| Compound ID |
Compound Name |
Compound Formula |
|
CP0454974
|
N-[(1R)-1-{4-[(2,4-dimethoxyphenyl)methyl]-5-[2-(1H-indol-3-yl)ethyl]-4H-1,2,4-triazol-3-yl}-2-(1H-indol-3-yl)ethyl]piperidine-4-carboxamide
Show/Hide
|
C37H41N7O3
|
1
|
| 1 |
EC50 = 0.6 nM
|
|
|
|
CP0870851
|
(R)-N-(1-(4-(4-methoxybenzyl)-5-phenethyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)piperidine-4-carboxamide
Show/Hide
|
C34H40N6O2
|
1
|
| 1 |
EC50 = 1.6 nM
|
|
|
|
CP0454969
|
N-[(1R)-2-(1H-indol-3-yl)-1-[5-[2-(1H-indol-3-yl)ethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]ethyl]piperidine-4-carboxamide
Show/Hide
|
C36H39N7O2
|
3
|
| 1 |
EC50 = 1.6 nM
|
|
|
| 2 |
EC50 = 3 nM
|
|
|
| 3 |
IC50 = 0.3 nM
|
|
|
|
CP0454968
|
N-[(1R)-2-(1H-indol-3-yl)-1-{5-[2-(1H-indol-3-yl)ethyl]-4-phenyl-4H-1,2,4-triazol-3-yl}ethyl]piperidine-4-carboxamide
Show/Hide
|
C34H35N7O
|
1
|
| 1 |
EC50 = 2.3 nM
|
|
|
|
CP0454970
|
(3S)-N-[(1R)-2-(1H-indol-3-yl)-1-{5-[2-(1H-indol-3-yl)ethyl]-4-[(4-methoxyphenyl)methyl]-4H-1,2,4-triazol-3-yl}ethyl]piperidine-3-carboxamide
Show/Hide
|
C36H39N7O2
|
1
|
| 1 |
EC50 = 2.5 nM
|
|
|
|
CP0420539
|
(R)-N-(1-(5-(2-(1H-indol-3-yl)ethyl)-4-(3-methoxybenzyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide
Show/Hide
|
C34H37N7O2
|
1
|
| 1 |
EC50 = 4 nM
|
|
|
|
CP0510818
|
N-[(1R)-1-{4-[(2,4-dimethoxyphenyl)methyl]-5-[2-(1H-indol-3-yl)ethyl]-4H-1,2,4-triazol-3-yl}-2-(1H-indol-3-yl)ethyl]piperidine-3-carboxamide
Show/Hide
|
C37H41N7O3
|
1
|
| 1 |
EC50 = 5.3 nM
|
|
|
|
CP0454973
|
N-[(1R)-1-{4-benzyl-5-[2-(1H-indol-3-yl)ethyl]-4H-1,2,4-triazol-3-yl}-2-(1H-indol-3-yl)ethyl]piperidine-4-carboxamide
Show/Hide
|
C35H37N7O
|
1
|
| 1 |
EC50 = 5.4 nM
|
|
|
|
CP0424338
|
(2S)-N-[(1R)-2-(1H-indol-3-yl)-1-{5-[2-(1H-indol-3-yl)ethyl]-4-[(4-methoxyphenyl)methyl]-4H-1,2,4-triazol-3-yl}ethyl]pyrrolidine-2-carboxamide
Show/Hide
|
C35H37N7O2
|
1
|
| 1 |
EC50 = 6 nM
|
|
|
|
CP0910551
|
(R)-N-(1-(4-(2,4-dimethoxybenzyl)-5-phenethyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)piperidine-4-carboxamide
Show/Hide
|
C35H42N6O3
|
1
|
| 1 |
EC50 = 6.1 nM
|
|
|
|
CP0434205
|
N-[(1R)-1-{4-[(4-ethylphenyl)methyl]-5-(2-phenylethyl)-4H-1,2,4-triazol-3-yl}-2-(1H-indol-3-yl)ethyl]piperidine-4-carboxamide
Show/Hide
|
C35H40N6O
|
1
|
| 1 |
EC50 = 7.7 nM
|
|
|
|
CP0882982
|
(R,S)-N-((R)-1-(5-((1H-indol-3-yl)methyl)-4-(4-methoxybenzyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)piperazine-2-carboxamide
Show/Hide
|
C35H40N8O2
|
1
|
| 1 |
EC50 = 8.7 nM
|
|
|
|
CP0454971
|
N-[(1R)-1-{4-benzyl-5-[2-(1H-indol-3-yl)ethyl]-4H-1,2,4-triazol-3-yl}-2-(1H-indol-3-yl)ethyl]piperidine-3-carboxamide
Show/Hide
|
C35H37N7O
|
1
|
| 1 |
EC50 = 9.9 nM
|
|
|
|
CP0428458
|
(R)-N-(1-(4-(4-ethylbenzyl)-5-phenethyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide
Show/Hide
|
C33H38N6O
|
1
|
| 1 |
EC50 = 11 nM
|
|
|
|
CP0890894
|
N-((R)-1-(4-(4-methoxybenzyl)-5-phenethyl-4,5-dihydro-1H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)piperazine-2-carboxamide
Show/Hide
|
C33H39N7O2
|
1
|
| 1 |
EC50 = 12 nM
|
|
|
|
CP0457704
|
(R)-N-(1-(5-(2-(1H-indol-3-yl)ethyl)-4-(4-methoxybenzyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)picolinamide
Show/Hide
|
C36H33N7O2
|
1
|
| 1 |
EC50 = 12 nM
|
|
|
|
CP0378565
|
(R)-N-(1-(4-(4-methylbenzyl)-5-(3-phenylpropyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide
Show/Hide
|
C33H38N6O
|
1
|
| 1 |
EC50 = 12 nM
|
|
|
|
CP0879905
|
N-((R)-1-(4-(2,4-dimethoxyphenyl)-5-phenethyl-4,5-dihydro-1H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)piperidine-4-carboxamide
Show/Hide
|
C34H40N6O3
|
1
|
| 1 |
EC50 = 14 nM
|
|
|
|
CP0485811
|
N-[(1R)-1-[4-(4-ethylphenyl)-5-[2-(1H-indol-3-yl)ethyl]-4H-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]piperidine-4-carboxamide
Show/Hide
|
C36H39N7O
|
1
|
| 1 |
EC50 = 15 nM
|
|
|
|
CP0378569
|
(R)-N-(1-(5-(3-(1H-indol-3-yl)propyl)-4-phenethyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide
Show/Hide
|
C35H39N7O
|
1
|
| 1 |
EC50 = 15 nM
|
|
|
|
CP0403076
|
(R)-N-((4-(2,4-dimethoxybenzyl)-5-phenethyl-4H-1,2,4-triazol-3-yl)(1H-indol-3-yl)methyl)benzamide
Show/Hide
|
C35H33N5O3
|
1
|
| 1 |
EC50 = 16 nM
|
|
|
|
CP0475200
|
(R)-N-(1-(5-(3-(1H-indol-3-yl)propyl)-4-(3-methoxybenzyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide
Show/Hide
|
C35H39N7O2
|
1
|
| 1 |
EC50 = 18 nM
|
|
|
|
CP0877433
|
N-((R)-1-(4-(2,4-dimethoxybenzyl)-5-phenethyl-4,5-dihydro-1H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)piperazine-2-carboxamide
Show/Hide
|
C34H41N7O3
|
1
|
| 1 |
EC50 = 19.6 nM
|
|
|
|
CP0378563
|
(R)-2-amino-N-(1-(4-(furan-2-ylmethyl)-5-phenethyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-methylpropanamide
Show/Hide
|
C29H32N6O2
|
1
|
| 1 |
EC50 = 23 nM
|
|
|
|
CP0486752
|
(R)-tetrahydro-2H-pyran-4-yl 1-(5-(2-(1H-indol-3-yl)ethyl)-4-(4-methoxybenzyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethylcarbamate
Show/Hide
|
C36H38N6O4
|
1
|
| 1 |
EC50 = 24 nM
|
|
|
|
CP0486754
|
(S)-tetrahydro-2H-pyran-4-yl 1-(5-(2-(1H-indol-3-yl)ethyl)-4-(4-methoxybenzyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethylcarbamate
Show/Hide
|
C36H38N6O4
|
1
|
| 1 |
EC50 = 24 nM
|
|
|
|
CP0489342
|
(S)-N-(1-(5-(2-(1H-indol-3-yl)ethyl)-4-(4-methoxybenzyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)piperidine-4-carboxamide
Show/Hide
|
C36H39N7O2
|
1
|
| 1 |
EC50 = 32 nM
|
|
|
|
CP0454975
|
(3R)-N-[(1R)-2-(1H-indol-3-yl)-1-{4-[(4-methoxyphenyl)methyl]-5-(2-phenylethyl)-4H-1,2,4-triazol-3-yl}ethyl]piperidine-3-carboxamide
Show/Hide
|
C34H38N6O2
|
1
|
| 1 |
EC50 = 36 nM
|
|
|
|
CP0378577
|
(R)-N-(1-(5-(2-(1H-indol-3-yl)ethyl)-4-phenyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide
Show/Hide
|
C32H33N7O
|
1
|
| 1 |
EC50 = 41 nM
|
|
|
|
CP0419726
|
(R)-N-(1-(4-(3-methoxybenzyl)-5-phenethyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide
Show/Hide
|
C32H36N6O2
|
1
|
| 1 |
EC50 = 45 nM
|
|
|
|
CP0378570
|
(R)-N-(1-(5-(3-(1H-indol-3-yl)propyl)-4-benzyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide
Show/Hide
|
C34H37N7O
|
1
|
| 1 |
EC50 = 49 nM
|
|
|
|
CP0467750
|
(R)-N-(1-(5-(2-(1H-Indol-3-yl)ethyl)-4-benzyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide
Show/Hide
|
C33H35N7O
|
1
|
| 1 |
EC50 = 64 nM
|
|
|
|
CP0489341
|
(R)-pyridin-2-yl 1-(5-(2-(1H-indol-3-yl)ethyl)-4-(4-methoxybenzyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethylcarbamate
Show/Hide
|
C36H33N7O3
|
1
|
| 1 |
EC50 = 75 nM
|
|
|
|
CP0464296
|
(S)-N-(1-(5-(2-(1H-indol-3-yl)ethyl)-4-(4-methoxybenzyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)picolinamide
Show/Hide
|
C36H33N7O2
|
1
|
| 1 |
EC50 = 88 nM
|
|
|
|
CP0436918
|
(R)-N-(1-(4-(2-methoxybenzyl)-5-phenethyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide
Show/Hide
|
C32H36N6O2
|
1
|
| 1 |
EC50 = 98 nM
|
|
|
|
CP0378566
|
(R)-N-(1-(4-(2-(1H-indol-3-yl)ethyl)-5-(3-(1H-indol-3-yl)propyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide
Show/Hide
|
C37H40N8O
|
1
|
| 1 |
EC50 = 140 nM
|
|
|
|
CP0906073
|
N-((R)-1-(4-(4-ethylbenzyl)-5-phenethyl-4,5-dihydro-1H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)piperazine-2-carboxamide
Show/Hide
|
C34H41N7O
|
1
|
| 1 |
EC50 = 143 nM
|
|
|
|
CP0879903
|
N-((R)-1-(4-(furan-2-ylmethyl)-5-phenethyl-4,5-dihydro-1H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)piperidine-4-carboxamide
Show/Hide
|
C31H36N6O2
|
1
|
| 1 |
EC50 = 183 nM
|
|
|
|
CP0495967
|
(R)-N-(1-(5-(2-(1H-indol-3-yl)ethyl)-4-(4-fluorobenzyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide
Show/Hide
|
C33H34FN7O
|
1
|
| 1 |
EC50 = 210 nM
|
|
|
|
CP0906077
|
(R)-N-(1-(4-(4-methoxybenzyl)-5-phenethyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-3-aminopropanamide
Show/Hide
|
C31H36N6O2
|
1
|
| 1 |
EC50 = 256 nM
|
|
|
|
CP0454976
|
(2-aminoethyl)[(1R)-1-{4-[(2,4-dimethoxyphenyl)methyl]-5-(2-phenylethyl)-4H-1,2,4-triazol-3-yl}-2-(1H-indol-3-yl)ethyl]amine
Show/Hide
|
C31H36N6O2
|
1
|
| 1 |
EC50 = 279 nM
|
|
|
|
CP0906075
|
N-((R)-1-(4-(4-methoxybenzyl)-5-phenethyl-4,5-dihydro-1H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)cyclohexanecarboxamide
Show/Hide
|
C35H41N5O2
|
1
|
| 1 |
EC50 = 390 nM
|
|
|
|
CP0897607
|
(S)-N-((S)-1-(5-(2-(1H-indol-3-yl)ethyl)-4-(4-methoxybenzyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)pyrrolidine-2-carboxamide
Show/Hide
|
C35H37N7O2
|
1
|
| 1 |
EC50 = 440 nM
|
|
|
|
CP0511871
|
(R)-N-(1-(5-(2-(1H-indol-2-yl)ethyl)-4-(4-methylbenzyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide
Show/Hide
|
C34H37N7O
|
1
|
| 1 |
EC50 = 630 nM
|
|
|
|
CP0455070
|
(S)-pyridin-2-yl 1-(5-(2-(1H-indol-3-yl)ethyl)-4-(4-methoxybenzyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethylcarbamate
Show/Hide
|
C36H33N7O3
|
1
|
| 1 |
EC50 = 1580 nM
|
|
|
|
CP0865055
|
5-((1R,5S)-8-Acetyl-8-azabicyclo[3.2.1]oct-3-en-3-yl)-2-((benzo[d][1,3]dioxol-5-ylmethyl)amino)-N-(3-chloro-4-methoxybenzyl)nicotinamide
Show/Hide
|
C32H33ClN4O5
|
1
|
| 1 |
IC50 = 0.3 nM
|
|
|
|
CP0884346
|
5-(8-Acetyl-8-azabicyclo[3.2.1]oct-3-en-3-yl)-N-(((S)-2,3-dihydrobenzo[b][1,4]dioxin-2-yl)methyl)-2-(((2,3-dihydrobenzofuran-6-yl)methyl)amino)nicotinamide
Show/Hide
|
C34H36N4O5
|
1
|
| 1 |
IC50 = 0.39 nM
|
|
|
|
CP0873715
|
5-(8-Acetyl-8-azabicyclo[3.2.1]oct-3-en-3-yl)-N-(3-chloro-4-methoxybenzyl)-2-(((2,3-dihydrobenzofuran-6-yl)methyl)amino)nicotinamide
Show/Hide
|
C33H35ClN4O4
|
1
|
| 1 |
IC50 = 0.42 nM
|
|
|
|
CP0849540
|
3-(Difluoromethyl)-4-methylbenzyl 2-((benzo[d][1,3]-dioxol-5-ylmethyl)amino)-5-(3-hydroxy-3-methylbut-1-yn-1-yl)nicotinate
Show/Hide
|
C28H27F2N3O4
|
1
|
| 1 |
IC50 = 0.44 nM
|
|
|
|
CP0229128
|
US8546435, 6
Show/Hide
|
C32H34N6O4
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
|
CP0284845
|
US8546435, 4
Show/Hide
|
C36H35N7O3
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
|
CP0475559
|
N-[(1R)-1-[5-[(1R)-1-acetamido-2-phenylethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]-3-fluoropyridine-2-carboxamide
Show/Hide
|
C36H34FN7O3
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
|
CP0852605
|
5-(3-Acetamido-3-methylbut-1-yn-1-yl)-2-((benzo[d]-[1,3]dioxol-5-ylmethyl)amino)-N-(3-chloro-4-methoxybenzyl)-nicotinamide
Show/Hide
|
C29H29ClN4O5
|
1
|
| 1 |
IC50 = 3 nM
|
|
|
|
CP0126988
|
US8546435, 5
Show/Hide
|
C35H33N7O3
|
1
|
| 1 |
IC50 = 3 nM
|
|
|
|
CP0419825
|
US8546435, 3
Show/Hide
|
C38H36N8O3
|
1
|
| 1 |
IC50 = 3 nM
|
|
|
|
CP0475496
|
US8546435, 7
Show/Hide
|
C35H39N7O4
|
1
|
| 1 |
IC50 = 3 nM
|
|
|
|
CP0455241
|
N-[(1R)-1-[5-[(1R)-1-amino-2-phenylethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]pyridine-2-carboxamide
Show/Hide
|
C34H33N7O2
|
1
|
| 1 |
IC50 = 4 nM
|
|
|
|
CP0475492
|
N-[(1R)-1-[5-[(1R)-1-acetamido-2-phenylethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]-3,4-dihydro-2H-pyran-6-carboxamide
Show/Hide
|
C36H38N6O4
|
1
|
| 1 |
IC50 = 4 nM
|
|
|
|
CP0475493
|
N-[(1R)-1-[5-[(1R)-1-acetamido-2-phenylethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]-4,6-difluoropyridine-2-carboxamide
Show/Hide
|
C36H33F2N7O3
|
1
|
| 1 |
IC50 = 4 nM
|
|
|
|
CP0510760
|
US8546435, 8
Show/Hide
|
C36H40N8O3
|
1
|
| 1 |
IC50 = 19 nM
|
|
|
|
CP0663159
|
5-((1R,5S)-8-acetyl-8-azabicyclo[3.2.1]oct-3-en-3-yl)-N-(((S)-2,3-dihydrobenzo[b][1,4]dioxin-2-yl)methyl)-2-((2,3-dihydrobenzofuran-6-yl)methylamino)nicotinamide
Show/Hide
|
C33H34N4O5
|
1
|
| 1 |
IC50 = 31 nM
|
|
|
|
CP0327955
|
US8546435, 9
Show/Hide
|
C35H38N8O3
|
1
|
| 1 |
IC50 = 33 nM
|
|
|
|
CP0475747
|
2-amino-N-[(1R)-1-[5-[(1R)-1-formamido-2-phenylethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]-2-methylpropanamide
Show/Hide
|
C33H37N7O3
|
1
|
| 1 |
IC50 = 43 nM
|
|
|
|
CP0475494
|
N-[(1R)-1-[5-[(1S)-1-acetamido-2-phenylethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]pyridine-2-carboxamide
Show/Hide
|
C36H35N7O3
|
1
|
| 1 |
IC50 = 70 nM
|
|
|
|
CP0475560
|
N-[(1R)-1-[5-[(1R)-1-acetamido-2-phenylethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]-2-amino-2-methylpropanamide
Show/Hide
|
C34H39N7O3
|
1
|
| 1 |
IC50 = 90 nM
|
|
|
|
CP0475562
|
2-amino-N-[(1R)-1-[5-[(1R)-1-amino-2-(1H-indol-3-yl)ethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]-2-methylpropanamide
Show/Hide
|
C34H38N8O2
|
1
|
| 1 |
IC50 = 90 nM
|
|
|
|
CP0447867
|
2-amino-N-[(1R)-1-[5-[(1R)-1-amino-2-phenylethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]-2-methylpropanamide
Show/Hide
|
C32H37N7O2
|
1
|
| 1 |
IC50 = 135 nM
|
|
|
|
CP0475749
|
N-[(1R)-1-[5-[(1S)-1-amino-2-phenylethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]pyridine-2-carboxamide
Show/Hide
|
C34H33N7O2
|
1
|
| 1 |
IC50 = 150 nM
|
|
|
|
CP0420542
|
2-amino-N-[(1R)-2-(1H-indol-3-yl)-1-{5-[2-(1H-indol-3-yl)ethyl]-4-[(4-methoxyphenyl)methyl]-4H-1,2,4-triazol-3-yl}ethyl]-2-methylpropanamide
Show/Hide
|
C34H37N7O2
|
1
|
| 1 |
IC50 = 190 nM
|
|
|
|
CP0414782
|
N-[(1R)-1-[5-[(1S)-1-acetamido-2-(1H-indol-3-yl)ethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]pyridine-2-carboxamide
Show/Hide
|
C38H36N8O3
|
1
|
| 1 |
IC50 = 190 nM
|
|
|
|
CP0424823
|
(R)-N-(1-(4-(4-methoxybenzyl)-5-phenethyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide
Show/Hide
|
C32H36N6O2
|
1
|
| 1 |
IC50 = 275 nM
|
|
|
|
CP0424824
|
(R)-N-(1-(4-(4-methoxybenzyl)-5-(3-phenylpropyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide
Show/Hide
|
C33H38N6O2
|
1
|
| 1 |
IC50 = 600 nM
|
|
|
|
CP0454068
|
(R)-N-(1-(5-(2-(1H-indol-3-yl)ethyl)-4-(2,4-dimethoxybenzyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide
Show/Hide
|
C35H39N7O3
|
1
|
| 1 |
IC50 = 620 nM
|
|
|
|
CP0454074
|
(R)-N-(1-(4-(2,4-dimethoxybenzyl)-5-phenethyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide
Show/Hide
|
C33H38N6O3
|
1
|
| 1 |
IC50 = 800 nM
|
|
|
|
CP0455074
|
(R)-N-(1-(4-(4-methoxybenzyl)-5-benzyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide
Show/Hide
|
C31H34N6O2
|
1
|
| 1 |
IC50 = 870 nM
|
|
|
|
CP0475561
|
N-[(1R)-1-[5-[(1S)-1-formamido-2-(1H-indol-3-yl)ethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]pyridine-2-carboxamide
Show/Hide
|
C37H34N8O3
|
1
|
| 1 |
IC50 = 1200 nM
|
|
|
|
CP0455042
|
(S)-N-(1-(5-(2-(1H-indol-3-yl)ethyl)-4-(2,4-dimethoxybenzyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide
Show/Hide
|
C35H39N7O3
|
1
|
| 1 |
IC50 = 3200 nM
|
|
|
|
CP0379866
|
N-[(1R)-1-[5-[(1S)-1-acetamido-2-(1H-indol-3-yl)ethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]-2-amino-2-methylpropanamide
Show/Hide
|
C36H40N8O3
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0385352
|
N-[(1R)-1-[5-[(1S)-1-acetamido-2-phenylethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]-2-amino-2-methylpropanamide
Show/Hide
|
C34H39N7O3
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0419823
|
2-amino-N-[(1R)-1-[5-[(1S)-1-amino-2-phenylethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]-2-methylpropanamide
Show/Hide
|
C32H37N7O2
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0561894
|
2-amino-N-[(1R)-1-[5-[(1S)-1-amino-2-(1H-indol-3-yl)ethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]-2-methylpropanamide
Show/Hide
|
C34H38N8O2
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
