Sub[-Tyr-Arg-Leu-Arg-Tyr-NH2]2

Sub[-Trp-Arg-Nva-Arg-Tyr-NH2]2

6-((5-ethyl-4-(fluoromethyl)thiazol-2-ylthio)methyl)-N-((6-methylpyridin-2-yl)methyl)-4-morpholinopyridin-2-amine

6-((4,5-dimethyloxazol-2-ylthio)methyl)-N-((6-methylpyridin-2-yl)methyl)-4-thiomorpholinopyridin-2-amine

6-((4-(fluoromethyl)-5-methylthiazol-2-ylthio)methyl)-N-((6-methylpyridin-2-yl)methyl)-4-morpholinopyridin-2-amine

6-((4,5-dimethylthiazol-2-ylthio)methyl)-N-((6-methylpyridin-2-yl)methyl)-4-morpholinopyridin-2-amine

6-((4,5-dimethyloxazol-2-ylthio)methyl)-N-((6-fluoropyridin-2-yl)methyl)-4-thiomorpholinopyridin-2-amine

6-((5-ethyl-4-methyloxazol-2-ylthio)methyl)-N-((6-methylpyridin-2-yl)methyl)-4-morpholinopyridin-2-amine

N-[(6-methylpyridin-2-yl)methyl]-4-morpholin-4-yl-6-(4,5,6,7-tetrahydro-1,3-benzoxazol-2-ylsulfanylmethyl)pyridin-2-amine

6-((5-(fluoromethyl)-4-methylthiazol-2-ylthio)methyl)-N-((6-methylpyridin-2-yl)methyl)-4-morpholinopyridin-2-amine

6-((4,5-dimethyloxazol-2-ylthio)methyl)-N-((6-methylpyridin-2-yl)methyl)-4-morpholinopyridin-2-amine

propan-2-yl N-[3-chloro-5-[1-[[6-[2-(5-ethyl-4-methyl-1,3-thiazol-2-yl)ethyl]-4-morpholin-4-ylpyridin-2-yl]amino]ethyl]phenyl]carbamate

6-((4,5-dimethyloxazol-2-ylthio)methyl)-N-((6-fluoropyridin-2-yl)methyl)-4-morpholinopyridin-2-amine

6-[(4,5-dimethyl-1,3-oxazol-2-yl)sulfanylmethyl]-4-(1,1-dioxo-1,4-thiazinan-4-yl)-N-[(6-methylpyridin-2-yl)methyl]pyridin-2-amine

6-((4,5-dimethyloxazol-2-ylthio)methyl)-N-((6-(fluoromethyl)pyridin-2-yl)methyl)-4-morpholinopyridin-2-amine

6-((4,5-dimethyloxazol-2-ylthio)methyl)-N-((6-(methoxymethyl)pyridin-2-yl)methyl)-4-morpholinopyridin-2-amine

6-((4,5-dimethyloxazol-2-ylthio)methyl)-N-((2-fluoropyridin-4-yl)methyl)-4-morpholinopyridin-2-amine

6-((4,5-dimethyloxazol-2-ylthio)methyl)-N-((2-fluoropyridin-3-yl)methyl)-4-morpholinopyridin-2-amine

6-[(4,5-dimethyl-1,3-oxazol-2-yl)sulfanylmethyl]-4-(1,1-dioxo-1,4-thiazinan-4-yl)-N-[(6-fluoropyridin-2-yl)methyl]pyridin-2-amine

6-((4,5-dimethyloxazol-2-ylthio)methyl)-N-((6-((2-fluoroethoxy)methyl)pyridin-2-yl)methyl)-4-morpholinopyridin-2-amine

(1-(4-chlorophenoxy)-9-((1-methylpiperidin-4-yl)methyl)-9H-carbazol-3-yl)(4-methylpiperazin-1-yl)methanone

2-(4-((1-(4-chlorophenoxy)-3-(1-methylpiperazine-4-carbonyl)-9H-carbazol-9-yl)methyl)piperidin-1-yl)-N,N-dimethylacetamide

(1-(4-chlorophenoxy)-9-(piperidin-4-ylmethyl)-9H-carbazol-3-yl)(4-methylpiperazin-1-yl)methanone

6-((4,5-dimethyloxazol-2-ylthio)methyl)-N-((6-(2-fluoroethoxy)pyridin-2-yl)methyl)-4-morpholinopyridin-2-amine

6-((4,5-dimethyloxazol-2-ylthio)methyl)-N-((6-fluoropyridin-3-yl)methyl)-4-morpholinopyridin-2-amine

(1R,3S)-1-(4-chlorophenoxy)-3-(4-methylpiperidin-1-yl)-9-(piperidin-4-ylmethyl)-2,3-dihydro-1H-carbazol-4-one

(1-(4-chlorophenoxy)-9-(((3R,4S)-3-fluoro-1-methylpiperidin-4-yl)methyl)-9H-carbazol-3-yl)(4-methylpiperazin-1-yl)methanone

(1R)-1-(4-chlorophenoxy)-3-(4-methylpiperazin-1-yl)-9-[(1-methylpiperidin-4-yl)methyl]-2,3-dihydro-1H-carbazol-4-one

(1R)-1-(4-chlorophenoxy)-3-[4-(2-hydroxyethyl)piperazin-1-yl]-9-(piperidin-4-ylmethyl)-2,3-dihydro-1H-carbazol-4-one

(1-(4-chlorophenoxy)-9-((3-fluoro-1,2,5,6-tetrahydropyridin-4-yl)methyl)-9H-carbazol-3-yl)(4-methylpiperazin-1-yl)methanone

(1R,3S)-1-(4-chlorophenoxy)-3-(4-methylpiperazin-1-yl)-9-(piperidin-4-ylmethyl)-2,3-dihydro-1H-carbazol-4-one

(1-(4-chlorophenoxy)-9-(3-(piperidin-1-yl)propyl)-9H-carbazol-3-yl)(4-methylpiperazin-1-yl)methanone

1-(4-chlorophenoxy)-N-(2-(dimethylamino)ethyl)-9-(((3S,4S)-3-fluoropiperidin-4-yl)methyl)-9H-carbazole-3-carboxamide

(1-(4-chlorophenoxy)-9-(((3R,4S)-3-fluoropiperidin-4-yl)methyl)-9H-carbazol-3-yl)(4-methylpiperazin-1-yl)methanone

(1-(4-chlorophenoxy)-9-(((3S,4S)-3-fluoropiperidin-4-yl)methyl)-9H-carbazol-3-yl)(4-methylpiperazin-1-yl)methanone

(1R)-1-(4-chlorophenoxy)-9-[[4-(methylamino)cyclohexyl]methyl]-3-(4-methylpiperazin-1-yl)-2,3-dihydro-1H-carbazol-4-one

(1-(4-chlorophenoxy)-9-(((3S,4S)-3-fluoro-1-methylpiperidin-4-yl)methyl)-9H-carbazol-3-yl)(4-methylpiperazin-1-yl)methanone

(1R,3R)-1-(4-chlorophenoxy)-3-(4-methylpiperidin-1-yl)-9-(piperidin-4-ylmethyl)-2,3-dihydro-1H-carbazol-4-one

(1R)-1-(4-chlorophenoxy)-3-(4-fluoro-4-methylpiperidin-1-yl)-9-(piperidin-4-ylmethyl)-2,3-dihydro-1H-carbazol-4-one

(1-(4-chlorophenoxy)-9-(piperidin-3-ylmethyl)-9H-carbazol-3-yl)(4-methylpiperazin-1-yl)methanone

(1R)-1-(4-chlorophenoxy)-9-[[(3R,4S)-3-fluoro-1-methylpiperidin-4-yl]methyl]-3-(4-methylpiperazin-1-yl)-2,3-dihydro-1H-carbazol-4-one

(1-(4-chlorophenoxy)-9-(((3R,4S)-1-cyclopropyl-3-fluoropiperidin-4-yl)methyl)-9H-carbazol-3-yl)(4-methylpiperazin-1-yl)methanone

(1R)-1-(4-chlorophenoxy)-9-[[(3R,4S)-3-fluoropiperidin-4-yl]methyl]-3-(4-methylpiperazin-1-yl)-2,3-dihydro-1H-carbazol-4-one

1-(4-chlorophenoxy)-N-(2-(dimethylamino)ethyl)-9-(((3S,4S)-3-fluoropiperidin-4-yl)methyl)-N-methyl-9H-carbazole-3-carboxamide

(1R)-1-(4-chlorophenoxy)-9-[[(3R,4R)-3-fluoropiperidin-4-yl]methyl]-3-(4-methylpiperazin-1-yl)-2,3-dihydro-1H-carbazol-4-one

1-(4-chlorophenoxy)-N-((1-ethylpyrrolidin-2-yl)methyl)-9-(((3S,4S)-3-fluoropiperidin-4-yl)methyl)-9H-carbazole-3-carboxamide

(1R)-1-(4-chlorophenoxy)-3-piperazin-1-yl-9-(3-piperidin-1-ylpropyl)-2,3-dihydro-1H-carbazol-4-one

(1R)-1-(4-chlorophenoxy)-9-[[(3R,4R)-3-fluoro-1-methylpiperidin-4-yl]methyl]-3-(4-methylpiperazin-1-yl)-2,3-dihydro-1H-carbazol-4-one

(1-(4-chlorophenoxy)-9-(((3S,4S)-3-fluoropiperidin-4-yl)methyl)-9H-carbazol-3-yl)(3-(dimethylamino)pyrrolidin-1-yl)methanone

(1R)-1-(4-chlorophenoxy)-3-(4-methylpiperidin-1-yl)-9-(3-piperidin-1-ylpropyl)-2,3-dihydro-1H-carbazol-4-one

(1R,3R)-1-(4-chlorophenoxy)-3-(4-methylpiperazin-1-yl)-9-(piperidin-4-ylmethyl)-2,3-dihydro-1H-carbazol-4-one

(1-(4-chlorophenoxy)-9-(((3R,4S)-3-fluoropiperidin-4-yl)methyl)-9H-carbazol-3-yl)(4-(2-hydroxyethyl)piperazin-1-yl)methanone

(1-(4-chlorophenoxy)-9-(((3S,4S)-3-fluoropiperidin-4-yl)methyl)-9H-carbazol-3-yl)(4-cyclopropylpiperazin-1-yl)methanone

(1R)-1-(4-chlorophenoxy)-3-(4-methylpiperazin-1-yl)-9-(3-piperidin-1-ylpropyl)-2,3-dihydro-1H-carbazol-4-one

1-(4-chlorophenoxy)-9-(((3S,4S)-3-fluoropiperidin-4-yl)methyl)-N-(2-(1-methylpyrrolidin-2-yl)ethyl)-9H-carbazole-3-carboxamide

(1R)-1-(4-chlorophenoxy)-3-(4,4-difluoropiperidin-1-yl)-9-(piperidin-4-ylmethyl)-2,3-dihydro-1H-carbazol-4-one

(1-(4-chlorophenoxy)-9-(((3R,4S)-3-fluoropiperidin-4-yl)methyl)-9H-carbazol-3-yl)(5,6-dihydroimidazo[1,2-a]pyrazin-7(8H)-yl)methanone

(1-(4-chlorophenoxy)-9-(((3R,4S)-3-fluoropiperidin-4-yl)methyl)-9H-carbazol-3-yl)(6,7-dihydro-1H-imidazo[4,5-c]pyridin-5(4H)-yl)methanone

(1R)-1-(4-chlorophenoxy)-3-piperidin-1-yl-9-(3-piperidin-1-ylpropyl)-2,3-dihydro-1H-carbazol-4-one

(1R)-1-(4-chlorophenoxy)-3-(4-methyl-3-oxopiperazin-1-yl)-9-(piperidin-4-ylmethyl)-2,3-dihydro-1H-carbazol-4-one

6-(2-(5-ethyl-4-methyloxazol-2-yl)ethyl)-4-morpholino-N-(2,2,2-trifluoroethyl)pyridin-2-amine

(1R)-1-(4-chlorophenoxy)-9-(3-piperidin-1-ylpropyl)-2,3-dihydro-1H-carbazol-4-one

(1-(4-chlorophenoxy)-9-(((3R,4S)-3-fluoropiperidin-4-yl)methyl)-9H-carbazol-3-yl)(4-hydroxypiperidin-1-yl)methanone

6-(2-(5-ethyl-4-methyloxazol-2-yl)ethyl)-4-morpholino-N-propylpyridin-2-amine

(1-(4-chlorophenoxy)-9-(((3R,4S)-3-fluoropiperidin-4-yl)methyl)-9H-carbazol-3-yl)(4-(2,2,2-trifluoroethyl)piperazin-1-yl)methanone

1-(4-chlorophenoxy)-9-(((3S,4S)-3-fluoropiperidin-4-yl)methyl)-N,N-dimethyl-9H-carbazole-3-carboxamide

6-(2-(5-ethyl-4-methyloxazol-2-yl)ethyl)-N-(2-methoxyethyl)-4-morpholinopyridin-2-amine

2-(6-((4,5-dimethylthiazol-2-ylthio)methyl)-4-morpholinopyridin-2-ylamino)acetonitrile

ethyl 2-[[6-[2-(5-ethyl-4-methyl-1,3-oxazol-2-yl)ethyl]-4-morpholin-4-ylpyridin-2-yl]amino]acetate

(1R)-1-(4-chlorophenoxy)-3-morpholin-4-yl-9-(3-piperidin-1-ylpropyl)-2,3-dihydro-1H-carbazol-4-one

N-ethyl-6-[2-(5-ethyl-4-methyl-1,3-oxazol-2-yl)ethyl]-4-morpholin-4-ylpyridin-2-amine

2-(6-((5-ethyl-4-methyloxazol-2-ylthio)methyl)-4-morpholinopyridin-2-ylamino)acetonitrile

2-(6-(2-(5-ethyl-4-methyloxazol-2-yl)ethyl)-4-morpholinopyridin-2-ylamino)acetonitrile

3-(6-(2-(5-ethyl-4-methyloxazol-2-yl)ethyl)-4-morpholinopyridin-2-ylamino)propanenitrile

6-(2-(5-ethyl-4-methyloxazol-2-yl)ethyl)-N-isopropyl-4-morpholinopyridin-2-amine

(1R)-1-(4-chlorophenoxy)-9-methyl-3-(4-methylpiperazin-1-yl)-2,3-dihydro-1H-carbazol-4-one

6-(2-(5-ethyl-4-methyloxazol-2-yl)ethyl)-N-methyl-4-morpholinopyridin-2-amine

2-(4-morpholino-6-((1,4,5-trimethyl-1H-imidazol-2-ylthio)methyl)pyridin-2-ylamino)acetonitrile

2-(6-((4,5-dimethyloxazol-2-ylthio)methyl)-4-morpholinopyridin-2-ylamino)acetonitrile

(1-((1R,4R)-4-((R)-1-(4-methoxyphenyl)ethylamino)-2,2-dimethylcyclohexanecarbonyl)-4-phenylpiperidin-4-yl)(pyrrolidin-1-yl)methanone

(4,4-diphenylpiperidin-1-yl)((1R,4R)-4-((R)-1-(4-methoxyphenyl)ethylamino)-2,2-dimethylcyclohexyl)methanone

(1-((1R,4R)-2,2-dimethyl-4-((R)-1-p-tolylethylamino)cyclohexanecarbonyl)-4-phenylpiperidin-4-yl)(pyrrolidin-1-yl)methanone

1-((1R,4R)-4-((R)-1-(4-methoxyphenyl)ethylamino)-2,2-dimethylcyclohexanecarbonyl)-N,N-dimethyl-4-phenylpiperidine-4-carboxamide

1'-((1R,4R)-4-((R)-1-(4-methoxyphenyl)ethylamino)-2,2-dimethylcyclohexanecarbonyl)-4'-phenyl-1,4'-bipiperidin-2-one

(1-((1R,4R)-4-((S)-2,2-difluoro-1-(4-methoxyphenyl)ethylamino)-2,2-dimethylcyclohexanecarbonyl)-4-phenylpiperidin-4-yl)(pyrrolidin-1-yl)methanone

((1R,4R)-4-((R)-1-(4-methoxyphenyl)ethylamino)-2,2-dimethylcyclohexyl)(4-(6-methoxypyridin-3-yl)-4-phenylpiperidin-1-yl)methanone

(1-((1R,4R)-4-((R)-1-(4-chlorophenyl)ethylamino)-2,2-dimethylcyclohexanecarbonyl)-4-phenylpiperidin-4-yl)(pyrrolidin-1-yl)methanone

((1R,4R)-4-((R)-1-(4-methoxyphenyl)ethylamino)-2,2-dimethylcyclohexyl)(4-phenyl-4-(pyridin-3-yl)piperidin-1-yl)methanone

(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-amino-1-hydroxy-3-(1H-indol-3-yl)propylidene]amino]-5-carbamimidamido-1-hydroxypentylidene]amino]-1-hydroxypentylidene]amino]-5-carbamimidamido-1-hydroxypentylidene]amino]-1-hydroxy-3-(4-hydroxyphenyl)propylidene]amino]-1-hydroxy-3-(1H-indol-3-yl)propylidene]amino]-5-carbamimidamido-1-hydroxypentylidene]amino]-1-hydroxypentylidene]amino]-5-carbamimidamido-1-hydroxypentylidene]amino]-1-hydroxy-3-(4-hydroxyphenyl)propylidene]amino]-1-hydroxy-3-(1H-indol-3-yl)propylidene]amino]-5-carbamimidamido-1-hydroxypentylidene]amino]-1-hydroxypentylidene]amino]-5-carbamimidamido-N-[(2S)-1-hydroxy-3-(4-hydroxyphenyl)-1-iminopropan-2-yl]pentanimidic acid

(4-(6-chloropyridin-3-yl)-4-phenylpiperidin-1-yl)((1R,4R)-4-((R)-1-(4-methoxyphenyl)ethylamino)-2,2-dimethylcyclohexyl)methanone

3-(1-((1R,4R)-4-((R)-1-(4-methoxyphenyl)ethylamino)-2,2-dimethylcyclohexanecarbonyl)-4-phenylpiperidin-4-yl)-1,3-oxazinan-2-one

(1-((1R,4R)-2,2-dimethyl-4-((S)-2,2,2-trifluoro-1-(4-methoxyphenyl)ethylamino)cyclohexanecarbonyl)-4-phenylpiperidin-4-yl)(pyrrolidin-1-yl)methanone

(1-((1R,4R)-4-((R)-1-(4-fluorophenyl)ethylamino)-2,2-dimethylcyclohexanecarbonyl)-4-phenylpiperidin-4-yl)(pyrrolidin-1-yl)methanone

1-(1-((1R,4R)-4-((R)-1-(4-methoxyphenyl)ethylamino)-2,2-dimethylcyclohexanecarbonyl)-4-phenylpiperidin-4-yl)tetrahydropyrimidin-2(1H)-one

N-[4-[(1R,4R)-4-[[(1R)-1-(4-methoxyphenyl)ethyl]amino]-2,2-dimethylcyclohexanecarbonyl]-1-phenylcyclohexyl]acetamide

N-[4-[(1R,4R)-4-[[(1R)-1-(4-methoxyphenyl)ethyl]amino]-2,2-dimethylcyclohexanecarbonyl]-1-phenylcyclohexyl]-N-methylacetamide

((1R,4R)-4-((R)-1-(4-methoxyphenyl)ethylamino)-2,2-dimethylcyclohexyl)(4-(5-methyl-1,3,4-oxadiazol-2-yl)-4-phenylpiperidin-1-yl)methanone

Adp[-Trp-Arg-Nva-Arg-Tyr-NH2]2

(1-((1R,4R)-4-((R)-1-(4-methoxyphenyl)ethylamino)-2,2-dimethylcyclohexanecarbonyl)-4-phenylpiperidin-4-yl)(piperidin-1-yl)methanone

(1-((1R,4R)-2,2-dimethyl-4-((R)-1-phenylethylamino)cyclohexanecarbonyl)-4-phenylpiperidin-4-yl)(pyrrolidin-1-yl)methanone

(1-((1R,4R)-4-((R)-1-(3-methoxyphenyl)ethylamino)-2,2-dimethylcyclohexanecarbonyl)-4-phenylpiperidin-4-yl)(pyrrolidin-1-yl)methanone

(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-amino-1-hydroxy-3-(1H-indol-3-yl)propylidene]amino]-5-carbamimidamido-1-hydroxypentylidene]amino]-1-hydroxypentylidene]amino]-5-carbamimidamido-1-hydroxypentylidene]amino]-1-hydroxy-3-(4-hydroxyphenyl)propylidene]amino]-1-hydroxy-3-(1H-indol-3-yl)propylidene]amino]-5-carbamimidamido-1-hydroxypentylidene]amino]-1-hydroxypentylidene]amino]-5-carbamimidamido-N-[(2S)-1-hydroxy-3-(4-hydroxyphenyl)-1-iminopropan-2-yl]pentanimidic acid

((1R,4R)-4-((R)-1-(4-methoxyphenyl)ethylamino)-2,2-dimethylcyclohexyl)(4-(5-methyl-1,3,4-thiadiazol-2-yl)-4-phenylcyclohexyl)methanone

(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2R)-2-amino-3-[[(2R)-2-amino-3-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-amino-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-1-oxopentan-2-yl]amino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-3-(1H-indol-3-yl)-1-oxopropan-2-yl]amino]-3-oxopropyl]disulfanyl]propanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]pentanoyl]amino]-N-[(2S)-1-amino-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]-5-(diaminomethylideneamino)pentanamide

(1-((1R,4R)-4-(4-methoxybenzylamino)-2,2-dimethylcyclohexanecarbonyl)-4-phenylpiperidin-4-yl)(pyrrolidin-1-yl)methanone

(1-((1R,4R)-4-((R)-1-(2-methoxyphenyl)ethylamino)-2,2-dimethylcyclohexanecarbonyl)-4-phenylpiperidin-4-yl)(pyrrolidin-1-yl)methanone

(4-(1,3,4-oxadiazol-2-yl)-4-phenylpiperidin-1-yl)((1R,4R)-4-((R)-1-(4-methoxyphenyl)ethylamino)-2,2-dimethylcyclohexyl)methanone

(1-((1R,4R)-4-((S)-1-(4-methoxyphenyl)ethylamino)-2,2-dimethylcyclohexanecarbonyl)-4-phenylpiperidin-4-yl)(pyrrolidin-1-yl)methanone

((1R,4R)-4-((R)-1-(4-methoxyphenyl)ethylamino)-2,2-dimethylcyclohexyl)(4'-phenyl-1,4'-bipiperidin-1'-yl)methanone

N-[4-(4-benzoylpiperazin-1-yl)-3-chlorophenyl]-2,2-dimethylpropanamide

N-(3-chloro-4-(4-(3-methoxypicolinoyl)piperazin-1-yl)phenyl)-2-methyl-2-phenylpropanamide Hydrochloride salt

N-[3-chloro-4-[2-(cyclopropylmethyl)-2,8-diazaspiro[4.5]decan-8-yl]phenyl]-2-methyl-2-[4-(trifluoromethyl)pyrimidin-2-yl]propanamide