-benzyloxy-phenyl)-propionic acid
Show/Hide
|
C29H29NO4
|
1
|
| 1 |
EC50 = 10232.93 nM
|
|
|
|
CP0125654
|
2-[(2E)-3,7-dimethylocta-2,6-dienyl]-5-[(E)-2-(4-fluorophenyl)ethenyl]benzene-1,3-diol
Show/Hide
|
C24H27FO2
|
1
|
| 1 |
EC50 = 11000 nM
|
|
|
|
CP0845746
|
5-[(4-{2-[5-(1,2-Dithiolan-3-yl)pentylmethylamino]ethoxy}-phenyl)methyl]-1,3-thiazolidine-2,4-dione tartarate
Show/Hide
|
C24H34N2O9S3
|
1
|
| 1 |
EC50 = 11050 nM
|
|
|
|
CP0846915
|
5-[(4-{2-[5-(1,2-dithiolan-3-yl)pentylmethylamino]ethoxy}-phenyl)methyl]-1,3-thiazolidine-2,4-dione hydrochloride
Show/Hide
|
C20H29ClN2O3S3
|
1
|
| 1 |
EC50 = 11050 nM
|
|
|
|
CP0499697
|
2-[3-chloro-4-[3-[5-(dithiolan-3-yl)pentanoyl-methylamino]propoxy]phenyl]acetic acid
Show/Hide
|
C20H28ClNO4S2
|
1
|
| 1 |
EC50 = 12300 nM
|
|
|
|
CP0188635
|
2-[(2E)-3,7-dimethylocta-2,6-dienyl]-5-[(E)-2-(4-methoxyphenyl)ethenyl]benzene-1,3-diol
Show/Hide
|
C25H30O3
|
1
|
| 1 |
EC50 = 14000 nM
|
|
|
|
CP0505001
|
2-[3-[2-[2-(2-Hydroxyphenyl)-5-isopropyl-4-oxazolyl]ethyl]-1,2-benzisoxazol-6-yloxy]-2-methylpropionic acid
Show/Hide
|
C25H26N2O6
|
1
|
| 1 |
EC50 = 14600 nM
|
|
|
|
CP0114689
|
(2S)-2-(2-benzoylanilino)-3-(4-phenylmethoxyphenyl)propanoic acid
Show/Hide
|
C29H25NO4
|
1
|
| 1 |
EC50 = 16595.87 nM
|
|
|
|
CP0376410
|
methyl 2-[3-chloro-4-[3-[5-(dithiolan-3-yl)pentanoyl-methylamino]propoxy]phenyl]acetate
Show/Hide
|
C21H30ClNO4S2
|
1
|
| 1 |
EC50 = 18490 nM
|
|
|
|
CP0441423
|
2-[3-[2-[2-Phenyl-5-propyl-4-oxazolyl]ethyl]-1,2-benzisoxazol-6-yloxy]-2-methylpropionic acid
Show/Hide
|
C25H26N2O5
|
1
|
| 1 |
EC50 = 19100 nM
|
|
|
|
CP0390775
|
2-[3-[2-[5-Methyl-2-phenyl-4-oxazolyl]ethyl]-1,2-benzisoxazol-6-yloxy]-2-methylpropionic acid
Show/Hide
|
C23H22N2O5
|
1
|
| 1 |
EC50 = 20800 nM
|
|
|
|
CP0037303
|
ADD-3878
Show/Hide
|
C18H23NO3S
|
1
|
| 1 |
EC50 = 22908.68 nM
|
|
|
|
CP0409330
|
2-methyl-2-phenoxypropanoic acid, 25i
Show/Hide
|
C23H21F3N2O4S
|
1
|
| 1 |
EC50 > 25000 nM
|
|
|
|
CP0445956
|
2-methyl-2-phenoxypropanoic acid, 25j
Show/Hide
|
C23H21F3N2O4S
|
1
|
| 1 |
EC50 > 25000 nM
|
|
|
|
CP0378649
|
(R)-2-Ethoxy-3-(3-(4,5-dihydro-5-phenethylisoxazol-3-yl)phenyl-)propanoic Acid
Show/Hide
|
C22H25NO4
|
1
|
| 1 |
EC50 = 25100 nM
|
|
|
|
CP0482211
|
2-[3-[2-[5-Ethyl-2-phenyl-4-oxazolyl]ethyl]-1,2-benzisoxazol-6-yloxy]-2-methylpropionic acid
Show/Hide
|
C24H24N2O5
|
1
|
| 1 |
EC50 = 25100 nM
|
|
|
|
CP0415748
|
(R)-2-Ethoxy-3-(3-(4,5-dihydro-5-phenylisoxazole-3-yl)phenyl-)propanoic Acid
Show/Hide
|
C20H21NO4
|
1
|
| 1 |
EC50 = 25400 nM
|
|
|
|
CP0459248
|
2-[3-[2-[2-(2,4-Dichlorophenyl)-5-isopropyl-4-oxazolyl]ethyl]-1,2-benzisoxazol-6-yloxy]-2-methylpropionic acid
Show/Hide
|
C25H24Cl2N2O5
|
1
|
| 1 |
EC50 = 26300 nM
|
|
|
|
CP0376049
|
2-[3-[2-[2-(2-Chlorophenyl)-5-propyl-4-oxazolyl]ethyl]-1,2-benzisoxazol-6-yloxy]-2-methylpropionic acid
Show/Hide
|
C25H25ClN2O5
|
1
|
| 1 |
EC50 = 26400 nM
|
|
|
|
CP0917983
|
5-[(4-{2-[5-(1,2-dithiolan-3-yl)pentylmethylamino]ethoxy}-phenyl)methyl]-1,3-thiazolidine-2,4-dione
Show/Hide
|
C20H28N2O3S3
|
1
|
| 1 |
EC50 = 28000 nM
|
|
|
|
CP0378651
|
(S)-2-Ethoxy-3-(3-(5-(4-methanesulfonyloxyphenyl)-4,5-dihydroisoxazol-3-yl)phenyl)propanoic Acid
Show/Hide
|
C21H23NO7S
|
1
|
| 1 |
EC50 = 28100 nM
|
|
|
|
CP0444307
|
2-methyl-5-[4-(5-methyl-2-phenyl-1,3-oxazol-4-yl)butyl]-1,3-dioxane-2-carboxylic acid
Show/Hide
|
C20H25NO5
|
1
|
| 1 |
EC50 = 30000 nM
|
|
|
|
CP0376050
|
2-[3-[2-[2-(2-Chlorophenyl)-5-isopropyl-4-oxazolyl]ethyl]-1,2-benzisoxazol-6-yloxy]-2-methylpropionic acid
Show/Hide
|
C25H25ClN2O5
|
1
|
| 1 |
EC50 = 31100 nM
|
|
|
|
CP0495628
|
(R)-2-Ethoxy-3-(3-(5-phenylisoxazole-3-yl)phenyl)propanoic Acid
Show/Hide
|
C20H19NO4
|
1
|
| 1 |
EC50 = 37400 nM
|
|
|
|
CP0415750
|
(S)-2-Ethoxy-3-(3-(5-(4-hydroxyphenyl)-4,5-dihydroisoxazol-3-yl)phenyl)propanoic Acid
Show/Hide
|
C20H21NO5
|
1
|
| 1 |
EC50 = 38600 nM
|
|
|
|
CP0433389
|
(R)-3-(3-(5-Benzyl-4,5-dihydroisoxazol-3-yl)phenyl)-2-ethoxypropanoicAcid
Show/Hide
|
C21H23NO4
|
1
|
| 1 |
EC50 = 41400 nM
|
|
|
|
CP0042877
|
2-(4-(4-Chlorobenzoyl)phenoxy)-2-methylpropionic acid
Show/Hide
|
C17H15ClO4
|
2
|
| 1 |
EC50 > 100000 nM
|
|
|
| 2 |
EC50 = 100000 nM
|
|
|
|
CP0422670
|
2-methyl-5-[4-(5-methyl-2-phenyl-1,3-oxazol-4-yl)butyl]-1,3-dioxane-2-carboxylic acid
Show/Hide
|
C20H25NO5
|
1
|
| 1 |
EC50 = 100000 nM
|
|
|
|
CP0420999
|
(3R)-3-methyl-6-[2-[[5-(trifluoromethyl)-2-[4-(trifluoromethyl)phenyl]imidazol-1-yl]methyl]phenoxy]hexanoic acid
Show/Hide
|
C25H24F6N2O3
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0421003
|
(3R)-6-[2-[[2-(4-cyanophenyl)-5-(trifluoromethyl)imidazol-1-yl]methyl]phenoxy]-3-methylhexanoic acid
Show/Hide
|
C25H24F3N3O3
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0517564
|
(3R)-6-[2-[[5-chloro-2-[4-(trifluoromethyl)phenyl]imidazol-1-yl]methyl]phenoxy]-3-methylhexanoic acid
Show/Hide
|
C24H24ClF3N2O3
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0054286
|
2-(2-methyl-4-((4-methyl-2-(4-(trifluoromethyl)phenyl)thiazol-5-yl)methylselanyl)phenoxy)acetic acid
Show/Hide
|
C21H18F3NO3SSe
|
1
|
| 1 |
EC50 > 1000 nM
|
|
|
|
CP0381218
|
2-(2-methyl-4-((4-methyl-2-(4-(trifluoromethyl)phenyl)thiazol-5-yl)methylselanyl)phenoxy)propanoic acid
Show/Hide
|
C22H20F3NO3SSe
|
1
|
| 1 |
EC50 > 1000 nM
|
|
|
|
CP0437343
|
2-(2-methyl-4-((4-methyl-2-(4-(trifluoromethyl)phenyl)thiazol-5-yl)methylselanyl)phenoxy)butanoic acid
Show/Hide
|
C23H22F3NO3SSe
|
1
|
| 1 |
EC50 > 1000 nM
|
|
|
|
CP0437344
|
2-(4-((2-(3-fluoro-4-(trifluoromethyl)phenyl)-4-methylthiazol-5-yl)methylselanyl)-2-methylphenoxy)propanoic acid
Show/Hide
|
C22H19F4NO3SSe
|
1
|
| 1 |
EC50 > 1000 nM
|
|
|
|
CP0498362
|
2-(4-((2-(3-fluoro-4-(trifluoromethyl)phenyl)-4-methylthiazol-5-yl)methylselanyl)-2-methylphenoxy)acetic acid
Show/Hide
|
C21H17F4NO3SSe
|
1
|
| 1 |
EC50 > 1000 nM
|
|
|
|
CP0040604
|
2-[4-[3-[[(2S)-2-(2-benzoylanilino)-3-[4-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]propyl]amino]-3-oxopropyl]phenyl]sulfanyl-2-methylpropanoic acid
Show/Hide
|
C47H47N3O6S
|
2
|
| 1 |
EC50 < 10000 nM
|
|
|
| 2 |
IC50 = 1995.26 nM
|
|
|
|
CP0145160
|
4-[[(2S)-2-(2-benzoylanilino)-3-[4-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]propyl]amino]-2-methyl-4-oxobutanoic acid
Show/Hide
|
C39H39N3O6
|
2
|
| 1 |
EC50 < 10000 nM
|
|
|
| 2 |
IC50 = 1000 nM
|
|
|
|
CP0146855
|
N-[(2S)-2-(2-benzoylanilino)-3-[4-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]propyl]-3-[2-(dimethylamino)ethoxy]benzamide
Show/Hide
|
C45H46N4O5
|
2
|
| 1 |
EC50 < 10000 nM
|
|
|
| 2 |
IC50 = 6309.57 nM
|
|
|
|
CP0256084
|
2-(3-aminophenoxy)-N-[(2S)-2-(2-benzoylanilino)-3-[4-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]propyl]acetamide
Show/Hide
|
C42H40N4O5
|
2
|
| 1 |
EC50 < 10000 nM
|
|
|
| 2 |
IC50 = 6309.57 nM
|
|
|
|
CP0673789
|
2-(4-(2-chloro-4-((4-(trifluoromethyl)phenoxy)methyl)phenylthio)-5,6,7,8-tetrahydronaphthalen-1-yloxy)acetic acid
Show/Hide
|
C26H22ClF3O4S
|
1
|
| 1 |
Ki = 460 nM
|
|
|
