| Compound ID |
Compound Name |
Compound Formula |
|
CP0844786
|
N-(cyclohexylmethyl)-2-(3-((R)-2-((R)-2-hydroxy-2-(4-hydroxy-3-(hydroxymethyl)phenyl)ethylamino)propyl)phenyl)acetamide
Show/Hide
|
C27H38N2O4
|
1
|
| 1 |
Activity = 0.02 nM
|
|
|
|
CP0372313
|
N-[(3,4-dichlorophenyl)methyl]-2-[3-[(2R)-2-[[(2R)-2-hydroxy-2-[4-hydroxy-3-(hydroxymethyl)phenyl]ethyl]amino]propyl]phenyl]acetamide
Show/Hide
|
C27H30Cl2N2O4
|
3
|
| 1 |
Activity = 0.03 nM
|
|
|
| 2 |
EC50 = 0.024 nM
|
|
|
| 3 |
EC50 = 1.1 nM
|
|
|
|
CP0440913
|
N-(1-adamantyl)-2-[3-[(2R)-2-[[(2R)-2-hydroxy-2-[4-hydroxy-3-(hydroxymethyl)phenyl]ethyl]amino]propyl]phenyl]acetamide
Show/Hide
|
C30H40N2O4
|
2
|
| 1 |
Activity = 0.06 nM
|
|
|
| 2 |
EC50 = 0.064 nM
|
|
|
|
CP0065062
|
1-hydroxy-2-naphthoic acid;4-[1-hydroxy-2-[6-(4-phenylbutoxy)hexylamino]ethyl]-2-methylol-phenol
Show/Hide
|
C25H37NO4
|
8
|
| 1 |
Activity = 0.07 nM
|
|
|
| 2 |
EC50 = 0.07 nM
|
|
|
| 3 |
EC50 = 0.2512 nM
|
|
|
| 4 |
Kd = 1100 nM
|
|
|
| 5 |
Ki = 0.18 nM
|
|
|
| 6 |
Ki = 0.25 nM
|
|
|
| 7 |
Ki = 0.39 nM
|
|
|
| 8 |
Ki = 3.2 nM
|
|
|
|
CP0922071
|
N-(cycloheptylmethyl)-2-(3-((R)-2-((R)-2-hydroxy-2-(4-hydroxy-3-(hydroxymethyl)phenyl)ethylamino)propyl)phenyl)acetamide
Show/Hide
|
C28H40N2O4
|
1
|
| 1 |
Activity = 0.118 nM
|
|
|
|
CP0882544
|
N-adamantan-2-yl-2-(3-{(R)-2-[(R)-2-hydroxy-2-(4-hydroxy-3-hydroxymethyl-phenyl)-ethylamino]-propyl}-phenyl)-acetamide
Show/Hide
|
C30H40N2O4
|
1
|
| 1 |
Activity = 0.19 nM
|
|
|
|
CP0880756
|
N-cyclooctyl-2-(3-((R)-2-((R)-2-hydroxy-2-(4-hydroxy-3-(hydroxymethyl)phenyl)ethylamino)propyl)phenyl)acetamide
Show/Hide
|
C28H40N2O4
|
1
|
| 1 |
Activity = 0.2 nM
|
|
|
|
CP0850169
|
N-adamantan-1-ylmethyl-2-(3-{(R)-2-[(R)-2-hydroxy-2-(4-hydroxy-3-hydroxymethyl-phenyl)-ethylamino]-propyl}-phenyl)-acetamide
Show/Hide
|
C31H42N2O4
|
1
|
| 1 |
Activity = 0.25 nM
|
|
|
|
CP0144504
|
5-[(2R)-2-[[(2R)-2-hydroxy-2-[4-hydroxy-3-(hydroxymethyl)phenyl]ethyl]amino]propyl]-N-[(2-methoxyphenyl)methyl]-1H-indole-2-carboxamide
Show/Hide
|
C29H33N3O5
|
1
|
| 1 |
EC50 = 0.02 nM
|
|
|
|
CP0372621
|
(R)-N-(2-chloro-4-hydroxybenzyl)-2-(3-(2-(2-hydroxy-2-(4-hydroxy-3-(methylsulfonamido)phenyl)ethylamino)-2-methylpropyl)phenyl)acetamide
Show/Hide
|
C28H34ClN3O6S
|
1
|
| 1 |
EC50 = 0.02 nM
|
|
|
|
CP0229160
|
N-benzyl-5-[(2R)-2-[[(2R)-2-hydroxy-2-[4-hydroxy-3-(hydroxymethyl)phenyl]ethyl]amino]propyl]-N-methyl-1H-indole-2-carboxamide
Show/Hide
|
C29H33N3O4
|
1
|
| 1 |
EC50 = 0.022 nM
|
|
|
|
CP0520867
|
(R)-N-benzyl-2-(3-(2-(2-hydroxy-2-(4-hydroxy-3-(methylsulfonamido)phenyl)ethylamino)-2-methylpropyl)phenyl)acetamide
Show/Hide
|
C28H35N3O5S
|
1
|
| 1 |
EC50 = 0.023 nM
|
|
|
|
CP0507603
|
N-benzyl-2-[3-[(2R)-2-[[(2R)-2-hydroxy-2-[4-hydroxy-3-(methanesulfonamido)phenyl]ethyl]amino]propyl]phenyl]acetamide
Show/Hide
|
C27H33N3O5S
|
1
|
| 1 |
EC50 = 0.027 nM
|
|
|
|
CP0459845
|
5-{(R)-2-[(R)-2-hydroxy-2-(4-hydroxy-3-hydroxymethyl-phenyl)-ethylamino]-propyl}-1H-indole-2-carboxylic acid (4H-1lambda*4*-thiazol-2-ylmethyl)-amide
Show/Hide
|
C25H28N4O4S
|
1
|
| 1 |
EC50 = 0.031 nM
|
|
|
|
CP0505984
|
N-(cyclohexylmethyl)-2-[3-[(2R)-2-[[(2R)-2-hydroxy-2-[4-hydroxy-3-(methanesulfonamido)phenyl]ethyl]amino]propyl]phenyl]acetamide
Show/Hide
|
C27H39N3O5S
|
1
|
| 1 |
EC50 = 0.032 nM
|
|
|
|
CP0459846
|
5-((R)-2-((R)-2-hydroxy-2-(4-hydroxy-3-(hydroxymethyl)phenyl)ethylamino)propyl)-N-(pyridin-2-ylmethyl)-1H-indole-2-carboxamide
Show/Hide
|
C27H30N4O4
|
1
|
| 1 |
EC50 = 0.038 nM
|
|
|
|
CP0511140
|
5-[(2R)-2-[[(2R)-2-hydroxy-2-[4-hydroxy-3-(hydroxymethyl)phenyl]ethyl]amino]propyl]-N-[(2-methylsulfanylphenyl)methyl]-1H-indole-2-carboxamide
Show/Hide
|
C29H33N3O4S
|
1
|
| 1 |
EC50 = 0.038 nM
|
|
|
|
CP0372622
|
2-(3-((R)-2-((R)-2-hydroxy-2-(4-hydroxy-3-(methylsulfonamido)phenyl)ethylamino)propyl)phenyl)-N-(2-methoxybenzyl)acetamide
Show/Hide
|
C28H35N3O6S
|
1
|
| 1 |
EC50 = 0.04 nM
|
|
|
|
CP0507954
|
2-(3-((R)-2-((R)-2-hydroxy-2-(4-hydroxy-3-(methylsulfonamido)phenyl)ethylamino)propyl)phenyl)-N-phenethylacetamide
Show/Hide
|
C28H35N3O5S
|
1
|
| 1 |
EC50 = 0.04 nM
|
|
|
|
CP0504447
|
2-(3-((R)-2-((R)-2-hydroxy-2-(4-hydroxy-3-(methylsulfonamido)phenyl)ethylamino)propyl)phenyl)-N-(3-phenylpropyl)acetamide
Show/Hide
|
C29H37N3O5S
|
1
|
| 1 |
EC50 = 0.042 nM
|
|
|
|
CP0404074
|
(R)-N-(4-hydroxy-2,6-dimethylbenzyl)-2-(3-(2-(2-hydroxy-2-(4-hydroxy-3-(methylsulfonamido)phenyl)ethylamino)-2-methylpropyl)phenyl)acetamide
Show/Hide
|
C30H39N3O6S
|
1
|
| 1 |
EC50 = 0.045 nM
|
|
|
|
CP0416324
|
N-[(2-ethoxyphenyl)methyl]-2-[3-[(2R)-2-[[(2R)-2-hydroxy-2-[4-hydroxy-3-(methanesulfonamido)phenyl]ethyl]amino]propyl]phenyl]acetamide
Show/Hide
|
C29H37N3O6S
|
1
|
| 1 |
EC50 = 0.048 nM
|
|
|
|
CP0510689
|
N-benzyl-5-[(2R)-2-[[(2R)-2-hydroxy-2-[4-hydroxy-3-(hydroxymethyl)phenyl]ethyl]amino]propyl]-1H-indole-2-carboxamide
Show/Hide
|
C28H31N3O4
|
1
|
| 1 |
EC50 = 0.049 nM
|
|
|
|
CP0505412
|
N-(cyclobutylmethyl)-5-[(2R)-2-[[(2R)-2-hydroxy-2-[4-hydroxy-3-(hydroxymethyl)phenyl]ethyl]amino]propyl]-1H-indole-2-carboxamide
Show/Hide
|
C26H33N3O4
|
1
|
| 1 |
EC50 = 0.051 nM
|
|
|
|
CP0505413
|
N-[(2,6-difluorophenyl)methyl]-5-[(2R)-2-[[(2R)-2-hydroxy-2-[4-hydroxy-3-(hydroxymethyl)phenyl]ethyl]amino]propyl]-1H-indole-2-carboxamide
Show/Hide
|
C28H29F2N3O4
|
1
|
| 1 |
EC50 = 0.053 nM
|
|
|
|
CP0386941
|
N-[2-hydroxy-5-[1-hydroxy-2-[(2-methyl-1-phenylpropan-2-yl)amino]ethyl]phenyl]methanesulfonamide
Show/Hide
|
C19H26N2O4S
|
1
|
| 1 |
EC50 = 0.054 nM
|
|
|
|
CP0404075
|
N-[(3,4-dimethylphenyl)methyl]-2-[3-[(2R)-2-[[(2R)-2-hydroxy-2-[4-hydroxy-3-(methanesulfonamido)phenyl]ethyl]amino]propyl]phenyl]acetamide
Show/Hide
|
C29H37N3O5S
|
1
|
| 1 |
EC50 = 0.056 nM
|
|
|
|
CP0296443
|
N-[(2,6-dimethoxyphenyl)methyl]-5-[(2R)-2-[[(2R)-2-hydroxy-2-[4-hydroxy-3-(hydroxymethyl)phenyl]ethyl]amino]propyl]-1H-indole-2-carboxamide
Show/Hide
|
C30H35N3O6
|
1
|
| 1 |
EC50 = 0.058 nM
|
|
|
|
CP0306158
|
5-((R)-2-((R)-2-hydroxy-2-(4-hydroxy-3-(hydroxymethyl)phenyl)ethylamino)propyl)-N-((R)-1-phenylethyl)-1H-indole-2-carboxamide
Show/Hide
|
C29H33N3O4
|
1
|
| 1 |
EC50 = 0.058 nM
|
|
|
|
CP0504446
|
(R)-N-(3,4-dichlorobenzyl)-2-(3-(2-(2-hydroxy-2-(4-hydroxy-3-(methylsulfonamido)phenyl)ethylamino)-2-methylpropyl)phenyl)acetamide
Show/Hide
|
C28H33Cl2N3O5S
|
1
|
| 1 |
EC50 = 0.066 nM
|
|
|
|
CP0510345
|
(R)-N-(3,5-dichloro-4-hydroxybenzyl)-2-(3-(2-(2-hydroxy-2-(4-hydroxy-3-(methylsulfonamido)phenyl)ethylamino)-2-methylpropyl)phenyl)acetamide
Show/Hide
|
C28H33Cl2N3O6S
|
1
|
| 1 |
EC50 = 0.091 nM
|
|
|
|
CP0539700
|
5-{(R)-2-[(R)-2-hydroxy-2-(4-hydroxy-3-hydroxymethyl-phenyl)-ethylamino]-propyl}-1H-indole-2-carboxylic acid 4-sulfamoyl-benzylamide
Show/Hide
|
C28H32N4O6S
|
1
|
| 1 |
EC50 = 0.122 nM
|
|
|
|
CP0853347
|
2-(Hydroxymethyl)-4-((1R)-1-hydroxy-2-{[6-({2-[(1-naphthalenylmethyl)oxy]ethyl}oxy)hexyl]amino}ethyl)phenolAcetate Salt
Show/Hide
|
C30H41NO7
|
1
|
| 1 |
EC50 = 0.1259 nM
|
|
|
|
CP0514462
|
(R)-N-(3,5-dichloro-2-hydroxybenzyl)-2-(3-(2-(2-hydroxy-2-(4-hydroxy-3-(methylsulfonamido)phenyl)ethylamino)-2-methylpropyl)phenyl)acetamide
Show/Hide
|
C28H33Cl2N3O6S
|
1
|
| 1 |
EC50 = 0.13 nM
|
|
|
|
CP0068209
|
4-[1-hydroxy-2-(isopropylamino)ethyl]pyrocatechol;hydrochloride
Show/Hide
|
C11H17NO3
|
9
|
| 1 |
EC50 = 0.1585 nM
|
|
|
| 2 |
EC50 = 0.84 nM
|
|
|
| 3 |
EC50 = 2 nM
|
|
|
| 4 |
EC50 = 3 nM
|
|
|
| 5 |
EC50 = 13 nM
|
|
|
| 6 |
EC50 = 39.81 nM
|
|
|
| 7 |
Kd = 740 nM
|
|
|
| 8 |
Ki = 46 nM
|
|
|
| 9 |
Ki = 676.08 nM
|
|
|
|
CP0847406
|
3-(4-{[6-({(2R)-2-[3-(Formylamino)-4-hydroxyphenyl]-2-hydroxyethyl}amino)hexyl]oxy}butyl)benzenesulfonamide fumarate salt
Show/Hide
|
C29H41N3O10S
|
1
|
| 1 |
EC50 = 0.1585 nM
|
|
|
|
CP0859379
|
3-(4-{[6-({(2R)-2-Hydroxy-2-[4-hydroxy-3-(hydroxymethyl)phenyl]ethyl}amino)-hexyl]oxy}butyl)benzenesulfonamide cinnamate salt
Show/Hide
|
C34H46N2O8S
|
1
|
| 1 |
EC50 = 0.1585 nM
|
|
|
|
CP0851887
|
N-[3-(4-{[6-({(2R)-2-Hydroxy-2-[4-hydroxy-3-(hydroxymethyl)phenyl]ethyl}amino)hexyl]oxy}butyl)-5-methylphenyl]urea acetate salt
Show/Hide
|
C29H45N3O7
|
1
|
| 1 |
EC50 = 0.1585 nM
|
|
|
|
CP0459847
|
5-[(2R)-2-[[(2R)-2-hydroxy-2-[4-hydroxy-3-(hydroxymethyl)phenyl]ethyl]amino]propyl]-N-[(4-hydroxyphenyl)methyl]-1H-indole-2-carboxamide
Show/Hide
|
C28H31N3O5
|
1
|
| 1 |
EC50 = 0.164 nM
|
|
|
|
CP0505983
|
(R)-N-(5-chloro-2-hydroxybenzyl)-2-(3-(2-(2-hydroxy-2-(4-hydroxy-3-(methylsulfonamido)phenyl)ethylamino)-2-methylpropyl)phenyl)acetamide
Show/Hide
|
C28H34ClN3O6S
|
1
|
| 1 |
EC50 = 0.17 nM
|
|
|
|
CP0850211
|
N-Cyclohexyl-3-(4-{[6-({(2R)-2-hydroxy-2-[4-hydroxy-3-(hydroxymethyl)phenyl]ethyl}amino)hexyl]oxy}butyl)benzenesulfonamide acetate salt
Show/Hide
|
C33H52N2O8S
|
1
|
| 1 |
EC50 = 0.1995 nM
|
|
|
|
CP0386940
|
(R)-2-(3-(2-(2-hydroxy-2-(4-hydroxy-3-(methylsulfonamido)phenyl)ethylamino)-2-methylpropyl)phenyl)-N-((6-hydroxynaphthalen-2-yl)methyl)acetamide
Show/Hide
|
C32H37N3O6S
|
1
|
| 1 |
EC50 = 0.21 nM
|
|
|
|
CP0504445
|
(R)-2-(3-(2-(2-hydroxy-2-(4-hydroxy-3-(methylsulfonamido)phenyl)ethylamino)-2-methylpropyl)phenyl)-N-((4'-hydroxybiphenyl-4-yl)methyl)acetamide
Show/Hide
|
C34H39N3O6S
|
1
|
| 1 |
EC50 = 0.24 nM
|
|
|
|
CP0853348
|
N-(3-{[(2-{[6-({(2R)-2-Hydroxy-2-[4-hydroxy-3-(hydroxymethyl)-phenyl]-ethyl}amino)hexyl]oxy}ethyl)oxy]methyl}phenyl)methanesulfonamideAcetate Salt
Show/Hide
|
C27H42N2O9S
|
1
|
| 1 |
EC50 = 0.2512 nM
|
|
|
|
CP0871785
|
2-{3-[3-(4-{[6-({(2R)-2-Hydroxy-2-[4-hydroxy-3-(hydroxymethyl)phenyl]ethyl}amino)hexyl]oxy}butyl)phenyl]-2,5-dioxo-1-imidazolidinyl}acetamide acetate salt
Show/Hide
|
C32H46N4O9
|
1
|
| 1 |
EC50 = 0.2512 nM
|
|
|
|
CP0851889
|
(R)-2-(3-(3-(4-(6-(2-hydroxy-2-(4-hydroxy-3-(hydroxymethyl)phenyl)ethylamino)hexyloxy)butyl)phenyl)ureido)acetamide formate
Show/Hide
|
C29H44N4O8
|
1
|
| 1 |
EC50 = 0.2512 nM
|
|
|
|
CP0539658
|
5-[(2R)-2-[[(2R)-2-hydroxy-2-[4-hydroxy-3-(hydroxymethyl)phenyl]ethyl]amino]propyl]-N-[2-(3-methoxyphenyl)ethyl]-1H-indole-2-carboxamide
Show/Hide
|
C30H35N3O5
|
1
|
| 1 |
EC50 = 0.254 nM
|
|
|
|
CP0505414
|
N-[(2,6-dimethoxyphenyl)methyl]-5-[(2R)-2-[[(2R)-2-hydroxy-2-[4-hydroxy-3-(hydroxymethyl)phenyl]ethyl]amino]butyl]-1H-indole-2-carboxamide
Show/Hide
|
C31H37N3O6
|
1
|
| 1 |
EC50 = 0.258 nM
|
|
|
|
CP0545497
|
(R)-2-(3-(2-(2-hydroxy-2-(4-hydroxy-3-(methylsulfonamido)phenyl)ethylamino)-2-methylpropyl)phenyl)-N-((4'-hydroxybiphenyl-3-yl)methyl)acetamide
Show/Hide
|
C34H39N3O6S
|
1
|
| 1 |
EC50 = 0.26 nM
|
|
|
|
CP0849999
|
(R)-N-cyclopentyl-2-(3-(3-(4-(6-(2-hydroxy-2-(4-hydroxy-3-(hydroxymethyl)phenyl)ethylamino)hexyloxy)butyl)phenyl)ureido)acetamide acetate
Show/Hide
|
C35H54N4O8
|
1
|
| 1 |
EC50 = 0.3162 nM
|
|
|
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CP0372757
|
(R)-N-(2-chloro-4-hydroxybenzyl)-N-ethyl-2-(3-(2-(2-hydroxy-2-(4-hydroxy-3-(methylsulfonamido)phenyl)ethylamino)-2-methylpropyl)phenyl)acetamide
Show/Hide
|
C30H38ClN3O6S
|
1
|
| 1 |
EC50 = 0.37 nM
|
|
|
|
CP0708199
|
Vilanterol
Show/Hide
|
C26H37Cl2NO7
|
1
|
| 1 |
EC50 = 0.3981 nM
|
|
|
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CP0874631
|
4-[(1R)-2-({6-[(2-{[(2,5-Dichlorophenyl)methyl]oxy}ethyl)oxy]-hexyl}-amino)-1-hydroxyethyl]-2-(hydroxymethyl)phenol Acetate Salt
Show/Hide
|
C26H37Cl2NO7
|
1
|
| 1 |
EC50 = 0.3981 nM
|
|
|
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CP0906725
|
4-[(1R)-2-({6-[(2-{[(3,5-Dimethylphenyl)methyl]oxy}ethyl)oxy]-hexyl}-amino)-1-hydroxyethyl]-2-(hydroxymethyl)phenol Acetate Salt
Show/Hide
|
C28H43NO7
|
1
|
| 1 |
EC50 = 0.3981 nM
|
|
|
|
CP0847073
|
SID93576620
Show/Hide
|
C23H30N2O9
|
1
|
| 1 |
EC50 = 0.4 nM
|
|
|
|
CP0066323
|
CAS_73573-87-2
Show/Hide
|
C19H24N2O4
|
4
|
| 1 |
EC50 = 0.5012 nM
|
|
|
| 2 |
Ki = 2.6 nM
|
|
|
| 3 |
Ki = 23 nM
|
|
|
| 4 |
Ki = 26 nM
|
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CP0847408
|
3-(4-{[6-({(2R)-2-Hydroxy-2-[4-hydroxy-3-(hydroxymethyl)-phenyl]ethyl}amino)hexyl]oxy}butyl)-N-isopropylbenzenesulfonamide acetate salt
Show/Hide
|
C30H48N2O8S
|
1
|
| 1 |
EC50 = 0.5012 nM
|
|
|
|
CP0910906
|
4-(4-{[6-({(2R)-2-Hydroxy-2-[4-hydroxy-3-(hydroxymethyl)-phenyl]ethyl}amino)hexyl]oxy}butyl)benzenesulfonamide acetate salt
Show/Hide
|
C27H42N2O8S
|
1
|
| 1 |
EC50 = 0.5012 nM
|
|
|
|
CP0708203
|
(R,R)-formoterol fumarate
Show/Hide
|
C23H28N2O8
|
1
|
| 1 |
EC50 = 0.5012 nM
|
|
|
|
CP0850450
|
Formoterol fumarate
Show/Hide
|
C23H30N2O9
|
1
|
| 1 |
EC50 = 0.5012 nM
|
|
|
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CP0852279
|
(R)-1-ethyl-3-(4-(4-(6-(2-hydroxy-2-(4-hydroxy-3-(hydroxymethyl)phenyl)ethylamino)hexyloxy)butyl)phenyl)urea acetate
Show/Hide
|
C30H47N3O7
|
1
|
| 1 |
EC50 = 0.5012 nM
|
|
|
|
CP0888674
|
(R)-1-(3-(4-(6-(2-hydroxy-2-(4-hydroxy-3-(hydroxymethyl)phenyl)ethylamino)hexyloxy)butyl)benzyl)urea acetate
Show/Hide
|
C29H45N3O7
|
1
|
| 1 |
EC50 = 0.5012 nM
|
|
|
|
CP0898259
|
4-((1R)-2-{[6-({4-[3-(Cyclopentylsulfonyl)-5-methylphenyl]butyl}oxy)hexyl]amino}-1-hydroxyethyl)-2-(hydroxymethyl)phenol acetic acid salt
Show/Hide
|
C33H51NO8S
|
1
|
| 1 |
EC50 = 0.5012 nM
|
|
|
|
CP0847407
|
3-(4-{[6-({(2R)-2-Hydroxy-2-[4-hydroxy-3-(hydroxymethyl)-phenyl]ethyl}amino)hexyl]oxy}butyl)-N-methylbenzenesulfonamide acetate salt
Show/Hide
|
C28H44N2O8S
|
1
|
| 1 |
EC50 = 0.631 nM
|
|
|
|
CP0913516
|
1-{[3-(4-{[6-({(2R)-2-Hydroxy-2-[4-hydroxy-3-(hydroxymethyl)phenyl]ethyl}amino)hexyl]oxy}butyl)phenyl]methyl}-2,4-imidazolidinedione acetate salt
Show/Hide
|
C31H45N3O8
|
1
|
| 1 |
EC50 = 0.631 nM
|
|
|
|
CP0917314
|
3-[3-(4-{[6-([(2R)-2-Hydroxy-2-[4-hydroxy-3-(hydroxymethyl)phenyl]ethyl]amino)hexyl]oxy}butyl)phenyl]imidazolidine-2,4-dione acetate
Show/Hide
|
C30H43N3O8
|
1
|
| 1 |
EC50 = 0.631 nM
|
|
|
|
CP0870890
|
(R)-1-ethyl-3-(3-(4-(6-(2-hydroxy-2-(4-hydroxy-3-(hydroxymethyl)phenyl)ethylamino)hexyloxy)butyl)benzyl)urea acetate
Show/Hide
|
C31H49N3O7
|
1
|
| 1 |
EC50 = 0.631 nM
|
|
|
|
CP0510690
|
1-benzyl-N-[(2,6-dimethoxyphenyl)methyl]-5-[(2R)-2-[[(2R)-2-hydroxy-2-[4-hydroxy-3-(hydroxymethyl)phenyl]ethyl]amino]propyl]indole-2-carboxamide
Show/Hide
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C37H41N3O6
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1
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| 1 |
EC50 = 0.687 nM
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CP0371922
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6-hydroxy-8-[1-hydroxy-2-[[2-methyl-1-(2-methylphenyl)propan-2-yl]amino]ethyl]-4H-1,4-benzoxazin-3-one
Show/Hide
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C21H26N2O4
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1
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| 1 |
EC50 = 0.7 nM
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CP0485251
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N-[(2,6-dimethoxyphenyl)methyl]-5-[(2R)-2-[[(2R)-2-hydroxy-2-[4-hydroxy-3-(hydroxymethyl)phenyl]ethyl]amino]propyl]-1-methylindole-2-carboxamide
Show/Hide
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C31H37N3O6
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1
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| 1 |
EC50 = 0.706 nM
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CP0871038
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2-(4-{[6-({(2R)-2-Hydroxy-2-[4-hydroxy-3-(hydroxymethyl)-phenyl]ethyl}amino)hexyl]oxy}butyl)benzenesulfonamide acetate salt
Show/Hide
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C27H42N2O8S
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1
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| 1 |
EC50 = 0.7943 nM
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CP0847188
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4-[(1R)-1-Hydroxy-2-({6-[(2-{[(3-hydroxyphenyl)methyl]oxy}-ethyl)oxy]-hexyl}amino)ethyl]-2-(hydroxymethyl)phenol Acetate Salt
Show/Hide
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C26H39NO8
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1
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| 1 |
EC50 = 0.7943 nM
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CP0499227
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3-[3-[4-[6-[[(2R)-2-hydroxy-2-[4-hydroxy-3-(hydroxymethyl)phenyl]ethyl]amino]hexoxy]butyl]phenyl]-1H-pyrimidine-2,4-dione
Show/Hide
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C29H39N3O6
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1
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| 1 |
EC50 = 0.7943 nM
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CP0884854
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3-[3-(4-{[6-({(2R)-2-Hydroxy-2-[4-hydroxy-3-(hydroxymethyl)phenyl]ethyl}amino)hexyl]oxy}butyl)phenyl]-5,5-dimethyl-2,4-imidazolidinedione acetate salt
Show/Hide
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C32H47N3O8
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1
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| 1 |
EC50 = 0.7943 nM
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CP0917315
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1-{[3-(4-{[6-({(2R)-2-Hydroxy-2-[4-hydroxy-3-(hydroxymethyl)phenyl]ethyl}amino)hexyl]oxy}butyl)phenyl]methyl}-2,4,5-imidazolidinetrione formate salt
Show/Hide
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C30H41N3O9
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1
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| 1 |
EC50 = 0.7943 nM
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CP0903932
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(R)-1-(3-(4-(6-(2-hydroxy-2-(4-hydroxy-3-(hydroxymethyl)phenyl)ethylamino)hexyloxy)butyl)phenyl)urea acetate
Show/Hide
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C28H43N3O7
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1
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| 1 |
EC50 = 0.7943 nM
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CP0449097
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2-[4-[[(2R)-2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]propyl]amino]phenyl]-N-[(4-methylphenyl)methyl]acetamide
Show/Hide
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C27H32ClN3O2
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1
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| 1 |
EC50 = 1 nM
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CP0850324
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2-(Hydroxymethyl)-4-{(1R)-1-hydroxy-2-[(6-{4-[3-(piperidin-1-ylsulfonyl)phenyl]butoxy}hexyl)amino]ethyl}phenol
Show/Hide
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C32H50N2O8S
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1
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| 1 |
EC50 = 1 nM
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CP0888635
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3-(4-{[6-({(2R)-2-Hydroxy-2-[4-hydroxy-3-(hydroxymethyl)-phenyl]ethyl}amino)hexyl]oxy}butyl)-N,N-dimethylbenzenesulfonamide acetate salt
Show/Hide
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C29H46N2O8S
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1
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| 1 |
EC50 = 1 nM
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CP0451500
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2-[[3-[4-[6-[[(2R)-2-hydroxy-2-[4-hydroxy-3-(hydroxymethyl)phenyl]ethyl]amino]hexoxy]butyl]phenyl]carbamoylamino]acetic acid
Show/Hide
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C28H41N3O7
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1
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| 1 |
EC50 = 1 nM
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CP0851886
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(R)-1-ethyl-3-(3-(4-(6-(2-hydroxy-2-(4-hydroxy-3-(hydroxymethyl)phenyl)ethylamino)hexyloxy)butyl)phenyl)urea acetate
Show/Hide
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C30H47N3O7
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1
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| 1 |
EC50 = 1 nM
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CP0851888
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(R)-1-cyclohexyl-3-(3-(4-(6-(2-hydroxy-2-(4-hydroxy-3-(hydroxymethyl)phenyl)ethylamino)hexyloxy)butyl)phenyl)urea acetate
Show/Hide
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C34H53N3O7
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1
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| 1 |
EC50 = 1 nM
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CP0888673
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(R)-1-(3-(4-(6-(2-hydroxy-2-(4-hydroxy-3-(hydroxymethyl)phenyl)ethylamino)hexyloxy)butyl)-5-(trifluoromethyl)phenyl)urea acetate
Show/Hide
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C29H42F3N3O7
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1
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| 1 |
EC50 = 1 nM
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CP0875710
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4-((1R)-2-{[6-({4-[3-(3-Cyclopenten-1-ylsulfonyl)phenyl]butyl}oxy)hexyl]amino}-1-hydroxyethyl)-2-(hydroxymethyl)phenol acetate salt
Show/Hide
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C32H47NO8S
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1
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| 1 |
EC50 = 1 nM
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CP0118781
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[3-[(2R)-2-[[(2R)-2-hydroxy-2-[3-(thiophen-2-ylsulfonylamino)phenyl]ethyl]amino]propyl]-1H-indol-7-yl] thiophene-2-sulfonate
Show/Hide
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C27H27N3O6S4
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1
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| 1 |
EC50 = 1.2 nM
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CP0877391
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2-(Hydroxymethyl)-4-{(1R)-1-hydroxy-2-[(6-{4-[3-(morpholin-4-ylsulfonyl)phenyl]butoxy}hexyl)amino]ethyl}phenol acetate salt
Show/Hide
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C31H48N2O9S
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1
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| 1 |
EC50 = 1.259 nM
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CP0851858
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1-[3-(4-{[6-({(2R)-2-Hydroxy-2-[4-hydroxy-3-(hydroxymethyl)phenyl]ethyl}amino)hexyl]oxy}butyl)phenyl]-2,4(1H,3H)-pyrimidinedione acetate salt
Show/Hide
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C31H43N3O8
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1
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| 1 |
EC50 = 1.259 nM
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CP0884855
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3-{[3-(4-{[6-({(2R)-2-Hydroxy-2-[4-hydroxy-3-(hydroxymethyl)phenyl]ethyl}amino)hexyl]oxy}butyl)phenyl]methyl}-2,4-imidazolidinedione acetate salt
Show/Hide
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C31H45N3O8
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1
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| 1 |
EC50 = 1.259 nM
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CP0103438
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[3-[(2R)-2-[[(2R)-2-hydroxy-2-[3-(thiophen-2-ylsulfonylamino)phenyl]ethyl]amino]propyl]-1H-indol-7-yl] pyridine-3-sulfonate
Show/Hide
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C28H28N4O6S3
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1
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| 1 |
EC50 = 1.3 nM
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CP0387196
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8-[2-[[1-(4-chlorophenyl)-2-methylpropan-2-yl]amino]-1-hydroxyethyl]-6-hydroxy-4H-1,4-benzoxazin-3-one
Show/Hide
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C20H23ClN2O4
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1
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| 1 |
EC50 = 1.3 nM
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CP0402051
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6-hydroxy-8-[1-hydroxy-2-[[2-methyl-1-[2-(trifluoromethyl)phenyl]propan-2-yl]amino]ethyl]-4H-1,4-benzoxazin-3-one
Show/Hide
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C21H23F3N2O4
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1
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| 1 |
EC50 = 1.4 nM
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CP0844800
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rac-6-hydroxy-8-(1-hydroxy-2-(1-(4-methoxyphenyl)-2-methylpropan-2-ylamino)ethyl)-2H-benzo[b][1,4]oxazin-3(4H)-one
Show/Hide
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C21H26N2O5
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1
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| 1 |
EC50 = 1.4 nM
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CP0378048
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[3-[(2R)-2-[[(2R)-2-hydroxy-2-[3-(2-methylprop-2-enylamino)phenyl]ethyl]amino]propyl]-1H-indol-7-yl] methanesulfonate
Show/Hide
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C24H31N3O4S
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1
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| 1 |
EC50 = 1.5 nM
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CP0481594
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[3-[4-[6-[[(2R)-2-hydroxy-2-[4-hydroxy-3-(hydroxymethyl)phenyl]ethyl]amino]hexoxy]butyl]phenyl]methanesulfonamide
Show/Hide
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C26H40N2O6S
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1
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| 1 |
EC50 = 1.585 nM
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CP0859375
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3-{[(2-{[6-({(2R)-2-Hydroxy-2-[4-hydroxy-3-(hydroxymethyl)-phenyl]-ethyl}amino)hexyl]oxy}ethyl)oxy]methyl}benzenesulfonamideacetate salt
Show/Hide
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C26H40N2O9S
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1
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| 1 |
EC50 = 1.585 nM
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CP0924345
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N-(3-{[(2-{[6-({(2R)-2-Hydroxy-2-[4-hydroxy-3-(hydroxymethyl)-phenyl]ethyl}amino)hexyl]oxy}ethyl)oxy]methyl}phenyl)urea Acetate salt
Show/Hide
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C27H41N3O8
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1
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| 1 |
EC50 = 1.585 nM
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CP0875711
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4-((1R)-2-{[6-({4-[3-(Cyclohexylsulfonyl)phenyl]butyl}oxy)hexyl]amino}-1-hydroxyethyl)-2-(hydroxymethyl)phenol acetate salt
Show/Hide
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C33H51NO8S
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1
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| 1 |
EC50 = 1.585 nM
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CP0390982
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4-[2-[6-[[(2R)-2-hydroxy-2-[4-hydroxy-3-(hydroxymethyl)phenyl]ethyl]amino]hexoxy]ethoxymethyl]benzenesulfonamide
Show/Hide
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C24H36N2O7S
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1
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| 1 |
EC50 = 1.995 nM
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CP0890908
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3-[4-(4-{[6-({(2R)-2-Hydroxy-2-[4-hydroxy-3-(hydroxymethyl)phenyl]ethyl}amino)hexyl]oxy}butyl)phenyl]-2,4-imidazolidinedione acetate salt
Show/Hide
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C30H43N3O8
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1
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| 1 |
EC50 = 1.995 nM
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CP0708202
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4-((1R)-2-{[6-({4-[3-(Cyclopentylsulfonyl)phenyl]butyl}oxy)-hexyl]amino}-1-hydroxyethyl)-2-(hydroxymethyl)phenol acetate salt
Show/Hide
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C32H49NO8S
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1
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| 1 |
EC50 = 1.995 nM
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CP0467168
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[3-[(2R)-2-[[(2R)-2-hydroxy-2-[3-(prop-2-enylamino)phenyl]ethyl]amino]propyl]-1H-indol-7-yl] methanesulfonate
Show/Hide
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C23H29N3O4S
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1
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| 1 |
EC50 = 2.2 nM
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CP0409670
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(S)-6-(4-(2-(3-(3-(2-cyclopentylethyl)-2-oxo-2,3-dihydro-1H-benzo[d]imidazol-4-yloxy)-2-hydroxypropylamino)-2-methylpropyl)phenoxy)nicotinamide
Show/Hide
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C33H41N5O5
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1
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| 1 |
EC50 = 2.4 nM
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CP0371926
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6-hydroxy-8-[1-hydroxy-2-[(2-methyl-1-phenylpropan-2-yl)amino]ethyl]-4H-1,4-benzoxazin-3-one
Show/Hide
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C20H24N2O4
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1
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| 1 |
EC50 = 2.4 nM
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CP0224386
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5-((R)-2-(4-(4-(3-((R)-3-(diisopropylamino)-1-phenylpropyl)-4-hydroxyphenyl)butoxy)phenethylamino)-1-hydroxyethyl)-8-hydroxyquinolin-2(1H)-one
Show/Hide
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C44H55N3O5
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1
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| 1 |
EC50 = 2.4 nM
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CP0850210
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3-(3-{[7-({(2R)-2-Hydroxy-2-[4-hydroxy-3-(hydroxymethyl)-phenyl]ethyl}amino)heptyl]oxy}propyl)benzenesulfonamide sulfamate salt
Show/Hide
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C25H41N3O9S2
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1
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| 1 |
EC50 = 2.512 nM
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CP0849916
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2-(Hydroxymethyl)-4-[(1R)-1-hydroxy-2-({6-[(2-{[(4-methylphenyl)methyl]oxy}ethyl)oxy]hexyl}amino)ethyl]phenol Acetate Salt
Show/Hide
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C27H41NO7
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1
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| 1 |
EC50 = 2.512 nM
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CP0867970
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4-[(1R)-2-({6-[(2-{[(4-Chlorophenyl)methyl]oxy}ethyl)oxy]-hexyl}amino)-1-hydroxyethyl]-2-(hydroxymethyl)phenol Acetate Salt
Show/Hide
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C26H38ClNO7
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1
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| 1 |
EC50 = 2.512 nM
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CP0874619
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2-(Hydroxymethyl)-4-((1R)-1-hydroxy-2-{[6-({2-[(phenylmethyl)-oxy]ethyl}oxy)hexyl]amino}ethyl)phenol
Show/Hide
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C26H39NO7
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1
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| 1 |
EC50 = 2.512 nM
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CP0884853
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3-[2-(4-{[6-({(2R)-2-Hydroxy-2-[4-hydroxy-3-(hydroxymethyl)phenyl]ethyl}amino)hexyl]oxy}butyl)phenyl]-2,4-imidazolidinedione
Show/Hide
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C28H39N3O6
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1
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| 1 |
EC50 = 2.512 nM
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CP0917316
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1-[3-(4-{[6-({(2R)-2-Hydroxy-2-[4-hydroxy-3-(hydroxymethyl)phenyl]ethyl}amino)hexyl]oxy}butyl)phenyl]-2,4-imidazolidinedione acetate salt
Show/Hide
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C30H43N3O8
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1
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| 1 |
EC50 = 2.512 nM
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CP0485250
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N-[(2,6-dimethoxyphenyl)methyl]-1-ethyl-5-[(2R)-2-[[(2R)-2-hydroxy-2-[4-hydroxy-3-(hydroxymethyl)phenyl]ethyl]amino]propyl]indole-2-carboxamide
Show/Hide
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C32H39N3O6
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1
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| 1 |
EC50 = 2.55 nM
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CP0418660
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3-(2-(2-hydroxy-2-(5-hydroxy-3-oxo-3,4-dihydro-2H-benzo[b][1,4]oxazin-8-yl)ethylamino)-2-methylpropyl)benzoic acid
Show/Hide
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C21H24N2O6
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1
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| 1 |
EC50 = 2.9 nM
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CP0103437
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Benzenesulfonic acid 3-(2-{(R)-(R)-2-hydroxy-2-[3-(thiophene-2-sulfonylamino)-phenyl]-ethylamino}-propyl)-1H-indol-7-yl ester
Show/Hide
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C29H29N3O6S3
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1
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| 1 |
EC50 = 3.1 nM
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CP0404412
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N-[[4-[[(2R)-2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]propyl]amino]phenyl]methyl]acetamide
Show/Hide
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C20H26ClN3O2
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1
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| 1 |
EC50 = 3.162 nM
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CP0371867
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8-[2-[[1-(4-fluorophenyl)-2-methylpropan-2-yl]amino]-1-hydroxyethyl]-6-hydroxy-4H-1,4-benzoxazin-3-one
Show/Hide
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C20H23FN2O4
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1
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| 1 |
EC50 = 3.4 nM
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CP0488648
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6-hydroxy-8-[1-hydroxy-2-[[2-methyl-1-[3-(trifluoromethyl)phenyl]propan-2-yl]amino]ethyl]-4H-1,4-benzoxazin-3-one
Show/Hide
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C21H23F3N2O4
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1
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| 1 |
EC50 = 3.4 nM
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CP0761842
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(R)-(3'-Chloro-4'-hydroxy-biphenyl-2-yl)-carbamic acid 1-{9-[2-hydroxy-2-(4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-nonyl}-piperidin-4-yl ester
Show/Hide
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C36H49ClN4O7S
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1
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| 1 |
EC50 = 3.7 nM
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CP0235763
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[1-[9-[[(2R)-2-hydroxy-2-(8-hydroxy-2-oxo-1H-quinolin-5-yl)ethyl]amino]nonyl]piperidin-4-yl] N-[2-(3-chloro-4-hydroxyphenyl)phenyl]carbamate
Show/Hide
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C38H47ClN4O6
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1
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| 1 |
EC50 = 3.7 nM
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CP0481497
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6-hydroxy-8-[1-hydroxy-2-[[2-methyl-1-(3-methylphenyl)propan-2-yl]amino]ethyl]-4H-1,4-benzoxazin-3-one
Show/Hide
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C21H26N2O4
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1
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| 1 |
EC50 = 4.1 nM
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CP0383083
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4-Aminomethylpiperidine substituted analogue
Show/Hide
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C26H34N4O9S
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1
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| 1 |
EC50 = 5 nM
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CP0374871
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N-[[4-[[(2R)-2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]propyl]amino]phenyl]methyl]methanesulfonamide
Show/Hide
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C19H26ClN3O3S
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1
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| 1 |
EC50 = 5.012 nM
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CP0374720
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(R)-1-((R)-3-Chloro-phenyl)-2-[2-(7-methoxy-1H-indol-3-yl)-1-methyl-ethylamino]-ethanol
Show/Hide
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C20H23ClN2O2
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1
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| 1 |
EC50 = 5.2 nM
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CP0039163
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[3-[(2R)-2-[[(2R)-2-hydroxy-2-[3-(thiophen-2-ylsulfonylamino)phenyl]ethyl]amino]propyl]-1H-indol-7-yl] octane-1-sulfonate
Show/Hide
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C31H41N3O6S3
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1
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| 1 |
EC50 = 5.6 nM
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CP0378245
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N-[5-[(1R)-2-[6-[4-[3-[(1R)-3-[di(propan-2-yl)amino]-1-phenylpropyl]-4-hydroxyphenyl]butoxy]hexylamino]-1-hydroxyethyl]-2-hydroxyphenyl]methanesulfonamide
Show/Hide
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C40H61N3O6S
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1
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| 1 |
EC50 = 5.7 nM
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CP0118799
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[3-[(2R)-2-[[(2R)-2-hydroxy-2-[3-(thiophen-2-ylsulfonylamino)phenyl]ethyl]amino]propyl]-1H-indol-7-yl] propane-2-sulfonate
Show/Hide
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C26H31N3O6S3
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1
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| 1 |
EC50 = 6.2 nM
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CP0071878
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N-[3-[(1R)-1-hydroxy-2-[[(2R)-1-(7-methoxy-1H-indol-3-yl)propan-2-yl]amino]ethyl]phenyl]thiophene-2-sulfonamide
Show/Hide
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C24H27N3O4S2
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1
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| 1 |
EC50 = 6.6 nM
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CP0071879
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N-[3-[(1R)-1-hydroxy-2-[[(2R)-1-(7-phenylmethoxy-1H-indol-3-yl)propan-2-yl]amino]ethyl]phenyl]thiophene-2-sulfonamide
Show/Hide
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C30H31N3O4S2
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1
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| 1 |
EC50 = 6.6 nM
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CP0486040
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2-[3-(2-{(R)-(R)-2-Hydroxy-2-[3-(thiophene-2-sulfonylamino)-phenyl]-ethylamino}-propyl)-1H-indol-7-yloxy]-N,N-dimethyl-acetamide
Show/Hide
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C27H32N4O5S2
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1
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| 1 |
EC50 = 6.8 nM
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CP0497035
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4-[3-(2-{(R)-(R)-2-Hydroxy-2-[3-(thiophene-2-sulfonylamino)-phenyl]-ethylamino}-propyl)-1H-indol-7-yloxysulfonyl]-benzoic acid ethyl ester
Show/Hide
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C32H33N3O8S3
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1
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| 1 |
EC50 = 7.2 nM
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CP0279836
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Butane-1-sulfonic acid 3-(2-{(R)-(R)-2-hydroxy-2-[3-(thiophene-2-sulfonylamino)-phenyl]-ethylamino}-propyl)-1H-indol-7-yl ester
Show/Hide
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C27H33N3O6S3
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1
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| 1 |
EC50 = 7.3 nM
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CP0198056
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[3-[(2R)-2-[[(2R)-2-hydroxy-2-[3-(naphthalen-2-ylmethylamino)phenyl]ethyl]amino]propyl]-1H-indol-7-yl] methanesulfonate
Show/Hide
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C31H33N3O4S
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1
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| 1 |
EC50 = 7.6 nM
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CP0378083
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N-[3-[(1R)-2-[[(2R)-1-(7-ethoxy-1H-indol-3-yl)propan-2-yl]amino]-1-hydroxyethyl]phenyl]thiophene-2-sulfonamide
Show/Hide
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C25H29N3O4S2
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1
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| 1 |
EC50 = 7.7 nM
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CP0405573
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2-[4-[[(2R)-2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]propyl]amino]phenyl]-N-(1,3-thiazol-2-yl)acetamide
Show/Hide
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C22H25ClN4O2S
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1
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| 1 |
EC50 = 7.943 nM
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CP0871071
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3-(5-{[5-({(2R)-2-Hydroxy-2-[4-hydroxy-3-(hydroxymethyl)-phenyl]ethyl}amino)pentyl]oxy}pentyl)benzenesulfonamide acetate salt
Show/Hide
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C27H42N2O8S
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1
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| 1 |
EC50 = 7.943 nM
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CP0482973
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4-[(1R)-1-hydroxy-2-[6-[2-[(4-hydroxyphenyl)methoxy]ethoxy]hexylamino]ethyl]-2-(hydroxymethyl)phenol
Show/Hide
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C24H35NO6
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1
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| 1 |
EC50 = 7.943 nM
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CP0853673
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4-[(1R)-2-({6-[4-(1,1-Dioxo-2,3-dihydro-1-benzothien-6-yl)butoxy]hexyl}amino)-1-hydroxyethyl]-2-(hydroxymethyl)phenol acetate salt
Show/Hide
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C29H43NO8S
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1
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| 1 |
EC50 = 7.943 nM
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CP0452021
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N-[3-[3-[(1R)-3-[di(propan-2-yl)amino]-1-phenylpropyl]-4-hydroxyphenyl]propyl]-2-[3-[2-[[(2R)-2-hydroxy-2-[4-hydroxy-3-(methanesulfonamido)phenyl]ethyl]amino]-2-methylpropyl]phenyl]acetamide
Show/Hide
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C45H62N4O6S
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1
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| 1 |
EC50 = 8.1 nM
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CP0058497
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[3-[(2R)-2-[[(2R)-2-hydroxy-2-[3-(prop-2-ynylamino)phenyl]ethyl]amino]propyl]-1H-indol-7-yl] methanesulfonate
Show/Hide
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C23H27N3O4S
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1
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| 1 |
EC50 = 9.6 nM
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CP0448280
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(1R)-2-[[(2R)-1-anilinopropan-2-yl]amino]-1-(3-chlorophenyl)ethanol
Show/Hide
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C17H21ClN2O
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1
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| 1 |
EC50 = 10 nM
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CP0488117
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N-[2-[4-[[(2R)-2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]propyl]amino]phenyl]ethyl]-4-methylbenzenesulfonamide
Show/Hide
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C26H32ClN3O3S
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1
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| 1 |
EC50 = 10 nM
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CP0403823
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1-[4-(4-{[2-Hydroxy-2-(4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-methyl}-piperidine-1-sulfonyl)-phenyl]-1H-pyrazole-4-carboxylic acid
Show/Hide
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C25H31N5O8S2
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1
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| 1 |
EC50 = 10 nM
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CP0039162
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[3-[(2R)-2-[[(2R)-2-[3-[[(E)-but-2-enyl]amino]phenyl]-2-hydroxyethyl]amino]propyl]-1H-indol-7-yl] methanesulfonate
Show/Hide
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C24H31N3O4S
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1
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| 1 |
EC50 = 10 nM
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CP0847405
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3-(4-{[6-({(2S)-2-Hydroxy-2-[4-hydroxy-3-(hydroxymethyl)-phenyl]ethyl}amino)hexyl]oxy}butyl)benzenesulfonamide acetate salt
Show/Hide
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C27H42N2O8S
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1
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| 1 |
EC50 = 10 nM
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CP0452020
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N-[5-[(1R)-2-[2-[3-[(1R)-3-[di(propan-2-yl)amino]-1-phenylpropyl]-4-hydroxyphenyl]ethylamino]-1-hydroxyethyl]-2-hydroxyphenyl]methanesulfonamide
Show/Hide
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C32H45N3O5S
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1
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| 1 |
EC50 = 10 nM
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CP0492744
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8-[2-[[1-(4-bromophenyl)-2-methylpropan-2-yl]amino]-1-hydroxyethyl]-6-hydroxy-4H-1,4-benzoxazin-3-one
Show/Hide
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C20H23BrN2O4
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1
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| 1 |
EC50 = 10.7 nM
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CP0431043
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[3-[(2R)-2-[[(2R)-2-hydroxy-2-[3-[[(E)-pent-2-enyl]amino]phenyl]ethyl]amino]propyl]-1H-indol-7-yl] methanesulfonate
Show/Hide
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C25H33N3O4S
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1
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| 1 |
EC50 = 11 nM
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CP0470913
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6-hydroxy-8-[1-hydroxy-2-[[2-methyl-1-[4-(trifluoromethoxy)phenyl]propan-2-yl]amino]ethyl]-4H-1,4-benzoxazin-3-one
Show/Hide
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C21H23F3N2O5
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1
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| 1 |
EC50 = 11.9 nM
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CP0458862
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1-[(2,5-difluorophenyl)methyl]-3-[4-[4-[[[(2R)-2-hydroxy-2-[4-hydroxy-3-(methanesulfonamido)phenyl]ethyl]amino]methyl]piperidin-1-yl]sulfonylphenyl]-1-propan-2-ylurea
Show/Hide
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C32H41F2N5O7S2
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1
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| 1 |
EC50 = 12 nM
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CP0378084
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N-[3-[(1R)-1-hydroxy-2-[[(2R)-1-(7-propan-2-yloxy-1H-indol-3-yl)propan-2-yl]amino]ethyl]phenyl]thiophene-2-sulfonamide
Show/Hide
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C26H31N3O4S2
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1
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| 1 |
EC50 = 12 nM
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CP0371868
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8-[2-[[1-(3,5-difluorophenyl)-2-methylpropan-2-yl]amino]-1-hydroxyethyl]-6-hydroxy-4H-1,4-benzoxazin-3-one
Show/Hide
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C20H22F2N2O4
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1
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| 1 |
EC50 = 12.1 nM
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CP0501365
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6-hydroxy-8-[1-hydroxy-2-[[2-methyl-1-[4-(trifluoromethyl)phenyl]propan-2-yl]amino]ethyl]-4H-1,4-benzoxazin-3-one
Show/Hide
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C21H23F3N2O4
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1
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| 1 |
EC50 = 12.4 nM
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CP0375681
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(3-{2-[(R)-2-((R)-3-Chloro-phenyl)-2-hydroxy-ethylamino]-propyl}-1H-indol-7-yloxy)-acetic acid
Show/Hide
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C21H23ClN2O4
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1
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| 1 |
EC50 = 13 nM
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CP0133061
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3-Amino-N-(3-{(R)-1-hydroxy-2-[(R)-2-(7-methanesulfonyl-1H-indol-3-yl)-1-methyl-ethylamino]-ethyl}-phenyl)-benzenesulfonamide
Show/Hide
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C26H30N4O5S2
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1
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| 1 |
EC50 = 13 nM
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CP0405841
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[3-[(2R)-2-[[(2R)-2-hydroxy-2-[3-[[(E)-3-phenylprop-2-enyl]amino]phenyl]ethyl]amino]propyl]-1H-indol-7-yl] methanesulfonate
Show/Hide
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C29H33N3O4S
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1
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| 1 |
EC50 = 13 nM
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CP0473363
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N-[5-[(1R)-2-[2-[4-[4-[3-[(1R)-3-[di(propan-2-yl)amino]-1-phenylpropyl]-4-hydroxyphenyl]butoxy]phenyl]ethylamino]-1-hydroxyethyl]-2-hydroxyphenyl]methanesulfonamide
Show/Hide
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C42H57N3O6S
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1
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| 1 |
EC50 = 13 nM
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CP0116358
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(R)-1-(9-(2-hydroxy-2-(8-hydroxy-2-oxo-1,2-dihydroquinolin-5-yl)ethylamino)nonyl)piperidin-4-yl biphenyl-2-ylcarbamate
Show/Hide
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C38H48N4O5
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1
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| 1 |
EC50 = 13 nM
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CP0761844
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(R)-(3'-Chloro-4'-hydroxy-biphenyl-2-yl)-carbamic acid 1-[3-(4-{2-[2-hydroxy-2-(4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-ethyl}-phenoxy)-propyl]-piperidin-4-yl ester
Show/Hide
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C38H45ClN4O8S
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1
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| 1 |
EC50 = 13 nM
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CP0065058
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8-hydroxy-5-[(1R)-1-hydroxy-2-[9-[4-[[3-[hydroxy(diphenyl)methyl]-1,2,4-triazol-1-yl]methyl]piperidin-1-yl]nonylamino]ethyl]-1H-quinolin-2-one
Show/Hide
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C41H52N6O4
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1
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| 1 |
EC50 = 13 nM
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CP0771494
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(R)-(3'-Chloro-4'-hydroxy-4-methyl-biphenyl-2-yl)-carbamic acid 1-{9-[2-hydroxy-2-(4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-nonyl}-piperidin-4-yl ester
Show/Hide
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C37H51ClN4O7S
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1
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| 1 |
EC50 = 14 nM
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CP0054748
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5-[(1R)-2-[9-[4-[[3-[(R)-cyclohexyl-hydroxy-phenylmethyl]-1,2,4-triazol-1-yl]methyl]piperidin-1-yl]nonylamino]-1-hydroxyethyl]-8-hydroxy-1H-quinolin-2-one
Show/Hide
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C41H58N6O4
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1
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| 1 |
EC50 = 14 nM
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CP0371866
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6-hydroxy-8-[1-hydroxy-2-[[1-(3-methoxyphenyl)-2-methylpropan-2-yl]amino]ethyl]-4H-1,4-benzoxazin-3-one
Show/Hide
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C21H26N2O5
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1
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| 1 |
EC50 = 14.3 nM
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CP0460724
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2-(3-((R)-2-((R)-2-(3,5-dihydroxyphenyl)-2-hydroxyethylamino)propyl)phenyl)-N-(3-(3-((R)-3-(diisopropylamino)-1-phenylpropyl)-4-hydroxyphenyl)propyl)acetamide
Show/Hide
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C43H57N3O5
|
1
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| 1 |
EC50 = 15 nM
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CP0426955
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8-[2-[[1-(4-ethoxyphenyl)-2-methylpropan-2-yl]amino]-1-hydroxyethyl]-6-hydroxy-4H-1,4-benzoxazin-3-one
Show/Hide
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C22H28N2O5
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1
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| 1 |
EC50 = 15.4 nM
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CP0461634
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[3-[(2R)-2-[[(2R)-2-[3-(benzylamino)phenyl]-2-hydroxyethyl]amino]propyl]-1H-indol-7-yl] methanesulfonate
Show/Hide
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C27H31N3O4S
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1
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| 1 |
EC50 = 16 nM
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CP0473364
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N-[3-[3-[(1R)-3-[di(propan-2-yl)amino]-1-phenylpropyl]-4-hydroxyphenyl]propyl]-2-[3-[2-[[(2R)-2-hydroxy-2-[4-hydroxy-3-(hydroxymethyl)phenyl]ethyl]amino]-2-methylpropyl]phenyl]acetamide
Show/Hide
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C45H61N3O5
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1
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| 1 |
EC50 = 17 nM
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CP0725692
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((1S,5S)-3-(9-((R)-2-hydroxy-2-(4-hydroxy-3-(methylsulfonamido)phenyl)ethylamino)nonyl)-3-azabicyclo[3.1.0]hexan-1-yl)methyl 3'-chloro-4'-hydroxybiphenyl-2-ylcarbamate
Show/Hide
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C37H49ClN4O7S
|
1
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| 1 |
EC50 = 17 nM
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CP0039168
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[3-[(2R)-2-[[(2R)-2-hydroxy-2-[3-(thiophen-2-ylsulfonylamino)phenyl]ethyl]amino]propyl]-1H-indol-7-yl] methanesulfonate
Show/Hide
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C24H27N3O6S3
|
1
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| 1 |
EC50 = 18 nM
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CP0442324
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[3-[(2R)-2-[[(2R)-2-[3-(but-2-ynylamino)phenyl]-2-hydroxyethyl]amino]propyl]-1H-indol-7-yl] methanesulfonate
Show/Hide
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C24H29N3O4S
|
1
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| 1 |
EC50 = 18 nM
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CP0075978
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2-[[3-[(2R)-2-[[(2R)-2-hydroxy-2-[3-(thiophen-2-ylsulfonylamino)phenyl]ethyl]amino]propyl]-1H-indol-7-yl]oxy]acetic acid
Show/Hide
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C25H27N3O6S2
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1
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| 1 |
EC50 = 19 nM
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CP0430587
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2-[4-[[(2R)-2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]propyl]amino]phenyl]-N-methylsulfonylacetamide
Show/Hide
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C20H26ClN3O4S
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1
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| 1 |
EC50 = 19.95 nM
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CP0853659
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2-(Hydroxymethyl)-4-((1R)-1-hydroxy-2-{[6-({4-[4-(methylsulfonyl)phenyl]butyl}oxy)hexyl]amino}ethyl)phenol acetate salt
Show/Hide
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C28H43NO8S
|
1
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| 1 |
EC50 = 19.95 nM
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CP0047480
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(S)-4-(3-hexylureido)-N-(4-(2-(1-hydroxy-2-(4-hydroxyphenoxy)ethylamino)ethyl)phenyl)benzenesulfonamide
Show/Hide
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C30H40N4O6S
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2
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| 1 |
EC50 = 20 nM
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| 2 |
IC50 = 3000 nM
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CP0478306
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1-(4-{4-[2-Hydroxy-2-(4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-piperidin-1-yl}-benzoyl)-pyrrolidine-2-carboxylic acid
Show/Hide
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C26H34N4O7S
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1
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| 1 |
EC50 = 20 nM
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CP0401690
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4-Aminomethylpiperidine substituted analogue
Show/Hide
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C31H39N5O9S2
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1
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| 1 |
EC50 = 20 nM
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CP0716118
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(R)-(3'-Chloro-4'-hydroxy-biphenyl-2-yl)-carbamic acid 1-{8-[2-hydroxy-2-(4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-octyl}-piperidin-4-yl ester
Show/Hide
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C35H47ClN4O7S
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1
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| 1 |
EC50 = 20 nM
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CP0054749
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5-[(1R)-2-[2-[4-[2-[4-[[3-[(R)-cyclohexyl-hydroxy-phenylmethyl]-1,2,4-triazol-1-yl]methyl]piperidin-1-yl]ethyl]phenyl]ethylamino]-1-hydroxyethyl]-8-hydroxy-1H-quinolin-2-one
Show/Hide
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C42H52N6O4
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1
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| 1 |
EC50 = 20.9 nM
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CP0071873
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N-[3-[(1R)-1-hydroxy-2-[[(2R)-1-(1H-indol-3-yl)propan-2-yl]amino]ethyl]phenyl]thiophene-2-sulfonamide
Show/Hide
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C23H25N3O3S2
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1
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| 1 |
EC50 = 21 nM
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CP0659243
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(R)-(3'-Chloro-4'-hydroxy-biphenyl-2-yl)-carbamic acid 1-{10-[2-hydroxy-2-(4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-decyl}-piperidin-4-yl ester
Show/Hide
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C37H51ClN4O7S
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1
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| 1 |
EC50 = 21 nM
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CP0231612
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5-[(1R)-2-[9-[4-[[3-(cyclohexyl-hydroxy-phenylmethyl)-1,2,4-triazol-1-yl]methyl]piperidin-1-yl]nonylamino]-1-hydroxyethyl]-8-hydroxy-1H-quinolin-2-one
Show/Hide
|
C41H58N6O4
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1
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| 1 |
EC50 = 21 nM
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CP0881304
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(2',5'-Difluoro-4'-hydroxy-biphenyl-2-yl)-carbamic acid 1-{(R)-9-[2-hydroxy-2-(4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-nonyl}-piperidin-4-yl ester
Show/Hide
|
C36H48F2N4O7S
|
1
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| 1 |
EC50 = 22 nM
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CP0375678
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1-(3-Chloro-phenyl)-2-[2-(1H-indol-3-yl)-1-methyl-ethylamino]-ethanol
Show/Hide
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C19H21ClN2O
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1
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| 1 |
EC50 = 23 nM
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CP0677104
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(R)-(3'-Chloro-4'-hydroxy-biphenyl-2-yl)-carbamic acid 8-{9-[2-hydroxy-2-(4-hydroxy-3-methanesulfonylaminophenyl)-ethylamino]-nonyl}-8-azabicyclo[3.2.1]oct-3-yl ester
Show/Hide
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C38H51ClN4O7S
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1
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| 1 |
EC50 = 23 nM
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CP0761843
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(R)-(3'-Chloro-5-fluoro-4'-hydroxy-biphenyl-2-yl)-carbamic acid 1-{9-[2-hydroxy-2-(4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-nonyl}-piperidin-4-yl ester
Show/Hide
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C36H48ClFN4O7S
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1
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| 1 |
EC50 = 23 nM
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CP0841972
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(R)-1-(9-((R)-2-hydroxy-2-(4-hydroxy-3-(methylsulfonamido)phenyl)ethylamino)nonyl)pyrrolidin-3-yl 3'-chloro-4'-hydroxybiphenyl-2-ylcarbamate
Show/Hide
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C35H47ClN4O7S
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1
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| 1 |
EC50 = 24 nM
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CP0198066
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(R)-1-((R)-3-Chloro-phenyl)-2-[2-(1H-indol-3-yl)-1-methyl-ethylamino]-ethanol
Show/Hide
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C19H21ClN2O
|
1
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| 1 |
EC50 = 25 nM
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CP0673932
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(R)-(3'-Fluoro-4'-hydroxy-biphenyl-2-yl)-carbamic acid 1-{9-[2-hydroxy-2-(4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-nonyl}-piperidin-4-yl ester
Show/Hide
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C36H49FN4O7S
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1
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| 1 |
EC50 = 26 nM
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CP0841971
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(R)-(4'-Hydroxy-biphenyl-2-yl)-carbamic acid 1-{9-[2-hydroxy-2-(4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-nonyl}-piperidin-4-yl ester
Show/Hide
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C36H50N4O7S
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1
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| 1 |
EC50 = 26 nM
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CP0189834
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N-[4-[4-[[[(2R)-2-hydroxy-2-[4-hydroxy-3-(methanesulfonamido)phenyl]ethyl]amino]methyl]piperidin-1-yl]sulfonylphenyl]nonanamide
Show/Hide
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C30H46N4O7S2
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1
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| 1 |
EC50 = 30 nM
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CP0318599
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2-[1-[4-[4-[[[(2R)-2-hydroxy-2-[4-hydroxy-3-(methanesulfonamido)phenyl]ethyl]amino]methyl]piperidin-1-yl]sulfonylphenyl]indol-3-yl]acetic acid
Show/Hide
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C31H36N4O8S2
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1
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| 1 |
EC50 = 30 nM
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CP0467627
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1-[(2,5-difluorophenyl)methyl]-3-[4-[4-[[[(2R)-2-hydroxy-2-[4-hydroxy-3-(methanesulfonamido)phenyl]ethyl]amino]methyl]piperidin-1-yl]sulfonylphenyl]urea
Show/Hide
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C29H35F2N5O7S2
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1
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| 1 |
EC50 = 30 nM
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CP0441102
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N-(benzenesulfonyl)-2-[4-[[(2R)-2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]propyl]amino]phenyl]acetamide
Show/Hide
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C25H28ClN3O4S
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1
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| 1 |
EC50 = 31.62 nM
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CP0875712
|
4-{(1R)-2-[(6-{4-[4-(Cyclopentylsulfonyl)phenyl]butoxy}hexyl)amino]-1-hydroxyethyl}-2-(hydroxymethyl)phenol acetate salt
Show/Hide
|
C32H49NO8S
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1
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| 1 |
EC50 = 31.62 nM
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CP0434354
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6-[4-(2-{[(2S)-2-hydroxy-3-{2'-oxo-1',2'-dihydrospiro[cyclopropane-1,3'-indole]-4'-yloxy}propyl]amino}-2-methylpropyl)phenoxy]pyridine-3-carboxamide
Show/Hide
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C29H32N4O5
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1
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| 1 |
EC50 = 35.2 nM
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CP0039161
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[3-[(2R)-2-[[(2R)-2-hydroxy-2-[3-(3-methylbut-2-enylamino)phenyl]ethyl]amino]propyl]-1H-indol-7-yl] methanesulfonate
Show/Hide
|
C25H33N3O4S
|
1
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| 1 |
EC50 = 36 nM
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CP0677100
|
(R)-(3'-Chloro-4'-hydroxy-3,5-dimethyl-biphenyl-2-yl)-carbamic acid 1-{9-[2-hydroxy-2-(4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-nonyl}-piperidin-4-yl ester
Show/Hide
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C38H53ClN4O7S
|
1
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| 1 |
EC50 = 36 nM
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CP0106025
|
(-)ISOPROTERENOL
Show/Hide
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C11H17NO3
|
2
|
| 1 |
EC50 = 39.81 nM
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| 2 |
Ki = 46 nM
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CP0853672
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4-[(1R)-2-({6-[4-(1,1-Dioxido-3,4-dihydro-2H-thiochromen-7-yl)butoxy]hexyl}amino)-1-hydroxyethyl]-2-(hydroxymethyl)phenol formate salt
Show/Hide
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C29H43NO8S
|
1
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| 1 |
EC50 = 39.81 nM
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CP0135421
|
(4-{4-[2-Hydroxy-2-(4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-piperidin-1-yl}-benzoylamino)-acetic acid
Show/Hide
|
C23H30N4O7S
|
1
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| 1 |
EC50 = 40 nM
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CP0688667
|
((1R,6R)-3-(9-((R)-2-hydroxy-2-(4-hydroxy-3-(methylsulfonamido)phenyl)ethylamino)nonyl)-3-azabicyclo[3.1.0]hexan-6-yl)methyl 3'-chloro-4'-hydroxybiphenyl-2-ylcarbamate
Show/Hide
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C37H49ClN4O7S
|
1
|
| 1 |
EC50 = 42 nM
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CP0492962
|
[3-[(2R)-2-[[(2R)-2-hydroxy-2-(3-phenylmethoxyphenyl)ethyl]amino]propyl]-1H-indol-7-yl] methanesulfonate
Show/Hide
|
C27H30N2O5S
|
1
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| 1 |
EC50 = 46 nM
|
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CP0371869
|
8-[2-[[1-(4-ethylphenyl)-2-methylpropan-2-yl]amino]-1-hydroxyethyl]-6-hydroxy-4H-1,4-benzoxazin-3-one
Show/Hide
|
C22H28N2O4
|
1
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| 1 |
EC50 = 49.7 nM
|
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CP0382237
|
2-[4-[[(2R)-2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]propyl]amino]phenyl]acetic acid
Show/Hide
|
C19H23ClN2O3
|
1
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| 1 |
EC50 = 50.12 nM
|
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CP0386623
|
sodium;2-[4-[(2R)-2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]propyl]phenoxy]acetate
Show/Hide
|
C19H21ClNO4-
|
1
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| 1 |
EC50 = 50.12 nM
|
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CP0455408
|
2-[3-[[(2R)-2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]propyl]amino]phenyl]acetic acid
Show/Hide
|
C19H23ClN2O3
|
1
|
| 1 |
EC50 = 50.12 nM
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CP0457574
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2-[4-[[(2R)-2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]propyl]amino]phenyl]-1,3-thiazole-4-carboxylic acid
Show/Hide
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C21H22ClN3O3S
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1
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| 1 |
EC50 = 50.12 nM
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CP0464671
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4-[4-[[(2R)-2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]propyl]amino]phenyl]-1,3-thiazole-2-carboxylic acid
Show/Hide
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C21H22ClN3O3S
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1
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| 1 |
EC50 = 50.12 nM
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CP0466916
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3-[3-[[(2R)-2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]propyl]amino]phenyl]benzoic acid
Show/Hide
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C24H25ClN2O3
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1
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| 1 |
EC50 = 50.12 nM
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CP0677102
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(R)-(3'-Chloro-4-fluoro-4'-hydroxy-biphenyl-2-yl)-carbamic acid 1-{9-[2-hydroxy-2-(4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-nonyl}-piperidin-4-yl ester
Show/Hide
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C36H48ClFN4O7S
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1
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| 1 |
EC50 = 57 nM
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CP0371925
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6-hydroxy-8-[1-hydroxy-2-[[2-methyl-1-(4-propan-2-ylphenyl)propan-2-yl]amino]ethyl]-4H-1,4-benzoxazin-3-one
Show/Hide
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C23H30N2O4
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1
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| 1 |
EC50 = 58 nM
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CP0213665
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3-[N-butyl-4-[4-[[(2R)-2-hydroxy-2-[4-hydroxy-3-(methanesulfonamido)phenyl]ethyl]amino]piperidin-1-yl]anilino]-3-oxopropanoic acid
Show/Hide
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C27H38N4O7S
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1
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| 1 |
EC50 = 60 nM
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CP0463273
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1-[4-(4-{[2-Hydroxy-2-(4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-methyl}-piperidine-1-sulfonyl)-phenyl]-1H-indole-4-carboxylic acid
Show/Hide
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C30H34N4O8S2
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1
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| 1 |
EC50 = 60 nM
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CP0467150
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4-[3-(2-{(R)-(R)-2-Hydroxy-2-[3-(thiophene-2-sulfonylamino)-phenyl]-ethylamino}-propyl)-1H-indol-7-yloxysulfonyl]-benzoic acid
Show/Hide
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C30H29N3O8S3
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1
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| 1 |
EC50 = 60 nM
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CP0688665
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(R)-(5'-Fluoro-3'-hydroxy-biphenyl-2-yl)-carbamic acid 1-{9-[2-hydroxy-2-(4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-nonyl}-piperidin-4-yl ester
Show/Hide
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C36H49FN4O7S
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1
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| 1 |
EC50 = 65 nM
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CP0371924
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6-hydroxy-8-[1-hydroxy-2-[[2-methyl-1-(4-phenylphenyl)propan-2-yl]amino]ethyl]-4H-1,4-benzoxazin-3-one
Show/Hide
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C26H28N2O4
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1
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| 1 |
EC50 = 68 nM
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CP0429984
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[3-[(2R)-2-[[(2R)-2-(3-benzamidophenyl)-2-hydroxyethyl]amino]propyl]-1H-indol-7-yl] methanesulfonate
Show/Hide
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C27H29N3O5S
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1
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| 1 |
EC50 = 69 nM
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CP0903933
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(R)-Biphenyl-2-yl-carbamic acid 1-{9-[2-hydroxy-2-(4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-nonyl}-piperidin-4-yl ester
Show/Hide
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C36H50N4O6S
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1
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| 1 |
EC50 = 74 nM
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CP0378418
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2-[4-[[(2R)-2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]propyl]amino]phenyl]-N-(4-methylphenyl)sulfonylacetamide
Show/Hide
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C26H30ClN3O4S
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1
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| 1 |
EC50 = 79.43 nM
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CP0382240
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2-[4-[[(2R)-2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]propyl]amino]phenyl]furan-3-carboxylic acid
Show/Hide
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C22H23ClN2O4
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1
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| 1 |
EC50 = 79.43 nM
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CP0208046
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2-(4-{4-[2-Hydroxy-2-(4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-piperidin-1-yl}-benzoylamino)-4-methyl-pentanoic acid
Show/Hide
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C27H38N4O7S
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1
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| 1 |
EC50 = 80 nM
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CP0691421
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(2'-Hydroxy-biphenyl-2-yl)-carbamic acid 1-{(R)-9-[2-hydroxy-2-(4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-nonyl}-piperidin-4-yl ester
Show/Hide
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C36H50N4O7S
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1
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| 1 |
EC50 = 90 nM
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CP0371923
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(S)-6-hydroxy-8-(1-hydroxy-2-(1-(4-methoxyphenyl)-2-methylpropan-2-ylamino)ethyl)-2H-benzo[b][1,4]oxazin-3(4H)-one
Show/Hide
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C21H26N2O5
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1
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| 1 |
EC50 = 97.7 nM
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CP0382239
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4-[3-[[(2R)-2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]propyl]amino]phenyl]-1,3-thiazole-2-carboxylic acid
Show/Hide
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C21H22ClN3O3S
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1
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| 1 |
EC50 = 100 nM
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CP0464672
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2-[4-[[(2R)-2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]propyl]amino]phenyl]-1,3-oxazole-4-carboxylic acid
Show/Hide
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C21H22ClN3O4
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1
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| 1 |
EC50 = 100 nM
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CP0754218
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(3',5'-Difluoro-2'-hydroxy-biphenyl-2-yl)-carbamic acid 1-{(R)-9-[2-hydroxy-2-(4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-nonyl}-piperidin-4-yl ester
Show/Hide
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C36H48F2N4O7S
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1
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| 1 |
EC50 = 102 nM
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CP0373204
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N-[3-[3-[(1R)-3-[di(propan-2-yl)amino]-1-phenylpropyl]-4-hydroxyphenyl]propyl]-11-[[(2R)-2-hydroxy-2-[4-hydroxy-3-(methanesulfonamido)phenyl]ethyl]amino]undecanamide
Show/Hide
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C44H68N4O6S
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1
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| 1 |
EC50 = 116 nM
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CP0174576
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8-hydroxy-5-[(1R)-1-hydroxy-2-[2-[4-[2-[4-[[3-[hydroxy(diphenyl)methyl]-1,2,4-triazol-1-yl]methyl]piperidin-1-yl]ethyl]phenyl]ethylamino]ethyl]-1H-quinolin-2-one
Show/Hide
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C42H46N6O4
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1
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| 1 |
EC50 = 116 nM
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CP0382242
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2-[3-[[(2R)-2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]propyl]amino]phenyl]-1,3-oxazole-4-carboxylic acid
Show/Hide
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C21H22ClN3O4
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1
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| 1 |
EC50 = 125.89 nM
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CP0399444
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2-[3-[[(2R)-2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]propyl]amino]phenyl]furan-3-carboxylic acid
Show/Hide
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C22H23ClN2O4
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1
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| 1 |
EC50 = 125.89 nM
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CP0473365
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2-((R)-3-(diisopropylamino)-1-phenylpropyl)-4-(4-(4-(2-((R)-2-hydroxy-2-(4-hydroxy-3-(hydroxymethyl)phenyl)ethylamino)ethyl)phenoxy)butyl)phenol
Show/Hide
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C42H56N2O5
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1
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| 1 |
EC50 = 129 nM
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CP0691423
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(R)-(3'-Hydroxy-biphenyl-2-yl)-carbamic acid 1-{9-[2-hydroxy-2-(4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-nonyl}-piperidin-4-yl ester
Show/Hide
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C36H50N4O7S
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1
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| 1 |
EC50 = 129 nM
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CP0457573
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2-[3-[[(2R)-2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]propyl]amino]phenyl]-1,3-thiazole-4-carboxylic acid
Show/Hide
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C21H22ClN3O3S
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1
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| 1 |
EC50 = 158.49 nM
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CP0460723
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4-((R)-2-(4-(4-(3-((R)-3-(diisopropylamino)-1-phenylpropyl)-4-hydroxyphenyl)butoxy)phenethylamino)-1-hydroxyethyl)benzene-1,2-diol
Show/Hide
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C41H54N2O5
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1
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| 1 |
EC50 = 173 nM
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CP0673933
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(R)-(3'-Chloro-4'-hydroxy-biphenyl-2-yl)-carbamic acid 1-{11-[2-hydroxy-2-(4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-undecyl}-piperidin-4-yl ester
Show/Hide
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C38H53ClN4O7S
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1
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| 1 |
EC50 = 195 nM
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CP0449854
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1-(benzenesulfonyl)-3-[[3-[[(2R)-2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]propyl]amino]phenyl]methyl]urea
Show/Hide
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C25H29ClN4O4S
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1
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| 1 |
EC50 = 251.19 nM
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CP0460647
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4-{4-[2-Hydroxy-2-(4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-piperidin-1-yl}-benzamide
Show/Hide
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C21H28N4O5S
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1
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| 1 |
EC50 = 270 nM
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CP0071877
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(+/-)-2-(4-((R)-2-((R)-2-(3-chlorophenyl)-2-hydroxyethylamino)propyl)phenoxy)acetic acid
Show/Hide
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C19H22ClNO4
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4
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| 1 |
EC50 = 290 nM
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| 2 |
IC50 = 3000 nM
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| 3 |
Ki = 630 nM
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| 4 |
Ki = 2850 nM
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CP0877319
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4'-(2-{[(2R)-2-(6-Aminopyridin-3-yl)-2-hydroxyethyl]amino}ethyl)-3-(cyclohexyloxy)-N-(methylsulfonyl)biphenyl-4-carboxamide Dihydrochloride
Show/Hide
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C29H38Cl2N4O5S
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1
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| 1 |
EC50 = 290 nM
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CP0374848
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N-[2-[4-[[(2R)-2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]propyl]amino]phenyl]ethylsulfonyl]benzamide
Show/Hide
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C26H30ClN3O4S
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1
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| 1 |
EC50 = 316.23 nM
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CP0449742
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5-[3-[[(2R)-2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]propyl]amino]phenyl]-1,3-oxazole-4-carboxylic acid
Show/Hide
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C21H22ClN3O4
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1
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| 1 |
EC50 = 316.23 nM
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CP0039165
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(S)-1-((R)-3-Chloro-phenyl)-2-[2-(1H-indol-3-yl)-1-methyl-ethylamino]-ethanol
Show/Hide
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C19H21ClN2O
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1
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| 1 |
EC50 = 330 nM
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CP0382238
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3-[4-[[(2R)-2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]propyl]amino]phenyl]propanoic acid
Show/Hide
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C20H25ClN2O3
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1
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| 1 |
EC50 = 398.11 nM
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CP0457575
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5-[4-[[(2R)-2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]propyl]amino]phenyl]-1,3-oxazole-4-carboxylic acid
Show/Hide
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C21H22ClN3O4
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1
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| 1 |
EC50 = 398.11 nM
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CP0399929
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1-[(2,5-difluorophenyl)methyl]-3-[4-[4-[[[(2S)-2-hydroxy-3-[4-hydroxy-3-(methanesulfonamido)phenoxy]propyl]amino]methyl]piperidin-1-yl]sulfonylphenyl]urea
Show/Hide
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C30H37F2N5O8S2
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1
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| 1 |
EC50 = 454 nM
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CP0386625
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methyl 3-[3-[2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]ethylamino]phenyl]benzoate
Show/Hide
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C24H25ClN2O3
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1
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| 1 |
EC50 = 501.19 nM
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CP0495955
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(R)-4'-(2-(2-hydroxy-2-phenylethylamino)ethyl)-3-(isopropylamino)biphenyl-4-carboxylic acid
Show/Hide
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C26H30N2O3
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1
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| 1 |
EC50 = 586 nM
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CP0857860
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N-[5-(2-{1-[4-((R)-2,4-Dioxo-thiazolidin-5-ylmethyl)-phenyl]-piperidin-4-ylamino}-1-hydroxy-ethyl)-2-hydroxy-phenyl]-benzenesulfonamide
Show/Hide
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C29H32N4O6S2
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1
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| 1 |
EC50 = 620 nM
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CP0382241
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2-[4-[[(2R)-2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]propyl]amino]phenyl]thiophene-3-carboxylic acid
Show/Hide
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C22H23ClN2O3S
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1
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| 1 |
EC50 = 630.96 nM
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CP0386624
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3-[3-[2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]ethylamino]phenyl]-4-methylbenzoic acid
Show/Hide
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C24H25ClN2O3
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1
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| 1 |
EC50 = 630.96 nM
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CP0375236
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1-[4-(4-{[(S)-2-Hydroxy-3-(8-hydroxy-2-oxo-1,2,3,4-tetrahydro-quinolin-5-yloxy)-propylamino]-methyl}-piperidine-1-sulfonyl)-phenyl]-3-octyl-urea
Show/Hide
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C33H49N5O7S
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1
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| 1 |
EC50 = 680 nM
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CP0440993
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2-[3-[[(2R)-2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]propyl]amino]phenyl]thiophene-3-carboxylic acid
Show/Hide
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C22H23ClN2O3S
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1
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| 1 |
EC50 = 794.33 nM
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CP0437478
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3-[4-[4-[[(2R)-2-hydroxy-2-[4-hydroxy-3-(methanesulfonamido)phenyl]ethyl]amino]piperidin-1-yl]anilino]-3-oxopropanoic acid
Show/Hide
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C23H30N4O7S
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1
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| 1 |
EC50 = 900 nM
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CP0036332
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4-{(R)-2-[1-(4-Butoxy-benzenesulfonyl)-azetidin-3-ylamino]-1-hydroxy-ethyl}-phenol
Show/Hide
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C21H28N2O5S
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1
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| 1 |
EC50 = 920 nM
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CP0166797
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1-hexyl-3-[4-[4-[[(2R)-2-hydroxy-2-[4-hydroxy-3-(methanesulfonamido)phenyl]ethyl]amino]piperidin-1-yl]sulfonylphenyl]urea
Show/Hide
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C27H41N5O7S2
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1
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| 1 |
EC50 = 920 nM
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CP0371725
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N-[2-[3-[[(2R)-2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]propyl]amino]phenyl]ethylsulfonyl]benzenesulfonamide
Show/Hide
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C25H30ClN3O5S2
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1
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| 1 |
EC50 = 1000 nM
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CP0463635
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4-Aminomethylpiperidine substituted analogue
Show/Hide
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C28H40N4O7S
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1
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| 1 |
EC50 = 1000 nM
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CP0483335
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2-[3-[[(2R)-2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]propyl]amino]phenyl]benzoic acid
Show/Hide
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C24H25ClN2O3
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1
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| 1 |
EC50 = 1000 nM
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CP0443504
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(R)-4'-(2-(2-(4-aminopyridin-3-yl)-2-hydroxyethylamino)ethyl)-3-(cyclohexyloxy)biphenyl-4-carboxylic acid
Show/Hide
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C28H33N3O4
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1
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| 1 |
EC50 = 1100 nM
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CP0418058
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4-(2-{[(2R)-2-(6-Amino-3-pyridinyl)-2-hydroxyethyl]amino}ethyl)-3-(cyclohexyloxy)-4-biphenylcarboxylic acid
Show/Hide
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C28H33N3O4
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1
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| 1 |
EC50 = 1100 nM
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CP0889313
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N-[5-(2-{1-[4-((R)-2,4-Dioxo-thiazolidin-5-ylmethyl)-phenyl]-piperidin-4-ylamino}-1-hydroxy-ethyl)-2-hydroxy-phenyl]-methanesulfonamide
Show/Hide
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C24H30N4O6S2
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1
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| 1 |
EC50 = 1190 nM
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CP0443398
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4'-[2-[[(2R)-2-(6-Amino-3-pyridinyl)-2-hydroxyethyl]amino]ethyl]-3-(isopropylthio)-N-(methylsulfonyl)-4-biphenylcarboxamide
Show/Hide
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C26H32N4O4S2
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1
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| 1 |
EC50 = 1200 nM
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CP0403282
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Solabegron
Show/Hide
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C23H23ClN2O3
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1
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| 1 |
EC50 = 1258.93 nM
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CP0393191
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N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-[4-[4-(trifluoromethoxy)phenyl]-1,3-thiazol-2-yl]benzenesulfonamide
Show/Hide
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C31H27F3N4O4S2
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2
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| 1 |
EC50 = 1400 nM
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| 2 |
IC50 = 1200 nM
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CP0136837
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2-(4-{4-[2-Hydroxy-2-(4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-piperidin-1-yl}-benzoylamino)-3-phenyl-propionic acid
Show/Hide
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C30H36N4O7S
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1
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| 1 |
EC50 = 1500 nM
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CP0441823
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2-[3-[[(2R)-2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]propyl]amino]phenyl]pyridine-3-carboxylic acid
Show/Hide
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C23H24ClN3O3
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1
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| 1 |
EC50 = 1584.89 nM
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CP0451649
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4-[3-[[(2R)-2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]propyl]amino]phenyl]benzoic acid
Show/Hide
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C24H25ClN2O3
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1
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| 1 |
EC50 = 1584.89 nM
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CP0377642
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4-[4-(3,4-Difluoro-phenyl)-thiazol-2-yl]-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
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C30H26F2N4O3S2
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2
|
| 1 |
EC50 = 1800 nM
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| 2 |
IC50 = 1700 nM
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CP0156740
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(R)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)-4-(4-(4-(trifluoromethyl)phenyl)thiazol-2-yl)benzenesulfonamide
Show/Hide
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C31H27F3N4O3S2
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2
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| 1 |
EC50 = 2400 nM
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| 2 |
IC50 = 2300 nM
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CP0457572
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2-[3-[2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]ethylamino]phenyl]furan-3-carboxylic acid
Show/Hide
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C21H21ClN2O4
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1
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| 1 |
EC50 = 2511.89 nM
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CP0853349
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4-[(1R)-1-Hydroxy-2-({6-[(2-hydroxyethyl)oxy]hexyl}amino)-ethyl]-2-(hydroxymethyl)phenol Acetate Salt
Show/Hide
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C19H33NO7
|
1
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| 1 |
EC50 = 2511.89 nM
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CP0401348
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4-[[(2R)-2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]propyl]amino]benzoic acid
Show/Hide
|
C18H21ClN2O3
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1
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| 1 |
EC50 = 3162.28 nM
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CP0438096
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(4-{4-[2-Hydroxy-2-(4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-piperidin-1-yl}-benzoylamino)-acetic acid ethyl ester
Show/Hide
|
C25H34N4O7S
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1
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| 1 |
EC50 = 3200 nM
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CP0474560
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(R)-4'-(2-(2-(4-aminopyridin-3-yl)-2-hydroxyethylamino)ethyl)-3-isobutylbiphenyl-4-carboxylic acid
Show/Hide
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C26H31N3O3
|
1
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| 1 |
EC50 = 3200 nM
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CP0375138
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4-(2-{[(2R)-2-(6-Amino-3-pyridinyl)-2-hydroxyethyl]amino}ethyl)-3-isobutyl-4-biphenylcarboxylic acid
Show/Hide
|
C26H31N3O3
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1
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| 1 |
EC50 = 3200 nM
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CP0420505
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5-[3-[2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]ethylamino]phenyl]pyridine-3-carboxylic acid
Show/Hide
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C22H22ClN3O3
|
1
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| 1 |
EC50 = 3981.07 nM
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CP0420451
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3-(4-{4-[2-Hydroxy-2-(4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-piperidin-1-yl}-phenyl)-propionic acid
Show/Hide
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C23H31N3O6S
|
1
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| 1 |
EC50 = 4700 nM
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CP0448512
|
2-[butyl-[4-[4-[[(2R)-2-hydroxy-2-[4-hydroxy-3-(methanesulfonamido)phenyl]ethyl]amino]piperidin-1-yl]phenyl]sulfamoyl]acetic acid
Show/Hide
|
C26H38N4O8S2
|
1
|
| 1 |
EC50 = 5000 nM
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CP0440991
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2-[3-[2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]ethylamino]phenyl]thiophene-3-carboxylic acid
Show/Hide
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C21H21ClN2O3S
|
1
|
| 1 |
EC50 = 5011.87 nM
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CP0430852
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8-[2-[[1-(4-tert-butylphenyl)-2-methylpropan-2-yl]amino]-1-hydroxyethyl]-6-hydroxy-4H-1,4-benzoxazin-3-one
Show/Hide
|
C24H32N2O4
|
1
|
| 1 |
EC50 = 5167 nM
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CP0422142
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(4-{4-[2-Hydroxy-2-(4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-piperidin-1-yl}-benzyloxy)-acetic acid
Show/Hide
|
C23H31N3O7S
|
1
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| 1 |
EC50 = 6000 nM
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CP0345975
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2-(4-{4-[2-Hydroxy-2-(4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-piperidin-1-yl}-benzoylamino)-3-methyl-butyric acid
Show/Hide
|
C26H36N4O7S
|
1
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| 1 |
EC50 > 10000 nM
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CP0845050
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4'-(2-{[(2R)-2-Hydroxy-2-phenylethyl]amino}ethyl)-3-(isopropylamino)-N-(methylsulfonyl)biphenyl-4-carboxamide Dihydrochloride
Show/Hide
|
C27H35Cl2N3O4S
|
1
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| 1 |
EC50 > 10000 nM
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CP0845051
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4'-(2-{[(2R)-2-Hydroxy-2-phenylethyl]amino}ethyl)-3-(isopropylsulfanyl)-N-(methylsulfonyl)biphenyl-4-carboxamide Hydrochloride
Show/Hide
|
C27H33ClN2O4S2
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1
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| 1 |
EC50 > 10000 nM
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CP0851070
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3-(Cyclohexylamino)-4'-(2-{[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino}ethyl)-N-(methylsulfonyl)biphenyl-4-carboxamide Trihydrochloride
Show/Hide
|
C29H39Cl3N4O4S
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1
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| 1 |
EC50 > 10000 nM
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CP0882007
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4'-(2-{[(2R)-2-Hydroxy-2-phenylethyl]amino}ethyl)-3-isobutyl-N-(methylsulfonyl)biphenyl-4-carboxamide Hydrochloride
Show/Hide
|
C28H35ClN2O4S
|
1
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| 1 |
EC50 > 10000 nM
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CP0900959
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3-(Cyclohexyloxy)-4'-(2-{[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino}ethyl)-N-(methylsulfonyl)biphenyl-4-carboxamide Dihydrochloride
Show/Hide
|
C29H37Cl2N3O5S
|
1
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| 1 |
EC50 > 10000 nM
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CP0409159
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(S)-6-(4-(2-(3-(3-ethyl-2-oxo-2,3-dihydro-1H-benzo[d]imidazol-4-yloxy)-2-hydroxypropylamino)-2-methylpropyl)phenoxy)nicotinamide
Show/Hide
|
C28H33N5O5
|
1
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| 1 |
EC50 > 10000 nM
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CP0409669
|
(S)-6-(4-(2-(3-(3-(2-cyclobutylethyl)-2-oxo-2,3-dihydro-1H-benzo[d]imidazol-4-yloxy)-2-hydroxypropylamino)-2-methylpropyl)phenoxy)nicotinamide
Show/Hide
|
C32H39N5O5
|
1
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| 1 |
EC50 > 10000 nM
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|
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CP0419619
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(S)-6-(4-(2-(2-hydroxy-3-(2-oxo-3-propyl-2,3-dihydro-1H-benzo[d]imidazol-4-yloxy)propylamino)-2-methylpropyl)phenoxy)nicotinamide
Show/Hide
|
C29H35N5O5
|
1
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| 1 |
EC50 > 10000 nM
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CP0424777
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(S)-6-(4-(2-(3-(3-(2-cyclopropylethyl)-2-oxo-2,3-dihydro-1H-benzo[d]imidazol-4-yloxy)-2-hydroxypropylamino)-2-methylpropyl)phenoxy)nicotinamide
Show/Hide
|
C31H37N5O5
|
1
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| 1 |
EC50 > 10000 nM
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|
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CP0437372
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(S)-6-(4-(2-(2-hydroxy-3-(3-methyl-2-oxo-2,3-dihydro-1H-benzo[d]imidazol-4-yloxy)propylamino)-2-methylpropyl)phenoxy)nicotinamide
Show/Hide
|
C27H31N5O5
|
1
|
| 1 |
EC50 > 10000 nM
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|
|
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CP0371753
|
6-(4-(2-((S)-3-(3-benzyl-2-oxoindolin-4-yloxy)-2-hydroxypropylamino)-2-methylpropyl)phenoxy)nicotinamide
Show/Hide
|
C34H36N4O5
|
1
|
| 1 |
EC50 > 10000 nM
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|
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CP0371757
|
6-[4-(2-{[(2S)-2-hydroxy-3-{2'-oxo-1',2'-dihydrospiro[cyclohexane-1,3'-indole]-4'-yloxy}propyl]amino}-2-methylpropyl)phenoxy]pyridine-3-carboxamide
Show/Hide
|
C32H38N4O5
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
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CP0371758
|
(S)-6-(4-(2-(2-hydroxy-3-(2-oxoindolin-4-yloxy)propylamino)-2-methylpropyl)phenoxy)nicotinamide
Show/Hide
|
C27H30N4O5
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
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CP0417209
|
6-(4-(2-((S)-2-hydroxy-3-(3-methyl-2-oxoindolin-4-yloxy)propylamino)-2-methylpropyl)phenoxy)nicotinamide
Show/Hide
|
C28H32N4O5
|
1
|
| 1 |
EC50 > 10000 nM
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|
|
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CP0424778
|
6-(4-(2-((S)-2-hydroxy-3-(3-isopropyl-2-oxoindolin-4-yloxy)propylamino)-2-methylpropyl)phenoxy)nicotinamide
Show/Hide
|
C30H36N4O5
|
1
|
| 1 |
EC50 > 10000 nM
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|
|
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CP0424781
|
(S)-6-(4-(2-(3-(3,3-dibenzyl-2-oxoindolin-4-yloxy)-2-hydroxypropylamino)-2-methylpropyl)phenoxy)nicotinamide
Show/Hide
|
C41H42N4O5
|
1
|
| 1 |
EC50 > 10000 nM
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|
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CP0434351
|
6-[4-(2-{[(2S)-2-hydroxy-3-{2'-oxo-1',2'-dihydrospiro[cyclopentane-1,3'-indole]-4'-yloxy}propyl]amino}-2-methylpropyl)phenoxy]pyridine-3-carboxamide
Show/Hide
|
C31H36N4O5
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0434352
|
6-[4-(2-{[(2S)-2-hydroxy-3-{2'-oxo-1',2'-dihydrospiro[cyclobutane-1,3'-indole]-4'-yloxy}propyl]amino}-2-methylpropyl)phenoxy]pyridine-3-carboxamide
Show/Hide
|
C30H34N4O5
|
1
|
| 1 |
EC50 > 10000 nM
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|
|
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CP0436369
|
6-(4-(2-((S)-2-hydroxy-3-(3-isobutyl-2-oxoindolin-4-yloxy)propylamino)-2-methylpropyl)phenoxy)nicotinamide
Show/Hide
|
C31H38N4O5
|
1
|
| 1 |
EC50 > 10000 nM
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|
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CP0458653
|
(S)-6-(4-(2-(3-(3,3-diethyl-2-oxoindolin-4-yloxy)-2-hydroxypropylamino)-2-methylpropyl)phenoxy)nicotinamide
Show/Hide
|
C31H38N4O5
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
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CP0458654
|
(S)-6-(4-(2-(3-(3,3-dimethyl-2-oxoindolin-4-yloxy)-2-hydroxypropylamino)-2-methylpropyl)phenoxy)nicotinamide
Show/Hide
|
C29H34N4O5
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
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CP0288880
|
ethyl 2-[[(6S)-6-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]-6,7,8,9-tetrahydro-5H-benzo[7]annulen-3-yl]oxy]acetate
Show/Hide
|
C23H28ClNO4
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
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CP0373035
|
4'-{2-[(R)-2-(3-Chloro-phenyl)-2-hydroxy-ethylamino]-ethyl}-biphenyl-4-carboxylic acid
Show/Hide
|
C23H22ClNO3
|
2
|
| 1 |
EC50 > 10000 nM
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|
|
| 2 |
EC50 > 1000 nM
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CP0500725
|
4-[4-[2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]ethyl]phenyl]-3-methylbenzoic acid
Show/Hide
|
C24H24ClNO3
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
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CP0456857
|
6-[3-[2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]ethylamino]phenyl]pyridine-2-carboxylic acid
Show/Hide
|
C22H22ClN3O3
|
1
|
| 1 |
EC50 = 10000 nM
|
|
|
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CP0217241
|
4'-(2-((1R,2S)-1-hydroxy-1-(4-hydroxyphenyl)propan-2-ylamino)ethyl)-3-isopropoxy-N-(methylsulfonyl)biphenyl-4-carboxamide
Show/Hide
|
C28H34N2O6S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0514692
|
3-(cyclohexyloxy)-4'-(2-((1R,2S)-1-hydroxy-1-(4-hydroxyphenyl)propan-2-ylamino)ethyl)-N-(methylsulfonyl)biphenyl-4-carboxamide
Show/Hide
|
C31H38N2O6S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
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CP0423025
|
2-((S)-7-((R)-2-(3-chlorophenyl)-2-hydroxyethylamino)-5,6,7,8-tetrahydronaphthalen-2-yloxy)acetic acid
Show/Hide
|
C20H22ClNO4
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
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CP0037154
|
(R)-4'-(2-(2-(3-chlorophenyl)-2-hydroxyethylamino)ethyl)-3-isopropoxybiphenyl-4-carboxylic acid
Show/Hide
|
C26H28ClNO4
|
2
|
| 1 |
EC50 > 10000 nM
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|
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| 2 |
EC50 > 1000 nM
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CP0137177
|
(R)-4'-(2-(2-hydroxy-2-phenylethylamino)ethyl)-3-isopropoxybiphenyl-4-carboxylic acid
Show/Hide
|
C26H29NO4
|
2
|
| 1 |
EC50 > 10000 nM
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|
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| 2 |
EC50 > 1000 nM
|
|
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CP0375139
|
(R)-4'-(2-(2-hydroxy-2-phenylethylamino)ethyl)-3-isobutylbiphenyl-4-carboxylic acid
Show/Hide
|
C27H31NO3
|
2
|
| 1 |
EC50 > 10000 nM
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|
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| 2 |
EC50 > 1000 nM
|
|
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CP0389986
|
4-((2R)-2-{[(2R)-2-Hydroxy-2-phenylethyl]amino}propyl)-3-isopropoxy-4-biphenylcarboxylic acid
Show/Hide
|
C27H31NO4
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0399297
|
(R)-4'-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)-3-isopropoxybiphenyl-4-carboxylic acid
Show/Hide
|
C25H28N2O4
|
2
|
| 1 |
EC50 > 10000 nM
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|
|
| 2 |
EC50 > 1000 nM
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|
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CP0418057
|
4-(2-{[(2R)-2-(6-Amino-3-pyridinyl)-2-hydroxyethyl]amino}ethyl)-3-isopropoxy-4-biphenylcarboxylic acid
Show/Hide
|
C25H29N3O4
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
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CP0418059
|
(R)-3-(cyclohexyloxy)-4'-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)biphenyl-4-carboxylic acid
Show/Hide
|
C28H32N2O4
|
2
|
| 1 |
EC50 > 10000 nM
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|
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| 2 |
EC50 > 1000 nM
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|
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CP0474707
|
4-(2-{[(1S,2R)-2-Hydroxy-1-methyl-2-phenylethyl]amino}ethyl)-3-propoxy-4-biphenylcarboxylic acid
Show/Hide
|
C27H31NO4
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0484975
|
4-(2-{[(1S,2R)-2-Hydroxy-1-methyl-2-phenylethyl]amino}ethyl)-3-isopropoxy-4-biphenylcarboxylic acid
Show/Hide
|
C27H31NO4
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
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CP0059008
|
N-[3-[(1R)-1-hydroxy-2-[2-[(3-methyl-2H-indazol-6-yl)oxy]ethylamino]ethyl]phenyl]methanesulfonamide
Show/Hide
|
C19H24N4O4S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0155749
|
N-[3-[(1R)-1-hydroxy-2-[2-[(3-propan-2-yl-2H-indazol-6-yl)oxy]ethylamino]ethyl]phenyl]methanesulfonamide
Show/Hide
|
C21H28N4O4S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
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CP0382114
|
N-[3-[(1R)-2-[2-[(3-cyclopropyl-2H-indazol-6-yl)oxy]ethylamino]-1-hydroxyethyl]phenyl]methanesulfonamide
Show/Hide
|
C21H26N4O4S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0382115
|
N-[3-[(1R)-2-[2-[(3-ethyl-2H-indazol-6-yl)oxy]ethylamino]-1-hydroxyethyl]phenyl]methanesulfonamide
Show/Hide
|
C20H26N4O4S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0085893
|
N-[3-[(1R)-1-hydroxy-2-[2-[(3-methyl-2H-indazol-6-yl)oxy]ethylamino]ethyl]phenyl]cyclobutanesulfonamide
Show/Hide
|
C22H28N4O4S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0216696
|
N-[3-[(1R)-1-hydroxy-2-[2-[(3-methyl-2H-indazol-6-yl)oxy]ethylamino]ethyl]phenyl]benzenesulfonamide
Show/Hide
|
C24H26N4O4S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0454822
|
2-[butyl-[4-[4-[[(2R)-2-hydroxy-2-[4-hydroxy-3-(methanesulfonamido)phenyl]ethyl]amino]piperidin-1-yl]benzoyl]amino]acetic acid
Show/Hide
|
C27H38N4O7S
|
1
|
| 1 |
EC50 = 10500 nM
|
|
|
|
CP0432795
|
4-Aminomethylpiperidine substituted analogue
Show/Hide
|
C31H38N4O7S
|
1
|
| 1 |
EC50 = 20000 nM
|
|
|
|
CP0850325
|
3-{6-[4-({(2R)-2-Hydroxy-2-[4-hydroxy-3-(hydroxymethyl)-phenyl]ethyl}amino)butoxy]hexyl}benzenesulfonamide acetate salt
Show/Hide
|
C27H42N2O8S
|
1
|
| 1 |
EC50 = 25118.86 nM
|
|
|
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CP0460947
|
4-{4-[2-Hydroxy-2-(4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-piperidin-1-yl}-benzoic acid
Show/Hide
|
C21H27N3O6S
|
1
|
| 1 |
EC50 > 50000 nM
|
|
|
|
CP0372199
|
(S)-4'-{2-[(2-Hydroxy-3-phenoxypropyl)amino]ethyl}-2-(1H-imidazol-2-yl)acetanilide
Show/Hide
|
C22H26N4O3
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0372204
|
(S)-4'-(2-{[2-Hydroxy-3-phenoxypropyl]amino}ethyl)-2-(4,6-dimethyl-2-pyridyl)-acetanilide
Show/Hide
|
C26H31N3O3
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0372205
|
(S)-N-Propyl-4'-{2-[(2-hydroxy-3-phenoxypropyl)-amino]ethyl}-2-(1-benzylimidazol-2-yl)acetanilide
Show/Hide
|
C32H38N4O3
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0372410
|
(S)-4'-(2-{[2-Hydroxy-3-(4-methylsulfonamidophenoxy)-propyl]amino}ethyl)-2-(2-pyridyl)acetanilide
Show/Hide
|
C25H30N4O5S
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0372411
|
(S)-4'-{2-[(2-Hydroxy-3-phenoxypropyl)amino]ethyl}-2-(1-benzylimidazol-2-yl)-acetanilide
Show/Hide
|
C29H32N4O3
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0372412
|
(S)-4'-(2-{[2-Hydroxy-3-phenoxypropyl]amino}ethyl)-2-(1-benzyl-benzimidazol-2-yl)-acetanilide
Show/Hide
|
C33H34N4O3
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0372413
|
(S)-4'-(2-{[2-Hydroxy-3-(4-hydroxyphenoxy)propyl]amino}ethyl)-2-(2-pyridyl)acetanilide
Show/Hide
|
C24H27N3O4
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0372414
|
(S)-4'-{2-[(2-Hydroxy-3-phenoxypropyl)amino]ethyl}-2-[1-(2-naphtylmethyl)imidazol-2-yl]acetanilide
Show/Hide
|
C33H34N4O3
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0382049
|
(S)-N-Methyl-4'-{2-[(2-hydroxy-3-phenoxypropyl)-amino]ethyl}-2-(1-benzylimidazol-2-yl)acetanilide
Show/Hide
|
C30H34N4O3
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0388089
|
(S)-4'-{2-[(2-Hydroxy-3-phenoxypropyl)amino]ethyl}-2-(1-benzylimidazol-4-yl)-acetanilide
Show/Hide
|
C29H32N4O3
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0388090
|
(S)-4'-{2-[(2-Hydroxy-3-phenoxypropyl)amino]ethyl}-2-[1-(4-chlorobenzyl)imidazol-2-yl]acetanilide
Show/Hide
|
C29H31ClN4O3
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0388092
|
(S)-4'-(2-{[2-Hydroxy-3-phenoxypropyl]amino}ethyl)-2-(3-methyl-2-pyridyl)acetanilide
Show/Hide
|
C25H29N3O3
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0388094
|
(S)-4'-{2-[(2-Hydroxy-3-phenoxypropyl)amino]ethyl}-2-(6-chloro-2-pyridyl)acetanilide
Show/Hide
|
C24H26ClN3O3
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0388095
|
(S)-4'-{2-[(2-Hydroxy-3-phenoxypropyl)amino]ethyl}-2-[1-(4-bromobenzyl)imidazol-2-yl]acetanilide
Show/Hide
|
C29H31BrN4O3
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0427161
|
(S)-4'-(2-{[2-Hydroxy-3-(carbazol-4-yloxy)propyl]-amino}ethyl)-2-(2-pyridyl)acetanilide
Show/Hide
|
C26H28N4O3
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0431167
|
(S)-1-[(2-{1-[(1-Benzylimidazol-2-yl)acetyl]-1,2,3,4-tetrahydroquinolin-6-yl}ethyl)-amino]-3-phenoxy-2-propanol
Show/Hide
|
C32H36N4O3
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0431169
|
(S)-4'-{2-[(2-Hydroxy-3-phenoxypropyl)amino]ethyl}-2-(1-phenylimidazol-2-yl)-acetanilide
Show/Hide
|
C28H30N4O3
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0439488
|
(S)-4'-(2-{[2-Hydroxy-3-(carbazol-4-yloxy)propyl]-amino}ethyl)-2-(2-pyridyl)acetanilide
Show/Hide
|
C30H30N4O3
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0439490
|
(S)-4'-(2-{[2-Hydroxy-3-(indol-4-yloxy)propyl]amino}-ethyl)-2-(2-pyridyl)acetanilide
Show/Hide
|
C25H27N5O4
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0443470
|
(S)-4'-(2-{[2-Hydroxy-3-phenoxypropyl]amino}ethyl)-2-(2-pyridyl)acetanilide
Show/Hide
|
C24H27N3O3
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0443472
|
(S)-4'-(2-{[2-Hydroxy-3-(2-benzimidazolon-4-yloxy)-propyl]amino}ethyl)-2-(2-pyridyl)-acetanilide
Show/Hide
|
C23H26N4O3
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0443473
|
(S)-4'-{2-[(2-Hydroxy-3-phenoxypropyl)amino]ethyl}-2-(6-benzyloxy-2-pyridyl)-acetanilide
Show/Hide
|
C31H33N3O4
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0044683
|
4-{(S)-2-Hydroxy-3-[1-(4-methoxy-benzenesulfonyl)-piperidin-4-ylamino]-propoxy}-phenol
Show/Hide
|
C21H28N2O6S
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0094903
|
(S)-1-(9H-Carbazol-4-yloxy)-3-[1-(4-methoxy-benzenesulfonyl)-piperidin-4-ylamino]-propan-2-ol
Show/Hide
|
C27H31N3O5S
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
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CP0097140
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4-{(S)-2-Hydroxy-3-[1-(4-methoxy-benzenesulfonyl)-piperidin-4-ylamino]-propoxy}-1,3-dihydro-benzoimidazol-2-one
Show/Hide
|
C22H28N4O6S
|
1
|
| 1 |
EC50 > 100000 nM
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|
|
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CP0130252
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4-{(S)-3-[1-(3,4-Dimethoxy-benzenesulfonyl)-piperidin-4-ylamino]-2-hydroxy-propoxy}-1,3-dihydro-benzoimidazol-2-one
Show/Hide
|
C23H30N4O7S
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
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CP0139363
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(S)-1-(9H-Carbazol-4-yloxy)-3-[1-(3,4-dimethoxy-benzenesulfonyl)-piperidin-4-ylamino]-propan-2-ol
Show/Hide
|
C28H33N3O6S
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
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CP0270078
|
(S)-1-[1-(4-Butoxy-benzenesulfonyl)-piperidin-4-ylamino]-3-(9H-carbazol-4-yloxy)-propan-2-ol
Show/Hide
|
C30H37N3O5S
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
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CP0279642
|
(S)-N-(4-(2-(2-hydroxy-3-(4-hydroxyphenoxy)propylamino)ethyl)phenyl)benzenesulfonamide
Show/Hide
|
C23H26N2O5S
|
2
|
| 1 |
EC50 > 100000 nM
|
|
|
| 2 |
IC50 = 190 nM
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|
|
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CP0404751
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(S)-N-(4-(2-(2-hydroxy-3-phenoxypropylamino)ethyl)phenyl)benzenesulfonamide
Show/Hide
|
C23H26N2O4S
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0844961
|
(S)-1-(4-{2-[(2-Hydroxy-3-phenoxypropyl)amino]ethyl}-phenyl)-3-phenylthiourea hydrochloride
Show/Hide
|
C24H28ClN3O2S
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0844962
|
(S)-1-(4-{2-[(2-Hydroxy-3-phenoxypropyl)amino]ethyl}-phenyl)-3-(4-methoxycarbonylphenyl)thiourea hydrochloride
Show/Hide
|
C26H30ClN3O4S
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
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CP0844965
|
(S)-2-Cyano-1-(4-{2-[(2-hydroxy-3-phenoxypropyl)-amino]ethyl}phenyl)-3-phenylguanidine hydrochloride
Show/Hide
|
C25H28ClN5O2
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0844967
|
(S)-1-(4-Bromophenyl)-3-(4-{2-[(2-hydroxy-3-phenoxypropyl)amino]ethyl}phenyl)thiourea hydrochloride
Show/Hide
|
C24H27BrClN3O2S
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0844968
|
(S)-1-Benzyl-3-(4-{2-[(2-hydroxy-3-phenoxypropyl)amino]-ethyl}phenyl)thiourea hydrochloride
Show/Hide
|
C25H30ClN3O2S
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0851797
|
(S)-1-(4-{2-[(2-Hydroxy-3-phenoxypropyl)amino]ethyl}-phenyl)-3-(3-nitrophenyl)thiourea hydrochloride
Show/Hide
|
C24H27ClN4O4S
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0851798
|
(S)-1-(4-{2-[(2-Hydroxy-3-phenoxypropyl)amino]ethyl}-phenyl)-3-(4-iodophenyl)thiourea hydrochloride
Show/Hide
|
C24H27ClIN3O2S
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0851799
|
(S)-1-(4-{2-[(2-Hydroxy-3-phenoxypropyl)amino]ethyl}-phenyl)-3-(4-methylphenyl)thiourea hydrochloride
Show/Hide
|
C25H30ClN3O2S
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0851800
|
(S)-1-Phenoxy-3-({2-[4-(phenylamino)phenyl]ethyl}amino)-2-propanol hydrochloride
Show/Hide
|
C23H27ClN2O2
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0851807
|
(S)-1-(3-Chlorophenyl)-3-(4-{2-[(2-hydroxy-3-phenoxypropyl)amino]ethyl}phenyl)thiourea hydrochloride
Show/Hide
|
C24H27Cl2N3O2S
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0851810
|
Phenyl (S)-(4-{2-[(2-hydroxy-3-phenoxypropyl)amino]ethyl}phenyl)carbamate hydrochloride
Show/Hide
|
C24H27ClN2O4
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0858640
|
(S)-1-(4-{2-[(2-Hydroxy-3-phenoxypropyl)amino]ethyl}-phenyl)-3-(3-methoxyphenyl)thiourea hydrochloride
Show/Hide
|
C25H30ClN3O3S
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0858641
|
(S)-1-(4-{2-[(2-Hydroxy-3-phenoxypropyl)amino]ethyl}-phenyl)-3-(4-sulfamoylphenyl)thiourea hydrochloride
Show/Hide
|
C24H29ClN4O4S2
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0858642
|
(S)-1-Cyclohexyl-3-(4-{2-[(2-hydroxy-3-phenoxypropyl)-amino]ethyl}phenyl)thiourea hydrochloride
Show/Hide
|
C24H34ClN3O2S
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0858643
|
(S)-1-(2-Chlorophenyl)-3-(4-{2-[(2-hydroxy-3-phenoxypropyl)amino]ethyl}phenyl)thiourea hydrochloride
Show/Hide
|
C24H27Cl2N3O2S
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0858644
|
(S)-1-(4-{2-[(2-Hydroxy-3-phenoxypropyl)amino]ethyl}-phenyl)-3-(2-nitrophenyl)thiourea hydrochloride
Show/Hide
|
C24H27ClN4O4S
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0861800
|
(S)-1-(4-Chlorophenyl)-3-(4-{2-[(2-hydroxy-3-phenoxypropyl)amino]ethyl}phenyl)thiourea hydrochloride
Show/Hide
|
C24H27Cl2N3O2S
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0861819
|
(S)-1-(4-{2-[(2-Hydroxy-3-phenoxypropyl)amino]ethyl}-phenyl)-3-(2-methoxyphenyl)thiourea hydrochloride
Show/Hide
|
C25H30ClN3O3S
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0861821
|
(S)-1-(4-{2-[(2-Hydroxy-3-phenoxypropyl)amino]ethyl}phenyl)-3-phenylurea hydrochloride
Show/Hide
|
C24H28ClN3O3
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0861826
|
(S)-N-Phenyl-4-{2-[(2-hydroxy-3-phenoxypropyl)amino]-ethyl}benzenesulfonamide hydrochloride
Show/Hide
|
C23H27ClN2O4S
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0873011
|
(S)-1-(4-{2-[(2-Hydroxy-3-phenoxypropyl)amino]ethyl}-phenyl)-3-(2-phenylethyl)thiourea hydrochloride
Show/Hide
|
C26H32ClN3O2S
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0873012
|
(S)-1-(4-{2-[(2-Hydroxy-3-phenoxypropyl)amino]ethyl}-phenyl)-3-(4-nitrophenyl)thiourea hydrochloride
Show/Hide
|
C24H27ClN4O4S
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0873014
|
(S)-1-(4-Fluorophenyl)-3-(4-{2-[(2-hydroxy-3-phenoxypropyl)amino]ethyl}phenyl)thiourea hydrochloride
Show/Hide
|
C24H27ClFN3O2S
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0891546
|
(S)-N-(4-{2-[(2-Hydroxy-3-phenoxypropyl)amino]ethyl}phenyl)benzamide hydrochloride
Show/Hide
|
C24H27ClN2O3
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0372784
|
(S)-4'-(2-{[2-Hydroxy-3-(4-hydroxyphenoxy)propyl]amino}ethyl)-2,2-diphenylacetanilide
Show/Hide
|
C31H32N2O4
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0372785
|
(S)-4'-(2-{[2-Hydroxy-3-(4-hydroxyphenoxy)propyl]amino}ethyl)-2-(4-pyridyl)acetanilide
Show/Hide
|
C24H27N3O4
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0375758
|
(S)-4'-(2-{[2-Hydroxy-3-(4-hydroxyphenoxy)propyl]amino}ethyl)-2-(3-chlorophenyl)acetanilide
Show/Hide
|
C25H27ClN2O4
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0375759
|
(S)-4'-(2-{[2-Hydroxy-3-(4-hydroxyphenoxy)propyl]amino}ethyl)-2-(3-pyridyl)acetanilide
Show/Hide
|
C24H27N3O4
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0375760
|
(S)-4'-(2-{[2-Hydroxy-3-(4-hydroxyphenoxy)propyl]amino}ethyl)-2-phenylacetanilide
Show/Hide
|
C25H28N2O4
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0375775
|
(S)-4'-(2-{[2-Hydroxy-3-(4-hydroxyphenoxy)propyl]amino}ethyl)-2-(2-methoxyphenyl)acetanilide
Show/Hide
|
C26H30N2O5
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0377688
|
(S)-4'-(2-{[2-Hydroxy-3-(4-hydroxyphenoxy)propyl]amino}ethyl)-2-(isoquinolin-3-yl)acetanilide
Show/Hide
|
C28H29N3O4
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0377695
|
(S)-4'-(2-{[2-Hydroxy-3-(4-hydroxyphenoxy)propyl]amino}ethyl)-2-amino-2-phenylacetanilide
Show/Hide
|
C25H29N3O4
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0377697
|
(S)-4'-(2-{[2-Hydroxy-3-(4-hydroxyphenoxy)propyl]amino}ethyl)-2-(quinolin-2-yl)acetanilide
Show/Hide
|
C28H29N3O4
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0377700
|
(S)-4'-(2-{[2-Hydroxy-3-(4-hydroxyphenoxy)propyl]amino}ethyl)-2-(2-naphthyl)acetanilide
Show/Hide
|
C29H30N2O4
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0377701
|
(S)-4'-(2-{[2-Hydroxy-3-(4-hydroxyphenoxy)propyl]amino}ethyl)-2-(3-thenyl)acetanilide
Show/Hide
|
C23H26N2O4S
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0377702
|
(S)-4'-(2-{[2-Hydroxy-3-(4-hydroxyphenoxy)propyl]amino}ethyl)-2-hydroxy-2-phenylacetanilide
Show/Hide
|
C25H28N2O5
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0387789
|
(S)-4'-(2-{[2-Hydroxy-3-(4-hydroxyphenoxy)propyl]amino}ethyl)-2-(pyrazin-2-yl)acetanilide
Show/Hide
|
C23H26N4O4
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0387792
|
(S)-4'-(2-{[2-Hydroxy-3-(4-hydroxyphenoxy)propyl]amino}ethyl)-2-(2-chlorophenyl)acetanilide
Show/Hide
|
C25H27ClN2O4
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0387797
|
(S)-4'-(2-{[2-Hydroxy-3-(4-hydroxyphenoxy)propyl]amino}ethyl)-2-(4-methoxyphenyl)acetanilide
Show/Hide
|
C26H30N2O5
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0388477
|
(S)-4'-(2-{[2-Hydroxy-3-(4-hydroxyphenoxy)propyl]amino}ethyl)-2-(pyrimidin-2-yl)acetanilide
Show/Hide
|
C23H26N4O4
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0431466
|
(S)-4'-(2-{[2-Hydroxy-3-(4-hydroxyphenoxy)propyl]amino}ethyl)-2-(3-methoxyphenyl)acetanilide
Show/Hide
|
C26H30N2O5
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0431469
|
(S)-4'-(2-{[2-Hydroxy-3-(4-hydroxyphenoxy)propyl]amino}ethyl)-2-(2-thenyl)acetanilide
Show/Hide
|
C23H26N2O4S
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0474045
|
(S)-4'-(2-{[2-Hydroxy-3-(4-hydroxyphenoxy)propyl]amino}ethyl)-2-(4-chlorophenyl)acetanilide
Show/Hide
|
C25H27ClN2O4
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0504027
|
(S)-4'-(2-{[2-Hydroxy-3-(4-hydroxyphenoxy)propyl]amino}ethyl)-2-(1-naphthyl)acetanilide
Show/Hide
|
C29H30N2O4
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0851904
|
(S)-4'-(2-{[2-Hydroxy-3-(4-hydroxyphenoxy)propyl]amino}ethyl)-2-(indol-3-yl)acetanilide
Show/Hide
|
C27H29N3O4
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0849414
|
1-(4-{(S)-3-Hydroxy-2-[2-hydroxy-3-((S)-phenoxy)-propylamino]-propyl}-phenyl)-3-phenyl-urea
Show/Hide
|
C25H29N3O4
|
1
|
| 1 |
EC50 > 100 nM
|
|
|
|
CP0403861
|
1-(9H-Carbazol-4-yloxy)-3-[(1-hexyl-piperidin-4-ylmethyl)-amino]-propan-2-ol
Show/Hide
|
C27H39N3O2
|
1
|
| 1 |
EC50 > 1000 nM
|
|
|
|
CP0403918
|
1-(9H-Carbazol-4-yloxy)-3-{[1-(3,3,3-trifluoro-propyl)-piperidin-4-ylmethyl]-amino}-propan-2-ol
Show/Hide
|
C24H30F3N3O2
|
1
|
| 1 |
EC50 > 1000 nM
|
|
|
|
CP0430919
|
1-[(S)-4-(4-{[3-(9H-Carbazol-4-yloxy)-2-hydroxy-propylamino]-methyl}-piperidine-1-sulfonyl)-phenyl]-3-hexyl-urea
Show/Hide
|
C34H45N5O5S
|
1
|
| 1 |
EC50 > 1000 nM
|
|
|
|
CP0472259
|
3-[((S)-4-{[3-(9H-Carbazol-4-yloxy)-2-hydroxy-propylamino]-methyl}-piperidine-1-carbonyl)-amino]-benzoic acid
Show/Hide
|
C29H32N4O5
|
1
|
| 1 |
EC50 > 1000 nM
|
|
|
|
CP0419581
|
2-[3-[[(2R)-2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]propyl]amino]phenyl]-N-(4-methylphenyl)sulfonylacetamide
Show/Hide
|
C26H30ClN3O4S
|
1
|
| 1 |
EC50 < 1000 nM
|
|
|
|
CP0372880
|
(R)-4'-(2-(2-hydroxy-2-phenylethylamino)ethyl)-3-(isopropylthio)biphenyl-4-carboxylic acid
Show/Hide
|
C26H29NO3S
|
1
|
| 1 |
EC50 > 1000 nM
|
|
|
|
CP0381824
|
(R)-4'-(2-(2-(3-chlorophenyl)-2-hydroxyethylamino)ethyl)-3-methoxybiphenyl-4-carboxylic acid
Show/Hide
|
C24H24ClNO4
|
1
|
| 1 |
EC50 > 1000 nM
|
|
|
|
CP0504380
|
(R)-4'-(2-(2-(4-aminopyridin-3-yl)-2-hydroxyethylamino)ethyl)-3-isopropoxybiphenyl-4-carboxylic acid
Show/Hide
|
C25H29N3O4
|
1
|
| 1 |
EC50 > 1000 nM
|
|
|
|
CP0372774
|
5-[((7S)-7-{[(2R)-2-(6-Chloro-3-pyridinyl)-2-hydroxyethyl]amino}-5,6,7,8-tetrahydro-2-naphthalenyl)oxy]-2-methoxybenzoic Acid
Show/Hide
|
C25H25ClN2O5
|
1
|
| 1 |
EC50 > 1000 nM
|
|
|
|
CP0372799
|
5-[((7S)-7-{[(2R)-2-(3-Chlorophenyl)-2-hydroxyethyl]amino}-5,6,7,8-tetrahydro-2-naphthalenyl)oxy]-2-methoxybenzoic Acid
Show/Hide
|
C26H26ClNO5
|
1
|
| 1 |
EC50 > 1000 nM
|
|
|
|
CP0381359
|
4-((S)-7-((R)-2-(6-chloropyridin-3-yl)-2-hydroxyethylamino)-5,6,7,8-tetrahydronaphthalen-2-yl)benzoic acid
Show/Hide
|
C24H23ClN2O3
|
1
|
| 1 |
EC50 > 1000 nM
|
|
|
|
CP0387764
|
4-((7S)-7-{[(2R)-2-(3-Chlorophenyl)-2-hydroxyethyl]amino}-5,6,7,8-tetrahydro-2-naphthalenyl)benzoic Acid
Show/Hide
|
C25H24ClNO3
|
1
|
| 1 |
EC50 > 1000 nM
|
|
|
|
CP0387892
|
3-[((7S)-7-{[(2R)-2-(3-Chlorophenyl)-2-hydroxyethyl]amino}-5,6,7,8-tetrahydro-2-naphthalenyl)oxy]-5-(dimethylamino)benzoicAcid
Show/Hide
|
C27H29ClN2O4
|
1
|
| 1 |
EC50 > 1000 nM
|
|
|
|
CP0387894
|
4-((S)-7-((R)-2-hydroxy-2-(4-(trifluoromethyl)phenyl)ethylamino)-5,6,7,8-tetrahydronaphthalen-2-yl)benzoic acid
Show/Hide
|
C26H24F3NO3
|
1
|
| 1 |
EC50 > 1000 nM
|
|
|
|
CP0393173
|
6-[((7S)-7-{[(2R)-2-(3-Chlorophenyl)-2-hydroxyethyl]amino}-5,6,7,8-tetrahydro-2-naphthalenyl)oxy]nicotinic Acid
Show/Hide
|
C24H23ClN2O4
|
1
|
| 1 |
EC50 > 1000 nM
|
|
|
|
CP0393188
|
4-((7S)-7-{[(2R)-2-(3-Chlorophenyl)-2-hydroxyethyl]amino}-5,6,7,8-tetrahydro-2-naphthalenyl)phenoxy]acetic Acid
Show/Hide
|
C26H26ClNO4
|
1
|
| 1 |
EC50 > 1000 nM
|
|
|
|
CP0399816
|
5-[((7S)-7-{[(2R)-2-(3-Chlorophenyl)-2-hydroxyethyl]amino}-5,6,7,8-tetrahydro-2-naphthalenyl)oxy]-2-thiophenecarboxylic Acid
Show/Hide
|
C23H22ClNO4S
|
1
|
| 1 |
EC50 > 1000 nM
|
|
|
|
CP0456745
|
5-[((7S)-7-{[(2R)-2-(4-Chlorophenyl)-2-hydroxyethyl]amino}-5,6,7,8-tetrahydro-2-naphthalenyl)oxy]-2-methoxybenzoic Acid
Show/Hide
|
C26H26ClNO5
|
1
|
| 1 |
EC50 > 1000 nM
|
|
|
|
CP0493893
|
4-((S)-7-((R)-2-(4-chlorophenyl)-2-hydroxyethylamino)-5,6,7,8-tetrahydronaphthalen-2-yl)benzoic acid
Show/Hide
|
C25H24ClNO3
|
1
|
| 1 |
EC50 > 1000 nM
|
|
|
|
CP0500727
|
3-[((7S)-7-{[(2R)-2-(3-Chlorophenyl)-2-hydroxyethyl]amino}-5,6,7,8-tetrahydro-2-naphthalenyl)oxy]-5-methoxybenzoic Acid
Show/Hide
|
C26H26ClNO5
|
1
|
| 1 |
EC50 > 1000 nM
|
|
|
|
CP0503536
|
3-[((7S)-7-{[(2R)-2-(3-Chlorophenyl)-2-hydroxyethyl]amino}-5,6,7,8-tetrahydro-2-naphthalenyl)oxy]benzoic Acid
Show/Hide
|
C25H24ClNO4
|
1
|
| 1 |
EC50 > 1000 nM
|
|
|
|
CP0504227
|
3-[((8S)-8-{[(2R)-2-(3-Chlorophenyl)-2-hydroxyethyl]amino}-6,7,8,9-tetrahydro-5H-benzo[a]cyclohepten-2-yl)oxy]benzoic Acid
Show/Hide
|
C26H26ClNO4
|
1
|
| 1 |
EC50 > 1000 nM
|
|
|
|
CP0375141
|
4-[(2R)-2-{[(2R)-2-Hydroxy-2-phenylethyl]amino}propyl]biphenyl-4-carboxylic acid
Show/Hide
|
C24H25NO3
|
1
|
| 1 |
EC50 > 1000 nM
|
|
|
|
CP0375142
|
4-((2R)-2-{[(2R)-2-Hydroxy-2-(3-pyridinyl)ethyl]amino}propyl)-3-propoxy-4-biphenylcarboxylic acid
Show/Hide
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C26H30N2O4
|
1
|
| 1 |
EC50 > 1000 nM
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CP0400939
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4-((2R)-2-{[(2R)-2-Hydroxy-2-(3-pyridyl)ethyl]amino}propyl)-3-isopropyloxy-1,1-biphenyl-4-carboxylic acid
Show/Hide
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C26H30N2O4
|
1
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| 1 |
EC50 > 1000 nM
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CP0484987
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4-((2R)-2-{[(2R)-2-Hydroxy-2-(3-pyridinyl)ethyl]amino}propyl)-1,1-biphenyl-4-carboxylic acid
Show/Hide
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C23H24N2O3
|
1
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| 1 |
EC50 > 1000 nM
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CP0403283
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4-[3-[[(2R)-2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]propyl]amino]phenyl]benzene-1,3-dicarboxylic acid
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C25H25ClN2O5
|
1
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| 1 |
EC50 < 10000 nM
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CP0439425
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3-[3-[2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]ethylamino]phenyl]pyridine-4-carboxylic acid
Show/Hide
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C22H22ClN3O3
|
1
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| 1 |
EC50 < 10000 nM
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CP0068490
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1-[(7-methyl-2,3-dihydro-1H-inden-4-yl)oxy]-3-(propan-2-ylamino)butan-2-ol
Show/Hide
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C17H27NO2
|
1
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| 1 |
IC50 = 0.74 nM
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CP0101662
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(2R,3S)-1-[(7-methyl-2,3-dihydro-1H-inden-4-yl)oxy]-3-(propan-2-ylamino)butan-2-ol
Show/Hide
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C17H27NO2
|
1
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| 1 |
IC50 = 0.74 nM
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CP0072120
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(-)-(S)-Propranolol
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C16H21NO2
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2
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| 1 |
IC50 = 0.78 nM
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| 2 |
Ki = 0.54 nM
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CP0044877
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1-(3,4,5-Trimethoxy-benzyl)-1,2,3,4-tetrahydro-isoquinoline-6,7-diol
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C19H23NO5
|
2
|
| 1 |
IC50 = 6.1 nM
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| 2 |
Ki = 43.65 nM
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CP0419183
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4-((3S)-3-{[(2S)-2-hydroxy-3-(4-hydroxyphenoxy)propyl]amino}butyl)phenol
Show/Hide
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C19H25NO4
|
1
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| 1 |
IC50 = 10 nM
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CP0437272
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N-[4-[2-[[(2S)-2-hydroxy-3-(4-hydroxyphenoxy)propyl]amino]ethyl]phenyl]acetamide
Show/Hide
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C19H24N2O4
|
1
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| 1 |
IC50 = 11 nM
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CP0464087
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4-{(S)-2-Hydroxy-3-[(S)-3-(4-methoxy-phenyl)-1-methyl-propylamino]-propoxy}-phenol
Show/Hide
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C20H27NO4
|
1
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| 1 |
IC50 = 20 nM
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CP0375012
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N-[4-[2-[[(2S)-2-hydroxy-3-(4-hydroxyphenoxy)propyl]amino]ethyl]phenyl]-1-phenylmethanesulfonamide
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C24H28N2O5S
|
1
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| 1 |
IC50 = 21 nM
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CP0422411
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N-[4-[2-[[(2S)-3-(6-aminopyridin-3-yl)oxy-2-hydroxypropyl]amino]ethyl]phenyl]-4-iodobenzenesulfonamide
Show/Hide
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C22H25IN4O4S
|
1
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| 1 |
IC50 = 28 nM
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CP0245933
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1-cyano-2-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-3-(3-phenoxyphenyl)guanidine
Show/Hide
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C29H28N6O2
|
1
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| 1 |
IC50 = 40 nM
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CP0487112
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1-[5-(3-cyclopentylpropyl)-1,2,4-oxadiazol-3-yl]-N-phenyl-2,3-dihydro-1H-indole-5-sulfonamide
Show/Hide
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C24H28N4O3S
|
1
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| 1 |
IC50 = 42 nM
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CP0457043
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N-[4-[2-[[(2S)-2-hydroxy-3-phenoxypropyl]amino]ethyl]phenyl]-4-iodobenzenesulfonamide
Show/Hide
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C23H25IN2O4S
|
1
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| 1 |
IC50 = 50 nM
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CP0149413
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1-cyano-2-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-3-[1-(4-octyl-1,3-thiazol-2-yl)-2,3-dihydroindol-5-yl]guanidine
Show/Hide
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C36H44N8OS
|
1
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| 1 |
IC50 = 50 nM
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CP0299564
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1-cyano-2-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-3-naphthalen-2-ylguanidine
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C27H26N6O
|
1
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| 1 |
IC50 = 50 nM
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CP0530370
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1-(5-hexyl-1,2,4-oxadiazol-3-yl)-N-phenyl-2,3-dihydro-1H-indole-5-sulfonamide
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C22H26N4O3S
|
1
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| 1 |
IC50 = 52 nM
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CP0406365
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4-(3,5-Diiodo-4-methoxy-benzyl)-4,5,6,7-tetrahydro-thiazolo[5,4-c]pyridin-2-ylamine
Show/Hide
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C14H15I2N3OS
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2
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| 1 |
IC50 = 56 nM
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| 2 |
Ki = 426.58 nM
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CP0408503
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N-[4-[2-[[(2S)-2-hydroxy-3-(4-hydroxyphenoxy)propyl]amino]ethyl]phenyl]propane-2-sulfonamide
Show/Hide
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C20H28N2O5S
|
1
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| 1 |
IC50 = 58 nM
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CP0373740
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(R)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)biphenyl-4-carboxamide
Show/Hide
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C28H27N3O2
|
1
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| 1 |
IC50 = 60 nM
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CP0498157
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4-{(S)-2-Hydroxy-3-[3-(4-methoxy-phenyl)-propylamino]-propoxy}-phenol
Show/Hide
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C19H25NO4
|
1
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| 1 |
IC50 = 63 nM
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CP0432925
|
1-(6-octylpyridin-2-yl)-N-phenyl-2,3-dihydro-1H-indole-5-sulfonamide
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C27H33N3O2S
|
1
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| 1 |
IC50 = 63 nM
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CP0110208
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1-cyano-2-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-3-[1-(4-octyl-1,3-thiazol-2-yl)-2,3-dihydroindol-6-yl]guanidine
Show/Hide
|
C36H44N8OS
|
1
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| 1 |
IC50 = 66 nM
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CP0267922
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1-cyano-2-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-3-(3-iodophenyl)guanidine
Show/Hide
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C23H23IN6O
|
1
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| 1 |
IC50 = 67 nM
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CP0447775
|
4-((2S)-2-{[(2S)-2-hydroxy-3-(4-hydroxyphenoxy)propyl]amino}propyl)phenol
Show/Hide
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C18H23NO4
|
1
|
| 1 |
IC50 = 84 nM
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CP0400966
|
4-Ethyl-N-(4-{2-[(S)-2-hydroxy-3-(pyridin-3-yloxy)-propylamino]-ethyl}-phenyl)-benzenesulfonamide
Show/Hide
|
C24H29N3O4S
|
1
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| 1 |
IC50 = 94 nM
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CP0406510
|
2-Chloro-N-(4-{2-[(S)-2-hydroxy-3-(4-hydroxy-phenoxy)-propylamino]-ethyl}-phenyl)-benzenesulfonamide
Show/Hide
|
C23H25ClN2O5S
|
1
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| 1 |
IC50 = 100 nM
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CP0495433
|
N-[4-[2-[[(2S)-3-(4-fluorophenoxy)-2-hydroxypropyl]amino]ethyl]phenyl]-4-iodobenzenesulfonamide
Show/Hide
|
C23H24FIN2O4S
|
1
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| 1 |
IC50 = 100 nM
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CP0409910
|
1-(5-octyl-1,2,4-oxadiazol-3-yl)-N-phenyl-2,3-dihydro-1H-indole-5-sulfonamide
Show/Hide
|
C24H30N4O3S
|
1
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| 1 |
IC50 = 100 nM
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CP0447499
|
(R)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)-4-phenethylbenzamide
Show/Hide
|
C30H31N3O2
|
1
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| 1 |
IC50 = 100 nM
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CP0377226
|
3-(2-hydroxy-3-(1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propoxy)phenol
Show/Hide
|
C26H28N4O3S
|
2
|
| 1 |
IC50 = 100 nM
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| 2 |
Ki = 6 nM
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CP0039159
|
N-[4-[2-[[(2S)-2-hydroxy-3-pyridin-3-yloxypropyl]amino]ethyl]phenyl]-4-iodobenzenesulfonamide
Show/Hide
|
C22H24IN3O4S
|
1
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| 1 |
IC50 = 110 nM
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CP0501166
|
N-[4-[2-[[(2S)-3-(6-aminopyridin-3-yl)oxy-2-hydroxypropyl]amino]ethyl]phenyl]-4-ethylbenzenesulfonamide
Show/Hide
|
C24H30N4O4S
|
1
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| 1 |
IC50 = 110 nM
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CP0406511
|
N-[4-[2-[[(2S)-2-hydroxy-3-(4-hydroxyphenoxy)propyl]amino]ethyl]phenyl]-4-iodobenzenesulfonamide
Show/Hide
|
C23H25IN2O5S
|
1
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| 1 |
IC50 = 120 nM
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CP0406530
|
2-Phenyl-ethanesulfonic acid (4-{2-[(S)-2-hydroxy-3-(4-hydroxy-phenoxy)-propylamino]-ethyl}-phenyl)-amide
Show/Hide
|
C25H30N2O5S
|
1
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| 1 |
IC50 = 120 nM
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CP0388522
|
1-(1-(5-(4-fluorophenyl)thieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)-3-phenoxypropan-2-ol
Show/Hide
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C26H27FN4O2S
|
2
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| 1 |
IC50 = 123 nM
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| 2 |
Ki = 19 nM
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CP0405254
|
3-Phenyl-propane-1-sulfonic acid (4-{2-[(S)-2-hydroxy-3-(4-hydroxy-phenoxy)-propylamino]-ethyl}-phenyl)-amide
Show/Hide
|
C26H32N2O5S
|
1
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| 1 |
IC50 = 130 nM
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CP0448240
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1-(6-hexylpyridin-2-yl)-N-phenyl-2,3-dihydro-1H-indole-5-sulfonamide
Show/Hide
|
C25H29N3O2S
|
1
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| 1 |
IC50 = 140 nM
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CP0360976
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1-cyano-3-(3,5-dichlorophenyl)-2-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]guanidine
Show/Hide
|
C23H22Cl2N6O
|
1
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| 1 |
IC50 = 140 nM
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CP0410916
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4-(2-{[(2S)-2-hydroxy-3-(4-hydroxyphenoxy)propyl]amino}ethyl)phenol
Show/Hide
|
C17H21NO4
|
1
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| 1 |
IC50 = 150 nM
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CP0530324
|
N-[4-[2-[[(2S)-2-hydroxy-3-(4-methoxyphenoxy)propyl]amino]ethyl]phenyl]-4-iodobenzenesulfonamide
Show/Hide
|
C24H27IN2O5S
|
1
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| 1 |
IC50 = 150 nM
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CP0299165
|
1-[4-[[4-[4-[(6,7-dihydroxy-1,2,3,4-tetrahydroisoquinolin-1-yl)methoxy]phenyl]phenyl]sulfamoyl]phenyl]-3-hexylurea
Show/Hide
|
C35H40N4O6S
|
1
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| 1 |
IC50 = 160 nM
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CP0380549
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N-[4-[2-[[(2S)-2-hydroxy-3-(4-hydroxyphenoxy)propyl]amino]ethyl]phenyl]-4-methylbenzenesulfonamide
Show/Hide
|
C24H28N2O5S
|
1
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| 1 |
IC50 = 170 nM
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CP0106484
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1-cyano-2-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-3-(4-iodophenyl)guanidine
Show/Hide
|
C23H23IN6O
|
1
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| 1 |
IC50 = 170 nM
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CP0480631
|
4-Bromo-N-(4-{2-[(S)-2-hydroxy-3-(4-hydroxy-phenoxy)-propylamino]-ethyl}-phenyl)-benzenesulfonamide
Show/Hide
|
C23H25BrN2O5S
|
1
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| 1 |
IC50 = 180 nM
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CP0459230
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1-(5-octyl-1,3-oxazol-2-yl)-N-phenyl-2,3-dihydro-1H-indole-5-sulfonamide
Show/Hide
|
C25H31N3O3S
|
1
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| 1 |
IC50 = 180 nM
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CP0362780
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1-cyano-2-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-3-[1-[4-[4-(trifluoromethoxy)phenyl]-1,3-thiazol-2-yl]-2,3-dihydroindol-5-yl]guanidine
Show/Hide
|
C35H31F3N8O2S
|
1
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| 1 |
IC50 = 180 nM
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CP0525981
|
N-[4-[2-[[(2S)-2-hydroxy-3-(4-hydroxyphenoxy)propyl]amino]ethyl]phenyl]-4-methoxybenzenesulfonamide
Show/Hide
|
C24H28N2O6S
|
1
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| 1 |
IC50 = 190 nM
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CP0436821
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1-[4-[[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]sulfamoyl]phenyl]-3-(2-phenylethyl)urea
Show/Hide
|
C30H33N5O4S
|
1
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| 1 |
IC50 = 200 nM
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CP0453193
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1-[4-[[4-[(6,7-dihydroxy-1,2,3,4-tetrahydroisoquinolin-1-yl)methyl]phenyl]sulfamoyl]phenyl]-3-hexylurea
Show/Hide
|
C29H36N4O5S
|
1
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| 1 |
IC50 = 200 nM
|
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CP0364013
|
1-cyano-3-(3-fluorophenyl)-2-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]guanidine
Show/Hide
|
C23H23FN6O
|
1
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| 1 |
IC50 = 200 nM
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CP0374173
|
1-(2-methoxyphenoxy)-3-(1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propan-2-ol
Show/Hide
|
C27H30N4O3S
|
2
|
| 1 |
IC50 = 205 nM
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| 2 |
Ki = 11 nM
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CP0404587
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N-[4-[2-[[(2S)-2-hydroxy-3-(4-hydroxyphenoxy)propyl]amino]ethyl]phenyl]methanesulfonamide
Show/Hide
|
C18H24N2O5S
|
1
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| 1 |
IC50 = 220 nM
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CP0862655
|
(R)-2-(2-{4-[2-Nitro-1-(3-phenoxy-phenylamino)-vinylamino]-phenyl}-ethylamino)-1-pyridin-3-yl-ethanol
Show/Hide
|
C29H29N5O4
|
1
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| 1 |
IC50 = 220 nM
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CP0406259
|
1-(2-fluorophenoxy)-3-(1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propan-2-ol
Show/Hide
|
C26H27FN4O2S
|
2
|
| 1 |
IC50 = 220 nM
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| 2 |
Ki = 25 nM
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CP0441536
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N-[4-[2-[[(2S)-2-hydroxy-3-(4-hydroxyphenoxy)propyl]amino]ethyl]phenyl]benzamide
Show/Hide
|
C24H26N2O4
|
1
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| 1 |
IC50 = 230 nM
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CP0463785
|
4-Bromo-N-(4-{2-[(S)-2-hydroxy-3-(pyridin-3-yloxy)-propylamino]-ethyl}-phenyl)-benzenesulfonamide
Show/Hide
|
C22H24BrN3O4S
|
1
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| 1 |
IC50 = 230 nM
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CP0403330
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N-[4-[2-[[(2S)-2-hydroxy-3-(4-hydroxyphenoxy)propyl]amino]ethyl]phenyl]quinoline-3-sulfonamide
Show/Hide
|
C26H27N3O5S
|
1
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| 1 |
IC50 = 240 nM
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CP0409911
|
1-(5-hexylpyridin-2-yl)-N-phenyl-2,3-dihydro-1H-indole-5-sulfonamide
Show/Hide
|
C25H29N3O2S
|
1
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| 1 |
IC50 = 240 nM
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CP0377154
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1-(3-(hydroxymethyl)phenoxy)-3-(1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propan-2-ol
Show/Hide
|
C27H30N4O3S
|
2
|
| 1 |
IC50 = 245 nM
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| 2 |
Ki = 18 nM
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CP0377715
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N-[4-[2-[[(2S)-2-hydroxy-3-(4-hydroxyphenoxy)propyl]amino]ethyl]phenyl]pentane-1-sulfonamide
Show/Hide
|
C22H32N2O5S
|
1
|
| 1 |
IC50 = 250 nM
|
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CP0374193
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1-(3-methoxyphenoxy)-3-(1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propan-2-ol
Show/Hide
|
C27H30N4O3S
|
2
|
| 1 |
IC50 = 250 nM
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|
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| 2 |
Ki = 30 nM
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CP0222316
|
1-{4-[2-((R)-2-Hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-3-[1-(4-octyl-thiazol-2-yl)-2,3-dihydro-1H-indol-5-yl]-thiourea
Show/Hide
|
C35H44N6OS2
|
1
|
| 1 |
IC50 = 260 nM
|
|
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CP0460262
|
4-Chloro-N-(4-{2-[(S)-2-hydroxy-3-(4-hydroxy-phenoxy)-propylamino]-ethyl}-phenyl)-benzenesulfonamide
Show/Hide
|
C23H25ClN2O5S
|
1
|
| 1 |
IC50 = 280 nM
|
|
|
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CP0160155
|
1-[4-[[4-[(6,7-dihydroxy-1,2,3,4-tetrahydroisoquinolin-1-yl)methoxy]phenyl]sulfamoyl]phenyl]-3-hexylurea
Show/Hide
|
C29H36N4O6S
|
1
|
| 1 |
IC50 = 300 nM
|
|
|
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CP0361078
|
1-[4-[[6-[(6,7-dihydroxy-1,2,3,4-tetrahydroisoquinolin-1-yl)methyl]naphthalen-2-yl]sulfamoyl]phenyl]-3-hexylurea
Show/Hide
|
C33H38N4O5S
|
1
|
| 1 |
IC50 = 300 nM
|
|
|
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CP0388516
|
4-(2-hydroxy-3-(1-(5-(thiophen-2-yl)thieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propoxy)phenol
Show/Hide
|
C24H26N4O3S2
|
2
|
| 1 |
IC50 = 327 nM
|
|
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| 2 |
Ki = 28 nM
|
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CP0258437
|
N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-(3-octyl-2-oxoimidazol-1-yl)benzenesulfonamide
Show/Hide
|
C32H41N5O4S
|
1
|
| 1 |
IC50 = 330 nM
|
|
|
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CP0460849
|
4-[(4-octyl-1,3-thiazol-2-yl)amino]-N-phenylbenzene-1-sulfonamide
Show/Hide
|
C23H29N3O2S2
|
1
|
| 1 |
IC50 = 340 nM
|
|
|
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CP0400965
|
3,4-Dichloro-N-(4-{2-[(S)-2-hydroxy-3-(pyridin-3-yloxy)-propylamino]-ethyl}-phenyl)-benzenesulfonamide
Show/Hide
|
C22H23Cl2N3O4S
|
1
|
| 1 |
IC50 = 360 nM
|
|
|
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CP0464054
|
3-Chloro-N-(4-{2-[(S)-2-hydroxy-3-(4-hydroxy-phenoxy)-propylamino]-ethyl}-phenyl)-benzenesulfonamide
Show/Hide
|
C23H25ClN2O5S
|
1
|
| 1 |
IC50 = 370 nM
|
|
|
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CP0714856
|
N-{4-[2-(2-Hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-4-(3-octyl-2,4-dioxo-imidazolidin-1-yl)-benzenesulfonamide
Show/Hide
|
C32H41N5O5S
|
1
|
| 1 |
IC50 = 370 nM
|
|
|
|
CP0688072
|
(R)-2-(2-{4-[1-(Naphthalen-1-ylamino)-2-nitro-vinylamino]-phenyl}-ethylamino)-1-pyridin-3-yl-ethanol
Show/Hide
|
C27H27N5O3
|
1
|
| 1 |
IC50 = 370 nM
|
|
|
|
CP0403004
|
N-[4-[2-[[(2S)-3-(6-aminopyridin-3-yl)oxy-2-hydroxypropyl]amino]ethyl]phenyl]-4-bromobenzenesulfonamide
Show/Hide
|
C22H25BrN4O4S
|
1
|
| 1 |
IC50 = 380 nM
|
|
|
|
CP0502498
|
N-[4-[2-[[(2S)-3-(6-aminopyridin-3-yl)oxy-2-hydroxypropyl]amino]ethyl]phenyl]-3,4-dichlorobenzenesulfonamide
Show/Hide
|
C22H24Cl2N4O4S
|
1
|
| 1 |
IC50 = 380 nM
|
|
|
|
CP0333214
|
N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-(3-octyl-2-oxoimidazolidin-1-yl)benzenesulfonamide
Show/Hide
|
C32H43N5O4S
|
1
|
| 1 |
IC50 = 380 nM
|
|
|
|
CP0404004
|
4-[4-(3-Fluoro-benzyl)-[1,2,3]triazol-2-yl]-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
|
C30H29FN6O3S
|
1
|
| 1 |
IC50 = 380 nM
|
|
|
|
CP0197394
|
3-[[N-cyano-N'-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]carbamimidoyl]amino]benzamide
Show/Hide
|
C24H25N7O2
|
1
|
| 1 |
IC50 = 400 nM
|
|
|
|
CP0373738
|
(R)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)biphenyl-3-carboxamide
Show/Hide
|
C28H27N3O2
|
1
|
| 1 |
IC50 = 400 nM
|
|
|
|
CP0428937
|
(R)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)-3-(1H-imidazol-2-yl)benzamide
Show/Hide
|
C25H25N5O2
|
1
|
| 1 |
IC50 = 400 nM
|
|
|
|
CP0428938
|
(R)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)-3-phenethylbenzamide
Show/Hide
|
C30H31N3O2
|
1
|
| 1 |
IC50 = 400 nM
|
|
|
|
CP0457339
|
N-[4-[2-[[(2S)-2-hydroxy-3-pyridin-3-yloxypropyl]amino]ethyl]phenyl]-4-propan-2-ylbenzenesulfonamide
Show/Hide
|
C25H31N3O4S
|
1
|
| 1 |
IC50 = 410 nM
|
|
|
|
CP0441620
|
1-[4-[[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]sulfamoyl]phenyl]-3-octylurea
Show/Hide
|
C30H41N5O4S
|
1
|
| 1 |
IC50 = 410 nM
|
|
|
|
CP0438071
|
4-(3-Hexyl-ureido)-N-(4-{2-[(S)-2-hydroxy-3-(pyridin-3-yloxy)-propylamino]-ethyl}-phenyl)-benzenesulfonamide
Show/Hide
|
C29H39N5O5S
|
1
|
| 1 |
IC50 = 430 nM
|
|
|
|
CP0466340
|
4-Chloro-N-(4-{2-[(S)-2-hydroxy-3-(pyridin-3-yloxy)-propylamino]-ethyl}-phenyl)-benzenesulfonamide
Show/Hide
|
C22H24ClN3O4S
|
1
|
| 1 |
IC50 = 430 nM
|
|
|
|
CP0448298
|
4-[methyl(4-octyl-1,3-thiazol-2-yl)amino]-N-phenylbenzene-1-sulfonamide
Show/Hide
|
C24H31N3O2S2
|
1
|
| 1 |
IC50 = 440 nM
|
|
|
|
CP0403534
|
1-[6-(3-cyclopentylpropyl)pyridin-2-yl]-N-phenyl-2,3-dihydro-1H-indole-5-sulfonamide
Show/Hide
|
C27H31N3O2S
|
1
|
| 1 |
IC50 = 450 nM
|
|
|
|
CP0409506
|
1-(3-hexylphenyl)-N-phenyl-2,3-dihydro-1H-indole-5-sulfonamide
Show/Hide
|
C26H30N2O2S
|
1
|
| 1 |
IC50 = 460 nM
|
|
|
|
CP0497049
|
N-[4-[2-[[(2S)-2-hydroxy-3-pyridin-3-yloxypropyl]amino]ethyl]phenyl]quinoline-3-sulfonamide
Show/Hide
|
C25H26N4O4S
|
1
|
| 1 |
IC50 = 490 nM
|
|
|
|
CP0431268
|
4-[5-(4-Fluoro-phenoxymethyl)-[1,2,4]oxadiazol-3-yl]-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
|
C30H28FN5O5S
|
1
|
| 1 |
IC50 = 490 nM
|
|
|
|
CP0405223
|
4-{(S)-3-[2-(4-Amino-phenyl)-ethylamino]-2-hydroxy-propoxy}-phenol
Show/Hide
|
C17H22N2O3
|
1
|
| 1 |
IC50 = 500 nM
|
|
|
|
CP0465353
|
N-[4-[2-[[(2S)-2-hydroxy-3-(4-hydroxyphenoxy)propyl]amino]ethyl]phenyl]propane-1-sulfonamide
Show/Hide
|
C20H28N2O5S
|
1
|
| 1 |
IC50 = 500 nM
|
|
|
|
CP0378009
|
1-(4-hexyl-1,3-thiazol-2-yl)-N-phenyl-2,3-dihydro-1H-indole-5-sulfonamide
Show/Hide
|
C23H27N3O2S2
|
1
|
| 1 |
IC50 = 510 nM
|
|
|
|
CP0454848
|
N-[4-[2-[[(2S)-2-hydroxy-3-pyridin-3-yloxypropyl]amino]ethyl]phenyl]-4-methoxybenzenesulfonamide
Show/Hide
|
C23H27N3O5S
|
1
|
| 1 |
IC50 = 520 nM
|
|
|
|
CP0429158
|
1-(4-octylpyrimidin-2-yl)-N-phenyl-2,3-dihydro-1H-indole-5-sulfonamide
Show/Hide
|
C26H32N4O2S
|
1
|
| 1 |
IC50 = 530 nM
|
|
|
|
CP0383033
|
N-[4-[2-[[(2S)-3-(6-aminopyridin-3-yl)oxy-2-hydroxypropyl]amino]ethyl]phenyl]-4-propan-2-ylbenzenesulfonamide
Show/Hide
|
C25H32N4O4S
|
1
|
| 1 |
IC50 = 540 nM
|
|
|
|
CP0498143
|
1-cyano-3-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-2-naphthalen-1-ylguanidine
Show/Hide
|
C27H26N6O
|
1
|
| 1 |
IC50 = 570 nM
|
|
|
|
CP0428931
|
(R)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)pyrazolo[1,5-a]pyridine-7-carboxamide
Show/Hide
|
C23H23N5O2
|
1
|
| 1 |
IC50 = 600 nM
|
|
|
|
CP0428936
|
(R)-3-(2-(1H-pyrrol-1-yl)ethyl)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)benzamide
Show/Hide
|
C28H30N4O2
|
1
|
| 1 |
IC50 = 600 nM
|
|
|
|
CP0422190
|
N-[4-[2-[[(2S)-3-(6-aminopyridin-3-yl)oxy-2-hydroxypropyl]amino]ethyl]phenyl]-4-methoxybenzenesulfonamide
Show/Hide
|
C23H28N4O5S
|
1
|
| 1 |
IC50 = 620 nM
|
|
|
|
CP0383247
|
1-(4-hexylpyrimidin-2-yl)-N-phenyl-2,3-dihydro-1H-indole-5-sulfonamide
Show/Hide
|
C24H28N4O2S
|
1
|
| 1 |
IC50 = 620 nM
|
|
|
|
CP0434375
|
4-(4-Hexyl-thiazol-2-yl)-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
|
C30H36N4O3S2
|
1
|
| 1 |
IC50 = 620 nM
|
|
|
|
CP0439361
|
N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-[4-[[4-(trifluoromethoxy)phenoxy]methyl]triazol-2-yl]benzenesulfonamide
Show/Hide
|
C31H29F3N6O5S
|
1
|
| 1 |
IC50 = 620 nM
|
|
|
|
CP0456599
|
N-[4-[2-[[(2S)-2-hydroxy-3-(4-hydroxyphenoxy)propyl]amino]ethyl]phenyl]naphthalene-2-sulfonamide
Show/Hide
|
C27H28N2O5S
|
1
|
| 1 |
IC50 = 630 nM
|
|
|
|
CP0437496
|
N-[4-[2-[[(2S)-3-(6-aminopyridin-3-yl)oxy-2-hydroxypropyl]amino]ethyl]phenyl]benzenesulfonamide
Show/Hide
|
C22H26N4O4S
|
1
|
| 1 |
IC50 = 630 nM
|
|
|
|
CP0393665
|
N-octyl-5-(phenylsulfamoyl)-2,3-dihydroindole-1-carboxamide
Show/Hide
|
C23H31N3O3S
|
1
|
| 1 |
IC50 = 630 nM
|
|
|
|
CP0461347
|
1-[4-[[4-[2-[[(2S)-3-(6-aminopyridin-3-yl)oxy-2-hydroxypropyl]amino]ethyl]phenyl]sulfamoyl]phenyl]-3-hexylurea
Show/Hide
|
C29H40N6O5S
|
1
|
| 1 |
IC50 = 640 nM
|
|
|
|
CP0496357
|
4-[5-(3-Cyclohexyl-propyl)-[1,2,4]oxadiazol-3-yl]-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
|
C32H39N5O4S
|
1
|
| 1 |
IC50 = 660 nM
|
|
|
|
CP0471480
|
4-[4-(3,4-Difluoro-phenoxymethyl)-[1,2,3]triazol-2-yl]-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
|
C30H28F2N6O4S
|
1
|
| 1 |
IC50 = 690 nM
|
|
|
|
CP0447792
|
4-[5-(3-Fluoro-benzyl)-[1,2,4]oxadiazol-3-yl]-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
|
C30H28FN5O4S
|
1
|
| 1 |
IC50 = 695 nM
|
|
|
|
CP0441818
|
1-[4-[[3-[3-[(6,7-dihydroxy-1,2,3,4-tetrahydroisoquinolin-1-yl)methyl]phenyl]phenyl]sulfamoyl]phenyl]-3-hexylurea
Show/Hide
|
C35H40N4O5S
|
1
|
| 1 |
IC50 = 710 nM
|
|
|
|
CP0381012
|
1-cyano-2-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-3-[1-[4-[4-(trifluoromethoxy)phenyl]-1,3-thiazol-2-yl]-2,3-dihydroindol-6-yl]guanidine
Show/Hide
|
C35H31F3N8O2S
|
1
|
| 1 |
IC50 = 710 nM
|
|
|
|
CP0492342
|
N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-[5-[(3,4,5-trifluorophenyl)methyl]-1,2,4-oxadiazol-3-yl]benzenesulfonamide
Show/Hide
|
C30H26F3N5O4S
|
1
|
| 1 |
IC50 = 720 nM
|
|
|
|
CP0392836
|
N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-(4-octyl-5-oxo-1,2,4-triazol-1-yl)benzenesulfonamide
Show/Hide
|
C31H40N6O4S
|
1
|
| 1 |
IC50 = 730 nM
|
|
|
|
CP0372587
|
N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-[4-[[4-(trifluoromethyl)phenoxy]methyl]triazol-2-yl]benzenesulfonamide
Show/Hide
|
C31H29F3N6O4S
|
1
|
| 1 |
IC50 = 730 nM
|
|
|
|
CP0422412
|
N-[4-[2-[[(2S)-2-hydroxy-3-pyridin-3-yloxypropyl]amino]ethyl]phenyl]benzenesulfonamide
Show/Hide
|
C22H25N3O4S
|
1
|
| 1 |
IC50 = 750 nM
|
|
|
|
CP0535177
|
1-(4-methyl-1,3-thiazol-2-yl)-N-phenyl-2,3-dihydro-1H-indole-5-sulfonamide
Show/Hide
|
C18H17N3O2S2
|
1
|
| 1 |
IC50 = 750 nM
|
|
|
|
CP0421070
|
4-[3-(3-Cyclopentyl-propyl)-2-oxo-imidazolidin-1-yl]-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
|
C32H41N5O4S
|
1
|
| 1 |
IC50 = 760 nM
|
|
|
|
CP0492821
|
4-[3-(3-Cyclopentyl-propyl)-2-oxo-2,3-dihydro-imidazol-1-yl]-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
|
C32H39N5O4S
|
1
|
| 1 |
IC50 = 760 nM
|
|
|
|
CP0391419
|
1-(3',4',5'-Trimethoxy-biphenyl-4-ylmethyl)-1,2,3,4-tetrahydro-isoquinoline-6,7-diol
Show/Hide
|
C25H27NO5
|
1
|
| 1 |
IC50 = 760 nM
|
|
|
|
CP0501622
|
4-[4-(2,3-Difluoro-phenyl)-thiazol-2-yl]-N-{4-[2-(2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
|
C30H26F2N4O3S2
|
1
|
| 1 |
IC50 = 760 nM
|
|
|
|
CP0376379
|
4-[4-(4-Fluoro-benzyl)-[1,2,3]triazol-2-yl]-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
|
C30H29FN6O3S
|
1
|
| 1 |
IC50 = 780 nM
|
|
|
|
CP0506110
|
(4-{4-[2-((R)-2-Hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenylsulfamoyl}-phenyl)-carbamic acid phenethyl ester
Show/Hide
|
C30H32N4O5S
|
1
|
| 1 |
IC50 = 820 nM
|
|
|
|
CP0424633
|
N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-[4-[[4-(trifluoromethoxy)phenyl]methyl]triazol-2-yl]benzenesulfonamide
Show/Hide
|
C31H29F3N6O4S
|
1
|
| 1 |
IC50 = 860 nM
|
|
|
|
CP0388524
|
1-phenoxy-3-(1-(thieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propan-2-ol
Show/Hide
|
C20H24N4O2S
|
2
|
| 1 |
IC50 = 862 nM
|
|
|
| 2 |
Ki = 189 nM
|
|
|
|
CP0495441
|
4-Fluoro-N-(4-{2-[(S)-2-hydroxy-3-(pyridin-3-yloxy)-propylamino]-ethyl}-phenyl)-benzenesulfonamide
Show/Hide
|
C22H24FN3O4S
|
1
|
| 1 |
IC50 = 900 nM
|
|
|
|
CP0402511
|
1-[4-(3-cyclopentylpropyl)-1,3-thiazol-2-yl]-N-phenyl-2,3-dihydro-1H-indole-5-sulfonamide
Show/Hide
|
C25H29N3O2S2
|
1
|
| 1 |
IC50 = 900 nM
|
|
|
|
CP0377145
|
N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-[4-(2-phenylethyl)-1,3-thiazol-2-yl]benzenesulfonamide
Show/Hide
|
C32H32N4O3S2
|
1
|
| 1 |
IC50 = 910 nM
|
|
|
|
CP0131163
|
1-cyano-3-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-2-[1-(4-octyl-1,3-thiazol-2-yl)-2,3-dihydroindol-4-yl]guanidine
Show/Hide
|
C36H44N8OS
|
1
|
| 1 |
IC50 = 930 nM
|
|
|
|
CP0461455
|
4-[5-(3-Cyclopentyl-propyl)-[1,2,4]oxadiazol-3-yl]-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
|
C31H37N5O4S
|
1
|
| 1 |
IC50 = 962 nM
|
|
|
|
CP0409613
|
4-[5-(3,4-Difluoro-benzyl)-[1,2,4]oxadiazol-3-yl]-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
|
C30H27F2N5O4S
|
1
|
| 1 |
IC50 = 980 nM
|
|
|
|
CP0486017
|
N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-[4-[3-(trifluoromethyl)phenyl]-1,3-thiazol-2-yl]benzenesulfonamide
Show/Hide
|
C31H27F3N4O3S2
|
1
|
| 1 |
IC50 = 980 nM
|
|
|
|
CP0503040
|
N-[4-[2-[[(2S)-3-(6-aminopyridin-3-yl)oxy-2-hydroxypropyl]amino]ethyl]phenyl]-4-chlorobenzenesulfonamide
Show/Hide
|
C22H25ClN4O4S
|
1
|
| 1 |
IC50 = 990 nM
|
|
|
|
CP0460293
|
1-[4-[[3-[4-[(6,7-dihydroxy-1,2,3,4-tetrahydroisoquinolin-1-yl)methoxy]phenyl]phenyl]sulfamoyl]phenyl]-3-hexylurea
Show/Hide
|
C35H40N4O6S
|
1
|
| 1 |
IC50 = 990 nM
|
|
|
|
CP0460042
|
N-[4-[2-[[(2S)-3-(6-aminopyridin-3-yl)oxy-2-hydroxypropyl]amino]ethyl]phenyl]-4-fluorobenzenesulfonamide
Show/Hide
|
C22H25FN4O4S
|
1
|
| 1 |
IC50 = 1000 nM
|
|
|
|
CP0404196
|
N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]naphthalene-2-sulfonamide
Show/Hide
|
C25H25N3O3S
|
1
|
| 1 |
IC50 = 1000 nM
|
|
|
|
CP0534841
|
N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]quinoline-3-sulfonamide
Show/Hide
|
C24H24N4O3S
|
1
|
| 1 |
IC50 = 1000 nM
|
|
|
|
CP0393663
|
1-nonanoyl-N-phenyl-2,3-dihydro-1H-indole-5-sulfonamide
Show/Hide
|
C23H30N2O3S
|
1
|
| 1 |
IC50 = 1000 nM
|
|
|
|
CP0529098
|
N-methyl-N-octyl-5-(phenylsulfamoyl)-2,3-dihydroindole-1-carboxamide
Show/Hide
|
C24H33N3O3S
|
1
|
| 1 |
IC50 = 1000 nM
|
|
|
|
CP0434368
|
4-[3-(3-Cyclohexyl-propyl)-2-oxo-imidazolidin-1-yl]-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
|
C33H43N5O4S
|
1
|
| 1 |
IC50 = 1000 nM
|
|
|
|
CP0480524
|
4-(3-Heptyl-2-oxo-imidazolidin-1-yl)-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
|
C31H41N5O4S
|
1
|
| 1 |
IC50 = 1000 nM
|
|
|
|
CP0528122
|
4-[3-(2-Cyclohexyl-ethyl)-2-oxo-imidazolidin-1-yl]-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
|
C32H41N5O4S
|
1
|
| 1 |
IC50 = 1000 nM
|
|
|
|
CP0395012
|
N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-[5-(4-methylpentyl)-1,2,4-oxadiazol-3-yl]benzenesulfonamide
Show/Hide
|
C29H35N5O4S
|
1
|
| 1 |
IC50 = 1000 nM
|
|
|
|
CP0422347
|
4-(5-Hexyl-[1,2,4]oxadiazol-3-yl)-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
|
C29H35N5O4S
|
1
|
| 1 |
IC50 = 1000 nM
|
|
|
|
CP0406380
|
N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-[(4-octyl-1,3-thiazol-2-yl)methyl]benzenesulfonamide
Show/Hide
|
C33H42N4O3S2
|
1
|
| 1 |
IC50 = 1000 nM
|
|
|
|
CP0451356
|
4-[4-(3,4-Difluoro-benzyl)-[1,2,3]triazol-2-yl]-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
|
C30H28F2N6O3S
|
1
|
| 1 |
IC50 = 1000 nM
|
|
|
|
CP0373727
|
(R)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)-1H-benzo[d]imidazole-2-carboxamide
Show/Hide
|
C23H23N5O2
|
1
|
| 1 |
IC50 = 1100 nM
|
|
|
|
CP0400357
|
(R)-2-(benzo[d]oxazol-2-yl)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)acetamide
Show/Hide
|
C24H24N4O3
|
1
|
| 1 |
IC50 = 1100 nM
|
|
|
|
CP0716783
|
3-(1-{4-[2-((R)-2-Hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenylamino}-2-nitro-vinylamino)-benzamide
Show/Hide
|
C24H26N6O4
|
1
|
| 1 |
IC50 = 1200 nM
|
|
|
|
CP0777882
|
(R)-2-(2-{4-[1-(3-Iodo-phenylamino)-2-nitro-vinylamino]-phenyl}-ethylamino)-1-pyridin-3-yl-ethanol
Show/Hide
|
C23H24IN5O3
|
1
|
| 1 |
IC50 = 1200 nM
|
|
|
|
CP0374199
|
1-(3-(2-hydroxy-3-(1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propoxy)phenyl)urea
Show/Hide
|
C27H30N6O3S
|
2
|
| 1 |
IC50 = 1280 nM
|
|
|
| 2 |
Ki = 139 nM
|
|
|
|
CP0383518
|
N-[4-[2-[[(2S)-3-(6-aminopyridin-3-yl)oxy-2-hydroxypropyl]amino]ethyl]phenyl]quinoline-3-sulfonamide
Show/Hide
|
C25H27N5O4S
|
1
|
| 1 |
IC50 = 1300 nM
|
|
|
|
CP0395300
|
1-(4-octyl-1,3-thiazol-2-yl)-N-phenyl-2,3-dihydro-1H-indole-5-sulfonamide
Show/Hide
|
C25H31N3O2S2
|
1
|
| 1 |
IC50 = 1300 nM
|
|
|
|
CP0376057
|
4-[4-(3,4-Difluoro-phenyl)-[1,2,3]triazol-2-yl]-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
|
C29H26F2N6O3S
|
1
|
| 1 |
IC50 = 1300 nM
|
|
|
|
CP0308845
|
1-(4-Octyl-thiazol-2-yl)-2,3-dihydro-1H-indole-5-sulfonic acid {4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-amide
Show/Hide
|
C34H43N5O3S2
|
1
|
| 1 |
IC50 = 1300 nM
|
|
|
|
CP0517113
|
4-(5-Heptyl-[1,2,4]oxadiazol-3-yl)-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
|
C30H37N5O4S
|
1
|
| 1 |
IC50 = 1415 nM
|
|
|
|
CP0399813
|
4-[5-(3,4-Difluoro-phenoxymethyl)-[1,2,4]oxadiazol-3-yl]-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
|
C30H27F2N5O5S
|
1
|
| 1 |
IC50 = 1430 nM
|
|
|
|
CP0374130
|
1-(3-octylphenyl)-N-phenyl-2,3-dihydro-1H-indole-5-sulfonamide
Show/Hide
|
C28H34N2O2S
|
1
|
| 1 |
IC50 = 1500 nM
|
|
|
|
CP0409587
|
4-{5-[(4-Fluoro-phenyl)-(3-methyl-ureido)-methyl]-[1,2,4]oxadiazol-3-yl}-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
|
C32H32FN7O5S
|
1
|
| 1 |
IC50 = 1500 nM
|
|
|
|
CP0414877
|
N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-[5-(naphthalen-2-ylmethyl)-1,2,4-oxadiazol-3-yl]benzenesulfonamide
Show/Hide
|
C34H31N5O4S
|
1
|
| 1 |
IC50 = 1500 nM
|
|
|
|
CP0498929
|
N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-[4-[4-(trifluoromethoxy)phenyl]triazol-2-yl]benzenesulfonamide
Show/Hide
|
C30H27F3N6O4S
|
1
|
| 1 |
IC50 = 1600 nM
|
|
|
|
CP0383690
|
4-[5-(4-Fluoro-benzyl)-[1,2,4]oxadiazol-3-yl]-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
|
C30H28FN5O4S
|
1
|
| 1 |
IC50 = 1660 nM
|
|
|
|
CP0373718
|
(R)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)-2-(4-phenylthiazol-2-yl)acetamide
Show/Hide
|
C26H26N4O2S
|
1
|
| 1 |
IC50 = 1700 nM
|
|
|
|
CP0428922
|
(R)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)-2-(2-phenylthiazol-4-yl)acetamide
Show/Hide
|
C26H26N4O2S
|
1
|
| 1 |
IC50 = 1700 nM
|
|
|
|
CP0428934
|
(R)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)-2-phenethylbenzamide
Show/Hide
|
C30H31N3O2
|
1
|
| 1 |
IC50 = 1700 nM
|
|
|
|
CP0377071
|
N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-[4-[2-(trifluoromethyl)phenyl]-1,3-thiazol-2-yl]benzenesulfonamide
Show/Hide
|
C31H27F3N4O3S2
|
1
|
| 1 |
IC50 = 1800 nM
|
|
|
|
CP0404462
|
4-[4-(4-Fluoro-phenyl)-thiazol-2-yl]-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
|
C30H27FN4O3S2
|
1
|
| 1 |
IC50 = 1900 nM
|
|
|
|
CP0496292
|
N-[4-[[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]sulfamoyl]phenyl]-4-phenylbutanamide
Show/Hide
|
C31H34N4O4S
|
1
|
| 1 |
IC50 = 2000 nM
|
|
|
|
CP0403724
|
1-heptanoyl-N-phenyl-2,3-dihydro-1H-indole-5-sulfonamide
Show/Hide
|
C21H26N2O3S
|
1
|
| 1 |
IC50 = 2000 nM
|
|
|
|
CP0537923
|
N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-(1-octyl-5-oxo-1,2,4-triazol-4-yl)benzenesulfonamide
Show/Hide
|
C31H40N6O4S
|
1
|
| 1 |
IC50 = 2000 nM
|
|
|
|
CP0661196
|
4-(3-Hexyl-2,4-dioxo-imidazolidin-1-yl)-N-{4-[2-(2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
|
C30H37N5O5S
|
1
|
| 1 |
IC50 = 2000 nM
|
|
|
|
CP0399960
|
N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-(3-methyl-2-oxoimidazolidin-1-yl)benzenesulfonamide
Show/Hide
|
C25H29N5O4S
|
1
|
| 1 |
IC50 = 2000 nM
|
|
|
|
CP0415378
|
4-{3-[3-(4-Chloro-phenyl)-propyl]-2-oxo-imidazolidin-1-yl}-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
|
C33H36ClN5O4S
|
1
|
| 1 |
IC50 = 2000 nM
|
|
|
|
CP0508553
|
N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-[2-oxo-3-(3-phenylpropyl)imidazolidin-1-yl]benzenesulfonamide
Show/Hide
|
C33H37N5O4S
|
1
|
| 1 |
IC50 = 2000 nM
|
|
|
|
CP0440071
|
4-{5-[Amino-(4-fluoro-phenyl)-methyl]-[1,2,4]oxadiazol-3-yl}-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
|
C30H29FN6O4S
|
1
|
| 1 |
IC50 = 2000 nM
|
|
|
|
CP0454745
|
N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-[5-[[4-(trifluoromethyl)phenyl]methyl]-1,2,4-oxadiazol-3-yl]benzenesulfonamide
Show/Hide
|
C31H28F3N5O4S
|
1
|
| 1 |
IC50 = 2000 nM
|
|
|
|
CP0402246
|
4-[4-(4-tert-Butyl-phenyl)-thiazol-2-yl]-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
|
C34H36N4O3S2
|
1
|
| 1 |
IC50 = 2000 nM
|
|
|
|
CP0460921
|
N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-[[4-(naphthalen-2-ylmethyl)-1,3-thiazol-2-yl]methyl]benzenesulfonamide
Show/Hide
|
C36H34N4O3S2
|
1
|
| 1 |
IC50 = 2000 nM
|
|
|
|
CP0421152
|
N-[4-[2-[4-[[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]sulfamoyl]phenyl]-1,3-thiazol-4-yl]phenyl]acetamide
Show/Hide
|
C32H31N5O4S2
|
1
|
| 1 |
IC50 = 2100 nM
|
|
|
|
CP0105792
|
4-(2-hydroxy-3-(1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propoxy)-2-(hydroxymethyl)phenol
Show/Hide
|
C27H30N4O4S
|
2
|
| 1 |
IC50 = 2250 nM
|
|
|
| 2 |
Ki = 14 nM
|
|
|
|
CP0309666
|
4-(3-Hexyl-2-oxo-imidazolidin-1-yl)-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
|
C30H39N5O4S
|
1
|
| 1 |
IC50 = 2300 nM
|
|
|
|
CP0499569
|
N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-[4-(naphthalen-2-ylmethyl)-1,3-thiazol-2-yl]benzenesulfonamide
Show/Hide
|
C35H32N4O3S2
|
1
|
| 1 |
IC50 = 2300 nM
|
|
|
|
CP0801117
|
(R)-2-(2-{4-[1-(3-Fluoro-phenylamino)-2-nitro-vinylamino]-phenyl}-ethylamino)-1-pyridin-3-yl-ethanol
Show/Hide
|
C23H24FN5O3
|
1
|
| 1 |
IC50 = 2400 nM
|
|
|
|
CP0856438
|
(R)-2-(4-Fluorophenyl)-N-(4-(((2S,5R)-5-((R)-hydroxy(pyridin-3-yl)methyl)pyrrolidin-2-yl)methyl)phenyl)-5,6-dihydro-4Hcyclopenta[d]thiazole-4-carboxamide
Show/Hide
|
C30H29FN4O2S
|
1
|
| 1 |
IC50 = 2471 nM
|
|
|
|
CP0429222
|
N-methyl-N-(2-phenylethyl)-5-(phenylsulfamoyl)-2,3-dihydroindole-1-carboxamide
Show/Hide
|
C24H25N3O3S
|
1
|
| 1 |
IC50 = 2500 nM
|
|
|
|
CP0461167
|
N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-(5-octyl-1,2,4-oxadiazol-3-yl)benzenesulfonamide
Show/Hide
|
C31H39N5O4S
|
1
|
| 1 |
IC50 = 2500 nM
|
|
|
|
CP0375247
|
4-{5-[(4-Fluoro-phenyl)-hydroxy-methyl]-[1,2,4]oxadiazol-3-yl}-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
|
C30H28FN5O5S
|
1
|
| 1 |
IC50 = 2500 nM
|
|
|
|
CP0399921
|
4-[3-(3,4-Difluoro-benzyl)-[1,2,4]oxadiazol-5-yl]-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
|
C30H27F2N5O4S
|
1
|
| 1 |
IC50 = 2500 nM
|
|
|
|
CP0416046
|
4-{5-[(4-Fluoro-phenyl)-methanesulfonylamino-methyl]-[1,2,4]oxadiazol-3-yl}-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
|
C31H31FN6O6S2
|
1
|
| 1 |
IC50 = 2500 nM
|
|
|
|
CP0502500
|
4-[5-(2-Hydroxy-phenoxymethyl)-[1,2,4]oxadiazol-3-yl]-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
|
C30H29N5O6S
|
1
|
| 1 |
IC50 = 2500 nM
|
|
|
|
CP0392506
|
4-[4-(4-Fluoro-benzyl)-thiazol-2-yl]-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
|
C31H29FN4O3S2
|
1
|
| 1 |
IC50 = 2500 nM
|
|
|
|
CP0384184
|
4-[4-(3-Fluoro-4-methoxy-phenyl)-[1,2,3]triazol-2-yl]-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
|
C30H29FN6O4S
|
1
|
| 1 |
IC50 = 2500 nM
|
|
|
|
CP0893925
|
(R)-2-(4-Fluorophenyl)-N-(4-(((2S,5R)-5-((R)-hydroxy(phenyl)-methyl)pyrrolidin-2-yl)methyl)phenyl)-5,6-dihydro-4Hcyclopenta[d]thiazole-4-carboxamide
Show/Hide
|
C31H30FN3O2S
|
1
|
| 1 |
IC50 = 2513 nM
|
|
|
|
CP0431336
|
4-[4-(2,4-Difluoro-phenyl)-thiazol-2-yl]-N-{4-[2-(2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
|
C30H26F2N4O3S2
|
1
|
| 1 |
IC50 = 2600 nM
|
|
|
|
CP0422182
|
4-[5-(2-Cyclopentyloxy-ethyl)-[1,2,4]oxadiazol-3-yl]-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
|
C30H35N5O5S
|
1
|
| 1 |
IC50 = 2667 nM
|
|
|
|
CP0403989
|
N-[4-[2-[[(2S)-2-hydroxy-3-(4-hydroxyphenoxy)propyl]amino]ethyl]phenyl]cyclohexanesulfonamide
Show/Hide
|
C23H32N2O5S
|
1
|
| 1 |
IC50 = 3000 nM
|
|
|
|
CP0432447
|
3,4-Dichloro-N-(4-{2-[(S)-2-hydroxy-3-(4-hydroxy-phenoxy)-propylamino]-ethyl}-phenyl)-benzenesulfonamide
Show/Hide
|
C23H24Cl2N2O5S
|
1
|
| 1 |
IC50 = 3000 nM
|
|
|
|
CP0279585
|
4-(3-Hexyl-ureido)-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
|
C28H37N5O4S
|
1
|
| 1 |
IC50 = 3000 nM
|
|
|
|
CP0430314
|
N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-(4-octyl-3,5-dioxo-1,2,4-triazolidin-1-yl)benzenesulfonamide
Show/Hide
|
C31H40N6O5S
|
1
|
| 1 |
IC50 = 3000 nM
|
|
|
|
CP0393943
|
N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-(5-pentyl-1,2,4-oxadiazol-3-yl)benzenesulfonamide
Show/Hide
|
C28H33N5O4S
|
1
|
| 1 |
IC50 = 3000 nM
|
|
|
|
CP0440078
|
N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-[5-[[4-(methanesulfonamido)phenyl]methyl]-1,2,4-oxadiazol-3-yl]benzenesulfonamide
Show/Hide
|
C31H32N6O6S2
|
1
|
| 1 |
IC50 = 3000 nM
|
|
|
|
CP0376537
|
N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-(4-pyridin-3-yl-1,3-thiazol-2-yl)benzenesulfonamide
Show/Hide
|
C29H27N5O3S2
|
1
|
| 1 |
IC50 = 3000 nM
|
|
|
|
CP0393166
|
N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-(4-octyl-1,3-thiazol-2-yl)benzenesulfonamide
Show/Hide
|
C32H40N4O3S2
|
1
|
| 1 |
IC50 = 3000 nM
|
|
|
|
CP0467467
|
4-[4-(3-Cyclopentyl-propyl)-thiazol-2-yl]-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
|
C32H38N4O3S2
|
1
|
| 1 |
IC50 = 3000 nM
|
|
|
|
CP0452934
|
(R)-2-cyclohexyl-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)benzamide
Show/Hide
|
C28H33N3O2
|
1
|
| 1 |
IC50 = 3000 nM
|
|
|
|
CP0412012
|
4-(3-(1-(5-(4-fluorophenyl)thieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)-2-hydroxypropoxy)phenol
Show/Hide
|
C26H27FN4O3S
|
2
|
| 1 |
IC50 = 3000 nM
|
|
|
| 2 |
Ki = 175 nM
|
|
|
|
CP0448510
|
1-[4-[[4-[4-[(6,7-dihydroxy-1,2,3,4-tetrahydroisoquinolin-1-yl)methyl]phenyl]phenyl]sulfamoyl]phenyl]-3-hexylurea
Show/Hide
|
C35H40N4O5S
|
1
|
| 1 |
IC50 = 3400 nM
|
|
|
|
CP0658182
|
(R)-2-(2-{4-[1-(Naphthalen-2-ylamino)-2-nitro-vinylamino]-phenyl}-ethylamino)-1-pyridin-3-yl-ethanol
Show/Hide
|
C27H27N5O3
|
1
|
| 1 |
IC50 = 3400 nM
|
|
|
|
CP0421068
|
4-[3-(3,4-Difluoro-benzyl)-2-oxo-imidazolidin-1-yl]-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
|
C31H31F2N5O4S
|
1
|
| 1 |
IC50 = 3500 nM
|
|
|
|
CP0453406
|
4-[3-(3,4-Difluoro-phenoxymethyl)-[1,2,4]oxadiazol-5-yl]-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
|
C30H27F2N5O5S
|
1
|
| 1 |
IC50 = 3500 nM
|
|
|
|
CP0490952
|
(R)-2-(3,5-diphenyl-1H-pyrazol-1-yl)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)acetamide
Show/Hide
|
C32H31N5O2
|
1
|
| 1 |
IC50 = 3600 nM
|
|
|
|
CP0506458
|
4-[3-(4-Fluoro-benzyl)-[1,2,4]oxadiazol-5-yl]-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
|
C30H28FN5O4S
|
1
|
| 1 |
IC50 = 4000 nM
|
|
|
|
CP0449007
|
N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-(4-pyridin-2-yl-1,3-thiazol-2-yl)benzenesulfonamide
Show/Hide
|
C29H27N5O3S2
|
1
|
| 1 |
IC50 = 4000 nM
|
|
|
|
CP0220943
|
4-(4-Hexyl-5-oxo-4,5-dihydro-[1,2,4]triazol-1-yl)-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
|
C29H36N6O4S
|
1
|
| 1 |
IC50 = 4500 nM
|
|
|
|
CP0375151
|
N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-[5-[(4-pyridin-2-ylphenyl)methyl]-1,2,4-oxadiazol-3-yl]benzenesulfonamide
Show/Hide
|
C35H32N6O4S
|
1
|
| 1 |
IC50 = 4500 nM
|
|
|
|
CP0447745
|
N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-[4-[[4-(trifluoromethyl)phenyl]methyl]triazol-2-yl]benzenesulfonamide
Show/Hide
|
C31H29F3N6O3S
|
1
|
| 1 |
IC50 = 4700 nM
|
|
|
|
CP0428935
|
(R)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)-2-(phenoxymethyl)benzamide
Show/Hide
|
C29H29N3O3
|
1
|
| 1 |
IC50 = 4700 nM
|
|
|
|
CP0438951
|
4-Bromo-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
|
C21H22BrN3O3S
|
1
|
| 1 |
IC50 = 5000 nM
|
|
|
|
CP0801317
|
N-{4-[2-(2-Hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-4-(3-octyl-2,5-dioxo-imidazolidin-1-yl)-benzenesulfonamide
Show/Hide
|
C32H41N5O5S
|
1
|
| 1 |
IC50 = 5000 nM
|
|
|
|
CP0420930
|
4-[3-(2,2-Dimethyl-hexyl)-2-oxo-imidazolidin-1-yl]-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
|
C32H43N5O4S
|
1
|
| 1 |
IC50 = 5000 nM
|
|
|
|
CP0464739
|
4-[3-(2-Cyclopentyl-ethyl)-2-oxo-imidazolidin-1-yl]-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
|
C31H39N5O4S
|
1
|
| 1 |
IC50 = 5000 nM
|
|
|
|
CP0524162
|
N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-(2-oxo-3-pentylimidazolidin-1-yl)benzenesulfonamide
Show/Hide
|
C29H37N5O4S
|
1
|
| 1 |
IC50 = 5000 nM
|
|
|
|
CP0380788
|
N-[4-[[3-[4-[[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]sulfamoyl]phenyl]-1,2,4-oxadiazol-5-yl]methyl]phenyl]acetamide
Show/Hide
|
C32H32N6O5S
|
1
|
| 1 |
IC50 = 5000 nM
|
|
|
|
CP0403739
|
N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-[5-[(4-methoxyphenoxy)methyl]-1,2,4-oxadiazol-3-yl]benzenesulfonamide
Show/Hide
|
C31H31N5O6S
|
1
|
| 1 |
IC50 = 5000 nM
|
|
|
|
CP0406150
|
N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-[5-[[4-(trifluoromethoxy)phenoxy]methyl]-1,2,4-oxadiazol-3-yl]benzenesulfonamide
Show/Hide
|
C31H28F3N5O6S
|
1
|
| 1 |
IC50 = 5000 nM
|
|
|
|
CP0419359
|
4-[4-(2,6-Difluoro-benzyl)-[1,2,3]triazol-2-yl]-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
|
C30H28F2N6O3S
|
1
|
| 1 |
IC50 = 5000 nM
|
|
|
|
CP0448737
|
N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-[4-(3,4,5-trifluorophenyl)-1,3-thiazol-2-yl]benzenesulfonamide
Show/Hide
|
C30H25F3N4O3S2
|
1
|
| 1 |
IC50 = 5000 nM
|
|
|
|
CP0100405
|
N-[(2-amino-1,3-thiazol-4-yl)methyl]-4-[[(2S,5R)-5-[(R)-hydroxy(phenyl)methyl]pyrrolidin-2-yl]methyl]benzamide
Show/Hide
|
C23H26N4O2S
|
1
|
| 1 |
IC50 = 5200 nM
|
|
|
|
CP0504031
|
4-(3-Butyl-2-oxo-imidazolidin-1-yl)-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
|
C28H35N5O4S
|
1
|
| 1 |
IC50 = 5300 nM
|
|
|
|
CP0373741
|
(R)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)-2-(pyrrolidin-1-yl)benzamide
Show/Hide
|
C26H30N4O2
|
1
|
| 1 |
IC50 = 5300 nM
|
|
|
|
CP0408753
|
methyl N-[(4-fluorophenyl)-[3-[4-[[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]sulfamoyl]phenyl]-1,2,4-oxadiazol-5-yl]methyl]carbamate
Show/Hide
|
C32H31FN6O6S
|
1
|
| 1 |
IC50 = 5400 nM
|
|
|
|
CP0483633
|
N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-[5-[[3-(trifluoromethoxy)phenyl]methyl]-1,2,4-oxadiazol-3-yl]benzenesulfonamide
Show/Hide
|
C31H28F3N5O5S
|
1
|
| 1 |
IC50 = 5500 nM
|
|
|
|
CP0377155
|
4-(2-hydroxy-3-(1-(5-methylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propoxy)phenol
Show/Hide
|
C21H26N4O3S
|
2
|
| 1 |
IC50 = 5500 nM
|
|
|
| 2 |
Ki = 2600 nM
|
|
|
|
CP0806796
|
(R)-2-(2-{4-[1-(3,5-Dichloro-phenylamino)-2-nitro-vinylamino]-phenyl}-ethylamino)-1-pyridin-3-yl-ethanol
Show/Hide
|
C23H23Cl2N5O3
|
1
|
| 1 |
IC50 = 5600 nM
|
|
|
|
CP0225356
|
8-[4-[[(2S,5R)-5-[(R)-hydroxy(phenyl)methyl]pyrrolidin-2-yl]methyl]benzoyl]-2-oxa-8-azaspiro[4.5]decan-1-one
Show/Hide
|
C27H32N2O4
|
1
|
| 1 |
IC50 = 5600 nM
|
|
|
|
CP0383394
|
4-[4-(4-Hydroxy-phenyl)-thiazol-2-yl]-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
|
C30H28N4O4S2
|
1
|
| 1 |
IC50 = 5700 nM
|
|
|
|
CP0460906
|
N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-propan-2-ylbenzenesulfonamide
Show/Hide
|
C24H29N3O3S
|
1
|
| 1 |
IC50 = 6000 nM
|
|
|
|
CP0373717
|
(R)-2-(1H-benzo[d]imidazol-2-yl)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)acetamide
Show/Hide
|
C24H25N5O2
|
1
|
| 1 |
IC50 = 6000 nM
|
|
|
|
CP0421404
|
N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-(4-naphthalen-2-yl-1,3-thiazol-2-yl)benzenesulfonamide
Show/Hide
|
C34H30N4O3S2
|
1
|
| 1 |
IC50 = 6300 nM
|
|
|
|
CP0383192
|
N-hexyl-N-methyl-5-(phenylsulfamoyl)-2,3-dihydroindole-1-carboxamide
Show/Hide
|
C22H29N3O3S
|
1
|
| 1 |
IC50 = 6500 nM
|
|
|
|
CP0095132
|
N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-[2-oxo-3-(4,4,4-trifluorobutyl)imidazolidin-1-yl]benzenesulfonamide
Show/Hide
|
C28H32F3N5O4S
|
1
|
| 1 |
IC50 = 6500 nM
|
|
|
|
CP0469997
|
4-(5-Butyl-[1,2,4]oxadiazol-3-yl)-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
|
C27H31N5O4S
|
1
|
| 1 |
IC50 = 6500 nM
|
|
|
|
CP0373723
|
N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-2-(2-oxo-4-phenylpyrrolidin-1-yl)acetamide
Show/Hide
|
C27H30N4O3
|
1
|
| 1 |
IC50 = 6700 nM
|
|
|
|
CP0428933
|
(R)-2-(2-(1H-pyrrol-1-yl)ethyl)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)benzamide
Show/Hide
|
C28H30N4O2
|
1
|
| 1 |
IC50 = 6900 nM
|
|
|
|
CP0484749
|
N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-iodobenzenesulfonamide
Show/Hide
|
C21H22IN3O3S
|
1
|
| 1 |
IC50 = 7000 nM
|
|
|
|
CP0448813
|
N,N-dimethyl-5-(phenylsulfamoyl)-2,3-dihydroindole-1-carboxamide
Show/Hide
|
C17H19N3O3S
|
1
|
| 1 |
IC50 = 7000 nM
|
|
|
|
CP0125773
|
N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-(4-methyl-3-octyl-2-oxoimidazol-1-yl)benzenesulfonamide
Show/Hide
|
C33H43N5O4S
|
1
|
| 1 |
IC50 = 7000 nM
|
|
|
|
CP0163835
|
4-(3-Hexyl-4-methyl-2-oxo-2,3-dihydro-imidazol-1-yl)-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
|
C31H39N5O4S
|
1
|
| 1 |
IC50 = 7000 nM
|
|
|
|
CP0122668
|
1-cyano-2-[6-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]naphthalen-2-yl]-3-[1-[4-[4-(trifluoromethoxy)phenyl]-1,3-thiazol-2-yl]-2,3-dihydroindol-5-yl]guanidine
Show/Hide
|
C39H33F3N8O2S
|
1
|
| 1 |
IC50 = 7100 nM
|
|
|
|
CP0378309
|
N-methyl-5-(phenylsulfamoyl)-2,3-dihydroindole-1-carboxamide
Show/Hide
|
C16H17N3O3S
|
1
|
| 1 |
IC50 = 7300 nM
|
|
|
|
CP0395094
|
1-[3-(3-cyclopentylpropyl)phenyl]-N-phenyl-2,3-dihydro-1H-indole-5-sulfonamide
Show/Hide
|
C28H32N2O2S
|
1
|
| 1 |
IC50 = 7500 nM
|
|
|
|
CP0403717
|
4-[3-(4-Fluoro-phenoxymethyl)-[1,2,4]oxadiazol-5-yl]-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
|
C30H28FN5O5S
|
1
|
| 1 |
IC50 = 7500 nM
|
|
|
|
CP0376678
|
N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-[5-[[4-(trifluoromethoxy)phenyl]methyl]-1,2,4-oxadiazol-3-yl]benzenesulfonamide
Show/Hide
|
C31H28F3N5O5S
|
1
|
| 1 |
IC50 = 7600 nM
|
|
|
|
CP0373724
|
(R)-2-(5,6-dimethyl-4-oxothieno[2,3-d]pyrimidin-3(4H)-yl)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)acetamide
Show/Hide
|
C25H27N5O3S
|
1
|
| 1 |
IC50 = 7800 nM
|
|
|
|
CP0484629
|
2-Phenyl-ethanesulfonic acid {4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-amide
Show/Hide
|
C23H27N3O3S
|
1
|
| 1 |
IC50 = 8000 nM
|
|
|
|
CP0505800
|
1-[4-[[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]sulfamoyl]phenyl]-3-methylurea
Show/Hide
|
C23H27N5O4S
|
1
|
| 1 |
IC50 = 8000 nM
|
|
|
|
CP0514433
|
1-[4-[[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]sulfamoyl]phenyl]-3-propylurea
Show/Hide
|
C25H31N5O4S
|
1
|
| 1 |
IC50 = 8000 nM
|
|
|
|
CP0518414
|
N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]benzenesulfonamide
Show/Hide
|
C21H23N3O3S
|
1
|
| 1 |
IC50 = 8000 nM
|
|
|
|
CP0438279
|
N-methyl-N-(2-methyl-1-phenylpropan-2-yl)-5-(phenylsulfamoyl)-2,3-dihydroindole-1-carboxamide
Show/Hide
|
C26H29N3O3S
|
1
|
| 1 |
IC50 = 8000 nM
|
|
|
|
CP0860176
|
N-{4-[2-((R)-2-Hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-4-{5-[4-(5H-tetrazol-5-yl)-phenoxymethyl]-[1,2,4]oxadiazol-3-yl}-benzenesulfonamide
Show/Hide
|
C31H29N9O5S
|
1
|
| 1 |
IC50 = 8000 nM
|
|
|
|
CP0480430
|
N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-(4-quinolin-6-yl-1,3-thiazol-2-yl)benzenesulfonamide
Show/Hide
|
C33H29N5O3S2
|
1
|
| 1 |
IC50 = 8000 nM
|
|
|
|
CP0765379
|
(R)-2-Amino-N-(4-(((2S,5R)-5-((R)-(3-chlorophenyl)(hydroxy)-methyl)pyrrolidin-2-yl)methyl)phenyl)-5,6-dihydro-4Hcyclopenta[d]thiazole-4-carboxamide
Show/Hide
|
C25H27ClN4O2S
|
1
|
| 1 |
IC50 = 8451 nM
|
|
|
|
CP0186827
|
4-(1-Hexyl-5-oxo-1,5-dihydro-[1,2,4]triazol-4-yl)-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
|
C29H36N6O4S
|
1
|
| 1 |
IC50 = 8500 nM
|
|
|
|
CP0463492
|
N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-(5-propyl-1,2,4-oxadiazol-3-yl)benzenesulfonamide
Show/Hide
|
C26H29N5O4S
|
1
|
| 1 |
IC50 = 8500 nM
|
|
|
|
CP0428928
|
(R)-2-(2-aminothiazol-4-yl)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)acetamide
Show/Hide
|
C20H23N5O2S
|
1
|
| 1 |
IC50 = 8700 nM
|
|
|
|
CP0404091
|
4-[4-(3-Fluoro-phenyl)-[1,2,3]triazol-2-yl]-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
|
C29H27FN6O3S
|
1
|
| 1 |
IC50 = 8800 nM
|
|
|
|
CP0432468
|
N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-[4-[(2,4,6-trifluorophenyl)methyl]triazol-2-yl]benzenesulfonamide
Show/Hide
|
C30H27F3N6O3S
|
1
|
| 1 |
IC50 = 8800 nM
|
|
|
|
CP0418526
|
N-[4-[[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]sulfamoyl]phenyl]pentanamide
Show/Hide
|
C26H32N4O4S
|
1
|
| 1 |
IC50 = 9000 nM
|
|
|
|
CP0193453
|
N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-[2-oxo-3-(4,4,5,5,5-pentafluoropentyl)imidazolidin-1-yl]benzenesulfonamide
Show/Hide
|
C29H32F5N5O4S
|
1
|
| 1 |
IC50 = 9000 nM
|
|
|
|
CP0495477
|
4-[4-(4-Fluoro-phenyl)-[1,2,3]triazol-2-yl]-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
|
C29H27FN6O3S
|
1
|
| 1 |
IC50 = 9300 nM
|
|
|
|
CP0440122
|
N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-[5-[(4-methylsulfanylphenyl)methyl]-1,2,4-oxadiazol-3-yl]benzenesulfonamide
Show/Hide
|
C31H31N5O4S2
|
1
|
| 1 |
IC50 = 9500 nM
|
|
|
|
CP0441693
|
N-[4-[[3-[4-[[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]sulfamoyl]phenyl]-1,2,4-oxadiazol-5-yl]methoxy]phenyl]acetamide
Show/Hide
|
C32H32N6O6S
|
1
|
| 1 |
IC50 = 9500 nM
|
|
|
|
CP0397752
|
4-Chloro-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
|
C21H22ClN3O3S
|
1
|
| 1 |
IC50 = 10000 nM
|
|
|
|
CP0441426
|
N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]methanesulfonamide
Show/Hide
|
C16H21N3O3S
|
1
|
| 1 |
IC50 = 10000 nM
|
|
|
|
CP0451013
|
N-[4-[[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]sulfamoyl]phenyl]octanamide
Show/Hide
|
C29H38N4O4S
|
1
|
| 1 |
IC50 = 10000 nM
|
|
|
|
CP0495089
|
(4-{4-[2-((R)-2-Hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenylsulfamoyl}-phenyl)-carbamic acid propyl ester
Show/Hide
|
C25H30N4O5S
|
1
|
| 1 |
IC50 = 10000 nM
|
|
|
|
CP0402512
|
3-hexyl-1-(4-{[4-(2-{[(2R)-2-hydroxy-2-(pyridin-3-yl)ethyl]amino}ethyl)phenyl]sulfamoyl}phenyl)-1-methylurea
Show/Hide
|
C29H39N5O4S
|
1
|
| 1 |
IC50 = 10000 nM
|
|
|
|
CP0431683
|
4-(4-Hexyl-3,5-dioxo-[1,2,4]triazolidin-1-yl)-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
|
C29H36N6O5S
|
1
|
| 1 |
IC50 = 10000 nM
|
|
|
|
CP0777212
|
4-(3-Hexyl-2,5-dioxo-imidazolidin-1-yl)-N-{4-[2-(2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
|
C30H37N5O5S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0392936
|
N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-[2-oxo-3-(4,4,4-trifluorobutyl)imidazol-1-yl]benzenesulfonamide
Show/Hide
|
C28H30F3N5O4S
|
1
|
| 1 |
IC50 = 10000 nM
|
|
|
|
CP0454640
|
N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-(5-methyl-1,2,4-oxadiazol-3-yl)benzenesulfonamide
Show/Hide
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C24H25N5O4S
|
1
|
| 1 |
IC50 = 10000 nM
|
|
|
|
CP0258480
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1-cyano-3-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-2-[1-[4-[4-(trifluoromethoxy)phenyl]-1,3-thiazol-2-yl]-2,3-dihydroindol-4-yl]guanidine
Show/Hide
|
C35H31F3N8O2S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
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CP0373722
|
(R)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)-2-(5-phenyl-4H-1,2,4-triazol-3-yl)acetamide
Show/Hide
|
C25H26N6O2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
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CP0373726
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(R)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)-2-(2H-indazol-2-yl)acetamide
Show/Hide
|
C24H25N5O2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
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CP0373729
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(R)-(1H-benzo[d]imidazol-2-yl)methyl 4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenylcarbamate
Show/Hide
|
C24H25N5O3
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0373743
|
(R)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)-2-(1H-imidazol-2-yl)benzamide
Show/Hide
|
C25H25N5O2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0373982
|
(R)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)-2-(4-oxoquinazolin-3(4H)-yl)acetamide
Show/Hide
|
C25H25N5O3
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0400358
|
(R)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)-2-(4-methylthiazol-2-yl)acetamide
Show/Hide
|
C21H24N4O2S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
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CP0428923
|
(R)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)-2-phenylacetamide
Show/Hide
|
C23H25N3O2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0428924
|
(R)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)-2-(2-oxoquinazolin-1(2H)-yl)acetamide
Show/Hide
|
C25H25N5O3
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0428927
|
(R)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)-2-(2-methylthiazol-4-yl)acetamide
Show/Hide
|
C21H24N4O2S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0429875
|
(R)-2-(1H-benzo[d]imidazol-2-yl)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)benzamide
Show/Hide
|
C29H27N5O2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0429887
|
(R)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)-2-(2H-1,2,3-triazol-2-yl)benzamide
Show/Hide
|
C24H24N6O2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0429905
|
(R)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)-2-(1H-indazol-3-yl)acetamide
Show/Hide
|
C24H25N5O2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0795225
|
1-(3-Thiophen-2-yl-phenyl)-ethanone, O-(phenylaminocarbonyl)oxime
Show/Hide
|
C19H16N2O2S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0231692
|
ethyl 1-[4-[[(2S,5R)-5-[(R)-hydroxy(phenyl)methyl]pyrrolidin-2-yl]methyl]benzoyl]piperidine-4-carboxylate
Show/Hide
|
C27H34N2O4
|
1
|
| 1 |
IC50 = 10900 nM
|
|
|
|
CP0452014
|
8-[4-[[(2S,5R)-5-[(R)-hydroxy(phenyl)methyl]pyrrolidin-2-yl]methyl]benzoyl]-3,3-dimethyl-2-oxa-8-azaspiro[4.5]decan-1-one
Show/Hide
|
C29H36N2O4
|
1
|
| 1 |
IC50 = 11000 nM
|
|
|
|
CP0277683
|
4-(3-Hexyl-2-oxo-2,3-dihydro-imidazol-1-yl)-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
|
C30H37N5O4S
|
1
|
| 1 |
IC50 = 12000 nM
|
|
|
|
CP0438564
|
N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-[5-(3-oxopentyl)-1,2,4-oxadiazol-3-yl]benzenesulfonamide
Show/Hide
|
C28H31N5O5S
|
1
|
| 1 |
IC50 = 12000 nM
|
|
|
|
CP0464804
|
4-[3-(3,4-Difluoro-benzyl)-2-oxo-2,3-dihydro-imidazol-1-yl]-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
|
C31H29F2N5O4S
|
1
|
| 1 |
IC50 = 13000 nM
|
|
|
|
CP0428926
|
(R)-2-(2H-benzo[d][1,2,3]triazol-2-yl)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)acetamide
Show/Hide
|
C23H24N6O2
|
1
|
| 1 |
IC50 = 13000 nM
|
|
|
|
CP0224385
|
ethyl (1S,5R)-3-[4-[[(2S,5R)-5-[(R)-hydroxy(phenyl)methyl]pyrrolidin-2-yl]methyl]benzoyl]-3-azabicyclo[3.1.0]hexane-6-carboxylate
Show/Hide
|
C27H32N2O4
|
1
|
| 1 |
IC50 = 13400 nM
|
|
|
|
CP0454388
|
4-[5-(4-Fluoro-benzoyl)-[1,2,4]oxadiazol-3-yl]-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
|
C30H26FN5O5S
|
1
|
| 1 |
IC50 = 15000 nM
|
|
|
|
CP0373746
|
(R)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)-5-methyl-2-(pyrrolidin-1-yl)benzamide
Show/Hide
|
C27H32N4O2
|
1
|
| 1 |
IC50 = 15000 nM
|
|
|
|
CP0417913
|
(R)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)-2-(1H-indazol-1-yl)acetamide
Show/Hide
|
C24H25N5O2
|
1
|
| 1 |
IC50 = 15000 nM
|
|
|
|
CP0377641
|
N-[5-[2-[4-[[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]sulfamoyl]phenyl]-1,3-thiazol-4-yl]pentyl]acetamide
Show/Hide
|
C31H37N5O4S2
|
1
|
| 1 |
IC50 = 16000 nM
|
|
|
|
CP0373736
|
(R)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)-2-(2-(methylamino)thiazol-4-yl)acetamide
Show/Hide
|
C21H25N5O2S
|
1
|
| 1 |
IC50 = 16000 nM
|
|
|
|
CP0430396
|
(R)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)-4-methyl-2-(pyrrolidin-1-yl)benzamide
Show/Hide
|
C27H32N4O2
|
1
|
| 1 |
IC50 = 16000 nM
|
|
|
|
CP0373719
|
(R)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)-2-(5-methyl-4H-1,2,4-triazol-3-yl)acetamide
Show/Hide
|
C20H24N6O2
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0373721
|
(R)-2-(3-amino-1H-1,2,4-triazol-1-yl)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)acetamide
Show/Hide
|
C19H23N7O2
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0373730
|
(R)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)-2-(1H-pyrazol-1-yl)acetamide
Show/Hide
|
C20H23N5O2
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0373731
|
(R)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)-2-(3-methyl-1H-pyrazol-1-yl)acetamide
Show/Hide
|
C21H25N5O2
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0373733
|
N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-2-pyrazol-1-ylpropanamide
Show/Hide
|
C21H25N5O2
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0373734
|
(R)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)-2-methyl-2-(1H-pyrazol-1-yl)propanamide
Show/Hide
|
C22H27N5O2
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0373735
|
2-(3,5-dimethyl-1H-pyrazol-1-yl)-N-(4-(2-((R)-2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)propanamide
Show/Hide
|
C23H29N5O2
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0373737
|
(R)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)biphenyl-2-carboxamide
Show/Hide
|
C28H27N3O2
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0373744
|
(R)-2-(benzo[d]thiazol-2-yl)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)benzamide
Show/Hide
|
C29H26N4O2S
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0373745
|
(R)-2-(furan-2-yl)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)benzamide
Show/Hide
|
C26H25N3O3
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0417833
|
(R)-2-(3,5-dimethyl-1H-pyrazol-1-yl)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)acetamide
Show/Hide
|
C22H27N5O2
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0417912
|
(R)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)-2,5-dimethylbenzamide
Show/Hide
|
C24H27N3O2
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0417917
|
2-(2-aminothiazol-4-yl)-N-(4-(2-((R)-2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)propanamide
Show/Hide
|
C21H25N5O2S
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0428929
|
(R)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)-2-(1H-1,2,4-triazol-1-yl)acetamide
Show/Hide
|
C19H22N6O2
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0428930
|
(R)-3-(1H-benzo[d]imidazol-2-yl)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)propanamide
Show/Hide
|
C25H27N5O2
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0428932
|
(R)-2-(2,5-dimethylthiazol-4-yl)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)acetamide
Show/Hide
|
C22H26N4O2S
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0429908
|
(R)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)-3-(1-methyl-1H-benzo[d]imidazol-2-yl)propanamide
Show/Hide
|
C26H29N5O2
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0447473
|
(R)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)-2-methylbenzamide
Show/Hide
|
C23H25N3O2
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0452933
|
(R)-2-(4,5-diphenyl-1H-pyrazol-1-yl)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)acetamide
Show/Hide
|
C32H31N5O2
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0845306
|
N-(4-(2-((R)-2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)-2-(1H-pyrazol-1-yl)propanamide hydrochloride
Show/Hide
|
C21H26ClN5O2
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0051719
|
2-(2-aminothiazol-4-yl)-N-(4-(((2S,5R)-5-((R)-hydroxy(phenyl)methyl)pyrrolidin-2-yl)methyl)phenyl)acetamide
Show/Hide
|
C23H26N4O2S
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0105651
|
(6S)-N-[4-[[(2S,5R)-5-[(R)-hydroxy(pyridin-3-yl)methyl]pyrrolidin-2-yl]methyl]phenyl]-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazole-6-carboxamide
Show/Hide
|
C24H27N5O2
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0135425
|
(4R)-N-[4-[[(2S,5R)-5-[(R)-hydroxy(pyridin-3-yl)methyl]pyrrolidin-2-yl]methyl]phenyl]-2-methyl-5,6-dihydro-4H-cyclopenta[d][1,3]thiazole-4-carboxamide
Show/Hide
|
C25H28N4O2S
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0135426
|
(4R)-N-[4-[[(2S,5R)-5-[(R)-hydroxy(pyridin-3-yl)methyl]pyrrolidin-2-yl]methyl]phenyl]-5,6-dihydro-4H-cyclopenta[d][1,3]thiazole-4-carboxamide
Show/Hide
|
C24H26N4O2S
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0135429
|
(4R)-2-amino-N-[4-[[(2S,5R)-5-[(R)-hydroxy(phenyl)methyl]pyrrolidin-2-yl]methyl]phenyl]-5,6-dihydro-4H-cyclopenta[d][1,3]thiazole-4-carboxamide
Show/Hide
|
C25H28N4O2S
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0699562
|
(R)-2-Amino-N-(4-(((2S,5R)-5-((R)-(3-fluorophenyl)(hydroxy)-methyl)pyrrolidin-2-yl)methyl)phenyl)-5,6-dihydro-4Hcyclopenta[d]thiazole-4-carboxamide
Show/Hide
|
C25H27FN4O2S
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0717837
|
(R)-2-Amino-N-(4-(((2S,5R)-5-((R)-(4-fluorophenyl)(hydroxy)-methyl)pyrrolidin-2-yl)methyl)phenyl)-5,6-dihydro-4Hcyclopenta[d]thiazole-4-carboxamide
Show/Hide
|
C25H27FN4O2S
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0869699
|
(R)-2-Ethyl-N-(4-(((2S,5R)-5-((R)-hydroxy(pyridin-3-yl)-methyl)pyrrolidin-2-yl)methyl)phenyl)-5,6-dihydro-4Hcyclopenta[d]thiazole-4-carboxamide
Show/Hide
|
C26H30N4O2S
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0869700
|
N-(4-(((2S,5R)-5-((R)-Hydroxy(pyridin-3-yl)methyl)pyrrolidin-2-yl)methyl)phenyl)-2-(1H-pyrazol-1-yl)acetamide
Show/Hide
|
C22H25N5O2
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0869756
|
(R)-2-(2-Aminothiazol-4-yl)-N-(4-(((2S,5R)-5-((R)-hydroxy-(phenyl)methyl)pyrrolidin-2-yl)methyl)phenyl)butanamide
Show/Hide
|
C25H30N4O2S
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0869757
|
(R)-2-Ethyl-N-(4-(((2S,5R)-5-((R)-hydroxy(phenyl)methyl)-pyrrolidin-2-yl)methyl)phenyl)-5,6-dihydro-4H-cyclopenta[d]-thiazole-4-carboxamide
Show/Hide
|
C27H31N3O2S
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0869758
|
(R)-2-(2-Aminothiazol-4-yl)-N-(4-(((2S,5R)-5-((R)-hydroxy-(phenyl)methyl)pyrrolidin-2-yl)methyl)phenyl)pentanamide
Show/Hide
|
C26H32N4O2S
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0869783
|
(R)-N-(4-(((2S,5R)-5-((R)-Hydroxy(phenyl)methyl)pyrrolidin-2-yl)methyl)phenyl)-2-methyl-5,6-dihydro-4H-cyclopenta[d]-thiazole-4-carboxamide
Show/Hide
|
C26H29N3O2S
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0869784
|
(R)-2-Cyclopropyl-N-(4-(((2S,5R)-5-((R)-hydroxy(pyridin-3-yl)-methyl)pyrrolidin-2-yl)methyl)phenyl)-5,6-dihydro-4Hcyclopenta[d]thiazole-4-carboxamide
Show/Hide
|
C27H30N4O2S
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0869787
|
(R)-2-Amino-N-(4-(((2S,5R)-5-((R)-hydroxy(phenyl)methyl)-pyrrolidin-2-yl)methyl)phenyl)-4,5,6,7-tetrahydrobenzo[d]-thiazole-4-carboxamide
Show/Hide
|
C26H30N4O2S
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0881853
|
(S)-2-(2-Aminothiazol-4-yl)-N-(4-(((2S,5R)-5-((R)-hydroxy(phenyl)methyl)pyrrolidin-2-yl)methyl)phenyl)-propanamide
Show/Hide
|
C24H28N4O2S
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0881856
|
(R)-2-(2-Aminothiazol-4-yl)-N-(4-(((2S,5R)-5-((R)-hydroxy-(phenyl)methyl)pyrrolidin-2-yl)methyl)phenyl)propanamide
Show/Hide
|
C24H28N4O2S
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0881884
|
(R)-2-Amino-N-(4-(((2S,5R)-5-((R)-hydroxy(pyridin-3-yl)-methyl)pyrrolidin-2-yl)methyl)phenyl)-5,6-dihydro-4Hcyclopenta[d]thiazole-4-carboxamide
Show/Hide
|
C24H27N5O2S
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0893924
|
(S)-N-(4-(((2S,5R)-5-((R)-Hydroxy(pyridin-3-yl)methyl)-pyrrolidin-2-yl)methyl)phenyl)-2-(1H-pyrazol-1-yl)-propanamide
Show/Hide
|
C23H27N5O2
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0901747
|
(R)-2-(2-Aminothiazol-4-yl)-N-(4-(((2S,5R)-5-((R)-hydroxy-(phenyl)methyl)pyrrolidin-2-yl)methyl)phenyl)-3-methylbutanamide
Show/Hide
|
C26H32N4O2S
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0903641
|
(R)-2-Amino-N-(4-(((2S,5R)-5-((R)-hydroxy(phenyl)methyl)-pyrrolidin-2-yl)methyl)phenyl)-5,6,7,8-tetrahydro-4Hcyclohepta[d]thiazole-4-carboxamide
Show/Hide
|
C27H32N4O2S
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0908527
|
(R)-N-(4-(((2S,5R)-5-((R)-Hydroxy(phenyl)methyl)pyrrolidin-2-yl)methyl)phenyl)-5,6-dihydro-4H-cyclopenta[d]thiazole-4-carboxamide
Show/Hide
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C25H27N3O2S
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1
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| 1 |
IC50 > 20000 nM
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CP0937943
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(S)-2-Amino-N-(4-(((2S,5R)-5-((R)-hydroxy(phenyl)methyl)-pyrrolidin-2-yl)methyl)phenyl)-5,6-dihydro-4H-cyclopenta[d]-thiazole-4-carboxamide
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C25H28N4O2S
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1
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| 1 |
IC50 > 20000 nM
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CP0148856
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[4-[[(2S,5R)-5-[(R)-hydroxy(phenyl)methyl]pyrrolidin-2-yl]methyl]phenyl]-[(1R,5S)-6-(2-methyltetrazol-5-yl)-3-azabicyclo[3.1.0]hexan-3-yl]methanone
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C26H30N6O2
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1
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| 1 |
IC50 > 20000 nM
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CP0203142
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(4-ethylsulfonylpiperidin-1-yl)-[4-[[(2S,5R)-5-[(R)-hydroxy(phenyl)methyl]pyrrolidin-2-yl]methyl]phenyl]methanone
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C26H34N2O4S
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1
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| 1 |
IC50 > 20000 nM
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CP0407116
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[4-[[(2S,5R)-5-[(R)-hydroxy(phenyl)methyl]pyrrolidin-2-yl]methyl]phenyl]-[(1R,5S)-6-(1,3,4-oxadiazol-2-yl)-3-azabicyclo[3.1.0]hexan-3-yl]methanone
Show/Hide
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C26H28N4O3
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1
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| 1 |
IC50 > 20000 nM
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CP0452015
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[(1R,5S)-6-(5-ethyl-1,3,4-oxadiazol-2-yl)-3-azabicyclo[3.1.0]hexan-3-yl]-[4-[[(2S,5R)-5-[(R)-hydroxy(phenyl)methyl]pyrrolidin-2-yl]methyl]phenyl]methanone
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C28H32N4O3
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1
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| 1 |
IC50 > 20000 nM
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CP0472576
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ethyl (1S,5R)-3-[4-[[(2S,5R)-5-[(R)-hydroxy(phenyl)methyl]pyrrolidin-2-yl]methyl]benzoyl]-3-azabicyclo[3.1.0]hexane-6-carboxylate
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C27H32N2O4
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1
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| 1 |
IC50 > 20000 nM
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CP0453458
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N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-[4-[4-(trifluoromethyl)phenyl]triazol-2-yl]benzenesulfonamide
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C30H27F3N6O3S
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1
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| 1 |
IC50 = 21000 nM
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CP0438779
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4-[5-(3-Hydroxy-pentyl)-[1,2,4]oxadiazol-3-yl]-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
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C28H33N5O5S
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1
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| 1 |
IC50 = 24000 nM
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CP0415331
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1-[4-[[3-[4-[(6,7-dihydroxy-1,2,3,4-tetrahydroisoquinolin-1-yl)methyl]phenyl]phenyl]sulfamoyl]phenyl]-3-hexylurea
Show/Hide
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C35H40N4O5S
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1
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| 1 |
IC50 = 32000 nM
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CP0488859
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N-hexyl-5-(phenylsulfamoyl)-2,3-dihydroindole-1-carboxamide
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C21H27N3O3S
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1
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| 1 |
IC50 = 36000 nM
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CP0497882
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4-[5-(4-Hydroxy-pentyl)-[1,2,4]oxadiazol-3-yl]-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
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C28H33N5O5S
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1
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| 1 |
IC50 = 44000 nM
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CP0399955
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N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-(4-quinolin-3-yl-1,3-thiazol-2-yl)benzenesulfonamide
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C33H29N5O3S2
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1
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| 1 |
IC50 = 47000 nM
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CP0492302
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4-(4-Benzofuran-2-yl-thiazol-2-yl)-N-{4-[2-(2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
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C32H28N4O4S2
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1
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| 1 |
IC50 = 49000 nM
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CP0480481
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N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]propane-2-sulfonamide
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C18H25N3O3S
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1
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| 1 |
IC50 = 50000 nM
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CP0415443
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N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-[3-(4-methoxybutyl)-2-oxoimidazolidin-1-yl]benzenesulfonamide
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C29H37N5O5S
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1
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| 1 |
IC50 = 50000 nM
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CP0383393
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N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-[4-(1H-indol-3-yl)-1,3-thiazol-2-yl]benzenesulfonamide
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C32H29N5O3S2
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1
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| 1 |
IC50 = 50000 nM
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CP0460764
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N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-[5-(3-oxo-3-pyrrolidin-1-ylpropyl)-1,2,4-oxadiazol-3-yl]benzenesulfonamide
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C30H34N6O5S
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1
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| 1 |
IC50 = 51000 nM
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CP0507494
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N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-[5-(4-oxopentyl)-1,2,4-oxadiazol-3-yl]benzenesulfonamide
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C28H31N5O5S
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1
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| 1 |
IC50 = 57000 nM
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CP0447728
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N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-[5-(naphthalen-2-yloxymethyl)-1,2,4-oxadiazol-3-yl]benzenesulfonamide
Show/Hide
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C34H31N5O5S
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1
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| 1 |
IC50 = 90000 nM
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CP0492498
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4-[4-(4-Hexyl-phenyl)-thiazol-2-yl]-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
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C36H40N4O3S2
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1
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| 1 |
IC50 = 90000 nM
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CP0455443
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4-(4-Benzo[b]thiophen-2-yl-thiazol-2-yl)-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
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C32H28N4O3S3
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1
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| 1 |
IC50 = 93000 nM
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CP0089815
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N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-[2-oxo-3-(3-oxo-3-pyrrolidin-1-ylpropyl)imidazolidin-1-yl]benzenesulfonamide
Show/Hide
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C31H38N6O5S
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1
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| 1 |
IC50 = 100000 nM
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CP0399931
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1-[4-[[6-[(6,7-dihydroxy-1,2,3,4-tetrahydroisoquinolin-1-yl)methoxy]naphthalen-2-yl]sulfamoyl]phenyl]-3-hexylurea
Show/Hide
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C33H38N4O6S
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1
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| 1 |
IC50 > 100000 nM
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CP0515960
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1-[4-[[4-[3-[(6,7-dihydroxy-1,2,3,4-tetrahydroisoquinolin-1-yl)methyl]phenyl]phenyl]sulfamoyl]phenyl]-3-hexylurea
Show/Hide
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C35H40N4O5S
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1
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| 1 |
IC50 = 100000 nM
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CP0378898
|
CAS_155346
Show/Hide
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C16H21N3O2
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1
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| 1 |
Kd = 0.7 nM
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CP0383039
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4-[3-(tert-butylamino)-2-hydroxypropoxy]-2,3-dihydro-1H-1,3-benzodiazol-2-one hydrochloride
Show/Hide
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C14H21N3O3
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1
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| 1 |
Kd = 19 nM
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CP0390295
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5-[3-(tert-butylamino)-2-hydroxypropoxy]-1,2,3,4-tetrahydronaphthalene-2,3-diol
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C17H27NO4
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1
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| 1 |
Kd = 70 nM
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CP0041613
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Anapriline
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C16H21NO2
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2
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| 1 |
Kd = 150 nM
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| 2 |
Ki = 0.32 nM
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CP0421581
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(2S,3S)-1-[(7-methyl-2,3-dihydro-1H-inden-4-yl)oxy]-3-(propan-2-ylamino)butan-2-ol
Show/Hide
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C17H27NO2
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1
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| 1 |
Kd = 630 nM
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CP0087906
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2-{4-[2-hydroxy-3-(propan-2-ylamino)propoxy]phenyl}acetamide
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C14H22N2O3
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1
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| 1 |
Kd = 1200 nM
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CP0065922
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4-[2-(tert-butylamino)-1-hydroxyethyl]-2-(hydroxymethyl)phenol
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C13H21NO3
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2
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| 1 |
Kd = 1400 nM
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| 2 |
Ki = 1828 nM
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CP0048177
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(2R,3R)-2,3-dihydroxysuccinic acid;1-(isopropylamino)-3-[4-(2-methoxyethyl)phenoxy]propan-2-ol
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C15H25NO3
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2
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| 1 |
Kd = 15500 nM
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| 2 |
Ki = 220 nM
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CP0192811
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Bisoprolol
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C18H31NO4
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2
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| 1 |
Kd = 33000 nM
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| 2 |
Ki = 250 nM
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CP0156994
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1-(9H-Carbazol-4-yloxy)-3-isopropylamino-propan-2-ol
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C18H22N2O2
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1
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| 1 |
Ki = 0.03 nM
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CP0384606
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(2S)-1-(9H-carbazol-4-yloxy)-3-[2-(2-methoxyphenoxy)ethylamino]propan-2-ol
Show/Hide
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C24H26N2O4
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2
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| 1 |
Ki = 0.03 nM
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| 2 |
Ki = 0.034 nM
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CP0567672
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(2S)-1-[2-[4-[3-(2-aminoethyldisulfanyl)propoxy]-3-methoxyphenyl]ethylamino]-3-naphthalen-1-yloxypropan-2-ol
Show/Hide
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C27H36N2O4S2
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1
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| 1 |
Ki = 0.073 nM
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CP0566044
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(2S)-1-[2-[4-[2-(2-aminoethyldisulfanyl)ethoxy]-3-methoxyphenyl]ethylamino]-3-naphthalen-1-yloxypropan-2-ol
Show/Hide
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C26H34N2O4S2
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1
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| 1 |
Ki = 0.16 nM
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CP0401112
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5-hydroxy-8-[(1R)-1-hydroxy-2-[2-[3-methoxy-4-(3-phenylpropoxy)phenyl]ethylamino]ethyl]-4H-1,4-benzoxazin-3-one
Show/Hide
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C28H32N2O6
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1
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| 1 |
Ki = 0.25 nM
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CP0217089
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1-[(3,5-diiodophenyl)methyl]-1,2,3,4-tetrahydroisoquinoline-6,7-diol
Show/Hide
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C16H15I2NO2
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1
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| 1 |
Ki = 0.302 nM
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CP0548583
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4-hydroxy-7-[(1R)-1-hydroxy-2-[[(1R,2R)-2-(2-phenylethyl)cyclopentyl]amino]ethyl]-3H-1,3-benzothiazol-2-one
Show/Hide
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C22H26N2O3S
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1
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| 1 |
Ki = 0.4 nM
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CP0399132
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8-hydroxy-5-[(1R)-1-hydroxy-2-[2-[3-methoxy-4-(3-phenylpropoxy)phenyl]ethylamino]ethyl]-1H-quinolin-2-one
Show/Hide
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C29H32N2O5
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1
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| 1 |
Ki = 0.48 nM
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CP0459850
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7-[(1R)-2-[[(1S,2R)-2-cyclopentylcyclopentyl]amino]-1-hydroxyethyl]-4-hydroxy-3H-1,3-benzothiazol-2-one
Show/Hide
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C19H26N2O3S
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1
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| 1 |
Ki = 0.6 nM
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CP0258990
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7-((R)-2-((cis)-bi(cyclopentan)-2-ylamino)-1-hydroxyethyl)-4-hydroxybenzo[d]thiazol-2(3H)-one
Show/Hide
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C19H26N2O3S
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1
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| 1 |
Ki = 0.8 nM
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CP0384610
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(2R)-1-(9H-carbazol-4-yloxy)-3-[2-(2-methoxyphenoxy)ethylamino]propan-2-ol
Show/Hide
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C24H26N2O4
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1
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| 1 |
Ki = 0.88 nM
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CP0533002
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(2R)-1-[2-[4-[3-(2-aminoethyldisulfanyl)propoxy]-3-methoxyphenyl]ethylamino]-3-naphthalen-1-yloxypropan-2-ol
Show/Hide
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C27H36N2O4S2
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1
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| 1 |
Ki = 1.1 nM
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CP0058651
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7-[(1R)-2-[2-(3-butylphenyl)ethylamino]-1-hydroxyethyl]-4-hydroxy-3H-1,3-benzothiazol-2-one
Show/Hide
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C21H26N2O3S
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1
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| 1 |
Ki = 1.4 nM
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CP0105976
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1-[(3,4,5-triiodophenyl)methyl]-1,2,3,4-tetrahydroisoquinoline-6,7-diol
Show/Hide
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C16H14I3NO2
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1
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| 1 |
Ki = 1.514 nM
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CP0078129
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1-[(4-amino-3,5-diiodophenyl)methyl]-1,2,3,4-tetrahydroisoquinoline-6,7-diol
Show/Hide
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C16H16I2N2O2
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1
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| 1 |
Ki = 1.549 nM
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CP0064477
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7-[(1R)-2-[2-(3-butoxyphenyl)ethylamino]-1-hydroxyethyl]-4-hydroxy-3H-1,3-benzothiazol-2-one
Show/Hide
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C21H26N2O4S
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1
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| 1 |
Ki = 1.7 nM
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CP0201486
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N-[4-[(6,7-dihydroxy-1,2,3,4-tetrahydroisoquinolin-1-yl)methyl]-2-iodophenyl]benzamide
Show/Hide
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C23H21IN2O3
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1
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| 1 |
Ki = 1.995 nM
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CP0093810
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7-[(1R)-2-[[(1R,2R)-2-cyclohexylcyclopentyl]amino]-1-hydroxyethyl]-4-hydroxy-3H-1,3-benzothiazol-2-one
Show/Hide
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C20H28N2O3S
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1
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| 1 |
Ki = 2 nM
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CP0039258
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TMQ, 3',5'-Diiodo
Show/Hide
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C17H17I2NO3
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1
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| 1 |
Ki = 2.042 nM
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CP0187238
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7-((R)-2-((1S,2S)-2-(benzyloxy)cyclopentylamino)-1-hydroxyethyl)-4-hydroxybenzo[d]thiazol-2(3H)-one
Show/Hide
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C21H24N2O4S
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1
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| 1 |
Ki = 2.5 nM
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CP0401110
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5-hydroxy-8-[2-[2-[3-methoxy-4-(3-phenylpropoxy)phenyl]ethylamino]ethyl]-4H-1,4-benzoxazin-3-one
Show/Hide
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C28H32N2O5
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1
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| 1 |
Ki = 2.8 nM
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CP0483868
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(S,R)-(-)-ethyl {4-[2-{[2-(3-bromoisoxazol-5-yl)-2-hydroxyethyl]amino}propyl]phenoxy} acetate
Show/Hide
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C18H23BrN2O5
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1
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| 1 |
Ki = 2.82 nM
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CP0315065
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5-[(1R)-1-hydroxy-2-[[(2R)-1-(4-methoxyphenyl)propan-2-yl]azaniumyl]ethyl]-2-oxo-1H-quinolin-8-olate
Show/Hide
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C21H24N2O4
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1
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| 1 |
Ki = 3.19 nM
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CP0520584
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(4-{(R)-2-[(R)-2-(3-Chloro-phenyl)-2-hydroxy-ethylamino]-propyl}-phenoxy)-acetic acid methyl ester
Show/Hide
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C20H24ClNO4
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1
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| 1 |
Ki = 3.2 nM
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CP0322398
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4-hydroxy-7-[(1R)-1-hydroxy-2-[2-(3-propylphenyl)ethylamino]ethyl]-3H-1,3-benzothiazol-2-one
Show/Hide
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C20H24N2O3S
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1
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| 1 |
Ki = 3.2 nM
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CP0384604
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(1R)-1-(9H-carbazol-4-yl)-2-[2-(2-methoxyphenoxy)ethylamino]ethanol
Show/Hide
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C23H24N2O3
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1
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| 1 |
Ki = 3.3 nM
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CP0418025
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(2R)-1-[2-[4-[2-(2-aminoethyldisulfanyl)ethoxy]-3-methoxyphenyl]ethylamino]-3-naphthalen-1-yloxypropan-2-ol
Show/Hide
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C26H34N2O4S2
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1
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| 1 |
Ki = 3.4 nM
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CP0517044
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7-[(1R)-2-[2-(4-butoxyphenyl)ethylamino]-1-hydroxyethyl]-4-hydroxy-3H-1,3-benzothiazol-2-one
Show/Hide
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C21H26N2O4S
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1
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| 1 |
Ki = 3.9 nM
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CP0435325
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1-phenoxy-3-(1-(5-(thiophen-2-yl)thieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propan-2-ol
Show/Hide
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C24H26N4O2S2
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1
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| 1 |
Ki = 4 nM
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CP0245845
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4-hydroxy-7-[(1R)-1-hydroxy-2-[[(1R,2R)-2-propan-2-ylcyclopentyl]amino]ethyl]-3H-1,3-benzothiazol-2-one
Show/Hide
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C17H24N2O3S
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1
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| 1 |
Ki = 4.2 nM
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CP0377225
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4-(2-hydroxy-3-(1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propoxy)-2-(methoxymethyl)phenol
Show/Hide
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C28H32N4O4S
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1
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| 1 |
Ki = 4.9 nM
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CP0384601
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3-(9H-carbazol-4-yloxy)-N-[2-(2-methoxyphenoxy)ethyl]propan-1-amine
Show/Hide
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C24H26N2O3
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1
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| 1 |
Ki = 5.4 nM
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CP0115242
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4-hydroxy-7-[(1R)-1-hydroxy-2-[[(1R,2R)-2-phenylcyclopentyl]amino]ethyl]-3H-1,3-benzothiazol-2-one
Show/Hide
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C20H22N2O3S
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1
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| 1 |
Ki = 5.5 nM
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CP0435332
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1-(2-allylphenoxy)-3-(1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propan-2-ol
Show/Hide
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C29H32N4O2S
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1
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| 1 |
Ki = 6 nM
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CP0401111
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8-hydroxy-5-[2-[2-[3-methoxy-4-(3-phenylpropoxy)phenyl]ethylamino]ethyl]-1H-quinolin-2-one
Show/Hide
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C29H32N2O4
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1
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| 1 |
Ki = 6.3 nM
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CP0079656
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1-[(4-amino-3-iodophenyl)methyl]-1,2,3,4-tetrahydroisoquinoline-6,7-diol
Show/Hide
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C16H17IN2O2
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1
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| 1 |
Ki = 6.457 nM
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CP0379809
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4-hydroxy-7-[(1R)-1-hydroxy-2-[2-[4-(2-methylpropyl)phenyl]ethylamino]ethyl]-3H-1,3-benzothiazol-2-one
Show/Hide
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C21H26N2O3S
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1
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| 1 |
Ki = 6.8 nM
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CP0406254
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3-ethyl-4-(2-hydroxy-3-(1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propoxy)phenol
Show/Hide
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C28H32N4O3S
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1
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| 1 |
Ki = 7 nM
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CP0463313
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4-hydroxy-7-[(1R)-1-hydroxy-2-[[(1R,2R)-2-(2-methylphenyl)cyclopentyl]amino]ethyl]-3H-1,3-benzothiazol-2-one
Show/Hide
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C21H24N2O3S
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1
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| 1 |
Ki = 7.1 nM
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CP0384602
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4-[(2S)-2-hydroxy-3-[2-[3-methoxy-4-(3-phenylpropoxy)phenyl]ethylamino]propoxy]benzene-1,2-diol
Show/Hide
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C27H33NO6
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1
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| 1 |
Ki = 7.2 nM
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CP0080005
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N-[4-[(6,7-dihydroxy-1,2,3,4-tetrahydroisoquinolin-1-yl)methyl]-2-iodophenyl]acetamide
Show/Hide
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C18H19IN2O3
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1
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| 1 |
Ki = 7.762 nM
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CP0272444
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N-[4-[(6,7-dihydroxy-1,2,3,4-tetrahydroisoquinolin-1-yl)methyl]-2,6-diiodophenyl]acetamide
Show/Hide
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C18H18I2N2O3
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1
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| 1 |
Ki = 8.71 nM
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CP0388489
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1-phenoxy-3-(1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propan-2-ol
Show/Hide
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C26H28N4O2S
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1
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| 1 |
Ki = 9 nM
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CP0229485
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(R)-1-(pyridin-3-yl)-2-(2-(4-(thiazol-4-yl)phenoxy)ethylamino)ethanol
Show/Hide
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C18H19N3O2S
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1
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| 1 |
Ki = 10 nM
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CP0378407
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(R)-2-(2-(4-(oxazol-4-yl)phenoxy)ethylamino)-1-(pyridin-3-yl)ethanol
Show/Hide
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C18H19N3O3
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1
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| 1 |
Ki = 10 nM
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CP0377223
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1-(2-isopropylphenoxy)-3-(1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propan-2-ol
Show/Hide
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C29H34N4O2S
|
1
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| 1 |
Ki = 10 nM
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CP0388475
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1-(3-ethylphenoxy)-3-(1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propan-2-ol
Show/Hide
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C28H32N4O2S
|
1
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| 1 |
Ki = 10 nM
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CP0469324
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2-ethyl-4-(2-hydroxy-3-(1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propoxy)phenol
Show/Hide
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C28H32N4O3S
|
1
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| 1 |
Ki = 11 nM
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CP0162255
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1-[(4-hydroxy-3,5-diiodophenyl)methyl]-1,2,3,4-tetrahydroisoquinoline-6,7-diol
Show/Hide
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C16H15I2NO3
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1
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| 1 |
Ki = 11.75 nM
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CP0093802
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7-[(1R)-2-[[(1R,2R)-2-(3-ethylphenyl)cyclopentyl]amino]-1-hydroxyethyl]-4-hydroxy-3H-1,3-benzothiazol-2-one
Show/Hide
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C22H26N2O3S
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1
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| 1 |
Ki = 12 nM
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CP0384608
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4-[(2S)-2-hydroxy-3-(propan-2-ylamino)propoxy]benzene-1,2-diol
Show/Hide
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C12H19NO4
|
1
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| 1 |
Ki = 12 nM
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CP0419868
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5-hydroxy-8-[(1S)-1-hydroxy-2-[2-[3-methoxy-4-(3-phenylpropoxy)phenyl]ethylamino]ethyl]-4H-1,4-benzoxazin-3-one
Show/Hide
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C28H32N2O6
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1
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| 1 |
Ki = 13 nM
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CP0439745
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(S,R)-(-)-{4-[2-{[2-(3-bromoisoxazol-5-yl)-2-hydroxyethyl]-amino}propyl]phenoxy}acetic acid
Show/Hide
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C16H19BrN2O5
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1
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| 1 |
Ki = 13.9 nM
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CP0388617
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1-phenoxy-3-(1-(thieno[3,2-d]pyrimidin-4-yl)piperidin-4-ylamino)propan-2-ol
Show/Hide
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C20H24N4O2S
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1
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| 1 |
Ki = 14 nM
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CP0123458
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4-hydroxy-7-[(1R)-1-hydroxy-2-[[(1R,2R)-2-(3-methylphenyl)cyclopentyl]amino]ethyl]-3H-1,3-benzothiazol-2-one
Show/Hide
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C21H24N2O3S
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1
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| 1 |
Ki = 15 nM
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CP0483832
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(S,R)-(-)-1-(3-bromoisoxazol-5-yl)-2-{[2-(4-butoxyphenyl)-1-methylethyl]amino}ethanol
Show/Hide
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C18H25BrN2O3
|
1
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| 1 |
Ki = 15.5 nM
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CP0384600
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4-[(1R)-1-hydroxy-2-[2-[3-methoxy-4-(3-phenylpropoxy)phenyl]ethylamino]ethyl]benzene-1,2-diol
Show/Hide
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C26H31NO5
|
1
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| 1 |
Ki = 18 nM
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CP0259163
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4-hydroxy-7-[(1R)-1-hydroxy-2-[2-(4-propylphenyl)ethylamino]ethyl]-3H-1,3-benzothiazol-2-one
Show/Hide
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C20H24N2O3S
|
1
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| 1 |
Ki = 19 nM
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CP0406244
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4-(2-hydroxy-3-(1-(5-(thiophen-2-yl)thieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propoxy)-2-(hydroxymethyl)phenol
Show/Hide
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C25H28N4O4S2
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1
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| 1 |
Ki = 20 nM
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CP0542944
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(2S)-1-[2-[4-[3-(2-aminoethyldisulfanyl)propoxy]-3-methoxyphenyl]ethylamino]-3-[4-(2-methoxyethyl)phenoxy]propan-2-ol
Show/Hide
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C26H40N2O5S2
|
1
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| 1 |
Ki = 20 nM
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CP0159295
|
8-Hydroxy-5-[(R)-1-hydroxy-2-(5,6-diethylindan-2-ylamino)-ethyl]-1H-quinolin-2-one
Show/Hide
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C24H28N2O3
|
2
|
| 1 |
Ki = 20.6 nM
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| 2 |
Ki = 76 nM
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CP0378414
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(R)-2-(2-(4-(2-methyloxazol-4-yl)phenoxy)ethylamino)-1-(pyridin-3-yl)ethanol
Show/Hide
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C19H21N3O3
|
1
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| 1 |
Ki = 21 nM
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CP0384701
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4-[(2S)-2-hydroxy-3-[2-(2-methoxyphenoxy)ethylamino]propoxy]benzene-1,2-diol
Show/Hide
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C18H23NO6
|
1
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| 1 |
Ki = 21 nM
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CP0399136
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8-hydroxy-5-[(1S)-1-hydroxy-2-[2-[3-methoxy-4-(3-phenylpropoxy)phenyl]ethylamino]ethyl]-1H-quinolin-2-one
Show/Hide
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C29H32N2O5
|
1
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| 1 |
Ki = 23 nM
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CP0091266
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N-[5-[(2S)-3-[[(1S)-1-(3,4-dimethoxyphenyl)-2-phenylethyl]amino]-2-hydroxypropyl]-2-hydroxyphenyl]methanesulfonamide
Show/Hide
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C26H32N2O6S
|
1
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| 1 |
Ki = 24 nM
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CP0406252
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4-(2-hydroxy-3-(1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propoxy)-3-(hydroxymethyl)phenol
Show/Hide
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C27H30N4O4S
|
1
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| 1 |
Ki = 25 nM
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CP0453931
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N-[5-[(2R)-3-[[(1S)-3-(3-chlorophenyl)-1-(3,4-dimethoxyphenyl)propyl]amino]-2-hydroxypropyl]-2-hydroxyphenyl]methanesulfonamide
Show/Hide
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C27H33ClN2O6S
|
1
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| 1 |
Ki = 26 nM
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CP0570008
|
2-(9H-carbazol-4-yl)-N-[2-(2-methoxyphenoxy)ethyl]ethanamine
Show/Hide
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C23H24N2O2
|
1
|
| 1 |
Ki = 26 nM
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CP0378409
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(R)-2-(2-(4-(2-(hydroxymethyl)oxazol-4-yl)phenoxy)ethylamino)-1-(pyridin-3-yl)ethanol
Show/Hide
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C19H21N3O4
|
1
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| 1 |
Ki = 30 nM
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CP0377222
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1-(3-fluorophenoxy)-3-(1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propan-2-ol
Show/Hide
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C26H27FN4O2S
|
1
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| 1 |
Ki = 30 nM
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CP0517045
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7-[(1R)-2-[2-(3,4-dimethylphenyl)ethylamino]-1-hydroxyethyl]-4-hydroxy-3H-1,3-benzothiazol-2-one
Show/Hide
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C19H22N2O3S
|
1
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| 1 |
Ki = 32 nM
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CP0295726
|
Procaterol
Show/Hide
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C16H22N2O3
|
1
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| 1 |
Ki = 33 nM
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CP0434384
|
(R)-2-(2-(4-(2-ethyloxazol-4-yl)phenoxy)ethylamino)-1-(pyridin-3-yl)ethanol
Show/Hide
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C20H23N3O3
|
1
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| 1 |
Ki = 37 nM
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CP0536378
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N-[5-[(2S)-3-[[(1R)-1-(3,4-dichlorophenyl)-2-phenylethyl]amino]-2-hydroxypropyl]-2-hydroxyphenyl]methanesulfonamide
Show/Hide
|
C24H26Cl2N2O4S
|
1
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| 1 |
Ki = 38 nM
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CP0377227
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3-(2-hydroxy-3-(1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propoxy)benzonitrile
Show/Hide
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C27H27N5O2S
|
1
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| 1 |
Ki = 42 nM
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CP0399131
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4-[(1S)-1-hydroxy-2-[2-[3-methoxy-4-(3-phenylpropoxy)phenyl]ethylamino]ethyl]benzene-1,2-diol
Show/Hide
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C26H31NO5
|
1
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| 1 |
Ki = 47 nM
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CP0378410
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(R)-2-(2-(4-(2-isopropyloxazol-4-yl)phenoxy)ethylamino)-1-(pyridin-3-yl)ethanol
Show/Hide
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C21H25N3O3
|
1
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| 1 |
Ki = 49 nM
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CP0492226
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(2S)-1-[2-[4-[2-(2-aminoethyldisulfanyl)ethoxy]-3-methoxyphenyl]ethylamino]-3-[4-(2-propan-2-yloxyethoxymethyl)phenoxy]propan-2-ol
Show/Hide
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C28H44N2O6S2
|
1
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| 1 |
Ki = 51 nM
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CP0399133
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4-[2-[2-[3-methoxy-4-(3-phenylpropoxy)phenyl]ethylamino]ethyl]benzene-1,2-diol
Show/Hide
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C26H31NO4
|
1
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| 1 |
Ki = 53 nM
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CP0374195
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1-(4-fluorophenoxy)-3-(1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propan-2-ol
Show/Hide
|
C26H27FN4O2S
|
1
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| 1 |
Ki = 55 nM
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CP0452776
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N-[5-[(2R)-3-[[(1S)-3-(2-chlorophenyl)-1-(3,4-dimethoxyphenyl)propyl]amino]-2-hydroxypropyl]-2-hydroxyphenyl]methanesulfonamide
Show/Hide
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C27H33ClN2O6S
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1
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| 1 |
Ki = 57 nM
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CP0542945
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(2S)-1-[2-[4-[2-(2-aminoethyldisulfanyl)ethoxy]-3-methoxyphenyl]ethylamino]-3-[4-(2-methoxyethyl)phenoxy]propan-2-ol
Show/Hide
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C25H38N2O5S2
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1
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| 1 |
Ki = 57 nM
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CP0309177
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N-[5-[(2S)-3-[[(1R)-1-(3,4-dimethoxyphenyl)-2-phenylethyl]amino]-2-hydroxypropyl]-2-hydroxyphenyl]methanesulfonamide
Show/Hide
|
C26H32N2O6S
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1
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| 1 |
Ki = 66 nM
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CP0388490
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1-(1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)-3-(3-(trifluoromethoxy)phenoxy)propan-2-ol
Show/Hide
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C27H27F3N4O3S
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1
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| 1 |
Ki = 68 nM
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CP0510848
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N-[5-[(2R)-3-[[(1S)-1-[3,4-bis(difluoromethoxy)phenyl]-3-phenylpropyl]amino]-2-hydroxypropyl]-2-hydroxyphenyl]methanesulfonamide
Show/Hide
|
C27H30F4N2O6S
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1
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| 1 |
Ki = 71 nM
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CP0377153
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1-(1-(5-methylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)-3-phenoxypropan-2-ol
Show/Hide
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C21H26N4O2S
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1
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| 1 |
Ki = 80 nM
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CP0374122
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4-(2-hydroxy-3-(1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propoxy)phenol
Show/Hide
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C26H28N4O3S
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1
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| 1 |
Ki = 81 nM
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CP0457725
|
(R,R)-(+)-ethyl {4-[2-{[2-(3-bromoisoxazol-5-yl)-2-hydroxyethyl]amino}propyl]phenoxy} acetate
Show/Hide
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C18H23BrN2O5
|
1
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| 1 |
Ki = 81.4 nM
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CP0388474
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1-(4-ethylphenoxy)-3-(1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propan-2-ol
Show/Hide
|
C28H32N4O2S
|
1
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| 1 |
Ki = 88 nM
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CP0388521
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1-(4-(hydroxymethyl)phenoxy)-3-(1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propan-2-ol
Show/Hide
|
C27H30N4O3S
|
1
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| 1 |
Ki = 93 nM
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CP0388613
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4-(2-hydroxy-3-(1-(5-methyl-6-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propoxy)-2-(hydroxymethyl)phenol
Show/Hide
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C28H32N4O4S
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1
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| 1 |
Ki = 94 nM
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CP0517043
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7-[(1R)-2-[[(1S,2S)-2-cyclohexylcyclopentyl]amino]-1-hydroxyethyl]-4-hydroxy-3H-1,3-benzothiazol-2-one
Show/Hide
|
C20H28N2O3S
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1
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| 1 |
Ki = 97 nM
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CP0384609
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4-[(1R)-1-hydroxy-2-[2-(2-methoxyphenoxy)ethylamino]ethyl]benzene-1,2-diol
Show/Hide
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C17H21NO5
|
1
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| 1 |
Ki = 97 nM
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CP0388603
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1-(1-(5-methyl-6-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)-3-phenoxypropan-2-ol
Show/Hide
|
C27H30N4O2S
|
1
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| 1 |
Ki = 100 nM
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CP0490367
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N-[5-[(2S)-3-[[(1R)-1-[3,4-bis(difluoromethoxy)phenyl]-2-phenylethyl]amino]-2-hydroxypropyl]-2-hydroxyphenyl]methanesulfonamide
Show/Hide
|
C26H28F4N2O6S
|
1
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| 1 |
Ki = 102 nM
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CP0375479
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2-(4-{(R)-2-[(R)-2-(3-Chloro-phenyl)-2-hydroxy-ethylamino]-propyl}-phenoxy)-N-hydroxy-acetamide
Show/Hide
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C19H23ClN2O4
|
1
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| 1 |
Ki = 112 nM
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CP0354617
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8-Hydroxy-5-[(R)-1-hydroxy-2-(5,6-di-n-butylindan-2-ylamino)-ethyl]-1H-quinolin-2-one
Show/Hide
|
C28H36N2O3
|
1
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| 1 |
Ki = 112 nM
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CP0388476
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N-[3-[2-hydroxy-3-[[1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-yl]amino]propoxy]phenyl]acetamide
Show/Hide
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C28H31N5O3S
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1
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| 1 |
Ki = 117 nM
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CP0128002
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8-Hydroxy-5-[(R)-1-hydroxy-2-(5,6-di-n-propylindan-2-ylamino)-ethyl]-1H-quinolin-2-one
Show/Hide
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C26H32N2O3
|
1
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| 1 |
Ki = 119 nM
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CP0309024
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(R)-2-(2-(4-(2-methylthiazol-4-yl)phenoxy)ethylamino)-1-(pyridin-3-yl)ethanol
Show/Hide
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C19H21N3O2S
|
1
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| 1 |
Ki = 120 nM
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CP0467205
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N-[5-[(2R)-3-[[(1S)-3-(4-chlorophenyl)-1-(3,4-dimethoxyphenyl)propyl]amino]-2-hydroxypropyl]-2-hydroxyphenyl]methanesulfonamide
Show/Hide
|
C27H33ClN2O6S
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1
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| 1 |
Ki = 120 nM
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CP0543720
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4-[(2R)-2-hydroxy-3-[2-[3-methoxy-4-(3-phenylpropoxy)phenyl]ethylamino]propoxy]benzene-1,2-diol
Show/Hide
|
C27H33NO6
|
1
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| 1 |
Ki = 120 nM
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CP0377150
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(3-(2-hydroxy-3-(1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propoxy)phenyl)(morpholino)methanone
Show/Hide
|
C31H35N5O4S
|
1
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| 1 |
Ki = 135 nM
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CP0517042
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4-hydroxy-7-[(1R)-1-hydroxy-2-[[(1R,2R)-2-(4-methylphenyl)cyclopentyl]amino]ethyl]-3H-1,3-benzothiazol-2-one
Show/Hide
|
C21H24N2O3S
|
1
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| 1 |
Ki = 149 nM
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CP0392741
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5-{2-[(R)-2-((S)-2-Hydroxy-3-phenoxy-propylamino)-propyl]-thiazol-5-yl}-pentanoic acid
Show/Hide
|
C20H28N2O4S
|
1
|
| 1 |
Ki = 150 nM
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CP0406256
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4-(2-hydroxy-3-(1-(thieno[3,2-d]pyrimidin-4-yl)piperidin-4-ylamino)propoxy)-2-(hydroxymethyl)phenol
Show/Hide
|
C21H26N4O4S
|
1
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| 1 |
Ki = 165 nM
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CP0498432
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2-(4-{(R)-2-[(R)-2-(3-Chloro-phenyl)-2-hydroxy-ethylamino]-propyl}-phenoxy)-acetamide
Show/Hide
|
C19H23ClN2O3
|
1
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| 1 |
Ki = 170 nM
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CP0473252
|
(1S)-1-(9H-carbazol-4-yl)-2-[2-(2-methoxyphenoxy)ethylamino]ethanol
Show/Hide
|
C23H24N2O3
|
1
|
| 1 |
Ki = 170 nM
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CP0452808
|
N-[2-hydroxy-5-[(2R)-2-hydroxy-3-[[(1S)-1-(3-methoxyphenyl)-3-phenylpropyl]amino]propyl]phenyl]methanesulfonamide
Show/Hide
|
C26H32N2O5S
|
1
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| 1 |
Ki = 200 nM
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CP0150288
|
8-Hydroxy-5-[(R)-1-hydroxy-2-(indan-2-ylamino)-ethyl]-1H-quinolin-2-one
Show/Hide
|
C20H20N2O3
|
1
|
| 1 |
Ki = 218 nM
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CP0469323
|
4-(2-hydroxy-3-(1-(5-methylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propoxy)-2-(hydroxymethyl)phenol
Show/Hide
|
C22H28N4O4S
|
1
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| 1 |
Ki = 223 nM
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CP0388503
|
5-(2-hydroxy-3-(1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propoxy)-2-(hydroxymethyl)phenol
Show/Hide
|
C27H30N4O4S
|
1
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| 1 |
Ki = 259 nM
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CP0416729
|
(R)-1-(3-Chloro-phenyl)-2-{(R)-2-[4-(2-hydroxy-ethoxy)-phenyl]-1-methyl-ethylamino}-ethanol
Show/Hide
|
C19H24ClNO3
|
1
|
| 1 |
Ki = 260 nM
|
|
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CP0448417
|
7-[(1R)-2-[[(1R,2R)-2-(3-ethoxyphenyl)cyclopentyl]amino]-1-hydroxyethyl]-4-hydroxy-3H-1,3-benzothiazol-2-one
Show/Hide
|
C22H26N2O4S
|
1
|
| 1 |
Ki = 266 nM
|
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CP0388612
|
4-(2-hydroxy-3-(1-(5-methyl-6-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propoxy)phenol
Show/Hide
|
C27H30N4O3S
|
1
|
| 1 |
Ki = 270 nM
|
|
|
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CP0453908
|
N-[2-hydroxy-5-[(2R)-2-hydroxy-3-[[(1S)-1-(4-methoxyphenyl)-3-phenylpropyl]amino]propyl]phenyl]methanesulfonamide
Show/Hide
|
C26H32N2O5S
|
1
|
| 1 |
Ki = 280 nM
|
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CP0470971
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(2R)-1-[2-[4-[3-(2-aminoethyldisulfanyl)propoxy]-3-methoxyphenyl]ethylamino]-3-[4-(2-methoxyethyl)phenoxy]propan-2-ol
Show/Hide
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C26H40N2O5S2
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1
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| 1 |
Ki = 320 nM
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CP0224884
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8-Hydroxy-5-[(R)-1-hydroxy-2-(5,6-dimethoxyindan-2-ylamino)-ethyl]-1H-quinolin-2-one
Show/Hide
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C22H24N2O5
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1
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| 1 |
Ki = 342 nM
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CP0535407
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N-[2-hydroxy-5-[(2S)-2-hydroxy-3-[[(1R)-1-(3-methoxyphenyl)-2-phenylethyl]amino]propyl]phenyl]methanesulfonamide
Show/Hide
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C25H30N2O5S
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1
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| 1 |
Ki = 350 nM
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CP0042352
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2,3-bis(oxidanyl)butanedioic acid;4-[(1R)-2-(methylamino)-1-oxidanyl-ethyl]benzene-1,2-diol
Show/Hide
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C9H13NO3
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1
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| 1 |
Ki = 360 nM
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CP0412043
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3-(2-hydroxy-3-(1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propoxy)-N-methylbenzamide
Show/Hide
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C28H31N5O3S
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1
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| 1 |
Ki = 370 nM
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CP0538610
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N-[5-[(2R)-3-[[(1S)-1-(3,4-dimethoxyphenyl)-3-phenylpropyl]amino]-2-hydroxypropyl]-2-hydroxyphenyl]methanesulfonamide
Show/Hide
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C27H34N2O6S
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1
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| 1 |
Ki = 390 nM
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CP0533400
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4-[(2R)-2-hydroxy-3-(propan-2-ylamino)propoxy]benzene-1,2-diol
Show/Hide
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C12H19NO4
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1
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| 1 |
Ki = 420 nM
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CP0406249
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4-(2-hydroxy-3-(1-(thieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propoxy)-2-(hydroxymethyl)phenol
Show/Hide
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C21H26N4O4S
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1
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| 1 |
Ki = 440 nM
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CP0454267
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(R,R)-(+)-1-(3-bromoisoxazol-5-yl)-2-{[2-(4-butoxyphenyl)-1-methylethyl]amino}ethanol
Show/Hide
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C18H25BrN2O3
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1
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| 1 |
Ki = 458 nM
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CP0378402
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(R)-2-(2-(4-(2-phenylthiazol-4-yl)phenoxy)ethylamino)-1-(pyridin-3-yl)ethanol
Show/Hide
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C24H23N3O2S
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1
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| 1 |
Ki = 500 nM
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CP0501137
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(R,R)-(+)-{4-[2-{[2-(3-bromoisoxazol-5-yl)-2-hydroxyethyl]-amino}propyl]phenoxy}acetic acid
Show/Hide
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C16H19BrN2O5
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1
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| 1 |
Ki = 501 nM
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CP0457458
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N-[2-hydroxy-5-[(2S)-2-hydroxy-3-[[(1R)-1-(4-methoxyphenyl)-2-phenylethyl]amino]propyl]phenyl]methanesulfonamide
Show/Hide
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C25H30N2O5S
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1
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| 1 |
Ki = 510 nM
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CP0472738
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4-hydroxy-2-(2-hydroxy-3-(1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propoxy)benzoic acid
Show/Hide
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C27H28N4O5S
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1
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| 1 |
Ki = 517 nM
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CP0122545
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8-Hydroxy-5-[(R)-1-hydroxy-2-(5,6-dimethylindan-2-ylamino)-ethyl]-1H-quinolin-2-one
Show/Hide
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C22H24N2O3
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1
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| 1 |
Ki = 522 nM
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CP0388618
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4-(2-hydroxy-3-(1-(thieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propoxy)phenol
Show/Hide
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C20H24N4O3S
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1
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| 1 |
Ki = 589 nM
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CP0399135
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4-[2-[2-(2-methoxyphenoxy)ethylamino]ethyl]benzene-1,2-diol
Show/Hide
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C17H21NO4
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1
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| 1 |
Ki = 610 nM
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CP0403859
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4-[(3,4,5-trimethoxyphenyl)methyl]-4,5,6,7-tetrahydro-[1,3]thiazolo[5,4-c]pyridin-2-amine
Show/Hide
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C16H21N3O3S
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1
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| 1 |
Ki = 616.6 nM
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CP0224883
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8-Hydroxy-5-[(R)-1-hydroxy-2-(4,7-diethylindan-2-ylamino)-ethyl]-1H-quinolin-2-one
Show/Hide
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C24H28N2O3
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1
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| 1 |
Ki = 692 nM
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CP0388508
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1-(4-methoxyphenoxy)-3-(1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propan-2-ol
Show/Hide
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C27H30N4O3S
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1
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| 1 |
Ki = 700 nM
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CP0384605
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4-[3-[2-[3-methoxy-4-(3-phenylpropoxy)phenyl]ethylamino]propoxy]benzene-1,2-diol
Show/Hide
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C27H33NO5
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1
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| 1 |
Ki = 700 nM
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CP0533398
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4-[(2S)-2-hydroxy-3-[2-(2-methoxyphenoxy)ethylamino]propyl]benzene-1,2-diol
Show/Hide
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C18H23NO5
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1
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| 1 |
Ki = 740 nM
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CP0333937
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N-[5-[(2R)-3-[[(1S)-1-(3,4-dimethoxyphenyl)-2-phenylethyl]amino]-2-hydroxypropyl]-2-hydroxyphenyl]methanesulfonamide
Show/Hide
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C26H32N2O6S
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1
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| 1 |
Ki = 820 nM
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CP0399134
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4-[(1S)-1-hydroxy-2-[2-(2-methoxyphenoxy)ethylamino]ethyl]benzene-1,2-diol
Show/Hide
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C17H21NO5
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1
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| 1 |
Ki = 850 nM
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CP0377224
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4-(2-hydroxy-3-(1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propoxy)benzene-1,2-diol
Show/Hide
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C26H28N4O4S
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1
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| 1 |
Ki = 873 nM
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CP0479748
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4-[3-[2-(2-methoxyphenoxy)ethylamino]propyl]benzene-1,2-diol
Show/Hide
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C18H23NO4
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1
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| 1 |
Ki = 920 nM
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CP0472744
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4-(2-hydroxy-3-(1-(thieno[3,2-d]pyrimidin-4-yl)piperidin-4-ylamino)propoxy)phenol
Show/Hide
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C20H24N4O3S
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1
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| 1 |
Ki = 961 nM
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CP0378904
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2-hydroxy-5-{2-[(2-hydroxy-3-{4-[1-methyl-4-(trifluoromethyl)-1H-imidazol-2-yl]phenoxy}propyl)amino]ethoxy}benzamide; methanesulfonic acid
Show/Hide
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C23H25F3N4O5
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1
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| 1 |
Ki = 1000 nM
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CP0461704
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N-[2-hydroxy-5-[(2S)-2-hydroxy-3-[[(1R)-1-(3-hydroxy-4-methoxyphenyl)-2-phenylethyl]amino]propyl]phenyl]methanesulfonamide
Show/Hide
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C25H30N2O6S
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1
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| 1 |
Ki = 1070 nM
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CP0480559
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3-{2-[(R)-2-((S)-2-Hydroxy-3-phenoxy-propylamino)-propyl]-thiazol-5-yl}-propionic acid
Show/Hide
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C18H24N2O4S
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1
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| 1 |
Ki = 1230 nM
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CP0492227
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(2R)-1-[2-[4-[2-(2-aminoethyldisulfanyl)ethoxy]-3-methoxyphenyl]ethylamino]-3-[4-(2-methoxyethyl)phenoxy]propan-2-ol
Show/Hide
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C25H38N2O5S2
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1
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| 1 |
Ki = 1300 nM
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CP0533517
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2-[3-(2-aminoethyldisulfanyl)propoxy]-5-[2-[[(2S)-2-hydroxy-3-[4-[1-methyl-4-(trifluoromethyl)imidazol-2-yl]phenoxy]propyl]amino]ethoxy]benzamide
Show/Hide
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C28H36F3N5O5S2
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1
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| 1 |
Ki = 1400 nM
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CP0364380
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N-[5-[(2R)-3-[[(1R)-1-(3,4-dimethoxyphenyl)-2-phenylethyl]amino]-2-hydroxypropyl]-2-hydroxyphenyl]methanesulfonamide
Show/Hide
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C26H32N2O6S
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1
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| 1 |
Ki = 1500 nM
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CP0373483
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4-{2-[(R)-2-((S)-2-Hydroxy-3-phenoxy-propylamino)-propyl]-thiazol-5-yl}-butyric acid
Show/Hide
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C19H26N2O4S
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1
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| 1 |
Ki = 1600 nM
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CP0533001
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2-[2-(2-aminoethyldisulfanyl)ethoxy]-5-[2-[[(2S)-2-hydroxy-3-[4-[1-methyl-4-(trifluoromethyl)imidazol-2-yl]phenoxy]propyl]amino]ethoxy]benzamide
Show/Hide
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C27H34F3N5O5S2
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1
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| 1 |
Ki = 2000 nM
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CP0396810
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(2S)-1-[2-[4-[2-(2-aminoethyldisulfanyl)ethoxy]-3-methoxyphenyl]ethylamino]-3-[4-[1-methyl-4-(trifluoromethyl)imidazol-2-yl]phenoxy]propan-2-ol
Show/Hide
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C27H35F3N4O4S2
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1
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| 1 |
Ki = 2200 nM
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CP0144828
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(4-{(R)-2-[(R)-2-(3-Chloro-phenyl)-2-hydroxy-ethylamino]-propyl}-phenoxy)-methanesulfonic acid
Show/Hide
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C18H22ClNO5S
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1
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| 1 |
Ki = 2250 nM
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CP0388359
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N-[3-[(5-chloro-6-oxo-4-piperazin-1-ylpyridazin-1-yl)methyl]phenyl]-4-phenylbenzamide
Show/Hide
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C28H26ClN5O2
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1
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| 1 |
Ki = 2290.87 nM
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CP0440458
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2-[4-[2-[[(2S)-2-hydroxy-3-phenoxypropyl]amino]ethoxy]phenoxy]acetic acid
Show/Hide
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C19H23NO6
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1
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| 1 |
Ki = 2350 nM
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CP0399906
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N-[5-[(5-chloro-6-oxo-4-piperazin-1-ylpyridazin-1-yl)methyl]-2-methylphenyl]-4-phenylbenzamide
Show/Hide
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C29H28ClN5O2
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1
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| 1 |
Ki = 2398.83 nM
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CP0333936
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N-[2-hydroxy-5-[(2R)-2-hydroxy-3-[[(1R)-1-(3-methoxyphenyl)-2-phenylethyl]amino]propyl]phenyl]methanesulfonamide
Show/Hide
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C25H30N2O5S
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1
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| 1 |
Ki = 2700 nM
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CP0490366
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N-[2-hydroxy-5-[(2R)-2-hydroxy-3-[[(1R)-1-(4-methoxyphenyl)-2-phenylethyl]amino]propyl]phenyl]methanesulfonamide
Show/Hide
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C25H30N2O5S
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1
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| 1 |
Ki = 3100 nM
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CP0039930
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(-)-arterenol
Show/Hide
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C8H11NO3
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1
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| 1 |
Ki = 3300 nM
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CP0567612
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4-[3-[2-(2-methoxyphenoxy)ethylamino]propoxy]benzene-1,2-diol
Show/Hide
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C18H23NO5
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1
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| 1 |
Ki = 3800 nM
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CP0046448
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1-[[3,5-bis(trifluoromethyl)phenyl]methyl]-1,2,3,4-tetrahydroisoquinoline-6,7-diol
Show/Hide
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C18H15F6NO2
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1
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| 1 |
Ki = 4365.16 nM
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CP0384603
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4-[(2R)-2-hydroxy-3-[2-(2-methoxyphenoxy)ethylamino]propyl]benzene-1,2-diol
Show/Hide
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C18H23NO5
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1
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| 1 |
Ki = 5200 nM
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CP0440420
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4-[3-(propan-2-ylamino)propoxy]benzene-1,2-diol
Show/Hide
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C12H19NO3
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1
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| 1 |
Ki = 6900 nM
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CP0384611
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4-[(2R)-2-hydroxy-3-[2-(2-methoxyphenoxy)ethylamino]propoxy]benzene-1,2-diol
Show/Hide
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C18H23NO6
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1
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| 1 |
Ki = 7900 nM
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CP0383399
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(2S,3S,4S,5R,6S)-6-(5-((R)-2-(5,6-diethyl-2,3-dihydro-1H-inden-2-ylamino)-1-hydroxyethyl)-2-oxo-1,2-dihydroquinolin-8-yloxy)-3,4,5-trihydroxytetrahydro-2H-pyran-2-carboxylic acid
Show/Hide
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C30H36N2O9
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1
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| 1 |
Ki > 10000 nM
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CP0388502
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3-(2-hydroxy-3-(1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propoxy)benzoic acid
Show/Hide
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C27H28N4O4S
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1
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| 1 |
Ki > 10000 nM
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CP0451232
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3-(2-{(R)-2-[2-(3-Chloro-phenyl)-2-hydroxy-ethylamino]-propyl}-thiazol-5-yl)-propionic acid
Show/Hide
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C17H21ClN2O3S
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1
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| 1 |
Ki = 11400 nM
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CP0412982
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4-(2-{(R)-2-[2-(3-Chloro-phenyl)-2-hydroxy-ethylamino]-propyl}-thiazol-5-yl)-butyric acid
Show/Hide
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C18H23ClN2O3S
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1
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| 1 |
Ki = 13900 nM
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CP0404156
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2-(4-{(R)-2-[(R)-2-(3-Chloro-phenyl)-2-hydroxy-ethylamino]-propyl}-phenoxy)-malonic acid
Show/Hide
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C20H22ClNO6
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1
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| 1 |
Ki = 17100 nM
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CP0374790
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(4-{(R)-2-[(R)-2-(3-Chloro-phenyl)-2-hydroxy-ethylamino]-propyl}-phenoxymethyl)-phosphonic acid
Show/Hide
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C18H23ClNO5P
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1
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| 1 |
Ki = 39700 nM
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CP0413983
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(2R,3R)-6-Dipropylamino-5,6,7,8-tetrahydro-naphthalen-1-ol
Show/Hide
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C16H25NO
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1
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| 1 |
Ki = 40000 nM
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CP0518305
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(4-{(R)-2-[(R)-2-(3-Chloro-phenyl)-2-hydroxy-ethylamino]-propyl}-phenoxymethyl)-phosphonic acid monoisopropyl ester
Show/Hide
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C21H29ClNO5P
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1
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| 1 |
Ki = 42600 nM
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CP0036921
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3-HYDROXYTYRAMINE HYDROCHLORIDE
Show/Hide
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C8H11NO2
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1
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| 1 |
Ki = 61000 nM
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CP0448909
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(4-{(R)-2-[(R)-2-(3-Chloro-phenyl)-2-hydroxy-ethylamino]-propyl}-phenoxymethyl)-methyl-phosphinic acid
Show/Hide
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C19H25ClNO4P
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1
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| 1 |
Ki = 73700 nM
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CP0044536
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(2R)-7-Dipropylamino-5,6,7,8-tetrahydro-naphthalen-2-ol
Show/Hide
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C16H25NO
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1
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| 1 |
Ki = 86000 nM
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CP0461669
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(+/-)-N-[5-(2-bromo-1-hydroxyethyl)isoxazol-3-yl]methanesulfonamide
Show/Hide
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C10H19N3O4S
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1
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| 1 |
Ki > 100000 nM
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CP0006107
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CAS_85760-74-3
Show/Hide
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C13H21N3
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1
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| 1 |
Ki = 100000 nM
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CP0127400
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(-)-Pramipexole
Show/Hide
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C10H17N3S
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1
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| 1 |
Ki = 100000 nM
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CP0388360
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N-[3-[(5-chloro-6-oxo-4-piperazin-1-ylpyridazin-1-yl)methyl]-2-methylphenyl]-4-phenylbenzamide
Show/Hide
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C29H28ClN5O2
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1
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| 1 |
Ki > 6309.57 nM
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