Brief Information of the Compound and Protein
Compound Name
(R)-3-(4-(3-(1-(5-chloro-1,3-dimethyl-1H-indole-2-carboxamido)ethyl)-5-fluorophenoxy)-2-ethylphenyl)propanoic acid
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PubChem ID
CID: 24754924
SID: 49657721
Canonical SMILES
CCc1cc(Oc2cc(F)cc(c2)[C@@H](C)NC(=O)c2c(C)c3cc(Cl)ccc3n2C)ccc1CCC(O)=O
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Compound Formula C30H30ClFN2O4
Compound Structure
Protein Name
Peroxisome proliferator-activated receptor delta
Protein Classification
Transcription factor
>
Nuclear receptor
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Nuclear hormone receptor subfamily 1
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Nuclear hormone receptor subfamily 1 group C
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Nuclear hormone receptor subfamily 1 group C member 2
Uniprot ID
Q03181
Gene Name
PPARD
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000044 CV-1 Chlorocebus aethiops (Green monkey)  1
1
EC50 = 1 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 IC50 = 5 nM