| Compound ID |
Compound Name |
Compound Formula |
|
CP0041416
|
(6alpha)-17-(Acetyloxy)-6-methylpreg-4-ene-3,20-dione
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|
C24H34O4
|
2
|
| 1 |
EC50 = 0.15 nM
|
|
|
| 2 |
IC50 < 10000 nM
|
|
|
|
CP0351334
|
(6S,8S,10R,14S,15S)-17-Acetyl-6,10-dimethyl-13-(R)-methyl-17-(2-oxo-propyl)-1,2,6,7,8,9,10,11,12,13,14,15,16,17-tetradecahydro-cyclopenta[a]phenanthren-3-one
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|
C25H36O3
|
1
|
| 1 |
EC50 = 0.15 nM
|
|
|
|
CP0035186
|
(10S,11S,14S,15S,17R)-17-[4-(dimethylamino)phenyl]-14-hydroxy-15-methyl-14-(prop-1-yn-1-yl)tetracyclo[8.7.0.0^{2,7}.0^{11,15}]heptadeca-1,6-dien-5-one
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|
C29H35NO2
|
7
|
| 1 |
EC50 = 0.3 nM
|
|
|
| 2 |
EC50 > 10000 nM
|
|
|
| 3 |
IC50 = 0.18 nM
|
|
|
| 4 |
IC50 = 0.2512 nM
|
|
|
| 5 |
IC50 = 0.3 nM
|
|
|
| 6 |
IC50 = 0.6 nM
|
|
|
| 7 |
Ki = 0.2512 nM
|
|
|
|
CP0197932
|
(S)-2-chloro-4-((2-chlorobenzyl)(1-(cyanomethyl)pyrrolidin-3-yl)amino)benzonitrile
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|
C20H18Cl2N4
|
1
|
| 1 |
EC50 = 0.5 nM
|
|
|
|
CP0088155
|
9-Fluoro-2,2,4-trimethyl-5-[1-thiophen-3-yl-meth-(Z)-ylidene]-2,5-dihydro-1H-6-oxa-1-aza-chrysene
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|
C24H20FNOS
|
1
|
| 1 |
EC50 = 0.71 nM
|
|
|
|
CP0284048
|
4-chloro-13-(2-chlorophenyl)-6-methyl-11-oxo-8-thia-3,10-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5-tetraene-5-carbonitrile
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|
C18H11Cl2N3OS
|
1
|
| 1 |
EC50 = 0.7943 nM
|
|
|
|
CP0185600
|
9-Fluoro-5-[1-(2-methoxy-phenyl)-meth-(Z)-ylidene]-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
|
C27H24FNO2
|
1
|
| 1 |
EC50 = 0.93 nM
|
|
|
|
CP0063848
|
7-Fluoro-2,2,4-trimethyl-5-[1-o-tolyl-meth-(Z)-ylidene]-2,5-dihydro-1H-6-oxa-1-aza-chrysene
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|
C27H24FNO
|
1
|
| 1 |
EC50 = 1.4 nM
|
|
|
|
CP0038813
|
(1S,2R,10S,11S,14S,15S)-14-acetyl-2,15-dimethyltetracyclo[8.7.0.0^{2,7}.0^{11,15}]heptadec-6-en-5-one
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|
C21H30O2
|
7
|
| 1 |
EC50 = 1.5 nM
|
|
|
| 2 |
EC50 = 2.89 nM
|
|
|
| 3 |
EC50 = 2.9 nM
|
|
|
| 4 |
EC50 = 15.2 nM
|
|
|
| 5 |
IC50 > 10000 nM
|
|
|
| 6 |
IC50 < 10000 nM
|
|
|
| 7 |
Ki = 3.8 nM
|
|
|
|
CP0294954
|
(S)-2-chloro-4-((2-chlorobenzyl)(1-methylpyrrolidin-3-yl)amino)benzonitrile
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|
C19H19Cl2N3
|
1
|
| 1 |
EC50 = 1.6 nM
|
|
|
|
CP0207627
|
9-Fluoro-2,2,4-trimethyl-5-((Z)-3-methyl-but-2-enylidene)-2,5-dihydro-1H-6-oxa-1-aza-chrysene
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|
C24H24FNO
|
1
|
| 1 |
EC50 = 1.7 nM
|
|
|
|
CP0100985
|
9-Fluoro-5-[1-furan-2-yl-meth-(Z)-ylidene]-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
|
C24H20FNO2
|
1
|
| 1 |
EC50 = 1.7 nM
|
|
|
|
CP0063871
|
9-Fluoro-2,2,4-trimethyl-5-[1-(3-methyl-pyridin-4-yl)-meth-(Z)-ylidene]-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
|
C26H23FN2O
|
1
|
| 1 |
EC50 = 2 nM
|
|
|
|
CP0101021
|
5-[1-(2-Ethyl-phenyl)-meth-(Z)-ylidene]-9-fluoro-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
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|
C28H26FNO
|
1
|
| 1 |
EC50 = 2 nM
|
|
|
|
CP0083695
|
5-[1,3]Dithian-2-ylidene-9-fluoro-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
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|
C23H22FNOS2
|
1
|
| 1 |
EC50 = 2.1 nM
|
|
|
|
CP0162846
|
7-Fluoro-2,2,4-trimethyl-5-[1-phenyl-meth-(Z)-ylidene]-2,5-dihydro-1H-6-oxa-1-aza-chrysene
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|
C26H22FNO
|
1
|
| 1 |
EC50 = 2.1 nM
|
|
|
|
CP0036228
|
17-ethynyl-17beta-hydroxyestr-4-en-3-one
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|
C20H26O2
|
1
|
| 1 |
EC50 = 2.2 nM
|
|
|
|
CP0164939
|
(Z)-5-(bromomethylene)-9-fluoro-2,2,4-trimethyl-2,5-dihydro-1H-chromeno[3,4-f]quinoline
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|
C20H17BrFNO
|
1
|
| 1 |
EC50 = 2.2 nM
|
|
|
|
CP0055012
|
ONAPRISTONE
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|
C29H39NO3
|
3
|
| 1 |
EC50 = 2.2 nM
|
|
|
| 2 |
IC50 = 1.6 nM
|
|
|
| 3 |
IC50 = 2.2 nM
|
|
|
|
CP0117375
|
5-(4-Chloro-3-methyl-phenyl)-9-fluoro-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene; sulfate
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|
C26H23ClFNO
|
2
|
| 1 |
EC50 = 2.7 nM
|
|
|
| 2 |
Ki = 0.49 nM
|
|
|
|
CP0112566
|
2-[(Z)-(9-fluoro-2,2,4-trimethyl-1H-chromeno[3,4-f]quinolin-5-ylidene)methyl]-N,N-dimethylaniline
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|
C28H27FN2O
|
1
|
| 1 |
EC50 = 2.7 nM
|
|
|
|
CP0286195
|
7-Fluoro-5-[1-(3-fluoro-phenyl)-meth-(Z)-ylidene]-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
|
C26H21F2NO
|
1
|
| 1 |
EC50 = 2.7 nM
|
|
|
|
CP0172383
|
5-(3-Chloro-phenyl)-9-fluoro-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
|
C25H21ClFNO
|
1
|
| 1 |
EC50 = 2.8 nM
|
|
|
|
CP0038907
|
(S)-2-chloro-4-((1-methylpyrrolidin-3-yl)(2-(trifluoromethyl)benzyl)amino)benzonitrile
Show/Hide
|
C20H19ClF3N3
|
1
|
| 1 |
EC50 = 3 nM
|
|
|
|
CP0437620
|
5-(4-Chloro-phenyl)-9-methoxy-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
|
C26H24ClNO2
|
1
|
| 1 |
EC50 = 3.1 nM
|
|
|
|
CP0175610
|
9-Chloro-2,2,4,5-tetramethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
|
C20H20ClNO
|
1
|
| 1 |
EC50 = 3.2 nM
|
|
|
|
CP0301650
|
9-Chloro-5-(3-chloro-phenyl)-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
|
C25H21Cl2NO
|
2
|
| 1 |
EC50 = 3.6 nM
|
|
|
| 2 |
Ki = 0.48 nM
|
|
|
|
CP0182597
|
9-Fluoro-2,2,4-trimethyl-5-[1-o-tolyl-meth-(Z)-ylidene]-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
|
C27H24FNO
|
1
|
| 1 |
EC50 = 3.6 nM
|
|
|
|
CP0465325
|
9-Chloro-5-(3-fluoro-phenyl)-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
|
C25H21ClFNO
|
1
|
| 1 |
EC50 = 3.7 nM
|
|
|
|
CP0193172
|
7-Fluoro-5-[1-(4-fluoro-phenyl)-meth-(Z)-ylidene]-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
|
C26H21F2NO
|
1
|
| 1 |
EC50 = 4 nM
|
|
|
|
CP0453719
|
9-Fluoro-5-[1-(2-isopropyl-phenyl)-meth-(Z)-ylidene]-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
|
C29H28FNO
|
1
|
| 1 |
EC50 = 4 nM
|
|
|
|
CP0107815
|
(4S,5S)-5-(4-Chloro-phenyl)-2,2,4-trimethyl-1,2,4,5-tetrahydro-6-oxa-1-aza-chrysen-3-one
Show/Hide
|
C25H22ClNO2
|
1
|
| 1 |
EC50 = 4.5 nM
|
|
|
|
CP0095680
|
9-Fluoro-2,2,4-trimethyl-5-[1-(2-propyl-phenyl)-meth-(Z)-ylidene]-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
|
C29H28FNO
|
1
|
| 1 |
EC50 = 4.5 nM
|
|
|
|
CP0185145
|
9-Fluoro-2,2,4-trimethyl-5-[1-(3-methyl-pyridin-2-yl)-meth-(Z)-ylidene]-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
|
C26H23FN2O
|
1
|
| 1 |
EC50 = 4.5 nM
|
|
|
|
CP0437035
|
9-Fluoro-2,2,4-trimethyl-5-m-tolyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
|
C26H24FNO
|
1
|
| 1 |
EC50 = 5 nM
|
|
|
|
CP0372871
|
5-(4-Bromo-phenyl)-9-chloro-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
|
C25H21BrClNO
|
1
|
| 1 |
EC50 = 5.2 nM
|
|
|
|
CP0148252
|
(4R,5S)-5-(4-Chloro-phenyl)-2,2,4-trimethyl-1,2,4,5-tetrahydro-6-oxa-1-aza-chrysen-3-one
Show/Hide
|
C25H22ClNO2
|
1
|
| 1 |
EC50 = 5.3 nM
|
|
|
|
CP0200504
|
9-Fluoro-2,2,4-trimethyl-5-[1-phenyl-meth-(Z)-ylidene]-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
|
C26H22FNO
|
1
|
| 1 |
EC50 = 5.3 nM
|
|
|
|
CP0104425
|
2,2,4-Trimethyl-5-[1-o-tolyl-meth-(Z)-ylidene]-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
|
C27H25NO
|
1
|
| 1 |
EC50 = 5.7 nM
|
|
|
|
CP0361748
|
9-Fluoro-2,2,4-trimethyl-5-[1-pyridin-4-yl-meth-(Z)-ylidene]-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
|
C25H21FN2O
|
1
|
| 1 |
EC50 = 5.8 nM
|
|
|
|
CP0185170
|
9-Fluoro-2,2,4-trimethyl-5-[1-(2-methylsulfanyl-phenyl)-meth-(Z)-ylidene]-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
|
C27H24FNOS
|
1
|
| 1 |
EC50 = 6.2 nM
|
|
|
|
CP0106426
|
(4S,5S)-5-(3-Fluoro-phenyl)-2,2,4-trimethyl-1,2,4,5-tetrahydro-6-oxa-1-aza-chrysen-3-one
Show/Hide
|
C25H22FNO2
|
1
|
| 1 |
EC50 = 6.3 nM
|
|
|
|
CP0099719
|
9-Chloro-2,2,4-trimethyl-5-phenyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
|
C25H22ClNO
|
1
|
| 1 |
EC50 = 6.9 nM
|
|
|
|
CP0460156
|
9-Chloro-2,2,4-trimethyl-5-m-tolyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
|
C26H24ClNO
|
1
|
| 1 |
EC50 = 7.1 nM
|
|
|
|
CP0257394
|
9-Fluoro-5-[1-(2-fluoro-phenyl)-meth-(Z)-ylidene]-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
|
C26H21F2NO
|
1
|
| 1 |
EC50 = 7.3 nM
|
|
|
|
CP0401478
|
9-Fluoro-2,2,4-trimethyl-5-phenyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
|
C25H22FNO
|
1
|
| 1 |
EC50 = 7.4 nM
|
|
|
|
CP0431461
|
9-Chloro-2,2,4-trimethyl-5-(3-trifluoromethyl-phenyl)-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
|
C26H21ClF3NO
|
1
|
| 1 |
EC50 = 7.4 nM
|
|
|
|
CP0301665
|
5-[1-(3-Fluoro-phenyl)-meth-(Z)-ylidene]-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
|
C26H22FNO
|
1
|
| 1 |
EC50 = 7.6 nM
|
|
|
|
CP0205607
|
5-(3-Bromo-phenyl)-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
|
C25H22BrNO
|
2
|
| 1 |
EC50 = 8 nM
|
|
|
| 2 |
IC50 = 1136 nM
|
|
|
|
CP0212996
|
5-(3-Fluoro-phenyl)-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
|
C25H22FNO
|
2
|
| 1 |
EC50 = 8 nM
|
|
|
| 2 |
IC50 = 150 nM
|
|
|
|
CP0333217
|
5-(4-Fluoro-phenyl)-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
|
C25H22FNO
|
2
|
| 1 |
EC50 = 8 nM
|
|
|
| 2 |
IC50 = 342 nM
|
|
|
|
CP0475782
|
5-(4-Chloro-phenyl)-9-fluoro-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
|
C25H21ClFNO
|
1
|
| 1 |
EC50 = 8.1 nM
|
|
|
|
CP0107672
|
(4R,5S)-5-(3-Fluoro-phenyl)-2,2,4-trimethyl-1,2,4,5-tetrahydro-6-oxa-1-aza-chrysen-3-one
Show/Hide
|
C25H22FNO2
|
1
|
| 1 |
EC50 = 8.7 nM
|
|
|
|
CP0184486
|
5-[1-(3-Fluoro-phenyl)-meth-(Z)-ylidene]-2,2,4-trimethyl-1,2,4,5-tetrahydro-6-oxa-1-aza-chrysen-3-one
Show/Hide
|
C26H22FNO2
|
1
|
| 1 |
EC50 = 8.7 nM
|
|
|
|
CP0437687
|
9-Chloro-5-(4-chloro-phenyl)-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
|
C25H21Cl2NO
|
1
|
| 1 |
EC50 = 9 nM
|
|
|
|
CP0164908
|
(4R,5S)-2,2,4-Trimethyl-5-phenyl-1,2,4,5-tetrahydro-6-oxa-1-aza-chrysen-3-one
Show/Hide
|
C25H23NO2
|
1
|
| 1 |
EC50 = 9 nM
|
|
|
|
CP0301589
|
5-[1-(2-Bromo-phenyl)-meth-(Z)-ylidene]-9-fluoro-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
|
C26H21BrFNO
|
1
|
| 1 |
EC50 = 9 nM
|
|
|
|
CP0104422
|
9-Chloro-5-(4-chloro-3-methyl-phenyl)-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
|
C26H23Cl2NO
|
2
|
| 1 |
EC50 = 9.4 nM
|
|
|
| 2 |
Ki = 0.5 nM
|
|
|
|
CP0416578
|
9-Chloro-5-(4-fluoro-3-methyl-phenyl)-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
|
C26H23ClFNO
|
1
|
| 1 |
EC50 = 9.5 nM
|
|
|
|
CP0279772
|
5-(4-Chloro-phenyl)-2,2,4,4-tetramethyl-1,2,4,5-tetrahydro-6-oxa-1-aza-chrysen-3-one
Show/Hide
|
C26H24ClNO2
|
1
|
| 1 |
EC50 = 9.8 nM
|
|
|
|
CP0401479
|
9-Fluoro-2,2,4-trimethyl-5-(3-trifluoromethyl-phenyl)-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
|
C26H21F4NO
|
1
|
| 1 |
EC50 = 10 nM
|
|
|
|
CP0405238
|
5-(4-Chloro-phenyl)-8-fluoro-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
|
C25H21ClFNO
|
1
|
| 1 |
EC50 = 10 nM
|
|
|
|
CP0114693
|
(4S,5S)-2,2,4-Trimethyl-5-phenyl-1,2,4,5-tetrahydro-6-oxa-1-aza-chrysen-3-one
Show/Hide
|
C25H23NO2
|
1
|
| 1 |
EC50 = 10 nM
|
|
|
|
CP0322395
|
(S)-ethyl 2-(3-((3-chloro-4-cyanophenyl)(2-chlorobenzyl)amino)pyrrolidin-1-yl)acetate
Show/Hide
|
C22H23Cl2N3O2
|
1
|
| 1 |
EC50 = 10 nM
|
|
|
|
CP0082075
|
(Z)-5-(butan-2-ylidene)-9-fluoro-2,2,4-trimethyl-2,5-dihydro-1H-chromeno[3,4-f]quinoline
Show/Hide
|
C23H24FNO
|
1
|
| 1 |
EC50 = 11 nM
|
|
|
|
CP0137848
|
9-Fluoro-2,2,4-trimethyl-5-[1-(2-trifluoromethoxy-phenyl)-meth-(Z)-ylidene]-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
|
C27H21F4NO2
|
1
|
| 1 |
EC50 = 11 nM
|
|
|
|
CP0201054
|
2-[9-Fluoro-2,2,4-trimethyl-1,2-dihydro-6-oxa-1-aza-chrysen-(5Z)-ylidenemethyl]-benzaldehyde
Show/Hide
|
C27H22FNO2
|
1
|
| 1 |
EC50 = 11 nM
|
|
|
|
CP0305346
|
2-[9-Fluoro-2,2,4-trimethyl-1,2-dihydro-6-oxa-1-aza-chrysen-(5Z)-ylidenemethyl]-benzonitrile
Show/Hide
|
C27H21FN2O
|
1
|
| 1 |
EC50 = 11 nM
|
|
|
|
CP0318485
|
5-[1-(2-Chloro-phenyl)-meth-(Z)-ylidene]-9-fluoro-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
|
C26H21ClFNO
|
1
|
| 1 |
EC50 = 12 nM
|
|
|
|
CP0449427
|
9-Chloro-5-(4-methoxy-phenyl)-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
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C26H24ClNO2
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1
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| 1 |
EC50 = 13 nM
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CP0163667
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2,2,4-Trimethyl-5-(3-trifluoromethyl-phenyl)-2,5-dihydro-1H-6-oxa-1-aza-chrysene
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C26H22F3NO
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2
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| 1 |
EC50 = 13 nM
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| 2 |
IC50 > 10000 nM
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CP0103435
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9-Chloro-7-fluoro-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
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C19H17ClFNO
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1
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| 1 |
EC50 = 13.5 nM
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CP0134558
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5-(4-Chloro-3-methyl-phenyl)-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
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C26H24ClNO
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2
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| 1 |
EC50 = 14 nM
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| 2 |
IC50 > 10000 nM
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CP0185464
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5-(4-Chloro-phenyl)-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
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C25H22ClNO
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3
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| 1 |
EC50 = 14 nM
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| 2 |
EC50 = 15 nM
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| 3 |
IC50 = 600 nM
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CP0235429
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5-(4-Bromo-phenyl)-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
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C25H22BrNO
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2
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| 1 |
EC50 = 14 nM
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| 2 |
IC50 = 3138 nM
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CP0147609
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(4S,5S)-2,2,4-Trimethyl-5-(3-trifluoromethyl-phenyl)-1,2,4,5-tetrahydro-6-oxa-1-aza-chrysen-3-one
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C26H22F3NO2
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1
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| 1 |
EC50 = 14 nM
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CP0193258
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9-Fluoro-2,2,4-trimethyl-5-[1-(2-trifluoromethyl-phenyl)-meth-(Z)-ylidene]-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
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C27H21F4NO
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1
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| 1 |
EC50 = 14 nM
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CP0134269
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5-[1-(2,5-Difluoro-phenyl)-meth-(Z)-ylidene]-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
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C26H21F2NO
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1
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| 1 |
EC50 = 14.7 nM
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CP0146748
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5-[1-(3,4-Difluoro-phenyl)-meth-(Z)-ylidene]-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
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C26H21F2NO
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1
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| 1 |
EC50 = 14.7 nM
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CP0377309
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9-Fluoro-5-(4-fluoro-3-methyl-phenyl)-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
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C26H23F2NO
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1
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| 1 |
EC50 = 15 nM
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CP0361542
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9-Fluoro-2,2,4-trimethyl-5-[1-pyridin-2-yl-meth-(Z)-ylidene]-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
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C25H21FN2O
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1
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| 1 |
EC50 = 15 nM
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CP0057358
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5-(3-Fluoro-4-methyl-phenyl)-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
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C26H24FNO
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2
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| 1 |
EC50 = 16 nM
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| 2 |
IC50 > 10000 nM
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CP0097577
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(4R,5S)-2,2,4-Trimethyl-5-(3-trifluoromethyl-phenyl)-1,2,4,5-tetrahydro-6-oxa-1-aza-chrysen-3-one
Show/Hide
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C26H22F3NO2
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1
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| 1 |
EC50 = 16 nM
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CP0341518
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7-Fluoro-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene-9-carbonitrile
Show/Hide
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C20H17FN2O
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1
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| 1 |
EC50 = 16.7 nM
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CP0295932
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5-Benzyl-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
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C26H25NO
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1
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| 1 |
EC50 = 16.8 nM
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CP0051168
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5-(4-Chloro-3-fluoro-phenyl)-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
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C25H21ClFNO
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2
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| 1 |
EC50 = 17 nM
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| 2 |
IC50 > 10000 nM
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CP0051650
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5-(3-Bromo-5-methyl-phenyl)-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
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C26H24BrNO
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2
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| 1 |
EC50 = 17 nM
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| 2 |
IC50 = 1100 nM
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CP0148253
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2,2,4-Trimethyl-5-[1-phenyl-meth-(Z)-ylidene]-1,2,4,5-tetrahydro-6-oxa-1-aza-chrysen-3-one
Show/Hide
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C26H23NO2
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1
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| 1 |
EC50 = 17 nM
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CP0063640
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5-(3-Chloro-phenyl)-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
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C25H22ClNO
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2
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| 1 |
EC50 = 18 nM
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| 2 |
IC50 = 930 nM
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CP0200882
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5-(3,4-Dichloro-phenyl)-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
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C25H21Cl2NO
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2
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| 1 |
EC50 = 18 nM
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| 2 |
IC50 = 720 nM
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CP0404026
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5-[1-(2,4-Difluoro-phenyl)-meth-(Z)-ylidene]-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
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C26H21F2NO
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1
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| 1 |
EC50 = 22 nM
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CP0193631
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2,2,4-Trimethyl-5-[1-phenyl-meth-(Z)-ylidene]-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
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C26H23NO
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1
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| 1 |
EC50 = 24.4 nM
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CP0367405
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5-(4-Fluoro-3-trifluoromethyl-phenyl)-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
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C26H21F4NO
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2
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| 1 |
EC50 = 25 nM
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| 2 |
IC50 = 4600 nM
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CP0349897
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7,9-Difluoro-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
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C19H17F2NO
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1
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| 1 |
EC50 = 25.4 nM
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CP0292289
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5-[1-(2,3-Difluoro-phenyl)-meth-(Z)-ylidene]-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
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C26H21F2NO
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1
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| 1 |
EC50 = 26.3 nM
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CP0285558
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5-(3-Bromo-5-fluoro-phenyl)-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
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C25H21BrFNO
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2
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| 1 |
EC50 = 27 nM
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| 2 |
IC50 = 1207 nM
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CP0237182
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(E)-5-(butan-2-ylidene)-9-fluoro-2,2,4-trimethyl-2,5-dihydro-1H-chromeno[3,4-f]quinoline
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C23H24FNO
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2
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| 1 |
EC50 = 27 nM
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| 2 |
IC50 = 980 nM
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CP0184604
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(Z)-5-butylidene-9-fluoro-2,2,4-trimethyl-2,5-dihydro-1H-chromeno[3,4-f]quinoline
Show/Hide
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C23H24FNO
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1
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| 1 |
EC50 = 28 nM
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CP0295910
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2,2,4-Trimethyl-9-nitro-2,5-dihydro-1H-6-oxa-1-aza-chrysene
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C19H18N2O3
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1
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| 1 |
EC50 = 28.6 nM
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CP0515006
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5-[1-(2-Fluoro-phenyl)-meth-(Z)-ylidene]-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
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C26H22FNO
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1
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| 1 |
EC50 = 29 nM
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CP0345411
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9-Fluoro-2,2,4-trimethyl-5-(3-methyl-2-methylene-butylidene)-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
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C25H26FNO
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1
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| 1 |
EC50 = 29 nM
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CP0099192
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9-Fluoro-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
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C19H18FNO
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1
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| 1 |
EC50 = 30.3 nM
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CP0531862
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5-[1-(4-Bromo-phenyl)-meth-(Z)-ylidene]-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
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C26H22BrNO
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1
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| 1 |
EC50 = 31.5 nM
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CP0303823
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5-[1-(2,6-Difluoro-phenyl)-meth-(Z)-ylidene]-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
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C26H21F2NO
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1
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| 1 |
EC50 = 32 nM
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CP0267194
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2,2,4-Trimethyl-5-(4-trifluoromethyl-phenyl)-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
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C26H22F3NO
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2
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| 1 |
EC50 = 33 nM
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| 2 |
IC50 = 150 nM
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CP0161503
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5-Bromo-2-((1R,3R)-3-bromo-2,2-dimethyl-6-methylene-cyclohexylmethyl)-4-methoxy-phenol
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C17H22Br2O2
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1
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| 1 |
EC50 = 35 nM
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CP0082132
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9-Chloro-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
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C19H18ClNO
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1
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| 1 |
EC50 = 35.7 nM
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CP0246143
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5-[1-(3-Bromo-phenyl)-meth-(Z)-ylidene]-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
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C26H22BrNO
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1
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| 1 |
EC50 = 37 nM
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CP0184222
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2,2,4-Trimethyl-5-p-tolyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
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C26H25NO
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2
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| 1 |
EC50 = 37 nM
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| 2 |
IC50 = 250 nM
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CP0301450
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(4S,5S)-5-(4-Chloro-phenyl)-2,2,4-trimethyl-2,3,4,5-tetrahydro-1H-6-oxa-1-aza-chrysene
Show/Hide
|
C25H24ClNO
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1
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| 1 |
EC50 = 39 nM
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CP0107714
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7,9-Difluoro-2,2,4-trimethyl-2,3,4,5-tetrahydro-1H-6-oxa-1-aza-chrysene
Show/Hide
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C19H19F2NO
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1
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| 1 |
EC50 = 40 nM
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CP0110330
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9-Bromo-7-methoxy-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
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C20H20BrNO2
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1
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| 1 |
EC50 = 43 nM
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CP0134207
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9-Bromo-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
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C19H18BrNO
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1
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| 1 |
EC50 = 45 nM
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CP0183553
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5-[1-(3-Fluoro-phenyl)-meth-(Z)-ylidene]-2,2,4-trimethyl-2,3,4,5-tetrahydro-1H-6-oxa-1-aza-chrysene
Show/Hide
|
C26H24FNO
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1
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| 1 |
EC50 = 47 nM
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CP0270576
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5-[1-(3,5-Difluoro-phenyl)-meth-(Z)-ylidene]-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
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C26H21F2NO
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1
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| 1 |
EC50 = 47.7 nM
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CP0369770
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(4R,5S)-5-(4-Chloro-phenyl)-2,2,4-trimethyl-2,3,4,5-tetrahydro-1H-6-oxa-1-aza-chrysene
Show/Hide
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C25H24ClNO
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2
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| 1 |
EC50 = 48 nM
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| 2 |
IC50 = 3100 nM
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CP0420410
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5-Cyclohexylmethylene-9-fluoro-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
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C26H28FNO
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2
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| 1 |
EC50 = 48 nM
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| 2 |
IC50 = 800 nM
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CP0250549
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5-(3,5-Dichloro-phenyl)-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
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C25H21Cl2NO
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2
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| 1 |
EC50 = 50 nM
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| 2 |
IC50 > 10000 nM
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CP0275372
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(S)-2-chloro-4-((2-chlorobenzyl)(1-(2-methoxyethyl)pyrrolidin-3-yl)amino)benzonitrile
Show/Hide
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C21H23Cl2N3O
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1
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| 1 |
EC50 = 50 nM
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CP0266550
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2,2,4-Trimethyl-9-nitro-2,3,4,5-tetrahydro-1H-6-oxa-1-aza-chrysene
Show/Hide
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C19H20N2O3
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1
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| 1 |
EC50 = 52 nM
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CP0035629
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9-Bromo-7-fluoro-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
|
C19H17BrFNO
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1
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| 1 |
EC50 = 57 nM
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CP0268369
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5-[1-(2-Chloro-phenyl)-meth-(Z)-ylidene]-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
|
C26H22ClNO
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1
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| 1 |
EC50 = 57.8 nM
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CP0334888
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5-[1-(2-Bromo-phenyl)-meth-(Z)-ylidene]-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
|
C26H22BrNO
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1
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| 1 |
EC50 = 57.8 nM
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CP0221030
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5-[1-(4-Fluoro-phenyl)-meth-(Z)-ylidene]-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
|
C26H22FNO
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1
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| 1 |
EC50 = 59.5 nM
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CP0334590
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2,2,4-Trimethyl-5-[1-m-tolyl-meth-(Z)-ylidene]-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
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C27H25NO
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1
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| 1 |
EC50 = 75 nM
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CP0082128
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2,2,4,9-Tetramethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
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C20H21NO
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1
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| 1 |
EC50 = 76 nM
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CP0082133
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2,2,4-Trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
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C19H19NO
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1
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| 1 |
EC50 = 111 nM
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CP0268090
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5-[1-(3-Chloro-phenyl)-meth-(Z)-ylidene]-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
|
C26H22ClNO
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1
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| 1 |
EC50 = 117 nM
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CP0082129
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7-Fluoro-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
|
C19H18FNO
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1
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| 1 |
EC50 = 118 nM
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CP0353353
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5-(4-Chloro-phenyl)-2,2-dimethyl-4-methylene-2,3,4,5-tetrahydro-1H-6-oxa-1-aza-chrysene
Show/Hide
|
C25H22ClNO
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2
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| 1 |
EC50 = 124 nM
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| 2 |
IC50 = 1755 nM
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CP0295084
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5-[1-(4-Chloro-phenyl)-meth-(Z)-ylidene]-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
|
C26H22ClNO
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1
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| 1 |
EC50 = 139 nM
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CP0050558
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2,2,4-Trimethyl-5-phenyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
|
C25H23NO
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2
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| 1 |
EC50 = 156 nM
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| 2 |
IC50 = 290 nM
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CP0106007
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9-Methoxy-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
|
C20H21NO2
|
1
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| 1 |
EC50 = 170 nM
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CP0110332
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9-Chloro-2,2,4,7-tetramethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
|
C20H20ClNO
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1
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| 1 |
EC50 = 178 nM
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CP0288560
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8-Methoxy-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
|
C20H21NO2
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1
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| 1 |
EC50 = 193 nM
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CP0299302
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(13S)-4-amino-13-(2-chlorophenyl)-6-methyl-11-oxo-8-thia-3,10-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5-tetraene-5-carbonitrile
Show/Hide
|
C18H13ClN4OS
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1
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| 1 |
EC50 = 199.53 nM
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CP0167379
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(S)-2-chloro-4-((2-methylbenzyl)(1-methylpyrrolidin-3-yl)amino)benzonitrile
Show/Hide
|
C20H22ClN3
|
1
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| 1 |
EC50 = 200 nM
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CP0358631
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(S)-2-chloro-4-((2-chlorobenzyl)(1-isopropylpyrrolidin-3-yl)amino)benzonitrile
Show/Hide
|
C21H23Cl2N3
|
1
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| 1 |
EC50 = 200 nM
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CP0358632
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(S)-2-chloro-4-((2-chlorobenzyl)(1-(3,3,3-trifluoropropyl)pyrrolidin-3-yl)amino)benzonitrile
Show/Hide
|
C21H20Cl2F3N3
|
1
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| 1 |
EC50 = 200 nM
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CP0358634
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(S)-2-(3-((3-chloro-4-cyanophenyl)(2-chlorobenzyl)amino)pyrrolidin-1-yl)acetamide
Show/Hide
|
C20H20Cl2N4O
|
1
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| 1 |
EC50 = 200 nM
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CP0399510
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9-Fluoro-5-(4-methoxy-phenyl)-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
|
C26H24FNO2
|
1
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| 1 |
EC50 = 270 nM
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CP0063641
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4-Methyl-5-(2,2,4,4-tetramethyl-3-oxo-1,2,3,4-tetrahydro-quinolin-6-yl)-thiophene-2-carbonitrile
Show/Hide
|
C19H20N2OS
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2
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| 1 |
EC50 = 350 nM
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| 2 |
IC50 = 10 nM
|
|
|
|
CP0046946
|
5-Bromo-4-methoxy-2-((1S,4R)-2,2,4-trimethyl-6-methylene-cyclohexylmethyl)-phenol
Show/Hide
|
C18H25BrO2
|
1
|
| 1 |
EC50 = 458 nM
|
|
|
|
CP0099191
|
7-Chloro-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
|
C19H18ClNO
|
1
|
| 1 |
EC50 = 576 nM
|
|
|
|
CP0104457
|
9-Bromo-7-fluoro-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene-8-carbaldehyde
Show/Hide
|
C20H17BrFNO2
|
1
|
| 1 |
EC50 = 576 nM
|
|
|
|
CP0166403
|
4-amino-13-(2-chlorophenyl)-6-methyl-11-oxo-8-thia-3,10-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5-tetraene-5-carbonitrile
Show/Hide
|
C18H13ClN4OS
|
1
|
| 1 |
EC50 = 630.96 nM
|
|
|
|
CP0216130
|
9-Fluoro-2,2,4,7-tetramethyl-2,3,4,5-tetrahydro-1H-6-oxa-1-aza-chrysene
Show/Hide
|
C20H22FNO
|
1
|
| 1 |
EC50 = 637 nM
|
|
|
|
CP0058423
|
5,8-difluoro-2,2,4-trimethyl-2,10-dihydro-1H-indeno[1,2-g]quinoline
Show/Hide
|
C19H17F2N
|
1
|
| 1 |
EC50 = 650 nM
|
|
|
|
CP0299601
|
9-Fluoro-2,2,4-trimethyl-7-nitro-2,3,4,5-tetrahydro-1H-6-oxa-1-aza-chrysene
Show/Hide
|
C19H19FN2O3
|
1
|
| 1 |
EC50 = 781 nM
|
|
|
|
CP0135117
|
9-Fluoro-2,2,4-trimethyl-5-methylene-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
|
C20H18FNO
|
1
|
| 1 |
EC50 = 1000 nM
|
|
|
|
CP0040470
|
4-(2,2,4,4-Tetramethyl-3-oxo-1,2,3,4-tetrahydro-quinolin-6-yl)-thiophene-2-carbonitrile
Show/Hide
|
C18H18N2OS
|
2
|
| 1 |
EC50 = 1190 nM
|
|
|
| 2 |
IC50 = 14 nM
|
|
|
|
CP0214131
|
5-Bromo-4-methoxy-2-(4,6,6-trimethyl-2-methylene-cyclohex-3-enylmethyl)-phenol
Show/Hide
|
C18H23BrO2
|
2
|
| 1 |
EC50 = 1295 nM
|
|
|
| 2 |
IC50 = 3567 nM
|
|
|
|
CP0183300
|
5-(4-Chloro-phenyl)-2,2-dimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
|
C24H20ClNO
|
2
|
| 1 |
EC50 = 1300 nM
|
|
|
| 2 |
IC50 = 140 nM
|
|
|
|
CP0071628
|
2-[4-cyano-N-(2,2,2-trifluoroethyl)-3-(trifluoromethyl)anilino]-N,N-dimethylpropanamide
Show/Hide
|
C15H15F6N3O
|
1
|
| 1 |
EC50 = 1300 nM
|
|
|
|
CP0136434
|
(S)-4-(benzyl(1-methylpyrrolidin-3-yl)amino)-2-chlorobenzonitrile
Show/Hide
|
C19H20ClN3
|
1
|
| 1 |
EC50 = 1300 nM
|
|
|
|
CP0055056
|
Acetic acid 5-bromo-4-methoxy-2-(4,6,6-trimethyl-2-methylene-cyclohex-3-enylmethyl)-phenyl ester
Show/Hide
|
C20H25BrO3
|
2
|
| 1 |
EC50 = 1457 nM
|
|
|
| 2 |
IC50 = 710 nM
|
|
|
|
CP0217116
|
5-(6-Bromo-pyridin-2-yl)-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
|
C24H21BrN2O
|
2
|
| 1 |
EC50 = 1700 nM
|
|
|
| 2 |
IC50 = 71 nM
|
|
|
|
CP0301622
|
4-(2,2,4-Trimethyl-1,2-dihydro-quinolin-6-yl)-thiophene-2-carbonitrile
Show/Hide
|
C17H16N2S
|
2
|
| 1 |
EC50 = 1800 nM
|
|
|
| 2 |
IC50 = 24 nM
|
|
|
|
CP0215570
|
7,9-Dibromo-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
|
C19H17Br2NO
|
1
|
| 1 |
EC50 = 1871 nM
|
|
|
|
CP0309710
|
2,2,4-Trimethyl-9-phenyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
|
C25H23NO
|
1
|
| 1 |
EC50 = 2030 nM
|
|
|
|
CP0150643
|
Acetic acid 5-bromo-4-methoxy-2-(5,5,7-trimethyl-spiro[2.5]oct-7-en-4-ylmethyl)-phenyl ester
Show/Hide
|
C21H27BrO3
|
2
|
| 1 |
EC50 = 2117 nM
|
|
|
| 2 |
IC50 = 160 nM
|
|
|
|
CP0156852
|
4-Methyl-5-(2,2,4-trimethyl-1,2,3,4-tetrahydro-quinolin-6-yl)-thiophene-2-carbonitrile
Show/Hide
|
C18H20N2S
|
2
|
| 1 |
EC50 = 2290 nM
|
|
|
| 2 |
IC50 = 31 nM
|
|
|
|
CP0110334
|
6-(4-Bromo-thiophen-2-yl)-2,2,4-trimethyl-1,2-dihydro-quinoline
Show/Hide
|
C16H16BrNS
|
2
|
| 1 |
EC50 = 2700 nM
|
|
|
| 2 |
IC50 = 105 nM
|
|
|
|
CP0082976
|
(Z)-2-(9-fluoro-2,2,4-trimethyl-1,2-dihydrochromeno[3,4-f]quinolin-5-ylidene)acetonitrile
Show/Hide
|
C21H17FN2O
|
2
|
| 1 |
EC50 = 2700 nM
|
|
|
| 2 |
IC50 = 65 nM
|
|
|
|
CP0311285
|
5-(2,2,4-Trimethyl-1,2-dihydro-quinolin-6-yl)-thiophene-2-carbonitrile
Show/Hide
|
C17H16N2S
|
2
|
| 1 |
EC50 = 2900 nM
|
|
|
| 2 |
IC50 = 27 nM
|
|
|
|
CP0161504
|
Acetic acid 5-bromo-2-((1S,6R)-4,6-dimethyl-2-methylene-cyclohex-3-enylmethyl)-4-methoxy-phenyl ester
Show/Hide
|
C19H23BrO3
|
2
|
| 1 |
EC50 = 3005 nM
|
|
|
| 2 |
IC50 = 350 nM
|
|
|
|
CP0184235
|
5-Bromo-4-methoxy-2-((1S,2R)-2-methyl-6-methylene-cyclohexylmethyl)-phenol
Show/Hide
|
C16H21BrO2
|
2
|
| 1 |
EC50 = 3011 nM
|
|
|
| 2 |
IC50 = 320 nM
|
|
|
|
CP0123765
|
5-Bromo-2-((S)-2,2-dimethyl-6-methylene-cyclohexylmethyl)-4-methoxy-phenol
Show/Hide
|
C17H23BrO2
|
2
|
| 1 |
EC50 = 3264 nM
|
|
|
| 2 |
IC50 = 597 nM
|
|
|
|
CP0150432
|
5-Bromo-4-methoxy-2-[(E)-3-(4,6,6-trimethyl-2-methylene-cyclohex-3-enyl)-propenyl]-phenol
Show/Hide
|
C20H25BrO2
|
1
|
| 1 |
EC50 = 3300 nM
|
|
|
|
CP0060893
|
5-(6-Bromo-pyridin-3-yl)-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
|
C24H21BrN2O
|
2
|
| 1 |
EC50 = 3900 nM
|
|
|
| 2 |
IC50 = 54 nM
|
|
|
|
CP0089139
|
4-amino-13-(2-chloro-6-fluorophenyl)-6-methyl-11-oxo-8-thia-3,10-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5-tetraene-5-carbonitrile
Show/Hide
|
C18H12ClFN4OS
|
1
|
| 1 |
EC50 = 3981.07 nM
|
|
|
|
CP0267637
|
4-amino-13-(2-fluorophenyl)-6-methyl-11-oxo-8-thia-3,10-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5-tetraene-5-carbonitrile
Show/Hide
|
C18H13FN4OS
|
1
|
| 1 |
EC50 = 3981.07 nM
|
|
|
|
CP0207843
|
5-Bromo-2-(2,2-dimethyl-6-methylene-cyclohexylmethyl)-4-methoxy-phenol
Show/Hide
|
C17H23BrO2
|
2
|
| 1 |
EC50 = 4020 nM
|
|
|
| 2 |
IC50 = 405 nM
|
|
|
|
CP0185326
|
5-[1-(3-Methoxy-phenyl)-meth-(Z)-ylidene]-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
|
C27H25NO2
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0303783
|
2,2,4-Trimethyl-5-[1-p-tolyl-meth-(Z)-ylidene]-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
|
C27H25NO
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0097002
|
1-[4-(2,2,4-Trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysen-5-yl)-phenyl]-ethanone
Show/Hide
|
C27H25NO2
|
2
|
| 1 |
EC50 > 10000 nM
|
|
|
| 2 |
IC50 = 132 nM
|
|
|
|
CP0284433
|
5-(4-Methoxy-phenyl)-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene
Show/Hide
|
C26H25NO2
|
2
|
| 1 |
EC50 > 10000 nM
|
|
|
| 2 |
IC50 = 105 nM
|
|
|
|
CP0136432
|
(S)-2-chloro-4-((1-methylpyrrolidin-3-yl)(propyl)amino)benzonitrile
Show/Hide
|
C15H20ClN3
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0136435
|
(S)-2-chloro-4-((1-methylpyrrolidin-3-yl)(pyridin-2-ylmethyl)amino)benzonitrile
Show/Hide
|
C18H19ClN4
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0147279
|
(S)-2-chloro-4-(ethyl(1-methylpyrrolidin-3-yl)amino)benzonitrile
Show/Hide
|
C14H18ClN3
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0197930
|
(S)-2-chloro-4-((2,6-dichlorobenzyl)(1-methylpyrrolidin-3-yl)amino)benzonitrile
Show/Hide
|
C19H18Cl3N3
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0254446
|
(S)-2-chloro-4-((4-chlorobenzyl)(1-methylpyrrolidin-3-yl)amino)benzonitrile
Show/Hide
|
C19H19Cl2N3
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0358627
|
(S)-4-(butyl(1-methylpyrrolidin-3-yl)amino)-2-chlorobenzonitrile
Show/Hide
|
C16H22ClN3
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0358629
|
(S)-2-chloro-4-((3-chlorobenzyl)(1-methylpyrrolidin-3-yl)amino)benzonitrile
Show/Hide
|
C19H19Cl2N3
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0358635
|
(S)-2-chloro-4-((2-chlorobenzyl)(1-(pyridin-2-ylmethyl)pyrrolidin-3-yl)amino)benzonitrile
Show/Hide
|
C24H22Cl2N4
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0517059
|
(S)-2-chloro-4-((cyclohexylmethyl)(1-methylpyrrolidin-3-yl)amino)benzonitrile
Show/Hide
|
C19H26ClN3
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0221290
|
4-amino-6-methyl-11-oxo-13-phenyl-8-thia-3,10-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5-tetraene-5-carbonitrile
Show/Hide
|
C18H14N4OS
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0233971
|
(13R)-4-amino-13-(2-chlorophenyl)-6-methyl-11-oxo-8-thia-3,10-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5-tetraene-5-carbonitrile
Show/Hide
|
C18H13ClN4OS
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0265651
|
4-amino-13-(2,4-dichlorophenyl)-6-methyl-11-oxo-8-thia-3,10-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5-tetraene-5-carbonitrile
Show/Hide
|
C18H12Cl2N4OS
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0265653
|
13-(2-chlorophenyl)-6-methyl-4,11-dioxo-8-thia-3,10-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-triene-5-carbonitrile
Show/Hide
|
C18H12ClN3O2S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0272503
|
4-amino-6-methyl-13-(2-methylphenyl)-11-oxo-8-thia-3,10-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5-tetraene-5-carbonitrile
Show/Hide
|
C19H16N4OS
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0272505
|
4-amino-13-(2,5-dichlorophenyl)-6-methyl-11-oxo-8-thia-3,10-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5-tetraene-5-carbonitrile
Show/Hide
|
C18H12Cl2N4OS
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0287545
|
4-amino-13-(2-methoxyphenyl)-6-methyl-11-oxo-8-thia-3,10-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5-tetraene-5-carbonitrile
Show/Hide
|
C19H16N4O2S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0350721
|
4-amino-13-(2,3-dichlorophenyl)-6-methyl-11-oxo-8-thia-3,10-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5-tetraene-5-carbonitrile
Show/Hide
|
C18H12Cl2N4OS
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0371224
|
4-amino-13-(3-methoxyphenyl)-6-methyl-11-oxo-8-thia-3,10-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5-tetraene-5-carbonitrile
Show/Hide
|
C19H16N4O2S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0244609
|
4-chloro-N-[[4-(3,5-dimethyl-1,2-oxazol-4-yl)phenyl]methyl]-1,3-dimethylpyrazolo[3,4-b]pyridine-5-carboxamide
Show/Hide
|
C21H20ClN5O2
|
2
|
| 1 |
EC50 > 10000 nM
|
|
|
| 2 |
IC50 = 3162.28 nM
|
|
|
|
CP0294482
|
4-chloro-N-[(2,4-dimethylphenyl)methyl]-1-ethylpyrazolo[3,4-b]pyridine-5-carboxamide
Show/Hide
|
C18H19ClN4O
|
2
|
| 1 |
EC50 > 10000 nM
|
|
|
| 2 |
IC50 = 1258.93 nM
|
|
|
|
CP0301835
|
4-chloro-N-(2,3-dihydro-1H-inden-2-ylmethyl)-3-ethyl-1-methylpyrazolo[3,4-b]pyridine-5-carboxamide
Show/Hide
|
C20H21ClN4O
|
2
|
| 1 |
EC50 > 10000 nM
|
|
|
| 2 |
IC50 > 10000 nM
|
|
|
|
CP0090808
|
3-(3-fluorophenyl)-1-(4-methylphenyl)-3-(4-nitroanilino)propan-1-one
Show/Hide
|
C22H19FN2O3
|
2
|
| 1 |
EC50 > 10000 nM
|
|
|
| 2 |
IC50 = 6064 nM
|
|
|
|
CP0092869
|
3-(3-fluorophenyl)-1-(4-fluorophenyl)-3-(4-nitroanilino)propan-1-one
Show/Hide
|
C21H16F2N2O3
|
2
|
| 1 |
EC50 > 10000 nM
|
|
|
| 2 |
IC50 = 805 nM
|
|
|
|
CP0226268
|
3-cyclohexyl-1-(4-methoxyphenyl)-3-(4-nitroanilino)propan-1-one
Show/Hide
|
C22H26N2O4
|
2
|
| 1 |
EC50 > 10000 nM
|
|
|
| 2 |
IC50 = 139 nM
|
|
|
|
CP0226271
|
1-(3-chlorophenyl)-3-(3-fluorophenyl)-3-(4-nitroanilino)propan-1-one
Show/Hide
|
C21H16ClFN2O3
|
2
|
| 1 |
EC50 > 10000 nM
|
|
|
| 2 |
IC50 = 3538 nM
|
|
|
|
CP0288608
|
1-(3-methoxyphenyl)-3-(4-nitroanilino)-3-[4-(trifluoromethyl)phenyl]propan-1-one
Show/Hide
|
C23H19F3N2O4
|
2
|
| 1 |
EC50 > 10000 nM
|
|
|
| 2 |
IC50 = 1831 nM
|
|
|
|
CP0294140
|
1-(4-bromophenyl)-3-(4-nitroanilino)-3-[4-(trifluoromethyl)phenyl]propan-1-one
Show/Hide
|
C22H16BrF3N2O3
|
2
|
| 1 |
EC50 > 10000 nM
|
|
|
| 2 |
IC50 = 1213 nM
|
|
|
|
CP0294141
|
1-(4-chlorophenyl)-3-cyclohexyl-3-(4-nitroanilino)propan-1-one
Show/Hide
|
C21H23ClN2O3
|
2
|
| 1 |
EC50 > 10000 nM
|
|
|
| 2 |
IC50 = 216 nM
|
|
|
|
CP0302211
|
1-(4-methoxyphenyl)-3-(4-nitroanilino)-3-[4-(trifluoromethyl)phenyl]propan-1-one
Show/Hide
|
C23H19F3N2O4
|
2
|
| 1 |
EC50 > 10000 nM
|
|
|
| 2 |
IC50 = 2696 nM
|
|
|
|
CP0308057
|
3-cyclohexyl-1-(3-fluorophenyl)-3-(4-nitroanilino)propan-1-one
Show/Hide
|
C21H23FN2O3
|
2
|
| 1 |
EC50 > 10000 nM
|
|
|
| 2 |
IC50 = 193 nM
|
|
|
|
CP0315062
|
1-(4-bromophenyl)-3-cyclohexyl-3-(4-nitroanilino)propan-1-one
Show/Hide
|
C21H23BrN2O3
|
2
|
| 1 |
EC50 > 10000 nM
|
|
|
| 2 |
IC50 = 1555 nM
|
|
|
|
CP0294481
|
4-chloro-N-[[2-(3-methoxyphenyl)phenyl]methyl]-1,3-dimethylpyrazolo[3,4-b]pyridine-5-carboxamide
Show/Hide
|
C23H21ClN4O2
|
2
|
| 1 |
EC50 > 19952.62 nM
|
|
|
| 2 |
IC50 > 5011.87 nM
|
|
|
|
CP0493508
|
6-(3-Chloro-5-fluoro-phenyl)-4,4-dimethyl-1,4-dihydro-benzo[d][1,3]oxazin-2-one
Show/Hide
|
C16H13ClFNO2
|
1
|
| 1 |
IC50 = 2.6 nM
|
|
|
|
CP0453570
|
6-(3-Fluoro-phenyl)-4,4-dimethyl-1,4-dihydro-benzo[d][1,3]oxazin-2-one
Show/Hide
|
C16H14FNO2
|
1
|
| 1 |
IC50 = 3.8 nM
|
|
|
|
CP0503518
|
4-(4,4-Dimethyl-2-oxo-1,4-dihydro-2H-benzo[d][1,3]oxazin-6-yl)-thiophene-2-carbonitrile
Show/Hide
|
C15H12N2O2S
|
1
|
| 1 |
IC50 = 6.7 nM
|
|
|
|
CP0102421
|
6-(3-Chloro-phenyl)-4,4-dimethyl-1,4-dihydro-benzo[d][1,3]oxazin-2-one
Show/Hide
|
C16H14ClNO2
|
1
|
| 1 |
IC50 = 9.3 nM
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CP0408419
|
3-(4,4-Dimethyl-2-oxo-1,4-dihydro-2H-benzo[d][1,3]oxazin-6-yl)-benzonitrile
Show/Hide
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C17H14N2O2
|
1
|
| 1 |
IC50 = 9.9 nM
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CP0082146
|
8-Fluoro-2,2,4-trimethyl-2,10-dihydro-1H-indeno[1,2-g]quinoline
Show/Hide
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C19H18FN
|
1
|
| 1 |
IC50 = 10 nM
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CP0496251
|
3-(4,4-Dimethyl-2-oxo-1,4-dihydro-2H-benzo[d][1,3]oxazin-6-yl)-5-fluoro-benzonitrile
Show/Hide
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C17H13FN2O2
|
2
|
| 1 |
IC50 = 15.9 nM
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| 2 |
IC50 = 16 nM
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CP0038093
|
3-Fluoro-5-(2,2,4-trimethyl-1,2-dihydro-quinolin-6-yl)-benzonitrile
Show/Hide
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C19H17FN2
|
1
|
| 1 |
IC50 = 30 nM
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CP0194317
|
2,2,4-Trimethyl-6-(5-nitro-thiophen-2-yl)-1,2-dihydro-quinoline
Show/Hide
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C16H16N2O2S
|
1
|
| 1 |
IC50 = 31 nM
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CP0196605
|
4-Methyl-5-(2,2,4-trimethyl-1,2-dihydro-quinolin-6-yl)-thiophene-2-carbonitrile
Show/Hide
|
C18H18N2S
|
1
|
| 1 |
IC50 = 33 nM
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CP0392781
|
6-(3-Chloro-4-fluoro-phenyl)-4,4-dimethyl-1,4-dihydro-benzo[d][1,3]oxazin-2-one
Show/Hide
|
C16H13ClFNO2
|
1
|
| 1 |
IC50 = 37 nM
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CP0038634
|
3-(2,2,4-Trimethyl-1,2-dihydro-quinolin-6-yl)-benzonitrile
Show/Hide
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C19H18N2
|
1
|
| 1 |
IC50 = 38 nM
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CP0392791
|
6-(3-Methoxy-phenyl)-4,4-dimethyl-1,4-dihydro-benzo[d][1,3]oxazin-2-one
Show/Hide
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C17H17NO3
|
1
|
| 1 |
IC50 = 38.3 nM
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CP0273183
|
4-(4,4-Dimethyl-2-oxo-1,4-dihydro-2H-benzo[d][1,3]oxazin-6-yl)-furan-2-carbonitrile
Show/Hide
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C15H12N2O3
|
1
|
| 1 |
IC50 = 40.2 nM
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CP0049604
|
2,2,4-Trimethyl-6-(3-nitro-phenyl)-1,2-dihydro-quinoline
Show/Hide
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C18H18N2O2
|
1
|
| 1 |
IC50 = 42 nM
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CP0254309
|
6-(5-Chloro-thiophen-2-yl)-2,2,4-trimethyl-1,2-dihydro-quinoline
Show/Hide
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C16H16ClNS
|
1
|
| 1 |
IC50 = 43 nM
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CP0352043
|
(5,8-difluoro-2,2,4-trimethyl-1,10-dihydroindeno[1,2-g]quinolin-10-yl) 2,2,2-trifluoroacetate
Show/Hide
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C21H16F5NO2
|
1
|
| 1 |
IC50 = 46 nM
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CP0106239
|
6,8,8-Trimethyl-4-trifluoromethyl-8,9-dihydro-1H-pyrido[3,2-g]quinolin-2-one
Show/Hide
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C16H15F3N2O
|
1
|
| 1 |
IC50 = 49 nM
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CP0082134
|
4-Bromo-5-(2,2,4-trimethyl-1,2-dihydro-quinolin-6-yl)-thiophene-2-carbonitrile
Show/Hide
|
C17H15BrN2S
|
1
|
| 1 |
IC50 = 52 nM
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CP0304316
|
5-(4,4-Dimethyl-2-oxo-1,4-dihydro-2H-benzo[d][1,3]oxazin-6-yl)-2-fluoro-benzonitrile
Show/Hide
|
C17H13FN2O2
|
1
|
| 1 |
IC50 = 55 nM
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CP0051504
|
2,2,4-Trimethyl-2,10-dihydro-1H-pyrido[2,3-b]carbazole
Show/Hide
|
C18H18N2
|
1
|
| 1 |
IC50 = 59 nM
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CP0110333
|
6-(5-Bromo-thiophen-2-yl)-2,2,4-trimethyl-1,2-dihydro-quinoline
Show/Hide
|
C16H16BrNS
|
1
|
| 1 |
IC50 = 65 nM
|
|
|
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CP0110336
|
6-(3-Fluoro-5-nitro-phenyl)-2,2,4-trimethyl-1,2-dihydro-quinoline
Show/Hide
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C18H17FN2O2
|
1
|
| 1 |
IC50 = 70 nM
|
|
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CP0332398
|
7,9-Difluoro-2,2,4-trimethyl-2,10-dihydro-1H-indeno[1,2-g]quinolin-10-ol
Show/Hide
|
C19H17F2NO
|
1
|
| 1 |
IC50 = 74 nM
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|
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CP0173385
|
6-(3,5-Difluoro-phenyl)-2,2,4-trimethyl-1,2-dihydro-quinoline
Show/Hide
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C18H17F2N
|
1
|
| 1 |
IC50 = 79 nM
|
|
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CP0245642
|
6,8-Difluoro-2,2,4-trimethyl-2,10-dihydro-1H-indeno[1,2-g]quinolin-10-ol
Show/Hide
|
C19H17F2NO
|
1
|
| 1 |
IC50 = 80 nM
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|
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CP0048931
|
2,2,4-trimethyl-8-nitro-2,10-dihydro-1H-indeno[1,2-g]quinoline
Show/Hide
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C19H18N2O2
|
1
|
| 1 |
IC50 = 90 nM
|
|
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CP0379086
|
3-Fluoro-5-(8-fluoro-4,4-dimethyl-2-oxo-1,4-dihydro-2H-benzo[d][1,3]oxazin-6-yl)-benzonitrile
Show/Hide
|
C17H12F2N2O2
|
1
|
| 1 |
IC50 = 98.8 nM
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CP0305347
|
6-Fluoro-2,2,4-trimethyl-2,10-dihydro-1H-indeno[1,2-g]quinolin-10-ol
Show/Hide
|
C19H18FNO
|
1
|
| 1 |
IC50 = 99 nM
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|
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CP0047802
|
7-Fluoro-2,2,4-trimethyl-8-nitro-2,10-dihydro-1H-indeno[1,2-g]quinoline
Show/Hide
|
C19H17FN2O2
|
1
|
| 1 |
IC50 = 100 nM
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CP0130624
|
4,6,8,8-Tetramethyl-8,9-dihydro-1H-pyrido[3,2-g]quinolin-2-one
Show/Hide
|
C16H18N2O
|
1
|
| 1 |
IC50 = 109 nM
|
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CP0040461
|
5-Methyl-4-(2,2,4-trimethyl-1,2-dihydro-quinolin-6-yl)-thiophene-2-carbonitrile
Show/Hide
|
C18H18N2S
|
1
|
| 1 |
IC50 = 109 nM
|
|
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CP0061790
|
8-Fluoro-2,2,4-trimethyl-2,10-dihydro-1H-indeno[1,2-g]quinolin-10-ol
Show/Hide
|
C19H18FNO
|
1
|
| 1 |
IC50 = 122 nM
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|
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CP0082136
|
3,5-Dimethyl-4-(2,2,4-trimethyl-1,2-dihydro-quinolin-6-yl)-thiophene-2-carbonitrile
Show/Hide
|
C19H20N2S
|
1
|
| 1 |
IC50 = 124 nM
|
|
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|
CP0778920
|
1-[9-Fluoro-2,2,4-trimethyl-1,2-dihydro-6-oxa-1-aza-chrysen-(5Z)-ylidene]-propan-2-one
Show/Hide
|
C22H20FNO2
|
1
|
| 1 |
IC50 = 124 nM
|
|
|
|
CP0101361
|
1,6,8,8,9-Pentamethyl-4-trifluoromethyl-8,9-dihydro-1H-pyrido[3,2-g]quinolin-2-one
Show/Hide
|
C18H19F3N2O
|
1
|
| 1 |
IC50 = 136 nM
|
|
|
|
CP0037261
|
6-fluoro-2,2,4-trimethyl-2,10-dihydro-1H-indeno[1,2-g]quinoline
Show/Hide
|
C19H18FN
|
1
|
| 1 |
IC50 = 146 nM
|
|
|
|
CP0079841
|
6,9-difluoro-2,2,4-trimethyl-2,10-dihydro-1H-indeno[1,2-g]quinoline
Show/Hide
|
C19H17F2N
|
1
|
| 1 |
IC50 = 146 nM
|
|
|
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CP0377494
|
(5bR,9aR)-1-Methyl-4-trifluoromethyl-1,5b,6,7,8,9,9a,10-octahydro-pyrido[2,3-b]carbazol-2-one
Show/Hide
|
C17H17F3N2O
|
1
|
| 1 |
IC50 = 150 nM
|
|
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CP0082141
|
6-Fluoro-2,2,4-trimethyl-1,2-dihydro-indeno[1,2-g]quinolin-10-one
Show/Hide
|
C19H16FNO
|
1
|
| 1 |
IC50 = 158 nM
|
|
|
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CP0283242
|
7-(4-nitrophenyl)-2-[4-(trifluoromethoxy)phenyl]sulfonyl-3,4,5,6-tetrahydrodiazepine
Show/Hide
|
C18H16F3N3O5S
|
1
|
| 1 |
IC50 = 158.49 nM
|
|
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CP0079750
|
5-Chloro-2,2,4-trimethyl-2,10-dihydro-1H-indeno[1,2-g]quinolin-10-ol
Show/Hide
|
C19H18ClNO
|
1
|
| 1 |
IC50 = 163 nM
|
|
|
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CP0082148
|
1-(2,2,4-Trimethyl-2,10-dihydro-1H-indeno[1,2-g]quinolin-8-yl)-ethanone
Show/Hide
|
C21H21NO
|
1
|
| 1 |
IC50 = 164 nM
|
|
|
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CP0460983
|
(5bR,9aR)-4-Trifluoromethyl-1,5b,6,7,8,9,9a,10-octahydro-pyrido[2,3-b]carbazol-2-one
Show/Hide
|
C16H15F3N2O
|
1
|
| 1 |
IC50 = 170 nM
|
|
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CP0308090
|
7-(3,4-dichlorophenyl)-2-(2,4-dichlorophenyl)sulfonyl-3,4,5,6-tetrahydrodiazepine
Show/Hide
|
C17H14Cl4N2O2S
|
1
|
| 1 |
IC50 = 199.53 nM
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CP0058424
|
2,2,4-Trimethyl-2,10-dihydro-1H-indeno[1,2-g]quinoline
Show/Hide
|
C19H19N
|
1
|
| 1 |
IC50 = 220 nM
|
|
|
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CP0041137
|
6,8,8-Trimethyl-4-trifluoromethyl-6,7,8,9-tetrahydro-1H-pyrido[3,2-g]quinolin-2-one
Show/Hide
|
C16H17F3N2O
|
1
|
| 1 |
IC50 = 231 nM
|
|
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CP0194318
|
2,2,4-Trimethyl-6-(3-methyl-thiophen-2-yl)-1,2-dihydro-quinoline
Show/Hide
|
C17H19NS
|
1
|
| 1 |
IC50 = 232 nM
|
|
|
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CP0295804
|
1,6,8,8-Tetramethyl-4-trifluoromethyl-8,9-dihydro-1H-pyrido[3,2-g]quinolin-2-one
Show/Hide
|
C17H17F3N2O
|
1
|
| 1 |
IC50 = 233 nM
|
|
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CP0041367
|
3-Bromo-5-(2,2,4-trimethyl-1,2-dihydro-quinolin-6-yl)-thiophene-2-carbonitrile
Show/Hide
|
C17H15BrN2S
|
1
|
| 1 |
IC50 = 242 nM
|
|
|
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CP0226810
|
(2Z)-2-(9-fluoro-2,2,4-trimethyl-1H-chromeno[3,4-f]quinolin-5-ylidene)acetaldehyde
Show/Hide
|
C21H18FNO2
|
1
|
| 1 |
IC50 = 243 nM
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|
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CP0082137
|
4-(2,2,4-Trimethyl-1,2-dihydro-quinolin-6-yl)-thiophene-2-carbaldehyde
Show/Hide
|
C17H17NOS
|
1
|
| 1 |
IC50 = 245 nM
|
|
|
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CP0194320
|
8-chloro-2,2,4-trimethyl-2,10-dihydro-1H-indeno[1,2-g]quinoline
Show/Hide
|
C19H18ClN
|
1
|
| 1 |
IC50 = 248 nM
|
|
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CP0453010
|
7-(3-bromophenyl)-2-(5-bromothiophen-2-yl)sulfonyl-3,4,5,6-tetrahydrodiazepine
Show/Hide
|
C15H14Br2N2O2S2
|
1
|
| 1 |
IC50 = 251.19 nM
|
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CP0150490
|
4,6,6-trimethyl-2-methylidene-1-[(4-nitrophenyl)methyl]cyclohex-3-en-1-ol
Show/Hide
|
C17H21NO3
|
1
|
| 1 |
IC50 = 260 nM
|
|
|
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CP0332143
|
6-Ethyl-8,8-dimethyl-4-trifluoromethyl-6,7,8,9-tetrahydro-1H-pyrido[3,2-g]quinolin-2-one
Show/Hide
|
C17H19F3N2O
|
1
|
| 1 |
IC50 = 274 nM
|
|
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CP0134882
|
11-Ethyl-1,3,3-trimethyl-4,11-dihydro-3H-pyrido[3,2-a]carbazole
Show/Hide
|
C20H22N2
|
1
|
| 1 |
IC50 = 284 nM
|
|
|
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CP0161755
|
(6R,7S)-6,7,8,8-Tetramethyl-4-trifluoromethyl-6,7,8,9-tetrahydro-1H-pyrido[3,2-g]quinolin-2-one
Show/Hide
|
C17H19F3N2O
|
1
|
| 1 |
IC50 = 310 nM
|
|
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CP0084521
|
2-(5-bromothiophen-2-yl)sulfonyl-7-(3,4-dichlorophenyl)-3,4,5,6-tetrahydrodiazepine
Show/Hide
|
C15H13BrCl2N2O2S2
|
1
|
| 1 |
IC50 = 316.23 nM
|
|
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CP0164926
|
3-(2,2,4-Trimethyl-1,2-dihydro-quinolin-6-yl)-thiophene-2-carbonitrile
Show/Hide
|
C17H16N2S
|
1
|
| 1 |
IC50 = 318 nM
|
|
|
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CP0187275
|
8,8-Dimethyl-4-trifluoromethyl-6,7,8,9-tetrahydro-1H-pyrido[3,2-g]quinolin-2-one
Show/Hide
|
C15H15F3N2O
|
1
|
| 1 |
IC50 = 330 nM
|
|
|
|
CP0220774
|
7,8,8-Trimethyl-4-trifluoromethyl-6,7,8,9-tetrahydro-1H-pyrido[3,2-g]quinolin-2-one
Show/Hide
|
C16H17F3N2O
|
1
|
| 1 |
IC50 = 348 nM
|
|
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|
CP0183617
|
2,2,4-Trimethyl-1,2-dihydro-indeno[1,2-g]quinolin-10-one
Show/Hide
|
C19H17NO
|
1
|
| 1 |
IC50 = 353 nM
|
|
|
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CP0368335
|
6,7,7,8,8-Pentamethyl-4-trifluoromethyl-6,7,8,9-tetrahydro-1H-pyrido[3,2-g]quinolin-2-one
Show/Hide
|
C18H21F3N2O
|
1
|
| 1 |
IC50 = 362 nM
|
|
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|
CP0307544
|
5,8-Difluoro-2,2,4-trimethyl-1,2-dihydro-indeno[1,2-g]quinolin-10-one
Show/Hide
|
C19H15F2NO
|
1
|
| 1 |
IC50 = 365 nM
|
|
|
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CP0062175
|
5-(4-Chloro-phenyl)-2,2-dimethyl-2,3-dihydro-1H,5H-6-oxa-1-aza-chrysen-4-one
Show/Hide
|
C24H20ClNO2
|
1
|
| 1 |
IC50 = 376 nM
|
|
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|
CP0377889
|
(5bR,7S,9aR)-1,7-Dimethyl-4-trifluoromethyl-1,5b,6,7,8,9,9a,10-octahydro-pyrido[2,3-b]carbazol-2-one
Show/Hide
|
C18H19F3N2O
|
1
|
| 1 |
IC50 = 380 nM
|
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CP0163588
|
8,8-dimethyl-4-(trifluoromethyl)-1H,2H,8H,9H-pyrido[3,2-g]quinolin-2-one
Show/Hide
|
C15H13F3N2O
|
1
|
| 1 |
IC50 = 390 nM
|
|
|
|
CP0088296
|
6,7,8,8-Tetramethyl-4-trifluoromethyl-8,9-dihydro-1H-pyrido[3,2-g]quinolin-2-one
Show/Hide
|
C17H17F3N2O
|
1
|
| 1 |
IC50 = 393 nM
|
|
|
|
CP0352184
|
3a,10-Dimethyl-7-trifluoromethyl-1,2,3a,4,5,10-hexahydro-3H-10,11b-diaza-cyclopenta[a]anthracen-9-one
Show/Hide
|
C18H19F3N2O
|
1
|
| 1 |
IC50 = 398 nM
|
|
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|
CP0308089
|
4-[2-(2-fluorophenyl)sulfonyl-3,4,5,6-tetrahydrodiazepin-7-yl]benzonitrile
Show/Hide
|
C18H16FN3O2S
|
1
|
| 1 |
IC50 = 398.11 nM
|
|
|
|
CP0077038
|
11-butyl-1,3,3-trimethyl-4,11-dihydro-3H-pyrido[3,2-a]carbazole
Show/Hide
|
C22H26N2
|
1
|
| 1 |
IC50 = 416 nM
|
|
|
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CP0110335
|
2,2,4-Trimethyl-6-thiophen-2-yl-1,2-dihydro-quinoline
Show/Hide
|
C16H17NS
|
1
|
| 1 |
IC50 = 416 nM
|
|
|
|
CP0060654
|
2,2,4-Trimethyl-2,3,4,10-tetrahydro-1H-indeno[1,2-g]quinoline
Show/Hide
|
C19H21N
|
1
|
| 1 |
IC50 = 424 nM
|
|
|
|
CP0375432
|
(5bR,9aR)-5b,9,9-Trimethyl-4-trifluoromethyl-1,5b,6,7,8,9,9a,10-octahydro-pyrido[2,3-b]carbazol-2-one
Show/Hide
|
C19H21F3N2O
|
1
|
| 1 |
IC50 = 430 nM
|
|
|
|
CP0149090
|
8-bromo-2,2,4-trimethyl-2,10-dihydro-1H-indeno[1,2-g]quinoline
Show/Hide
|
C19H18BrN
|
1
|
| 1 |
IC50 = 434 nM
|
|
|
|
CP0213900
|
(3R,4S,5S)-5-(4-Chloro-phenyl)-2,2,4-trimethyl-2,3,4,5-tetrahydro-1H-6-oxa-1-aza-chrysen-3-ol
Show/Hide
|
C25H24ClNO2
|
1
|
| 1 |
IC50 = 460 nM
|
|
|
|
CP0352052
|
10-Fluoro-1,3,3-trimethyl-4,11-dihydro-3H-indeno[2,1-f]quinoline
Show/Hide
|
C19H18FN
|
1
|
| 1 |
IC50 = 496 nM
|
|
|
|
CP0436398
|
6-(2-Chloro-phenyl)-4,4-dimethyl-1,4-dihydro-benzo[d][1,3]oxazin-2-one
Show/Hide
|
C16H14ClNO2
|
1
|
| 1 |
IC50 = 500 nM
|
|
|
|
CP0285450
|
2-(4-chlorophenyl)sulfonyl-7-(3-fluorophenyl)-3,4,5,6-tetrahydrodiazepine
Show/Hide
|
C17H16ClFN2O2S
|
1
|
| 1 |
IC50 = 501.19 nM
|
|
|
|
CP0276572
|
8-Ethyl-8-methyl-4-trifluoromethyl-6,7,8,9-tetrahydro-1H-pyrido[3,2-g]quinolin-2-one
Show/Hide
|
C16H17F3N2O
|
1
|
| 1 |
IC50 = 543 nM
|
|
|
|
CP0123816
|
5-Bromo-2-((1S,3R)-3-bromo-2,2-dimethyl-6-methylene-cyclohexylmethyl)-4-methoxy-phenol
Show/Hide
|
C17H22Br2O2
|
1
|
| 1 |
IC50 = 549 nM
|
|
|
|
CP0293868
|
1,3,3-trimethyl-4,11-dihydro-3H-indeno[2,1-f]quinoline
Show/Hide
|
C19H19N
|
1
|
| 1 |
IC50 = 549 nM
|
|
|
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CP0214113
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5-Bromo-4-methoxy-2-(2,6,6-trimethyl-4-methylene-cyclohex-2-enylmethyl)-phenol
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C18H23BrO2
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1
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| 1 |
IC50 = 580 nM
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CP0198388
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1,6,8,8-Tetramethyl-4-trifluoromethyl-6,7,8,9-tetrahydro-1H-pyrido[3,2-g]quinolin-2-one
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C17H19F3N2O
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1
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| 1 |
IC50 = 585 nM
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CP0104916
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2,2,4-Trimethyl-2,10-dihydro-1H-indeno[1,2-g]quinolin-10-ol
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C19H19NO
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1
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| 1 |
IC50 = 609 nM
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CP0276908
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7-(2-chlorophenyl)-2-(5-chlorothiophen-2-yl)sulfonyl-3,4,5,6-tetrahydrodiazepine
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C15H14Cl2N2O2S2
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1
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| 1 |
IC50 = 630.96 nM
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CP0448642
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6-(4-Chloro-phenyl)-4,4-dimethyl-1,4-dihydro-benzo[d][1,3]oxazin-2-one
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C16H14ClNO2
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1
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| 1 |
IC50 = 642 nM
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CP0276761
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Acetic acid 5-bromo-4-methoxy-2-((S)-3,6,6-trimethyl-2-methylene-cyclohex-3-enylmethyl)-phenyl ester
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C20H25BrO3
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1
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| 1 |
IC50 = 660 nM
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CP0292001
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1,3,3-Trimethyl-4,11-dihydro-3H-pyrido[3,2-a]carbazole
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C18H18N2
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1
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| 1 |
IC50 = 662 nM
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CP0377845
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5-(2,2,4-Trimethyl-1,2-dihydro-quinolin-6-yl)-thiophene-2-carbaldehyde
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C17H17NOS
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1
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| 1 |
IC50 = 729 nM
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CP0463444
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(5bR,9aR)-5b-Methyl-4-trifluoromethyl-1,5b,6,7,8,9,9a,10-octahydro-pyrido[2,3-b]carbazol-2-one
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C17H17F3N2O
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1
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| 1 |
IC50 = 730 nM
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CP0208002
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(6S,7S)-6,7,8,8-Tetramethyl-4-trifluoromethyl-6,7,8,9-tetrahydro-1H-pyrido[3,2-g]quinolin-2-one
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C17H19F3N2O
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1
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| 1 |
IC50 = 735 nM
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CP0037637
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(R)-5-bromo-2-((2,2-dimethyl-6-methylenecyclohexyl)methyl)-4-methoxyphenol
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C17H23BrO2
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1
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| 1 |
IC50 = 741 nM
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CP0393742
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(R)-2-Methyl-5-trifluoromethyl-1,2,3,8-tetrahydro-pyrrolo[3,2-g]quinolin-7-one
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C13H11F3N2O
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1
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| 1 |
IC50 = 750 nM
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CP0192843
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6-(3-Fluoro-phenyl)-2,2,4-trimethyl-1,2-dihydro-quinoline
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C18H18FN
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1
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| 1 |
IC50 = 750 nM
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CP0079027
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5-Bromo-2-(6,6-dimethyl-2-methylene-cyclohex-3-enylmethyl)-4-methoxy-phenol
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C17H21BrO2
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1
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| 1 |
IC50 = 783 nM
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CP0280284
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2,2,4-Trimethyl-6-phenyl-1,2-dihydro-quinoline
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C18H19N
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1
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| 1 |
IC50 = 783 nM
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CP0272980
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7,7,8,8-Tetramethyl-4-trifluoromethyl-6,7,8,9-tetrahydro-1H-pyrido[3,2-g]quinolin-2-one
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C17H19F3N2O
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1
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| 1 |
IC50 = 876 nM
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CP0079028
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5-Bromo-2-((1S,2R,4R)-2,4-dimethyl-6-methylene-cyclohexylmethyl)-4-methoxy-phenol
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C17H23BrO2
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1
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| 1 |
IC50 = 985 nM
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CP0374711
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(5bR,9aR)-1,10-Dimethyl-4-trifluoromethyl-1,5b,6,7,8,9,9a,10-octahydro-pyrido[2,3-b]carbazol-2-one
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C18H19F3N2O
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1
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| 1 |
IC50 = 1000 nM
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CP0102103
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5-Bromo-4-methoxy-2-((1R,2S)-2-methyl-6-methylene-cyclohexylmethyl)-phenol
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C16H21BrO2
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1
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| 1 |
IC50 = 1050 nM
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CP0184817
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1-Nitro-4-(4,6,6-trimethyl-2-methylene-cyclohex-3-enylmethyl)-benzene
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C17H21NO2
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1
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| 1 |
IC50 = 1050 nM
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CP0041439
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8-Ethyl-1,8,9-trimethyl-4-trifluoromethyl-6,7,8,9-tetrahydro-1H-pyrido[3,2-g]quinolin-2-one
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C18H21F3N2O
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1
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| 1 |
IC50 = 1105 nM
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CP0320204
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1,3,3-Trimethyl-3,4-dihydro-benzo[4,5]furo[2,3-f]quinoline
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C18H17NO
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1
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| 1 |
IC50 = 1144 nM
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CP0216906
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8-Methyl-8-propyl-4-trifluoromethyl-6,7,8,9-tetrahydro-1H-pyrido[3,2-g]quinolin-2-one
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C17H19F3N2O
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1
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| 1 |
IC50 = 1144 nM
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CP0150041
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5-Bromo-2-(2,2-dimethyl-5-methylene-cyclopentylmethyl)-4-methoxy-phenol
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C16H21BrO2
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1
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| 1 |
IC50 = 1200 nM
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CP0246106
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1,8,8-Trimethyl-4-trifluoromethyl-6,7,8,9-tetrahydro-1H-pyrido[3,2-g]quinolin-2-one
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C16H17F3N2O
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1
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| 1 |
IC50 = 1239 nM
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CP0285440
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7-(4-chlorophenyl)-2-(3-chlorophenyl)sulfonyl-3,4,5,6-tetrahydrodiazepine
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C17H16Cl2N2O2S
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1
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| 1 |
IC50 = 1258.93 nM
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CP0041214
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1-Nitro-4-(4,6,6-trimethyl-2-methylene-cyclohex-3-enylsulfanyl)-benzene
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C16H19NO2S
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1
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| 1 |
IC50 = 1350 nM
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CP0221713
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1,3,3-Trimethyl-9-nitro-4,11-dihydro-3H-indeno[2,1-f]quinoline
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C19H18N2O2
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1
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| 1 |
IC50 = 1674 nM
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CP0267990
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6,8,8,9-Tetramethyl-4-trifluoromethyl-8,9-dihydro-1H-pyrido[3,2-g]quinolin-2-one
Show/Hide
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C17H17F3N2O
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1
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| 1 |
IC50 = 1678 nM
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CP0043208
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1-Ethyl-6,8,8-trimethyl-4-trifluoromethyl-8,9-dihydro-1H-pyrido[3,2-g]quinolin-2-one
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C18H19F3N2O
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1
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| 1 |
IC50 = 1763 nM
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CP0082084
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9-Fluoro-2,2,4-trimethyl-2,10-dihydro-1H-indeno[1,2-g]quinoline
Show/Hide
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C19H18FN
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1
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| 1 |
IC50 = 1772 nM
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CP0142838
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2-Methyl-1-nitro-4-(4,6,6-trimethyl-2-methylene-cyclohex-3-enylmethyl)-benzene
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C18H23NO2
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1
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| 1 |
IC50 = 1800 nM
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CP0146696
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Bicalutamide
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C18H14F4N2O4S
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1
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| 1 |
IC50 = 1819 nM
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CP0041438
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6'-trifluoromethylspiro[cyclohexane-1,2'-(1',2',3',4',8',9'-hexahydropyrido[3,2-g]quinoline)]-8'-one
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C18H19F3N2O
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1
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| 1 |
IC50 = 1828 nM
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CP0082144
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2,2,4-Trimethyl-1,2-dihydro-benzo[4,5]furo[3,2-g]quinoline
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C18H17NO
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1
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| 1 |
IC50 = 1847 nM
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CP0407007
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(2R,3R)-2,3-Dimethyl-5-trifluoromethyl-1,2,3,8-tetrahydro-pyrrolo[3,2-g]quinolin-7-one
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C14H13F3N2O
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1
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| 1 |
IC50 = 1900 nM
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CP0185471
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5-diphenylmethylene-2,2,4-trimethyl-2,5-dihydro-1H-chromeno[3,4-f]quinolin-9-yl fluoride
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C32H26FNO
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1
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| 1 |
IC50 = 1930 nM
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CP0041695
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5-(4,6,6-Trimethyl-2-methylene-cyclohex-3-enylmethyl)-benzo[1,2,5]oxadiazole
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C17H20N2O
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1
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| 1 |
IC50 = 1950 nM
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CP0285449
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2-(3-chloro-2-methylphenyl)sulfonyl-7-(3-chlorophenyl)-3,4,5,6-tetrahydrodiazepine
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C18H18Cl2N2O2S
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1
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| 1 |
IC50 = 1995.26 nM
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CP0122190
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5-Bromo-2-((1S,5R)-5-hydroxy-2,2,5-trimethyl-6-methylene-cyclohexylmethyl)-4-methoxy-phenol
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C18H25BrO3
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1
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| 1 |
IC50 = 2000 nM
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CP0040191
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2-Hydroxy-2-methyl-N-(4-nitro-3-trifluoromethyl-phenyl)-propionamide
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C11H11F3N2O4
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1
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| 1 |
IC50 = 2013 nM
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CP0215260
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1,8,8,9-Tetramethyl-4-trifluoromethyl-6,7,8,9-tetrahydro-1H-pyrido[3,2-g]quinolin-2-one
Show/Hide
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C17H19F3N2O
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1
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| 1 |
IC50 = 2200 nM
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CP0206243
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9-Bromo-1,3,3-trimethyl-4,11-dihydro-3H-indeno[2,1-f]quinoline
Show/Hide
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C19H18BrN
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1
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| 1 |
IC50 = 2330 nM
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CP0292537
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7-Ethyl-8,8-dimethyl-4-trifluoromethyl-6,7,8,9-tetrahydro-1H-pyrido[3,2-g]quinolin-2-one
Show/Hide
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C17H19F3N2O
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1
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| 1 |
IC50 = 2334 nM
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CP0041245
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3-Ethoxy-5,5-dimethyl-6-(4-nitro-benzyl)-cyclohex-2-enone
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C17H21NO4
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1
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| 1 |
IC50 = 2443 nM
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CP0102250
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8,8-Diethyl-4-trifluoromethyl-6,7,8,9-tetrahydro-1H-pyrido[3,2-g]quinolin-2-one
Show/Hide
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C17H19F3N2O
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1
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| 1 |
IC50 = 2708 nM
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CP0237260
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1,6,8,8,10-Pentamethyl-4-trifluoromethyl-6,7,8,9-tetrahydro-1H-pyrido[3,2-g]quinolin-2-one
Show/Hide
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C18H21F3N2O
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1
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| 1 |
IC50 = 2931 nM
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CP0141600
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6-Isopropyl-8,8-dimethyl-4-trifluoromethyl-6,7,8,9-tetrahydro-1H-pyrido[3,2-g]quinolin-2-one
Show/Hide
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C18H21F3N2O
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1
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| 1 |
IC50 = 3162 nM
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CP0049970
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(3S,4R,5S)-5-(4-Chloro-phenyl)-2,2,4-trimethyl-2,3,4,5-tetrahydro-1H-6-oxa-1-aza-chrysen-3-ol
Show/Hide
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C25H24ClNO2
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1
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| 1 |
IC50 = 3200 nM
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CP0036037
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8-Ethyl-1,8-dimethyl-4-trifluoromethyl-6,7,8,9-tetrahydro-1H-pyrido[3,2-g]quinolin-2-one
Show/Hide
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C17H19F3N2O
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1
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| 1 |
IC50 = 3277 nM
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CP0043286
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5-Bromo-2-((1S,4R)-4-hydroxymethyl-2,2-dimethyl-6-methylene-cyclohexylmethyl)-4-methoxy-phenol
Show/Hide
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C18H25BrO3
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1
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| 1 |
IC50 = 3300 nM
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CP0289340
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8-fluoro-1,3,3-trimethyl-9-nitro-4,11-dihydro-3H-indeno[2,1-f]quinoline
Show/Hide
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C19H17FN2O2
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1
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| 1 |
IC50 = 3331 nM
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CP0328159
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6,8,8,10-Tetramethyl-4-trifluoromethyl-8,9-dihydro-1H-pyrido[3,2-g]quinolin-2-one
Show/Hide
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C17H17F3N2O
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1
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| 1 |
IC50 = 3346 nM
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CP0088803
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5-Bromo-2-((1S,5R)-5-hydroxy-2,2-dimethyl-6-methylene-cyclohexylmethyl)-4-methoxy-phenol
Show/Hide
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C17H23BrO3
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1
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| 1 |
IC50 = 3400 nM
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CP0037585
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8-Bromo-2,2,4-trimethyl-2,10-dihydro-1H-indeno[1,2-g]quinolin-10-ol
Show/Hide
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C19H18BrNO
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1
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| 1 |
IC50 = 3443 nM
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CP0316819
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6,8,8,10-Tetramethyl-4-trifluoromethyl-6,7,8,9-tetrahydro-1H-pyrido[3,2-g]quinolin-2-one
Show/Hide
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C17H19F3N2O
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1
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| 1 |
IC50 = 3726 nM
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CP0259897
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1,6,8,8,10-Pentamethyl-4-trifluoromethyl-8,9-dihydro-1H-pyrido[3,2-g]quinolin-2-one
Show/Hide
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C18H19F3N2O
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1
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| 1 |
IC50 = 4395 nM
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CP0267930
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6,9-Difluoro-1,3,3-trimethyl-4,11-dihydro-3H-indeno[2,1-f]quinoline
Show/Hide
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C19H17F2N
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1
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| 1 |
IC50 = 5685 nM
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CP0134478
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8-Bromo-2,2,4,10-tetramethyl-2,10-dihydro-1H-indeno[1,2-g]quinoline
Show/Hide
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C20H20BrN
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1
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| 1 |
IC50 = 10000 nM
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CP0183440
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5,8-Difluoro-2,2,4,10-tetramethyl-2,10-dihydro-1H-indeno[1,2-g]quinolin-10-ol
Show/Hide
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C20H19F2NO
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1
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| 1 |
IC50 = 10000 nM
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CP0298284
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6,9-Difluoro-1,3,3-trimethyl-4,11-dihydro-3H-indeno[2,1-f]quinolin-11-ol
Show/Hide
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C19H17F2NO
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1
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| 1 |
IC50 = 10000 nM
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CP0307445
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(2,2,4-Trimethyl-2,10-dihydro-1H-indeno[1,2-g]quinolin-9-yl)-methanol
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C20H21NO
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1
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| 1 |
IC50 = 10000 nM
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CP0332290
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10-Benzyl-8-bromo-2,2,4-trimethyl-2,10-dihydro-1H-indeno[1,2-g]quinoline
Show/Hide
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C26H24BrN
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1
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| 1 |
IC50 = 10000 nM
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CP0087434
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3a-Methyl-7-trifluoromethyl-1,2,3a,4,5,10-hexahydro-3H-10,11b-diaza-cyclopenta[a]anthracen-9-one
Show/Hide
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C17H17F3N2O
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1
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| 1 |
IC50 > 10000 nM
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CP0060594
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WAY-362450
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C25H24F2N2O3
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1
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| 1 |
IC50 = 10000 nM
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CP0041854
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6-chloro-3,20-dioxo-1beta,2beta-dihydro-3'H-cyclopropa[1,2]pregna-4,6-dien-17-yl acetate
Show/Hide
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C24H29ClO4
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1
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| 1 |
IC50 > 1000 nM
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CP0333121
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(4S)-2-(4-chlorophenyl)sulfonyl-5-(3,4-dichlorophenyl)-4-methyl-3,4-dihydropyrazole
Show/Hide
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C16H13Cl3N2O2S
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1
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| 1 |
Ki = 25.12 nM
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CP0318808
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2-(4-chlorophenyl)sulfonyl-5-(3,4-dichlorophenyl)-3-methyl-3,4-dihydropyrazole
Show/Hide
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C16H13Cl3N2O2S
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1
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| 1 |
Ki = 199.53 nM
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CP0295424
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2-(4-chlorophenyl)sulfonyl-5-(3,4-dichlorophenyl)-3-phenyl-3,4-dihydropyrazole
Show/Hide
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C21H15Cl3N2O2S
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1
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| 1 |
Ki = 398.11 nM
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CP0276747
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4-[2-(4-chlorophenyl)sulfonyl-5-(3,4-dichlorophenyl)-3,4-dihydropyrazol-4-yl]-N,N-dimethylaniline
Show/Hide
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C23H20Cl3N3O2S
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1
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| 1 |
Ki = 794.33 nM
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CP0269257
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4-[(4R)-2-(4-chlorophenyl)sulfonyl-5-(3,4-dichlorophenyl)-3,4-dihydropyrazol-4-yl]-N,N-dimethylaniline
Show/Hide
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C23H20Cl3N3O2S
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1
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| 1 |
Ki = 1584.89 nM
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CP0273126
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(4R)-2-(4-chlorophenyl)sulfonyl-5-(3,4-dichlorophenyl)-4-methyl-3,4-dihydropyrazole
Show/Hide
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C16H13Cl3N2O2S
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1
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| 1 |
Ki = 5011.87 nM
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CP0246097
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4-[(4S)-2-(4-chlorophenyl)sulfonyl-5-(3,4-dichlorophenyl)-3,4-dihydropyrazol-4-yl]-N,N-dimethylaniline
Show/Hide
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C23H20Cl3N3O2S
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1
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| 1 |
Ki < 3162.28 nM
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