Brief Information of the Compound and Protein
Compound Name
(3R)-1-cyclohexyl-3-(4-(pyrazin-2-yl)-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole
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PubChem ID
CID: 122179455
Canonical SMILES
c1ccc2c3c([nH]c2c1)C(C1CCCCC1)N[C@@H](c1nc(-c2cnccn2)c[nH]1)C3
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Compound Formula C24H26N6
Compound Structure
Protein Name
Somatostatin receptor type 3
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Peptide receptor (family A GPCR)
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Short peptide receptor (family A GPCR)
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Somatostatin receptor
Uniprot ID
P32745
Gene Name
SSTR3
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  2
1
IC50 = 53.3 nM
   TI
   LI
   LO
   TS
2
IC50 = 134.6 nM
   TI
   LI
   LO
   TS