| Compound ID |
Compound Name |
Compound Formula |
|
CP0049684
|
5-(4-Fluoro-phenyl)-6-(4-methanesulfonyl-phenyl)-spiro[2.4]hept-5-ene
Show/Hide
|
C20H19FO2S
|
1
|
| 1 |
IC50 = 1.1 nM
|
|
|
|
CP0470554
|
1-Methanesulfonyl-4-(3-methylene-2-phenyl-cyclobut-1-enyl)-benzene
Show/Hide
|
C18H16O2S
|
1
|
| 1 |
IC50 = 1.2 nM
|
|
|
|
CP0061060
|
5-Bromo-2-(4-fluoro-phenyl)-3-(4-methanesulfonyl-phenyl)-thiophene
Show/Hide
|
C17H12BrFO2S2
|
3
|
| 1 |
IC50 = 2 nM
|
|
|
| 2 |
IC50 = 2.1 nM
|
|
|
| 3 |
IC50 < 200 nM
|
|
|
|
CP0011191
|
4-[5-(4-methylphenyl)-3-(trifluoromethyl)-1H-pyrazol-1-yl]benzene-1-sulfonamide
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|
C17H14F3N3O2S
|
2
|
| 1 |
IC50 = 2 nM
|
|
|
| 2 |
IC50 = 36 nM
|
|
|
|
CP0460409
|
1-(4,4-Dimethyl-3-methylene-2-phenyl-cyclobut-1-enyl)-4-methanesulfonyl-benzene
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|
C20H20O2S
|
1
|
| 1 |
IC50 = 2.2 nM
|
|
|
|
CP0475726
|
3-(4-Methanesulfonyl-phenyl)-4,4-dimethyl-2-phenyl-cyclobut-2-enone
Show/Hide
|
C19H18O3S
|
1
|
| 1 |
IC50 = 2.8 nM
|
|
|
|
CP0401298
|
5-(4-Methanesulfonyl-phenyl)-6-phenyl-2-trifluoromethyl-thiazolo[3,2-b][1,2,4]triazole
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|
C18H12F3N3O2S2
|
1
|
| 1 |
IC50 = 3 nM
|
|
|
|
CP0449755
|
5-(4-Methanesulfonyl-phenyl)-6-m-tolyl-2-trifluoromethyl-thiazolo[3,2-b][1,2,4]triazole
Show/Hide
|
C19H14F3N3O2S2
|
1
|
| 1 |
IC50 = 3 nM
|
|
|
|
CP0374182
|
2-Benzyl-4-cyclopropylmethoxy-5-(4-methanesulfonyl-phenyl)-2H-pyridazin-3-one
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|
C22H22N2O4S
|
1
|
| 1 |
IC50 = 3 nM
|
|
|
|
CP0377648
|
2-(4-Fluoro-phenyl)-3-(4-methanesulfonyl-phenyl)-4,4-dimethyl-cyclobut-2-enone
Show/Hide
|
C19H17FO3S
|
1
|
| 1 |
IC50 = 5 nM
|
|
|
|
CP0430344
|
5-(4-Methanesulfonyl-phenyl)-6-phenyl-2-vinyl-thiazolo[3,2-b][1,2,4]triazole
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|
C19H15N3O2S2
|
1
|
| 1 |
IC50 = 6 nM
|
|
|
|
CP0442097
|
3-(4-Methanesulfonyl-phenyl)-2-(3,4,5-trichloro-phenyl)-cyclopent-2-enone
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|
C18H13Cl3O3S
|
1
|
| 1 |
IC50 = 6 nM
|
|
|
|
CP0538370
|
3-(4-Methanesulfonyl-phenyl)-2-phenylethynyl-cyclopent-2-enone
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|
C20H16O3S
|
1
|
| 1 |
IC50 = 6 nM
|
|
|
|
CP0529605
|
2-(3-Chloro-4-fluoro-phenyl)-3-(4-methanesulfonyl-phenyl)-cyclopent-2-enone
Show/Hide
|
C18H14ClFO3S
|
1
|
| 1 |
IC50 = 9 nM
|
|
|
|
CP0158195
|
3-(4-Fluoro-phenyl)-4-(4-methanesulfonyl-phenyl)-5H-furan-2-one
Show/Hide
|
C17H13FO4S
|
1
|
| 1 |
IC50 = 10 nM
|
|
|
|
CP0412211
|
3-(3,4-Difluoro-phenoxy)-4-(4-methanesulfonyl-phenyl)-5,5-dimethyl-5H-furan-2-one
Show/Hide
|
C19H16F2O5S
|
1
|
| 1 |
IC50 = 10 nM
|
|
|
|
CP0494798
|
3-(4-Chloro-phenoxy)-4-(4-methanesulfonyl-phenyl)-5,5-dimethyl-5H-furan-2-one
Show/Hide
|
C19H17ClO5S
|
1
|
| 1 |
IC50 = 10 nM
|
|
|
|
CP0428132
|
2-Isopropyl-5-(4-methanesulfonyl-phenyl)-6-phenyl-thiazolo[3,2-b][1,2,4]triazole
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|
C20H19N3O2S2
|
1
|
| 1 |
IC50 = 11 nM
|
|
|
|
CP0453531
|
3-(4-Methanesulfonyl-phenyl)-2-phenoxy-cyclopent-2-enone
Show/Hide
|
C18H16O4S
|
1
|
| 1 |
IC50 = 11 nM
|
|
|
|
CP0506598
|
3-(4-Methanesulfonyl-phenyl)-2-phenyl-cyclopent-2-enone
Show/Hide
|
C18H16O3S
|
1
|
| 1 |
IC50 = 11 nM
|
|
|
|
CP0395145
|
3-(4-Methanesulfonyl-phenyl)-2-phenyl-spiro[3.4]oct-2-en-1-one
Show/Hide
|
C21H20O3S
|
1
|
| 1 |
IC50 = 12 nM
|
|
|
|
CP0492730
|
6-(3,4-Difluoro-phenyl)-5-(4-methanesulfonyl-phenyl)-imidazo[2,1-b]thiazole
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|
C18H12F2N2O2S2
|
1
|
| 1 |
IC50 = 12 nM
|
|
|
|
CP0527628
|
5-(4-Methanesulfonyl-phenyl)-2-methyl-6-phenyl-imidazo[2,1-b]thiazole
Show/Hide
|
C19H16N2O2S2
|
1
|
| 1 |
IC50 = 12 nM
|
|
|
|
CP0498180
|
6-(3-Fluoro-phenyl)-5-(4-methanesulfonyl-phenyl)-2-trifluoromethyl-thiazolo[3,2-b][1,2,4]triazole
Show/Hide
|
C18H11F4N3O2S2
|
1
|
| 1 |
IC50 = 13 nM
|
|
|
|
CP0222382
|
N-[6-[(4-ethyl-1,3-thiazol-2-yl)sulfanyl]-1-oxo-3H-2-benzofuran-5-yl]methanesulfonamide
Show/Hide
|
C14H14N2O4S3
|
1
|
| 1 |
IC50 = 13 nM
|
|
|
|
CP0502348
|
6-(4-Fluoro-phenyl)-5-(4-methanesulfonyl-phenyl)-imidazo[2,1-b]thiazole
Show/Hide
|
C18H13FN2O2S2
|
1
|
| 1 |
IC50 = 14 nM
|
|
|
|
CP0464094
|
2-(3-Fluoro-phenyl)-3-(4-methanesulfonyl-phenyl)-cyclopent-2-enone
Show/Hide
|
C18H15FO3S
|
1
|
| 1 |
IC50 = 14 nM
|
|
|
|
CP0497560
|
2-(3,4-Difluoro-phenyl)-3-(4-methanesulfonyl-phenyl)-cyclopent-2-enone
Show/Hide
|
C18H14F2O3S
|
1
|
| 1 |
IC50 = 14 nM
|
|
|
|
CP0536032
|
2-(3,5-Dichloro-phenyl)-3-(4-methanesulfonyl-phenyl)-cyclopent-2-enone
Show/Hide
|
C18H14Cl2O3S
|
1
|
| 1 |
IC50 = 14 nM
|
|
|
|
CP0551260
|
2-(3H-1lambda*4*-Benzo[b]thiophen-2-yl)-3-(4-methanesulfonyl-phenyl)-cyclopent-2-enone
Show/Hide
|
C20H16O3S2
|
1
|
| 1 |
IC50 = 14 nM
|
|
|
|
CP0449758
|
2-Ethyl-5-(4-methanesulfonyl-phenyl)-6-phenyl-thiazolo[3,2-b][1,2,4]triazole
Show/Hide
|
C19H17N3O2S2
|
1
|
| 1 |
IC50 = 15 nM
|
|
|
|
CP0394274
|
2-(4-Chloro-3-fluoro-phenyl)-3-(4-methanesulfonyl-phenyl)-cyclopent-2-enone
Show/Hide
|
C18H14ClFO3S
|
1
|
| 1 |
IC50 = 15 nM
|
|
|
|
CP0559515
|
2-(3,5-Difluoro-phenyl)-3-(4-methanesulfonyl-phenyl)-cyclopent-2-enone
Show/Hide
|
C18H14F2O3S
|
1
|
| 1 |
IC50 = 15 nM
|
|
|
|
CP0383382
|
2-Chloro-6-(4-chloro-phenyl)-5-(4-methanesulfonyl-phenyl)-imidazo[2,1-b]thiazole
Show/Hide
|
C18H12Cl2N2O2S2
|
1
|
| 1 |
IC50 = 16 nM
|
|
|
|
CP0402569
|
5-(4-Methanesulfonyl-phenyl)-6-phenyl-3,5-dihydro-1lambda*4*-imidazo[2,1-b]thiazole
Show/Hide
|
C18H14N2O2S2
|
1
|
| 1 |
IC50 = 16 nM
|
|
|
|
CP0451741
|
5-Chloro-6'-cyclopropyl-3-(4-methanesulfonyl-phenyl)-[2,3']bipyridinyl
Show/Hide
|
C20H17ClN2O2S
|
1
|
| 1 |
IC50 = 16 nM
|
|
|
|
CP0514173
|
2-(3,5-Difluoro-phenoxy)-3-(4-methanesulfonyl-phenyl)-cyclopent-2-enone
Show/Hide
|
C18H14F2O4S
|
1
|
| 1 |
IC50 = 17 nM
|
|
|
|
CP0465116
|
2-(4-Fluoro-phenyl)-3-(4-methanesulfonyl-phenyl)-cyclopent-2-enone
Show/Hide
|
C18H15FO3S
|
1
|
| 1 |
IC50 = 19 nM
|
|
|
|
CP0419384
|
5-(4-Methanesulfonyl-phenyl)-2-methyl-6-phenyl-thiazolo[3,2-b][1,2,4]triazole
Show/Hide
|
C18H15N3O2S2
|
1
|
| 1 |
IC50 = 20 nM
|
|
|
|
CP0037144
|
4-(4-methanesulfonylphenyl)-3-phenyl-2,5-dihydrofuran-2-one
Show/Hide
|
C17H14O4S
|
1
|
| 1 |
IC50 = 20 nM
|
|
|
|
CP0063951
|
3-(3-Fluoro-phenyl)-4-(4-methanesulfonyl-phenyl)-5H-furan-2-one
Show/Hide
|
C17H13FO4S
|
1
|
| 1 |
IC50 = 20 nM
|
|
|
|
CP0456602
|
3-(5-Chloro-pyridin-2-yloxy)-4-(4-methanesulfonyl-phenyl)-5,5-dimethyl-5H-furan-2-one
Show/Hide
|
C18H16ClNO5S
|
1
|
| 1 |
IC50 = 20 nM
|
|
|
|
CP0495468
|
3-(Benzo[b]thiophen-5-yloxy)-4-(4-methanesulfonyl-phenyl)-5,5-dimethyl-5H-furan-2-one
Show/Hide
|
C21H18O5S2
|
1
|
| 1 |
IC50 = 20 nM
|
|
|
|
CP0514059
|
3-(5-Bromo-pyridin-2-yloxy)-4-(4-methanesulfonyl-phenyl)-5,5-dimethyl-5H-furan-2-one
Show/Hide
|
C18H16BrNO5S
|
1
|
| 1 |
IC50 = 20 nM
|
|
|
|
CP0394392
|
3-(3-Fluoro-phenoxy)-4-(4-methanesulfonyl-phenyl)-5,5-dimethyl-5H-furan-2-one
Show/Hide
|
C19H17FO5S
|
1
|
| 1 |
IC50 = 20 nM
|
|
|
|
CP0405345
|
3-(2,4-Difluoro-phenoxy)-4-(4-methanesulfonyl-phenyl)-5,5-dimethyl-5H-furan-2-one
Show/Hide
|
C19H16F2O5S
|
1
|
| 1 |
IC50 = 20 nM
|
|
|
|
CP0442056
|
4-(4-Methanesulfonyl-phenyl)-5,5-dimethyl-3-p-tolyloxy-5H-furan-2-one
Show/Hide
|
C20H20O5S
|
1
|
| 1 |
IC50 = 20 nM
|
|
|
|
CP0465037
|
4-(4-Methanesulfonyl-phenyl)-5,5-dimethyl-3-phenoxy-5H-furan-2-one
Show/Hide
|
C19H18O5S
|
1
|
| 1 |
IC50 = 20 nM
|
|
|
|
CP0492368
|
4-(4-Methanesulfonyl-phenyl)-5,5-dimethyl-3-o-tolyloxy-5H-furan-2-one
Show/Hide
|
C20H20O5S
|
1
|
| 1 |
IC50 = 20 nM
|
|
|
|
CP0542544
|
4-(4-Methanesulfonyl-phenyl)-5,5-dimethyl-3-m-tolyloxy-5H-furan-2-one
Show/Hide
|
C20H20O5S
|
1
|
| 1 |
IC50 = 20 nM
|
|
|
|
CP0471121
|
2-Benzyl-4-isopropoxy-5-(4-methanesulfonyl-phenyl)-2H-pyridazin-3-one
Show/Hide
|
C21H22N2O4S
|
1
|
| 1 |
IC50 = 20 nM
|
|
|
|
CP0503643
|
2-Benzyl-4-(4-fluoro-phenoxy)-5-(4-methanesulfonyl-phenyl)-2H-pyridazin-3-one
Show/Hide
|
C24H19FN2O4S
|
1
|
| 1 |
IC50 = 20 nM
|
|
|
|
CP0507346
|
2-Benzyl-5-(4-methanesulfonyl-phenyl)-4-p-tolyl-2H-pyridazin-3-one
Show/Hide
|
C25H22N2O3S
|
1
|
| 1 |
IC50 = 20 nM
|
|
|
|
CP0449757
|
6-(3-Fluoro-phenyl)-5-(4-methanesulfonyl-phenyl)-thiazolo[3,2-b][1,2,4]triazole
Show/Hide
|
C17H12FN3O2S2
|
1
|
| 1 |
IC50 = 22 nM
|
|
|
|
CP0333574
|
4-(5-Chloro-6'-methyl-[2,3']bipyridinyl-3-yl)-benzenesulfonamide
Show/Hide
|
C17H14ClN3O2S
|
1
|
| 1 |
IC50 = 23 nM
|
|
|
|
CP0010057
|
2-{1-[(4-chlorophenyl)carbonyl]-5-methoxy-2-methyl-1H-indol-3-yl}acetic acid
Show/Hide
|
C19H16ClNO4
|
4
|
| 1 |
IC50 = 26 nM
|
|
|
| 2 |
IC50 = 30 nM
|
|
|
| 3 |
IC50 = 49 nM
|
|
|
| 4 |
IC50 < 200 nM
|
|
|
|
CP0216451
|
N-[1-oxo-6-(1,3-thiazol-2-ylsulfanyl)-3H-2-benzofuran-5-yl]methanesulfonamide
Show/Hide
|
C12H10N2O4S3
|
1
|
| 1 |
IC50 = 27 nM
|
|
|
|
CP0048346
|
N-[6-(2,4-difluorophenyl)sulfanyl-1-oxo-2,3-dihydroinden-5-yl]methanesulfonamide
Show/Hide
|
C16H13F2NO3S2
|
1
|
| 1 |
IC50 = 29 nM
|
|
|
|
CP0092588
|
3-(3,4-Difluoro-phenyl)-4-(4-methanesulfonyl-phenyl)-5H-furan-2-one
Show/Hide
|
C17H12F2O4S
|
1
|
| 1 |
IC50 = 30 nM
|
|
|
|
CP0514065
|
3-(5-Cyclopropyl-pyridin-2-yloxy)-4-(4-methanesulfonyl-phenyl)-5,5-dimethyl-5H-furan-2-one
Show/Hide
|
C21H21NO5S
|
1
|
| 1 |
IC50 = 30 nM
|
|
|
|
CP0535080
|
3-(1H-Indol-5-yloxy)-4-(4-methanesulfonyl-phenyl)-5,5-dimethyl-5H-furan-2-one
Show/Hide
|
C21H19NO5S
|
1
|
| 1 |
IC50 = 30 nM
|
|
|
|
CP0332572
|
N-[6-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]-1-oxo-2,3-dihydroinden-5-yl]methanesulfonamide
Show/Hide
|
C14H14N2O3S3
|
1
|
| 1 |
IC50 = 30 nM
|
|
|
|
CP0461479
|
2-Benzyl-5-(4-methanesulfonyl-phenyl)-4-phenyl-2H-pyridazin-3-one
Show/Hide
|
C24H20N2O3S
|
1
|
| 1 |
IC50 = 30 nM
|
|
|
|
CP0476692
|
2-(2,2-Dimethyl-cyclopropylmethyl)-4-(4-fluoro-phenyl)-5-(4-methanesulfonyl-phenyl)-2H-pyridazin-3-one
Show/Hide
|
C23H23FN2O3S
|
1
|
| 1 |
IC50 = 30 nM
|
|
|
|
CP0459216
|
6-(4-Methanesulfonyl-phenyl)-5-phenyl-thiazolo[3,2-b][1,2,4]triazole
Show/Hide
|
C17H13N3O2S2
|
1
|
| 1 |
IC50 = 32 nM
|
|
|
|
CP0289794
|
5-Chloro-3-(4-methanesulfonyl-phenyl)-[2,3']bipyridinyl
Show/Hide
|
C17H13ClN2O2S
|
1
|
| 1 |
IC50 = 34 nM
|
|
|
|
CP0502197
|
6-(4-Fluoro-phenyl)-5-(4-methanesulfonyl-phenyl)-thiazolo[3,2-b][1,2,4]triazole
Show/Hide
|
C17H12FN3O2S2
|
1
|
| 1 |
IC50 = 36 nM
|
|
|
|
CP0497673
|
3-(3,5-Dichloro-pyridin-2-yloxy)-4-(4-methanesulfonyl-phenyl)-5,5-dimethyl-5H-furan-2-one
Show/Hide
|
C18H15Cl2NO5S
|
1
|
| 1 |
IC50 = 40 nM
|
|
|
|
CP0502451
|
3-(5-Fluoro-pyridin-2-yloxy)-4-(4-methanesulfonyl-phenyl)-5,5-dimethyl-5H-furan-2-one
Show/Hide
|
C18H16FNO5S
|
1
|
| 1 |
IC50 = 40 nM
|
|
|
|
CP0503156
|
3-(3-Fluoro-phenyl)-4-(4-methanesulfonyl-phenyl)-5,5-dimethyl-5H-furan-2-one
Show/Hide
|
C19H17FO4S
|
1
|
| 1 |
IC50 = 40 nM
|
|
|
|
CP0562301
|
3-(3,5-Difluoro-phenoxy)-4-(4-methanesulfonyl-phenyl)-5,5-dimethyl-5H-furan-2-one
Show/Hide
|
C19H16F2O5S
|
1
|
| 1 |
IC50 = 40 nM
|
|
|
|
CP0541391
|
2-Cyclohexylmethyl-4-(4-fluoro-phenyl)-5-(4-methanesulfonyl-phenyl)-2H-pyridazin-3-one
Show/Hide
|
C24H25FN2O3S
|
1
|
| 1 |
IC50 = 40 nM
|
|
|
|
CP0036639
|
N-[6-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]-1-oxo-3H-2-benzofuran-5-yl]methanesulfonamide
Show/Hide
|
C13H12N2O4S3
|
1
|
| 1 |
IC50 = 43 nM
|
|
|
|
CP0096361
|
3-((3-fluoro-5-(1-methoxycyclohexyl)phenoxy)methyl)-1-(4-(methylsulfonyl)phenyl)-5-phenyl-1H-pyrazole
Show/Hide
|
C29H29FN2O5S
|
1
|
| 1 |
IC50 = 45 nM
|
|
|
|
CP0437782
|
6-(3,4-Difluoro-phenyl)-5-(4-methanesulfonyl-phenyl)-thiazolo[3,2-b][1,2,4]triazole
Show/Hide
|
C17H11F2N3O2S2
|
1
|
| 1 |
IC50 = 48 nM
|
|
|
|
CP0238803
|
N-[6-[(4-ethyl-1,3-thiazol-2-yl)sulfanyl]-1-oxo-2,3-dihydroinden-5-yl]methanesulfonamide
Show/Hide
|
C15H16N2O3S3
|
1
|
| 1 |
IC50 = 49 nM
|
|
|
|
CP0151492
|
5-Chloro-6'-ethyl-3-(4-methanesulfonyl-phenyl)-[2,3']bipyridinyl
Show/Hide
|
C19H17ClN2O2S
|
1
|
| 1 |
IC50 = 50 nM
|
|
|
|
CP0455359
|
4-(4-Fluoro-phenyl)-5-(4-methanesulfonyl-phenyl)-2-thiophen-2-ylmethyl-2H-pyridazin-3-one
Show/Hide
|
C22H17FN2O3S2
|
1
|
| 1 |
IC50 = 50 nM
|
|
|
|
CP0457141
|
4-(4-Fluoro-phenyl)-5-(4-methanesulfonyl-phenyl)-2-((1R,2S)-2-methyl-cyclopropylmethyl)-2H-pyridazin-3-one
Show/Hide
|
C22H21FN2O3S
|
1
|
| 1 |
IC50 = 50 nM
|
|
|
|
CP0479847
|
2-((2R,3R)-2,3-Dimethyl-cyclopropylmethyl)-4-(4-fluoro-phenyl)-5-(4-methanesulfonyl-phenyl)-2H-pyridazin-3-one
Show/Hide
|
C23H23FN2O3S
|
1
|
| 1 |
IC50 = 50 nM
|
|
|
|
CP0150082
|
3-(4-Methanesulfonyl-phenyl)-2-phenyl-pyridine
Show/Hide
|
C18H15NO2S
|
1
|
| 1 |
IC50 = 60 nM
|
|
|
|
CP0470044
|
4-(4-Fluoro-phenyl)-5-(4-methanesulfonyl-phenyl)-2-((1R,2R)-2-methyl-cyclopropylmethyl)-2H-pyridazin-3-one
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C22H21FN2O3S
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1
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| 1 |
IC50 = 60 nM
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CP0534429
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4-(4-Fluoro-phenyl)-5-(4-methanesulfonyl-phenyl)-2-((1S,2S)-2-methyl-cyclopropylmethyl)-2H-pyridazin-3-one
Show/Hide
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C22H21FN2O3S
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1
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| 1 |
IC50 = 60 nM
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CP0879971
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3-(4-Methanesulfonyl-phenyl)-4,4-dimethyl-2-phenyl-cyclobut-2-enone oxime
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C19H19NO3S
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1
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| 1 |
IC50 = 61 nM
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CP0371437
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5-Chloro-3-(4-methanesulfonyl-phenyl)-[2,2']bipyridinyl
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C17H13ClN2O2S
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1
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| 1 |
IC50 = 68 nM
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CP0304463
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3-(4-Fluoro-phenyl)-4-(4-methanesulfonyl-phenyl)-5-methoxy-5-methyl-5H-furan-2-one
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C19H17FO5S
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1
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| 1 |
IC50 = 69 nM
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CP0379346
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4-(4-Methanesulfonyl-phenyl)-5,5-dimethyl-3-phenylsulfanyl-5H-furan-2-one
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C19H18O4S2
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1
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| 1 |
IC50 = 70 nM
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CP0455358
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2-Cyclopropylmethyl-5-(4-methanesulfonyl-phenyl)-4-phenyl-2H-pyridazin-3-one
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C21H20N2O3S
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1
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| 1 |
IC50 = 70 nM
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CP0427268
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3-(3,4-Dichloro-phenyl)-5-hydroxy-4-(4-methanesulfonyl-phenyl)-5-methyl-5H-furan-2-one
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C18H14Cl2O5S
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1
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| 1 |
IC50 = 70 nM
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CP0505496
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6-(3,5-Difluoro-phenyl)-5-(4-methanesulfonyl-phenyl)-thiazolo[3,2-b][1,2,4]triazole
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C17H11F2N3O2S2
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1
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| 1 |
IC50 = 80 nM
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CP0393839
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5-(4-Methanesulfonyl-phenyl)-2,4-diphenyl-2H-pyridazin-3-one
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C23H18N2O3S
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1
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| 1 |
IC50 = 80 nM
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CP0132427
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5-Chloro-3-(4-methanesulfonyl-phenyl)-6''-methyl-[2,3'']bipyridinyl
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C18H15ClN2O2S
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1
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| 1 |
IC50 = 81 nM
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CP0041096
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5-Chloro-3-(4-methanesulfonyl-phenyl)-5'-methyl-[2,3']bipyridinyl
Show/Hide
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C18H15ClN2O2S
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1
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| 1 |
IC50 = 87 nM
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CP0529797
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2-(5-Chloro-pyridin-3-yl)-3-(4-methanesulfonyl-phenyl)-cyclopent-2-enone
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C17H14ClNO3S
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1
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| 1 |
IC50 = 87 nM
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CP0288956
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3-(4-Methanesulfonyl-phenyl)-5-trifluoromethyl-[2,3']bipyridinyl
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C18H13F3N2O2S
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1
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| 1 |
IC50 = 90 nM
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CP0428451
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3-(3-Chloro-pyridin-2-yloxy)-4-(4-methanesulfonyl-phenyl)-5,5-dimethyl-5H-furan-2-one
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C18H16ClNO5S
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1
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| 1 |
IC50 = 90 nM
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CP0383216
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2-(4-Methanesulfonyl-phenyl)-4,4-dimethyl-3-phenyl-cyclobut-2-enone
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C19H18O3S
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1
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| 1 |
IC50 = 96 nM
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CP0511113
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4-(4-Fluoro-phenyl)-5-(4-methanesulfonyl-phenyl)-2-(3-methyl-but-2-enyl)-2H-pyridazin-3-one
Show/Hide
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C22H21FN2O3S
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1
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| 1 |
IC50 = 100 nM
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CP0420193
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1-(4-aminosulfonylphenyl)-3-[3-fluoro-5-(4-methoxytetrahydropyran-4-yl)phenoxymethyl]-5-phenyl-1H-pyrazole
Show/Hide
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C28H28FN3O5S
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1
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| 1 |
IC50 = 100 nM
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CP0193706
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5-Chloro-3-(4-methanesulfonyl-phenyl)-[2,4']bipyridinyl
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C17H13ClN2O2S
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1
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| 1 |
IC50 = 101 nM
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CP0489046
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3-(4-Methanesulfonyl-phenyl)-2-phenyl-cyclobut-2-enone
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C17H14O3S
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1
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| 1 |
IC50 = 110 nM
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CP0403655
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2-Cyclopropyl-4-(4-fluoro-phenyl)-5-(4-methanesulfonyl-phenyl)-2H-pyridazin-3-one
Show/Hide
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C20H17FN2O3S
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1
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| 1 |
IC50 = 110 nM
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CP0373355
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5-Hydroxy-4-(4-methanesulfonyl-phenyl)-5-methyl-3-thiophen-3-yl-5H-furan-2-one
Show/Hide
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C16H14O5S2
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1
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| 1 |
IC50 = 110 nM
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CP0406476
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3-(4-Chloro-phenyl)-5-hydroxy-4-(4-methanesulfonyl-phenyl)-5-methyl-5H-furan-2-one
Show/Hide
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C18H15ClO5S
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1
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| 1 |
IC50 = 110 nM
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CP0442627
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3-(3-Chloro-4-fluoro-phenyl)-5-hydroxy-4-(4-methanesulfonyl-phenyl)-5-methyl-5H-furan-2-one
Show/Hide
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C18H14ClFO5S
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1
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| 1 |
IC50 = 110 nM
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CP0471950
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4-(4-Methanesulfonyl-phenyl)-5,5-dimethyl-3-(pyridin-2-yloxy)-5H-furan-2-one
Show/Hide
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C18H17NO5S
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1
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| 1 |
IC50 = 120 nM
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CP0196257
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N-[6-(3,5-dichloropyridin-2-yl)sulfanyl-1-oxo-2,3-dihydroinden-5-yl]methanesulfonamide
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C15H12Cl2N2O3S2
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1
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| 1 |
IC50 = 120 nM
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CP0409180
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6-(4-Methanesulfonyl-phenyl)-2-methyl-5-phenyl-imidazo[2,1-b]thiazole
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C19H16N2O2S2
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1
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| 1 |
IC50 = 140 nM
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CP0347870
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N-[6-[(4-ethenyl-1,3-thiazol-2-yl)sulfanyl]-1-oxo-3H-2-benzofuran-5-yl]methanesulfonamide
Show/Hide
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C14H12N2O4S3
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1
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| 1 |
IC50 = 140 nM
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CP0501248
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3-(4-Bromo-phenyl)-5-hydroxy-4-(4-methanesulfonyl-phenyl)-5-methyl-5H-furan-2-one
Show/Hide
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C18H15BrO5S
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1
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| 1 |
IC50 = 140 nM
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CP0449756
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6-(3-Fluoro-phenyl)-5-(4-methanesulfonyl-phenyl)-2-methyl-thiazolo[3,2-b][1,2,4]triazole
Show/Hide
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C18H14FN3O2S2
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1
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| 1 |
IC50 = 150 nM
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CP0511203
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4-(4-Methanesulfonyl-phenyl)-5,5-dimethyl-3-(5-methyl-pyridin-2-yloxy)-5H-furan-2-one
Show/Hide
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C19H19NO5S
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1
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| 1 |
IC50 = 150 nM
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CP0425983
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3-(4-Methanesulfonyl-phenyl)-2-(4-methoxy-pyridin-3-yl)-cyclopent-2-enone
Show/Hide
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C18H17NO4S
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1
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| 1 |
IC50 = 150 nM
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CP0536095
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2-(3,3-Dimethyl-but-1-ynyl)-3-(4-methanesulfonyl-phenyl)-cyclopent-2-enone
Show/Hide
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C18H20O3S
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1
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| 1 |
IC50 = 150 nM
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CP0454401
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5-Hydroxy-4-(4-methanesulfonyl-phenyl)-5-methyl-3-phenyl-5H-furan-2-one
Show/Hide
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C18H16O5S
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1
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| 1 |
IC50 = 160 nM
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CP0562353
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3-(4-Methanesulfonyl-phenyl)-2-pyridin-3-yl-cyclopent-2-enone
Show/Hide
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C17H15NO3S
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1
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| 1 |
IC50 = 170 nM
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CP0863041
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2-[(E)-2-(4-Fluoro-phenyl)-vinyl]-3-(4-methanesulfonyl-phenyl)-cyclopent-2-enone
Show/Hide
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C20H17FO3S
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1
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| 1 |
IC50 = 175 nM
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CP0420767
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2-(4-Chloro-pyridin-2-yl)-3-(4-methanesulfonyl-phenyl)-cyclopent-2-enone
Show/Hide
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C17H14ClNO3S
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1
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| 1 |
IC50 = 190 nM
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CP0412214
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3-(4-Fluoro-phenoxy)-4-(4-methanesulfonyl-phenyl)-5,5-dimethyl-5H-furan-2-one
Show/Hide
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C19H17FO5S
|
1
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| 1 |
IC50 = 200 nM
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CP0453302
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2-(2-Cyclopropyl-ethyl)-4-(4-fluoro-phenyl)-5-(4-methanesulfonyl-phenyl)-2H-pyridazin-3-one
Show/Hide
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C22H21FN2O3S
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1
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| 1 |
IC50 = 200 nM
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CP0491700
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2-Cyclopropylmethyl-4-(4-fluoro-phenyl)-5-(4-methanesulfonyl-phenyl)-2H-pyridazin-3-one
Show/Hide
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C21H19FN2O3S
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1
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| 1 |
IC50 = 200 nM
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CP0511114
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2-(1-Cyclopropyl-ethyl)-4-(4-fluoro-phenyl)-5-(4-methanesulfonyl-phenyl)-2H-pyridazin-3-one
Show/Hide
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C22H21FN2O3S
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1
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| 1 |
IC50 = 200 nM
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CP0535708
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4-(4-Fluoro-phenyl)-5-(4-methanesulfonyl-phenyl)-2-(1-methyl-cyclopropylmethyl)-2H-pyridazin-3-one
Show/Hide
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C22H21FN2O3S
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1
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| 1 |
IC50 = 200 nM
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CP0435658
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3-(3,4-Difluoro-phenyl)-5-hydroxy-4-(4-methanesulfonyl-phenyl)-5-methyl-5H-furan-2-one
Show/Hide
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C18H14F2O5S
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1
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| 1 |
IC50 = 200 nM
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CP0098763
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N-[6-(3-chloropyridin-2-yl)sulfanyl-1-oxo-2,3-dihydroinden-5-yl]methanesulfonamide
Show/Hide
|
C15H13ClN2O3S2
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1
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| 1 |
IC50 = 220 nM
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CP0437319
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1-(4-methanesulfonylphenyl)-3-[(3,4,5-trimethoxy)phenoxymethyl]-5-phenyl-1H-pyrazole
Show/Hide
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C26H26N2O6S
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1
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| 1 |
IC50 = 220 nM
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CP0441647
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5-(4-Methanesulfonyl-phenyl)-6-phenyl-thiazolo[2,3-c][1,2,4]triazole
Show/Hide
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C17H13N3O2S2
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1
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| 1 |
IC50 = 230 nM
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CP0398426
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3-(3-Fluoro-phenyl)-5-hydroxy-4-(4-methanesulfonyl-phenyl)-5-methyl-5H-furan-2-one
Show/Hide
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C18H15FO5S
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1
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| 1 |
IC50 = 250 nM
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CP0376342
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5-(4-Methanesulfonyl-phenyl)-6-(3-methoxy-phenyl)-thiazolo[3,2-b][1,2,4]triazole
Show/Hide
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C18H15N3O3S2
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1
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| 1 |
IC50 = 260 nM
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CP0490262
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4-(4-Methanesulfonyl-phenyl)-5,5-dimethyl-3-(pyridin-3-yloxy)-5H-furan-2-one
Show/Hide
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C18H17NO5S
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1
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| 1 |
IC50 = 260 nM
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CP0429115
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2-Benzyl-4-(5-chloro-pyridin-2-yloxy)-5-(4-methanesulfonyl-phenyl)-2H-pyridazin-3-one
Show/Hide
|
C23H18ClN3O4S
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1
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| 1 |
IC50 = 260 nM
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CP0510948
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4-(4-Methanesulfonyl-phenyl)-5,5-dimethyl-3-(pyridin-4-yloxy)-5H-furan-2-one
Show/Hide
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C18H17NO5S
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1
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| 1 |
IC50 = 270 nM
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CP0510663
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2-(5-Bromo-pyridin-3-yl)-3-(4-methanesulfonyl-phenyl)-cyclopent-2-enone
Show/Hide
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C17H14BrNO3S
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1
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| 1 |
IC50 = 300 nM
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CP0505297
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3-Benzyl-4-(4-methanesulfonyl-phenyl)-5,5-dimethyl-5H-furan-2-one
Show/Hide
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C20H20O4S
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1
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| 1 |
IC50 = 300 nM
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CP0384126
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5-(4-Methanesulfonyl-phenyl)-2-methyl-4-phenyl-2H-pyridazin-3-one
Show/Hide
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C18H16N2O3S
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1
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| 1 |
IC50 = 300 nM
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CP0511926
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3-[3-fluoro-5-(4-methoxytetrahydropyran-4-yl)phenoxymethyl]-1-(4-methoxyphenyl)-5-phenyl-1H-pyrazole
Show/Hide
|
C29H29FN2O4
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1
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| 1 |
IC50 = 300 nM
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CP0379192
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5-Hydroxy-4-(4-methanesulfonyl-phenyl)-5-methyl-3-(4-methylsulfanyl-phenyl)-5H-furan-2-one
Show/Hide
|
C19H18O5S2
|
1
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| 1 |
IC50 = 310 nM
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CP0427145
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3-[(3-fluoro-5-methoxy)phenoxymethyl]-1-(4-methanesulfonylphenyl)-5-phenyl-1H-pyrazole
Show/Hide
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C24H21FN2O4S
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1
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| 1 |
IC50 = 310 nM
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CP0244285
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N-[1-oxo-6-(1,3-thiazol-2-ylsulfanyl)-2,3-dihydroinden-5-yl]methanesulfonamide
Show/Hide
|
C13H12N2O3S3
|
1
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| 1 |
IC50 = 320 nM
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CP0504224
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3-(4-Fluoro-phenyl)-4-(4-methanesulfonyl-phenyl)-5-methyl-5-(2,2,2-trifluoro-ethoxy)-5H-furan-2-one
Show/Hide
|
C20H16F4O5S
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1
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| 1 |
IC50 = 320 nM
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CP0524560
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4-(4-Methanesulfonyl-phenyl)-5,5-dimethyl-3-(quinolin-2-yloxy)-5H-furan-2-one
Show/Hide
|
C22H19NO5S
|
1
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| 1 |
IC50 = 330 nM
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CP0288700
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3-(4-Methanesulfonyl-phenyl)-5-methyl-[2,3']bipyridinyl
Show/Hide
|
C18H16N2O2S
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1
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| 1 |
IC50 = 350 nM
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CP0383952
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3-(6-Chloro-pyridin-2-yloxy)-4-(4-methanesulfonyl-phenyl)-5,5-dimethyl-5H-furan-2-one
Show/Hide
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C18H16ClNO5S
|
1
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| 1 |
IC50 = 350 nM
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CP0554626
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5-(4-Methanesulfonyl-phenyl)-2-(2-methyl-benzyl)-4-phenyl-2H-pyridazin-3-one
Show/Hide
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C25H22N2O3S
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1
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| 1 |
IC50 = 350 nM
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CP0454876
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2-Benzyl-5-(4-methanesulfonyl-phenyl)-4-phenylsulfanyl-2H-pyridazin-3-one
Show/Hide
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C24H20N2O3S2
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1
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| 1 |
IC50 = 370 nM
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CP0379416
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3-(4-Fluoro-phenyl)-5-hydroxy-4-(4-methanesulfonyl-phenyl)-5-methyl-5H-furan-2-one
Show/Hide
|
C18H15FO5S
|
1
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| 1 |
IC50 = 380 nM
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CP0379193
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5-Hydroxy-3-(4-isopropyl-phenyl)-4-(4-methanesulfonyl-phenyl)-5-methyl-5H-furan-2-one
Show/Hide
|
C21H22O5S
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1
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| 1 |
IC50 = 410 nM
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CP0529372
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3-[3-fluoro-5-(4-methoxytetrahydropyran-4-yl)phenoxymethyl]-1-(3,4-dimethylphenyl)-5-phenyl-1H-pyrazole
Show/Hide
|
C30H31FN2O3
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1
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| 1 |
IC50 = 410 nM
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CP0404461
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5-(4-Methylsulfanyl-phenyl)-6-phenyl-imidazo[2,1-b]thiazole
Show/Hide
|
C18H14N2S2
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1
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| 1 |
IC50 = 420 nM
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CP0543976
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3-(4-Methanesulfonyl-phenyl)-2-(4-methyl-pyridin-3-yl)-cyclopent-2-enone
Show/Hide
|
C18H17NO3S
|
1
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| 1 |
IC50 = 440 nM
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CP0497173
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6-(4-Methanesulfonyl-phenyl)-5-phenyl-thiazolo[2,3-c][1,2,4]triazole
Show/Hide
|
C17H13N3O2S2
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1
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| 1 |
IC50 = 450 nM
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CP0409045
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5-Hydroxy-4-(4-methanesulfonyl-phenyl)-5-methyl-3-naphthalen-2-yl-5H-furan-2-one
Show/Hide
|
C22H18O5S
|
1
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| 1 |
IC50 = 450 nM
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CP0427141
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1-(4-methanesulfonylphenyl)-3-[(3,4-methylenedioxy)-phenoxymethyl]-5-phenyl-1H-pyrazole
Show/Hide
|
C24H20N2O5S
|
1
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| 1 |
IC50 = 450 nM
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CP0038355
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N-(1-oxo-6-pyridin-2-ylsulfanyl-2,3-dihydroinden-5-yl)methanesulfonamide
Show/Hide
|
C15H14N2O3S2
|
1
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| 1 |
IC50 = 500 nM
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CP0863089
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4-(4-Methanesulfonyl-phenyl)-5,5-dimethyl-3-phenylamino-5H-furan-2-one
Show/Hide
|
C19H19NO4S
|
1
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| 1 |
IC50 = 500 nM
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CP0449006
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5-(4-Methanesulfonyl-phenyl)-4-phenyl-2-(2,2,2-trifluoro-ethyl)-2H-pyridazin-3-one
Show/Hide
|
C19H15F3N2O3S
|
1
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| 1 |
IC50 = 500 nM
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CP0535156
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3-(4-Methanesulfonyl-phenyl)-4,4-dimethyl-2-phenyl-cyclobut-2-enol
Show/Hide
|
C19H20O3S
|
1
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| 1 |
IC50 = 530 nM
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CP0511117
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4-(4-Methanesulfonyl-phenyl)-5,5-dimethyl-3-(pyrazin-2-yloxy)-5H-furan-2-one
Show/Hide
|
C17H16N2O5S
|
1
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| 1 |
IC50 = 550 nM
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CP0429982
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3-(3,5-Difluoro-phenyl)-5-hydroxy-4-(4-methanesulfonyl-phenyl)-5-methyl-5H-furan-2-one
Show/Hide
|
C18H14F2O5S
|
1
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| 1 |
IC50 = 550 nM
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CP0427144
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3-[(5-cyano-3-fluoro)phenoxymethyl]-1-(4-methanesulfonylphenyl)-5-phenyl-1H-pyrazole
Show/Hide
|
C24H18FN3O3S
|
1
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| 1 |
IC50 = 570 nM
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CP0505182
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3-Benzoyl-4-(4-methanesulfonyl-phenyl)-5,5-dimethyl-5H-furan-2-one
Show/Hide
|
C20H18O5S
|
1
|
| 1 |
IC50 = 600 nM
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CP0463028
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4-(4-Fluoro-phenyl)-5-(4-methanesulfonyl-phenyl)-2-thiazol-2-ylmethyl-2H-pyridazin-3-one
Show/Hide
|
C21H16FN3O3S2
|
1
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| 1 |
IC50 = 600 nM
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CP0279521
|
3-(4-Methanesulfonyl-phenyl)-[2,3']bipyridinyl
Show/Hide
|
C17H14N2O2S
|
1
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| 1 |
IC50 = 610 nM
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CP0420498
|
3-[3-fluoro-5-(4-methoxytetrahydropyran-4-yl)phenoxymethyl]-1,5-diphenyl-1H-pyrazole
Show/Hide
|
C28H27FN2O3
|
1
|
| 1 |
IC50 = 610 nM
|
|
|
|
CP0453451
|
4-(4-Methanesulfonyl-phenyl)-5,5-dimethyl-3-(pyrimidin-2-yloxy)-5H-furan-2-one
Show/Hide
|
C17H16N2O5S
|
1
|
| 1 |
IC50 = 620 nM
|
|
|
|
CP0409133
|
2-(4-Bromo-pyridin-2-yl)-3-(4-methanesulfonyl-phenyl)-cyclopent-2-enone
Show/Hide
|
C17H14BrNO3S
|
1
|
| 1 |
IC50 = 630 nM
|
|
|
|
CP0214693
|
N-[6-(5-methylpyridin-2-yl)sulfanyl-1-oxo-2,3-dihydroinden-5-yl]methanesulfonamide
Show/Hide
|
C16H16N2O3S2
|
1
|
| 1 |
IC50 = 640 nM
|
|
|
|
CP0551566
|
3-Benzo[b]thiophen-2-yl-5-hydroxy-4-(4-methanesulfonyl-phenyl)-5-methyl-5H-furan-2-one
Show/Hide
|
C20H16O5S2
|
1
|
| 1 |
IC50 = 650 nM
|
|
|
|
CP0533028
|
3-(Isoquinolin-5-yloxy)-4-(4-methanesulfonyl-phenyl)-5,5-dimethyl-5H-furan-2-one
Show/Hide
|
C22H19NO5S
|
1
|
| 1 |
IC50 = 670 nM
|
|
|
|
CP0437318
|
1-(4-methanesulfonylphenyl)-3-[(3,4-dimethoxy)phenoxymethyl]-5-phenyl-1H-pyrazole
Show/Hide
|
C25H24N2O5S
|
1
|
| 1 |
IC50 = 700 nM
|
|
|
|
CP0437320
|
1-(3,4-dichlorophenyl)-3-[3-fluoro-5-(4-methoxytetrahydropyran-4-yl)phenoxymethyl]-5-phenyl-1H-pyrazole
Show/Hide
|
C28H25Cl2FN2O3
|
1
|
| 1 |
IC50 = 700 nM
|
|
|
|
CP0428151
|
1-(4-methanesulfonylphenyl)-3-[(3-nitro)phenoxymethyl]-5-phenyl-1H-pyrazole
Show/Hide
|
C23H19N3O5S
|
1
|
| 1 |
IC50 = 740 nM
|
|
|
|
CP0425190
|
1-(4-trifluoromethoxyphenyl)-3-[3-fluoro-5-(4-methoxytetrahydropyran-4-yl)phenoxymethyl]-5-phenyl-1H-pyrazole
Show/Hide
|
C29H26F4N2O4
|
1
|
| 1 |
IC50 = 820 nM
|
|
|
|
CP0299190
|
5-Chloro-3-(4-methanesulfonyl-phenyl)-4'-methyl-[2,3']bipyridinyl
Show/Hide
|
C18H15ClN2O2S
|
1
|
| 1 |
IC50 = 830 nM
|
|
|
|
CP0356874
|
N-[6-[(5-methyl-1,3-thiazol-2-yl)sulfanyl]-1-oxo-2,3-dihydroinden-5-yl]methanesulfonamide
Show/Hide
|
C14H14N2O3S3
|
1
|
| 1 |
IC50 = 870 nM
|
|
|
|
CP0522693
|
1-(4-methanesulfonylphenyl)-3-[(3,5-dimethoxy)phenoxymethyl]-5-phenyl-1H-pyrazole
Show/Hide
|
C25H24N2O5S
|
1
|
| 1 |
IC50 = 870 nM
|
|
|
|
CP0406295
|
5-(4-Methanesulfonyl-phenyl)-6-phenyl-imidazo[2,1-b]thiazole-3-carboxylic acid ethyl ester
Show/Hide
|
C21H18N2O4S2
|
1
|
| 1 |
IC50 = 900 nM
|
|
|
|
CP0511927
|
3-[(3-ethoxy)phenoxymethyl]-1-(4-methanesulfonylphenyl)-5-phenyl-1H-pyrazole
Show/Hide
|
C25H24N2O4S
|
1
|
| 1 |
IC50 = 900 nM
|
|
|
|
CP0427142
|
1-(4-methanesulfonylphenyl)-3-[3-(4-morpholino)phenoxymethyl]-5-phenyl-1H-pyrazole
Show/Hide
|
C27H27N3O4S
|
1
|
| 1 |
IC50 = 920 nM
|
|
|
|
CP0405546
|
1-(4-chlorophenyl)-3-[3-fluoro-5-(4-methoxytetrahydropyran-4-yl)phenoxymethyl]-5-phenyl-1H-pyrazole
Show/Hide
|
C28H26ClFN2O3
|
1
|
| 1 |
IC50 = 930 nM
|
|
|
|
CP0475206
|
3-[3-fluoro-5-(4-methoxytetrahydropyran-4-yl)phenoxymethyl]-1-(4-methylphenyl)-5-phenyl-1H-pyrazole
Show/Hide
|
C29H29FN2O3
|
1
|
| 1 |
IC50 = 930 nM
|
|
|
|
CP0405545
|
3-[3-fluoro-5-(4-methoxytetrahydropyran-4-yl)phenoxymethyl]-1-(4-fluorophenyl)-5-phenyl-1H-pyrazole
Show/Hide
|
C28H26F2N2O3
|
1
|
| 1 |
IC50 = 960 nM
|
|
|
|
CP0410010
|
6-(4-Methanesulfonyl-phenyl)-3-methyl-5-phenyl-imidazo[2,1-b]thiazole
Show/Hide
|
C19H16N2O2S2
|
1
|
| 1 |
IC50 = 1000 nM
|
|
|
|
CP0403632
|
2-Benzyl-5-(4-methanesulfonyl-phenyl)-4-(6-methyl-pyridin-3-yl)-2H-pyridazin-3-one
Show/Hide
|
C24H21N3O3S
|
1
|
| 1 |
IC50 = 1200 nM
|
|
|
|
CP0544001
|
3-(2,4-Dichloro-phenyl)-5-hydroxy-4-(4-methanesulfonyl-phenyl)-5-methyl-5H-furan-2-one
Show/Hide
|
C18H14Cl2O5S
|
1
|
| 1 |
IC50 = 1200 nM
|
|
|
|
CP0377852
|
5-(4-Methanesulfonyl-phenyl)-4-phenyl-2-pyridin-3-ylmethyl-2H-pyridazin-3-one
Show/Hide
|
C23H19N3O3S
|
1
|
| 1 |
IC50 = 1300 nM
|
|
|
|
CP0124380
|
5-Chloro-3-(4-methanesulfonyl-phenyl)-2'-methyl-[2,3']bipyridinyl
Show/Hide
|
C18H15ClN2O2S
|
1
|
| 1 |
IC50 = 1330 nM
|
|
|
|
CP0493881
|
3-(4-Methanesulfonyl-phenyl)-2-pyridin-2-yl-cyclopent-2-enone
Show/Hide
|
C17H15NO3S
|
1
|
| 1 |
IC50 = 1530 nM
|
|
|
|
CP0373335
|
5-Hydroxy-4-(4-methanesulfonyl-phenyl)-5-methyl-3-thiophen-2-yl-5H-furan-2-one
Show/Hide
|
C16H14O5S2
|
1
|
| 1 |
IC50 = 1900 nM
|
|
|
|
CP0509905
|
4-(4-Methanesulfonyl-phenyl)-5,5-dimethyl-3-(quinazolin-4-yloxy)-5H-furan-2-one
Show/Hide
|
C21H18N2O5S
|
1
|
| 1 |
IC50 = 2900 nM
|
|
|
|
CP0404472
|
5-(4-Methanesulfonyl-phenyl)-3-methyl-6-phenyl-imidazo[2,1-b]thiazole
Show/Hide
|
C19H16N2O2S2
|
1
|
| 1 |
IC50 = 3000 nM
|
|
|
|
CP0467337
|
6-(4-Methanesulfonyl-phenyl)-5-phenyl-imidazo[2,1-b]thiazole
Show/Hide
|
C18H14N2O2S2
|
1
|
| 1 |
IC50 = 3210 nM
|
|
|
|
CP0483637
|
2,3-Dichloro-6-(4-chloro-phenyl)-5-(4-methanesulfonyl-phenyl)-imidazo[2,1-b]thiazole
Show/Hide
|
C18H11Cl3N2O2S2
|
1
|
| 1 |
IC50 = 3600 nM
|
|
|
|
CP0437670
|
5-(4-Methanesulfonyl-phenyl)-2,3-dimethyl-6-phenyl-imidazo[2,1-b]thiazole
Show/Hide
|
C20H18N2O2S2
|
1
|
| 1 |
IC50 = 5000 nM
|
|
|
|
CP0448740
|
6-(4-Methylsulfanyl-phenyl)-5-phenyl-imidazo[2,1-b]thiazole
Show/Hide
|
C18H14N2S2
|
1
|
| 1 |
IC50 = 5000 nM
|
|
|
|
CP0215382
|
N-[6-[(4-methylsulfanyl-1,3-thiazol-2-yl)sulfanyl]-1-oxo-3H-2-benzofuran-5-yl]methanesulfonamide
Show/Hide
|
C13H12N2O4S4
|
1
|
| 1 |
IC50 = 11000 nM
|
|
|
|
CP0405020
|
6-(4-Methanesulfonyl-phenyl)-5-phenyl-2-trifluoromethyl-thiazolo[3,2-b][1,2,4]triazole
Show/Hide
|
C18H12F3N3O2S2
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
|
CP0341579
|
6-((3-fluoro-5-(4-methoxytetrahydro-2H-pyran-4-yl)phenoxy)methyl)-1-methylquinolin-2(1H)-one
Show/Hide
|
C23H24FNO4
|
1
|
| 1 |
IC50 > 100000 nM
|
|
|
|
CP0375888
|
3-(4-methylsulfonylphenyl)-2-phenoxy-5-(trifluoromethyl)pyridine
Show/Hide
|
C19H14F3NO3S
|
1
|
| 1 |
IC50 < 200 nM
|
|
|
|
CP0426034
|
3-(4-Methanesulfonyl-phenyl)-2-(2,2,2-trifluoro-ethoxy)-5-trifluoromethyl-pyridine
Show/Hide
|
C15H11F6NO3S
|
1
|
| 1 |
IC50 < 200 nM
|
|
|
|
CP0430495
|
(R)-2-[3-(4-Methanesulfonyl-phenyl)-5-trifluoromethyl-pyridin-2-ylsulfanyl]-propan-1-ol
Show/Hide
|
C16H16F3NO3S2
|
1
|
| 1 |
IC50 < 200 nM
|
|
|
|
CP0430496
|
[1-[3-(4-methylsulfonylphenyl)-5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl]methanol
Show/Hide
|
C19H21F3N2O3S
|
1
|
| 1 |
IC50 < 200 nM
|
|
|
|
CP0448538
|
2-(4-Chloro-benzyloxy)-3-(4-methanesulfonyl-phenyl)-5-trifluoromethyl-pyridine
Show/Hide
|
C20H15ClF3NO3S
|
1
|
| 1 |
IC50 < 200 nM
|
|
|
|
CP0448757
|
1-[3-(4-Methanesulfonyl-phenyl)-5-trifluoromethyl-pyridin-2-yloxy]-2-methyl-propan-2-ol
Show/Hide
|
C17H18F3NO4S
|
1
|
| 1 |
IC50 < 200 nM
|
|
|
|
CP0455670
|
(S)-3-[3-(4-Methanesulfonyl-phenyl)-5-trifluoromethyl-pyridin-2-yloxy]-2-methyl-butan-2-ol
Show/Hide
|
C18H20F3NO4S
|
1
|
| 1 |
IC50 < 200 nM
|
|
|
|
CP0464218
|
(1S,2R)-2-[3-(4-Methanesulfonyl-phenyl)-5-trifluoromethyl-pyridin-2-yloxy]-1-methyl-cyclopentanol
Show/Hide
|
C19H20F3NO4S
|
1
|
| 1 |
IC50 < 200 nM
|
|
|
|
CP0502697
|
1-[3-(4-Methanesulfonyl-phenyl)-5-trifluoromethyl-pyridin-2-ylsulfanyl]-2-methyl-propan-2-ol
Show/Hide
|
C17H18F3NO3S2
|
1
|
| 1 |
IC50 < 200 nM
|
|
|
|
CP0510029
|
3-(4-Methanesulfonyl-phenyl)-5-trifluoromethyl-2-(2,2,2-trifluoro-1-trifluoromethyl-ethoxy)-pyridine
Show/Hide
|
C16H10F9NO3S
|
1
|
| 1 |
IC50 < 200 nM
|
|
|
|
CP0510982
|
1-[3-(4-Methanesulfonyl-phenyl)-5-trifluoromethyl-pyridin-2-yloxymethyl]-cyclopentanol
Show/Hide
|
C19H20F3NO4S
|
1
|
| 1 |
IC50 < 200 nM
|
|
|
|
CP0530840
|
(S)-3-Ethyl-2-[3-(4-methanesulfonyl-phenyl)-5-trifluoromethyl-pyridin-2-yloxy]-pentan-3-ol
Show/Hide
|
C20H24F3NO4S
|
1
|
| 1 |
IC50 < 200 nM
|
|
|
|
CP0196302
|
N-[6-[(4,5-dimethyl-1,3-thiazol-2-yl)sulfanyl]-1-oxo-2,3-dihydroinden-5-yl]methanesulfonamide
Show/Hide
|
C15H16N2O3S3
|
1
|
| 1 |
IC50 > 1800 nM
|
|
|
|
CP0510619
|
1-Methanesulfonyl-4-(2-phenyl-cyclobut-1-enyl)-benzene
Show/Hide
|
C17H16O2S
|
1
|
| 1 |
IC50 > 5000 nM
|
|
|
|
CP0376557
|
6-(4-Methanesulfonyl-phenyl)-2,3-dimethyl-5-phenyl-imidazo[2,1-b]thiazole
Show/Hide
|
C20H18N2O2S2
|
1
|
| 1 |
IC50 > 5000 nM
|
|
|
|
CP0402232
|
5-(4-Methanesulfonyl-phenyl)-6-phenyl-imidazo[2,1-b]thiazole-3-carboxylic acid
Show/Hide
|
C19H14N2O4S2
|
1
|
| 1 |
IC50 > 5000 nM
|
|
|
|
CP0494744
|
2-(4-Methanesulfonyl-phenyl)-3-phenyl-benzo[d]imidazo[2,1-b]thiazole
Show/Hide
|
C22H16N2O2S2
|
1
|
| 1 |
IC50 > 5000 nM
|
|
|
|
CP0524161
|
3-(4-Methanesulfonyl-phenyl)-2-phenyl-benzo[d]imidazo[2,1-b]thiazole
Show/Hide
|
C22H16N2O2S2
|
1
|
| 1 |
IC50 > 5000 nM
|
|
|
|
CP0298848
|
4-(4-Methanesulfonyl-phenyl)-3-pyridin-3-yl-5H-furan-2-one
Show/Hide
|
C16H13NO4S
|
1
|
| 1 |
IC50 > 5000 nM
|
|
|
|
CP0463338
|
2-tert-Butyl-5-(4-methanesulfonyl-phenyl)-4-phenyl-2H-pyridazin-3-one
Show/Hide
|
C21H22N2O3S
|
1
|
| 1 |
IC50 > 5000 nM
|
|
|
|
CP0496313
|
5-(4-Methanesulfonyl-phenyl)-4-phenyl-2H-pyridazin-3-one
Show/Hide
|
C17H14N2O3S
|
1
|
| 1 |
IC50 > 5000 nM
|
|
|
|
CP0434021
|
5-Hydroxy-3-(4-hydroxy-phenyl)-4-(4-methanesulfonyl-phenyl)-5-methyl-5H-furan-2-one
Show/Hide
|
C18H16O6S
|
1
|
| 1 |
IC50 > 5000 nM
|
|
|
|
CP0511146
|
3-(3,4-Difluoro-phenoxy)-5-hydroxy-4-(4-methanesulfonyl-phenyl)-5-methyl-5H-furan-2-one
Show/Hide
|
C18H14F2O6S
|
1
|
| 1 |
IC50 > 5000 nM
|
|
|
|
CP0526034
|
5-Hydroxy-4-(4-methanesulfonyl-phenyl)-5-methyl-3-phenylsulfanyl-5H-furan-2-one
Show/Hide
|
C18H16O5S2
|
1
|
| 1 |
IC50 > 5000 nM
|
|
|
