General Information of the Protein
Protein ID
PT00806
Protein Name
Glucagon receptor
Gene Name
GCGR
Sequence
MALAPPQPSCLSQGLRIGGEDGKGRGRRWIPGGCSSFRRRLCHQAAWWLCQPAPRGGLRAVRAAGRRHRPWETQPAGRQDPSPVTGSEGLLLASSPSGSHFINRPGGSGGGLREAGQPAHHSRAQPGLLADGGPPTGPAALTEVRRGVRVPTRTLCPSCVAPARCGGRLLRGMPPARPRCPHLLLLLLACQPQASSAQVMDFLFEKWKLYGDQCLYNLSLLPPPTELVCNRTFDKYSCWPDTPPNTTANISCPWYLPWHHKVQHRLVFKKCGPDGQWVRGPRGQSWRNASQCQLDGQEIEVQKEVAKMYSSFQVMYTVGYSLSLGALLLALVVLLGLSKLRCTRNYIHANLFASFVLKAGSVLVIDALLKTRYSQKIGDDLSVSVWLSNGAVAGCRVAAVFMQYGVVANYCWLLVEGVYLHSLLGRATFPERSFFPLYLAVGWGAPVLFVVPWAVVKCLFENIQCWTSNDNMGFWWILRLPVFLAILINFFIFIRVLLILMAKLRARQMRYSDYKFRLAKSTLTLIPLLGVHEVVFAFVTDEHAQGTLRSAKLFFDLFLSSFQGLLVAVLYCFLNKEVQSELLRRWQRWRMGKRLREERPPSRHPDPGRPAGGAPSKKLLLSRGGDGAARDPSADTGLVGIPPGVAASPFESPQEPPGAPVGAGLRC
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Organism
Canis lupus familiaris, Dog, Canis familiaris
Protein Classification
Unclassified protein
Uniprot ID
E2R517
Subcellular Location
Cell membrane
Multi-pass membrane protein
Membrane
Multi-pass membrane protein
Map of Molecular Bioactivity Related to the Protein
Map of Molecular Bioactivity Related to the Protein

Protein
Cell Line
Compound

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Protein
Cell Line ID: CL000011 , CHO
Compound ID Compound Name Compound Formula
CP0120350
3-[[4-[(1S)-1-[3-(3,5-dichlorophenyl)-5-(6-methoxynaphthalen-2-yl)pyrazol-1-yl]ethyl]benzoyl]amino]propanoic acid
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C32H27Cl2N3O4
 1
1
IC50 = 104.5 nM
   TI
   LI
   LO
   TS