Compound ID |
Compound Name |
Compound Formula |
CP0567819
|
US9018211, 5
Show/Hide
|
C24H24Cl2N2O6
|
1
|
1 |
IC50 = 7 nM
|
|
|
CP0189728
|
US9018211, 2A
Show/Hide
|
C26H30N2O6
|
1
|
1 |
IC50 = 9 nM
|
|
|
CP0352199
|
US9018211, 2C
Show/Hide
|
C26H30N2O6
|
1
|
1 |
IC50 = 10 nM
|
|
|
CP0503622
|
US9018211, 2B
Show/Hide
|
C26H30N2O6
|
1
|
1 |
IC50 = 12 nM
|
|
|
CP0438215
|
US9056859, 11
Show/Hide
|
C24H26N6O3
|
1
|
1 |
IC50 = 12 nM
|
|
|
CP0224663
|
US9018211, 12
Show/Hide
|
C26H30N2O5
|
1
|
1 |
IC50 = 13 nM
|
|
|
CP0512075
|
US9018211, 20
Show/Hide
|
C24H27N3O4
|
1
|
1 |
IC50 = 14 nM
|
|
|
CP0490184
|
US9018211, 22 (isomer 2)
Show/Hide
|
C24H26FN3O4
|
1
|
1 |
IC50 = 15 nM
|
|
|
CP0046632
|
US9056859, 72
Show/Hide
|
C23H25N7O3
|
1
|
1 |
IC50 = 20 nM
|
|
|
CP0512076
|
US9018211, 55
Show/Hide
|
C26H28FN3O3
|
1
|
1 |
IC50 = 23 nM
|
|
|
CP0522195
|
US9056859, 48
Show/Hide
|
C25H26FN3O4
|
1
|
1 |
IC50 = 35 nM
|
|
|
CP0108863
|
US9018211, 52
Show/Hide
|
C24H28N4O5
|
1
|
1 |
IC50 = 36 nM
|
|
|
CP0484859
|
US9056859, 122
Show/Hide
|
C23H24FN7O
|
1
|
1 |
IC50 = 37 nM
|
|
|
CP0442905
|
US9062070, 22
Show/Hide
|
C24H22F2N8O2
|
1
|
1 |
IC50 = 40 nM
|
|
|
CP0520396
|
US9056859, 217
Show/Hide
|
C24H25N7O4
|
1
|
1 |
IC50 = 56 nM
|
|
|
CP0538774
|
US9062070, 25
Show/Hide
|
C24H22F2N8O2
|
1
|
1 |
IC50 = 60 nM
|
|
|
CP0563888
|
US9062070, 15
Show/Hide
|
C23H24N8O2S
|
1
|
1 |
IC50 = 60 nM
|
|
|
CP0133230
|
6-[2-[4-[2-[4-(tetrazol-1-yl)phenyl]acetyl]piperazin-1-yl]ethyl]-3,4-dihydroisochromen-1-one
Show/Hide
|
C24H26N6O3
|
1
|
1 |
IC50 = 61 nM
|
|
|
CP0515001
|
US9056859, 96
Show/Hide
|
C25H27N7O3
|
1
|
1 |
IC50 = 61 nM
|
|
|
CP0578697
|
US9056859, 39
Show/Hide
|
C22H22FN7O
|
1
|
1 |
IC50 = 63 nM
|
|
|
CP0069452
|
5-[2-[4-[2-[4-(tetrazol-1-yl)phenyl]acetyl]piperazin-1-yl]ethyl]-3H-2-benzofuran-1-one
Show/Hide
|
C23H24N6O3
|
1
|
1 |
IC50 = 65 nM
|
|
|
CP0554215
|
US9062070, 32
Show/Hide
|
C24H22ClFN8O2
|
1
|
1 |
IC50 = 70 nM
|
|
|
CP0442903
|
US9062070, 21
Show/Hide
|
C24H22F2N8O2
|
1
|
1 |
IC50 = 80 nM
|
|
|
CP0450165
|
US9062070, 20
Show/Hide
|
C24H22F2N8O2
|
1
|
1 |
IC50 = 80 nM
|
|
|
CP0488823
|
US9062070, 49
Show/Hide
|
C26H27N7O4
|
1
|
1 |
IC50 = 80 nM
|
|
|
CP0538776
|
US9062070, 31
Show/Hide
|
C24H22ClFN8O2
|
1
|
1 |
IC50 = 80 nM
|
|
|
CP0574817
|
US9062070, 83
Show/Hide
|
C23H21ClFN9O2
|
1
|
1 |
IC50 = 80 nM
|
|
|
CP0464460
|
US9062070, 19
Show/Hide
|
C24H22F2N8O2
|
1
|
1 |
IC50 = 90 nM
|
|
|
CP0488825
|
US9062070, 57
Show/Hide
|
C25H25N7O4
|
1
|
1 |
IC50 = 90 nM
|
|
|
CP0556002
|
US9062070, 97
Show/Hide
|
C25H26FN9O
|
1
|
1 |
IC50 = 90 nM
|
|
|
CP0507134
|
US9056859, 59
Show/Hide
|
C24H23F2N3O3
|
1
|
1 |
IC50 = 94 nM
|
|
|
CP0554240
|
US9062070, 102
Show/Hide
|
C24H25FN10O
|
1
|
1 |
IC50 = 100 nM
|
|
|
CP0563280
|
US9062070, 96A
Show/Hide
|
C25H26FN9O
|
1
|
1 |
IC50 = 100 nM
|
|
|
CP0563890
|
US9062070, 70
Show/Hide
|
C25H25FN8O3
|
1
|
1 |
IC50 = 100 nM
|
|
|
CP0573649
|
US9062070, 88
Show/Hide
|
C27H28FN7O4
|
1
|
1 |
IC50 = 100 nM
|
|
|
CP0578698
|
US9056859, 177
Show/Hide
|
C26H29N7O3
|
1
|
1 |
IC50 = 100 nM
|
|
|
CP0538773
|
US9062070, 18
Show/Hide
|
C24H22F2N8O2
|
1
|
1 |
IC50 = 110 nM
|
|
|
CP0524437
|
US9062070, 71
Show/Hide
|
C25H26N8O2
|
1
|
1 |
IC50 = 120 nM
|
|
|
CP0553589
|
US9062070, 1I
Show/Hide
|
C27H29N7O4
|
1
|
1 |
IC50 = 120 nM
|
|
|
CP0554239
|
US9062070, 80
Show/Hide
|
C23H22FN9O2
|
1
|
1 |
IC50 = 120 nM
|
|
|
CP0555350
|
US9062070, 89
Show/Hide
|
C27H28FN7O4
|
1
|
1 |
IC50 = 120 nM
|
|
|
CP0578132
|
US9062070, 76
Show/Hide
|
C24H24FN9O2
|
1
|
1 |
IC50 = 130 nM
|
|
|
CP0424201
|
US9062070, 66
Show/Hide
|
C26H27N7O4
|
1
|
1 |
IC50 = 140 nM
|
|
|
CP0520697
|
US9062070, 91
Show/Hide
|
C25H25FN8O2
|
1
|
1 |
IC50 = 140 nM
|
|
|
CP0506778
|
US9062070, 23
Show/Hide
|
C24H22F2N8O2
|
1
|
1 |
IC50 = 150 nM
|
|
|
CP0506941
|
US9062070, 58
Show/Hide
|
C25H25N7O4
|
1
|
1 |
IC50 = 150 nM
|
|
|
CP0550563
|
US9062070, 67
Show/Hide
|
C26H27N7O4
|
1
|
1 |
IC50 = 150 nM
|
|
|
CP0554238
|
US9062070, 75
Show/Hide
|
C24H24FN9O2
|
1
|
1 |
IC50 = 150 nM
|
|
|
CP0563275
|
US9062070, 50
Show/Hide
|
C26H27N7O4
|
1
|
1 |
IC50 = 150 nM
|
|
|
CP0450164
|
US9062070, 12
Show/Hide
|
C26H27FN8O2
|
1
|
1 |
IC50 = 160 nM
|
|
|
CP0524438
|
US9062070, 78
Show/Hide
|
C26H26FN7O4
|
1
|
1 |
IC50 = 160 nM
|
|
|
CP0553590
|
US9062070, 34
Show/Hide
|
C25H25FN8O2
|
1
|
1 |
IC50 = 160 nM
|
|
|
CP0506939
|
US9062070, 33
Show/Hide
|
C26H27N7O4
|
1
|
1 |
IC50 = 170 nM
|
|
|
CP0554237
|
US9062070, 44
Show/Hide
|
C25H25FN8O2
|
1
|
1 |
IC50 = 170 nM
|
|
|
CP0556003
|
US9062070, 98
Show/Hide
|
C25H26FN9O
|
1
|
1 |
IC50 = 170 nM
|
|
|
CP0488816
|
US9062070, 1G
Show/Hide
|
C27H29N7O4
|
1
|
1 |
IC50 = 180 nM
|
|
|
CP0563279
|
US9062070, 93
Show/Hide
|
C25H25FN8O2
|
1
|
1 |
IC50 = 180 nM
|
|
|
CP0575645
|
US9062070, 1K
Show/Hide
|
C27H29N7O4
|
1
|
1 |
IC50 = 180 nM
|
|
|
CP0488821
|
US9062070, 30
Show/Hide
|
C24H22ClFN8O2
|
1
|
1 |
IC50 = 190 nM
|
|
|
CP0550562
|
US9062070, 51
Show/Hide
|
C25H26N8O3
|
1
|
1 |
IC50 = 190 nM
|
|
|
CP0577838
|
US9062070, 79
Show/Hide
|
C23H22FN9O2
|
1
|
1 |
IC50 = 190 nM
|
|
|
CP0426604
|
US9062070, 24
Show/Hide
|
C24H22F2N8O2
|
1
|
1 |
IC50 = 200 nM
|
|
|
CP0488828
|
US9062070, 68
Show/Hide
|
C24H22F2N8O2
|
1
|
1 |
IC50 = 200 nM
|
|
|
CP0506942
|
US9062070, 86
Show/Hide
|
C27H28FN7O4
|
1
|
1 |
IC50 = 200 nM
|
|
|
CP0554825
|
US9062070, 1E
Show/Hide
|
C27H29N7O4
|
1
|
1 |
IC50 = 200 nM
|
|
|
CP0573648
|
US9062070, 87
Show/Hide
|
C27H28FN7O4
|
1
|
1 |
IC50 = 200 nM
|
|
|
CP0529265
|
US9062070, 14
Show/Hide
|
C27H29N7O4
|
1
|
1 |
IC50 = 210 nM
|
|
|
CP0506779
|
US9062070, 52
Show/Hide
|
C25H25FN8O3
|
1
|
1 |
IC50 = 220 nM
|
|
|
CP0563889
|
US9062070, 45
Show/Hide
|
C26H27N7O4
|
1
|
1 |
IC50 = 220 nM
|
|
|
CP0488832
|
US9062070, 101
Show/Hide
|
C26H28N8O3
|
1
|
1 |
IC50 = 230 nM
|
|
|
CP0488818
|
US9062070, 13
Show/Hide
|
C26H27FN8O2
|
1
|
1 |
IC50 = 260 nM
|
|
|
CP0424200
|
US9062070, 63
Show/Hide
|
C25H26N8O3
|
1
|
1 |
IC50 = 270 nM
|
|
|
CP0424202
|
US9062070, 74
Show/Hide
|
C26H28N8O3
|
1
|
1 |
IC50 = 280 nM
|
|
|
CP0450171
|
US9062070, 77
Show/Hide
|
C25H25FN8O3
|
1
|
1 |
IC50 = 290 nM
|
|
|
CP0488830
|
US9062070, 90
Show/Hide
|
C27H28FN7O4
|
1
|
1 |
IC50 = 310 nM
|
|
|
CP0488831
|
US9062070, 92
Show/Hide
|
C25H25FN8OS
|
1
|
1 |
IC50 = 310 nM
|
|
|
CP0424183
|
US9062070, 16
Show/Hide
|
C26H27N7O4
|
1
|
1 |
IC50 = 390 nM
|
|
|
CP0488822
|
US9062070, 39
Show/Hide
|
C25H25FN8O2
|
1
|
1 |
IC50 = 390 nM
|
|
|
CP0577836
|
US9062070, 3
Show/Hide
|
C25H26N8O4
|
1
|
1 |
IC50 = 530 nM
|
|
|
CP0556001
|
US9062070, 46
Show/Hide
|
C27H29N7O4
|
1
|
1 |
IC50 = 540 nM
|
|
|
CP0577837
|
US9062070, 69
Show/Hide
|
C27H29N7O4
|
1
|
1 |
IC50 = 630 nM
|
|
|