2-fluoro-N-[5-(trifluoromethyl)-1,3-oxazol-2-yl]-9H-xanthene-9-carboxamide

2,7-difluoro-N-(4-(trifluoromethyl)oxazol-2-yl)-9H-xanthene-9-carboxamide

4-fluoro-N-[4-(trifluoromethyl)-1,3-oxazol-2-yl]-9H-xanthene-9-carboxamide

4-fluoro-N-[5-(trifluoromethyl)-1,3-oxazol-2-yl]-9H-xanthene-9-carboxamide

2,7-difluoro-N-(oxazol-2-yl)-9H-xanthene-9-carboxamide

4,5-difluoro-N-(4-(trifluoromethyl)oxazol-2-yl)-9H-xanthene-9-carboxamide

4,5-difluoro-N-(5-(trifluoromethyl)oxazol-2-yl)-9H-xanthene-9-carboxamide

N-[4-(trifluoromethyl)-1,3-oxazol-2-yl]-9H-xanthene-9-carboxamide

N-(5-methyl-1,2,4-oxadiazol-3-yl)-9H-xanthene-9-carboxamide

3-fluoro-N-[4-(trifluoromethyl)-1,3-oxazol-2-yl]-9H-xanthene-9-carboxamide

N-[5-(trifluoromethyl)-1,3-oxazol-2-yl]-9H-xanthene-9-carboxamide

(1R,2R,3R,5R,6R)-2-Amino-3-(3,4-dichloro-benzyloxy)-6-fluoro-bicyclo[3.1.0]hexane-2,6-dicarboxylic acid

(1S,2S)-2-((S)-1-amino-1-carboxy-2-(9H-xanthen-9-yl)ethyl)cyclopropanecarboxylic acid

5-(1-(2,4-difluorophenyl)-5-methyl-1H-1,2,3-triazol-4-yl)-2-isopropylisoindolin-1-one

3-Methyl-1H-pyrrole-2,4-dicarboxylic acid 2-isopropyl ester 4-(1,2,2-trimethyl-propyl) ester

3,3-dimethylbutan-2-yl 2-[3-(1,3-dioxoisoindol-2-yl)propyl]-8-methyl-1-oxo-3,4-dihydropyrrolo[1,2-a]pyrazine-7-carboxylate

(S)-4-(3,3-dimethylbutan-2-yl) 2-propyl 3,5-dimethyl-1H-pyrrole-2,4-dicarboxylate

3-Methyl-1H-pyrrole-2,4-dicarboxylic acid 2-tert-butyl ester 4-(1,2,2-trimethyl-propyl) ester

3,3-dimethylbutan-2-yl 2-(2-fluoroethyl)-8-methyl-1-oxo-3,4-dihydropyrrolo[1,2-a]pyrazine-7-carboxylate

3,3-dimethylbutan-2-yl 2-(cyclopropylmethyl)-8-methyl-1-oxo-3,4-dihydropyrrolo[1,2-a]pyrazine-7-carboxylate

3,3-dimethylbutan-2-yl 8-methyl-1-oxo-2-prop-2-enyl-3,4-dihydropyrrolo[1,2-a]pyrazine-7-carboxylate

3,3-dimethylbutan-2-yl 2-(2,2-difluoroethyl)-8-methyl-1-oxo-3,4-dihydropyrrolo[1,2-a]pyrazine-7-carboxylate

3,3-dimethylbutan-2-yl 8-methyl-1-oxo-2-propyl-3,4-dihydropyrrolo[1,2-a]pyrazine-7-carboxylate

3-Methyl-1H-pyrrole-2,4-dicarboxylic acid 4-tert-butyl ester 2-cyclopropylmethyl ester

1-oxo-2,3,4,9-tetrahydro-1H-beta-carboline-6-carboxylic acid adamantan-1-ylamide

N-(1-oxo-2,3,4,9-tetrahydropyrido[3,4-b]indol-6-yl)adamantane-1-carboxamide

3-Methyl-1H-pyrrole-2,4-dicarboxylic acid 4-tert-butyl ester 2-propyl ester

1-oxo-2,3,4,9-tetrahydro-1H-beta-carboline-6-carboxylic acid adamantan-2-ylamide

3-Methyl-1H-pyrrole-2,4-dicarboxylic acid di-tert-butyl ester

6-(benzyloxy)-3,4-dihydro-2H-pyrido[3,4-b]indol-1(9H)-one

N-(3,3-dimethylbutan-2-yl)-N-methyl-1-oxo-2,3,4,9-tetrahydropyrido[3,4-b]indole-6-carboxamide

3-Methyl-1H-pyrrole-2,4-dicarboxylic acid 2-pentafluorophenyl ester 4-(1,2,2-trimethyl-propyl) ester

5-Chloro-3-methyl-1H-pyrrole-2,4-dicarboxylic acid 2-propyl ester 4-(1,2,2-trimethyl-propyl) ester

6-(benzyloxy)-7-methyl-3,4-dihydro-2H-pyrido[3,4-b]indol-1(9H)-one

N-(2-bicyclo[2.2.1]heptanyl)-1-oxo-2,3,4,9-tetrahydropyrido[3,4-b]indole-6-carboxamide

6-(3,3-dimethylbutan-2-yloxy)-3,4-dihydro-2H-pyrido[3,4-b]indol-1(9H)-one

3,3-dimethylbutan-2-yl 2-(2-methoxyethyl)-8-methyl-1-oxo-3,4-dihydropyrrolo[1,2-a]pyrazine-7-carboxylate

3,3-dimethylbutan-2-yl 2-benzyl-8-methyl-1-oxo-3,4-dihydropyrrolo[1,2-a]pyrazine-7-carboxylate

3-Methyl-1H-pyrrole-2,4-dicarboxylic acid 2-(1-ethyl-pyrrolidin-3-yl) ester 4-(1,2,2-trimethyl-propyl) ester

1-oxo-2,3,4,9-tetrahydro-1H-beta-carboline-6-carboxylic acid (adamantan-1-ylmethyl)-amide

3-Methyl-1H-pyrrole-2,4-dicarboxylic acid 4-tert-butyl ester 2-ethyl ester

6-(1-phenylethoxy)-3,4-dihydro-2H-pyrido[3,4-b]indol-1(9H)-one

3-Methyl-1H-pyrrole-2,4-dicarboxylic acid 2-(2-dimethylamino-1-methyl-ethyl) ester 4-(1,2,2-trimethyl-propyl) ester

3,3-dimethylbutan-2-yl 2-[3-(ethylcarbamoylamino)propyl]-8-methyl-1-oxo-3,4-dihydropyrrolo[1,2-a]pyrazine-7-carboxylate

3,3-dimethylbutan-2-yl 8-methyl-2-[2-[(2-methylpropan-2-yl)oxycarbonylamino]ethyl]-1-oxo-3,4-dihydropyrrolo[1,2-a]pyrazine-7-carboxylate

3,3-dimethylbutan-2-yl 8-methyl-1-oxo-2-[3-(pyridine-4-carbonylamino)propyl]-3,4-dihydropyrrolo[1,2-a]pyrazine-7-carboxylate

3,3-dimethylbutan-2-yl 2-(3-acetamidopropyl)-8-methyl-1-oxo-3,4-dihydropyrrolo[1,2-a]pyrazine-7-carboxylate

7-(benzyloxy)-1,2-dihydropyrrolo[3,4-b]indol-3(4H)-one

3-Methyl-1H-pyrrole-2,4-dicarboxylic acid 2-pyridin-3-yl ester 4-(1,2,2-trimethyl-propyl) ester

1,3,5-Trimethyl-1H-pyrrole-2,4-dicarboxylic acid 4-tert-butyl ester 2-propyl ester

8-benzyloxy-3,4a,5,9b-tetrahydro-pyridazino[4,5-b]indol-4-one

1-oxo-N-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-6-carboxamide

3-Methyl-1H-pyrrole-2,4-dicarboxylic acid 4-tert-butyl ester 2-furan-2-ylmethyl ester

3-Methyl-1H-pyrrole-2,4-dicarboxylic acid 2-pyrimidin-4-yl ester 4-(1,2,2-trimethyl-propyl) ester

6-benzyloxy-2,3,4,4a,9,9a-hexahydro-beta-carbolin-1-one

5-Formyl-3-methyl-1H-pyrrole-2,4-dicarboxylic acid 4-tert-butyl ester 2-propyl ester

3,5-Dimethyl-pyrrole-1,2,4-tricarboxylic acid 1,4-di-tert-butyl ester 2-propyl ester

5-(Cyclopropylmethyl-carbamoyl)-3-methyl-1H-pyrrole-2,4-dicarboxylic acid 4-tert-butyl ester 2-propyl ester

5-Acetoxymethyl-3-methyl-1H-pyrrole-2,4-dicarboxylic acid 4-tert-butyl ester 2-propyl ester

7-(benzyloxy)-3,4-dihydro-2H-pyrido[3,4-b]indol-1(9H)-one

4-Methyl-5-(pyridin-2-ylsulfanylcarbonyl)-1H-pyrrole-3-carboxylic acid tert-butyl ester

3,3-dimethylbutan-2-yl 8-methyl-2-morpholin-4-yl-1-oxo-3,4-dihydropyrrolo[1,2-a]pyrazine-7-carboxylate

3,3-dimethylbutan-2-yl 8-methyl-2-[3-[methyl(pyridine-4-carbonyl)amino]propyl]-1-oxo-3,4-dihydropyrrolo[1,2-a]pyrazine-7-carboxylate

3-Methyl-5-(pyridin-2-ylsulfanylcarbonyl)-1H-pyrrole-2,4-dicarboxylic acid 4-tert-butyl ester 2-propyl ester

4-Methyl-1H-pyrrole-2,3,5-tricarboxylic acid 3-tert-butyl ester 2-methyl ester 5-propyl ester

5-(benzyloxy)-3,4-dihydro-2H-pyrido[3,4-b]indol-1(9H)-one

6-phenoxy-3,4-dihydro-2H-pyrido[3,4-b]indol-1(9H)-one

1-adamantan-1-yl-3-(1-oxo-2,3,4,9-tetrahydro-1H-beta-carbolin-6-yl)-urea

6-(cyclohexylmethoxy)-3,4-dihydro-2H-pyrido[3,4-b]indol-1(9H)-one

1-(3-Methoxy-propyl)-3,5-dimethyl-1H-pyrrole-2,4-dicarboxylic acid 4-tert-butyl ester 2-propyl ester

5-Hydroxymethyl-3-methyl-1H-pyrrole-2,4-dicarboxylic acid 4-tert-butyl ester 2-propyl ester

6-hydroxy-3,4-dihydro-1-oxo-beta-carboline

6-Methoxy-2,3,4,9-tetrahydro-beta-carbolin-1-one

N-(3,3-dimethylbutan-2-yl)-1-oxo-2,3,4,9-tetrahydropyrido[3,4-b]indole-6-carboxamide

6-benzyloxy-2,3,4,4a,9,9a-hexahydro-1H-beta-carboline

6-(benzyloxy)-3,4-dihydro-2H-carbazol-1(9H)-one

6-(benzyloxy)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole

1-Allyloxycarbonylmethyl-3,5-dimethyl-1H-pyrrole-2,4-dicarboxylic acid 4-tert-butyl ester 2-propyl ester

3,5-Dimethyl-1H-pyrrole-2,4-dicarboxylic acid 2-propyl ester 4-(1,2,2-trimethyl-propyl) ester

N-(2-methyl-2-phenylpropyl)-5,6,7,8-tetrahydroquinoxaline-2-carboxamide

N-[2-(4-fluorophenyl)-2-methylpropyl]quinoxaline-2-carboxamide

N-(2-methyl-2-phenylpropyl)quinoxaline-2-carboxamide

N-(4-methylcyclohexyl)-5-piperidin-1-ylpyrazine-2-carboxamide

2-(2-(4-(2,3-dihydro-1H-inden-2-ylamino)pyrido[3,4-d]pyrimidin-6-ylamino)ethoxy)ethanol

4-N-(2,3-dihydro-1H-inden-2-yl)-6-N-(2-methoxyethyl)pyrido[3,4-d]pyrimidine-4,6-diamine

N-cycloheptyl-6-(2-morpholin-4-ylethoxy)pyrido[3,4-d]pyrimidin-4-amine

N-cycloheptyl-5-piperidin-1-ylpyrazine-2-carboxamide

5-(4-(hydroxymethyl)piperidin-1-yl)-N-((1r,4r)-4-methylcyclohexyl)pyrazine-2-carboxamide

4-N-cyclohexyl-6-N-(2-morpholin-4-ylethyl)pyrido[3,4-d]pyrimidine-4,6-diamine

N-(2-methyl-2-phenylpropyl)-6-piperidin-1-ylpyrazine-2-carboxamide

4-N-cyclohexyl-6-N-(2-methoxyethyl)pyrido[3,4-d]pyrimidine-4,6-diamine

5-((2-cyanoethyl)(methyl)amino)-N-(2-methyl-2-phenylpropyl)pyrazine-2-carboxamide

4-N-(2,3-dihydro-1H-inden-2-yl)-6-N-methylpyrido[3,4-d]pyrimidine-4,6-diamine

N-(2-methoxy-2-phenylpropyl)quinoxaline-2-carboxamide

N-(2-methyl-2-phenylpropyl)-5-piperidin-1-ylpyrazine-2-carboxamide

1-(2-(4-(cyclohexylamino)pyrido[3,4-d]pyrimidin-6-yloxy)ethyl)pyrrolidin-2-one

2-(4-(2,3-dihydro-1H-inden-2-ylamino)pyrido[3,4-d]pyrimidin-6-ylamino)ethanol

N-(2-phenylpropyl)quinoxaline-2-carboxamide

5-((1-(dimethylamino)propan-2-yl)(methyl)amino)-N-(2-methyl-2-phenylpropyl)pyrazine-2-carboxamide

(R)-6-(2-hydroxy-1-phenylethylamino)-N-(2-methyl-2-phenylpropyl)pyrazine-2-carboxamide

N-cyclohexylquinazolin-4-amine

6-(butyl(methyl)amino)-N-cycloheptylpyrazine-2-carboxamide

4-N,6-N-bis(2,3-dihydro-1H-inden-2-yl)pyrido[3,4-d]pyrimidine-4,6-diamine

3-(4-(cyclohexylamino)pyrido[3,4-d]pyrimidin-6-yloxy)propan-1-ol

N-(2,3-dihydro-1H-inden-2-yl)quinazolin-4-amine

5-(4-(hydroxymethyl)piperidin-1-yl)-N-(2-methyl-2-phenylpropyl)pyrazine-2-carboxamide

N-(2,3-dihydro-1H-inden-2-yl)-6-[ethyl(methyl)amino]pyrazine-2-carboxamide

N-(2-methyl-1-phenylpropan-2-yl)quinoxaline-2-carboxamide

N-(2-methyl-2-pyridin-2-ylpropyl)quinoxaline-2-carboxamide

N-cyclohexyl-6-(2-morpholin-4-ylethoxy)pyrido[3,4-d]pyrimidin-4-amine

6-((2-hydroxyethyl)(methyl)amino)-N-(2-methyl-2-phenylpropyl)pyrazine-2-carboxamide

6-(3-hydroxyphenethylamino)-N-(cyclopropylmethyl)pyrazine-2-carboxamide

4-N-(2,3-dihydro-1H-inden-2-yl)-4-N,6-N-dimethylpyrido[3,4-d]pyrimidine-4,6-diamine

6-(4-benzyl-1,4-diazepan-1-yl)-N-(cyclopropylmethyl)pyrazine-2-carboxamide

N-(2-phenylethyl)quinoxaline-2-carboxamide

N-cyclohexyl-6-(2-methoxyethoxy)pyrido[3,4-d]pyrimidin-4-amine

4-N-(2,3-dihydro-1H-inden-2-yl)-6-N-[2-(dimethylamino)ethyl]pyrido[3,4-d]pyrimidine-4,6-diamine

N-(2,3-dihydro-1H-inden-2-yl)-6-methoxypyrido[3,4-d]pyrimidin-4-amine

(3-phenylpiperidin-1-yl)(quinoxalin-2-yl)methanone

2-(6-(2,3-dihydro-1H-inden-2-ylamino)pyrido[3,4-d]pyrimidin-4-ylamino)ethanol

6-N-(2,3-dihydro-1H-inden-2-yl)-4-N-methylpyrido[3,4-d]pyrimidine-4,6-diamine

2-(4-(cyclohexylamino)pyrido[3,4-d]pyrimidin-6-yloxy)ethanol

N-(2-methyl-2-phenylpropyl)-5-phenylpyrazine-2-carboxamide

4-N-(2,3-dihydro-1H-inden-2-yl)-6-N,6-N-dimethylpyrido[3,4-d]pyrimidine-4,6-diamine

4-N-cyclohexyl-6-N,6-N-dimethylpyrido[3,4-d]pyrimidine-4,6-diamine

6-N-(3-aminopropyl)-4-N-cyclohexylpyrido[3,4-d]pyrimidine-4,6-diamine

4-N-(2,3-dihydro-1H-inden-2-yl)-4-N,6-N,6-N-trimethylpyrido[3,4-d]pyrimidine-4,6-diamine

N-(2-methyl-2-phenylpropyl)-6-phenylpyrazine-2-carboxamide

(8-(4-methylpiperazin-1-yl)imidazo[1,2-a]pyrazin-2-yl)(4-(pyridin-2-yl)-1,4-diazepan-1-yl)methanone

N-[2-(methylamino)-2-phenylpropyl]quinoxaline-2-carboxamide

(8-(4-methylpiperazin-1-yl)imidazo[1,2-a]pyrazin-2-yl)(4-(6-methylpyridin-2-yl)-1,4-diazepan-1-yl)methanone

4-(cyclohexyloxy)quinazoline

6-N,6-N-dimethyl-4-N-pentan-2-ylpyrido[3,4-d]pyrimidine-4,6-diamine

(8-(4-methylpiperazin-1-yl)imidazo[1,2-a]pyrazin-2-yl)(3-phenylpiperidin-1-yl)methanone

8-(4-methylpiperazin-1-yl)-N-(2-phenylpropyl)imidazo[1,2-a]pyrazine-2-carboxamide

2-methyl-2-phenyl-N-(quinoxalin-2-ylmethyl)propan-1-amine

(S)-N6,N6-dimethyl-N4-(1-phenylethyl)pyrido[3,4-d]pyrimidine-4,6-diamine

N-(2,3-dihydro-1H-inden-2-yl)isoquinolin-1-amine

6-N-(2-aminoethyl)-4-N-cyclohexylpyrido[3,4-d]pyrimidine-4,6-diamine

2,2'-(pyrido[3,4-d]pyrimidine-4,6-diylbis(azanediyl))diethanol

N-cyclohexylquinolin-4-amine

N-(2-methyl-2-phenylpropyl)pyrazine-2-carboxamide