Brief Information of the Compound and Protein
Compound Name
(1R,3R)-3-[5-(4-fluorophenyl)-1H-imidazol-2-yl]-1-(oxan-4-yl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole
    Show/Hide
PubChem ID
CID: 71452299
Canonical SMILES
Fc1ccc(cc1)-c1c[nH]c(n1)[C@H]1Cc2c([nH]c3ccccc23)[C@H](N1)C1CCOCC1
    Show/Hide
Compound Formula C25H25FN4O
Compound Structure
Protein Name
Somatostatin receptor type 3
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
>
Peptide receptor (family A GPCR)
>
Short peptide receptor (family A GPCR)
>
Somatostatin receptor
Uniprot ID
P32745
Gene Name
SSTR3
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  2
1
IC50 = 2.8 nM
   TI
   LI
   LO
   TS
2
IC50 = 5.7 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 EC50 = 5.7 nM
2 IC50 = 2.8 nM