General Information of the Protein
Protein ID
PT02856
Protein Name
Neuropeptide Y receptor type 5
Secondarily
Protein Name
NPY-Y5 receptor
Gene Name
NPY5R
Secondarily
Gene Name
Npy5
Sequence
MEVKLEEHFNKTFVTENNTAASQNTASPAWEDYRGTENNTSAARNTAFPVWEDYRGSVDDLQYFLIGLYTFVSLLGFMGNLLILMAVMKKRNQKTTVNFLIGNLAFSDILVVLFCSPFTLTSVLLDQWMFGKAMCHIMPFLQCVSVLVSTLILISIAIVRYHMIKHPISNNLTANHGYFLIATVWTLGFAICSPLPVFHSLVELKETFGSALLSSKYLCVESWPSDSYRIAFTISLLLVQYILPLVCLTVSHTSVCRSISCGLSHKENRLEENEMINLTLHPSKKSRDQAKPPSTQKWSYSFIRKHRRRYSKKTACVLPAPAGPSQEKHLTVPENPGSVRSQLSPSSKVIPGVPICFEVKPEESSDAQEMRVKRSLTRIKKRSRSVFYRLTILILVFAVSWMPLHVFHVVTDFNDNLISNRHFKLVYCICHLLGMMSCCLNPILYGFLNNGIKADLRALIHCLHMS
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Organism
Mus musculus, Mouse
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
>
Peptide receptor (family A GPCR)
>
Short peptide receptor (family A GPCR)
>
Neuropeptide Y receptor
Function
Receptor for neuropeptide Y and peptide YY. The activity of this receptor is mediated by G proteins that inhibit adenylate cyclase activity. Seems to be associated with food intake. Could be involved in feeding disorders (By similarity).
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Uniprot ID
Primary ID:
O70342

Secondarily ID:
O35380
Q9JMK1
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Subcellular Location
Cell membrane
Map of Molecular Bioactivity Related to the Protein
Map of Molecular Bioactivity Related to the Protein

Protein
Cell Line
Compound

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Protein
Cell Line ID: CL000011 , CHO
Compound ID Compound Name Compound Formula
CP0480738
US8916594, I-024
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C18H26N4O3S
 1
1
IC50 = 0.13 nM
   TI
   LI
   LO
   TS
CP0566447
US8916594, I-034
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C17H22F2N4O3S
 1
1
IC50 = 0.18 nM
   TI
   LI
   LO
   TS
CP0480737
US8916594, I-018
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C18H25FN4O3S
 1
1
IC50 = 0.2 nM
   TI
   LI
   LO
   TS
CP0442988
US8916594, I-017
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C17H23FN4O3S
 1
1
IC50 = 0.22 nM
   TI
   LI
   LO
   TS
CP0442989
US8916594, I-029
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C17H22F2N4O3S
 1
1
IC50 = 0.22 nM
   TI
   LI
   LO
   TS
CP0442990
US8916594, I-053
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C17H22F2N4O3S
 1
1
IC50 = 0.23 nM
   TI
   LI
   LO
   TS
CP0442157
US8653125, Ia-40
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C19H18Cl2N4O2
 1
1
IC50 = 0.26 nM
   TI
   LI
   LO
   TS
CP0480736
US8916594, I-006
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C17H23FN4O3S
 1
1
IC50 = 0.32 nM
   TI
   LI
   LO
   TS
CP0560659
US8916594, I-011
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C17H24N4O3S
 1
1
IC50 = 0.34 nM
   TI
   LI
   LO
   TS
CP0541860
US8653125, Ic-16
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C23H24F3N3O4
 1
1
IC50 = 0.41 nM
   TI
   LI
   LO
   TS
CP0480739
US8916594, I-138
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C16H27FN4O3S
 1
1
IC50 = 0.5 nM
   TI
   LI
   LO
   TS
CP0560615
US8653125, Ic-13
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C24H24ClN3O4
 1
1
IC50 = 0.56 nM
   TI
   LI
   LO
   TS
CP0557185
US8653125, Id-8
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C22H21FN4O4S
 1
1
IC50 = 0.58 nM
   TI
   LI
   LO
   TS
CP0560663
US8916594, I-147
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C17H28F2N4O3S
 1
1
IC50 = 0.61 nM
   TI
   LI
   LO
   TS
CP0549967
US8916594, I-152
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C14H21F5N4O3S
 1
1
IC50 = 0.65 nM
   TI
   LI
   LO
   TS
CP0512199
US8653125, Ia-35
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C23H23N3O3
 1
1
IC50 = 0.65 nM
   TI
   LI
   LO
   TS
CP0541859
US8653125, Ic-14
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C25H24F3N3O4
 1
1
IC50 = 0.68 nM
   TI
   LI
   LO
   TS
CP0484934
US8653125, Ic-17
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C21H20ClFN4O2
 1
1
IC50 = 0.69 nM
   TI
   LI
   LO
   TS
CP0446245
US8916594, I-130
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C22H34N4O3S
 1
1
IC50 = 0.7 nM
   TI
   LI
   LO
   TS
CP0560612
US8653125, Ia-30
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C23H22FN3O3
 1
1
IC50 = 0.71 nM
   TI
   LI
   LO
   TS
CP0529317
US8916594, I-143
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C18H30F2N4O3S
 1
1
IC50 = 0.8 nM
   TI
   LI
   LO
   TS
CP0566448
US8916594, I-099
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C17H24FN5O3S
 1
1
IC50 = 0.8 nM
   TI
   LI
   LO
   TS
CP0529316
US8916594, I-027
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C16H21FN4O3S
 1
1
IC50 = 0.86 nM
   TI
   LI
   LO
   TS
CP0442992
US8916594, I-081
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C16H21ClN4O3S
 1
1
IC50 = 0.9 nM
   TI
   LI
   LO
   TS
CP0551025
US8916594, I-100
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C18H26FN5O3S
 1
1
IC50 = 0.9 nM
   TI
   LI
   LO
   TS
CP0549966
US8916594, I-149
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C15H23F5N4O3S
 1
1
IC50 = 1.04 nM
   TI
   LI
   LO
   TS
CP0484939
US8653125, Ic-12
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C26H30ClN3O3
 1
1
IC50 = 1.1 nM
   TI
   LI
   LO
   TS
CP0560661
US8916594, I-023
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C16H21FN4O3S
 1
1
IC50 = 1.4 nM
   TI
   LI
   LO
   TS
CP0515684
US8916594, I-136
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C14H23F3N4O3S
 1
1
IC50 = 1.5 nM
   TI
   LI
   LO
   TS
CP0503728
US8653125, Ib-4
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C22H25FN4O3
 1
1
IC50 = 1.5 nM
   TI
   LI
   LO
   TS
CP0520453
US8653125, Ic-5
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C24H30ClN3O3
 1
1
IC50 = 1.5 nM
   TI
   LI
   LO
   TS
CP0512198
US8653125, Ia-2
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C22H21F2N5O2
 1
1
IC50 = 1.6 nM
   TI
   LI
   LO
   TS
CP0442993
US8916594, I-153
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C13H19F5N4O3S
 1
1
IC50 = 1.67 nM
   TI
   LI
   LO
   TS
CP0441913
US8653125, Ia-43
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C20H19F3N4O2
 1
1
IC50 = 1.8 nM
   TI
   LI
   LO
   TS
CP0521159
US8653125, Ic-11
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C27H30F3N3O3
 1
1
IC50 = 1.8 nM
   TI
   LI
   LO
   TS
CP0549969
US8916594, I-161
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C17H27F3N4O3S
 1
1
IC50 = 1.9 nM
   TI
   LI
   LO
   TS
CP0541858
US8653125, Ic-8
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C21H20F2N2O3
 1
1
IC50 = 2.3 nM
   TI
   LI
   LO
   TS
CP0512200
US8653125, Ib-1
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C21H21F2N5O
 1
1
IC50 = 2.9 nM
   TI
   LI
   LO
   TS
CP0530655
US8653125, Ia-24
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C24H22FN5O2
 1
1
IC50 = 2.9 nM
   TI
   LI
   LO
   TS
CP0560614
US8653125, Ia-42
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C19H19ClN4O2
 1
1
IC50 = 3 nM
   TI
   LI
   LO
   TS
CP0560662
US8916594, I-145
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C13H21F3N4O3S
 1
1
IC50 = 3.1 nM
   TI
   LI
   LO
   TS
CP0560613
US8653125, Ia-32
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C21H24N4O5
 1
1
IC50 = 3.3 nM
   TI
   LI
   LO
   TS
CP0560664
US8916594, I-150
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C14H22F3N3O3S
 1
1
IC50 = 3.6 nM
   TI
   LI
   LO
   TS
CP0578534
US8653125, Ia-4
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C22H21ClFN5O2
 1
1
IC50 = 3.8 nM
   TI
   LI
   LO
   TS
CP0465477
US8653125, Ia-28
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C23H22FN3O3
 1
1
IC50 = 4.1 nM
   TI
   LI
   LO
   TS
CP0541857
US8653125, Ia-14
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C26H25FN2O2
 1
1
IC50 = 4.1 nM
   TI
   LI
   LO
   TS
CP0549965
US8916594, I-146
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C15H24F3N3O3S
 1
1
IC50 = 4.21 nM
   TI
   LI
   LO
   TS
CP0560611
US8653125, Ia-15
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C24H27N3O4
 1
1
IC50 = 4.5 nM
   TI
   LI
   LO
   TS