General Information of the Compound
Compound ID
CP0497588
Compound Name
N-(3-benzyl-1,2,4,5-tetrahydro-3-benzazepin-7-yl)-4-butylbenzenesulfonamide
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Structure
Formula
C27H32N2O2S
Molecular Weight
448.632
Canonical SMILES
CCCCc1ccc(cc1)S(=O)(=O)Nc1ccc2CCN(Cc3ccccc3)CCc2c1
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InChI
InChI=1S/C27H32N2O2S/c1-2-3-7-22-10-14-27(15-11-22)32(30,31)28-26-13-12-24-16-18-29(19-17-25(24)20-26)21-23-8-5-4-6-9-23/h4-6,8-15,20,28H,2-3,7,16-19,21H2,1H3
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InChIKey
FWROZMQRBMGKLZ-UHFFFAOYSA-N
Physicochemical Property
logP
5.4308
Rotatable Bonds
8
Heavy Atom Count
32
Polar Areas
49.41
Hydrogen Bond Donor Count
1
Hydrogen Bond Acceptor Count
3
Complexity
32

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 46882348
ChEMBL ID
CHEMBL1078807
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT01121, Motilin receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
EC50 > 3162.28 nM
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   LI
   LO
   TS