Brief Information of the Compound and Protein
Compound Name
3,3-dimethylbutan-2-yl 8-methyl-2-[3-[methyl(pyridine-4-carbonyl)amino]propyl]-1-oxo-3,4-dihydropyrrolo[1,2-a]pyrazine-7-carboxylate
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PubChem ID
CID: 44408692
Canonical SMILES
CC(OC(=O)c1cn2CCN(CCCN(C)C(=O)c3ccncc3)C(=O)c2c1C)C(C)(C)C
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Compound Formula C25H34N4O4
Compound Structure
Protein Name
Metabotropic glutamate receptor 1
Protein Classification
Membrane receptor
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Family C G protein-coupled receptor
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Small molecule receptor (family C GPCR)
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Neurotransmitter receptor (family C GPCR)
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Metabotropic glutamate receptor
Uniprot ID
P23385
Gene Name
GRM1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
IC50 = 3162.28 nM
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