Brief Information of the Compound and Protein
Compound Name
(3R)-3-(4-(5-Fluoropyridin-2-yl)-1H-imidazol-2-yl)-1-(1-ethyl-pyrazol-4-yl)-1-(2-hydroxy-1,3,4-oxadiazol-5-yl)-2,3,4,9-tetrahydro-1H-beta-carboline
    Show/Hide
PubChem ID
CID: 46830055
SID: 99207687
Canonical SMILES
CCn1cc(C2(c3nn(C)c(=O)o3)N[C@@H](c3nc(-c4ccc(F)cn4)c[nH]3)Cc3c2[nH]c2ccccc32)cn1
    Show/Hide
Compound Formula C27H24FN9O2
Compound Structure
Protein Name
Somatostatin receptor type 3
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
>
Peptide receptor (family A GPCR)
>
Short peptide receptor (family A GPCR)
>
Somatostatin receptor
Uniprot ID
P32745
Gene Name
SSTR3
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  2
1
IC50 = 24.2 nM
   TI
   LI
   LO
   TS
2
IC50 = 137.9 nM
   TI
   LI
   LO
   TS