Brief Information of the Compound and Protein
Compound Name
 Compound Info 
(8-(4-methylpiperazin-1-yl)imidazo[1,2-a]pyrazin-2-yl)(4-(6-methylpyridin-2-yl)-1,4-diazepan-1-yl)methanone
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 PubChem ID
CID: 44438575
Canonical SMILES
CN1CCN(CC1)c1nccn2cc(nc12)C(=O)N1CCCN(CC1)c1cccc(C)n1
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Compound Formula C23H30N8O
Compound Structure
Protein Name
 Protein Info 
Metabotropic glutamate receptor 1
Protein Classification
Membrane receptor
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Family C G protein-coupled receptor
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Small molecule receptor (family C GPCR)
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Neurotransmitter receptor (family C GPCR)
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Metabotropic glutamate receptor
Uniprot ID
P23385
Gene Name
GRM1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO
 Cell Line Info 
Cricetulus griseus (Chinese hamster)  1
1
Ki = 650 nM
   TI
   LI
   LO
   TS