Brief Information of the Compound and Protein
Compound Name
(3R)-3-(4-(4-fluorophenyl)-1H-imidazol-2-yl)-1-phenyl-1-(trifluoromethyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole
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PubChem ID
CID: 122179451
Canonical SMILES
Fc1ccc(-c2c[nH]c([C@H]3Cc4c([nH]c5ccccc45)C(c4ccccc4)(C(F)(F)F)N3)n2)cc1
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Compound Formula C27H20F4N4
Compound Structure
Protein Name
Somatostatin receptor type 3
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
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Peptide receptor (family A GPCR)
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Short peptide receptor (family A GPCR)
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Somatostatin receptor
Uniprot ID
P32745
Gene Name
SSTR3
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  2
1
IC50 = 2.1 nM
   TI
   LI
   LO
   TS
2
IC50 = 13.3 nM
   TI
   LI
   LO
   TS