All Bioactivity

Brief Information of the Cell Line and Protein

Cell Line ID: CL000011 , CHO

Cell Line Info

Synonyms	Chinese Hamster Ovary CHO-ori
Category	Spontaneously immortalized cell line
Organism	Cricetulus griseus (Chinese hamster)
Cellosaurus ID	CVCL_0213

Protein ID: PT01693 , Somatostatin receptor type 3

Protein Info

Gene Name	SSTR3
Organism	Homo sapiens, Human
Protein Classification	Membrane receptor
Uniprot ID	P32745

Table of Molecular Bioactivities Related to the Cell Line and Protein

Cell Line ID: CL000011

Cell Line Info

Protein ID: PT01693

Protein Info

Compound ID	Compound Name	Compound Formula
CP0550776 Compound Info	1-[5-(4-methylphenyl)-1H-imidazol-2-yl]-N-(3-phenylpropyl)cyclopentan-1-amine Show/Hide	C24H29N3	2
1	EC50 = 5.2 nM Bioactivity Info	TI LI LO TS
2	Ki = 1.3 nM Bioactivity Info	TI LI LO TS
CP0386791 Compound Info	1-[5-(4-fluorophenyl)-1H-imidazol-2-yl]-N-(1H-indol-3-ylmethyl)cyclopentan-1-amine Show/Hide	C23H23FN4	2
1	EC50 = 8.1 nM Bioactivity Info	TI LI LO TS
2	Ki = 2 nM Bioactivity Info	TI LI LO TS
CP0392302 Compound Info	N-(1H-indol-3-ylmethyl)-1-[5-(4-methylphenyl)-1H-imidazol-2-yl]cyclopentan-1-amine Show/Hide	C24H26N4	2
1	EC50 = 11 nM Bioactivity Info	TI LI LO TS
2	Ki = 3.4 nM Bioactivity Info	TI LI LO TS
CP0388968 Compound Info	N-(1H-indol-2-ylmethyl)-1-[5-(4-methylphenyl)-1H-imidazol-2-yl]cyclopentan-1-amine Show/Hide	C24H26N4	2
1	EC50 = 15 nM Bioactivity Info	TI LI LO TS
2	Ki = 4.9 nM Bioactivity Info	TI LI LO TS
CP0392303 Compound Info	N-(1H-indol-3-ylmethyl)-1-(5-phenyl-1H-imidazol-2-yl)cyclopentan-1-amine Show/Hide	C23H24N4	2
1	EC50 = 20 nM Bioactivity Info	TI LI LO TS
2	Ki = 5.4 nM Bioactivity Info	TI LI LO TS
CP0443567 Compound Info	1-[5-(4-methylphenyl)-1H-imidazol-2-yl]-N-(1H-pyrrolo[3,2-b]pyridin-3-ylmethyl)cyclopentan-1-amine Show/Hide	C23H25N5	2
1	EC50 = 20 nM Bioactivity Info	TI LI LO TS
2	Ki = 24 nM Bioactivity Info	TI LI LO TS
CP0427963 Compound Info	N-[(4-fluorophenyl)methyl]-1-[5-(4-methylphenyl)-1H-imidazol-2-yl]cyclopentan-1-amine Show/Hide	C22H24FN3	2
1	EC50 = 26 nM Bioactivity Info	TI LI LO TS
2	Ki = 23 nM Bioactivity Info	TI LI LO TS
CP0402092 Compound Info	N-(cyclohexylmethyl)-1-[5-(4-methylphenyl)-1H-imidazol-2-yl]cyclopentan-1-amine Show/Hide	C22H31N3	2
1	EC50 = 34 nM Bioactivity Info	TI LI LO TS
2	Ki = 27 nM Bioactivity Info	TI LI LO TS
CP0388969 Compound Info	N-(3,3-dimethylbutyl)-1-[5-(4-methylphenyl)-1H-imidazol-2-yl]cyclopentan-1-amine Show/Hide	C21H31N3	2
1	EC50 = 35 nM Bioactivity Info	TI LI LO TS
2	Ki = 35 nM Bioactivity Info	TI LI LO TS
CP0443721 Compound Info	N-[(7-methoxy-1H-indol-3-yl)methyl]-1-[5-(4-methylphenyl)-1H-imidazol-2-yl]cyclopentan-1-amine Show/Hide	C25H28N4O	2
1	EC50 = 38 nM Bioactivity Info	TI LI LO TS
2	Ki = 24 nM Bioactivity Info	TI LI LO TS
CP0386764 Compound Info	N-(1H-indol-3-ylmethyl)-1-[5-(4-methylphenyl)-1H-imidazol-2-yl]cyclohexan-1-amine Show/Hide	C25H28N4	2
1	EC50 = 43 nM Bioactivity Info	TI LI LO TS
2	Ki = 5.3 nM Bioactivity Info	TI LI LO TS
CP0521107 Compound Info	N-[(1-methylindol-3-yl)methyl]-1-[5-(4-methylphenyl)-1H-imidazol-2-yl]cyclopentan-1-amine Show/Hide	C25H28N4	2
1	EC50 = 54 nM Bioactivity Info	TI LI LO TS
2	Ki = 26 nM Bioactivity Info	TI LI LO TS
CP0420331 Compound Info	N-benzyl-1-[5-(4-methylphenyl)-1H-imidazol-2-yl]cyclopentan-1-amine Show/Hide	C22H25N3	2
1	EC50 = 61 nM Bioactivity Info	TI LI LO TS
2	Ki = 90 nM Bioactivity Info	TI LI LO TS
CP0388972 Compound Info	N-[(3-fluorophenyl)methyl]-1-[5-(4-methylphenyl)-1H-imidazol-2-yl]cyclopentan-1-amine Show/Hide	C22H24FN3	2
1	EC50 = 93 nM Bioactivity Info	TI LI LO TS
2	Ki = 72 nM Bioactivity Info	TI LI LO TS
CP0420324 Compound Info	N-[(4-methoxyphenyl)methyl]-1-[5-(4-methylphenyl)-1H-imidazol-2-yl]cyclopentan-1-amine Show/Hide	C23H27N3O	2
1	EC50 = 96 nM Bioactivity Info	TI LI LO TS
2	Ki = 32 nM Bioactivity Info	TI LI LO TS
CP0431798 Compound Info	1-[5-(4-methylphenyl)-1H-imidazol-2-yl]-N-(2-phenylethyl)cyclopentan-1-amine Show/Hide	C23H27N3	2
1	EC50 = 103 nM Bioactivity Info	TI LI LO TS
2	Ki = 37 nM Bioactivity Info	TI LI LO TS
CP0472431 Compound Info	N-[2-(1H-indol-3-yl)ethyl]-1-[5-(4-methylphenyl)-1H-imidazol-2-yl]cyclopentan-1-amine Show/Hide	C25H28N4	2
1	EC50 = 110 nM Bioactivity Info	TI LI LO TS
2	Ki = 73 nM Bioactivity Info	TI LI LO TS
CP0420329 Compound Info	N-(1H-indol-3-ylmethyl)-1-[5-(4-methylphenyl)-1H-imidazol-2-yl]cyclobutan-1-amine Show/Hide	C23H24N4	2
1	EC50 = 160 nM Bioactivity Info	TI LI LO TS
2	Ki = 51 nM Bioactivity Info	TI LI LO TS
CP0386793 Compound Info	N-[(4-chlorophenyl)methyl]-1-[5-(4-methylphenyl)-1H-imidazol-2-yl]cyclopentan-1-amine Show/Hide	C22H24ClN3	2
1	EC50 = 170 nM Bioactivity Info	TI LI LO TS
2	Ki = 32 nM Bioactivity Info	TI LI LO TS
CP0392304 Compound Info	N-(1H-indol-3-ylmethyl)-1-[5-(4-phenylphenyl)-1H-imidazol-2-yl]cyclopentan-1-amine Show/Hide	C29H28N4	2
1	EC50 = 280 nM Bioactivity Info	TI LI LO TS
2	Ki = 31 nM Bioactivity Info	TI LI LO TS
CP0392306 Compound Info	1-[5-(4-methylphenyl)-1H-imidazol-2-yl]-N-[[4-(trifluoromethyl)phenyl]methyl]cyclopentan-1-amine Show/Hide	C23H24F3N3	2
1	EC50 = 370 nM Bioactivity Info	TI LI LO TS
2	Ki = 330 nM Bioactivity Info	TI LI LO TS
CP0392301 Compound Info	N-(1H-indol-3-ylmethyl)-2-[5-(4-methylphenyl)-1H-imidazol-2-yl]propan-2-amine Show/Hide	C22H24N4	2
1	EC50 = 390 nM Bioactivity Info	TI LI LO TS
2	Ki = 180 nM Bioactivity Info	TI LI LO TS
CP0472433 Compound Info	1-[5-(4-methylphenyl)-1H-imidazol-2-yl]-N-propylcyclopentan-1-amine Show/Hide	C18H25N3	2
1	EC50 = 770 nM Bioactivity Info	TI LI LO TS
2	Ki = 510 nM Bioactivity Info	TI LI LO TS
CP0386794 Compound Info	methyl 4-[[[1-[5-(4-methylphenyl)-1H-imidazol-2-yl]cyclopentyl]amino]methyl]benzoate Show/Hide	C24H27N3O2	2
1	EC50 = 970 nM Bioactivity Info	TI LI LO TS
2	Ki = 830 nM Bioactivity Info	TI LI LO TS
CP0392362 Compound Info	1-[5-(4-methylphenyl)-1H-imidazol-2-yl]-N-(oxan-4-ylmethyl)cyclopentan-1-amine Show/Hide	C21H29N3O	2
1	EC50 = 1200 nM Bioactivity Info	TI LI LO TS
2	Ki = 1200 nM Bioactivity Info	TI LI LO TS
CP0388971 Compound Info	1-[5-(4-methylphenyl)-1H-imidazol-2-yl]-N-(quinolin-6-ylmethyl)cyclopentan-1-amine Show/Hide	C25H26N4	2
1	EC50 = 1400 nM Bioactivity Info	TI LI LO TS
2	Ki = 1400 nM Bioactivity Info	TI LI LO TS
CP0392305 Compound Info	1-[5-(4-methylphenyl)-1H-imidazol-2-yl]-N-(3,3,3-trifluoropropyl)cyclopentan-1-amine Show/Hide	C18H22F3N3	2
1	EC50 = 1600 nM Bioactivity Info	TI LI LO TS
2	Ki = 2600 nM Bioactivity Info	TI LI LO TS
CP0388970 Compound Info	1-[5-(4-methylphenyl)-1H-imidazol-2-yl]-N-[(4-phenylphenyl)methyl]cyclopentan-1-amine Show/Hide	C28H29N3	2
1	EC50 = 2300 nM Bioactivity Info	TI LI LO TS
2	Ki = 160 nM Bioactivity Info	TI LI LO TS
CP0433177 Compound Info	N-(1H-indol-3-ylmethyl)-4-[5-(4-methylphenyl)-1H-imidazol-2-yl]piperidin-4-amine Show/Hide	C24H27N5	2
1	EC50 = 2500 nM Bioactivity Info	TI LI LO TS
2	Ki = 60 nM Bioactivity Info	TI LI LO TS
CP0392307 Compound Info	1-[5-(4-methylphenyl)-1H-imidazol-2-yl]-N-[(1-methylpyrazol-4-yl)methyl]cyclopentan-1-amine Show/Hide	C20H25N5	2
1	EC50 = 3700 nM Bioactivity Info	TI LI LO TS
2	Ki = 3400 nM Bioactivity Info	TI LI LO TS
CP0392300 Compound Info	N-[(3-ethylimidazol-4-yl)methyl]-1-[5-(4-methylphenyl)-1H-imidazol-2-yl]cyclopentan-1-amine Show/Hide	C21H27N5	2
1	EC50 = 4200 nM Bioactivity Info	TI LI LO TS
2	Ki = 8600 nM Bioactivity Info	TI LI LO TS
CP0427964 Compound Info	1-[5-(4-methylphenyl)-1H-imidazol-2-yl]-N-(pyridin-4-ylmethyl)cyclopentan-1-amine Show/Hide	C21H24N4	2
1	EC50 = 4200 nM Bioactivity Info	TI LI LO TS
2	Ki = 5600 nM Bioactivity Info	TI LI LO TS
CP0392298 Compound Info	1-[5-(4-methylphenyl)-1H-imidazol-2-yl]-N-(pyrimidin-5-ylmethyl)cyclopentan-1-amine Show/Hide	C20H23N5	1
1	EC50 = 4800 nM Bioactivity Info	TI LI LO TS
CP0844603 Compound Info	Ethyl5-((1R,3R)-3-(4-(4-fluorophenyl)-1H-imidazol-2-yl)-1-(1-methyl-1H-pyrazol-4-yl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indol-1-yl)nicotinate Show/Hide	C32H28FN7O2	2
1	IC50 = 0.15 nM Bioactivity Info	TI LI LO TS
2	IC50 = 0.78 nM Bioactivity Info	TI LI LO TS
CP0843104 Compound Info	2-(5-((1R,3R)-1-(1-ethyl-1H-pyrazol-4-yl)-3-(4-(5-fluoropyridin-2-yl)-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indol-1-yl)-2-oxo-1,3,4-oxadiazol-3(2H)-yl)acetamide Show/Hide	C28H25FN10O3	2
1	IC50 = 0.3 nM Bioactivity Info	TI LI LO TS
2	IC50 = 2.4 nM Bioactivity Info	TI LI LO TS
CP0783440 Compound Info	3-ethyl-5-((1R,3R)-1-(1-ethyl-1H-pyrazol-4-yl)-3-(4-(5-fluoropyridin-2-yl)-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indol-1-yl)-1,3,4-oxadiazol-2(3H)-one Show/Hide	C28H26FN9O2	2
1	IC50 = 0.4 nM Bioactivity Info	TI LI LO TS
2	IC50 = 3 nM Bioactivity Info	TI LI LO TS
CP0843102 Compound Info	3-((1R,3R)-1-(1-(cyclopropylmethyl)-1H-pyrazol-4-yl)-3-(4-(5-fluoropyridin-2-yl)-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indol-1-yl)-5-methyl-1,2,4-oxadiazole Show/Hide	C29H26FN9O	2
1	IC50 = 0.4 nM Bioactivity Info	TI LI LO TS
2	IC50 = 1.1 nM Bioactivity Info	TI LI LO TS
CP0776356 Compound Info	3-(2-(dimethylamino)ethyl)-5-((1R,3R)-1-(1-ethyl-1H-pyrazol-4-yl)-3-(4-(5-fluoropyridin-2-yl)-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indol-1-yl)-1,3,4-oxadiazol-2(3H)-one Show/Hide	C30H31FN10O2	2
1	IC50 = 0.5 nM Bioactivity Info	TI LI LO TS
2	IC50 = 2.1 nM Bioactivity Info	TI LI LO TS
CP0756633 Compound Info	5-((1R,3R)-3-(4-(4-fluorophenyl)-1H-imidazol-2-yl)-1-(1-methyl-1H-pyrazol-4-yl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indol-1-yl)nicotinicacid Show/Hide	C30H24FN7O2	2
1	IC50 = 0.52 nM Bioactivity Info	TI LI LO TS
2	IC50 = 1.22 nM Bioactivity Info	TI LI LO TS
CP0673513 Compound Info	Ethyl 2-((1S,3R)-3-(4-(4-fluorophenyl)-1H-imidazol-2-yl)-1-(1-methyl-1H-pyrazol-4-yl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indol-1-yl)isonicotinate Show/Hide	C32H28FN7O2	2
1	IC50 = 0.64 nM Bioactivity Info	TI LI LO TS
2	IC50 = 0.78 nM Bioactivity Info	TI LI LO TS
CP0072718 Compound Info	3-[(1R,3R)-3-[5-(4-fluorophenyl)-1H-imidazol-2-yl]-1-(1-methylpyrazol-4-yl)-2,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-5-methyl-1,2,4-oxadiazole Show/Hide	C27H23FN8O	4
1	IC50 = 0.66 nM Bioactivity Info	TI LI LO TS
2	IC50 = 0.7 nM Bioactivity Info	TI LI LO TS
3	IC50 = 0.9 nM Bioactivity Info	TI LI LO TS
4	IC50 = 0.95 nM Bioactivity Info	TI LI LO TS
CP0414056 Compound Info	(3R)-3-[5-(4-fluorophenyl)-1H-imidazol-2-yl]-1,1-bis(1-methylpyrazol-4-yl)-2,3,4,9-tetrahydropyrido[3,4-b]indole Show/Hide	C28H25FN8	2
1	IC50 = 0.7 nM Bioactivity Info	TI LI LO TS
2	IC50 = 0.74 nM Bioactivity Info	TI LI LO TS
CP0843103 Compound Info	2-((1R,3R)-1-(1-ethyl-1H-pyrazol-4-yl)-3-(4-(5-fluoropyridin-2-yl)-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indol-1-yl)-5-(methylthio)-1,3,4-oxadiazole Show/Hide	C27H24FN9OS	2
1	IC50 = 0.7 nM Bioactivity Info	TI LI LO TS
2	IC50 = 1.9 nM Bioactivity Info	TI LI LO TS
CP0305127 Compound Info	(3R)-3-[5-(4-fluorophenyl)-1H-imidazol-2-yl]-1,1-diphenyl-2,3,4,9-tetrahydropyrido[3,4-b]indole Show/Hide	C32H25FN4	2
1	IC50 = 0.76 nM Bioactivity Info	TI LI LO TS
2	IC50 = 7.3 nM Bioactivity Info	TI LI LO TS
CP0368917 Compound Info	3-[(1R,3S)-3-[5-(4-fluorophenyl)-1H-imidazol-2-yl]-1-(1-methylpyrazol-4-yl)-2,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-5-methyl-1,2,4-oxadiazole Show/Hide	C27H23FN8O	2
1	IC50 = 0.78 nM Bioactivity Info	TI LI LO TS
2	IC50 = 0.94 nM Bioactivity Info	TI LI LO TS
CP0045013 Compound Info	(3R)-1-cyclohexyl-3-(5-phenyl-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole Show/Hide	C26H28N4	3
1	IC50 = 0.8 nM Bioactivity Info	TI LI LO TS
2	IC50 = 26 nM Bioactivity Info	TI LI LO TS
3	IC50 = 26.1 nM Bioactivity Info	TI LI LO TS
CP0153442 Compound Info	5-[(1R,3R)-3-[5-(5-fluoropyridin-2-yl)-1H-imidazol-2-yl]-1-(1-methylpyrazol-4-yl)-2,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3-propan-2-yl-1,3,4-oxadiazol-2-one Show/Hide	C28H26FN9O2	2
1	IC50 = 0.8 nM Bioactivity Info	TI LI LO TS
2	IC50 = 2 nM Bioactivity Info	TI LI LO TS
CP0664424 Compound Info	2-(5-((1R,3R)-1-(1-ethyl-1H-pyrazol-4-yl)-3-(4-(5-fluoropyridin-2-yl)-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indol-1-yl)-2-oxo-1,3,4-oxadiazol-3(2H)-yl)acetic acid Show/Hide	C28H24FN9O4	2
1	IC50 = 0.8 nM Bioactivity Info	TI LI LO TS
2	IC50 = 4.9 nM Bioactivity Info	TI LI LO TS
CP0857552 Compound Info	Ethyl6-((1S,3R)-3-(4-(4-fluorophenyl)-1H-imidazol-2-yl)-1-(1-methyl-1H-pyrazol-4-yl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indol-1-yl)picolinate Show/Hide	C32H28FN7O2	2
1	IC50 = 0.83 nM Bioactivity Info	TI LI LO TS
2	IC50 = 1.97 nM Bioactivity Info	TI LI LO TS
CP0330210 Compound Info	3-[(3R)-3-[5-(4-fluorophenyl)-1H-imidazol-2-yl]-1-(5-methyl-1,2,4-oxadiazol-3-yl)-2,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-5-methyl-1,2,4-oxadiazole Show/Hide	C26H21FN8O2	2
1	IC50 = 0.97 nM Bioactivity Info	TI LI LO TS
2	IC50 = 1.2 nM Bioactivity Info	TI LI LO TS
CP0683295 Compound Info	5-((1R,3R)-1-(1-ethyl-1H-pyrazol-4-yl)-3-(4-(5-fluoropyridin-2-yl)-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indol-1-yl)-3-isopropyl-1,3,4-oxadiazol-2(3H)-one Show/Hide	C29H28FN9O2	2
1	IC50 = 1 nM Bioactivity Info	TI LI LO TS
2	IC50 = 2.1 nM Bioactivity Info	TI LI LO TS
CP0120411 Compound Info	3-[(1S,3R)-3-[5-(4-fluorophenyl)-1H-imidazol-2-yl]-1-(1-methylpyrazol-4-yl)-2,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-5-methyl-1,2,4-oxadiazole Show/Hide	C27H23FN8O	1
1	IC50 = 1.1 nM Bioactivity Info	TI LI LO TS
CP0651917 Compound Info	5-((1R,3R)-1-(1-ethyl-1H-pyrazol-4-yl)-3-(4-(5-fluoropyridin-2-yl)-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indol-1-yl)-3-methyl-1,3,4-oxadiazol-2(3H)-one Show/Hide	C27H24FN9O2	2
1	IC50 = 1.1 nM Bioactivity Info	TI LI LO TS
2	IC50 = 2.3 nM Bioactivity Info	TI LI LO TS
CP0761913 Compound Info	5-ethyl-3-((1R,3R)-3-(4-(5-fluoropyridin-2-yl)-1H-imidazol-2-yl)-1-(1-methyl-1H-pyrazol-4-yl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indol-1-yl)-1,2,4-oxadiazole Show/Hide	C27H24FN9O	2
1	IC50 = 1.2 nM Bioactivity Info	TI LI LO TS
2	IC50 = 2.9 nM Bioactivity Info	TI LI LO TS
CP0862026 Compound Info	3-((1R,3R)-1-(1-ethyl-1H-pyrazol-4-yl)-3-(4-(5-fluoropyridin-2-yl)-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indol-1-yl)-5-methyl-1,2,4-oxadiazole Show/Hide	C27H24FN9O	2
1	IC50 = 1.2 nM Bioactivity Info	TI LI LO TS
2	IC50 = 2.2 nM Bioactivity Info	TI LI LO TS
CP0698603 Compound Info	3-(cyclopropylmethyl)-5-((1R,3R)-1-(1-ethyl-1H-pyrazol-4-yl)-3-(4-(5-fluoropyridin-2-yl)-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indol-1-yl)-1,3,4-oxadiazol-2(3H)-one Show/Hide	C30H28FN9O2	2
1	IC50 = 1.3 nM Bioactivity Info	TI LI LO TS
2	IC50 = 1.4 nM Bioactivity Info	TI LI LO TS
CP0673514 Compound Info	Ethyl6-((1R,3R)-3-(4-(4-fluorophenyl)-1H-imidazol-2-yl)-1-(1-methyl-1H-pyrazol-4-yl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indol-1-yl)picolinate Show/Hide	C32H28FN7O2	2
1	IC50 = 1.52 nM Bioactivity Info	TI LI LO TS
2	IC50 = 5.36 nM Bioactivity Info	TI LI LO TS
CP0787642 Compound Info	3-ethyl-5-((1R,3R)-3-(4-(5-fluoropyridin-2-yl)-1H-imidazol-2-yl)-1-(1-methyl-1H-pyrazol-4-yl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indol-1-yl)-1,3,4-oxadiazol-2(3H)-one Show/Hide	C27H24FN9O2	2
1	IC50 = 1.6 nM Bioactivity Info	TI LI LO TS
2	IC50 = 2.9 nM Bioactivity Info	TI LI LO TS
CP0383431 Compound Info	(3R)-3-(5-phenyl-1H-imidazol-2-yl)-1-(thian-4-yl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole Show/Hide	C25H26N4S	2
1	IC50 = 1.7 nM Bioactivity Info	TI LI LO TS
2	IC50 = 10 nM Bioactivity Info	TI LI LO TS
CP0237736 Compound Info	2-[(1R,3R)-3-[5-(4-fluorophenyl)-1H-imidazol-2-yl]-1-(1-methylpyrazol-4-yl)-2,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]pyridine-4-carboxylic acid Show/Hide	C30H24FN7O2	2
1	IC50 = 1.71 nM Bioactivity Info	TI LI LO TS
2	IC50 = 2.13 nM Bioactivity Info	TI LI LO TS
CP0381489 Compound Info	ethyl 6-[(1R,3R)-3-[5-(4-fluorophenyl)-1H-imidazol-2-yl]-1-(1-methylpyrazol-4-yl)-2,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]pyridine-3-carboxylate Show/Hide	C32H28FN7O2	2
1	IC50 = 1.72 nM Bioactivity Info	TI LI LO TS
2	IC50 = 5.25 nM Bioactivity Info	TI LI LO TS
CP0731528 Compound Info	(3R)-3-(4-(4-fluorophenyl)-1H-imidazol-2-yl)-1-phenyl-1-(trifluoromethyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole Show/Hide	C27H20F4N4	2
1	IC50 = 2.1 nM Bioactivity Info	TI LI LO TS
2	IC50 = 13.3 nM Bioactivity Info	TI LI LO TS
CP0664423 Compound Info	2-((1R,3R)-1-(1-ethyl-1H-pyrazol-4-yl)-3-(4-(5-fluoropyridin-2-yl)-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indol-1-yl)-5-methyl-1,3,4-oxadiazole Show/Hide	C27H24FN9O	2
1	IC50 = 2.2 nM Bioactivity Info	TI LI LO TS
2	IC50 = 4.8 nM Bioactivity Info	TI LI LO TS
CP0664253 Compound Info	5-((1R,3R)-1-(1-ethyl-1H-pyrazol-4-yl)-3-(4-(5-fluoropyridin-2-yl)-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indol-1-yl)-N-methyl-1,3,4-oxadiazol-2-amine Show/Hide	C27H25FN10O	2
1	IC50 = 2.2 nM Bioactivity Info	TI LI LO TS
2	IC50 = 3.5 nM Bioactivity Info	TI LI LO TS
CP0057457 Compound Info	3-[(1S,3S)-3-[5-(4-fluorophenyl)-1H-imidazol-2-yl]-1-(1-methylpyrazol-4-yl)-2,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-5-methyl-1,2,4-oxadiazole Show/Hide	C27H23FN8O	2
1	IC50 = 2.3 nM Bioactivity Info	TI LI LO TS
2	IC50 = 3.6 nM Bioactivity Info	TI LI LO TS
CP0727500 Compound Info	6-((1S,3R)-3-(4-(4-fluorophenyl)-1H-imidazol-2-yl)-1-(1-methyl-1H-pyrazol-4-yl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indol-1-yl)nicotinicacid Show/Hide	C30H24FN7O2	4
1	IC50 = 2.4 nM Bioactivity Info	TI LI LO TS
2	IC50 = 7.9 nM Bioactivity Info	TI LI LO TS
3	IC50 = 23.7 nM Bioactivity Info	TI LI LO TS
4	IC50 = 87.2 nM Bioactivity Info	TI LI LO TS
CP0667449 Compound Info	3-((1R,3R)-3-(4-(5-fluoropyridin-2-yl)-1H-imidazol-2-yl)-1-(1-methyl-1H-pyrazol-4-yl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indol-1-yl)-5-methyl-1,2,4-oxadiazole Show/Hide	C26H22FN9O	2
1	IC50 = 2.5 nM Bioactivity Info	TI LI LO TS
2	IC50 = 3 nM Bioactivity Info	TI LI LO TS
CP0709139 Compound Info	(3R)-1-cyclohexyl-3-(4-(5-fluoropyridin-2-yl)-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole Show/Hide	C25H26FN5	2
1	IC50 = 2.6 nM Bioactivity Info	TI LI LO TS
2	IC50 = 4.8 nM Bioactivity Info	TI LI LO TS
CP0140617 Compound Info	(1R,3R)-3-[5-(4-fluorophenyl)-1H-imidazol-2-yl]-1-(oxan-4-yl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole Show/Hide	C25H25FN4O	2
1	IC50 = 2.8 nM Bioactivity Info	TI LI LO TS
2	IC50 = 5.7 nM Bioactivity Info	TI LI LO TS
CP0848007 Compound Info	ethyl6-((1R,3R)-3-(4-(4-fluorophenyl)-1H-imidazol-2-yl)-1-(1-methyl-1H-pyrazol-4-yl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indol-1-yl)nicotinate Show/Hide	C32H28FN7O2	2
1	IC50 = 2.91 nM Bioactivity Info	TI LI LO TS
2	IC50 = 31.6 nM Bioactivity Info	TI LI LO TS
CP0776355 Compound Info	5-((1R,3R)-1-(1-ethyl-1H-pyrazol-4-yl)-3-(4-(5-fluoropyridin-2-yl)-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indol-1-yl)-1,3,4-oxadiazole-2-thiol Show/Hide	C26H22FN9OS	2
1	IC50 = 3.3 nM Bioactivity Info	TI LI LO TS
2	IC50 = 7.6 nM Bioactivity Info	TI LI LO TS
CP0396794 Compound Info	ethyl 5-[(1S,3R)-3-[5-(4-fluorophenyl)-1H-imidazol-2-yl]-1-(1-methylpyrazol-4-yl)-2,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]pyridine-3-carboxylate Show/Hide	C32H28FN7O2	2
1	IC50 = 3.36 nM Bioactivity Info	TI LI LO TS
2	IC50 = 24 nM Bioactivity Info	TI LI LO TS
CP0767445 Compound Info	5-((1R,3R)-1-(1-ethyl-1H-pyrazol-4-yl)-3-(4-(5-fluoropyridin-2-yl)-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indol-1-yl)-1,3,4-oxadiazol-2-ol Show/Hide	C26H22FN9O2	2
1	IC50 = 3.5 nM Bioactivity Info	TI LI LO TS
2	IC50 = 5.4 nM Bioactivity Info	TI LI LO TS
CP0423874 Compound Info	methyl 4-[(3R)-3-(5-phenyl-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indol-1-yl]piperidine-1-carboxylate Show/Hide	C27H29N5O2	2
1	IC50 = 4 nM Bioactivity Info	TI LI LO TS
2	IC50 = 66 nM Bioactivity Info	TI LI LO TS
CP0664064 Compound Info	5-((1R,3R)-3-(4-(5-fluoropyridin-2-yl)-1H-imidazol-2-yl)-1-(1-methyl-1H-pyrazol-4-yl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indol-1-yl)-3-methyl-1,3,4-oxadiazol-2(3H)-one Show/Hide	C26H22FN9O2	2
1	IC50 = 4.3 nM Bioactivity Info	TI LI LO TS
2	IC50 = 4.5 nM Bioactivity Info	TI LI LO TS
CP0838810 Compound Info	6-((1S,3R)-3-(4-(4-fluorophenyl)-1H-imidazol-2-yl)-1-(1-methyl-1H-pyrazol-4-yl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indol-1-yl)picolinicacid Show/Hide	C30H24FN7O2	2
1	IC50 = 4.41 nM Bioactivity Info	TI LI LO TS
2	IC50 = 67 nM Bioactivity Info	TI LI LO TS
CP0651915 Compound Info	(3R)-3-(4-(4-fluorophenyl)-1H-imidazol-2-yl)-1-methyl-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole Show/Hide	C27H23FN4	2
1	IC50 = 4.6 nM Bioactivity Info	TI LI LO TS
2	IC50 = 15.7 nM Bioactivity Info	TI LI LO TS
CP0761914 Compound Info	5-((1R,3R)-1-(1-ethyl-1H-pyrazol-4-yl)-3-(4-(5-fluoropyridin-2-yl)-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indol-1-yl)-N,N-dimethyl-1,3,4-oxadiazol-2-amine Show/Hide	C28H27FN10O	2
1	IC50 = 4.6 nM Bioactivity Info	TI LI LO TS
2	IC50 = 4.7 nM Bioactivity Info	TI LI LO TS
CP0915242 Compound Info	2-ethyl-5-((1R,3R)-3-(4-(5-fluoropyridin-2-yl)-1H-imidazol-2-yl)-1-(1-methyl-1H-pyrazol-4-yl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indol-1-yl)-1,3,4-oxadiazole Show/Hide	C27H24FN9O	2
1	IC50 = 4.6 nM Bioactivity Info	TI LI LO TS
2	IC50 = 5.1 nM Bioactivity Info	TI LI LO TS
CP0362610 Compound Info	ethyl 2-[(1S,3R)-3-[5-(4-fluorophenyl)-1H-imidazol-2-yl]-1-(1-methylpyrazol-4-yl)-2,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]pyridine-4-carboxylate Show/Hide	C32H28FN7O2	2
1	IC50 = 4.87 nM Bioactivity Info	TI LI LO TS
2	IC50 = 47.1 nM Bioactivity Info	TI LI LO TS
CP0765589 Compound Info	2-((1R,3R)-3-(4-(5-fluoropyridin-2-yl)-1H-imidazol-2-yl)-1-(1-methyl-1H-pyrazol-4-yl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indol-1-yl)-5-methyl-1,3,4-oxadiazole Show/Hide	C26H22FN9O	2
1	IC50 = 4.9 nM Bioactivity Info	TI LI LO TS
2	IC50 = 6.9 nM Bioactivity Info	TI LI LO TS
CP0787641 Compound Info	5-((1R,3R)-3-(4-(5-fluoropyridin-2-yl)-1H-imidazol-2-yl)-1-(1-methyl-1H-pyrazol-4-yl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indol-1-yl)-1,3,4-oxadiazol-2-amine Show/Hide	C25H21FN10O	2
1	IC50 = 5.3 nM Bioactivity Info	TI LI LO TS
2	IC50 = 5.6 nM Bioactivity Info	TI LI LO TS
CP0857551 Compound Info	5-((1S,3R)-3-(4-(4-fluorophenyl)-1H-imidazol-2-yl)-1-(1-methyl-1H-pyrazol-4-yl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indol-1-yl)nicotinicacid Show/Hide	C30H24FN7O2	2
1	IC50 = 6.12 nM Bioactivity Info	TI LI LO TS
2	IC50 = 10.8 nM Bioactivity Info	TI LI LO TS
CP0145754 Compound Info	(1R,3R)-3-[5-(4-fluorophenyl)-1H-imidazol-2-yl]-1-(1-methylpyrazol-4-yl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole Show/Hide	C24H21FN6	2
1	IC50 = 6.9 nM Bioactivity Info	TI LI LO TS
2	IC50 = 9.3 nM Bioactivity Info	TI LI LO TS
CP0425384 Compound Info	tert-butyl 4-[(3R)-3-(5-phenyl-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indol-1-yl]piperidine-1-carboxylate Show/Hide	C30H35N5O2	2
1	IC50 = 7 nM Bioactivity Info	TI LI LO TS
2	IC50 = 1000 nM Bioactivity Info	TI LI LO TS
CP0283794 Compound Info	(1S,3R)-3-[5-(4-fluorophenyl)-1H-imidazol-2-yl]-1-(1-methylpyrazol-4-yl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole Show/Hide	C24H21FN6	2
1	IC50 = 7.2 nM Bioactivity Info	TI LI LO TS
2	IC50 = 33 nM Bioactivity Info	TI LI LO TS
CP0381316 Compound Info	3-[(1R,3R)-3-[5-(4-fluorophenyl)-1H-imidazol-2-yl]-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indol-1-yl]-5-methyl-1,2,4-oxadiazole Show/Hide	C23H19FN6O	2
1	IC50 = 9.2 nM Bioactivity Info	TI LI LO TS
2	IC50 = 58 nM Bioactivity Info	TI LI LO TS
CP0076698 Compound Info	(1R,3R)-1-(oxan-4-yl)-3-(5-phenyl-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole Show/Hide	C25H26N4O	3
1	IC50 = 11 nM Bioactivity Info	TI LI LO TS
2	IC50 = 14 nM Bioactivity Info	TI LI LO TS
3	IC50 = 22 nM Bioactivity Info	TI LI LO TS
CP0664062 Compound Info	3-((1R,3R)-3-(4-(5-fluoropyridin-2-yl)-1H-imidazol-2-yl)-1-(1H-pyrazol-4-yl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indol-1-yl)-5-methyl-1,2,4-oxadiazole Show/Hide	C25H20FN9O	2
1	IC50 = 11 nM Bioactivity Info	TI LI LO TS
2	IC50 = 20.4 nM Bioactivity Info	TI LI LO TS
CP0851110 Compound Info	(3-((1R,3R)-3-(4-(5-fluoropyridin-2-yl)-1H-imidazol-2-yl)-1-(1-methyl-1H-pyrazol-4-yl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indol-1-yl)-1,2,4-oxadiazol-5-yl)methanamine Show/Hide	C26H23FN10O	2
1	IC50 = 11.1 nM Bioactivity Info	TI LI LO TS
2	IC50 = 13.7 nM Bioactivity Info	TI LI LO TS
CP0709883 Compound Info	(3R)-1-cyclohexyl-3-(4-(pyridin-2-yl)-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole Show/Hide	C25H27N5	2
1	IC50 = 11.3 nM Bioactivity Info	TI LI LO TS
2	IC50 = 28.1 nM Bioactivity Info	TI LI LO TS
CP0717937 Compound Info	(R)-3-(4-(4-fluorophenyl)-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole Show/Hide	C20H17FN4	2
1	IC50 = 11.4 nM Bioactivity Info	TI LI LO TS
2	IC50 = 15 nM Bioactivity Info	TI LI LO TS
CP0667445 Compound Info	(3R)-1-cyclohexyl-3-(4-(pyridin-4-yl)-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole Show/Hide	C25H27N5	2
1	IC50 = 11.5 nM Bioactivity Info	TI LI LO TS
2	IC50 = 17.2 nM Bioactivity Info	TI LI LO TS
CP0452268 Compound Info	1-[4-[(3R)-3-(5-phenyl-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indol-1-yl]piperidin-1-yl]ethanone Show/Hide	C27H29N5O	2
1	IC50 = 16 nM Bioactivity Info	TI LI LO TS
2	IC50 = 46 nM Bioactivity Info	TI LI LO TS
CP0707930 Compound Info	5-((1R,3R)-3-(4-(5-fluoropyridin-2-yl)-1H-imidazol-2-yl)-1-(1H-pyrazol-4-yl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indol-1-yl)-3-methyl-1,3,4-oxadiazol-2(3H)-one Show/Hide	C25H20FN9O2	2
1	IC50 = 17.3 nM Bioactivity Info	TI LI LO TS
2	IC50 = 17.5 nM Bioactivity Info	TI LI LO TS
CP0381407 Compound Info	3-[(1S,3R)-3-[5-(4-fluorophenyl)-1H-imidazol-2-yl]-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indol-1-yl]-5-methyl-1,2,4-oxadiazole Show/Hide	C23H19FN6O	1
1	IC50 = 19 nM Bioactivity Info	TI LI LO TS
CP0691633 Compound Info	(3R)-1-cyclohexyl-3-(4-(pyridin-3-yl)-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole Show/Hide	C25H27N5	2
1	IC50 = 20 nM Bioactivity Info	TI LI LO TS
2	IC50 = 28.6 nM Bioactivity Info	TI LI LO TS
CP0787643 Compound Info	(3R)-3-(4-(5-Fluoropyridin-2-yl)-1H-imidazol-2-yl)-1-(1-ethyl-pyrazol-4-yl)-1-(2-hydroxy-1,3,4-oxadiazol-5-yl)-2,3,4,9-tetrahydro-1H-beta-carboline Show/Hide	C27H24FN9O2	2
1	IC50 = 24.2 nM Bioactivity Info	TI LI LO TS
2	IC50 = 137.9 nM Bioactivity Info	TI LI LO TS
CP0731527 Compound Info	(R)-3-(4-(4-fluorophenyl)-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-carbazole Show/Hide	C21H18FN3	2
1	IC50 = 24.9 nM Bioactivity Info	TI LI LO TS
2	IC50 = 538.6 nM Bioactivity Info	TI LI LO TS
CP0885987 Compound Info	(3R)-1-cyclohexyl-3-(4-phenyl-1H-imidazol-2-yl)-1,3,4,9-tetrahydropyrano[3,4-b]indole Show/Hide	C26H27N3O	2
1	IC50 = 25.3 nM Bioactivity Info	TI LI LO TS
2	IC50 = 156.6 nM Bioactivity Info	TI LI LO TS
CP0383434 Compound Info	N-methyl-4-[(3R)-3-(5-phenyl-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indol-1-yl]piperidine-1-carboxamide Show/Hide	C27H30N6O	2
1	IC50 = 35 nM Bioactivity Info	TI LI LO TS
2	IC50 = 180 nM Bioactivity Info	TI LI LO TS
CP0383433 Compound Info	(3R)-1-(1-methylsulfonylpiperidin-4-yl)-3-(5-phenyl-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole Show/Hide	C26H29N5O2S	1
1	IC50 = 44 nM Bioactivity Info	TI LI LO TS
CP0849068 Compound Info	2-((1R,3R)-3-(4-(4-fluorophenyl)-1H-imidazol-2-yl)-1-(1-methyl-1H-pyrazol-4-yl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indol-1-yl)isonicotinicacid Show/Hide	C30H24FN7O2	2
1	IC50 = 52.3 nM Bioactivity Info	TI LI LO TS
2	IC50 = 72.7 nM Bioactivity Info	TI LI LO TS
CP0839308 Compound Info	(3R)-1-cyclohexyl-3-(4-(pyrazin-2-yl)-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole Show/Hide	C24H26N6	2
1	IC50 = 53.3 nM Bioactivity Info	TI LI LO TS
2	IC50 = 134.6 nM Bioactivity Info	TI LI LO TS
CP0423873 Compound Info	(3R)-3-(5-phenyl-1H-imidazol-2-yl)-1-piperidin-4-yl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole Show/Hide	C25H27N5	2
1	IC50 = 63 nM Bioactivity Info	TI LI LO TS
2	IC50 = 220 nM Bioactivity Info	TI LI LO TS
CP0849099 Compound Info	6-((1R,3R)-3-(4-(4-fluorophenyl)-1H-imidazol-2-yl)-1-(1-methyl-1H-pyrazol-4-yl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indol-1-yl)picolinicacid Show/Hide	C30H24FN7O2	2
1	IC50 = 74.7 nM Bioactivity Info	TI LI LO TS
2	IC50 = 105 nM Bioactivity Info	TI LI LO TS
CP0914208 Compound Info	5-(1-(1-ethyl-1H-pyrazol-4-yl)-3-(4-(5-fluoropyridin-2-yl)-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indol-1-yl)-3-methyl-1,3,4-oxadiazol-2(3H)-one Show/Hide	C27H24FN9O2	2
1	IC50 = 75.4 nM Bioactivity Info	TI LI LO TS
2	IC50 = 76.7 nM Bioactivity Info	TI LI LO TS
CP0383432 Compound Info	4-[(3R)-3-(5-phenyl-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indol-1-yl]thiane 1,1-dioxide Show/Hide	C25H26N4O2S	2
1	IC50 = 120 nM Bioactivity Info	TI LI LO TS
2	IC50 = 290 nM Bioactivity Info	TI LI LO TS
CP0504796 Compound Info	(1S,3R)-1-(oxan-4-yl)-3-(5-phenyl-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole Show/Hide	C25H26N4O	2
1	IC50 = 390 nM Bioactivity Info	TI LI LO TS
2	IC50 = 1200 nM Bioactivity Info	TI LI LO TS
CP0864058 Compound Info	6-((1R,3R)-3-(4-(4-fluorophenyl)-1H-imidazol-2-yl)-1-(1-methyl-1H-pyrazol-4-yl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indol-1-yl)nicotinicacid Show/Hide	C30H24FN7O2	2
1	IC50 = 409 nM Bioactivity Info	TI LI LO TS
2	IC50 > 2000 nM Bioactivity Info	TI LI LO TS
CP0787640 Compound Info	3-((1R,3R)-3-(4-(5-fluoropyridin-2-yl)-1H-imidazol-2-yl)-1-(1-methyl-1H-pyrazol-4-yl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indol-1-yl)-1,2,4-oxadiazol-5-ol Show/Hide	C25H20FN9O2	2
1	IC50 = 888.4 nM Bioactivity Info	TI LI LO TS
2	IC50 = 1948 nM Bioactivity Info	TI LI LO TS
CP0049566 Compound Info	15-28-Somatostatin-28 Show/Hide	C76H104N18O19S2	2
1	Ki = 0.14 nM Bioactivity Info	TI LI LO TS
2	Ki = 0.2512 nM Bioactivity Info	TI LI LO TS
CP0403938 Compound Info	[(3S,6S,9S,12R,15S,18S,20R)-9-(4-aminobutyl)-3,15-dibenzyl-12-(1H-indol-3-ylmethyl)-2,5,8,11,14,17-hexaoxo-6-[(4-phenylmethoxyphenyl)methyl]-1,4,7,10,13,16-hexazabicyclo[16.3.0]henicosan-20-yl] N-[2-(dimethylamino)ethyl]carbamate Show/Hide	C61H72N10O9	1
1	Ki = 0.3162 nM Bioactivity Info	TI LI LO TS
CP0406383 Compound Info	(4R,7S,10S,13S,16S,19S,22S,25S,28S,31S,34S,37R)-19,34-bis(4-aminobutyl)-31-(2-amino-2-oxoethyl)-37-[[2-[[(2S)-2-aminopropanoyl]amino]acetyl]amino]-13,25,28-tribenzyl-16-[(1R)-1-hydroxyethyl]-7-(hydroxymethyl)-22-(1H-indol-3-ylmethyl)-10-methyl-6,9,12,15,18,21,24,27,30,33,36-undecaoxo-1,2-dithia-5,8,11,14,17,20,23,26,29,32,35-undecazacyclooctatriacontane-4-carboxamide Show/Hide	C75H103N19O17S2	1
1	Ki = 0.631 nM Bioactivity Info	TI LI LO TS
CP0425318 Compound Info	[(3S,6S,9S,12R,15S,18S,20R)-9-(4-aminobutyl)-3-benzyl-15-[(4-hydroxyphenyl)methyl]-12-(1H-indol-3-ylmethyl)-2,5,8,11,14,17-hexaoxo-6-[(4-phenylmethoxyphenyl)methyl]-1,4,7,10,13,16-hexazabicyclo[16.3.0]henicosan-20-yl] N-(2-aminoethyl)carbamate Show/Hide	C59H68N10O10	1
1	Ki = 0.631 nM Bioactivity Info	TI LI LO TS
CP0430413 Compound Info	(4R,7S,10S,13S,16S,19S,22S,25S,28S,31S,34S,37R)-19,34-bis(4-aminobutyl)-37-[[2-[[(2S)-2-aminopropanoyl]amino]acetyl]amino]-13,25,28-tribenzyl-10,16-bis[(1R)-1-hydroxyethyl]-7-(hydroxymethyl)-22-(1H-indol-3-ylmethyl)-31-methyl-6,9,12,15,18,21,24,27,30,33,36-undecaoxo-1,2-dithia-5,8,11,14,17,20,23,26,29,32,35-undecazacyclooctatriacontane-4-carboxamide Show/Hide	C75H104N18O17S2	1
1	Ki = 0.631 nM Bioactivity Info	TI LI LO TS
CP0432311 Compound Info	(4R,7S,10S,13S,16S,19S,22S,25S,28S,31S,34S,37R)-19,34-bis(4-aminobutyl)-31-(2-amino-2-oxoethyl)-37-[[2-[[(2S)-2-aminopropanoyl]amino]acetyl]amino]-13,25,28-tribenzyl-10,16-bis[(1R)-1-hydroxyethyl]-22-(1H-indol-3-ylmethyl)-7-methyl-6,9,12,15,18,21,24,27,30,33,36-undecaoxo-1,2-dithia-5,8,11,14,17,20,23,26,29,32,35-undecazacyclooctatriacontane-4-carboxamide Show/Hide	C76H105N19O17S2	1
1	Ki = 0.631 nM Bioactivity Info	TI LI LO TS
CP0403937 Compound Info	CHEBI:72312 Show/Hide	C58H66N10O9	1
1	Ki = 0.7943 nM Bioactivity Info	TI LI LO TS
CP0406372 Compound Info	[(3S,6S,9S,12R,15S,18S,20R)-9-(4-aminobutyl)-3-benzyl-15-(1H-imidazol-5-ylmethyl)-12-(1H-indol-3-ylmethyl)-2,5,8,11,14,17-hexaoxo-6-[(4-phenylmethoxyphenyl)methyl]-1,4,7,10,13,16-hexazabicyclo[16.3.0]henicosan-20-yl] N-(2-aminoethyl)carbamate Show/Hide	C56H66N12O9	1
1	Ki = 0.7943 nM Bioactivity Info	TI LI LO TS
CP0485884 Compound Info	(4R,7S,10S,13S,16S,19S,22S,25S,28S,31S,34S,37R)-19,34-bis(4-aminobutyl)-31-(2-amino-2-oxoethyl)-37-[[(2S)-2-[[(2S)-2-aminopropanoyl]amino]propanoyl]amino]-13,25,28-tribenzyl-10,16-bis[(1R)-1-hydroxyethyl]-7-(hydroxymethyl)-22-(1H-indol-3-ylmethyl)-6,9,12,15,18,21,24,27,30,33,36-undecaoxo-1,2-dithia-5,8,11,14,17,20,23,26,29,32,35-undecazacyclooctatriacontane-4-carboxamide Show/Hide	C77H107N19O18S2	1
1	Ki = 0.7943 nM Bioactivity Info	TI LI LO TS
CP0492743 Compound Info	[(3S,6S,9S,12R,15S,18S,20R)-9-(4-aminobutyl)-3,15-dibenzyl-12-(1H-indol-3-ylmethyl)-2,5,8,11,14,17-hexaoxo-6-[(4-phenylmethoxyphenyl)methyl]-1,4,7,10,13,16-hexazabicyclo[16.3.0]henicosan-20-yl] N-(2-aminoethyl)carbamate Show/Hide	C59H68N10O9	1
1	Ki = 0.7943 nM Bioactivity Info	TI LI LO TS
CP0470520 Compound Info	(4R,7S,10R,13S,16R,19S,22R,25S,28R,31S,34R,37S)-19,34-bis(4-aminobutyl)-31-(2-amino-2-oxoethyl)-37-[[2-[[(2S)-2-aminopropanoyl]amino]acetyl]amino]-13,25,28-tribenzyl-16-[(1S)-1-hydroxyethyl]-10-[(1R)-1-hydroxyethyl]-7-(hydroxymethyl)-22-(1H-indol-3-ylmethyl)-6,9,12,15,18,21,24,27,30,33,36-undecaoxo-1,2-dithia-5,8,11,14,17,20,23,26,29,32,35-undecazacyclooctatriacontane-4-carboxylic acid Show/Hide	C76H104N18O19S2	1
1	Ki = 1.2 nM Bioactivity Info	TI LI LO TS
CP0050675 Compound Info	(4R,7R,10S,13S,16S,19S,22S,25S,28S,31S,34S,37R)-37-{2-[(2S)-2-[(2S)-6-amino-2-[(2S)-2-[(2S)-2-[(2S)-2-{[(2S)-1-[(2S)-2-[(2S)-2-[(2S)-2-{[(2S)-1-[(2R)-2-[(2S)-2-[(2S)-2-[(2S)-2-[(2S)-2-amino-3-hydroxypropanamido]propanamido]-3-carbamoylpropanamido]-3-hydroxypropanamido]-3-carbamoylpropanoyl]pyrrolidin-2-yl]formamido}propanamido]-4-(methylsulfanyl)butanamido]propanoyl]pyrrolidin-2-yl]formamido}-5-carbamimidamidopentanamido]-4-carboxybutanamido]-5-carbamimidamidopentanamido]hexanamido]propanamido]a Show/Hide	C137H207N41O39S3	1
1	Ki = 1.3 nM Bioactivity Info	TI LI LO TS
CP0404418 Compound Info	(4R,7S,10S,13S,16S,19S,22S,25S,28S,31S,34S,37R)-19,34-bis(4-aminobutyl)-31-(2-amino-2-oxoethyl)-37-[[2-[[(2S)-2-aminopropanoyl]amino]acetyl]amino]-13,25,28-tribenzyl-10-[(1R)-1-hydroxyethyl]-7-(hydroxymethyl)-22-(1H-indol-3-ylmethyl)-16-methyl-6,9,12,15,18,21,24,27,30,33,36-undecaoxo-1,2-dithia-5,8,11,14,17,20,23,26,29,32,35-undecazacyclooctatriacontane-4-carboxamide Show/Hide	C75H103N19O17S2	1
1	Ki = 1.585 nM Bioactivity Info	TI LI LO TS
CP0416639 Compound Info	(3S,6S,9S,12R,15S,18S,20R)-9-(4-aminobutyl)-3,15-dibenzyl-20-hydroxy-12-(1H-indol-3-ylmethyl)-6-[(4-phenylmethoxyphenyl)methyl]-1,4,7,10,13,16-hexazabicyclo[16.3.0]henicosane-2,5,8,11,14,17-hexone Show/Hide	C56H62N8O8	1
1	Ki = 1.585 nM Bioactivity Info	TI LI LO TS
CP0375513 Compound Info	[(3S,6S,9S,12R,15S,18S,20R)-9-(4-aminobutyl)-3,15-dibenzyl-12-(1H-indol-3-ylmethyl)-2,5,8,11,14,17-hexaoxo-6-[(4-phenylmethoxyphenyl)methyl]-1,4,7,10,13,16-hexazabicyclo[16.3.0]henicosan-20-yl] N-(5-aminopentyl)carbamate Show/Hide	C62H74N10O9	1
1	Ki = 1.995 nM Bioactivity Info	TI LI LO TS
CP0398954 Compound Info	(4R,7S,10S,13S,16S,19S,22S,25S,28S,31S,34S,37R)-19-(4-aminobutyl)-31-(2-amino-2-oxoethyl)-37-[[2-[[(2S)-2-aminopropanoyl]amino]acetyl]amino]-13,25,28-tribenzyl-10,16-bis[(1R)-1-hydroxyethyl]-7-(hydroxymethyl)-22-(1H-indol-3-ylmethyl)-34-methyl-6,9,12,15,18,21,24,27,30,33,36-undecaoxo-1,2-dithia-5,8,11,14,17,20,23,26,29,32,35-undecazacyclooctatriacontane-4-carboxylic acid Show/Hide	C73H97N17O19S2	1
1	Ki = 2.512 nM Bioactivity Info	TI LI LO TS
CP0049568 Compound Info	(4R,7S,10S,13R,16S,19R)-10-(4-aminobutyl)-19-[[(2R)-2-amino-3-phenylpropanoyl]amino]-16-benzyl-N-[(2S,3R)-1,3-dihydroxybutan-2-yl]-7-[(1R)-1-hydroxyethyl]-13-(1H-indol-3-ylmethyl)-6,9,12,15,18-pentaoxo-1,2-dithia-5,8,11,14,17-pentazacycloicosane-4-carboxamide Show/Hide	C49H66N10O10S2	1
1	Ki = 5.012 nM Bioactivity Info	TI LI LO TS
CP0404159 Compound Info	(4R,7S,10S,13S,16S,19S,22S,25S,28S,31S,34S,37R)-19,34-bis(4-aminobutyl)-31-(2-amino-2-oxoethyl)-37-[[2-[[(2S)-2-aminopropanoyl]amino]acetyl]amino]-25,28-dibenzyl-10,16-bis[(1R)-1-hydroxyethyl]-7-(hydroxymethyl)-22-(1H-indol-3-ylmethyl)-13-methyl-6,9,12,15,18,21,24,27,30,33,36-undecaoxo-1,2-dithia-5,8,11,14,17,20,23,26,29,32,35-undecazacyclooctatriacontane-4-carboxamide Show/Hide	C70H101N19O18S2	1
1	Ki = 7.943 nM Bioactivity Info	TI LI LO TS
CP0375512 Compound Info	(4R,7S,10S,13R,16S,19R)-10-(4-aminobutyl)-N-[(2S)-1-amino-3-(1H-indol-3-yl)-1-oxopropan-2-yl]-19-[[(2R)-2-amino-3-phenylpropanoyl]amino]-16-[(4-hydroxyphenyl)methyl]-13-(1H-indol-3-ylmethyl)-6,9,12,15,18-pentaoxo-7-propan-2-yl-1,2-dithia-5,8,11,14,17-pentazacycloicosane-4-carboxamide Show/Hide	C57H70N12O9S2	1
1	Ki = 19.95 nM Bioactivity Info	TI LI LO TS
CP0463563 Compound Info	[(3S,6S,9S,12R,15S,18S,20R)-9-(4-aminobutyl)-3-benzyl-15-[3-(diaminomethylideneamino)propyl]-12-(1H-indol-3-ylmethyl)-2,5,8,11,14,17-hexaoxo-6-[(4-phenylmethoxyphenyl)methyl]-1,4,7,10,13,16-hexazabicyclo[16.3.0]henicosan-20-yl] N-(2-aminoethyl)carbamate Show/Hide	C56H71N13O9	1
1	Ki = 19.95 nM Bioactivity Info	TI LI LO TS
CP0845116 Compound Info	Cpa-cyclo(DCys-Pal-DTrp-Dab-Thr-Cys)-Nal-NH2 Show/Hide	C55H63ClN12O9S2	1
1	Ki = 23.6 nM Bioactivity Info	TI LI LO TS
CP0460931 Compound Info	(4R,7S,10S,13S,16S,19S,22S,25S,28S,31S,34S,37R)-19,34-bis(4-aminobutyl)-31-(2-amino-2-oxoethyl)-37-[[2-[[(2S)-2-aminopropanoyl]amino]acetyl]amino]-13,28-dibenzyl-10,16-bis[(1R)-1-hydroxyethyl]-7-(hydroxymethyl)-22-(1H-indol-3-ylmethyl)-25-methyl-6,9,12,15,18,21,24,27,30,33,36-undecaoxo-1,2-dithia-5,8,11,14,17,20,23,26,29,32,35-undecazacyclooctatriacontane-4-carboxamide Show/Hide	C70H101N19O18S2	1
1	Ki = 25.12 nM Bioactivity Info	TI LI LO TS
CP0151093 Compound Info	(3S,6S,9S,12R,15S,18S)-9-(4-Amino-butyl)-3-benzyl-15-(4-hydroxy-benzyl)-12-(1H-indol-3-ylmethyl)-6-isopropyl-1,18-dimethyl-1,4,7,10,13,16hexaaza-cyclooctadecane-2,5,8,11,14,17-hexaone Show/Hide	C44H56N8O7	1
1	Ki = 31.62 nM Bioactivity Info	TI LI LO TS
CP0421355 Compound Info	N'-[(1R)-2-(1H-indol-3-yl)-1-(5-phenyl-1H-imidazol-2-yl)ethyl]-4-methoxybenzenecarboximidamide Show/Hide	C27H25N5O	1
1	Ki = 36 nM Bioactivity Info	TI LI LO TS
CP0847340 Compound Info	Cpa-cyclo(DCys-Pal-DTrp-Lys-Thr-Cys)-Nal-NH2 Show/Hide	C57H67ClN12O9S2	1
1	Ki = 38.2 nM Bioactivity Info	TI LI LO TS
CP0854677 Compound Info	Tfm-cyclo(DCys-Pal-DTrp-NMeLys-Thr-Cys)-Nal-NH2 Show/Hide	C59H69F3N12O9S2	1
1	Ki = 40.2 nM Bioactivity Info	TI LI LO TS
CP0375444 Compound Info	3-(2-Naphtyl)-D-Ala-L-Cys(1)-L-Tyr-D-Trp-L-Lys-L-Val-L-Cys(1)-L-Thr-NH2 Show/Hide	C54H69N11O10S2	1
1	Ki = 63.1 nM Bioactivity Info	TI LI LO TS
CP0858062 Compound Info	Cpa-cyclo(DCys-Pal-DTrp-NMeLys-Thr-Cys)-Nal-NH2 Show/Hide	C58H69ClN12O9S2	1
1	Ki = 66 nM Bioactivity Info	TI LI LO TS
CP0861120 Compound Info	Cpa-cyclo(DCys-Pal-DTrp-Lys-NMeThr-Cys)-Nal-NH2 Show/Hide	C58H69ClN12O9S2	1
1	Ki = 68.7 nM Bioactivity Info	TI LI LO TS
CP0487505 Compound Info	4-Chloro-N-[(R)-2-(1H-indol-3-yl)-1-(4-phenyl-1H-imidazol-2-yl)-ethyl]-benzamidine Show/Hide	C26H22ClN5	1
1	Ki = 79 nM Bioactivity Info	TI LI LO TS
CP0847417 Compound Info	Cpa-cyclo(DCys-Pal-DTrp-NMeLys-Thr-Cys)-DTrp-NH2 Show/Hide	C56H68ClN13O9S2	1
1	Ki = 91.4 nM Bioactivity Info	TI LI LO TS
CP0136960 Compound Info	(4R,7S,10S,13R,16S,19S)-10-(4-aminobutyl)-19-[[(2S)-2-amino-3-(4-chlorophenyl)propanoyl]amino]-N-[(2S)-1-amino-3-naphthalen-2-yl-1-oxopropan-2-yl]-7-[(1R)-1-hydroxyethyl]-16-[(4-hydroxyphenyl)methyl]-13-(1H-indol-3-ylmethyl)-6,9,12,15,18-pentaoxo-1,2-dithia-5,8,11,14,17-pentazacycloicosane-4-carboxamide Show/Hide	C58H68ClN11O10S2	1
1	Ki = 115.1 nM Bioactivity Info	TI LI LO TS
CP0375504 Compound Info	(5S,8S,11S,14R,17S,19aS)-11-(4-Amino-butyl)-5,17-dibenzyl-8-((R)-1-hydroxy-ethyl)-14-(1H-indol-3-ylmethyl)-tetradecahydro-3a,6,9,12,15,18-hexaaza-cyclopentacyclooctadecene-4,7,10,13,16,19-hexaone Show/Hide	C44H54N8O7	1
1	Ki = 125.89 nM Bioactivity Info	TI LI LO TS
CP0912534 Compound Info	Cpa-cyclo(DCys-Pal-NMeDTrp-NMeLys-Thr-Cys)-Nal-NH2 Show/Hide	C59H71ClN12O9S2	1
1	Ki = 140 nM Bioactivity Info	TI LI LO TS
CP0902700 Compound Info	Nal-cyclo(DCys-Pal-DTrp-NMeLys-Thr-Cys)-DTrp-NH2 Show/Hide	C60H71N13O9S2	1
1	Ki = 148 nM Bioactivity Info	TI LI LO TS
CP0395005 Compound Info	1-(2,4-Difluoro-phenyl)-3-[(R)-2-(1H-indol-3-yl)-1-(4-phenyl-1H-imidazol-2-yl)-ethyl]-urea Show/Hide	C26H21F2N5O	1
1	Ki = 170 nM Bioactivity Info	TI LI LO TS
CP0412492 Compound Info	(3S,6S,9S,12R,15S,18S,20R)-9-(4-aminobutyl)-3,15-dibenzyl-20-hydroxy-6-[(1R)-1-hydroxyethyl]-12-(1H-indol-3-ylmethyl)-1,4,7,10,13,16-hexazabicyclo[16.3.0]henicosane-2,5,8,11,14,17-hexone Show/Hide	C44H54N8O8	1
1	Ki = 199.53 nM Bioactivity Info	TI LI LO TS
CP0485165 Compound Info	(4R,7S,10S,13S,16S,19S,22S,25S,28S,31S,34S,37R)-19,34-bis(4-aminobutyl)-31-(2-amino-2-oxoethyl)-37-[[2-[[(2S)-2-aminopropanoyl]amino]acetyl]amino]-13,25-dibenzyl-10,16-bis[(1R)-1-hydroxyethyl]-7-(hydroxymethyl)-22-(1H-indol-3-ylmethyl)-28-methyl-6,9,12,15,18,21,24,27,30,33,36-undecaoxo-1,2-dithia-5,8,11,14,17,20,23,26,29,32,35-undecazacyclooctatriacontane-4-carboxamide Show/Hide	C70H101N19O18S2	1
1	Ki = 199.53 nM Bioactivity Info	TI LI LO TS
CP0495082 Compound Info	2,4-Difluoro-N-[(R)-2-(1H-indol-3-yl)-1-(4-phenyl-1H-imidazol-2-yl)-ethyl]-benzamidine Show/Hide	C26H21F2N5	1
1	Ki = 200 nM Bioactivity Info	TI LI LO TS
CP0382365 Compound Info	tert-butyl N-[(1R)-2-(1H-indol-3-yl)-1-(5-phenyl-1H-imidazol-2-yl)ethyl]carbamate Show/Hide	C24H26N4O2	1
1	Ki = 210 nM Bioactivity Info	TI LI LO TS
CP0430098 Compound Info	N-[(1R)-2-(1H-indol-3-yl)-1-(5-phenyl-1H-imidazol-2-yl)ethyl]-2-[3-(trifluoromethyl)phenyl]acetamide Show/Hide	C28H23F3N4O	1
1	Ki = 240 nM Bioactivity Info	TI LI LO TS
CP0392901 Compound Info	N'-[(1R)-2-(1H-indol-3-yl)-1-(5-phenyl-1H-imidazol-2-yl)ethyl]benzenecarboximidamide Show/Hide	C26H23N5	1
1	Ki = 250 nM Bioactivity Info	TI LI LO TS
CP0862999 Compound Info	Cpa-cyclo(DCys-Pal-DTrp-Lys-NMeThr-Cys)-Nal-NH2 Show/Hide	C58H69ClN12O9S2	1
1	Ki = 315 nM Bioactivity Info	TI LI LO TS
CP0917823 Compound Info	NMeCpa-cyclo(DCys-Pal-DTrp-Lys-Thr-Cys)-Nal-NH2 Show/Hide	C58H69ClN12O9S2	1
1	Ki = 330 nM Bioactivity Info	TI LI LO TS
CP0847584 Compound Info	Cpa-cyclo(DCys-Pal-NMeDTrp-Lys-Thr-Cys)-Nal-NH2 Show/Hide	C58H69ClN12O9S2	1
1	Ki = 390 nM Bioactivity Info	TI LI LO TS
CP0376599 Compound Info	1-tert-Butyl-3-[(R)-2-(1H-indol-3-yl)-1-(4-phenyl-1H-imidazol-2-yl)-ethyl]-urea Show/Hide	C24H27N5O	1
1	Ki = 400 nM Bioactivity Info	TI LI LO TS
CP0421312 Compound Info	N'-[(1R)-2-(1H-indol-3-yl)-1-(5-phenyl-1H-imidazol-2-yl)ethyl]-4-(trifluoromethoxy)benzenecarboximidamide Show/Hide	C27H22F3N5O	1
1	Ki = 410 nM Bioactivity Info	TI LI LO TS
CP0888162 Compound Info	Cpa-cyclo(DCys-NMePal-DTrp-Lys-Thr-Cys)-Nal-NH2 Show/Hide	C58H69ClN12O9S2	1
1	Ki = 450 nM Bioactivity Info	TI LI LO TS
CP0404417 Compound Info	N'-[(1R)-2-(1H-indol-3-yl)-1-(5-phenyl-1H-imidazol-2-yl)ethyl]-4-(trifluoromethyl)benzenecarboximidamide Show/Hide	C27H22F3N5	1
1	Ki = 500 nM Bioactivity Info	TI LI LO TS
CP0880716 Compound Info	Pal-cyclo(DCys-Pal-DTrp-NMeLys-Thr-Cys)-DTrp-NH2 Show/Hide	C55H68N14O9S2	1
1	Ki = 537 nM Bioactivity Info	TI LI LO TS
CP0886292 Compound Info	Cpa-cyclo(NMeDCys-Pal-DTrp-Lys-Thr-Cys)-Nal-NH2 Show/Hide	C59H72N12O9S2	1
1	Ki = 576 nM Bioactivity Info	TI LI LO TS
CP0880603 Compound Info	Cpa-cyclo(NMeDCys-Pal-DTrp-Lys-Thr-Cys)-Dip-NHMe Show/Hide	C61H73ClN12O9S2	1
1	Ki = 584 nM Bioactivity Info	TI LI LO TS
CP0415095 Compound Info	N'-[(1R)-2-(1H-indol-3-yl)-1-(5-phenyl-1H-imidazol-2-yl)ethyl]ethanimidamide Show/Hide	C21H21N5	1
1	Ki = 700 nM Bioactivity Info	TI LI LO TS
CP0847290 Compound Info	Cpa-cyclo(DCys-Pal-DTrp-DDap-Thr-Cys)-Nal-NH2 Show/Hide	C54H61ClN12O9S2	1
1	Ki = 1000 nM Bioactivity Info	TI LI LO TS
CP0859471 Compound Info	Cpa-cyclo(DCys-Pal-DTrp-Lys-Thr-Cys)-NMeNal-NH2 Show/Hide	C58H69ClN12O9S2	1
1	Ki = 1000 nM Bioactivity Info	TI LI LO TS
CP0375876 Compound Info	(4R,7S,10S,13S,16S,19S,22S,25S,28S,31S,34S,37R)-19,34-bis(4-aminobutyl)-31-(2-amino-2-oxoethyl)-37-[[2-[[(2S)-2-aminopropanoyl]amino]acetyl]amino]-13,25,28-tribenzyl-10,16-bis[(1R)-1-hydroxyethyl]-7-(hydroxymethyl)-22-methyl-6,9,12,15,18,21,24,27,30,33,36-undecaoxo-1,2-dithia-5,8,11,14,17,20,23,26,29,32,35-undecazacyclooctatriacontane-4-carboxamide Show/Hide	C68H100N18O18S2	1
1	Ki = 1000 nM Bioactivity Info	TI LI LO TS
CP0425316 Compound Info	(4R,7S,10S,13S,16S,19S,22S,25S,28S,31S,34S,37R)-34-(4-aminobutyl)-31-(2-amino-2-oxoethyl)-37-[[2-[[(2S)-2-aminopropanoyl]amino]acetyl]amino]-13,25,28-tribenzyl-10,16-bis[(1R)-1-hydroxyethyl]-7-(hydroxymethyl)-22-(1H-indol-3-ylmethyl)-19-methyl-6,9,12,15,18,21,24,27,30,33,36-undecaoxo-1,2-dithia-5,8,11,14,17,20,23,26,29,32,35-undecazacyclooctatriacontane-4-carboxamide Show/Hide	C73H98N18O18S2	1
1	Ki = 1000 nM Bioactivity Info	TI LI LO TS
CP0377054 Compound Info	4-tert-Butyl-N-[(R)-2-(1H-indol-3-yl)-1-(4-phenyl-1H-imidazol-2-yl)-ethyl]-benzamidine Show/Hide	C30H31N5	1
1	Ki = 1400 nM Bioactivity Info	TI LI LO TS
CP0427962 Compound Info	N-(1H-indol-3-ylmethyl)-1-[5-(4-methylphenyl)-1H-imidazol-2-yl]cyclopropan-1-amine Show/Hide	C22H22N4	1
1	Ki = 1500 nM Bioactivity Info	TI LI LO TS

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About MolBiC

Correspondence

Prof. Feng ZHU

Prof. Leo, Lianyi Han