| Compound ID |
Compound Name |
Compound Formula |
|
CP0502246
|
CAS_52906-92-0
Show/Hide
|
C120H188N34O35S
|
1
|
| 1 |
EC50 = 0.03981 nM
|
|
|
|
CP0916579
|
MOTILIN_030
Show/Hide
|
C26H29FN4O
|
1
|
| 1 |
EC50 = 0.2512 nM
|
|
|
|
CP0941021
|
MOTILIN_050
Show/Hide
|
C26H29FN4O2
|
1
|
| 1 |
EC50 = 0.2512 nM
|
|
|
|
CP0950895
|
MOTILIN_055
Show/Hide
|
C25H26ClFN4O2
|
1
|
| 1 |
EC50 = 0.3162 nM
|
|
|
|
CP0916582
|
MOTILIN_056
Show/Hide
|
C26H29FN4O2
|
1
|
| 1 |
EC50 = 0.3981 nM
|
|
|
|
CP0954964
|
MOTILIN_023
Show/Hide
|
C27H31FN4O
|
1
|
| 1 |
EC50 = 0.3981 nM
|
|
|
|
CP0931906
|
MOTILIN_020
Show/Hide
|
C26H29FN4O
|
1
|
| 1 |
EC50 = 0.631 nM
|
|
|
|
CP0941020
|
MOTILIN_040
Show/Hide
|
C26H29FN4O
|
1
|
| 1 |
EC50 = 0.7943 nM
|
|
|
|
CP0952070
|
MOTILIN_068
Show/Hide
|
C25H31FN6O
|
1
|
| 1 |
EC50 = 0.7943 nM
|
|
|
|
CP0857174
|
MOTILIN_064
Show/Hide
|
C29H34FN5O
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0957584
|
MOTILIN_035
Show/Hide
|
C25H27FN4O2
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0851100
|
MOTILIN_067
Show/Hide
|
C26H33FN6O
|
1
|
| 1 |
EC50 = 1.259 nM
|
|
|
|
CP0952063
|
MOTILIN_019
Show/Hide
|
C25H27FN4O
|
1
|
| 1 |
EC50 = 1.259 nM
|
|
|
|
CP0954966
|
MOTILIN_039
Show/Hide
|
C25H26F2N4O
|
1
|
| 1 |
EC50 = 1.259 nM
|
|
|
|
CP0851099
|
MOTILIN_058
Show/Hide
|
C24H24F4N4O2S
|
1
|
| 1 |
EC50 = 1.585 nM
|
|
|
|
CP0869010
|
MOTILIN_026
Show/Hide
|
C25H28FN5O
|
1
|
| 1 |
EC50 = 1.585 nM
|
|
|
|
CP0931903
|
MOTILIN_015
Show/Hide
|
C25H27FN4O
|
1
|
| 1 |
EC50 = 1.585 nM
|
|
|
|
CP0952064
|
MOTILIN_022
Show/Hide
|
C27H29N5O
|
1
|
| 1 |
EC50 = 1.585 nM
|
|
|
|
CP0957586
|
MOTILIN_053
Show/Hide
|
C24H27FN4O2S
|
1
|
| 1 |
EC50 = 1.585 nM
|
|
|
|
CP0921486
|
MOTILIN_059
Show/Hide
|
C25H28FN5O2
|
1
|
| 1 |
EC50 = 1.995 nM
|
|
|
|
CP0952065
|
MOTILIN_024
Show/Hide
|
C26H29FN4O
|
1
|
| 1 |
EC50 = 1.995 nM
|
|
|
|
CP0954965
|
MOTILIN_037
Show/Hide
|
C26H27N5O2
|
1
|
| 1 |
EC50 = 1.995 nM
|
|
|
|
CP0954973
|
MOTILIN_061
Show/Hide
|
C26H34FN7
|
1
|
| 1 |
EC50 = 1.995 nM
|
|
|
|
CP0073984
|
4-butyl-N-[3-(1H-pyrazol-5-ylmethyl)-1,2,4,5-tetrahydro-3-benzazepin-7-yl]benzenesulfonamide
Show/Hide
|
C24H30N4O2S
|
1
|
| 1 |
EC50 = 2.512 nM
|
|
|
|
CP0916578
|
MOTILIN_021
Show/Hide
|
C26H28FN3O2
|
1
|
| 1 |
EC50 = 2.512 nM
|
|
|
|
CP0931902
|
MOTILIN_014
Show/Hide
|
C26H33F3N4O
|
1
|
| 1 |
EC50 = 2.512 nM
|
|
|
|
CP0952069
|
MOTILIN_066
Show/Hide
|
C26H33FN6O
|
1
|
| 1 |
EC50 = 2.512 nM
|
|
|
|
CP0360673
|
4-butyl-N-[3-[(5-methyl-1H-imidazol-4-yl)methyl]-1,2,4,5-tetrahydro-3-benzazepin-7-yl]benzenesulfonamide
Show/Hide
|
C25H32N4O2S
|
1
|
| 1 |
EC50 = 3.162 nM
|
|
|
|
CP0922273
|
MOTILIN_033
Show/Hide
|
C26H27N5O2
|
1
|
| 1 |
EC50 = 3.162 nM
|
|
|
|
CP0931901
|
MOTILIN_013
Show/Hide
|
C26H33N5O
|
1
|
| 1 |
EC50 = 3.162 nM
|
|
|
|
CP0931908
|
MOTILIN_036
Show/Hide
|
C25H26F2N4O2
|
1
|
| 1 |
EC50 = 3.162 nM
|
|
|
|
CP0035877
|
(3-(4-(((3R,5S)-3,5-dimethylpiperazin-1-yl)methyl)phenyl)pyridin-2-yl)(4-(4-fluorophenylamino)piperidin-1-yl)methanone
Show/Hide
|
C30H36FN5O
|
1
|
| 1 |
EC50 = 3.981 nM
|
|
|
|
CP0394499
|
3-((1-[(4-([(3S)-3-Methyl-1-piperazinyl]methyl)phenyl)acetyl]-4-piperidinyl)amino)benzonitrile
Show/Hide
|
C26H33N5O
|
1
|
| 1 |
EC50 = 3.981 nM
|
|
|
|
CP0354687
|
4-propan-2-yloxy-N-[3-(1H-pyrazol-5-ylmethyl)-1,2,4,5-tetrahydro-3-benzazepin-7-yl]benzenesulfonamide
Show/Hide
|
C23H28N4O3S
|
1
|
| 1 |
EC50 = 3.981 nM
|
|
|
|
CP0360495
|
7-((6-(4-fluorophenyl)pyridin-3-ylsulfonyl)methyl)-2,3,4,5-tetrahydro-1H-benzo[d]azepine
Show/Hide
|
C22H21FN2O2S
|
1
|
| 1 |
EC50 = 5.012 nM
|
|
|
|
CP0376525
|
2,2-dimethyl-N-[3-(1H-pyrazol-5-ylmethyl)-1,2,4,5-tetrahydro-3-benzazepin-7-yl]-3,4-dihydrochromene-6-sulfonamide
Show/Hide
|
C25H30N4O3S
|
1
|
| 1 |
EC50 = 5.012 nM
|
|
|
|
CP0857169
|
MOTILIN_028
Show/Hide
|
C25H32ClFN4O
|
1
|
| 1 |
EC50 = 5.012 nM
|
|
|
|
CP0921485
|
MOTILIN_018
Show/Hide
|
C25H27FN4O
|
1
|
| 1 |
EC50 = 5.012 nM
|
|
|
|
CP0931905
|
MOTILIN_017
Show/Hide
|
C26H35FN4O
|
1
|
| 1 |
EC50 = 5.012 nM
|
|
|
|
CP0952066
|
MOTILIN_027
Show/Hide
|
C24H26FN5O
|
1
|
| 1 |
EC50 = 5.012 nM
|
|
|
|
CP0957583
|
MOTILIN_025
Show/Hide
|
C26H28FN3O2
|
1
|
| 1 |
EC50 = 5.012 nM
|
|
|
|
CP0062907
|
6-morpholin-4-yl-N-[3-(1H-pyrazol-5-ylmethyl)-1,2,4,5-tetrahydro-3-benzazepin-7-yl]pyridine-3-sulfonamide
Show/Hide
|
C23H28N6O3S
|
1
|
| 1 |
EC50 = 6.31 nM
|
|
|
|
CP0857170
|
MOTILIN_034
Show/Hide
|
C25H26F2N4O
|
1
|
| 1 |
EC50 = 6.31 nM
|
|
|
|
CP0914292
|
MOTILIN_006
Show/Hide
|
C26H33F3N4O
|
1
|
| 1 |
EC50 = 6.31 nM
|
|
|
|
CP0921487
|
MOTILIN_065
Show/Hide
|
C26H33FN6O
|
1
|
| 1 |
EC50 = 6.31 nM
|
|
|
|
CP0225946
|
7-[[6-(4-chlorophenyl)pyridin-3-yl]sulfonylmethyl]-2,3,4,5-tetrahydro-1H-3-benzazepine
Show/Hide
|
C22H21ClN2O2S
|
1
|
| 1 |
EC50 = 7.943 nM
|
|
|
|
CP0271479
|
4-butyl-N-[3-(1H-imidazol-5-ylmethyl)-1,2,4,5-tetrahydro-3-benzazepin-7-yl]benzenesulfonamide
Show/Hide
|
C24H30N4O2S
|
1
|
| 1 |
EC50 = 7.943 nM
|
|
|
|
CP0271508
|
N-[3-(1H-pyrazol-5-ylmethyl)-1,2,4,5-tetrahydro-3-benzazepin-7-yl]-5-pyridin-2-ylthiophene-2-sulfonamide
Show/Hide
|
C23H23N5O2S2
|
1
|
| 1 |
EC50 = 7.943 nM
|
|
|
|
CP0857109
|
MOTILIN_044
Show/Hide
|
C25H27FN4O
|
1
|
| 1 |
EC50 = 7.943 nM
|
|
|
|
CP0857168
|
MOTILIN_002
Show/Hide
|
C25H32F2N4O
|
1
|
| 1 |
EC50 = 7.943 nM
|
|
|
|
CP0857937
|
MOTILIN_032
Show/Hide
|
C26H27N5O
|
1
|
| 1 |
EC50 = 7.943 nM
|
|
|
|
CP0857938
|
MOTILIN_049
Show/Hide
|
C26H30N4O2
|
1
|
| 1 |
EC50 = 7.943 nM
|
|
|
|
CP0931907
|
MOTILIN_029
Show/Hide
|
C25H27FN4O2
|
1
|
| 1 |
EC50 = 7.943 nM
|
|
|
|
CP0952067
|
MOTILIN_045
Show/Hide
|
C25H27FN4O
|
1
|
| 1 |
EC50 = 7.943 nM
|
|
|
|
CP0957585
|
MOTILIN_038
Show/Hide
|
C26H35FN4O
|
1
|
| 1 |
EC50 = 7.943 nM
|
|
|
|
CP0459694
|
1-[4-(4-fluoroanilino)piperidin-1-yl]-2-[4-[[(3S)-3-methylpiperazin-1-yl]methyl]phenyl]ethanone
Show/Hide
|
C25H33FN4O
|
1
|
| 1 |
EC50 = 10 nM
|
|
|
|
CP0131787
|
3-Cyclohexyl-1-[4'-((3R,5S)-3,5-dimethyl-piperazin-1-ylmethyl)-biphenyl-2-ylmethyl]-1-[2-(3-methoxy-phenyl)-ethyl]-urea
Show/Hide
|
C36H48N4O2
|
1
|
| 1 |
EC50 = 10 nM
|
|
|
|
CP0193948
|
4-phenyl-N-[3-(1H-pyrazol-5-ylmethyl)-1,2,4,5-tetrahydro-3-benzazepin-7-yl]benzenesulfonamide
Show/Hide
|
C26H26N4O2S
|
1
|
| 1 |
EC50 = 10 nM
|
|
|
|
CP0879735
|
MOTILIN_005
Show/Hide
|
C26H33F3N4O
|
1
|
| 1 |
EC50 = 10 nM
|
|
|
|
CP0136735
|
1-[4-(3-fluoroanilino)piperidin-1-yl]-2-[4-[[(3S)-3-methylpiperazin-1-yl]methyl]phenyl]ethanone
Show/Hide
|
C25H33FN4O
|
1
|
| 1 |
EC50 = 12.59 nM
|
|
|
|
CP0044015
|
7-((4'-fluorobiphenyl-4-ylsulfonyl)methyl)-2,3,4,5-tetrahydro-1H-benzo[d]azepine
Show/Hide
|
C23H22FNO2S
|
1
|
| 1 |
EC50 = 12.59 nM
|
|
|
|
CP0857110
|
MOTILIN_046
Show/Hide
|
C27H31FN4O
|
1
|
| 1 |
EC50 = 12.59 nM
|
|
|
|
CP0857935
|
MOTILIN_011
Show/Hide
|
C26H32N4O2
|
1
|
| 1 |
EC50 = 12.59 nM
|
|
|
|
CP0909411
|
MOTILIN_008
Show/Hide
|
C25H32F2N4O
|
1
|
| 1 |
EC50 = 12.59 nM
|
|
|
|
CP0957582
|
MOTILIN_009
Show/Hide
|
C25H32FN3O2
|
1
|
| 1 |
EC50 = 12.59 nM
|
|
|
|
CP0851098
|
MOTILIN_054
Show/Hide
|
C27H31FN4O3
|
1
|
| 1 |
EC50 = 15.85 nM
|
|
|
|
CP0857175
|
MOTILIN_070
Show/Hide
|
C27H37FN4O
|
1
|
| 1 |
EC50 = 15.85 nM
|
|
|
|
CP0857939
|
MOTILIN_051
Show/Hide
|
C27H31FN4O2
|
1
|
| 1 |
EC50 = 15.85 nM
|
|
|
|
CP0919771
|
MOTILIN_010
Show/Hide
|
C25H32FN3O2
|
1
|
| 1 |
EC50 = 15.85 nM
|
|
|
|
CP0921484
|
MOTILIN_012
Show/Hide
|
C26H33N5O
|
1
|
| 1 |
EC50 = 15.85 nM
|
|
|
|
CP0394501
|
1-[4-(3-fluoroanilino)piperidin-1-yl]-2-[4-[[(3R)-3-methylpiperazin-1-yl]methyl]phenyl]ethanone
Show/Hide
|
C25H33FN4O
|
1
|
| 1 |
EC50 = 19.95 nM
|
|
|
|
CP0208298
|
7-[[4-(4-chlorophenyl)phenyl]sulfonylmethyl]-2,3,4,5-tetrahydro-1H-3-benzazepine
Show/Hide
|
C23H22ClNO2S
|
1
|
| 1 |
EC50 = 19.95 nM
|
|
|
|
CP0362586
|
N-(4-fluorophenyl)-5-(2,3,4,5-tetrahydro-1H-3-benzazepin-7-ylmethylsulfonyl)pyridin-2-amine
Show/Hide
|
C22H22FN3O2S
|
1
|
| 1 |
EC50 = 19.95 nM
|
|
|
|
CP0857173
|
MOTILIN_063
Show/Hide
|
C29H35F2N5O2S
|
1
|
| 1 |
EC50 = 19.95 nM
|
|
|
|
CP0952062
|
MOTILIN_003
Show/Hide
|
C25H32FN3O2
|
1
|
| 1 |
EC50 = 19.95 nM
|
|
|
|
CP0952068
|
MOTILIN_060
Show/Hide
|
C24H27FN4O2S
|
1
|
| 1 |
EC50 = 19.95 nM
|
|
|
|
CP0954968
|
MOTILIN_048
Show/Hide
|
C28H28F3N3O2
|
1
|
| 1 |
EC50 = 19.95 nM
|
|
|
|
CP0459696
|
1-[4-(3-fluoroanilino)piperidin-1-yl]-3-[4-[[(3S)-3-methylpiperazin-1-yl]methyl]phenyl]propan-1-one
Show/Hide
|
C26H35FN4O
|
1
|
| 1 |
EC50 = 25.12 nM
|
|
|
|
CP0062902
|
7-((3',4'-difluorobiphenyl-4-ylsulfonyl)methyl)-2,3,4,5-tetrahydro-1H-benzo[d]azepine
Show/Hide
|
C23H21F2NO2S
|
1
|
| 1 |
EC50 = 25.12 nM
|
|
|
|
CP0869003
|
MOTILIN_004
Show/Hide
|
C25H32FN3O2
|
1
|
| 1 |
EC50 = 25.12 nM
|
|
|
|
CP0957581
|
MOTILIN_007
Show/Hide
|
C26H35FN4O2
|
1
|
| 1 |
EC50 = 25.12 nM
|
|
|
|
CP0957587
|
MOTILIN_062
Show/Hide
|
C27H34FN5S
|
1
|
| 1 |
EC50 = 25.12 nM
|
|
|
|
CP0961288
|
MOTILIN_071
Show/Hide
|
C28H39FN4O
|
1
|
| 1 |
EC50 = 25.12 nM
|
|
|
|
CP0415158
|
1-[2-(4-([(3R,5S)-3,5-Dimethyl-1-piperazinyl]methyl)phenyl)propanoyl]-N-(4-fluorophenyl)-4-piperidinamine
Show/Hide
|
C27H37FN4O
|
1
|
| 1 |
EC50 = 31.62 nM
|
|
|
|
CP0498741
|
1-[2-(4-([(3R,5S)-3,5-Dimethyl-1-piperazinyl]methyl)phenyl)-2-methylpropanoyl]-N-(4-fluorophenyl)-4-piperidinamine
Show/Hide
|
C28H39FN4O
|
1
|
| 1 |
EC50 = 31.62 nM
|
|
|
|
CP0497593
|
4-methyl-N-[3-(1H-pyrazol-5-ylmethyl)-1,2,4,5-tetrahydro-3-benzazepin-7-yl]-2,3-dihydro-1,4-benzoxazine-7-sulfonamide
Show/Hide
|
C23H27N5O3S
|
1
|
| 1 |
EC50 = 31.62 nM
|
|
|
|
CP0916581
|
MOTILIN_041
Show/Hide
|
C24H26FN5O2
|
1
|
| 1 |
EC50 = 31.62 nM
|
|
|
|
CP0950892
|
MOTILIN_001
Show/Hide
|
C26H33N5O
|
1
|
| 1 |
EC50 = 31.62 nM
|
|
|
|
CP0394496
|
1-[(4-([(3R,5S)-3,5-Dimethyl-1-piperazinyl]methyl)phenyl)acetyl]-N-(4-fluorophenyl)-4-piperidinamine
Show/Hide
|
C26H35FN4O
|
1
|
| 1 |
EC50 = 39.81 nM
|
|
|
|
CP0062919
|
3-chloro-4-methyl-N-[3-(1H-pyrazol-5-ylmethyl)-1,2,4,5-tetrahydro-3-benzazepin-7-yl]benzenesulfonamide
Show/Hide
|
C21H23ClN4O2S
|
1
|
| 1 |
EC50 = 39.81 nM
|
|
|
|
CP0469589
|
7-[[6-(2-methylpropoxy)pyridin-3-yl]sulfonylmethyl]-2,3,4,5-tetrahydro-1H-3-benzazepine
Show/Hide
|
C20H26N2O3S
|
1
|
| 1 |
EC50 = 39.81 nM
|
|
|
|
CP0851101
|
MOTILIN_069
Show/Hide
|
C27H37FN4O
|
1
|
| 1 |
EC50 = 39.81 nM
|
|
|
|
CP0857171
|
MOTILIN_042
Show/Hide
|
C27H35N5O
|
1
|
| 1 |
EC50 = 39.81 nM
|
|
|
|
CP0869011
|
MOTILIN_047
Show/Hide
|
C26H27N5O
|
1
|
| 1 |
EC50 = 39.81 nM
|
|
|
|
CP0931904
|
MOTILIN_016
Show/Hide
|
C26H28FN3O
|
1
|
| 1 |
EC50 = 39.81 nM
|
|
|
|
CP0055087
|
(3R,4S,5S,6R,7R,9R,11R,12R,13S,14R)-6-[(2S,3R,4S,6R)-4-(dimethylamino)-3-hydroxy-6-methyloxan-2-yl]oxy-14-ethyl-7,12,13-trihydroxy-4-[(2R,4R,5S,6S)-5-hydroxy-4-methoxy-4,6-dimethyloxan-2-yl]oxy-3,5,7,9,11,13-hexamethyl-oxacyclotetradecane-2,10-dione
Show/Hide
|
C37H67NO13
|
1
|
| 1 |
EC50 = 50.12 nM
|
|
|
|
CP0463803
|
3-[4-[[(3S,5R)-3,5-dimethylpiperazin-1-yl]methyl]phenyl]-1-[4-(4-fluoroanilino)piperidin-1-yl]propan-1-one
Show/Hide
|
C27H37FN4O
|
1
|
| 1 |
EC50 = 50.12 nM
|
|
|
|
CP0418599
|
3-cyclohexyl-1-[2-(3-methoxyphenyl)ethyl]-1-[[2-[4-(piperazin-1-ylmethyl)phenyl]phenyl]methyl]urea
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C34H44N4O2
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1
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| 1 |
EC50 = 50.12 nM
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CP0504591
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N-[5-[[7-[(4-butylphenyl)sulfonylamino]-1,2,4,5-tetrahydro-3-benzazepin-3-yl]methyl]thiophen-2-yl]acetamide
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C27H33N3O3S2
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1
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| 1 |
EC50 = 50.12 nM
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CP0373415
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1-[4-(4-fluoroanilino)piperidin-1-yl]-3-[4-[[(3S)-3-methylpiperazin-1-yl]methyl]phenyl]propan-1-one
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C26H35FN4O
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1
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| 1 |
EC50 = 63.1 nM
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CP0057206
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4-butyl-N-[3-[(2-methyl-1H-imidazol-5-yl)methyl]-1,2,4,5-tetrahydro-3-benzazepin-7-yl]benzenesulfonamide
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C25H32N4O2S
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1
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| 1 |
EC50 = 63.1 nM
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CP0271509
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7-((6-(piperidin-1-yl)pyridin-3-ylsulfonyl)methyl)-2,3,4,5-tetrahydro-1H-benzo[d]azepine
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C21H27N3O2S
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1
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| 1 |
EC50 = 63.1 nM
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CP0931909
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MOTILIN_043
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C27H35N5O
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1
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| 1 |
EC50 = 63.1 nM
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CP0950896
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MOTILIN_057
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C24H32FN5O
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1
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| 1 |
EC50 = 79.43 nM
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CP0916580
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MOTILIN_031
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C22H31N5O2S
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1
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| 1 |
EC50 = 100 nM
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CP0469067
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7-[(4-butylphenyl)sulfonylmethyl]-2,3,4,5-tetrahydro-1H-3-benzazepine
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C21H27NO2S
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1
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| 1 |
EC50 = 125.89 nM
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CP0044013
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7-((6-isopropoxypyridin-3-ylsulfonyl)methyl)-2,3,4,5-tetrahydro-1H-benzo[d]azepine
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C19H24N2O3S
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1
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| 1 |
EC50 = 158.49 nM
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CP0506557
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4-[5-(2,3,4,5-tetrahydro-1H-3-benzazepin-7-ylmethylsulfonyl)pyridin-2-yl]benzonitrile
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C23H21N3O2S
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1
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| 1 |
EC50 = 158.49 nM
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CP0950894
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MOTILIN_052
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C24H27FN4O2S
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1
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| 1 |
EC50 = 158.49 nM
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CP0411177
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4-butyl-N-(3-cyclopentyl-1,2,4,5-tetrahydro-3-benzazepin-7-yl)benzenesulfonamide
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C25H34N2O2S
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1
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| 1 |
EC50 = 199.53 nM
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CP0504205
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3-cyclohexyl-1-[2-(3-methoxyphenyl)ethyl]-1-[[2-[4-(piperidin-4-ylmethyl)phenyl]phenyl]methyl]urea
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C35H45N3O2
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1
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| 1 |
EC50 = 398.11 nM
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CP0192277
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4-(5-((2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-yl)methylsulfonyl)pyridin-2-yl)morpholine
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C20H25N3O3S
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1
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| 1 |
EC50 = 501.19 nM
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CP0360494
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7-((6-(4-fluorophenoxy)pyridin-3-ylsulfonyl)methyl)-2,3,4,5-tetrahydro-1H-benzo[d]azepine
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C22H21FN2O3S
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1
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| 1 |
EC50 = 501.19 nM
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CP0390054
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N-[3-[[7-[(4-butylphenyl)sulfonylamino]-1,2,4,5-tetrahydro-3-benzazepin-3-yl]methyl]phenyl]acetamide
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C29H35N3O3S
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1
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| 1 |
EC50 = 501.19 nM
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CP0375048
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N-(3-methoxypropyl)-2-phenyl-N-[[2-[4-(piperazin-1-ylmethyl)phenyl]phenyl]methyl]acetamide
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C30H37N3O2
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1
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| 1 |
EC50 = 794.33 nM
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CP0376526
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4-chloro-N-[3-(1H-pyrazol-5-ylmethyl)-1,2,4,5-tetrahydro-3-benzazepin-7-yl]benzenesulfonamide
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C20H21ClN4O2S
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1
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| 1 |
EC50 = 794.33 nM
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CP0402057
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7-(naphthalen-2-ylsulfonylmethyl)-2,3,4,5-tetrahydro-1H-3-benzazepine
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C21H21NO2S
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1
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| 1 |
EC50 = 1258.93 nM
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CP0157631
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4-butyl-N-(2,3,4,5-tetrahydro-1H-3-benzazepin-7-yl)benzenesulfonamide
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C20H26N2O2S
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1
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| 1 |
EC50 = 1584.89 nM
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CP0406687
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6-morpholin-4-yl-N-(2,3,4,5-tetrahydro-1H-3-benzazepin-7-yl)pyridine-3-sulfonamide
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C19H24N4O3S
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1
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| 1 |
EC50 = 1584.89 nM
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CP0381247
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N-(4-fluorophenyl)-5-(2,3,4,5-tetrahydro-1H-3-benzazepin-7-ylmethylsulfonyl)pyridine-2-carboxamide
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C23H22FN3O3S
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1
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| 1 |
EC50 = 1995.26 nM
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CP0411176
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4-butyl-N-[3-(oxolan-3-ylmethyl)-1,2,4,5-tetrahydro-3-benzazepin-7-yl]benzenesulfonamide
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C25H34N2O3S
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1
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| 1 |
EC50 = 1995.26 nM
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CP0411183
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N-(6-morpholin-4-ylpyridin-3-yl)-2,3,4,5-tetrahydro-1H-3-benzazepine-7-sulfonamide
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C19H24N4O3S
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1
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| 1 |
EC50 = 2511.89 nM
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CP0501686
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4-butyl-N-methyl-N-(2,3,4,5-tetrahydro-1H-3-benzazepin-7-yl)benzenesulfonamide
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C21H28N2O2S
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1
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| 1 |
EC50 = 2511.89 nM
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CP0501687
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1-phenyl-N-[3-(1H-pyrazol-5-ylmethyl)-1,2,4,5-tetrahydro-3-benzazepin-7-yl]methanesulfonamide
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C21H24N4O2S
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1
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| 1 |
EC50 = 2511.89 nM
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CP0510453
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4-butyl-N-[3-(thiophen-2-ylmethyl)-1,2,4,5-tetrahydro-3-benzazepin-7-yl]benzenesulfonamide
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C25H30N2O2S2
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1
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| 1 |
EC50 = 2511.89 nM
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CP0434025
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N-[[2-[4-[[2-(dimethylamino)ethyl-methylamino]methyl]phenyl]phenyl]methyl]-N-(3-methoxypropyl)-2-phenylacetamide
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C31H41N3O2
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1
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| 1 |
EC50 = 3162.28 nM
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CP0384095
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7-[(4-tert-butylphenyl)sulfonylmethyl]-2,3,4,5-tetrahydro-1H-3-benzazepine
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C21H27NO2S
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1
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| 1 |
EC50 = 3162.28 nM
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CP0538527
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4-butyl-N-[3-[(3-methylimidazol-4-yl)methyl]-1,2,4,5-tetrahydro-3-benzazepin-7-yl]benzenesulfonamide
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C25H32N4O2S
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1
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| 1 |
EC50 = 3162.28 nM
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CP0510507
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3-cyclohexyl-1-[2-(3-methoxyphenyl)ethyl]-1-[[2-(4-piperazin-1-ylphenyl)phenyl]methyl]urea
Show/Hide
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C33H42N4O2
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1
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| 1 |
EC50 = 5011.87 nM
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CP0060335
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4-cyano-N-[3-(1H-pyrazol-5-ylmethyl)-1,2,4,5-tetrahydro-3-benzazepin-7-yl]benzenesulfonamide
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C21H21N5O2S
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1
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| 1 |
EC50 = 7943.28 nM
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CP0491474
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N-[[2-[4-[(4-acetylpiperazin-1-yl)methyl]phenyl]phenyl]methyl]-N-(3-methoxypropyl)-2-phenylacetamide
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C32H39N3O3
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1
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| 1 |
EC50 > 12589.25 nM
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CP0494560
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N-(3-methoxypropyl)-2-phenyl-N-[[2-[4-(piperidin-1-ylmethyl)phenyl]phenyl]methyl]acetamide
Show/Hide
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C31H38N2O2
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1
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| 1 |
EC50 > 12589.25 nM
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CP0494562
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N-(3-methoxypropyl)-N-[[2-[4-[(4-methylpiperazin-1-yl)methyl]phenyl]phenyl]methyl]-2-phenylacetamide
Show/Hide
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C31H39N3O2
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1
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| 1 |
EC50 > 12589.25 nM
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CP0515821
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N-(3-methoxypropyl)-N-[[2-[4-(morpholin-4-ylmethyl)phenyl]phenyl]methyl]-2-phenylacetamide
Show/Hide
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C30H36N2O3
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1
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| 1 |
EC50 > 12589.25 nM
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CP0522405
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3-cyclohexyl-1-[2-(3-methoxyphenyl)ethyl]-1-[[2-[4-(2-piperazin-1-ylethyl)phenyl]phenyl]methyl]urea
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C35H46N4O2
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1
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| 1 |
EC50 > 12589.25 nM
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CP0362584
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N-[3-(1H-pyrazol-5-ylmethyl)-1,2,4,5-tetrahydro-3-benzazepin-7-yl]propane-2-sulfonamide
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C17H24N4O2S
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1
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| 1 |
EC50 > 12589.25 nM
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CP0411170
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6-morpholin-4-yl-N-(2,3,4,5-tetrahydro-1H-3-benzazepin-7-yl)pyridine-3-carboxamide
Show/Hide
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C20H24N4O2
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1
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| 1 |
EC50 > 12589.25 nM
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CP0469068
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N-methyl-6-morpholin-4-yl-N-(2,3,4,5-tetrahydro-1H-3-benzazepin-7-yl)pyridine-3-carboxamide
Show/Hide
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C21H26N4O2
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1
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| 1 |
EC50 > 12589.25 nM
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CP0504596
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7-(benzenesulfonylmethyl)-2,3,4,5-tetrahydro-1H-3-benzazepine
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C17H19NO2S
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1
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| 1 |
EC50 > 12589.25 nM
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CP0504611
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4-butyl-N-[3-(1-methylpiperidin-4-yl)-1,2,4,5-tetrahydro-3-benzazepin-7-yl]benzenesulfonamide
Show/Hide
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C26H37N3O2S
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1
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| 1 |
EC50 > 12589.25 nM
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CP0518937
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N-methyl-6-morpholin-4-yl-N-(2,3,4,5-tetrahydro-1H-3-benzazepin-7-ylmethyl)pyridine-3-carboxamide
Show/Hide
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C22H28N4O2
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1
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| 1 |
EC50 > 12589.25 nM
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CP0518938
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N-(6-morpholin-4-ylpyridin-3-yl)-2,3,4,5-tetrahydro-1H-3-benzazepine-7-carboxamide
Show/Hide
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C20H24N4O2
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1
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| 1 |
EC50 > 12589.25 nM
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CP0497589
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N-[3-(1-acetylpiperidin-4-yl)-1,2,4,5-tetrahydro-3-benzazepin-7-yl]-4-butylbenzenesulfonamide
Show/Hide
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C27H37N3O3S
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1
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| 1 |
EC50 > 2511.89 nM
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CP0485109
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N-(3-methoxypropyl)-2-phenyl-N-[[2-[4-(piperazine-1-carbonyl)phenyl]phenyl]methyl]acetamide
Show/Hide
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C30H35N3O3
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1
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| 1 |
EC50 > 3162.28 nM
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CP0497588
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N-(3-benzyl-1,2,4,5-tetrahydro-3-benzazepin-7-yl)-4-butylbenzenesulfonamide
Show/Hide
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C27H32N2O2S
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1
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| 1 |
EC50 > 3162.28 nM
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CP0465450
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(5R,8R,11S)-8-(propan-2-yl)-11-(pyrrolidin-1-ylmethyl)-5-{[3-(trifluoromethyl)phenyl]methyl}-3,4,5,6,7,8,9,10,11,12,13,14,15,16-tetradecahydro-2H-1,4,7,10,13-benzoxatetrazacyclooctadecine-6,9,12-trione
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C33H44F3N5O4
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1
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| 1 |
Ki = 4.6 nM
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CP0464246
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1-{[(5R,8R,11S)-6,9,12-trioxo-8-(propan-2-yl)-5-{[3-(trifluoromethyl)phenyl]methyl}-3,4,5,6,7,8,9,10,11,12,13,14,15,16-tetradecahydro-2H-1,4,7,10,13-benzoxatetrazacyclooctadecin-11-yl]methyl}guanidine
Show/Hide
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C30H40F3N7O4
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1
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| 1 |
Ki = 6 nM
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CP0466808
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1-{[(5R,8R,11S)-5-[(4-chlorophenyl)methyl]-6,9,12-trioxo-8-(propan-2-yl)-3,4,5,6,7,8,9,10,11,12,13,14,15,16-tetradecahydro-2H-1,4,7,10,13-benzoxatetrazacyclooctadecin-11-yl]methyl}guanidine
Show/Hide
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C29H40ClN7O4
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1
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| 1 |
Ki = 6 nM
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CP0485055
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(5R,8R,11S)-11-[(methylamino)methyl]-8-(propan-2-yl)-5-{[3-(trifluoromethyl)phenyl]methyl}-3,4,5,6,7,8,9,10,11,12,13,14,15,16-tetradecahydro-2H-1,4,7,10,13-benzoxatetrazacyclooctadecine-6,9,12-trione
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C30H40F3N5O4
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1
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| 1 |
Ki = 6 nM
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CP0466810
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(5R,8R,11S)-11-(aminomethyl)-8-(propan-2-yl)-5-{[3-(trifluoromethyl)phenyl]methyl}-3,4,5,6,7,8,9,10,11,12,13,14,15,16-tetradecahydro-2H-1,4,7,10,13-benzoxatetrazacyclooctadecine-6,9,12-trione
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C29H38F3N5O4
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1
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| 1 |
Ki = 15 nM
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CP0466809
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(5R,8R,11S)-5-[(4-chlorophenyl)methyl]-11-[(dimethylamino)methyl]-8-(propan-2-yl)-3,4,5,6,7,8,9,10,11,12,13,14,15,16-tetradecahydro-2H-1,4,7,10,13-benzoxatetrazacyclooctadecine-6,9,12-trione
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C30H42ClN5O4
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1
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| 1 |
Ki = 16 nM
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CP0562595
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(5R,8R,11S)-11-[(5-methyl-1H-1,2,3-triazol-1-yl)methyl]-8-(propan-2-yl)-5-{[3-(trifluoromethyl)phenyl]methyl}-3,4,5,6,7,8,9,10,11,12,13,14,15,16-tetradecahydro-2H-1,4,7,10,13-benzoxatetrazacyclooctadecine-6,9,12-trione
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C32H40F3N7O4
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1
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| 1 |
Ki = 17 nM
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CP0458668
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(5R,8R,11S)-5-[(3-chlorophenyl)methyl]-8-(propan-2-yl)-11-(1H-pyrazol-1-ylmethyl)-3,4,5,6,7,8,9,10,11,12,13,14,15,16-tetradecahydro-2H-1,4,7,10,13-benzoxatetrazacyclooctadecine-6,9,12-trione
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C31H39ClN6O4
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1
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| 1 |
Ki = 18 nM
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CP0466807
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(5R,8R,11S)-8-(propan-2-yl)-11-[(pyrimidin-2-ylamino)methyl]-5-{[3-(trifluoromethyl)phenyl]methyl}-3,4,5,6,7,8,9,10,11,12,13,14,15,16-tetradecahydro-2H-1,4,7,10,13-benzoxatetrazacyclooctadecine-6,9,12-trione
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C33H40F3N7O4
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1
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| 1 |
Ki = 20 nM
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CP0516654
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(5R,8R,11S)-11-[(5-methyl-1H-1,2,3,4-tetrazol-1-yl)methyl]-8-(propan-2-yl)-5-{[3-(trifluoromethyl)phenyl]methyl}-3,4,5,6,7,8,9,10,11,12,13,14,15,16-tetradecahydro-2H-1,4,7,10,13-benzoxatetrazacyclooctadecine-6,9,12-trione
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C31H39F3N8O4
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1
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| 1 |
Ki = 21 nM
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CP0485053
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(5R,8R,11S)-11-[(4,5-dimethyl-1H-1,2,3-triazol-1-yl)methyl]-8-(propan-2-yl)-5-{[3-(trifluoromethyl)phenyl]methyl}-3,4,5,6,7,8,9,10,11,12,13,14,15,16-tetradecahydro-2H-1,4,7,10,13-benzoxatetrazacyclooctadecine-6,9,12-trione
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C33H42F3N7O4
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1
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| 1 |
Ki = 23 nM
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CP0458644
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(5R,8R,11S)-5-[(3-chlorophenyl)methyl]-11-[(dimethylamino)methyl]-8-(propan-2-yl)-3,4,5,6,7,8,9,10,11,12,13,14,15,16-tetradecahydro-2H-1,4,7,10,13-benzoxatetrazacyclooctadecine-6,9,12-trione
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C30H42ClN5O4
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1
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| 1 |
Ki = 27 nM
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CP0511026
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3-[(5R,8R,11S)-5-[(3-chlorophenyl)methyl]-6,9,12-trioxo-8-(propan-2-yl)-3,4,5,6,7,8,9,10,11,12,13,14,15,16-tetradecahydro-2H-1,4,7,10,13-benzoxatetrazacyclooctadecin-11-yl]propanimidamide
Show/Hide
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C30H41ClN6O4
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1
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| 1 |
Ki = 27 nM
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CP0426874
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(5R,8R,11S)-5-[(4-chlorophenyl)methyl]-11-[(methylamino)methyl]-8-(propan-2-yl)-3,4,5,6,7,8,9,10,11,12,13,14,15,16-tetradecahydro-2H-1,4,7,10,13-benzoxatetrazacyclooctadecine-6,9,12-trione
Show/Hide
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C29H40ClN5O4
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1
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| 1 |
Ki = 31 nM
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CP0541529
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1-{2-[(5R,8R,11S)-5-[(3-chlorophenyl)methyl]-6,9,12-trioxo-8-(propan-2-yl)-3,4,5,6,7,8,9,10,11,12,13,14,15,16-tetradecahydro-2H-1,4,7,10,13-benzoxatetrazacyclooctadecin-11-yl]ethyl}guanidine
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C30H42ClN7O4
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1
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| 1 |
Ki = 33 nM
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CP0426869
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(5R,8R,11S)-5-[(3-chlorophenyl)methyl]-8-(propan-2-yl)-11-[(1,3-thiazol-2-ylamino)methyl]-3,4,5,6,7,8,9,10,11,12,13,14,15,16-tetradecahydro-2H-1,4,7,10,13-benzoxatetrazacyclooctadecine-6,9,12-trione
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C31H39ClN6O4S
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1
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| 1 |
Ki = 41 nM
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CP0466806
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(5R,8R,11S)-5-[(3-chlorophenyl)methyl]-11-[(4,5-dihydro-1H-imidazol-2-ylamino)methyl]-8-(propan-2-yl)-3,4,5,6,7,8,9,10,11,12,13,14,15,16-tetradecahydro-2H-1,4,7,10,13-benzoxatetrazacyclooctadecine-6,9,12-trione
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C31H42ClN7O4
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1
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| 1 |
Ki = 51 nM
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CP0458669
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1-{[(5R,8R,11S)-5-[(3-chlorophenyl)methyl]-6,9,12-trioxo-8-(propan-2-yl)-3,4,5,6,7,8,9,10,11,12,13,14,15,16-tetradecahydro-2H-1,4,7,10,13-benzoxatetrazacyclooctadecin-11-yl]methyl}guanidine
Show/Hide
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C29H40ClN7O4
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1
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| 1 |
Ki = 57 nM
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CP0458645
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(5R,8R,11S)-11-(aminomethyl)-5-[(4-chlorophenyl)methyl]-8-(propan-2-yl)-3,4,5,6,7,8,9,10,11,12,13,14,15,16-tetradecahydro-2H-1,4,7,10,13-benzoxatetrazacyclooctadecine-6,9,12-trione
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C28H38ClN5O4
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1
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| 1 |
Ki = 60 nM
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CP0485052
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(5R,8R,11S)-5-[(3-chlorophenyl)methyl]-11-(1H-imidazol-1-ylmethyl)-8-(propan-2-yl)-3,4,5,6,7,8,9,10,11,12,13,14,15,16-tetradecahydro-2H-1,4,7,10,13-benzoxatetrazacyclooctadecine-6,9,12-trione
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C31H39ClN6O4
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1
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| 1 |
Ki = 62 nM
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CP0434323
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(5R,8R,11S)-11-(aminomethyl)-5-[(3-chlorophenyl)methyl]-8-(propan-2-yl)-3,4,5,6,7,8,9,10,11,12,13,14,15,16-tetradecahydro-2H-1,4,7,10,13-benzoxatetrazacyclooctadecine-6,9,12-trione
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C28H38ClN5O4
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1
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| 1 |
Ki = 64 nM
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CP0562596
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(5R,8R,11S)-5-[(3-chlorophenyl)methyl]-8-(propan-2-yl)-11-[(1,4,5,6-tetrahydropyrimidin-2-ylamino)methyl]-3,4,5,6,7,8,9,10,11,12,13,14,15,16-tetradecahydro-2H-1,4,7,10,13-benzoxatetrazacyclooctadecine-6,9,12-trione
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C32H44ClN7O4
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1
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| 1 |
Ki = 87 nM
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CP0485054
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1-{[(5R,8R,11S)-5-[(3-chlorophenyl)methyl]-6,9,12-trioxo-8-(propan-2-yl)-3,4,5,6,7,8,9,10,11,12,13,14,15,16-tetradecahydro-2H-1,4,7,10,13-benzoxatetrazacyclooctadecin-11-yl]methyl}-2-cyanoguanidine
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C30H39ClN8O4
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1
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| 1 |
Ki = 100 nM
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CP0485051
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(5R,8R,11S)-5-[(3-fluorophenyl)methyl]-8-(propan-2-yl)-11-(1,3-thiazol-4-ylmethyl)-3,4,5,6,7,8,9,10,11,12,13,14,15,16-tetradecahydro-2H-1,4,7,10,13-benzoxatetrazacyclooctadecine-6,9,12-trione
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C31H38FN5O4S
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1
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| 1 |
Ki = 116 nM
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CP0134944
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(E)-(9R,12R,15S)-9-(4-hydroxy-benzyl)-12-isopropyl-15-propyl-6,7,8,9,11,12,14,15,17,18-decahydro-5-oxa-8,11,14,17-tetraaza-benzocyclooctadecene-10,13,16-trione
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C30H40N4O5
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1
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| 1 |
Ki = 137 nM
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CP0426871
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(5R,8R,11S)-11-(aminomethyl)-5-[(4-hydroxyphenyl)methyl]-8-(propan-2-yl)-3,4,5,6,7,8,9,10,11,12,13,14,15,16-tetradecahydro-2H-1,4,7,10,13-benzoxatetrazacyclooctadecine-6,9,12-trione
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C28H39N5O5
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1
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| 1 |
Ki = 171 nM
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CP0466811
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(5R,8R,11S)-11-(2-aminoethyl)-5-[(4-hydroxyphenyl)methyl]-8-(propan-2-yl)-3,4,5,6,7,8,9,10,11,12,13,14,15,16-tetradecahydro-2H-1,4,7,10,13-benzoxatetrazacyclooctadecine-6,9,12-trione
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C29H41N5O5
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1
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| 1 |
Ki = 342 nM
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CP0560279
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(5R,8R,11S)-5-[(4-hydroxyphenyl)methyl]-8-(propan-2-yl)-11-[(propan-2-ylamino)methyl]-3,4,5,6,7,8,9,10,11,12,13,14,15,16-tetradecahydro-2H-1,4,7,10,13-benzoxatetrazacyclooctadecine-6,9,12-trione
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C31H45N5O5
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1
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| 1 |
Ki = 376 nM
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CP0434322
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[(6R,9R,12S)-6-[(4-chlorophenyl)methyl]-7,10,13-trioxo-9-propan-2-yl-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),18,20-trien-12-yl]methylurea
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C29H39ClN6O5
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1
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| 1 |
Ki = 543 nM
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CP0333555
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(9R,12R,15S)-15-(4-amino-butyl)-9-(4-hydroxy-benzyl)-12-isopropyl-6,7,8,9,11,12,14,15,17,18-decahydro-5-oxa-8,11,14,17-tetraaza-benzocyclooctadecene-10,13,16-trione
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C31H43N5O5
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1
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| 1 |
Ki = 664 nM
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CP0511027
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(5R,8R,11S)-11-(3-aminopropyl)-5-[(4-hydroxyphenyl)methyl]-8-(propan-2-yl)-3,4,5,6,7,8,9,10,11,12,13,14-dodecahydro-2H-1,4,7,10,13-benzoxatetrazacyclooctadecine-6,9,12-trione
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C30H41N5O5
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1
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| 1 |
Ki = 889 nM
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CP0553920
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N-[[(6R,9R,12S)-6-[(4-hydroxyphenyl)methyl]-7,10,13-trioxo-9-propan-2-yl-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),18,20-trien-12-yl]methyl]acetamide
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C30H41N5O6
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1
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| 1 |
Ki = 1946 nM
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CP0453615
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(9R,12R,15S)-9-(4-hydroxy-benzyl)-12-isopropyl-10,13,16-trioxo-7,8,9,10,11,12,13,14,15,16,17,18-dodecahydro-6H-5-oxa-8,11,14,17-tetraaza-benzocyclooctadecen-15-yl]-acetic acid
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C29H36N4O7
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1
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| 1 |
Ki = 2553 nM
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