Brief Information of the Compound and Protein
Compound Name
US9163012, 65
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Canonical SMILES
N#Cc1ccc2[nH]c(=O)n([C@@H]3CCN(C(=O)O[C@H]4C5CC6CC4C[C@](C(N)=O)(C6)C5)C3)c2c1
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Compound Formula C24H27N5O4
Compound Structure
Protein Name
11-beta-hydroxysteroid dehydrogenase 1
Protein Classification
Enzyme
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Oxidoreductase
Uniprot ID
P28845
Gene Name
HSD11B1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
IC50 = 33.3 nM
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