| Compound ID |
Compound Name |
Compound Formula |
|
CP0390968
|
N-[4-(5,7-dihydro-4H-thieno[2,3-c]pyridin-6-yl)-2,6-dimethylphenyl]-3,3-dimethylbutanamide
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|
C21H28N2OS
|
1
|
| 1 |
EC50 = 20 nM
|
|
|
|
CP0396553
|
N-[4-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)-2,6-dimethylphenyl]-3,3-dimethylbutanamide
Show/Hide
|
C21H28N2OS
|
1
|
| 1 |
EC50 = 20 nM
|
|
|
|
CP0566192
|
N-[2,6-dimethyl-4-(2-methyl-5,7-dihydro-4H-thieno[2,3-c]pyridin-6-yl)phenyl]-3,3-dimethylbutanamide
Show/Hide
|
C22H30N2OS
|
1
|
| 1 |
EC50 = 30 nM
|
|
|
|
CP0396555
|
N-[4-(3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl)-2,6-dimethylphenyl]-3,3-dimethylbutanamide
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|
C21H29N3O
|
1
|
| 1 |
EC50 = 34 nM
|
|
|
|
CP0429370
|
N-[2,6-dimethyl-4-(7-methyl-2,3,4,5-tetrahydro-1-benzazepin-1-yl)phenyl]-3,3-dimethylbutanamide
Show/Hide
|
C25H34N2O
|
1
|
| 1 |
EC50 = 40 nM
|
|
|
|
CP0559564
|
N-[2,6-dimethyl-4-[2-(trifluoromethyl)-6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl]phenyl]-3,3-dimethylbutanamide
Show/Hide
|
C22H27F3N2OS
|
1
|
| 1 |
EC50 = 120 nM
|
|
|
|
CP0384877
|
N-[2,6-dimethyl-4-(4-oxopiperidin-1-yl)phenyl]-3,3-dimethylbutanamide
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|
C19H28N2O2
|
1
|
| 1 |
EC50 = 130 nM
|
|
|
|
CP0396557
|
N-[4-(7-chloro-2,3,4,5-tetrahydro-1-benzazepin-1-yl)-2,6-dimethylphenyl]-3,3-dimethylbutanamide
Show/Hide
|
C24H31ClN2O
|
1
|
| 1 |
EC50 = 140 nM
|
|
|
|
CP0462948
|
2-(3-chlorophenyl)-N-(2-pyrrolidin-1-ylphenyl)acetamide
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|
C18H19ClN2O
|
1
|
| 1 |
EC50 = 170 nM
|
|
|
|
CP0521058
|
N-[4-[4-(3-fluorophenyl)piperidin-1-yl]-2,6-dimethylphenyl]-3,3-dimethylbutanamide
Show/Hide
|
C25H33FN2O
|
1
|
| 1 |
EC50 = 220 nM
|
|
|
|
CP0539240
|
N-[4-(7-fluoro-2,3,4,5-tetrahydro-1-benzazepin-1-yl)-2,6-dimethylphenyl]-3,3-dimethylbutanamide
Show/Hide
|
C24H31FN2O
|
1
|
| 1 |
EC50 = 250 nM
|
|
|
|
CP0396554
|
N-[4-(2-cyano-6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)-2,6-dimethylphenyl]-3,3-dimethylbutanamide
Show/Hide
|
C22H27N3OS
|
1
|
| 1 |
EC50 = 290 nM
|
|
|
|
CP0558685
|
N-[2,6-dimethyl-4-(3-methyl-6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)phenyl]-3,3-dimethylbutanamide
Show/Hide
|
C22H30N2OS
|
1
|
| 1 |
EC50 = 300 nM
|
|
|
|
CP0521798
|
N-[4-(3,4-dihydro-2H-quinolin-1-ylmethyl)-2,6-dimethylphenyl]-3,3-dimethylbutanamide
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|
C24H32N2O
|
1
|
| 1 |
EC50 = 330 nM
|
|
|
|
CP0547749
|
N-(2-pyrrolidin-1-ylphenyl)-2-[3-(trifluoromethyl)phenyl]acetamide
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|
C19H19F3N2O
|
1
|
| 1 |
EC50 = 350 nM
|
|
|
|
CP0002667
|
ethyl N-[2-amino-4-[(4-fluorophenyl)methylamino]phenyl]carbamate
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|
C16H18FN3O2
|
1
|
| 1 |
EC50 = 350 nM
|
|
|
|
CP0449667
|
2-(3-fluorophenyl)-N-(2-pyrrolidin-1-ylphenyl)acetamide
Show/Hide
|
C18H19FN2O
|
1
|
| 1 |
EC50 = 490 nM
|
|
|
|
CP0369109
|
2-(4-fluorophenyl)-N-(2-pyrrolidin-1-ylphenyl)acetamide
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|
C18H19FN2O
|
1
|
| 1 |
EC50 = 700 nM
|
|
|
|
CP0332835
|
2-phenyl-N-(2-pyrrolidin-1-ylphenyl)acetamide
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|
C18H20N2O
|
1
|
| 1 |
EC50 = 743 nM
|
|
|
|
CP0423658
|
2-(4-chlorophenyl)-N-(2-pyrrolidin-1-ylphenyl)acetamide
Show/Hide
|
C18H19ClN2O
|
1
|
| 1 |
EC50 = 800 nM
|
|
|
|
CP0515843
|
2-(2-chlorophenyl)-N-(2-pyrrolidin-1-ylphenyl)acetamide
Show/Hide
|
C18H19ClN2O
|
1
|
| 1 |
EC50 = 950 nM
|
|
|
|
CP0449668
|
2-fluoro-2-phenyl-N-(2-pyrrolidin-1-ylphenyl)acetamide
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|
C18H19FN2O
|
1
|
| 1 |
EC50 = 990 nM
|
|
|
|
CP0527341
|
2-(3-chlorophenyl)-N-(3-pyrrolidin-1-ylphenyl)acetamide
Show/Hide
|
C18H19ClN2O
|
1
|
| 1 |
EC50 = 1020 nM
|
|
|
|
CP0449666
|
2-(3,4-dichlorophenyl)-N-(2-pyrrolidin-1-ylphenyl)acetamide
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|
C18H18Cl2N2O
|
1
|
| 1 |
EC50 = 1070 nM
|
|
|
|
CP0396556
|
N-[4-(7-bromo-2,3,4,5-tetrahydro-1-benzazepin-1-yl)-2,6-dimethylphenyl]-3,3-dimethylbutanamide
Show/Hide
|
C24H31BrN2O
|
1
|
| 1 |
EC50 = 1080 nM
|
|
|
|
CP0397409
|
2-(3-methylphenyl)-N-(2-pyrrolidin-1-ylphenyl)acetamide
Show/Hide
|
C19H22N2O
|
1
|
| 1 |
EC50 = 1320 nM
|
|
|
|
CP0521797
|
N-[4-(4,4-dimethylpiperidin-1-yl)-2,6-dimethylphenyl]-3,3-dimethylbutanamide
Show/Hide
|
C21H34N2O
|
1
|
| 1 |
EC50 = 1580 nM
|
|
|
|
CP0397410
|
2-(3,4-difluorophenyl)-N-(2-pyrrolidin-1-ylphenyl)acetamide
Show/Hide
|
C18H18F2N2O
|
1
|
| 1 |
EC50 = 1730 nM
|
|
|
|
CP0460497
|
2-(4-methoxyphenyl)-N-(2-pyrrolidin-1-ylphenyl)acetamide
Show/Hide
|
C19H22N2O2
|
1
|
| 1 |
EC50 = 1750 nM
|
|
|
|
CP0449665
|
2-(3-methoxyphenyl)-N-(2-pyrrolidin-1-ylphenyl)acetamide
Show/Hide
|
C19H22N2O2
|
1
|
| 1 |
EC50 = 2350 nM
|
|
|
|
CP0559565
|
N-[4-(2-fluoro-5,7-dihydro-4H-thieno[2,3-c]pyridin-6-yl)-2,6-dimethylphenyl]-3,3-dimethylbutanamide
Show/Hide
|
C21H27FN2OS
|
1
|
| 1 |
EC50 = 2930 nM
|
|
|
|
CP0497888
|
2-(3-chlorophenyl)-N-(2-piperidin-1-ylphenyl)acetamide
Show/Hide
|
C19H21ClN2O
|
1
|
| 1 |
EC50 = 7090 nM
|
|
|
|
CP0479540
|
2-(3-chlorophenyl)-N-(4-pyrrolidin-1-ylphenyl)acetamide
Show/Hide
|
C18H19ClN2O
|
1
|
| 1 |
EC50 = 8660 nM
|
|
|
|
CP0449664
|
2-(3-chlorophenyl)-N-(2-pyrrol-1-ylphenyl)acetamide
Show/Hide
|
C18H15ClN2O
|
1
|
| 1 |
EC50 = 12270 nM
|
|
|
|
CP0527340
|
2-(3-chlorophenyl)-N-[2-(dimethylamino)phenyl]acetamide
Show/Hide
|
C16H17ClN2O
|
1
|
| 1 |
EC50 = 27420 nM
|
|
|
|
CP0165878
|
(2R)-N-[4-(4-methoxyphenyl)-1,3-thiazol-2-yl]-1-(4-methylphenyl)sulfonylpiperidine-2-carboxamide
Show/Hide
|
C23H25N3O4S2
|
1
|
| 1 |
EC50 > 30000 nM
|
|
|
|
CP0423653
|
N-[2-[benzyl(methyl)amino]phenyl]-2-(3-chlorophenyl)acetamide
Show/Hide
|
C22H21ClN2O
|
1
|
| 1 |
EC50 > 30000 nM
|
|
|
|
CP0479539
|
N-methyl-2-phenyl-N-(2-pyrrolidin-1-ylphenyl)acetamide
Show/Hide
|
C19H22N2O
|
1
|
| 1 |
EC50 > 30000 nM
|
|
|
|
CP0499733
|
2-(3-chlorophenyl)-N-(2-morpholin-4-ylphenyl)acetamide
Show/Hide
|
C18H19ClN2O2
|
1
|
| 1 |
EC50 > 30000 nM
|
|
|
|
CP0527339
|
N-[2-(2,5-dimethylpyrrol-1-yl)phenyl]-2-phenylbutanamide
Show/Hide
|
C22H24N2O
|
1
|
| 1 |
EC50 > 30000 nM
|
|
|
|
CP0553555
|
2-(3-chlorophenyl)-N-[2-[ethyl(methyl)amino]phenyl]acetamide
Show/Hide
|
C17H19ClN2O
|
1
|
| 1 |
EC50 > 30000 nM
|
|
|
|
CP0565832
|
N-[2-(azepan-1-yl)phenyl]-2-(3-chlorophenyl)acetamide
Show/Hide
|
C20H23ClN2O
|
1
|
| 1 |
EC50 > 30000 nM
|
|
|
|
CP0010522
|
(2S)-2-phenyl-N-(2-pyrrolidin-1-ylphenyl)butanamide
Show/Hide
|
C20H24N2O
|
1
|
| 1 |
IC50 = 70 nM
|
|
|
|
CP0462950
|
2-(3-methoxyphenyl)-N-(2-pyrrolidin-1-ylphenyl)butanamide
Show/Hide
|
C21H26N2O2
|
1
|
| 1 |
IC50 = 120 nM
|
|
|
|
CP0423660
|
2-(4-fluorophenyl)-N-(2-pyrrolidin-1-ylphenyl)butanamide
Show/Hide
|
C20H23FN2O
|
1
|
| 1 |
IC50 = 130 nM
|
|
|
|
CP0449671
|
2-phenyl-N-(2-pyrrolidin-1-ylphenyl)butanamide
Show/Hide
|
C20H24N2O
|
1
|
| 1 |
IC50 = 163 nM
|
|
|
|
CP0479542
|
2-(3,4-difluorophenyl)-N-(2-pyrrolidin-1-ylphenyl)butanamide
Show/Hide
|
C20H22F2N2O
|
1
|
| 1 |
IC50 = 170 nM
|
|
|
|
CP0426070
|
2-phenyl-N-(4-pyrrolidin-1-ylphenyl)butanamide
Show/Hide
|
C20H24N2O
|
1
|
| 1 |
IC50 = 210 nM
|
|
|
|
CP0553557
|
2-(3-chlorophenyl)-N-(2-pyrrolidin-1-ylphenyl)butanamide
Show/Hide
|
C20H23ClN2O
|
1
|
| 1 |
IC50 = 240 nM
|
|
|
|
CP0499735
|
2-phenyl-N-(2-pyrrolidin-1-ylphenyl)propanamide
Show/Hide
|
C19H22N2O
|
1
|
| 1 |
IC50 = 260 nM
|
|
|
|
CP0462949
|
2-(4-chlorophenyl)-N-(2-pyrrolidin-1-ylphenyl)butanamide
Show/Hide
|
C20H23ClN2O
|
1
|
| 1 |
IC50 = 280 nM
|
|
|
|
CP0397411
|
2-phenyl-N-(2-pyrrolidin-1-ylphenyl)pentanamide
Show/Hide
|
C21H26N2O
|
1
|
| 1 |
IC50 = 320 nM
|
|
|
|
CP0497890
|
2-(3-methylphenyl)-N-(2-pyrrolidin-1-ylphenyl)butanamide
Show/Hide
|
C21H26N2O
|
1
|
| 1 |
IC50 = 330 nM
|
|
|
|
CP0553559
|
N-(2-pyrrolidin-1-ylphenyl)-2,3-dihydro-1H-indene-1-carboxamide
Show/Hide
|
C20H22N2O
|
1
|
| 1 |
IC50 = 330 nM
|
|
|
|
CP0553558
|
2-(3-fluorophenyl)-N-(2-pyrrolidin-1-ylphenyl)butanamide
Show/Hide
|
C20H23FN2O
|
1
|
| 1 |
IC50 = 360 nM
|
|
|
|
CP0449670
|
2-(4-methoxyphenyl)-N-(2-pyrrolidin-1-ylphenyl)butanamide
Show/Hide
|
C21H26N2O2
|
1
|
| 1 |
IC50 = 380 nM
|
|
|
|
CP0547750
|
N-(2-pyrrolidin-1-ylphenyl)-2-[3-(trifluoromethyl)phenyl]butanamide
Show/Hide
|
C21H23F3N2O
|
1
|
| 1 |
IC50 = 390 nM
|
|
|
|
CP0449669
|
2-(2-fluorophenyl)-N-(2-pyrrolidin-1-ylphenyl)butanamide
Show/Hide
|
C20H23FN2O
|
1
|
| 1 |
IC50 = 440 nM
|
|
|
|
CP0499734
|
2-(3,4-dichlorophenyl)-N-(2-pyrrolidin-1-ylphenyl)butanamide
Show/Hide
|
C20H22Cl2N2O
|
1
|
| 1 |
IC50 = 470 nM
|
|
|
|
CP0285161
|
2-phenyl-N-(2-phenylphenyl)butanamide
Show/Hide
|
C22H21NO
|
1
|
| 1 |
IC50 = 1320 nM
|
|
|
|
CP0423662
|
4-methyl-2-phenyl-N-(2-pyrrolidin-1-ylphenyl)pentanamide
Show/Hide
|
C22H28N2O
|
1
|
| 1 |
IC50 = 2220 nM
|
|
|
|
CP0479541
|
2-(2-chlorophenyl)-N-(2-pyrrolidin-1-ylphenyl)butanamide
Show/Hide
|
C20H23ClN2O
|
1
|
| 1 |
IC50 = 3310 nM
|
|
|
|
CP0547761
|
2-cyclopropyl-2-phenyl-N-(2-pyrrolidin-1-ylphenyl)acetamide
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|
C21H24N2O
|
1
|
| 1 |
IC50 = 3500 nM
|
|
|
|
CP0397407
|
2-phenyl-N-(2-pyrrol-1-ylphenyl)butanamide
Show/Hide
|
C20H20N2O
|
1
|
| 1 |
IC50 = 5270 nM
|
|
|
|
CP0527342
|
N-(2-morpholin-4-ylphenyl)-2-phenylbutanamide
Show/Hide
|
C20H24N2O2
|
1
|
| 1 |
IC50 = 12670 nM
|
|
|
|
CP0449663
|
N-(2-chlorophenyl)-2-phenylbutanamide
Show/Hide
|
C16H16ClNO
|
1
|
| 1 |
IC50 = 14990 nM
|
|
|
|
CP0547760
|
2-(3,4-dimethoxyphenyl)-N-(2-pyrrolidin-1-ylphenyl)butanamide
Show/Hide
|
C22H28N2O3
|
1
|
| 1 |
IC50 = 20230 nM
|
|
|
|
CP0397408
|
N-[2-(azepan-1-yl)phenyl]-2-phenylbutanamide
Show/Hide
|
C22H28N2O
|
1
|
| 1 |
IC50 > 30000 nM
|
|
|
|
CP0423654
|
N-(2-imidazol-1-ylphenyl)-2-phenylbutanamide
Show/Hide
|
C19H19N3O
|
1
|
| 1 |
IC50 > 30000 nM
|
|
|
|
CP0423655
|
N-[2-[ethyl(methyl)amino]phenyl]-2-phenylbutanamide
Show/Hide
|
C19H24N2O
|
1
|
| 1 |
IC50 > 30000 nM
|
|
|
|
CP0423656
|
2-phenyl-N-(3-pyrrolidin-1-ylphenyl)butanamide
Show/Hide
|
C20H24N2O
|
1
|
| 1 |
IC50 > 30000 nM
|
|
|
|
CP0462951
|
N-methyl-2-phenyl-N-(2-pyrrolidin-1-ylphenyl)butanamide
Show/Hide
|
C21H26N2O
|
1
|
| 1 |
IC50 > 30000 nM
|
|
|
|
CP0462952
|
N-(2-pyrrolidin-1-ylphenyl)-3,4-dihydro-2H-chromene-4-carboxamide
Show/Hide
|
C20H22N2O2
|
1
|
| 1 |
IC50 > 30000 nM
|
|
|
|
CP0462953
|
1-phenyl-N-(2-pyrrolidin-1-ylphenyl)cyclopropane-1-carboxamide
Show/Hide
|
C20H22N2O
|
1
|
| 1 |
IC50 > 30000 nM
|
|
|
|
CP0527344
|
2-methyl-2-phenyl-N-(2-pyrrolidin-1-ylphenyl)propanamide
Show/Hide
|
C20H24N2O
|
1
|
| 1 |
IC50 > 30000 nM
|
|
|
|
CP0940706
|
N-(2-(pyrrolidin-1-yl-2,5-dione)phenyl)-2-phenylbutanamide
Show/Hide
|
C20H20N2O3
|
1
|
| 1 |
IC50 > 30000 nM
|
|
|
