Brief Information of the Compound and Protein
Compound Name
2-[(1R,3R)-3-[5-(4-fluorophenyl)-1H-imidazol-2-yl]-1-(1-methylpyrazol-4-yl)-2,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]pyridine-4-carboxylic acid
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PubChem ID
CID: 86279005
Canonical SMILES
Cn1cc(cn1)[C@]1(N[C@H](Cc2c1[nH]c1ccccc21)c1nc(c[nH]1)-c1ccc(F)cc1)c1cc(ccn1)C(O)=O
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Compound Formula C30H24FN7O2
Compound Structure
Protein Name
Somatostatin receptor type 3
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Peptide receptor (family A GPCR)
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Short peptide receptor (family A GPCR)
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Somatostatin receptor
Uniprot ID
P32745
Gene Name
SSTR3
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  2
1
IC50 = 1.71 nM
   TI
   LI
   LO
   TS
2
IC50 = 2.13 nM
   TI
   LI
   LO
   TS