| Compound ID |
Compound Name |
Compound Formula |
|
CP0396582
|
N-[3-[5-methoxy-2-[2-(3-methoxyphenyl)ethyl]phenyl]propyl]propanamide
Show/Hide
|
C22H29NO3
|
2
|
| 1 |
EC50 = 0.024 nM
|
|
|
| 2 |
Ki = 0.55 nM
|
|
|
|
CP0409354
|
N-[3-[5-methoxy-2-[(3-methoxyphenyl)methoxy]phenyl]propyl]propanamide
Show/Hide
|
C21H27NO4
|
3
|
| 1 |
EC50 = 0.05 nM
|
|
|
| 2 |
Ki = 0.291 nM
|
|
|
| 3 |
Ki = 1.698 nM
|
|
|
|
CP0444081
|
N-[2-(2-ethoxy-7,8-dihydrofuro[2,3-g]benzimidazol-1-yl)ethyl]acetamide
Show/Hide
|
C15H19N3O3
|
2
|
| 1 |
EC50 = 0.05 nM
|
|
|
| 2 |
Ki = 0.24 nM
|
|
|
|
CP0520740
|
N-[2-(2-methoxy-7,8-dihydrofuro[2,3-g]benzimidazol-1-yl)ethyl]acetamide
Show/Hide
|
C14H17N3O3
|
2
|
| 1 |
EC50 = 0.06 nM
|
|
|
| 2 |
Ki = 0.38 nM
|
|
|
|
CP0034701
|
N-[2-(5-methoxy-1H-indol-3-yl)ethyl]acetamide
Show/Hide
|
C13H16N2O2
|
19
|
| 1 |
EC50 = 0.069 nM
|
|
|
| 2 |
EC50 = 0.07 nM
|
|
|
| 3 |
EC50 = 0.42 nM
|
|
|
| 4 |
EC50 = 0.47 nM
|
|
|
| 5 |
EC50 = 0.49 nM
|
|
|
| 6 |
EC50 = 0.82 nM
|
|
|
| 7 |
EC50 = 0.8511 nM
|
|
|
| 8 |
Ki = 0.12 nM
|
|
|
| 9 |
Ki = 0.13 nM
|
|
|
| 10 |
Ki = 0.15 nM
|
|
|
| 11 |
Ki = 0.21 nM
|
|
|
| 12 |
Ki = 0.23 nM
|
|
|
| 13 |
Ki = 0.29 nM
|
|
|
| 14 |
Ki = 0.35 nM
|
|
|
| 15 |
Ki = 0.41 nM
|
|
|
| 16 |
Ki = 0.429 nM
|
|
|
| 17 |
Ki = 0.52 nM
|
|
|
| 18 |
Ki = 0.741 nM
|
|
|
| 19 |
Ki = 0.955 nM
|
|
|
|
CP0178199
|
Agomelatine
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|
C15H17NO2
|
7
|
| 1 |
EC50 = 0.06918 nM
|
|
|
| 2 |
EC50 = 0.1 nM
|
|
|
| 3 |
EC50 = 0.18 nM
|
|
|
| 4 |
Ki = 0.2 nM
|
|
|
| 5 |
Ki = 0.21 nM
|
|
|
| 6 |
Ki = 0.27 nM
|
|
|
| 7 |
Ki = 0.3802 nM
|
|
|
|
CP0454903
|
1-[2-(2-methoxyquinolin-8-yl)ethyl]-3-methylurea
Show/Hide
|
C14H17N3O2
|
1
|
| 1 |
EC50 = 0.09 nM
|
|
|
|
CP0548271
|
N-[2-(2-ethoxy-6-methoxybenzimidazol-1-yl)ethyl]butanamide
Show/Hide
|
C16H23N3O3
|
2
|
| 1 |
EC50 = 0.09 nM
|
|
|
| 2 |
Ki = 0.28 nM
|
|
|
|
CP0045783
|
N-[2-(5-methoxy-2-phenyl-1-benzofuran-3-yl)ethyl]acetamide
Show/Hide
|
C19H19NO3
|
1
|
| 1 |
EC50 = 0.096 nM
|
|
|
|
CP0454899
|
1-[2-(2-methoxyquinolin-8-yl)ethyl]-3-methylthiourea
Show/Hide
|
C14H17N3OS
|
1
|
| 1 |
EC50 = 0.1 nM
|
|
|
|
CP0396581
|
N-[3-[5-methoxy-2-[2-(3-methoxyphenyl)ethynyl]phenyl]propyl]propanamide
Show/Hide
|
C22H25NO3
|
2
|
| 1 |
EC50 = 0.11 nM
|
|
|
| 2 |
Ki = 0.073 nM
|
|
|
|
CP0214091
|
But-3-enoic acid [2-(2-benzyl-5-methoxy-benzofuran-3-yl)-ethyl]-amide
Show/Hide
|
C22H23NO3
|
1
|
| 1 |
EC50 = 0.17 nM
|
|
|
|
CP0534038
|
N-[2-(2-ethoxy-6-methoxybenzimidazol-1-yl)ethyl]propanamide
Show/Hide
|
C15H21N3O3
|
2
|
| 1 |
EC50 = 0.19 nM
|
|
|
| 2 |
Ki = 1.4 nM
|
|
|
|
CP0417995
|
N-[3-[5-methoxy-2-(3-methoxyphenyl)phenyl]propyl]propanamide
Show/Hide
|
C20H25NO3
|
2
|
| 1 |
EC50 = 0.2 nM
|
|
|
| 2 |
Ki = 0.339 nM
|
|
|
|
CP0428960
|
2-(2-methoxyquinolin-8-yl)ethylurea
Show/Hide
|
C13H15N3O2
|
1
|
| 1 |
EC50 = 0.2 nM
|
|
|
|
CP0428961
|
1-ethyl-3-[2-(2-methoxyquinolin-8-yl)ethyl]urea
Show/Hide
|
C15H19N3O2
|
1
|
| 1 |
EC50 = 0.2 nM
|
|
|
|
CP0428962
|
N-[2-(2-methoxyquinolin-8-yl)ethyl]acetamide
Show/Hide
|
C14H16N2O2
|
1
|
| 1 |
EC50 = 0.2 nM
|
|
|
|
CP0429915
|
N-[(8-methoxy-1-methyl-2,3-dihydrocyclopenta[a]naphthalen-1-yl)methyl]acetamide
Show/Hide
|
C18H21NO2
|
2
|
| 1 |
EC50 = 0.2 nM
|
|
|
| 2 |
Ki = 0.1 nM
|
|
|
|
CP0459154
|
N-[(8-methoxy-2,3-dihydro-1H-cyclopenta[a]naphthalen-1-yl)methyl]acetamide
Show/Hide
|
C17H19NO2
|
2
|
| 1 |
EC50 = 0.2 nM
|
|
|
| 2 |
Ki = 0.2 nM
|
|
|
|
CP0514069
|
N-[3-[5-methoxy-2-[(3-methoxyphenyl)methyl]phenyl]propyl]propanamide
Show/Hide
|
C21H27NO3
|
2
|
| 1 |
EC50 = 0.24 nM
|
|
|
| 2 |
Ki = 3.39 nM
|
|
|
|
CP0534080
|
N-[2-(2-ethoxy-6-methoxybenzimidazol-1-yl)ethyl]acetamide
Show/Hide
|
C14H19N3O3
|
2
|
| 1 |
EC50 = 0.26 nM
|
|
|
| 2 |
Ki = 0.93 nM
|
|
|
|
CP0419698
|
US10781182, Compound IA2-121
Show/Hide
|
C14H18ClN3O3
|
2
|
| 1 |
EC50 = 0.27 nM
|
|
|
| 2 |
Ki = 0.93 nM
|
|
|
|
CP0485368
|
1-ethyl-3-[(8-methoxy-1-methyl-2,3-dihydrocyclopenta[a]naphthalen-1-yl)methyl]urea
Show/Hide
|
C19H24N2O2
|
2
|
| 1 |
EC50 = 0.3 nM
|
|
|
| 2 |
Ki = 0.3 nM
|
|
|
|
CP0419699
|
US10781182, Compound IA2-142
Show/Hide
|
C15H20ClN3O3
|
2
|
| 1 |
EC50 = 0.3 nM
|
|
|
| 2 |
Ki = 1.6 nM
|
|
|
|
CP0444082
|
US10781182, Compound IA2-120
Show/Hide
|
C15H21N3O3
|
2
|
| 1 |
EC50 = 0.35 nM
|
|
|
| 2 |
Ki = 4.5 nM
|
|
|
|
CP0847772
|
2,2-difluoro-N-(3-hydroxy-2-(7-methoxynaphthalen-1-yl)propyl)acetamide
Show/Hide
|
C16H17F2NO3
|
2
|
| 1 |
EC50 = 0.3715 nM
|
|
|
| 2 |
Ki = 0.3467 nM
|
|
|
|
CP0192453
|
But-3-enoic acid {2-[5-methoxy-2-(3-methoxy-benzyl)-benzofuran-3-yl]-ethyl}-amide
Show/Hide
|
C23H25NO4
|
1
|
| 1 |
EC50 = 0.39 nM
|
|
|
|
CP0454898
|
methyl N-[2-(2-methoxyquinolin-8-yl)ethyl]carbamate
Show/Hide
|
C14H16N2O3
|
1
|
| 1 |
EC50 = 0.4 nM
|
|
|
|
CP0429916
|
2-methoxy-N-[(8-methoxy-2,3-dihydro-1H-cyclopenta[a]naphthalen-1-yl)methyl]acetamide
Show/Hide
|
C18H21NO3
|
2
|
| 1 |
EC50 = 0.4 nM
|
|
|
| 2 |
Ki = 0.1 nM
|
|
|
|
CP0217078
|
N-[2-[5-methoxy-2-[(2-methoxyphenyl)methyl]-1-benzofuran-3-yl]ethyl]acetamide
Show/Hide
|
C21H23NO4
|
1
|
| 1 |
EC50 = 0.41 nM
|
|
|
|
CP0418574
|
N-[2-[7-methoxy-3-[3-(methylamino)phenyl]naphthalen-1-yl]ethyl]acetamide
Show/Hide
|
C22H24N2O2
|
2
|
| 1 |
EC50 = 0.5 nM
|
|
|
| 2 |
Ki = 0.51 nM
|
|
|
|
CP0565247
|
N-[2-(2,6-dimethoxybenzimidazol-1-yl)ethyl]acetamide
Show/Hide
|
C13H17N3O3
|
2
|
| 1 |
EC50 = 0.52 nM
|
|
|
| 2 |
Ki = 3.1 nM
|
|
|
|
CP0380668
|
N-[2-(4-ethyl-10-oxa-5,6-diazatricyclo[7.3.0.02,6]dodeca-1(9),2,4,7-tetraen-3-yl)ethyl]acetamide
Show/Hide
|
C15H19N3O2
|
2
|
| 1 |
EC50 = 0.53 nM
|
|
|
| 2 |
Ki = 0.42 nM
|
|
|
|
CP0419697
|
N-[2-(2-ethoxy-6-methoxybenzimidazol-1-yl)ethyl]cyclopropanecarboxamide
Show/Hide
|
C16H21N3O3
|
2
|
| 1 |
EC50 = 0.56 nM
|
|
|
| 2 |
Ki = 3.9 nM
|
|
|
|
CP0401351
|
N-[2-[3-[3-(hydroxymethyl)phenyl]-7-methoxynaphthalen-1-yl]ethyl]butanamide
Show/Hide
|
C24H27NO3
|
2
|
| 1 |
EC50 = 0.6 nM
|
|
|
| 2 |
Ki = 0.28 nM
|
|
|
|
CP0877970
|
rac-2-fluoro-N-(3-hydroxy-2-(7-methoxynaphthalen-1-yl)propyl)acetamide
Show/Hide
|
C16H18FNO3
|
2
|
| 1 |
EC50 = 0.631 nM
|
|
|
| 2 |
Ki = 0.537 nM
|
|
|
|
CP0424931
|
N-[2-[5-fluoro-2-(4-fluorophenyl)sulfanyl-1-benzothiophen-3-yl]ethyl]acetamide
Show/Hide
|
C18H15F2NOS2
|
2
|
| 1 |
EC50 = 0.64 nM
|
|
|
| 2 |
Ki = 0.87 nM
|
|
|
|
CP0452012
|
N-[2-(5-fluoro-1-benzothiophen-3-yl)ethyl]acetamide
Show/Hide
|
C12H12FNOS
|
2
|
| 1 |
EC50 = 0.68 nM
|
|
|
| 2 |
Ki = 4.87 nM
|
|
|
|
CP0401365
|
N-[2-[3-[3-(hydroxymethyl)phenyl]-7-methoxynaphthalen-1-yl]ethyl]propanamide
Show/Hide
|
C23H25NO3
|
2
|
| 1 |
EC50 = 0.7 nM
|
|
|
| 2 |
Ki = 0.52 nM
|
|
|
|
CP0462764
|
N-[2-(6-methoxypyrrolo[2,3-b]pyridin-1-yl)ethyl]butanamide
Show/Hide
|
C14H19N3O2
|
1
|
| 1 |
EC50 = 0.7 nM
|
|
|
|
CP0121891
|
N-[2-(8-methoxybenzo[e][1]benzofuran-1-yl)ethyl]acetamide
Show/Hide
|
C17H17NO3
|
2
|
| 1 |
EC50 = 0.7 nM
|
|
|
| 2 |
Ki = 0.09 nM
|
|
|
|
CP0406657
|
3-(2-methoxyquinolin-8-yl)-N-methylpropanamide
Show/Hide
|
C14H16N2O2
|
1
|
| 1 |
EC50 = 0.7 nM
|
|
|
|
CP0414939
|
1-[(8-methoxy-1-methyl-2,3-dihydrocyclopenta[a]naphthalen-1-yl)methyl]-3-propylurea
Show/Hide
|
C20H26N2O2
|
2
|
| 1 |
EC50 = 0.7 nM
|
|
|
| 2 |
Ki = 0.2 nM
|
|
|
|
CP0098513
|
N-[2-[5-methoxy-2-[(3-methoxyphenyl)methyl]-1-benzofuran-3-yl]ethyl]acetamide
Show/Hide
|
C21H23NO4
|
2
|
| 1 |
EC50 = 0.72 nM
|
|
|
| 2 |
Ki = 0.25 nM
|
|
|
|
CP0458570
|
N-[2-[3-[3-(hydroxymethyl)phenyl]-7-methoxynaphthalen-1-yl]ethyl]acetamide
Show/Hide
|
C22H23NO3
|
2
|
| 1 |
EC50 = 0.76 nM
|
|
|
| 2 |
Ki = 0.36 nM
|
|
|
|
CP0548268
|
N-[2-(6-methoxy-2-methylsulfanylbenzimidazol-1-yl)ethyl]acetamide
Show/Hide
|
C13H17N3O2S
|
2
|
| 1 |
EC50 = 0.76 nM
|
|
|
| 2 |
Ki = 3.2 nM
|
|
|
|
CP0847771
|
(R)-2-fluoro-N-(3-hydroxy-2-(7-methoxynaphthalen-1-yl)propyl)acetamide
Show/Hide
|
C16H18FNO3
|
2
|
| 1 |
EC50 = 0.7943 nM
|
|
|
| 2 |
Ki = 0.9772 nM
|
|
|
|
CP0488406
|
3-(2-methoxyquinolin-8-yl)-N-methylsulfonylpropanamide
Show/Hide
|
C14H16N2O4S
|
1
|
| 1 |
EC50 = 0.8 nM
|
|
|
|
CP0450973
|
US10781182, Compound IA2-143
Show/Hide
|
C13H16ClN3O3
|
2
|
| 1 |
EC50 = 0.86 nM
|
|
|
| 2 |
Ki = 0.8 nM
|
|
|
|
CP0410497
|
(8-methoxy-2,3-dihydro-1H-cyclopenta[a]naphthalen-1-yl)methylurea
Show/Hide
|
C16H18N2O2
|
2
|
| 1 |
EC50 = 0.9 nM
|
|
|
| 2 |
Ki = 0.1 nM
|
|
|
|
CP0105645
|
N-[(8-methoxybenzo[e][1]benzofuran-2-yl)methyl]cyclopropanecarboxamide
Show/Hide
|
C18H17NO3
|
2
|
| 1 |
EC50 = 0.98 nM
|
|
|
| 2 |
Ki = 0.6 nM
|
|
|
|
CP0414625
|
N-[(8-methoxybenzo[e][1]benzofuran-2-yl)methyl]acetamide
Show/Hide
|
C16H15NO3
|
2
|
| 1 |
EC50 = 0.98 nM
|
|
|
| 2 |
Ki = 0.4 nM
|
|
|
|
CP0433987
|
N-[2-[3-[3-(bromomethyl)phenyl]-7-methoxynaphthalen-1-yl]ethyl]acetamide
Show/Hide
|
C22H22BrNO2
|
2
|
| 1 |
EC50 = 1 nM
|
|
|
| 2 |
Ki = 0.56 nM
|
|
|
|
CP0432632
|
N-(1-phenyl-3,4-dihydro-2H-quinolin-3-yl)propanamide
Show/Hide
|
C18H20N2O
|
2
|
| 1 |
EC50 = 1 nM
|
|
|
| 2 |
Ki = 2 nM
|
|
|
|
CP0405073
|
N-[(8-methoxy-2,3-dihydro-1H-cyclopenta[a]naphthalen-1-yl)methyl]methanesulfonamide
Show/Hide
|
C16H19NO3S
|
2
|
| 1 |
EC50 = 1 nM
|
|
|
| 2 |
Ki = 0.1 nM
|
|
|
|
CP0458757
|
4-azamelatonin
Show/Hide
|
C12H15N3O2
|
1
|
| 1 |
EC50 = 1.1 nM
|
|
|
|
CP0121949
|
2-fluoro-N-[(8-methoxybenzo[e][1]benzofuran-2-yl)methyl]acetamide
Show/Hide
|
C16H14FNO3
|
2
|
| 1 |
EC50 = 1.1 nM
|
|
|
| 2 |
Ki = 0.7 nM
|
|
|
|
CP0474650
|
1-ethyl-3-[2-(2-methoxyquinolin-8-yl)ethyl]thiourea
Show/Hide
|
C15H19N3OS
|
1
|
| 1 |
EC50 = 1.1 nM
|
|
|
|
CP0847773
|
(R)-N-(3-hydroxy-2-(7-methoxynaphthalen-1-yl)propyl)propionamide
Show/Hide
|
C17H21NO3
|
2
|
| 1 |
EC50 = 1.259 nM
|
|
|
| 2 |
Ki = 0.3162 nM
|
|
|
|
CP0301499
|
N-[2-[5-methoxy-2-[[3-(trifluoromethyl)phenyl]methyl]-1-benzofuran-3-yl]ethyl]acetamide
Show/Hide
|
C21H20F3NO3
|
1
|
| 1 |
EC50 = 1.26 nM
|
|
|
|
CP0387872
|
N-[2-[3-(3-formylphenyl)-7-methoxynaphthalen-1-yl]ethyl]acetamide
Show/Hide
|
C22H21NO3
|
2
|
| 1 |
EC50 = 1.3 nM
|
|
|
| 2 |
Ki = 0.42 nM
|
|
|
|
CP0418572
|
N-[2-[3-(3-aminophenyl)-7-methoxynaphthalen-1-yl]ethyl]acetamide
Show/Hide
|
C21H22N2O2
|
2
|
| 1 |
EC50 = 1.3 nM
|
|
|
| 2 |
Ki = 0.27 nM
|
|
|
|
CP0486875
|
N-[2-(2-methoxy-5,6,7,8-tetrahydropyrido[2,3-b]indol-9-yl)ethyl]acetamide
Show/Hide
|
C16H21N3O2
|
1
|
| 1 |
EC50 = 1.3 nM
|
|
|
|
CP0377934
|
N-[2-[7-(cyclohexylmethyl)-2,6-dihydro-1H-cyclopenta[e][1]benzofuran-8-yl]ethyl]acetamide
Show/Hide
|
C22H29NO2
|
2
|
| 1 |
EC50 = 1.318 nM
|
|
|
| 2 |
Ki = 0.012 nM
|
|
|
|
CP0462765
|
N-[2-(6-methoxypyrrolo[2,3-b]pyridin-1-yl)ethyl]propanamide
Show/Hide
|
C13H17N3O2
|
1
|
| 1 |
EC50 = 1.4 nM
|
|
|
|
CP0406180
|
N-[(8-methoxybenzo[e][1]benzofuran-1-yl)methyl]acetamide
Show/Hide
|
C16H15NO3
|
2
|
| 1 |
EC50 = 1.4 nM
|
|
|
| 2 |
Ki = 0.7 nM
|
|
|
|
CP0435113
|
N-[2-[3-[3-(dimethylamino)phenyl]-7-methoxynaphthalen-1-yl]ethyl]acetamide
Show/Hide
|
C23H26N2O2
|
2
|
| 1 |
EC50 = 1.5 nM
|
|
|
| 2 |
Ki = 0.94 nM
|
|
|
|
CP0469375
|
1-ethyl-3-[(8-methoxy-1-methyl-2,3-dihydrocyclopenta[a]naphthalen-1-yl)methyl]thiourea
Show/Hide
|
C19H24N2OS
|
2
|
| 1 |
EC50 = 2 nM
|
|
|
| 2 |
Ki = 3 nM
|
|
|
|
CP0548270
|
US10781182, Compound IA2-140
Show/Hide
|
C14H19N3O3
|
2
|
| 1 |
EC50 = 2.01 nM
|
|
|
| 2 |
Ki = 11 nM
|
|
|
|
CP0467650
|
N-[2-(6-methoxypyrrolo[2,3-b]pyridin-1-yl)ethyl]acetamide
Show/Hide
|
C12H15N3O2
|
1
|
| 1 |
EC50 = 2.1 nM
|
|
|
|
CP0436558
|
N-[2-[5-fluoro-2-(4-fluorophenyl)sulfanyl-1-benzothiophen-3-yl]ethyl]but-3-enamide
Show/Hide
|
C20H17F2NOS2
|
2
|
| 1 |
EC50 = 2.15 nM
|
|
|
| 2 |
Ki = 0.24 nM
|
|
|
|
CP0399205
|
N-[2-(7-methoxy-3-phenylnaphthalen-1-yl)ethyl]acetamide
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C21H21NO2
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2
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| 1 |
EC50 = 2.4 nM
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| 2 |
Ki = 0.37 nM
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CP0419695
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N-[2-(2-ethoxy-6-methoxybenzimidazol-1-yl)ethyl]cyclobutanecarboxamide
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C17H23N3O3
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2
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| 1 |
EC50 = 2.49 nM
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| 2 |
Ki = 23 nM
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CP0877971
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rac-N-(1-hydroxy-3-(7-methoxynaphthalen-1-yl)propan-2-yl)propionamide
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C17H21NO3
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2
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| 1 |
EC50 = 2.754 nM
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| 2 |
Ki = 2.951 nM
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CP0385360
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3-(5-methoxy-1H-indol-3-yl)-N-prop-2-ynylpropanamide
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C15H16N2O2
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2
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| 1 |
EC50 = 3 nM
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| 2 |
Ki = 1 nM
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CP0389221
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N-[(1-benzyl-3,4-dihydro-2H-quinolin-3-yl)methyl]acetamide
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C19H22N2O
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2
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| 1 |
EC50 = 3 nM
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| 2 |
Ki = 1 nM
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CP0416460
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1-ethyl-3-[(8-methoxy-2,3-dihydro-1H-cyclopenta[a]naphthalen-1-yl)methyl]urea
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C18H22N2O2
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2
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| 1 |
EC50 = 3 nM
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| 2 |
Ki = 0.1 nM
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CP0429921
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1-[(8-methoxy-1-methyl-2,3-dihydrocyclopenta[a]naphthalen-1-yl)methyl]-3-methylthiourea
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C18H22N2OS
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2
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| 1 |
EC50 = 3 nM
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| 2 |
Ki = 0.2 nM
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CP0121948
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N-[2-(8-methoxybenzo[e][1]benzofuran-1-yl)ethyl]cyclopropanecarboxamide
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C19H19NO3
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2
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| 1 |
EC50 = 3.2 nM
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| 2 |
Ki = 13.3 nM
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CP0309822
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2-fluoro-N-[(8-methoxybenzo[e][1]benzofuran-1-yl)methyl]acetamide
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C16H14FNO3
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2
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| 1 |
EC50 = 3.4 nM
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| 2 |
Ki = 2.1 nM
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CP0405083
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1-[(8-methoxy-1-methyl-2,3-dihydrocyclopenta[a]naphthalen-1-yl)methyl]-3-propylthiourea
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C20H26N2OS
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2
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| 1 |
EC50 = 4 nM
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| 2 |
Ki = 0.3 nM
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CP0429925
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(8-methoxy-2,3-dihydro-1H-cyclopenta[a]naphthalen-1-yl)methylthiourea
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C16H18N2OS
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2
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| 1 |
EC50 = 5 nM
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| 2 |
Ki = 0.4 nM
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CP0429929
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methyl N-[(8-methoxy-2,3-dihydro-1H-cyclopenta[a]naphthalen-1-yl)methyl]carbamate
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C17H19NO3
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2
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| 1 |
EC50 = 5 nM
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| 2 |
Ki = 0.4 nM
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CP0381571
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5-[2-(5-methoxy-1H-indol-3-yl)ethyl]-3H-1,3,4-oxadiazol-2-one
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C13H13N3O3
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3
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| 1 |
EC50 = 5.5 nM
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| 2 |
EC50 = 29 nM
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| 3 |
Ki = 4 nM
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CP0414626
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N-[2-(8-methoxybenzo[e][1]benzofuran-2-yl)ethyl]cyclopropanecarboxamide
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C19H19NO3
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2
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| 1 |
EC50 = 5.8 nM
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| 2 |
Ki = 11 nM
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CP0429918
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1-[(8-methoxy-2,3-dihydro-1H-cyclopenta[a]naphthalen-1-yl)methyl]-3-methylthiourea
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C17H20N2OS
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1
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| 1 |
EC50 = 6 nM
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CP0105646
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1-ethyl-3-[2-(8-methoxybenzo[e][1]benzofuran-1-yl)ethyl]urea
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C18H20N2O3
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2
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| 1 |
EC50 = 6.2 nM
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| 2 |
Ki = 226 nM
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CP0426377
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N-[(1-ethyl-3,4-dihydro-2H-quinolin-3-yl)methyl]acetamide
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C14H20N2O
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2
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| 1 |
EC50 = 7 nM
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| 2 |
Ki = 1 nM
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CP0452013
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2-bromo-N-[2-[5-fluoro-2-(4-fluorophenyl)sulfanyl-1-benzothiophen-3-yl]ethyl]acetamide
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C18H14BrF2NOS2
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2
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| 1 |
EC50 = 7.27 nM
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| 2 |
Ki = 5.21 nM
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CP0847750
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(S)-N-(1-hydroxy-3-(7-methoxynaphthalen-1-yl)propan-2-yl)propionamide
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C17H21NO3
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2
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| 1 |
EC50 = 7.413 nM
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| 2 |
Ki = 5.495 nM
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CP0309821
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N-[(8-methoxybenzo[e][1]benzofuran-1-yl)methyl]cyclopropanecarboxamide
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C18H17NO3
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2
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| 1 |
EC50 = 8.8 nM
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| 2 |
Ki = 15 nM
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CP0472545
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N-[(8-methoxybenzo[e][1]benzofuran-1-yl)methyl]-2-methylpropanamide
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C18H19NO3
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2
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| 1 |
EC50 = 8.8 nM
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| 2 |
Ki = 24 nM
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CP0072976
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N-[2-[2-(cyclohexylmethyl)-5-methoxy-1-benzofuran-3-yl]ethyl]acetamide
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C20H27NO3
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1
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| 1 |
EC50 = 10 nM
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CP0436038
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N-[2-[6-methoxy-3-(2,2,2-trifluoroacetyl)pyrrolo[2,3-b]pyridin-1-yl]ethyl]acetamide
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C14H14F3N3O3
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1
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| 1 |
EC50 = 10 nM
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CP0443574
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1-ethyl-3-[(8-methoxybenzo[e][1]benzofuran-2-yl)methyl]urea
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C17H18N2O3
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2
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| 1 |
EC50 = 10 nM
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| 2 |
Ki = 4.2 nM
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CP0389226
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N-[(1-methyl-3,4-dihydro-2H-quinolin-3-yl)methyl]acetamide
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C13H18N2O
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2
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| 1 |
EC50 = 10 nM
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| 2 |
Ki = 15 nM
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CP0467651
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N-[2-(3-iodo-6-methoxypyrrolo[2,3-b]pyridin-1-yl)ethyl]acetamide
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C12H14IN3O2
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1
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| 1 |
EC50 = 11 nM
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CP0381574
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3-(5-methoxy-1H-indol-3-yl)-N-prop-2-enylpropanamide
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C15H18N2O2
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2
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| 1 |
EC50 = 11 nM
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| 2 |
Ki = 0.45 nM
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CP0297769
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N-[2-[5-ethyl-2-[(3-methoxyphenyl)methyl]-1-benzofuran-3-yl]ethyl]acetamide
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C22H25NO3
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1
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| 1 |
EC50 = 19 nM
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CP0391337
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1-[(8-methoxy-2,3-dihydro-1H-cyclopenta[a]naphthalen-1-yl)methyl]-3-propylurea
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C19H24N2O2
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2
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| 1 |
EC50 = 20 nM
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| 2 |
Ki = 0.2 nM
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CP0430453
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N-[2-[7-[4-[[3-(2-acetamidoethyl)-1-benzothiophen-5-yl]oxy]butoxy]naphthalen-1-yl]ethyl]acetamide
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C30H34N2O4S
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2
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| 1 |
EC50 = 20.6 nM
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| 2 |
Ki = 16.9 nM
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CP0877969
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(S)-2-fluoro-N-(3-hydroxy-2-(7-methoxynaphthalen-1-yl)propyl)acetamide
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C16H18FNO3
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2
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| 1 |
EC50 = 25.12 nM
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| 2 |
Ki = 52.48 nM
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CP0469064
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N-[2-[7-[4-[4-[4-(hydroxymethyl)phenyl]phenoxy]butoxy]naphthalen-1-yl]ethyl]acetamide
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C31H33NO4
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2
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| 1 |
EC50 = 26 nM
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| 2 |
Ki = 6.53 nM
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CP0373468
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N-[2-[7-[4-[8-[2-(but-3-enoylamino)ethyl]naphthalen-2-yl]oxybutoxy]naphthalen-1-yl]ethyl]but-3-enamide
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C36H40N2O4
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2
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| 1 |
EC50 = 40.2 nM
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| 2 |
Ki = 10.9 nM
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CP0405082
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1-ethyl-3-[(8-methoxy-2,3-dihydro-1H-cyclopenta[a]naphthalen-1-yl)methyl]thiourea
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C18H22N2OS
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2
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| 1 |
EC50 = 50 nM
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| 2 |
Ki = 2 nM
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CP0389326
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2-[(5-methoxy-1H-indol-3-yl)methyl]-5-methyl-1,3,4-oxadiazole
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C13H13N3O2
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2
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| 1 |
EC50 = 71 nM
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| 2 |
Ki = 16 nM
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CP0432631
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N-[[1-(2-phenylethyl)-3,4-dihydro-2H-quinolin-3-yl]methyl]acetamide
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C20H24N2O
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2
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| 1 |
EC50 = 80 nM
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| 2 |
Ki = 47 nM
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CP0382347
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2-(5-methoxy-1H-indol-3-yl)-N-prop-2-ynylacetamide
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C14H14N2O2
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2
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| 1 |
EC50 = 81 nM
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| 2 |
Ki = 3.8 nM
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CP0407040
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methyl 2-[6-[4-[8-(2-acetamidoethyl)naphthalen-2-yl]oxybutoxy]naphthalen-2-yl]propanoate
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C32H35NO5
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2
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| 1 |
EC50 = 88 nM
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| 2 |
Ki = 4.22 nM
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CP0401209
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N-ethyl-5-[(5-methoxy-1H-indol-3-yl)methyl]-1,3,4-thiadiazol-2-amine
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C14H16N4OS
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2
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| 1 |
EC50 = 110 nM
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| 2 |
Ki = 17 nM
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CP0071154
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2-(5-methoxy-1H-indol-3-yl)-N,N-dimethyl-ethanamine
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C13H18N2O
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2
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| 1 |
EC50 = 112 nM
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| 2 |
Ki = 16 nM
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CP0398561
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2-((S)-1'-((3S,4R)-1-tert-butyl-4-(2,4-difluorophenyl)pyrrolidine-3-carbonyl)-6-chloro-5-methyl-3H-spiro[isobenzofuran-1,4'-piperidine]-3-yl)-2-methylpropanenitrile
Show/Hide
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C32H38ClF2N3O2
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1
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| 1 |
EC50 = 115 nM
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CP0397791
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2-(5-methoxy-1H-indol-3-yl)-N-prop-2-enylacetamide
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C14H16N2O2
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2
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| 1 |
EC50 = 132 nM
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| 2 |
Ki = 4.9 nM
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CP0401703
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N-[2-[7-[4-[8-[2-(cyclopropanecarbonylamino)ethyl]naphthalen-2-yl]oxybutoxy]naphthalen-1-yl]ethyl]cyclopropanecarboxamide
Show/Hide
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C36H40N2O4
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2
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| 1 |
EC50 = 134 nM
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| 2 |
Ki = 13.6 nM
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CP0378677
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N-[3-hydroxy-2-(7-methoxynaphthalen-1-yl)propyl]acetamide
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C16H19NO3
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2
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| 1 |
EC50 = 144.54 nM
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| 2 |
Ki = 13.8 nM
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CP0400794
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2-[6-[4-[8-(2-acetamidoethyl)naphthalen-2-yl]oxybutoxy]naphthalen-2-yl]propanoic acid
Show/Hide
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C31H33NO5
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2
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| 1 |
EC50 = 161 nM
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| 2 |
Ki = 59.1 nM
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CP0415246
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2-((S)-6-chloro-1'-((3S,4R)-4-(2,4-difluorophenyl)-1-isopropylpyrrolidine-3-carbonyl)-5-methyl-3H-spiro[isobenzofuran-1,4'-piperidine]-3-yl)-2-methylpropanenitrile
Show/Hide
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C31H36ClF2N3O2
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1
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| 1 |
EC50 = 295 nM
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CP0382351
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5-[(5-methoxy-1H-indol-3-yl)methyl]-3-methyl-1,2,4-oxadiazole
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C13H13N3O2
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2
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| 1 |
EC50 = 295 nM
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| 2 |
Ki = 44 nM
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CP0493345
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2-((S)-6-chloro-1'-((3S,4R)-4-(2,4-difluorophenyl)-1-(1-hydroxy-2-methylpropan-2-yl)pyrrolidine-3-carbonyl)-5-methyl-3H-spiro[isobenzofuran-1,4'-piperidine]-3-yl)-2-methylpropanenitrile
Show/Hide
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C32H38ClF2N3O3
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1
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| 1 |
EC50 = 342.9 nM
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CP0436037
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7-azamelatonin
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C12H15N3O2
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1
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| 1 |
EC50 = 380 nM
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CP0400796
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N-[2-[7-[4-[8-(2-acetamidoethyl)naphthalen-2-yl]oxybutoxy]naphthalen-1-yl]ethyl]acetamide
Show/Hide
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C32H36N2O4
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3
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| 1 |
EC50 = 405 nM
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| 2 |
Ki = 72.7 nM
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| 3 |
Ki = 167 nM
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CP0389325
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2-[2-(5-methoxy-1H-indol-3-yl)ethyl]-1,3,4-oxadiazole
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C13H13N3O2
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2
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| 1 |
EC50 = 457 nM
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| 2 |
Ki = 68 nM
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CP0398563
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2-((S)-6-chloro-1'-((3S,4R)-4-(2,4-difluorophenyl)-1-(pentan-3-yl)pyrrolidine-3-carbonyl)-5-methyl-3H-spiro[isobenzofuran-1,4'-piperidine]-3-yl)-2-methylpropanenitrile
Show/Hide
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C33H40ClF2N3O2
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1
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| 1 |
EC50 = 465 nM
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CP0415040
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2-[2-(5-methoxy-1H-indol-3-yl)ethyl]-5-methyl-1,3-oxazole
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C15H16N2O2
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2
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| 1 |
EC50 = 503 nM
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| 2 |
Ki = 498 nM
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CP0398564
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2-((3S)-6-chloro-1'-((3S,4R)-4-(2,4-difluorophenyl)-1-(1-methoxypropan-2-yl)pyrrolidine-3-carbonyl)-5-methyl-3H-spiro[isobenzofuran-1,4'-piperidine]-3-yl)-2-methylpropanenitrile
Show/Hide
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C32H38ClF2N3O3
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1
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| 1 |
EC50 = 615 nM
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CP0493348
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2-((S)-6-chloro-1'-((3S,4R)-4-(2,4-difluorophenyl)-1-((tetrahydro-2H-pyran-4-yl)methyl)pyrrolidine-3-carbonyl)-5-methyl-3H-spiro[isobenzofuran-1,4'-piperidine]-3-yl)-2-methylpropanenitrile
Show/Hide
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C34H40ClF2N3O3
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1
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| 1 |
EC50 = 735 nM
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CP0072131
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2-[2-(5-methoxy-1H-indol-3-yl)ethyl]-5-methyl-1,3,4-oxadiazole
Show/Hide
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C14H15N3O2
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3
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| 1 |
EC50 = 881 nM
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| 2 |
EC50 = 1600 nM
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| 3 |
Ki = 190 nM
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CP0432491
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N-[(8-methoxy-2,3-dihydro-1H-cyclopenta[a]naphthalen-1-yl)methyl]ethanesulfonamide
Show/Hide
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C17H21NO3S
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2
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| 1 |
EC50 = 1000 nM
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| 2 |
Ki = 0.4 nM
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CP0398233
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5-[2-(5-methoxy-1H-indol-3-yl)ethyl]-3H-1,3,4-oxadiazole-2-thione
Show/Hide
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C13H13N3O2S
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2
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| 1 |
EC50 = 1096 nM
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| 2 |
Ki = 530 nM
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CP0283823
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2-((S)-6-chloro-1'-((3S,4R)-4-(2,4-difluorophenyl)-1-(tetrahydro-2H-pyran-4-yl)pyrrolidine-3-carbonyl)-5-methyl-3H-spiro[isobenzofuran-1,4'-piperidine]-3-yl)-2-methylpropanenitrile
Show/Hide
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C33H38ClF2N3O3
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1
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| 1 |
EC50 = 1697 nM
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CP0383642
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2-((S)-6-chloro-1'-((3S,4R)-4-(2,4-difluorophenyl)pyrrolidine-3-carbonyl)-5-methyl-3H-spiro[isobenzofuran-1,4'-piperidine]-3-yl)-2-methylpropanenitrile
Show/Hide
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C28H30ClF2N3O2
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1
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| 1 |
EC50 = 2100 nM
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CP0083725
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N-[2-(2-benzyl-5-methoxy-1-benzofuran-3-yl)ethyl]acetamide
Show/Hide
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C20H21NO3
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1
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| 1 |
EC50 > 10000 nM
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CP0095846
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N-[2-[5-methoxy-2-[(4-methoxyphenyl)methyl]-1-benzofuran-3-yl]ethyl]acetamide
Show/Hide
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C21H23NO4
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1
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| 1 |
EC50 > 10000 nM
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CP0100122
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N-[2-(2-benzyl-1-benzofuran-3-yl)ethyl]acetamide
Show/Hide
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C19H19NO2
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1
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| 1 |
EC50 > 10000 nM
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CP0452010
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N-[2-[5-fluoro-2-(4-fluorophenyl)sulfanyl-1-benzothiophen-3-yl]ethyl]propanamide
Show/Hide
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C19H17F2NOS2
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2
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| 1 |
EC50 > 10000 nM
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| 2 |
Ki = 4.4 nM
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CP0406181
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N-[2-(8-methoxybenzo[e][1]benzofuran-2-yl)ethyl]acetamide
Show/Hide
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C17H17NO3
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2
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| 1 |
EC50 > 10000 nM
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| 2 |
Ki = 1.7 nM
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CP0389225
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N-[(1-phenyl-3,4-dihydro-2H-quinolin-3-yl)methyl]acetamide
Show/Hide
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C18H20N2O
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1
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| 1 |
EC50 > 10000 nM
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CP0432630
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N-(1-benzyl-3,4-dihydro-2H-quinolin-3-yl)propanamide
Show/Hide
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C19H22N2O
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2
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| 1 |
EC50 > 10000 nM
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| 2 |
Ki = 6 nM
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CP0393387
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1-[(8-methoxy-2,3-dihydro-1H-cyclopenta[a]naphthalen-1-yl)methyl]-3-propylthiourea
Show/Hide
|
C19H24N2OS
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2
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| 1 |
EC50 > 10000 nM
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| 2 |
Ki = 3 nM
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CP0376623
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5-[(5-methoxy-1H-indol-3-yl)methyl]-3H-1,3,4-oxadiazole-2-thione
Show/Hide
|
C12H11N3O2S
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2
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| 1 |
EC50 > 1000 nM
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| 2 |
Ki = 535 nM
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CP0381569
|
5-[(5-methoxy-1H-indol-3-yl)methyl]-3H-1,3,4-oxadiazol-2-one
Show/Hide
|
C12H11N3O3
|
2
|
| 1 |
EC50 > 1000 nM
|
|
|
| 2 |
Ki = 160 nM
|
|
|
|
CP0381570
|
3-[(5-methoxy-1H-indol-3-yl)methyl]-4-methyl-1H-1,2,4-triazol-5-one
Show/Hide
|
C13H14N4O2
|
2
|
| 1 |
EC50 > 1000 nM
|
|
|
| 2 |
Ki = 560 nM
|
|
|
|
CP0398249
|
4-ethyl-3-[(5-methoxy-1H-indol-3-yl)methyl]-1H-1,2,4-triazole-5-thione
Show/Hide
|
C14H16N4OS
|
2
|
| 1 |
EC50 > 1000 nM
|
|
|
| 2 |
Ki = 220 nM
|
|
|
|
CP0521668
|
2,2,2-Trifluoro-N-[2-(7-isopropyl-1,6-dihydro-2H-indeno-[5,4-b]furan-8-yl)ethyl]acetamide
Show/Hide
|
C18H20F3NO2
|
1
|
| 1 |
Ki = 0.01 nM
|
|
|
|
CP0425880
|
N-[2-(7-propan-2-yl-2,6-dihydro-1H-cyclopenta[e][1]benzofuran-8-yl)ethyl]propanamide
Show/Hide
|
C19H25NO2
|
1
|
| 1 |
Ki = 0.011 nM
|
|
|
|
CP0425881
|
N-[2-[7-(3-propan-2-ylphenyl)-2,6-dihydro-1H-cyclopenta[e][1]benzofuran-8-yl]ethyl]acetamide
Show/Hide
|
C24H27NO2
|
1
|
| 1 |
Ki = 0.011 nM
|
|
|
|
CP0377935
|
N-[2-(7-bromo-2,6-dihydro-1H-cyclopenta[e][1]benzofuran-8-yl)ethyl]acetamide
Show/Hide
|
C15H16BrNO2
|
1
|
| 1 |
Ki = 0.014 nM
|
|
|
|
CP0499108
|
N-[2-(7-propan-2-yl-2,6-dihydro-1H-cyclopenta[e][1]benzofuran-8-yl)ethyl]acetamide
Show/Hide
|
C18H23NO2
|
1
|
| 1 |
Ki = 0.018 nM
|
|
|
|
CP0501489
|
N-[2-[7-(2-methoxyphenyl)-2,6-dihydro-1H-cyclopenta[e][1]benzofuran-8-yl]ethyl]acetamide
Show/Hide
|
C22H23NO3
|
1
|
| 1 |
Ki = 0.02 nM
|
|
|
|
CP0494363
|
N-[2-(2,6-dihydro-1H-cyclopenta[e][1]benzofuran-8-yl)ethyl]acetamide
Show/Hide
|
C15H17NO2
|
1
|
| 1 |
Ki = 0.022 nM
|
|
|
|
CP0532363
|
N-[3-[2-[(3,5-dimethoxyphenyl)methoxy]-5-methoxyphenyl]propyl]acetamide
Show/Hide
|
C21H27NO5
|
1
|
| 1 |
Ki = 0.0326 nM
|
|
|
|
CP0521667
|
N-[2-(7-pyridin-3-yl-2,6-dihydro-1H-cyclopenta[e][1]benzofuran-8-yl)ethyl]acetamide
Show/Hide
|
C20H20N2O2
|
1
|
| 1 |
Ki = 0.034 nM
|
|
|
|
CP0437994
|
N-[2-(7-propan-2-yl-2,6-dihydro-1H-cyclopenta[e][1]benzofuran-8-yl)ethyl]cyclopropanecarboxamide
Show/Hide
|
C20H25NO2
|
1
|
| 1 |
Ki = 0.035 nM
|
|
|
|
CP0377936
|
N-[2-[7-(4-methoxyphenyl)-2,6-dihydro-1H-cyclopenta[e][1]benzofuran-8-yl]ethyl]acetamide
Show/Hide
|
C22H23NO3
|
1
|
| 1 |
Ki = 0.037 nM
|
|
|
|
CP0504561
|
N-[3-(5-methoxy-2-phenylmethoxyphenyl)propyl]acetamide
Show/Hide
|
C19H23NO3
|
1
|
| 1 |
Ki = 0.04705 nM
|
|
|
|
CP0499107
|
1-ethyl-3-[2-(7-propan-2-yl-2,6-dihydro-1H-cyclopenta[e][1]benzofuran-8-yl)ethyl]urea
Show/Hide
|
C19H26N2O2
|
1
|
| 1 |
Ki = 0.084 nM
|
|
|
|
CP0458342
|
N-[2-(4-phenyl-10-oxa-5,6-diazatricyclo[7.3.0.02,6]dodeca-1(9),2,4,7-tetraen-3-yl)ethyl]acetamide
Show/Hide
|
C19H19N3O2
|
1
|
| 1 |
Ki = 0.085 nM
|
|
|
|
CP0485220
|
N-[3-(3-methoxyphenyl)-3-naphthalen-2-ylpropyl]acetamide
Show/Hide
|
C22H23NO2
|
1
|
| 1 |
Ki = 0.11 nM
|
|
|
|
CP0376971
|
N-[2-(4-cyclopropyl-10-oxa-5,6-diazatricyclo[7.3.0.02,6]dodeca-1(9),2,4,7-tetraen-3-yl)ethyl]propanamide
Show/Hide
|
C17H21N3O2
|
1
|
| 1 |
Ki = 0.14 nM
|
|
|
|
CP0055675
|
2-Iodomelatonin
Show/Hide
|
C13H15IN2O2
|
1
|
| 1 |
Ki = 0.15 nM
|
|
|
|
CP0186244
|
(4-Methoxy-6,7-dihydro-5H-dibenzo[a,c]cyclohepten-6-ylmethyl)-methoxymethyl-amine
Show/Hide
|
C20H23NO2
|
1
|
| 1 |
Ki = 0.16 nM
|
|
|
|
CP0501182
|
N-[2-(4-methyl-10-oxa-5,6-diazatricyclo[7.3.0.02,6]dodeca-1(9),2,4,7-tetraen-3-yl)ethyl]propanamide
Show/Hide
|
C15H19N3O2
|
1
|
| 1 |
Ki = 0.19 nM
|
|
|
|
CP0393386
|
1-[(2-methoxy-8,9-dihydro-7H-cyclopenta[h]quinolin-9-yl)methyl]-3-methylurea
Show/Hide
|
C16H19N3O2
|
1
|
| 1 |
Ki = 0.2 nM
|
|
|
|
CP0429924
|
N-[(2-methoxy-8,9-dihydro-7H-cyclopenta[h]quinolin-9-yl)methyl]acetamide
Show/Hide
|
C16H18N2O2
|
1
|
| 1 |
Ki = 0.2 nM
|
|
|
|
CP0508414
|
N-[(8-methoxy-1-methyl-2,3-dihydrocyclopenta[a]naphthalen-1-yl)methyl]methanesulfonamide
Show/Hide
|
C17H21NO3S
|
1
|
| 1 |
Ki = 0.2 nM
|
|
|
|
CP0441548
|
N-[2-(4-ethyl-10-oxa-5,6-diazatricyclo[7.3.0.02,6]dodeca-1(9),2,4,7-tetraen-3-yl)ethyl]propanamide
Show/Hide
|
C16H21N3O2
|
1
|
| 1 |
Ki = 0.22 nM
|
|
|
|
CP0389224
|
N-[[(1S,2R)-1-phenyl-1,2,3,4-tetrahydronaphthalen-2-yl]methyl]propanamide
Show/Hide
|
C20H23NO
|
1
|
| 1 |
Ki = 0.22 nM
|
|
|
|
CP0426376
|
N-[[(1R,2R)-1-phenyl-1,2,3,4-tetrahydronaphthalen-2-yl]methyl]propanamide
Show/Hide
|
C20H23NO
|
1
|
| 1 |
Ki = 0.23 nM
|
|
|
|
CP0455738
|
N-[2-(4-cyclopropyl-10-oxa-5,6-diazatricyclo[7.3.0.02,6]dodeca-1(9),2,4,7-tetraen-3-yl)ethyl]acetamide
Show/Hide
|
C16H19N3O2
|
1
|
| 1 |
Ki = 0.28 nM
|
|
|
|
CP0390104
|
N-[2-[4-(trifluoromethyl)-10-oxa-5,6-diazatricyclo[7.3.0.02,6]dodeca-1(9),2,4,7-tetraen-3-yl]ethyl]propanamide
Show/Hide
|
C15H16F3N3O2
|
1
|
| 1 |
Ki = 0.33 nM
|
|
|
|
CP0509534
|
N-[2-[7-(2-propan-2-yloxyphenyl)-2,6-dihydro-1H-cyclopenta[e][1]benzofuran-8-yl]ethyl]acetamide
Show/Hide
|
C24H27NO3
|
1
|
| 1 |
Ki = 0.34 nM
|
|
|
|
CP0040580
|
N-[2-(5-methoxy-1-benzofuran-3-yl)ethyl]acetamide
Show/Hide
|
C13H15NO3
|
1
|
| 1 |
Ki = 0.34 nM
|
|
|
|
CP0384067
|
N-[2-(2,7-dimethoxynaphthalen-1-yl)ethyl]propanamide
Show/Hide
|
C17H21NO3
|
1
|
| 1 |
Ki = 0.38 nM
|
|
|
|
CP0429922
|
1-[(2-methoxy-8,9-dihydro-7H-cyclopenta[h]quinolin-9-yl)methyl]-3-propylurea
Show/Hide
|
C18H23N3O2
|
1
|
| 1 |
Ki = 0.4 nM
|
|
|
|
CP0474642
|
N-[2-(6-methoxyquinolin-4-yl)ethyl]butanamide
Show/Hide
|
C16H20N2O2
|
1
|
| 1 |
Ki = 0.41 nM
|
|
|
|
CP0114370
|
4-P-PDOT
Show/Hide
|
C19H21NO
|
1
|
| 1 |
Ki = 0.46 nM
|
|
|
|
CP0475208
|
N-[[(3R,4S)-1-methyl-4-phenyl-3,4-dihydro-2H-quinolin-3-yl]methyl]propanamide
Show/Hide
|
C20H24N2O
|
1
|
| 1 |
Ki = 0.48 nM
|
|
|
|
CP0081204
|
N-[2-(11-methoxy-6,7-dihydro-5H-indolo[2,1-a][2]benzazepin-13-yl)ethyl]butanamide
Show/Hide
|
C24H28N2O2
|
1
|
| 1 |
Ki = 0.5 nM
|
|
|
|
CP0458343
|
N-[2-(4-methyl-10-oxa-5,6-diazatricyclo[7.3.0.02,6]dodeca-1(9),2,4,7-tetraen-3-yl)ethyl]acetamide
Show/Hide
|
C14H17N3O2
|
1
|
| 1 |
Ki = 0.53 nM
|
|
|
|
CP0456126
|
3-[4-(2-Acetylaminoethyl)-6-methoxynaphth-2-yl]benzoic acid methyl ester
Show/Hide
|
C23H23NO4
|
1
|
| 1 |
Ki = 0.64 nM
|
|
|
|
CP0443391
|
N-[2-[3-[3-(iodomethyl)phenyl]-7-methoxynaphthalen-1-yl]ethyl]acetamide
Show/Hide
|
C22H22INO2
|
1
|
| 1 |
Ki = 0.71 nM
|
|
|
|
CP0390102
|
N-[3-(3-methoxyphenyl)propyl]acetamide
Show/Hide
|
C12H17NO2
|
1
|
| 1 |
Ki = 0.751 nM
|
|
|
|
CP0501488
|
N-[2-[7-(4-tert-butylphenyl)-2,6-dihydro-1H-cyclopenta[e][1]benzofuran-8-yl]ethyl]acetamide
Show/Hide
|
C25H29NO2
|
1
|
| 1 |
Ki = 0.77 nM
|
|
|
|
CP0420022
|
1-[(8-methoxybenzo[e][1]benzofuran-2-yl)methyl]-3-methylthiourea
Show/Hide
|
C16H16N2O2S
|
1
|
| 1 |
Ki = 0.8 nM
|
|
|
|
CP0416462
|
N-[2-(2-methoxy-8,9-dihydro-7H-cyclopenta[h]quinolin-9-yl)ethyl]acetamide
Show/Hide
|
C17H20N2O2
|
1
|
| 1 |
Ki = 0.8 nM
|
|
|
|
CP0399886
|
N-[2-[(1R,3R)-7-methoxy-3-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]ethyl]cyclobutanecarboxamide
Show/Hide
|
C24H29NO2
|
1
|
| 1 |
Ki = 0.9 nM
|
|
|
|
CP0441549
|
N-[2-[4-(trifluoromethyl)-10-oxa-5,6-diazatricyclo[7.3.0.02,6]dodeca-1(9),2,4,7-tetraen-3-yl]ethyl]acetamide
Show/Hide
|
C14H14F3N3O2
|
1
|
| 1 |
Ki = 0.93 nM
|
|
|
|
CP0433988
|
N-[2-[7-methoxy-3-[3-(methoxymethyl)phenyl]naphthalen-1-yl]ethyl]acetamide
Show/Hide
|
C23H25NO3
|
1
|
| 1 |
Ki = 0.95 nM
|
|
|
|
CP0518308
|
N-[2-(6-methoxyquinolin-4-yl)ethyl]propanamide
Show/Hide
|
C15H18N2O2
|
1
|
| 1 |
Ki = 0.96 nM
|
|
|
|
CP0448964
|
N-[2-(2-hydroxy-7-methoxynaphthalen-1-yl)ethyl]propanamide
Show/Hide
|
C16H19NO3
|
1
|
| 1 |
Ki = 1.2 nM
|
|
|
|
CP0510962
|
N-[2-(2-ethoxy-7-methoxynaphthalen-1-yl)ethyl]propanamide
Show/Hide
|
C18H23NO3
|
1
|
| 1 |
Ki = 1.2 nM
|
|
|
|
CP0509510
|
N-[2-[2-(2-hydroxyethoxy)-7-methoxynaphthalen-1-yl]ethyl]propanamide
Show/Hide
|
C18H23NO4
|
1
|
| 1 |
Ki = 1.3 nM
|
|
|
|
CP0491332
|
N-[2-(6-methoxyquinolin-4-yl)ethyl]acetamide
Show/Hide
|
C14H16N2O2
|
1
|
| 1 |
Ki = 1.4 nM
|
|
|
|
CP0430666
|
N-[3-(2-ethoxy-5-methoxyphenyl)propyl]acetamide
Show/Hide
|
C14H21NO3
|
1
|
| 1 |
Ki = 1.59 nM
|
|
|
|
CP0430669
|
N-[3-[5-methoxy-2-(pyridin-2-ylmethoxy)phenyl]propyl]acetamide
Show/Hide
|
C18H22N2O3
|
1
|
| 1 |
Ki = 1.61 nM
|
|
|
|
CP0390834
|
methyl 2-[7-[4-[8-(2-acetamidoethyl)naphthalen-2-yl]oxybutoxy]naphthalen-1-yl]acetate
Show/Hide
|
C31H33NO5
|
1
|
| 1 |
Ki = 1.84 nM
|
|
|
|
CP0520030
|
N-[2-[3-[2-(hydroxymethyl)phenyl]-7-methoxynaphthalen-1-yl]ethyl]acetamide
Show/Hide
|
C22H23NO3
|
1
|
| 1 |
Ki = 1.86 nM
|
|
|
|
CP0432490
|
N-[2-(8-methoxy-2,3-dihydro-1H-cyclopenta[a]naphthalen-1-yl)ethyl]acetamide
Show/Hide
|
C18H21NO2
|
1
|
| 1 |
Ki = 2 nM
|
|
|
|
CP0470465
|
N-[3-(5-methoxy-2-propoxyphenyl)propyl]acetamide
Show/Hide
|
C15H23NO3
|
1
|
| 1 |
Ki = 2.12 nM
|
|
|
|
CP0849416
|
N-(2-(2-(isoindolin-2-ylmethyl)-5-methoxy-1H-indol-3-yl)ethyl)acetamide
Show/Hide
|
C22H25N3O2
|
1
|
| 1 |
Ki = 2.239 nM
|
|
|
|
CP0920948
|
N-[2-(5-Methoxy-2-{[(methyl(phenyl)amino]methyl}-1H-indol-3-yl)ethyl]acetamide
Show/Hide
|
C21H25N3O2
|
1
|
| 1 |
Ki = 2.291 nM
|
|
|
|
CP0375021
|
(E)-N-[3-(3-methoxyphenyl)-3-phenyl-2-propenyl]acetamide
Show/Hide
|
C18H19NO2
|
1
|
| 1 |
Ki = 2.5 nM
|
|
|
|
CP0388318
|
N-[2-[3-[3-(aminomethyl)phenyl]-7-methoxynaphthalen-1-yl]ethyl]acetamide
Show/Hide
|
C22H24N2O2
|
1
|
| 1 |
Ki = 3.4 nM
|
|
|
|
CP0866793
|
N-(2-(2-(isoindolin-2-ylmethyl)-5-methoxy-1H-indol-3-yl)ethyl)propionamide
Show/Hide
|
C23H27N3O2
|
1
|
| 1 |
Ki = 3.715 nM
|
|
|
|
CP0389223
|
N-[(1-phenyl-3,4-dihydronaphthalen-2-yl)methyl]propanamide
Show/Hide
|
C20H21NO
|
1
|
| 1 |
Ki = 3.8 nM
|
|
|
|
CP0458341
|
N-[2-(2-phenyl-7,8-dihydrofuro[2,3-g]benzimidazol-1-yl)ethyl]acetamide
Show/Hide
|
C19H19N3O2
|
1
|
| 1 |
Ki = 4.5 nM
|
|
|
|
CP0486794
|
5-[(E)-2-(7-methoxynaphthalen-1-yl)ethenyl]-3H-1,3,4-oxadiazol-2-one
Show/Hide
|
C15H12N2O3
|
1
|
| 1 |
Ki = 5.1 nM
|
|
|
|
CP0867260
|
N-(2-(2-((1H-indol-1-yl)methyl)-5-methoxy-1H-indol-3-yl)ethyl)acetamide
Show/Hide
|
C22H23N3O2
|
1
|
| 1 |
Ki = 5.754 nM
|
|
|
|
CP0376970
|
N-[2-(11-phenyl-5-oxa-1,10-diazatricyclo[7.3.0.02,6]dodeca-2(6),7,9,11-tetraen-12-yl)ethyl]acetamide
Show/Hide
|
C19H19N3O2
|
1
|
| 1 |
Ki = 6.1 nM
|
|
|
|
CP0467376
|
N-[2-(2-butoxy-7-methoxynaphthalen-1-yl)ethyl]propanamide
Show/Hide
|
C20H27NO3
|
1
|
| 1 |
Ki = 6.7 nM
|
|
|
|
CP0407039
|
N-[2-[7-[4-[8-(2-acetamidoethyl)naphthalen-2-yl]oxybutoxy]-1,2,3,4-tetrahydronaphthalen-1-yl]ethyl]acetamide
Show/Hide
|
C32H40N2O4
|
1
|
| 1 |
Ki = 6.79 nM
|
|
|
|
CP0372536
|
N-[2-(8-methoxy-2-methyl-3,4-dihydro-1H-pyrazino[1,2-a]indol-10-yl)ethyl]butanamide
Show/Hide
|
C19H27N3O2
|
1
|
| 1 |
Ki = 6.918 nM
|
|
|
|
CP0309824
|
1-ethyl-3-[(8-methoxybenzo[e][1]benzofuran-2-yl)methyl]thiourea
Show/Hide
|
C17H18N2O2S
|
1
|
| 1 |
Ki = 7 nM
|
|
|
|
CP0532362
|
N-[3-(3-methoxyphenyl)propyl]propanamide
Show/Hide
|
C13H19NO2
|
1
|
| 1 |
Ki = 7.07 nM
|
|
|
|
CP0423453
|
N-[2-[3-(3-acetamidophenyl)-7-methoxynaphthalen-1-yl]ethyl]acetamide
Show/Hide
|
C23H24N2O3
|
1
|
| 1 |
Ki = 7.54 nM
|
|
|
|
CP0874931
|
N-[2-(8-Methoxy-2-methyl-1,2,3,4-tetrahydropyrazino[1,2-a]indol-10-yl)ethyl]acetamide
Show/Hide
|
C17H23N3O2
|
1
|
| 1 |
Ki = 7.762 nM
|
|
|
|
CP0381636
|
2-((S)-2-Hydroxymethylindolin-1-ylmethyl)-melatonin
Show/Hide
|
C23H27N3O3
|
1
|
| 1 |
Ki = 7.8 nM
|
|
|
|
CP0474601
|
ethyl N-[3-[4-(2-acetamidoethyl)-6-methoxynaphthalen-2-yl]phenyl]carbamate
Show/Hide
|
C24H26N2O4
|
1
|
| 1 |
Ki = 8.3 nM
|
|
|
|
CP0373463
|
N-[2-[7-[4-[8-(2-acetamidoethyl)naphthalen-2-yl]oxybutoxy]naphthalen-1-yl]ethyl]but-3-enamide
Show/Hide
|
C34H38N2O4
|
1
|
| 1 |
Ki = 8.45 nM
|
|
|
|
CP0111066
|
N-[[1-[(4-chlorophenyl)methyl]-4-methoxyindol-2-yl]methyl]propanamide
Show/Hide
|
C20H21ClN2O2
|
1
|
| 1 |
Ki = 9 nM
|
|
|
|
CP0869995
|
N-(2-(2-(isoindolin-2-ylmethyl)-5-methoxy-1H-indol-3-yl)ethyl)but-3-enamide
Show/Hide
|
C24H27N3O2
|
1
|
| 1 |
Ki = 9.333 nM
|
|
|
|
CP0486386
|
N-[2-[2-[2-(dimethylamino)ethoxy]-7-methoxynaphthalen-1-yl]ethyl]propanamide
Show/Hide
|
C20H28N2O3
|
1
|
| 1 |
Ki = 10 nM
|
|
|
|
CP0524750
|
N-[2-[5-fluoro-2-(4-fluorophenyl)sulfanyl-1-benzothiophen-3-yl]ethyl]prop-2-enamide
Show/Hide
|
C19H15F2NOS2
|
1
|
| 1 |
Ki = 10.7 nM
|
|
|
|
CP0400713
|
N-[2-[7-[4-[8-(2-acetamidoethyl)naphthalen-2-yl]oxybutoxy]naphthalen-1-yl]ethyl]cyclopropanecarboxamide
Show/Hide
|
C34H38N2O4
|
1
|
| 1 |
Ki = 11.1 nM
|
|
|
|
CP0401701
|
N-[2-[7-[4-[8-(2-acetamidoethyl)naphthalen-2-yl]oxybutoxy]naphthalen-1-yl]ethyl]furan-2-carboxamide
Show/Hide
|
C35H36N2O5
|
1
|
| 1 |
Ki = 11.8 nM
|
|
|
|
CP0869937
|
5-[1-(5-Methoxy-1H-indol-3-yl)propan-2-yl]-1,3,4-oxadiazol-2(3H)-one
Show/Hide
|
C14H15N3O3
|
1
|
| 1 |
Ki = 12 nM
|
|
|
|
CP0447593
|
N-[3-(4-hydroxy-3-methoxyphenyl)propyl]acetamide
Show/Hide
|
C12H17NO3
|
1
|
| 1 |
Ki = 12.6 nM
|
|
|
|
CP0430667
|
N-[3-[5-methoxy-2-(2-phenylethoxy)phenyl]propyl]acetamide
Show/Hide
|
C20H25NO3
|
1
|
| 1 |
Ki = 13.4 nM
|
|
|
|
CP0400793
|
N-[2-[7-[4-[[3-(2-acetamidoethyl)-1-benzofuran-5-yl]oxy]butoxy]naphthalen-1-yl]ethyl]acetamide
Show/Hide
|
C30H34N2O5
|
1
|
| 1 |
Ki = 13.9 nM
|
|
|
|
CP0514684
|
N-[2-(6-methoxy-2-phenylquinazolin-4-yl)ethyl]acetamide
Show/Hide
|
C19H19N3O2
|
1
|
| 1 |
Ki = 15.6 nM
|
|
|
|
CP0383358
|
N-[2-(7-methoxy-2-propoxynaphthalen-1-yl)ethyl]propanamide
Show/Hide
|
C19H25NO3
|
1
|
| 1 |
Ki = 16 nM
|
|
|
|
CP0400795
|
methyl 4-[4-[4-[8-(2-acetamidoethyl)naphthalen-2-yl]oxybutoxy]phenyl]benzoate
Show/Hide
|
C32H33NO5
|
1
|
| 1 |
Ki = 19.1 nM
|
|
|
|
CP0947476
|
N-(2-(2-((3,4-dihydroisoquinolin-2(1H)-yl)methyl)-5-methoxy-1H-indol-3-yl)ethyl)acetamide
Show/Hide
|
C23H27N3O2
|
1
|
| 1 |
Ki = 21.38 nM
|
|
|
|
CP0548970
|
N-[2-(6-hexoxy-3,4-dihydro-2H-chromen-4-yl)ethyl]acetamide
Show/Hide
|
C19H29NO3
|
1
|
| 1 |
Ki = 21.4 nM
|
|
|
|
CP0047706
|
N-[3-[2-(4-phenylbutyl)-1,3-benzoxazol-7-yl]propyl]cyclopropanecarboxamide
Show/Hide
|
C24H28N2O2
|
1
|
| 1 |
Ki = 22 nM
|
|
|
|
CP0907712
|
{2-[7-Methoxy-1-(2-propionylamino-ethyl)-naphthalen-2-yloxy]-ethyl}-trimethyl-ammonium iodide
Show/Hide
|
C21H31IN2O3
|
1
|
| 1 |
Ki = 23 nM
|
|
|
|
CP0489804
|
N-[2-[3-[4-(hydroxymethyl)phenyl]-7-methoxynaphthalen-1-yl]ethyl]acetamide
Show/Hide
|
C22H23NO3
|
1
|
| 1 |
Ki = 23 nM
|
|
|
|
CP0452009
|
4-chloro-N-(2-(5-fluoro-2-(4-fluorophenylthio)benzo[b]thiophen-3-yl)ethyl)butanamide
Show/Hide
|
C20H18ClF2NOS2
|
1
|
| 1 |
Ki = 24.8 nM
|
|
|
|
CP0487668
|
N-[2-(2-cyclopropyl-6-methoxyquinazolin-4-yl)ethyl]acetamide
Show/Hide
|
C16H19N3O2
|
1
|
| 1 |
Ki = 25.9 nM
|
|
|
|
CP0400307
|
N-[3-(2,5-dimethoxyphenyl)propyl]acetamide
Show/Hide
|
C13H19NO3
|
1
|
| 1 |
Ki = 26.1 nM
|
|
|
|
CP0400306
|
N-[3-[5-methoxy-2-[(4-methoxyphenyl)methoxy]phenyl]propyl]acetamide
Show/Hide
|
C20H25NO4
|
1
|
| 1 |
Ki = 27.9 nM
|
|
|
|
CP0499033
|
(+/-)-2-(2-Hydroxymethyl-5-methoxyindolin-1-ylmethyl)-melatonin
Show/Hide
|
C24H29N3O4
|
1
|
| 1 |
Ki = 33.6 nM
|
|
|
|
CP0859463
|
N-(2-(2-(isoindolin-2-ylmethyl)-5-methoxy-1H-indol-3-yl)ethyl)cyclopropanecarboxamide
Show/Hide
|
C24H27N3O2
|
1
|
| 1 |
Ki = 33.88 nM
|
|
|
|
CP0514746
|
(+/-)-2-(2-Hydroxymethylindolin-1-ylmethyl)-melatonin
Show/Hide
|
C23H27N3O3
|
1
|
| 1 |
Ki = 36.2 nM
|
|
|
|
CP0513018
|
N-[2-(6-methoxyquinazolin-4-yl)ethyl]butanamide
Show/Hide
|
C15H19N3O2
|
1
|
| 1 |
Ki = 41 nM
|
|
|
|
CP0514689
|
N-[2-(6-methoxyquinazolin-4-yl)ethyl]propanamide
Show/Hide
|
C14H17N3O2
|
1
|
| 1 |
Ki = 41.1 nM
|
|
|
|
CP0914470
|
N-[2-(2-{[(4-Chlorophenyl)(methyl)amino]methyl}-5-methoxy-1H-indol-3-yl)ethyl]acetamide
Show/Hide
|
C21H24ClN3O2
|
1
|
| 1 |
Ki = 42.66 nM
|
|
|
|
CP0504015
|
3-(4-(2-Acetylaminoethyl)-6-methoxynaphth-2-yl)benzoic acid
Show/Hide
|
C22H21NO4
|
1
|
| 1 |
Ki = 43.3 nM
|
|
|
|
CP0400791
|
2-[7-[4-[8-(2-acetamidoethyl)naphthalen-2-yl]oxybutoxy]naphthalen-1-yl]acetic acid
Show/Hide
|
C30H31NO5
|
1
|
| 1 |
Ki = 45.8 nM
|
|
|
|
CP0105647
|
1-ethyl-3-[2-(8-methoxybenzo[e][1]benzofuran-2-yl)ethyl]urea
Show/Hide
|
C18H20N2O3
|
1
|
| 1 |
Ki = 46 nM
|
|
|
|
CP0514682
|
N-[2-[6-methoxy-2-(3-methoxyphenyl)quinazolin-4-yl]ethyl]acetamide
Show/Hide
|
C20H21N3O3
|
1
|
| 1 |
Ki = 46 nM
|
|
|
|
CP0447591
|
N-[3-(2-hydroxy-5-methoxyphenyl)propyl]acetamide
Show/Hide
|
C12H17NO3
|
1
|
| 1 |
Ki = 46.2 nM
|
|
|
|
CP0469724
|
N-[2-[3-[3-(hydroxymethyl)phenyl]-7-methoxynaphthalen-1-yl]ethyl]cyclobutanecarboxamide
Show/Hide
|
C25H27NO3
|
1
|
| 1 |
Ki = 48.3 nM
|
|
|
|
CP0415638
|
N-[2-[5-(3-phenylpropoxy)-1H-indol-3-yl]ethyl]acetamide
Show/Hide
|
C21H24N2O2
|
1
|
| 1 |
Ki = 49 nM
|
|
|
|
CP0402287
|
4-[4-[4-[8-(2-acetamidoethyl)naphthalen-2-yl]oxybutoxy]phenyl]benzoic acid
Show/Hide
|
C31H31NO5
|
1
|
| 1 |
Ki = 51.3 nM
|
|
|
|
CP0381637
|
N-[2-(7-methoxy-3,13-diazapentacyclo[11.7.0.03,11.04,9.014,19]icosa-4(9),5,7,10,14,16,18-heptaen-10-yl)ethyl]acetamide
Show/Hide
|
C23H25N3O2
|
2
|
| 1 |
Ki = 64.57 nM
|
|
|
| 2 |
Ki = 65.2 nM
|
|
|
|
CP0558022
|
5-[(E)-2-(6,7-dimethoxynaphthalen-1-yl)ethenyl]-3H-1,3,4-oxadiazol-2-one
Show/Hide
|
C16H14N2O4
|
1
|
| 1 |
Ki = 69 nM
|
|
|
|
CP0477491
|
N-[3-(3-methoxy-4-phenylmethoxyphenyl)propyl]acetamide
Show/Hide
|
C19H23NO3
|
1
|
| 1 |
Ki = 69.3 nM
|
|
|
|
CP0430668
|
N-[3-[5-methoxy-2-(3-phenylpropoxy)phenyl]propyl]acetamide
Show/Hide
|
C21H27NO3
|
1
|
| 1 |
Ki = 72.2 nM
|
|
|
|
CP0437583
|
N-[2-[2-(2-iodoethoxy)-7-methoxynaphthalen-1-yl]ethyl]propanamide
Show/Hide
|
C18H22INO3
|
1
|
| 1 |
Ki = 73 nM
|
|
|
|
CP0849192
|
N-(2-(2-((1H-indol-1-yl)methyl)-5-methoxy-1H-indol-3-yl)ethyl)cyclobutanecarboxamide
Show/Hide
|
C25H27N3O2
|
1
|
| 1 |
Ki = 81.28 nM
|
|
|
|
CP0373460
|
N-[2-[7-[4-[[3-(2-acetamidoethyl)-1H-indol-5-yl]oxy]butoxy]naphthalen-1-yl]ethyl]acetamide
Show/Hide
|
C30H35N3O4
|
1
|
| 1 |
Ki = 84.3 nM
|
|
|
|
CP0921467
|
N-[2-(2-Methyl-1,2,3,4-tetrahydropyrazino[1,2-a]indol-10-yl)ethyl]butanamide
Show/Hide
|
C18H25N3O
|
1
|
| 1 |
Ki = 85.11 nM
|
|
|
|
CP0385096
|
N-[2-[5-(3-phenoxypropoxy)-1H-indol-3-yl]ethyl]acetamide
Show/Hide
|
C21H24N2O3
|
1
|
| 1 |
Ki = 87 nM
|
|
|
|
CP0510641
|
N-[3-[2-[(4-bromo-2-fluorophenyl)methoxy]-5-methoxyphenyl]propyl]acetamide
Show/Hide
|
C19H21BrFNO3
|
1
|
| 1 |
Ki = 102 nM
|
|
|
|
CP0452111
|
N-[3-[3-methoxy-4-[(3-methoxyphenyl)methoxy]phenyl]propyl]acetamide
Show/Hide
|
C20H25NO4
|
1
|
| 1 |
Ki = 105 nM
|
|
|
|
CP0558328
|
N-[2-(7-methoxyphthalazin-1-yl)ethyl]butanamide
Show/Hide
|
C15H19N3O2
|
1
|
| 1 |
Ki = 108 nM
|
|
|
|
CP0473011
|
N-(1,2,3,4-tetrahydroquinolin-3-ylmethyl)acetamide
Show/Hide
|
C12H16N2O
|
1
|
| 1 |
Ki = 110 nM
|
|
|
|
CP0511802
|
5-[2-(5-methoxy-1H-indol-3-yl)ethyl]-N-methyl-1,3,4-oxadiazol-2-amine
Show/Hide
|
C14H16N4O2
|
1
|
| 1 |
Ki = 110 nM
|
|
|
|
CP0479258
|
N-[2-(6-methoxyquinazolin-4-yl)ethyl]acetamide
Show/Hide
|
C13H15N3O2
|
1
|
| 1 |
Ki = 115 nM
|
|
|
|
CP0470444
|
N-[3-(3-methoxy-4-phenylmethoxyphenyl)propyl]propanamide
Show/Hide
|
C20H25NO3
|
1
|
| 1 |
Ki = 121 nM
|
|
|
|
CP0193528
|
N-[2-[7-[3-[8-(2-acetamidoethyl)naphthalen-2-yl]oxypropoxy]naphthalen-1-yl]ethyl]acetamide
Show/Hide
|
C31H34N2O4
|
2
|
| 1 |
Ki = 149 nM
|
|
|
| 2 |
Ki = 354.81 nM
|
|
|
|
CP0452008
|
N-[2-[5-fluoro-2-(4-fluorophenyl)sulfanyl-1-benzothiophen-3-yl]ethyl]cyclobutanecarboxamide
Show/Hide
|
C21H19F2NOS2
|
1
|
| 1 |
Ki = 194 nM
|
|
|
|
CP0921994
|
N-(2-(2-(isoindolin-2-ylmethyl)-5-methoxy-1H-indol-3-yl)ethyl)cyclobutanecarboxamide
Show/Hide
|
C25H29N3O2
|
1
|
| 1 |
Ki = 199.53 nM
|
|
|
|
CP0844959
|
N-[2-(2-{[Ethyl(methyl)amino]methyl}-5-methoxy-1H-indol-3-yl)ethyl]acetamide
Show/Hide
|
C17H25N3O2
|
1
|
| 1 |
Ki = 223.87 nM
|
|
|
|
CP0258343
|
3-(cyclobutylmethyl)-5-[2-(5-methoxy-1H-indol-3-yl)ethyl]-1,3,4-oxadiazol-2-one
Show/Hide
|
C18H21N3O3
|
1
|
| 1 |
Ki = 230 nM
|
|
|
|
CP0375514
|
N-[2-[7-[8-(2-acetamidoethyl)naphthalen-2-yl]naphthalen-1-yl]ethyl]acetamide
Show/Hide
|
C28H28N2O2
|
1
|
| 1 |
Ki = 246 nM
|
|
|
|
CP0362932
|
5-[(E)-2-(7-methoxy-3,4-dihydronaphthalen-1-yl)ethenyl]-3H-1,3,4-oxadiazol-2-one
Show/Hide
|
C15H14N2O3
|
1
|
| 1 |
Ki = 260 nM
|
|
|
|
CP0511803
|
3-heptyl-5-[2-(5-methoxy-1H-indol-3-yl)ethyl]-1,3,4-oxadiazol-2-one
Show/Hide
|
C20H27N3O3
|
1
|
| 1 |
Ki = 300 nM
|
|
|
|
CP0422156
|
5-[2-(5-methoxy-1H-indol-3-yl)ethyl]-3-(3-phenylpropyl)-1,3,4-oxadiazol-2-one
Show/Hide
|
C22H23N3O3
|
1
|
| 1 |
Ki = 320 nM
|
|
|
|
CP0317553
|
3-(cyclopentylmethyl)-5-[2-(5-methoxy-1H-indol-3-yl)ethyl]-1,3,4-oxadiazol-2-one
Show/Hide
|
C19H23N3O3
|
1
|
| 1 |
Ki = 390 nM
|
|
|
|
CP0547557
|
N-[2-(6-methoxyquinazolin-4-yl)ethyl]cyclopropanecarboxamide
Show/Hide
|
C15H17N3O2
|
1
|
| 1 |
Ki = 398 nM
|
|
|
|
CP0094726
|
N-[2-(7,17-dimethoxy-3,13-diazapentacyclo[11.7.0.03,11.04,9.014,19]icosa-4(9),5,7,10,14(19),15,17-heptaen-10-yl)ethyl]acetamide
Show/Hide
|
C24H27N3O3
|
2
|
| 1 |
Ki = 407.38 nM
|
|
|
| 2 |
Ki = 410 nM
|
|
|
|
CP0514683
|
N-[2-(7-methoxyphthalazin-1-yl)ethyl]propanamide
Show/Hide
|
C14H17N3O2
|
1
|
| 1 |
Ki = 414 nM
|
|
|
|
CP0487632
|
3-hexyl-5-[2-(5-methoxy-1H-indol-3-yl)ethyl]-1,3,4-oxadiazol-2-one
Show/Hide
|
C19H25N3O3
|
1
|
| 1 |
Ki = 530 nM
|
|
|
|
CP0920290
|
N-[2-(2-{[(Benzyl(methyl)amino]methyl}-5-methoxy-1H-indol-3-yl)ethyl]acetamide
Show/Hide
|
C22H27N3O2
|
1
|
| 1 |
Ki = 660.69 nM
|
|
|
|
CP0552037
|
N-[2-(7-methoxyphthalazin-1-yl)ethyl]acetamide
Show/Hide
|
C13H15N3O2
|
1
|
| 1 |
Ki = 799 nM
|
|
|
|
CP0914471
|
N-[2-(9-Methoxy-2-methyl-2,3,4,5-tetrahydro-1H-[1,4]diazepino[1,2-a]indol-11-yl)ethyl]acetamide
Show/Hide
|
C18H25N3O2
|
1
|
| 1 |
Ki = 891.25 nM
|
|
|
|
CP0424907
|
N-[2-(7-methoxyphthalazin-1-yl)ethyl]cyclopropanecarboxamide
Show/Hide
|
C15H17N3O2
|
1
|
| 1 |
Ki = 1370 nM
|
|
|
|
CP0474655
|
N-[2-(3,13-diazapentacyclo[11.7.0.03,11.04,9.014,19]icosa-4,6,8,10,14,16,18-heptaen-10-yl)ethyl]acetamide
Show/Hide
|
C22H23N3O
|
1
|
| 1 |
Ki = 1700 nM
|
|
|
|
CP0498635
|
N-[3-(5-methoxy-2-phenylmethoxyphenyl)propyl]benzamide
Show/Hide
|
C24H25NO3
|
1
|
| 1 |
Ki = 2300 nM
|
|
|
|
CP0487667
|
N-ethyl-4-(6-methoxyquinazolin-4-yl)piperazine-1-carboxamide
Show/Hide
|
C16H21N5O2
|
1
|
| 1 |
Ki = 2800 nM
|
|
|
|
CP0547559
|
cyclopropyl-[4-(6-methoxyquinazolin-4-yl)piperazin-1-yl]methanone
Show/Hide
|
C17H20N4O2
|
1
|
| 1 |
Ki = 3295 nM
|
|
|
|
CP0036921
|
3-HYDROXYTYRAMINE HYDROCHLORIDE
Show/Hide
|
C8H11NO2
|
1
|
| 1 |
Ki = 9100 nM
|
|
|
|
CP0549637
|
5-[2-(5-methoxy-1H-indol-3-yl)ethyl]-3-propyl-1,3,4-oxadiazol-2-one
Show/Hide
|
C16H19N3O3
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0001238
|
14C-5-hydroxy tryptamine creatinine disulfate
Show/Hide
|
C10H12N2O
|
1
|
| 1 |
Ki > 100000 nM
|
|
|
|
CP0547558
|
N-[2-[(6-methoxyquinazolin-4-yl)amino]ethyl]acetamide
Show/Hide
|
C13H16N4O2
|
1
|
| 1 |
Ki > 100000 nM
|
|
|
|
CP0258344
|
5-[(E)-2-(5-methoxy-1H-indol-3-yl)ethenyl]-3H-1,3,4-oxadiazol-2-one
Show/Hide
|
C13H11N3O3
|
1
|
| 1 |
Ki > 100 nM
|
|
|
|
CP0478995
|
(E)-3-(5-methoxy-1H-indol-3-yl)-N-prop-2-ynylprop-2-enamide
Show/Hide
|
C15H14N2O2
|
1
|
| 1 |
Ki > 100 nM
|
|
|
|
CP0487486
|
5-[(E)-2-(5-methoxy-1H-indol-3-yl)ethenyl]-3-prop-2-ynyl-1,3,4-oxadiazol-2-one
Show/Hide
|
C16H13N3O3
|
1
|
| 1 |
Ki > 100 nM
|
|
|
|
CP0549638
|
(E)-3-(5-methoxy-1H-indol-3-yl)-N-prop-2-enylprop-2-enamide
Show/Hide
|
C15H16N2O2
|
1
|
| 1 |
Ki > 100 nM
|
|
|
|
CP0897694
|
6-Methoxy-1-methyl-4-(2-propionylamino-ethyl)-quinolinium iodide
Show/Hide
|
C16H21IN2O2
|
1
|
| 1 |
Ki > 1000 nM
|
|
|
|
CP0919223
|
4-(2-Acetylamino-ethyl)-6-methoxy-1-methyl-quinolinium iodide
Show/Hide
|
C15H19IN2O2
|
1
|
| 1 |
Ki > 1000 nM
|
|
|
|
CP0376624
|
2-[(5-methoxy-1H-indol-3-yl)methyl]-5-methyl-1,3-oxazole
Show/Hide
|
C14H14N2O2
|
1
|
| 1 |
Ki > 1000 nM
|
|
|
|
CP0433770
|
3-[2-(5-methoxy-1H-indol-3-yl)ethyl]-4-methyl-1H-1,2,4-triazol-5-one
Show/Hide
|
C14H16N4O2
|
1
|
| 1 |
Ki > 1000 nM
|
|
|
|
CP0449128
|
4-ethyl-3-[2-(5-methoxy-1H-indol-3-yl)ethyl]-1H-1,2,4-triazole-5-thione
Show/Hide
|
C15H18N4OS
|
1
|
| 1 |
Ki > 1000 nM
|
|
|
|
CP0482626
|
5-[2-(5-methoxy-1H-indol-3-yl)ethyl]-3-methyl-1,2,4-oxadiazole
Show/Hide
|
C14H15N3O2
|
1
|
| 1 |
Ki > 1000 nM
|
|
|
