| Compound ID |
Compound Name |
Compound Formula |
|
CP0001238
|
14C-5-hydroxy tryptamine creatinine disulfate
Show/Hide
|
C10H12N2O
|
4
|
| 1 |
EC50 = 43.6 nM
|
|
|
| 2 |
Ki = 33 nM
|
|
|
| 3 |
Ki = 75 nM
|
|
|
| 4 |
Ki = 78 nM
|
|
|
|
CP0081161
|
2-Phenyl-3-(1,2,3,6-tetrahydro-pyridin-4-yl)-1H-indole
Show/Hide
|
C19H18N2
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
|
CP0381514
|
3-(3-chlorophenyl)sulfonyl-N,5,7-trimethylpyrazolo[1,5-a]pyrimidin-2-amine
Show/Hide
|
C15H15ClN4O2S
|
2
|
| 1 |
IC50 = 2 nM
|
|
|
| 2 |
Ki = 0.1862 nM
|
|
|
|
CP0398640
|
N-[3-(4-methylpiperazin-1-yl)phenyl]-N-propan-2-ylnaphthalene-2-sulfonamide
Show/Hide
|
C24H29N3O2S
|
1
|
| 1 |
IC50 = 3 nM
|
|
|
|
CP0416325
|
N-ethyl-N-[3-(4-methylpiperazin-1-yl)phenyl]naphthalene-2-sulfonamide
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|
C23H27N3O2S
|
1
|
| 1 |
IC50 = 3 nM
|
|
|
|
CP0417851
|
N-benzyl-N-[3-(4-methylpiperazin-1-yl)phenyl]naphthalene-2-sulfonamide
Show/Hide
|
C28H29N3O2S
|
1
|
| 1 |
IC50 = 3 nM
|
|
|
|
CP0465482
|
3-(benzenesulfonyl)-N,7-dimethylpyrazolo[1,5-a]pyrimidin-2-amine
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|
C14H14N4O2S
|
2
|
| 1 |
IC50 = 3 nM
|
|
|
| 2 |
Ki = 0.2399 nM
|
|
|
|
CP0068819
|
3-(phenylsulfonyl)-N-(thiophen-2-ylmethyl)thieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-amine
Show/Hide
|
C18H13N5O2S3
|
3
|
| 1 |
IC50 = 3.6 nM
|
|
|
| 2 |
IC50 = 110 nM
|
|
|
| 3 |
Ki = 1.7 nM
|
|
|
|
CP0487098
|
N-[3-(4-methylpiperazin-1-yl)phenyl]-N-propylnaphthalene-2-sulfonamide
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|
C24H29N3O2S
|
1
|
| 1 |
IC50 = 4 nM
|
|
|
|
CP0043132
|
3-Benzenesulfonyl-2-methylsulfanyl-pyrido[1,2-a]pyrimidin-(4E)-ylideneamine
Show/Hide
|
C15H13N3O2S2
|
1
|
| 1 |
IC50 = 4 nM
|
|
|
|
CP0532668
|
3-(3-chloro-4-fluorophenyl)sulfonyl-N,5,7-trimethylpyrazolo[1,5-a]pyrimidin-2-amine
Show/Hide
|
C15H14ClFN4O2S
|
2
|
| 1 |
IC50 = 4 nM
|
|
|
| 2 |
Ki = 0.6026 nM
|
|
|
|
CP0465484
|
[3-(benzenesulfonyl)-5-methyl-2-(methylamino)pyrazolo[1,5-a]pyrimidin-7-yl]methanol
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|
C15H16N4O3S
|
2
|
| 1 |
IC50 = 4 nM
|
|
|
| 2 |
Ki = 0.2818 nM
|
|
|
|
CP0465485
|
US8618114, 1.2.8(8)
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|
C19H17N5O2S
|
1
|
| 1 |
IC50 = 4 nM
|
|
|
|
CP0539086
|
3-(benzenesulfonyl)-5-(methoxymethyl)-N,7-dimethylpyrazolo[1,5-a]pyrimidin-2-amine
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|
C16H18N4O3S
|
2
|
| 1 |
IC50 = 4 nM
|
|
|
| 2 |
Ki = 0.2692 nM
|
|
|
|
CP0105274
|
10-(benzenesulfonyl)-N-benzyl-N-methyl-5-thia-1,8,11,12-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaen-7-amine
Show/Hide
|
C21H17N5O2S2
|
3
|
| 1 |
IC50 = 5 nM
|
|
|
| 2 |
IC50 = 170 nM
|
|
|
| 3 |
Ki = 2.3 nM
|
|
|
|
CP0216239
|
3-(benzenesulfonyl)-N,5,7-trimethylpyrazolo[1,5-a]pyrimidin-2-amine
Show/Hide
|
C15H16N4O2S
|
3
|
| 1 |
IC50 = 5 nM
|
|
|
| 2 |
Ki = 0.257 nM
|
|
|
| 3 |
Ki = 0.26 nM
|
|
|
|
CP0379663
|
3-(3-fluorophenyl)sulfonyl-N,5,7-trimethylpyrazolo[1,5-a]pyrimidin-2-amine
Show/Hide
|
C15H15FN4O2S
|
2
|
| 1 |
IC50 = 5 nM
|
|
|
| 2 |
Ki = 0.5012 nM
|
|
|
|
CP0485301
|
2-(methylthio)-3-(phenylsulfonyl)-7,8-dihydro-6H-cyclopenta[e]pyrazolo[1,5-a]pyrimidine
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|
C16H15N3O2S2
|
2
|
| 1 |
IC50 = 6 nM
|
|
|
| 2 |
IC50 = 27 nM
|
|
|
|
CP0416326
|
N-(cyclopropylmethyl)-N-[3-(4-methylpiperazin-1-yl)phenyl]naphthalene-2-sulfonamide
Show/Hide
|
C25H29N3O2S
|
1
|
| 1 |
IC50 = 6 nM
|
|
|
|
CP0473511
|
3-(4-fluorophenyl)sulfonyl-N,5,7-trimethylpyrazolo[1,5-a]pyrimidin-2-amine
Show/Hide
|
C15H15FN4O2S
|
2
|
| 1 |
IC50 = 6 nM
|
|
|
| 2 |
Ki = 0.3981 nM
|
|
|
|
CP0416635
|
10-(benzenesulfonyl)-N-(furan-2-ylmethyl)-5-thia-1,8,11,12-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaen-7-amine
Show/Hide
|
C18H13N5O3S2
|
3
|
| 1 |
IC50 = 6.1 nM
|
|
|
| 2 |
IC50 = 40 nM
|
|
|
| 3 |
Ki = 2.8 nM
|
|
|
|
CP0504477
|
10-(benzenesulfonyl)-N-cyclohexyl-5-thia-1,8,11,12-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaen-7-amine
Show/Hide
|
C19H19N5O2S2
|
3
|
| 1 |
IC50 = 6.9 nM
|
|
|
| 2 |
IC50 = 200 nM
|
|
|
| 3 |
Ki = 3.2 nM
|
|
|
|
CP0377202
|
N-methyl-N-[3-(4-methylpiperazin-1-yl)phenyl]naphthalene-2-sulfonamide
Show/Hide
|
C22H25N3O2S
|
1
|
| 1 |
IC50 = 7 nM
|
|
|
|
CP0408044
|
(S)-2-methyl-5-(4-methylpiperazin-1-yl)-1-(naphthalen-2-ylsulfonyl)-2,3-dihydroquinolin-4(1H)-one
Show/Hide
|
C25H27N3O3S
|
1
|
| 1 |
IC50 = 7 nM
|
|
|
|
CP0077916
|
5-Chloro-2-methyl-3-(1,2,3,6-tetrahydro-pyridin-4-yl)-1H-indole
Show/Hide
|
C14H15ClN2
|
1
|
| 1 |
IC50 = 7.4 nM
|
|
|
|
CP0406285
|
2-(methylthio)-3-(phenylsulfonyl)-6,7,8,9-tetrahydropyrazolo[1,5-a]quinazoline
Show/Hide
|
C17H17N3O2S2
|
2
|
| 1 |
IC50 = 7.5 nM
|
|
|
| 2 |
IC50 = 35 nM
|
|
|
|
CP0125845
|
N-benzyl-10-(3-chlorophenyl)sulfonyl-N-methyl-5-thia-1,8,11,12-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaen-7-amine
Show/Hide
|
C21H16ClN5O2S2
|
3
|
| 1 |
IC50 = 7.5 nM
|
|
|
| 2 |
IC50 = 920 nM
|
|
|
| 3 |
Ki = 3.5 nM
|
|
|
|
CP0294753
|
9-methyl-2-(methylthio)-3-(phenylsulfonyl)-5,6,7,8-tetrahydropyrazolo[5,1-b]quinazoline
Show/Hide
|
C18H19N3O2S2
|
1
|
| 1 |
IC50 = 7.8 nM
|
|
|
|
CP0380601
|
2-methyl-5-(N-methyl-piperazin-1-yl)-1-(naphthalene-2-sulfonyl)-2,3-dihydro-1H-quinolin-4-one
Show/Hide
|
C25H27N3O3S
|
1
|
| 1 |
IC50 = 8 nM
|
|
|
|
CP0380597
|
2-ethyl-5-(N-methyl-piperazin-1-yl)-1-(naphthalene-2-sulfonyl)-2,3-dihydro-1H-quinolin-4-one
Show/Hide
|
C26H29N3O3S
|
1
|
| 1 |
IC50 = 9 nM
|
|
|
|
CP0898489
|
2-Methyl-5-(2-nitrophenoxy)-3-(1,2,3,6-tetrahydropyridin-4-yl)-1H-indole
Show/Hide
|
C20H19N3O3
|
1
|
| 1 |
IC50 = 9 nM
|
|
|
|
CP0392081
|
US8618114, 1.2.19(2).HCl
Show/Hide
|
C15H17N5O2S
|
2
|
| 1 |
IC50 = 9 nM
|
|
|
| 2 |
Ki = 0.5754 nM
|
|
|
|
CP0431340
|
US8618114, 1.2.22(2).HCl
Show/Hide
|
C16H19N5O2S
|
2
|
| 1 |
IC50 = 9 nM
|
|
|
| 2 |
Ki = 0.6457 nM
|
|
|
|
CP0483653
|
5-Chloro-2-methyl-3-(1-methyl-1,2,3,6-tetrahydro-pyridin-4-yl)-1H-indole
Show/Hide
|
C15H17ClN2
|
1
|
| 1 |
IC50 = 10 nM
|
|
|
|
CP0671076
|
2-Methyl-5-nitro-3-(1,2,3,6-tetrahydropyridin-4-yl)-1Hindole
Show/Hide
|
C14H15N3O2
|
1
|
| 1 |
IC50 = 10 nM
|
|
|
|
CP0681119
|
5-Bromo-2-methyl-3-(1,2,3,6-tetrahydropyridin-4-yl)-1Hindole
Show/Hide
|
C14H15BrN2
|
1
|
| 1 |
IC50 = 10 nM
|
|
|
|
CP0401198
|
US8618114, 1.2.22(5).HCl
Show/Hide
|
C16H18ClN5O2S
|
2
|
| 1 |
IC50 = 10 nM
|
|
|
| 2 |
Ki = 0.5495 nM
|
|
|
|
CP0530458
|
US8618114, 1.1.8(3)
Show/Hide
|
C19H16N4O3S2
|
1
|
| 1 |
IC50 < 10 nM
|
|
|
|
CP0380598
|
2,7-dimethyl-5-(4-methylpiperazin-1-yl)-1-(naphthalen-2-ylsulfonyl)-2,3-dihydroquinolin-4(1H)-one
Show/Hide
|
C26H29N3O3S
|
1
|
| 1 |
IC50 = 11 nM
|
|
|
|
CP0181403
|
US8618114, 1.2.22(1).HCl
Show/Hide
|
C15H17N5O2S
|
3
|
| 1 |
IC50 = 11.33 nM
|
|
|
| 2 |
Kd = 0.3981 nM
|
|
|
| 3 |
Ki = 0.5248 nM
|
|
|
|
CP0377182
|
10-(benzenesulfonyl)-N-cyclopentyl-5-thia-1,8,11,12-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaen-7-amine
Show/Hide
|
C18H17N5O2S2
|
3
|
| 1 |
IC50 = 11.9 nM
|
|
|
| 2 |
IC50 = 140 nM
|
|
|
| 3 |
Ki = 5.5 nM
|
|
|
|
CP0077216
|
US8618114, 1.2.11(1)
Show/Hide
|
C14H15N5O2S
|
3
|
| 1 |
IC50 = 12 nM
|
|
|
| 2 |
Kd = 0.5012 nM
|
|
|
| 3 |
Ki = 0.302 nM
|
|
|
|
CP0447454
|
US8618114, 1.2.12(2)
Show/Hide
|
C16H19N5O2S
|
2
|
| 1 |
IC50 = 12 nM
|
|
|
| 2 |
Ki = 0.3467 nM
|
|
|
|
CP0539246
|
US8618114, 1.2.10(3)
Show/Hide
|
C19H17N5O3S
|
1
|
| 1 |
IC50 = 12 nM
|
|
|
|
CP0377208
|
N-[3-(4-methylpiperazin-1-yl)phenyl]naphthalene-2-sulfonamide
Show/Hide
|
C21H23N3O2S
|
1
|
| 1 |
IC50 = 13 nM
|
|
|
|
CP0648533
|
N-(3-Fluorophenyl)-2-methyl-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole-8-sulfonamide hydrochloride
Show/Hide
|
C18H19ClFN3O2S
|
1
|
| 1 |
IC50 = 15 nM
|
|
|
|
CP0527677
|
2,6-dimethyl-5-(4-methylpiperazin-1-yl)-1-(naphthalen-2-ylsulfonyl)-2,3-dihydroquinolin-4(1H)-one
Show/Hide
|
C26H29N3O3S
|
1
|
| 1 |
IC50 = 15 nM
|
|
|
|
CP0398637
|
N-[3-(4-methylpiperazin-1-yl)phenyl]-N-propan-2-ylnaphthalene-1-sulfonamide
Show/Hide
|
C24H29N3O2S
|
1
|
| 1 |
IC50 = 16 nM
|
|
|
|
CP0381513
|
3-(benzenesulfonyl)-N,5-dimethylpyrazolo[1,5-a]pyrimidin-2-amine
Show/Hide
|
C14H14N4O2S
|
2
|
| 1 |
IC50 = 16 nM
|
|
|
| 2 |
Ki = 1.445 nM
|
|
|
|
CP0485300
|
5-methyl-2-(methylthio)-3-(phenylsulfonyl)-6,7,8,9-tetrahydropyrazolo[1,5-a]quinazoline
Show/Hide
|
C18H19N3O2S2
|
2
|
| 1 |
IC50 = 16.8 nM
|
|
|
| 2 |
IC50 = 32 nM
|
|
|
|
CP0527685
|
(S)-2-methyl-7-(4-methylpiperazin-1-yl)-1-(naphthalen-2-ylsulfonyl)-2,3-dihydroquinolin-4(1H)-one
Show/Hide
|
C25H27N3O3S
|
1
|
| 1 |
IC50 = 17 nM
|
|
|
|
CP0509330
|
3-(phenylsulfonyl)-N-((tetrahydrofuran-2-yl)methyl)thieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-amine
Show/Hide
|
C18H17N5O3S2
|
3
|
| 1 |
IC50 = 17.5 nM
|
|
|
| 2 |
IC50 = 63 nM
|
|
|
| 3 |
Ki = 8.1 nM
|
|
|
|
CP0530459
|
[3-(benzenesulfonyl)-7-methyl-2-(methylamino)pyrazolo[1,5-a]pyrimidin-5-yl]methanol
Show/Hide
|
C15H16N4O3S
|
2
|
| 1 |
IC50 = 19 nM
|
|
|
| 2 |
Ki = 0.4786 nM
|
|
|
|
CP0396616
|
3-(1,2,3,6-Tetrahydro-pyridin-4-yl)-1H-indole-5-carbonitrile
Show/Hide
|
C14H13N3
|
1
|
| 1 |
IC50 = 20 nM
|
|
|
|
CP0857428
|
2-Methyl-5-methylsulfanyl-3-(1,2,3,6-tetrahydropyridin-4-yl)-1H-indole
Show/Hide
|
C15H18N2S
|
1
|
| 1 |
IC50 = 20 nM
|
|
|
|
CP0025667
|
2-[4-(4-Methyl-benzyl)-piperazin-1-yl]-1-(2-methyl-2,3-dihydro-indol-1-yl)-ethanone
Show/Hide
|
C18H19ClN4
|
5
|
| 1 |
IC50 = 20 nM
|
|
|
| 2 |
Ki = 4 nM
|
|
|
| 3 |
Ki = 4.8 nM
|
|
|
| 4 |
Ki = 7.943 nM
|
|
|
| 5 |
Ki = 17 nM
|
|
|
|
CP0560640
|
US8618114, 1.2.22(11).HCl
Show/Hide
|
C15H16FN5O2S
|
1
|
| 1 |
IC50 = 22 nM
|
|
|
|
CP0505562
|
3-(3-chlorophenyl)sulfonyl-N-methylpyrazolo[1,5-a]pyrimidin-2-amine
Show/Hide
|
C13H11ClN4O2S
|
2
|
| 1 |
IC50 = 24 nM
|
|
|
| 2 |
Ki = 1.175 nM
|
|
|
|
CP0496117
|
US8618114, 1.2.22(6).HCl
Show/Hide
|
C16H18FN5O2S
|
2
|
| 1 |
IC50 = 25.19 nM
|
|
|
| 2 |
Ki = 1.413 nM
|
|
|
|
CP0379952
|
7-(4-methylpiperazin-1-yl)-1-(naphthalen-2-ylsulfonyl)-2,3-dihydroquinolin-4(1H)-one
Show/Hide
|
C24H25N3O3S
|
1
|
| 1 |
IC50 = 26 nM
|
|
|
|
CP0431341
|
US8618114, 1.2.22(10).HCl
Show/Hide
|
C18H23N5O2S
|
2
|
| 1 |
IC50 = 26 nM
|
|
|
| 2 |
Ki = 0.7079 nM
|
|
|
|
CP0487861
|
N-[4-(4-methylpiperazin-1-yl)phenyl]-N-propan-2-ylnaphthalene-2-sulfonamide
Show/Hide
|
C24H29N3O2S
|
1
|
| 1 |
IC50 = 27 nM
|
|
|
|
CP0380600
|
2-methyl-7-(N-methyl-piperazin-1-yl)-1-(naphthalene-2-sulfonyl)-2,3-dihydro-1H-quinolin-4-one
Show/Hide
|
C25H27N3O3S
|
1
|
| 1 |
IC50 = 28 nM
|
|
|
|
CP0523833
|
3-(2,5-dimethylphenylsulfonyl)-N-isopropylthieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-amine
Show/Hide
|
C18H19N5O2S2
|
2
|
| 1 |
IC50 = 28.3 nM
|
|
|
| 2 |
IC50 = 350 nM
|
|
|
|
CP0523843
|
3-(3-chlorophenylsulfonyl)-N-((tetrahydrofuran-2-yl)methyl)thieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-amine
Show/Hide
|
C18H16ClN5O3S2
|
1
|
| 1 |
IC50 = 29 nM
|
|
|
|
CP0393489
|
5-Chloro-3-(1-ethyl-1,2,3,6-tetrahydro-pyridin-4-yl)-2-methyl-1H-indole
Show/Hide
|
C16H19ClN2
|
1
|
| 1 |
IC50 = 30 nM
|
|
|
|
CP0441870
|
5-Chloro-2-ethyl-3-(1,2,3,6-tetrahydro-pyridin-4-yl)-1H-indole
Show/Hide
|
C15H17ClN2
|
1
|
| 1 |
IC50 = 30 nM
|
|
|
|
CP0658021
|
5-Fluoro-2-methyl-3-(1,2,3,6-tetrahydropyridin-4-yl)-1Hindole
Show/Hide
|
C14H15FN2
|
1
|
| 1 |
IC50 = 30 nM
|
|
|
|
CP0398823
|
3-(3-chlorophenylsulfonyl)-N-(pyridin-3-ylmethyl)thieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-amine
Show/Hide
|
C19H13ClN6O2S2
|
3
|
| 1 |
IC50 = 31.7 nM
|
|
|
| 2 |
IC50 = 1250 nM
|
|
|
| 3 |
Ki = 14.7 nM
|
|
|
|
CP0406029
|
10-(benzenesulfonyl)-N-[(2-chlorophenyl)methyl]-5-thia-1,8,11,12-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaen-7-amine
Show/Hide
|
C20H14ClN5O2S2
|
1
|
| 1 |
IC50 = 32 nM
|
|
|
|
CP0343626
|
3-(4-bromophenylsulfonyl)-N-isopentylthieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-amine
Show/Hide
|
C18H18BrN5O2S2
|
2
|
| 1 |
IC50 = 34.3 nM
|
|
|
| 2 |
Ki = 15.9 nM
|
|
|
|
CP0406030
|
10-(benzenesulfonyl)-N-(1-phenylethyl)-5-thia-1,8,11,12-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaen-7-amine
Show/Hide
|
C21H17N5O2S2
|
1
|
| 1 |
IC50 = 37 nM
|
|
|
|
CP0153460
|
2-(5-chloro-2-methyl-1H-indol-3-yl)-N,N-dimethylethanamine
Show/Hide
|
C13H17ClN2
|
1
|
| 1 |
IC50 = 40 nM
|
|
|
|
CP0392119
|
5-Chloro-2-methyl-3-(8-methyl-8-aza-bicyclo[3.2.1]oct-2-en-3-yl)-1H-indole
Show/Hide
|
C17H19ClN2
|
1
|
| 1 |
IC50 = 40 nM
|
|
|
|
CP0493361
|
5-Chloro-2-propyl-3-(1,2,3,6-tetrahydro-pyridin-4-yl)-1H-indole
Show/Hide
|
C16H19ClN2
|
1
|
| 1 |
IC50 = 40 nM
|
|
|
|
CP0957814
|
5-Chloro-1,2-dimethyl-3-(1,2,3,6-tetrahydropyridin-4-yl)-1H-indole
Show/Hide
|
C15H17ClN2
|
1
|
| 1 |
IC50 = 40 nM
|
|
|
|
CP0379950
|
2-methyl-1-(naphthalen-2-ylsulfonyl)-5-(piperazin-1-yl)-2,3-dihydroquinolin-4(1H)-one
Show/Hide
|
C24H25N3O3S
|
1
|
| 1 |
IC50 = 42 nM
|
|
|
|
CP0408043
|
(R)-2-methyl-7-(4-methylpiperazin-1-yl)-1-(naphthalen-2-ylsulfonyl)-2,3-dihydroquinolin-4(1H)-one
Show/Hide
|
C25H27N3O3S
|
1
|
| 1 |
IC50 = 43 nM
|
|
|
|
CP0437392
|
3-(4-fluorophenyl)sulfonyl-N-methylpyrazolo[1,5-a]pyrimidin-2-amine
Show/Hide
|
C13H11FN4O2S
|
2
|
| 1 |
IC50 = 45 nM
|
|
|
| 2 |
Ki = 11.75 nM
|
|
|
|
CP0465488
|
US8618114, 1.2.22(3).HCl
Show/Hide
|
C17H21N5O2S
|
2
|
| 1 |
IC50 = 45 nM
|
|
|
| 2 |
Ki = 1.38 nM
|
|
|
|
CP0406028
|
3-(3,4-dimethylphenylsulfonyl)-N-isopentylthieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-amine
Show/Hide
|
C20H23N5O2S2
|
1
|
| 1 |
IC50 = 46 nM
|
|
|
|
CP0505185
|
7-methyl-5-(4-methylpiperazin-1-yl)-1-(naphthalen-2-ylsulfonyl)-2,3-dihydroquinolin-4(1H)-one
Show/Hide
|
C25H27N3O3S
|
1
|
| 1 |
IC50 = 47 nM
|
|
|
|
CP0514268
|
3-(1-Butyl-1,2,3,6-tetrahydro-pyridin-4-yl)-5-chloro-2-methyl-1H-indole
Show/Hide
|
C18H23ClN2
|
1
|
| 1 |
IC50 = 50 nM
|
|
|
|
CP0671078
|
[2-Methyl-3-(1,2,3,6-tetrahydropyridin-4-yl)-1H-indol-5-yl]trifluoromethanesulfonate
Show/Hide
|
C15H15F3N2O3S
|
1
|
| 1 |
IC50 = 50 nM
|
|
|
|
CP0529057
|
US8618114, 1.2(1)
Show/Hide
|
C15H15ClN4O2S
|
1
|
| 1 |
IC50 = 52 nM
|
|
|
|
CP0485779
|
US8618114, 1.2.22(14).HCl
Show/Hide
|
C17H20FN5O2S
|
1
|
| 1 |
IC50 = 56.4 nM
|
|
|
|
CP0522767
|
10-(benzenesulfonyl)-N-(3,5-dimethyladamantan-1- yl)-5-thia-1,8,11,12- tetraazatricyclo[7.3.0.0^{2,6}]dodeca- 2(6),3,7,9,11-pentaen-7-amine
Show/Hide
|
C25H27N5O2S2
|
2
|
| 1 |
IC50 = 56.7 nM
|
|
|
| 2 |
Ki = 26.3 nM
|
|
|
|
CP0543853
|
7-bromo-5-(4-methylpiperazin-1-yl)-1-(naphthalen-2-ylsulfonyl)-2,3-dihydroquinolin-4(1H)-one
Show/Hide
|
C24H24BrN3O3S
|
1
|
| 1 |
IC50 = 58 nM
|
|
|
|
CP0504465
|
10-(benzenesulfonyl)-N-benzyl-5-thia-1,8,11,12-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaen-7-amine
Show/Hide
|
C20H15N5O2S2
|
1
|
| 1 |
IC50 = 59 nM
|
|
|
|
CP0514267
|
5-Chloro-2-methyl-3-(1-propyl-1,2,3,6-tetrahydro-pyridin-4-yl)-1H-indole
Show/Hide
|
C17H21ClN2
|
1
|
| 1 |
IC50 = 60 nM
|
|
|
|
CP0506203
|
N-butyl-10-(3-chlorophenyl)sulfonyl-5-thia-1,8,11,12-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaen-7-amine
Show/Hide
|
C17H16ClN5O2S2
|
1
|
| 1 |
IC50 = 60 nM
|
|
|
|
CP0408045
|
5-(N-methyl-piperazin-1-yl)-1-(naphthalene-2-sulfonyl)-2,3-dihydro-1H-quinolin-4-one
Show/Hide
|
C24H25N3O3S
|
1
|
| 1 |
IC50 = 61 nM
|
|
|
|
CP0238991
|
N-(1,3-benzodioxol-5-ylmethyl)-10-(4-bromophenyl)sulfonyl-5-thia-1,8,11,12-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaen-7-amine
Show/Hide
|
C21H14BrN5O4S2
|
2
|
| 1 |
IC50 = 62.1 nM
|
|
|
| 2 |
Ki = 28.8 nM
|
|
|
|
CP0406033
|
10-(benzenesulfonyl)-N-propan-2-yl-5-thia-1,8,11,12-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaen-7-amine
Show/Hide
|
C16H15N5O2S2
|
3
|
| 1 |
IC50 = 65 nM
|
|
|
| 2 |
IC50 = 370 nM
|
|
|
| 3 |
Ki = 30.2 nM
|
|
|
|
CP0523836
|
3-(3-chlorophenylsulfonyl)-N-isopentylthieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-amine
Show/Hide
|
C18H18ClN5O2S2
|
1
|
| 1 |
IC50 = 68 nM
|
|
|
|
CP0406026
|
10-(benzenesulfonyl)-N-butyl-5-thia-1,8,11,12-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaen-7-amine
Show/Hide
|
C17H17N5O2S2
|
1
|
| 1 |
IC50 = 69 nM
|
|
|
|
CP0509334
|
3-(3-chlorophenylsulfonyl)-N-cyclohexylthieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-amine
Show/Hide
|
C19H18ClN5O2S2
|
1
|
| 1 |
IC50 = 69 nM
|
|
|
|
CP0393498
|
5-Chloro-2-ethyl-3-(1-ethyl-1,2,3,6-tetrahydro-pyridin-4-yl)-1H-indole
Show/Hide
|
C17H21ClN2
|
1
|
| 1 |
IC50 = 70 nM
|
|
|
|
CP0539526
|
[3-(benzenesulfonyl)-5-methyl-2-methylsulfanylpyrazolo[1,5-a]pyrimidin-7-yl]methanol
Show/Hide
|
C15H15N3O3S2
|
2
|
| 1 |
IC50 = 73 nM
|
|
|
| 2 |
Ki = 0.5623 nM
|
|
|
|
CP0381512
|
3-(benzenesulfonyl)-N-methylpyrazolo[1,5-a]pyrimidin-2-amine
Show/Hide
|
C13H12N4O2S
|
2
|
| 1 |
IC50 = 76 nM
|
|
|
| 2 |
Ki = 3.89 nM
|
|
|
|
CP0647677
|
2,5-Dimethyl-8-(phenylsulfonyl)-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole hydrochloride
Show/Hide
|
C19H21ClN2O2S
|
1
|
| 1 |
IC50 = 78 nM
|
|
|
|
CP0560639
|
US8618114, 1.2.22(4).HCl
Show/Hide
|
C18H23N5O2S
|
1
|
| 1 |
IC50 = 78 nM
|
|
|
|
CP0056774
|
5-Methoxy-3-(1,2,3,6-tetrahydro-pyridin-4-yl)-1H-indole(RU-24969)
Show/Hide
|
C14H16N2O
|
1
|
| 1 |
IC50 = 79 nM
|
|
|
|
CP0099428
|
5-Methoxy-2-methyl-3-(1,2,3,6-tetrahydro-pyridin-4-yl)-1H-indole
Show/Hide
|
C15H18N2O
|
1
|
| 1 |
IC50 = 80 nM
|
|
|
|
CP0962765
|
5-Chloro-2-methyl-1-propyl-3-(1,2,3,6-tetrahydropyridin-4-yl)-1H-indole
Show/Hide
|
C17H21ClN2
|
1
|
| 1 |
IC50 = 80 nM
|
|
|
|
CP0080534
|
2-ethyl-5-methoxy-N,N-dimethyltryptamine
Show/Hide
|
C15H22N2O
|
3
|
| 1 |
IC50 = 85 nM
|
|
|
| 2 |
Ki = 16 nM
|
|
|
| 3 |
Ki = 52 nM
|
|
|
|
CP0494231
|
8-[(3-Fluorophenyl)sulfonyl]-2-methyl-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
Show/Hide
|
C18H17FN2O2S
|
1
|
| 1 |
IC50 = 85 nM
|
|
|
|
CP0150364
|
2,8-Dimethyl-5-((Z)-styryl)-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
Show/Hide
|
C21H22N2
|
1
|
| 1 |
IC50 = 87 nM
|
|
|
|
CP0392116
|
2-Ethyl-5-methoxy-3-(1,2,3,6-tetrahydro-pyridin-4-yl)-1H-indole
Show/Hide
|
C16H20N2O
|
1
|
| 1 |
IC50 = 90 nM
|
|
|
|
CP0487883
|
3-(3,4-dimethylphenylsulfonyl)-N-(thiophen-2-ylmethyl)thieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-amine
Show/Hide
|
C20H17N5O2S3
|
1
|
| 1 |
IC50 = 90 nM
|
|
|
|
CP0373093
|
2-Methylsulfanyl-3-phenylsulfonyl-5,6,7,8-tetrahydro-pyrazolo[5,1-b]quinazoline
Show/Hide
|
C17H17N3O2S2
|
2
|
| 1 |
IC50 = 98.5 nM
|
|
|
| 2 |
IC50 = 479 nM
|
|
|
|
CP0475431
|
3-(2,5-Dimethylphenylsulfonyl)thieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-amine
Show/Hide
|
C15H13N5O2S2
|
3
|
| 1 |
IC50 = 99.1 nM
|
|
|
| 2 |
IC50 = 1220 nM
|
|
|
| 3 |
Ki = 46 nM
|
|
|
|
CP0483652
|
5-Chloro-2-isopropyl-3-(1,2,3,6-tetrahydro-pyridin-4-yl)-1H-indole
Show/Hide
|
C16H19ClN2
|
1
|
| 1 |
IC50 = 100 nM
|
|
|
|
CP0886832
|
5-Chloro-1-ethyl-2-methyl-3-(1,2,3,6-tetrahydropyridin-4-yl)-1H-indole
Show/Hide
|
C16H19ClN2
|
1
|
| 1 |
IC50 = 100 nM
|
|
|
|
CP0898488
|
5-Isopropoxy-2-methyl-3-(1,2,3,6-tetrahydropyridin-4-yl)-1H-indole
Show/Hide
|
C17H22N2O
|
1
|
| 1 |
IC50 = 100 nM
|
|
|
|
CP0529058
|
3-(benzenesulfonyl)-7-(methoxymethyl)-N,5-dimethylpyrazolo[1,5-a]pyrimidin-2-amine
Show/Hide
|
C16H18N4O3S
|
2
|
| 1 |
IC50 = 101 nM
|
|
|
| 2 |
Ki = 7.586 nM
|
|
|
|
CP0523837
|
3-(3-chlorophenylsulfonyl)-N-(2-methoxyethyl)thieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-amine
Show/Hide
|
C16H14ClN5O3S2
|
1
|
| 1 |
IC50 = 110 nM
|
|
|
|
CP0509722
|
N-[(3-chlorophenyl)methyl]-10-(4-methylphenyl)sulfonyl-5-thia-1,8,11,12-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaen-7-amine
Show/Hide
|
C21H16ClN5O2S2
|
1
|
| 1 |
IC50 = 120 nM
|
|
|
|
CP0466805
|
5-(4-methylpiperazin-1-yl)-1-tosyl-2,3-dihydroquinolin-4(1H)-one
Show/Hide
|
C21H25N3O3S
|
1
|
| 1 |
IC50 = 129 nM
|
|
|
|
CP0507520
|
3-(3-chlorophenylsulfonyl)-N-cycloheptylthieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-amine
Show/Hide
|
C20H20ClN5O2S2
|
1
|
| 1 |
IC50 = 140 nM
|
|
|
|
CP0475404
|
3-(3-chlorophenylsulfonyl)-N-(3-methoxypropyl)thieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-amine
Show/Hide
|
C17H16ClN5O3S2
|
1
|
| 1 |
IC50 = 150 nM
|
|
|
|
CP0489488
|
3-(3-chlorophenylsulfonyl)-N-(1-phenylethyl)thieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-amine
Show/Hide
|
C21H16ClN5O2S2
|
1
|
| 1 |
IC50 = 150 nM
|
|
|
|
CP0509725
|
3-(3-chlorophenylsulfonyl)-N-(thiophen-2-ylmethyl)thieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-amine
Show/Hide
|
C18H12ClN5O2S3
|
1
|
| 1 |
IC50 = 150 nM
|
|
|
|
CP0472403
|
US8618114, 1.1.3(5)
Show/Hide
|
C14H11ClFN3O2S2
|
1
|
| 1 |
IC50 = 156 nM
|
|
|
|
CP0237538
|
2,8-Dimethyl-5-phenethyl-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
Show/Hide
|
C21H24N2
|
1
|
| 1 |
IC50 = 158 nM
|
|
|
|
CP0405290
|
6-methoxy-7-(4-methylpiperazin-1-yl)-1-(naphthalen-2-ylsulfonyl)-2,3-dihydroquinolin-4(1H)-one
Show/Hide
|
C25H27N3O4S
|
1
|
| 1 |
IC50 = 165 nM
|
|
|
|
CP0497226
|
3-(3-chlorophenylsulfonyl)-N-cyclopentylthieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-amine
Show/Hide
|
C18H16ClN5O2S2
|
1
|
| 1 |
IC50 = 170 nM
|
|
|
|
CP0509328
|
3-(2,5-dimethylphenylsulfonyl)-N-(1-phenylethyl)thieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-amine
Show/Hide
|
C23H21N5O2S2
|
1
|
| 1 |
IC50 = 170 nM
|
|
|
|
CP0523845
|
10-(benzenesulfonyl)-N-cycloheptyl-5-thia-1,8,11,12-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaen-7-amine
Show/Hide
|
C20H21N5O2S2
|
1
|
| 1 |
IC50 = 170 nM
|
|
|
|
CP0431339
|
US8618114, 1.2.12(4).HCl
Show/Hide
|
C19H24N6O2S
|
2
|
| 1 |
IC50 = 173 nM
|
|
|
| 2 |
Ki = 4.365 nM
|
|
|
|
CP0516421
|
[3-(benzenesulfonyl)-7-methyl-2-methylsulfanylpyrazolo[1,5-a]pyrimidin-5-yl]methanol
Show/Hide
|
C15H15N3O3S2
|
2
|
| 1 |
IC50 = 177 nM
|
|
|
| 2 |
Ki = 2.138 nM
|
|
|
|
CP0218398
|
6-[5-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]pentanoyl]-1-azatricyclo[6.3.1.04,12]dodeca-4,6,8(12)-trien-11-one
Show/Hide
|
C28H30FN3O3
|
1
|
| 1 |
IC50 = 177.6 nM
|
|
|
|
CP0430390
|
25-[(Z)-2-(4-Fluorophenyl)vinyl]-2,8-dimethyl-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
Show/Hide
|
C21H21FN2
|
1
|
| 1 |
IC50 = 180 nM
|
|
|
|
CP0124918
|
10-(4-methylphenyl)sulfonyl-N-(1-phenylethyl)-5-thia-1,8,11,12-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaen-7-amine
Show/Hide
|
C22H19N5O2S2
|
1
|
| 1 |
IC50 = 180 nM
|
|
|
|
CP0465480
|
3-(3-chloro-4-fluorophenyl)sulfonyl-5-methyl-2-methylsulfanylpyrazolo[1,5-a]pyrimidine
Show/Hide
|
C14H11ClFN3O2S2
|
2
|
| 1 |
IC50 = 187 nM
|
|
|
| 2 |
Ki = 7.943 nM
|
|
|
|
CP0377174
|
3-(Phenylsulfonyl)-5-pyrrolidin-1-ylthieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidine
Show/Hide
|
C17H15N5O2S2
|
2
|
| 1 |
IC50 = 188 nM
|
|
|
| 2 |
Ki = 87.5 nM
|
|
|
|
CP0502401
|
10-(benzenesulfonyl)-N-(2-methoxyethyl)-5-thia-1,8,11,12-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaen-7-amine
Show/Hide
|
C16H15N5O3S2
|
1
|
| 1 |
IC50 = 190 nM
|
|
|
|
CP0509332
|
3-(3-chlorophenylsulfonyl)-N-(furan-2-ylmethyl)thieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-amine
Show/Hide
|
C18H12ClN5O3S2
|
1
|
| 1 |
IC50 = 190 nM
|
|
|
|
CP0495047
|
US8618114, 1.1.12(5)
Show/Hide
|
C18H21N5O3S
|
2
|
| 1 |
IC50 = 197 nM
|
|
|
| 2 |
Ki = 16.6 nM
|
|
|
|
CP0055690
|
2-methyl-3-(1,2,3,6-tetrahydropyridin-4-yl)-1H-indole
Show/Hide
|
C14H16N2
|
1
|
| 1 |
IC50 = 200 nM
|
|
|
|
CP0522765
|
10-(4-methylphenyl)sulfonyl-N-(thiophen-2-ylmethyl)-5-thia-1,8,11,12-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaen-7-amine
Show/Hide
|
C19H15N5O2S3
|
1
|
| 1 |
IC50 = 220 nM
|
|
|
|
CP0475430
|
N-[1-(1-adamantyl)ethyl]-10-(benzenesulfonyl)-5-thia-1,8,11,12-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaen-7-amine
Show/Hide
|
C25H27N5O2S2
|
2
|
| 1 |
IC50 = 221 nM
|
|
|
| 2 |
Ki = 103 nM
|
|
|
|
CP0377171
|
10-(4-methylphenyl)sulfonyl-N-(oxolan-2-ylmethyl)-5-thia-1,8,11,12-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaen-7-amine
Show/Hide
|
C19H19N5O3S2
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1
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| 1 |
IC50 = 250 nM
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CP0386507
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3-(phenylsulfonyl)-N-(pyridin-3-ylmethyl)thieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-amine
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C19H14N6O2S2
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2
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| 1 |
IC50 = 260 nM
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| 2 |
IC50 > 30 nM
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CP0504461
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10-(benzenesulfonyl)-N-(3-methoxypropyl)-5-thia-1,8,11,12-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaen-7-amine
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C17H17N5O3S2
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1
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| 1 |
IC50 = 260 nM
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CP0523839
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N-benzyl-10-(4-methylphenyl)sulfonyl-5-thia-1,8,11,12-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaen-7-amine
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C21H17N5O2S2
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1
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| 1 |
IC50 = 260 nM
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CP0487881
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N-benzyl-10-(4-chlorophenyl)sulfonyl-5-thia-1,8,11,12-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaen-7-amine
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C20H14ClN5O2S2
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1
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| 1 |
IC50 = 270 nM
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CP0353494
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2,8-Dimethyl-5-(2-p-tolylethyl)-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
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C22H26N2
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1
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| 1 |
IC50 = 276 nM
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CP0487882
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3-(4-chlorophenylsulfonyl)-N-(1-phenylethyl)thieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-amine
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C21H16ClN5O2S2
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1
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| 1 |
IC50 = 280 nM
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CP0489485
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10-(benzenesulfonyl)-N-[(2-methoxyphenyl)methyl]-5-thia-1,8,11,12-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaen-7-amine
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C21H17N5O3S2
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1
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| 1 |
IC50 = 290 nM
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CP0509325
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10-(benzenesulfonyl)-N-(1,3-benzodioxol-5-ylmethyl)-5-thia-1,8,11,12-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaen-7-amine
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C21H15N5O4S2
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1
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| 1 |
IC50 = 290 nM
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CP0392115
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2-Ethyl-5-methoxy-3-piperidin-4-yl-1H-indole
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C16H22N2O
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1
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| 1 |
IC50 = 300 nM
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CP0454586
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N-benzyl-N-ethyl-10-(4-methylphenyl)sulfonyl-5-thia-1,8,11,12-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaen-7-amine
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C23H21N5O2S2
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1
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| 1 |
IC50 = 300 nM
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CP0564042
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US8618114, 1.1(4)
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C15H14ClN3O2S2
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1
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| 1 |
IC50 = 300 nM
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CP0529163
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6-(N-methyl-piperazin-1-yl)-1-(naphthalene-2-sulfonyl)-2,3-dihydro-1H-quinolin-4-one
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C24H25N3O3S
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1
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| 1 |
IC50 = 311 nM
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CP0539245
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US8618114, 1.2.9(7)
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C19H17N5O2S
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1
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| 1 |
IC50 = 341 nM
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CP0323299
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N-cycloheptyl-10-(3,4-dimethylphenyl)sulfonyl-5-thia-1,8,11,12-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaen-7-amine
Show/Hide
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C22H25N5O2S2
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1
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| 1 |
IC50 = 350 nM
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CP0466768
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(R)-2-methyl-5-(4-methylpiperazin-1-yl)-1-(naphthalen-2-ylsulfonyl)-2,3-dihydroquinolin-4(1H)-one
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C25H27N3O3S
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1
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| 1 |
IC50 = 353 nM
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CP0398761
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N,N-dimethyl-N'-[5-[(4-methylphenyl)sulfonylamino]-1,2-benzothiazol-3-yl]methanimidamide
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C17H18N4O2S2
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1
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| 1 |
IC50 = 360 nM
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CP0375182
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2,8-dimethyl-5-(2-(pyridin-4-yl)ethyl)-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
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C20H23N3
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1
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| 1 |
IC50 = 370 nM
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CP0509726
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3-(4-chlorophenylsulfonyl)-N-(furan-2-ylmethyl)thieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-amine
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C18H12ClN5O3S2
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1
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| 1 |
IC50 = 410 nM
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CP0472401
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3-(benzenesulfonyl)-5-(methoxymethyl)-7-methyl-2-methylsulfanylpyrazolo[1,5-a]pyrimidine
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C16H17N3O3S2
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2
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| 1 |
IC50 = 414 nM
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| 2 |
Ki = 3.236 nM
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CP0529164
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1-(5-chloro-3-methylbenzo[b]thiophen-2-ylsulfonyl)-7-(4-methylpiperazin-1-yl)-2,3-dihydroquinolin-4(1H)-one
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C23H24ClN3O3S2
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1
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| 1 |
IC50 = 419 nM
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CP0398638
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N-propan-2-yl-N-(6-pyridin-3-yloxypyridin-3-yl)naphthalene-2-sulfonamide
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C23H21N3O3S
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1
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| 1 |
IC50 = 422 nM
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CP0501165
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2,8-dimethyl-5-(2-(pyridin-3-yl)ethyl)-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
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C20H23N3
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1
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| 1 |
IC50 = 440 nM
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CP0544233
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3-(benzenesulfonyl)-5-methyl-2-methylsulfanylpyrazolo[1,5-a]pyrimidine
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C14H13N3O2S2
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2
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| 1 |
IC50 = 450 nM
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| 2 |
Ki = 16.6 nM
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CP0468668
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3-(3-chlorophenylsulfonyl)-N-isopropylthieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-amine
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C16H14ClN5O2S2
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1
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| 1 |
IC50 = 470 nM
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CP0523842
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3-(3,4-dimethylphenylsulfonyl)-N-(2-methoxybenzyl)thieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-amine
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C23H21N5O3S2
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1
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| 1 |
IC50 = 470 nM
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CP0503521
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3-(3-chlorophenyl)sulfonyl-2-methylsulfanylpyrazolo[1,5-a]pyrimidine
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C13H10ClN3O2S2
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2
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| 1 |
IC50 = 473 nM
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| 2 |
Ki = 15.14 nM
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CP0386509
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3-(4-chlorophenylsulfonyl)-N-((tetrahydrofuran-2-yl)methyl)thieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-amine
Show/Hide
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C18H16ClN5O3S2
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1
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| 1 |
IC50 = 480 nM
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CP0496037
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3-(3-Chlorophenylsulfonyl)-N-(4-fluorobenzyl)thieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-amine
Show/Hide
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C20H13ClFN5O2S2
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1
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| 1 |
IC50 = 480 nM
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CP0386508
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10-(benzenesulfonyl)-N-methyl-N-(pyridin-3-ylmethyl)-5-thia-1,8,11,12-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaen-7-amine
Show/Hide
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C20H16N6O2S2
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2
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| 1 |
IC50 = 500 nM
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| 2 |
IC50 > 30 nM
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CP0509331
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N-(furan-2-ylmethyl)-10-(4-methylphenyl)sulfonyl-5-thia-1,8,11,12-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaen-7-amine
Show/Hide
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C19H15N5O3S2
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1
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| 1 |
IC50 = 500 nM
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CP0484903
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US8618114, 1.1(7)
Show/Hide
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C20H18N4O3S2
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1
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| 1 |
IC50 = 514 nM
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CP0113868
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3-(3,4-dimethylphenylsulfonyl)-N-(4-fluorobenzyl)thieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-amine
Show/Hide
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C22H18FN5O2S2
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1
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| 1 |
IC50 = 520 nM
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CP0509327
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3-(4-bromophenylsulfonyl)-N-(1-phenylethyl)thieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-amine
Show/Hide
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C21H16BrN5O2S2
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1
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| 1 |
IC50 = 540 nM
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CP0509723
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N-benzyl-10-(3-chlorophenyl)sulfonyl-N-ethyl-5-thia-1,8,11,12-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaen-7-amine
Show/Hide
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C22H18ClN5O2S2
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1
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| 1 |
IC50 = 540 nM
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CP0446551
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5-[(Z)-2-(4-Methoxyphenyl)vinyl]-2,8-dimethyl-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
Show/Hide
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C22H24N2O
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1
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| 1 |
IC50 = 550 nM
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CP0497225
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N-benzyl-10-(4-chlorophenyl)sulfonyl-N-ethyl-5-thia-1,8,11,12-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaen-7-amine
Show/Hide
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C22H18ClN5O2S2
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1
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| 1 |
IC50 = 570 nM
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CP0386506
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N-[(2-methoxyphenyl)methyl]-10-(4-methylphenyl)sulfonyl-5-thia-1,8,11,12-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaen-7-amine
Show/Hide
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C22H19N5O3S2
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1
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| 1 |
IC50 = 580 nM
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CP0496036
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N'-[10-(3-chlorophenyl)sulfonyl-5-thia-1,8,11,12-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaen-7-yl]-N,N,N'-trimethylethane-1,2-diamine
Show/Hide
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C18H19ClN6O2S2
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1
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| 1 |
IC50 = 580 nM
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CP0496039
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N-benzyl-10-(4-bromophenyl)sulfonyl-N-ethyl-5-thia-1,8,11,12-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaen-7-amine
Show/Hide
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C22H18BrN5O2S2
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1
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| 1 |
IC50 = 580 nM
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CP0502402
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N-(3-methylbutyl)-10-(4-methylphenyl)sulfonyl-5-thia-1,8,11,12-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaen-7-amine
Show/Hide
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C19H21N5O2S2
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1
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| 1 |
IC50 = 580 nM
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CP0473045
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N-cyclopentyl-10-(2,5-dimethylphenyl)sulfonyl-5-thia-1,8,11,12-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaen-7-amine
Show/Hide
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C20H21N5O2S2
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1
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| 1 |
IC50 = 590 nM
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CP0489491
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3-(4-isopropylphenylsulfonyl)-N-m-tolylthieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-amine
Show/Hide
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C23H21N5O2S2
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1
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| 1 |
IC50 = 590 nM
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CP0507522
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N-(2,3-dimethylphenyl)-10-(4-methylphenyl)sulfonyl-5-thia-1,8,11,12-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaen-7-amine
Show/Hide
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C22H19N5O2S2
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1
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| 1 |
IC50 = 590 nM
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CP0493362
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3-(1-Benzyl-1,2,3,6-tetrahydro-pyridin-4-yl)-5-chloro-2-methyl-1H-indole
Show/Hide
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C21H21ClN2
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1
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| 1 |
IC50 = 600 nM
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CP0406032
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N-[(2-chlorophenyl)methyl]-10-(3,4-dimethylphenyl)sulfonyl-5-thia-1,8,11,12-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaen-7-amine
Show/Hide
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C22H18ClN5O2S2
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1
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| 1 |
IC50 = 600 nM
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CP0509336
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10-(benzenesulfonyl)-N-(4-fluorophenyl)-5-thia-1,8,11,12-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaen-7-amine
Show/Hide
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C19H12FN5O2S2
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1
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| 1 |
IC50 = 600 nM
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CP0406027
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3-(4-Bromophenylsulfonyl)thieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-amine
Show/Hide
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C13H8BrN5O2S2
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1
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| 1 |
IC50 = 610 nM
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CP0917036
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2-Methyl-8-(phenylsulfonyl)-5-(2-pyridin-2-ylethyl)-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole hydrochloride
Show/Hide
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C25H26ClN3O2S
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1
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| 1 |
IC50 = 620 nM
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CP0417858
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N-[3-(4-methylpiperazin-1-yl)phenyl]-N-propan-2-ylbenzenesulfonamide
Show/Hide
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C20H27N3O2S
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1
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| 1 |
IC50 = 644 nM
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CP0509333
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3-(4-chlorophenylsulfonyl)-N-(thiophen-2-ylmethyl)thieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-amine
Show/Hide
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C18H12ClN5O2S3
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1
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| 1 |
IC50 = 650 nM
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CP0439140
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5-[2-(4-Methoxyphenyl)ethyl]-2,8-dimethyl-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
Show/Hide
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C22H26N2O
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1
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| 1 |
IC50 = 666 nM
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CP0475425
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3-(2,5-dimethylphenylsulfonyl)-N-phenethylthieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-amine
Show/Hide
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C23H21N5O2S2
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1
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| 1 |
IC50 = 670 nM
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CP0504464
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3-(3,4-dimethylphenylsulfonyl)-N-(1-phenylpropan-2-yl)thieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-amine
Show/Hide
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C24H23N5O2S2
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1
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| 1 |
IC50 = 680 nM
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CP0217439
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10-(benzenesulfonyl)-N-[(4-fluorophenyl)methyl]-5-thia-1,8,11,12-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaen-7-amine
Show/Hide
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C20H14FN5O2S2
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1
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| 1 |
IC50 = 690 nM
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CP0509322
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3-(3-Chlorophenylsulfonyl)thieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-amine
Show/Hide
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C13H8ClN5O2S2
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1
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| 1 |
IC50 = 690 nM
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CP0446549
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8-Fluoro-2-methyl-5-phenethyl-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
Show/Hide
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C20H21FN2
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1
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| 1 |
IC50 = 692 nM
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CP0671077
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2-Methyl-3-(1,2,3,6-tetrahydropyridin-4-yl)-5-(3-thienyl)-1H-indole
Show/Hide
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C18H18N2S
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1
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| 1 |
IC50 = 700 nM
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CP0475426
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3-(2,5-dimethylphenylsulfonyl)-N-(thiophen-2-ylmethyl)thieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-amine
Show/Hide
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C20H17N5O2S3
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1
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| 1 |
IC50 = 710 nM
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CP0539528
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US8618114, 1.2(4)
Show/Hide
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C23H18N6O2S
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1
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| 1 |
IC50 = 723 nM
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CP0111211
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N-cyclohexyl-10-(4-methylphenyl)sulfonyl-5-thia-1,8,11,12-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaen-7-amine
Show/Hide
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C20H21N5O2S2
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1
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| 1 |
IC50 = 730 nM
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CP0345250
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N-[(4-fluorophenyl)methyl]-10-(4-methylphenyl)sulfonyl-5-thia-1,8,11,12-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaen-7-amine
Show/Hide
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C21H16FN5O2S2
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1
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| 1 |
IC50 = 740 nM
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CP0523850
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3-(3-chlorophenylsulfonyl)-N-(2,5-dimethylphenyl)thieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-amine
Show/Hide
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C21H16ClN5O2S2
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1
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| 1 |
IC50 = 740 nM
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CP0379359
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N'-[(E)-[1-(4-methoxyphenyl)sulfonyl-4-nitroindol-3-yl]methylideneamino]-N,N-dimethylmethanimidamide
Show/Hide
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C19H19N5O5S
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1
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| 1 |
IC50 = 740 nM
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CP0506204
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3-(3,4-dimethylphenylsulfonyl)-N-isopropylthieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-amine
Show/Hide
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C18H19N5O2S2
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1
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| 1 |
IC50 = 750 nM
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CP0507519
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3-(3,4-dimethylphenylsulfonyl)-N-(furan-2-ylmethyl)thieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-amine
Show/Hide
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C20H17N5O3S2
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1
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| 1 |
IC50 = 770 nM
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CP0406031
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3-(3-chlorophenylsulfonyl)-N-(2-methoxybenzyl)thieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-amine
Show/Hide
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C21H16ClN5O3S2
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1
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| 1 |
IC50 = 780 nM
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CP0935322
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N'-[3-(3-Chlorophenylsulfonyl)thieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-yl]-N,N-dimethylethane-1,2-diamine dihydrochloride
Show/Hide
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C18H22Cl4N6O2S2
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1
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| 1 |
IC50 = 780 nM
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CP0509728
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N-cycloheptyl-10-(4-methylphenyl)sulfonyl-5-thia-1,8,11,12-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaen-7-amine
Show/Hide
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C21H23N5O2S2
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1
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| 1 |
IC50 = 790 nM
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CP0489494
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3-(4-chlorophenylsulfonyl)-N-(2,3-dimethylphenyl)thieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-amine
Show/Hide
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C21H16ClN5O2S2
|
1
|
| 1 |
IC50 = 800 nM
|
|
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CP0475427
|
3-(phenylsulfonyl)-N-(3-(trifluoromethyl)phenyl)thieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-amine
Show/Hide
|
C20H12F3N5O2S2
|
1
|
| 1 |
IC50 = 820 nM
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|
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CP0509323
|
3-(3-chlorophenylsulfonyl)-N-phenethylthieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-amine
Show/Hide
|
C21H16ClN5O2S2
|
1
|
| 1 |
IC50 = 820 nM
|
|
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CP0509335
|
N-cyclohexyl-10-(3,4-dimethylphenyl)sulfonyl-5-thia-1,8,11,12-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaen-7-amine
Show/Hide
|
C21H23N5O2S2
|
1
|
| 1 |
IC50 = 820 nM
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|
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CP0468671
|
3-(2,5-dimethylphenylsulfonyl)-N-(2-methoxyethyl)thieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-amine
Show/Hide
|
C18H19N5O3S2
|
1
|
| 1 |
IC50 = 860 nM
|
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CP0497223
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3-(2,5-dimethylphenylsulfonyl)-N-isopentylthieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-amine
Show/Hide
|
C20H23N5O2S2
|
1
|
| 1 |
IC50 = 860 nM
|
|
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CP0509730
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3-(3,4-dimethylphenylsulfonyl)-N-(3-methoxyphenyl)thieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-amine
Show/Hide
|
C22H19N5O3S2
|
1
|
| 1 |
IC50 = 860 nM
|
|
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CP0494107
|
2,8-dimethyl-5-(2-(pyridin-2-yl)ethyl)-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
Show/Hide
|
C20H23N3
|
1
|
| 1 |
IC50 = 860 nM
|
|
|
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CP0520949
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N'-[10-(benzenesulfonyl)-5-thia-1,8,11,12-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaen-7-yl]-N,N,N'-trimethylethane-1,2-diamine
Show/Hide
|
C18H20N6O2S2
|
2
|
| 1 |
IC50 = 870 nM
|
|
|
| 2 |
IC50 > 300 nM
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CP0017601
|
2,8-dimethyl-5-[2-(6-methylpyridin-3-yl)ethyl]-3,4-dihydro-1H-pyrido[4,3-b]indole
Show/Hide
|
C21H25N3
|
2
|
| 1 |
IC50 = 890 nM
|
|
|
| 2 |
IC50 = 1160 nM
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|
|
|
CP0377172
|
3-(2,5-dimethylphenylsulfonyl)-N-((tetrahydrofuran-2-yl)methyl)thieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-amine
Show/Hide
|
C20H21N5O3S2
|
1
|
| 1 |
IC50 = 890 nM
|
|
|
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CP0507523
|
3-(4-isopropylphenylsulfonyl)-N-(3-methoxyphenyl)thieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-amine
Show/Hide
|
C23H21N5O3S2
|
1
|
| 1 |
IC50 = 900 nM
|
|
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CP0492828
|
2,8-Dimethyl-5-((Z)-2-p-tolylvinyl)-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
Show/Hide
|
C22H24N2
|
1
|
| 1 |
IC50 = 910 nM
|
|
|
|
CP0500564
|
3-(3-chloro-4-fluorophenyl)sulfonyl-2-methylsulfanylpyrazolo[1,5-a]pyrimidine
Show/Hide
|
C13H9ClFN3O2S2
|
2
|
| 1 |
IC50 = 912 nM
|
|
|
| 2 |
Ki = 44.67 nM
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CP0506207
|
3-(3-chlorophenylsulfonyl)-N-phenylthieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-amine
Show/Hide
|
C19H12ClN5O2S2
|
1
|
| 1 |
IC50 = 920 nM
|
|
|
|
CP0504466
|
3-(4-bromophenylsulfonyl)-N-(2-methoxybenzyl)thieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-amine
Show/Hide
|
C21H16BrN5O3S2
|
1
|
| 1 |
IC50 = 930 nM
|
|
|
|
CP0523835
|
10-(4-methylphenyl)sulfonyl-N-(2-phenylethyl)-5-thia-1,8,11,12-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaen-7-amine
Show/Hide
|
C22H19N5O2S2
|
1
|
| 1 |
IC50 = 960 nM
|
|
|
|
CP0523846
|
3-(4-chlorophenylsulfonyl)-N-cyclohexylthieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-amine
Show/Hide
|
C19H18ClN5O2S2
|
1
|
| 1 |
IC50 = 960 nM
|
|
|
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CP0439139
|
2-Methyl-5-phenethyl-8-trifluoromethyl-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
Show/Hide
|
C21H21F3N2
|
1
|
| 1 |
IC50 = 974 nM
|
|
|
|
CP0510498
|
5-[2-(4-Fluorophenyl)ethyl]-2,8-dimethyl-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
Show/Hide
|
C21H23FN2
|
1
|
| 1 |
IC50 = 977 nM
|
|
|
|
CP0530423
|
US8618114, 1.1.2(2)
Show/Hide
|
C14H12FN3O2S2
|
1
|
| 1 |
IC50 = 996 nM
|
|
|
|
CP0498602
|
8-Fluoro-2-methyl-5-((Z)-styryl)-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
Show/Hide
|
C20H19FN2
|
1
|
| 1 |
IC50 = 1000 nM
|
|
|
|
CP0523848
|
N-(2,3-dimethylphenyl)-10-(4-propan-2-ylphenyl)sulfonyl-5-thia-1,8,11,12-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaen-7-amine
Show/Hide
|
C24H23N5O2S2
|
1
|
| 1 |
IC50 = 1000 nM
|
|
|
|
CP0708856
|
2-Methyl-5-phenyl-3-(1,2,3,6-tetrahydropyridin-4-yl)-1Hindole
Show/Hide
|
C20H20N2
|
1
|
| 1 |
IC50 = 1000 nM
|
|
|
|
CP0484906
|
US8618114, 1.2.9(2)
Show/Hide
|
C18H15N5O2S
|
1
|
| 1 |
IC50 = 1037 nM
|
|
|
|
CP0416634
|
4-(3-(3-chlorophenylsulfonyl)thieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-yl)morpholine
Show/Hide
|
C17H14ClN5O3S2
|
1
|
| 1 |
IC50 = 1040 nM
|
|
|
|
CP0378180
|
8-bromo-2-methyl-5-(2-(pyridin-2-yl)ethyl)-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
Show/Hide
|
C19H20BrN3
|
1
|
| 1 |
IC50 = 1040 nM
|
|
|
|
CP0446548
|
8-Methoxy-2-methyl-5-phenethyl-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
Show/Hide
|
C21H24N2O
|
1
|
| 1 |
IC50 = 1050 nM
|
|
|
|
CP0502404
|
3-(4-ethylphenylsulfonyl)-N-phenethylthieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-amine
Show/Hide
|
C23H21N5O2S2
|
1
|
| 1 |
IC50 = 1050 nM
|
|
|
|
CP0523849
|
3-(3-chlorophenylsulfonyl)-N-(3-(trifluoromethyl)phenyl)thieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-amine
Show/Hide
|
C20H11ClF3N5O2S2
|
1
|
| 1 |
IC50 = 1070 nM
|
|
|
|
CP0468648
|
10-(benzenesulfonyl)-N-(1-phenylpropan-2-yl)-5-thia-1,8,11,12-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaen-7-amine
Show/Hide
|
C22H19N5O2S2
|
1
|
| 1 |
IC50 = 1080 nM
|
|
|
|
CP0509724
|
N-benzyl-10-(2,5-dimethylphenyl)sulfonyl-N-ethyl-5-thia-1,8,11,12-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaen-7-amine
Show/Hide
|
C24H23N5O2S2
|
1
|
| 1 |
IC50 = 1100 nM
|
|
|
|
CP0472464
|
N-(3,4-dimethylphenyl)-10-(4-propan-2-ylphenyl)sulfonyl-5-thia-1,8,11,12-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaen-7-amine
Show/Hide
|
C24H23N5O2S2
|
1
|
| 1 |
IC50 = 1110 nM
|
|
|
|
CP0511784
|
3-(benzenesulfonyl)-7-methyl-2-methylsulfanylpyrazolo[1,5-a]pyrimidine
Show/Hide
|
C14H13N3O2S2
|
2
|
| 1 |
IC50 = 1110 nM
|
|
|
| 2 |
Ki = 22.91 nM
|
|
|
|
CP0523832
|
3-(3-chlorophenylsulfonyl)-5-(4-methylpiperidin-1-yl)thieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidine
Show/Hide
|
C19H18ClN5O2S2
|
1
|
| 1 |
IC50 = 1120 nM
|
|
|
|
CP0513315
|
8-Fluoro-5-[2-(4-fluorophenyl)ethyl]-2-methyl-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
Show/Hide
|
C20H20F2N2
|
1
|
| 1 |
IC50 = 1130 nM
|
|
|
|
CP0489493
|
3-(4-chlorophenylsulfonyl)-N-(2-methoxyphenyl)thieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-amine
Show/Hide
|
C20H14ClN5O3S2
|
1
|
| 1 |
IC50 = 1150 nM
|
|
|
|
CP0496038
|
3-(4-chlorophenylsulfonyl)-N-(2-methoxybenzyl)thieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-amine
Show/Hide
|
C21H16ClN5O3S2
|
1
|
| 1 |
IC50 = 1150 nM
|
|
|
|
CP0497222
|
10-(benzenesulfonyl)-N-(2-phenylethyl)-5-thia-1,8,11,12-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaen-7-amine
Show/Hide
|
C21H17N5O2S2
|
1
|
| 1 |
IC50 = 1160 nM
|
|
|
|
CP0487880
|
10-(benzenesulfonyl)-N-[(4-chlorophenyl)methyl]-5-thia-1,8,11,12-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaen-7-amine
Show/Hide
|
C20H14ClN5O2S2
|
1
|
| 1 |
IC50 = 1170 nM
|
|
|
|
CP0503393
|
3-(benzenesulfonyl)-N,N,5,7-tetramethylpyrazolo[1,5-a]pyrimidin-2-amine
Show/Hide
|
C16H18N4O2S
|
2
|
| 1 |
IC50 = 1177 nM
|
|
|
| 2 |
Ki = 14.5 nM
|
|
|
|
CP0398639
|
N-(3-iodophenyl)-N-propan-2-ylnaphthalene-2-sulfonamide
Show/Hide
|
C19H18INO2S
|
1
|
| 1 |
IC50 = 1180 nM
|
|
|
|
CP0509326
|
N-benzyl-10-(4-chlorophenyl)sulfonyl-N-methyl-5-thia-1,8,11,12-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaen-7-amine
Show/Hide
|
C21H16ClN5O2S2
|
1
|
| 1 |
IC50 = 1190 nM
|
|
|
|
CP0377183
|
3-(4-chlorophenylsulfonyl)-N-isopropylthieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-amine
Show/Hide
|
C16H14ClN5O2S2
|
1
|
| 1 |
IC50 = 1200 nM
|
|
|
|
CP0509729
|
3-(3-chlorophenylsulfonyl)-N-p-tolylthieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-amine
Show/Hide
|
C20H14ClN5O2S2
|
1
|
| 1 |
IC50 = 1210 nM
|
|
|
|
CP0509324
|
3-(3-chlorophenylsulfonyl)-N,N-diethylthieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-amine
Show/Hide
|
C17H16ClN5O2S2
|
1
|
| 1 |
IC50 = 1220 nM
|
|
|
|
CP0523838
|
3-(2,5-dimethylphenylsulfonyl)-N-(3-phenylpropyl)thieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-amine
Show/Hide
|
C24H23N5O2S2
|
1
|
| 1 |
IC50 = 1220 nM
|
|
|
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CP0489487
|
N-(1,3-benzodioxol-5-ylmethyl)-10-(4-methylphenyl)sulfonyl-5-thia-1,8,11,12-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaen-7-amine
Show/Hide
|
C22H17N5O4S2
|
1
|
| 1 |
IC50 = 1250 nM
|
|
|
|
CP0475424
|
3-(2,5-dimethylphenylsulfonyl)-N-(3-methoxypropyl)thieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-amine
Show/Hide
|
C19H21N5O3S2
|
1
|
| 1 |
IC50 = 1290 nM
|
|
|
|
CP0509329
|
N-benzyl-10-(3,4-dimethylphenyl)sulfonyl-N-methyl-5-thia-1,8,11,12-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaen-7-amine
Show/Hide
|
C23H21N5O2S2
|
1
|
| 1 |
IC50 = 1330 nM
|
|
|
|
CP0504475
|
3-(2,5-dimethylphenylsulfonyl)-5-(1-methylpiperidin-4-yl)thieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidine
Show/Hide
|
C21H23N5O2S2
|
1
|
| 1 |
IC50 = 1340 nM
|
|
|
|
CP0496041
|
3-(4-bromophenylsulfonyl)-N-(3,4-dimethylphenyl)thieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-amine
Show/Hide
|
C21H16BrN5O2S2
|
1
|
| 1 |
IC50 = 1350 nM
|
|
|
|
CP0506205
|
10-(benzenesulfonyl)-N-[(3-methoxyphenyl)methyl]-5-thia-1,8,11,12-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaen-7-amine
Show/Hide
|
C21H17N5O3S2
|
1
|
| 1 |
IC50 = 1370 nM
|
|
|
|
CP0507521
|
N-(3-ethylphenyl)-10-(4-methylphenyl)sulfonyl-5-thia-1,8,11,12-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaen-7-amine
Show/Hide
|
C22H19N5O2S2
|
1
|
| 1 |
IC50 = 1380 nM
|
|
|
|
CP0433302
|
N,N-dimethyl-5-[3-[(E)-(4-methylpiperazin-1-yl)iminomethyl]-2-phenylindol-1-yl]sulfonylnaphthalen-1-amine
Show/Hide
|
C32H33N5O2S
|
1
|
| 1 |
IC50 = 1400 nM
|
|
|
|
CP0414658
|
N'-[(E)-[1-(2,5-dimethoxyphenyl)sulfonyl-4-nitroindol-3-yl]methylideneamino]-N,N-dimethylmethanimidamide
Show/Hide
|
C20H21N5O6S
|
1
|
| 1 |
IC50 = 1400 nM
|
|
|
|
CP0496042
|
N-(4-chlorophenyl)-10-(3,4-dimethylphenyl)sulfonyl-5-thia-1,8,11,12-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaen-7-amine
Show/Hide
|
C21H16ClN5O2S2
|
1
|
| 1 |
IC50 = 1430 nM
|
|
|
|
CP0513316
|
8-Fluoro-2-methyl-5-((Z)-2-p-tolylvinyl)-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
Show/Hide
|
C21H21FN2
|
1
|
| 1 |
IC50 = 1440 nM
|
|
|
|
CP0505520
|
N-benzyl-10-(2,5-dimethylphenyl)sulfonyl-N-methyl-5-thia-1,8,11,12-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaen-7-amine
Show/Hide
|
C23H21N5O2S2
|
1
|
| 1 |
IC50 = 1480 nM
|
|
|
|
CP0489461
|
N-(2-methoxyethyl)-10-(4-methylphenyl)sulfonyl-5-thia-1,8,11,12-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaen-7-amine
Show/Hide
|
C17H17N5O3S2
|
1
|
| 1 |
IC50 = 1490 nM
|
|
|
|
CP0421751
|
8-Fluoro-5-[(Z)-2-(4-methoxyphenyl)-vinyl]-2-methyl-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
Show/Hide
|
C21H21FN2O
|
1
|
| 1 |
IC50 = 1500 nM
|
|
|
|
CP0475428
|
3-(2,5-dimethylphenylsulfonyl)-5-(piperidin-1-yl)thieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidine
Show/Hide
|
C20H21N5O2S2
|
1
|
| 1 |
IC50 = 1520 nM
|
|
|
|
CP0377173
|
5-(azepan-1-yl)-3-(3-chlorophenylsulfonyl)thieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidine
Show/Hide
|
C19H18ClN5O2S2
|
1
|
| 1 |
IC50 = 1540 nM
|
|
|
|
CP0465486
|
US8618114, 1.2.12(3)
Show/Hide
|
C18H24N6O2S
|
2
|
| 1 |
IC50 = 1549 nM
|
|
|
| 2 |
Ki = 69.18 nM
|
|
|
|
CP0497224
|
3-(3,4-dimethylphenylsulfonyl)-N-(2-methoxyethyl)thieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-amine
Show/Hide
|
C18H19N5O3S2
|
1
|
| 1 |
IC50 = 1570 nM
|
|
|
|
CP0460301
|
2-methyl-5-(2-(pyridin-2-yl)ethyl)-8-(trifluoromethyl)-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
Show/Hide
|
C20H20F3N3
|
1
|
| 1 |
IC50 = 1590 nM
|
|
|
|
CP0502403
|
3-(4-ethylphenylsulfonyl)-N-isopropylthieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-amine
Show/Hide
|
C18H19N5O2S2
|
1
|
| 1 |
IC50 = 1600 nM
|
|
|
|
CP0523844
|
3-(4-bromophenylsulfonyl)-N-((tetrahydrofuran-2-yl)methyl)thieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-amine
Show/Hide
|
C18H16BrN5O3S2
|
1
|
| 1 |
IC50 = 1620 nM
|
|
|
|
CP0492829
|
2,8-Dimethyl-5-((E)-styryl)-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
Show/Hide
|
C21H24N2
|
1
|
| 1 |
IC50 = 1680 nM
|
|
|
|
CP0539529
|
US8618114, 1.2.19(2).HCl
Show/Hide
|
C23H32N6O3S
|
1
|
| 1 |
IC50 = 1683 nM
|
|
|
|
CP0430440
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8-Fluoro-2-methyl-5-((E)-styryl)-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
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C20H21FN2
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1
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| 1 |
IC50 = 1750 nM
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CP0506206
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3-(4-ethylphenylsulfonyl)-N-m-tolylthieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-amine
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C22H19N5O2S2
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1
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| 1 |
IC50 = 1750 nM
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CP0397526
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(E)-1-[1-(benzenesulfonyl)-2-phenylindol-3-yl]-N-(4-methylpiperazin-1-yl)methanimine
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C26H26N4O2S
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1
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| 1 |
IC50 = 1800 nM
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CP0523840
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N-[(2-chlorophenyl)methyl]-10-(4-propan-2-ylphenyl)sulfonyl-5-thia-1,8,11,12-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaen-7-amine
Show/Hide
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C23H20ClN5O2S2
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1
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| 1 |
IC50 = 1830 nM
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CP0382037
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N'-[(E)-[1-(benzenesulfonyl)-4-nitroindol-3-yl]methylideneamino]-N,N-dimethylmethanimidamide
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C18H17N5O4S
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1
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| 1 |
IC50 = 1830 nM
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CP0484905
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3-(4-fluorophenyl)sulfonyl-2-methylsulfanylpyrazolo[1,5-a]pyrimidine
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C13H10FN3O2S2
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2
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| 1 |
IC50 = 1870 nM
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| 2 |
Ki = 131.83 nM
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CP0502405
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N,N-diethyl-10-(4-ethylphenyl)sulfonyl-5-thia-1,8,11,12-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaen-7-amine
Show/Hide
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C19H21N5O2S2
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1
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| 1 |
IC50 = 1900 nM
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CP0496043
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4-(3-(2,5-dimethylphenylsulfonyl)thieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-yl)morpholine
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C19H19N5O3S2
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1
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| 1 |
IC50 = 1930 nM
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CP0523841
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N-benzyl-10-(4-bromophenyl)sulfonyl-N-methyl-5-thia-1,8,11,12-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaen-7-amine
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C21H16BrN5O2S2
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1
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| 1 |
IC50 = 1950 nM
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CP0532725
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8-Methyl-5-[(Z)-1-methyl-2-phenylvinyl]-2-methyl-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
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C22H24N2
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1
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| 1 |
IC50 = 1980 nM
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CP0475429
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3-(2,5-dimethylphenylsulfonyl)-5-(4-methylpiperidin-1-yl)thieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidine
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C21H23N5O2S2
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1
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| 1 |
IC50 = 1990 nM
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CP0504474
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1-(3-(phenylsulfonyl)thieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-yl)piperidine-4-carboxamide
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C19H18N6O3S2
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1
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| 1 |
IC50 = 1990 nM
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CP0509339
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3-(3-chlorophenylsulfonyl)-5-(3-methylpiperidin-1-yl)thieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidine
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C19H18ClN5O2S2
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1
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| 1 |
IC50 = 2000 nM
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CP0296155
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3-(4-bromophenylsulfonyl)-N-(2,5-dimethylphenyl)thieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-amine
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C21H16BrN5O2S2
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1
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| 1 |
IC50 = 2010 nM
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CP0509727
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N-cyclopentyl-10-(4-methylphenyl)sulfonyl-5-thia-1,8,11,12-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaen-7-amine
Show/Hide
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C19H19N5O2S2
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1
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| 1 |
IC50 = 2030 nM
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CP0522766
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5-(3-Methylpiperidin-1-yl)-3-(phenylsulfonyl)thieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidine
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C19H19N5O2S2
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1
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| 1 |
IC50 = 2030 nM
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CP0449776
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(E)-1-(2-methyl-1-naphthalen-2-ylsulfonylindol-3-yl)-N-(4-methylpiperazin-1-yl)methanimine
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C25H26N4O2S
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1
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| 1 |
IC50 = 2040 nM
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CP0524738
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2,8-dimethyl-5-(2-pyrazine-2-ylethyl)-gamma-carboline
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C19H22N4
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1
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| 1 |
IC50 = 2060 nM
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CP0379360
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N,N-dimethyl-N'-[(E)-[1-(4-methylphenyl)sulfonyl-4-nitroindol-3-yl]methylideneamino]methanimidamide
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C19H19N5O4S
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1
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| 1 |
IC50 = 2120 nM
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CP0504462
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3-(4-chlorophenylsulfonyl)-N-(2-methoxyethyl)thieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-amine
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C16H14ClN5O3S2
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1
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| 1 |
IC50 = 2170 nM
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CP0377207
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N-[2-(4-methylpiperazin-1-yl)phenyl]-N-propan-2-ylnaphthalene-2-sulfonamide
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C24H29N3O2S
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1
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| 1 |
IC50 = 2191 nM
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CP0465479
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US8618114, 1.1.1(6)
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C14H13N3O2S2
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1
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| 1 |
IC50 = 2200 nM
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CP0489486
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N-[(3-methoxyphenyl)methyl]-10-(4-methylphenyl)sulfonyl-5-thia-1,8,11,12-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaen-7-amine
Show/Hide
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C22H19N5O3S2
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1
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| 1 |
IC50 = 2210 nM
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CP0509338
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N-(3-chloro-5-methylphenyl)-10-(3,4-dimethylphenyl)sulfonyl-5-thia-1,8,11,12-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaen-7-amine
Show/Hide
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C22H18ClN5O2S2
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1
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| 1 |
IC50 = 2260 nM
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CP0506291
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8-Fluoro-2-methyl-5-(2-p-tolylethyl)-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
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C21H23FN2
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1
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| 1 |
IC50 = 2270 nM
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CP0465487
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US8618114, 1.2.19(3).HCl
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C24H34N6O3S
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1
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| 1 |
IC50 = 2277 nM
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CP0492826
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8-Fluoro-5-[2-(4-methoxyphenyl)ethyl]-2-methyl-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
Show/Hide
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C21H23FN2O
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1
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| 1 |
IC50 = 2350 nM
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CP0504463
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3-(3,4-dimethylphenylsulfonyl)-N-(3-methoxypropyl)thieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-amine
Show/Hide
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C19H21N5O3S2
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1
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| 1 |
IC50 = 2380 nM
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CP0470463
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(E)-1-[1-(5-chloro-2-methoxy-4-methylphenyl)sulfonyl-2-methylindol-3-yl]-N-(4-methylpiperazin-1-yl)methanimine
Show/Hide
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C23H27ClN4O3S
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1
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| 1 |
IC50 = 2400 nM
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CP0420210
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N'-[(E)-[1-(5-chloro-2-methoxyphenyl)sulfonyl-4-nitroindol-3-yl]methylideneamino]-N,N-dimethylmethanimidamide
Show/Hide
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C19H18ClN5O5S
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1
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| 1 |
IC50 = 2440 nM
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CP0489492
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3-(3-chlorophenylsulfonyl)-N-(4-fluorophenyl)thieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-amine
Show/Hide
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C19H11ClFN5O2S2
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1
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| 1 |
IC50 = 2500 nM
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CP0379358
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N,N-dimethyl-N'-[(E)-(1-naphthalen-2-ylsulfonyl-4-nitroindol-3-yl)methylideneamino]methanimidamide
Show/Hide
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C22H19N5O4S
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1
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| 1 |
IC50 = 2530 nM
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CP0430385
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2-Methyl-5-((E)-styryl)-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
Show/Hide
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C20H22N2
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1
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| 1 |
IC50 = 2580 nM
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CP0421755
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2,8-Dimethyl-5-[(Z)-2-(4-trifluoromethylphenyl)vinyl]-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
Show/Hide
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C22H21F3N2
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1
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| 1 |
IC50 = 2810 nM
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CP0397534
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(E)-1-[1-(4-fluorophenyl)sulfonyl-2-phenylindol-3-yl]-N-(4-methylpiperazin-1-yl)methanimine
Show/Hide
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C26H25FN4O2S
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1
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| 1 |
IC50 = 2900 nM
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CP0500633
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8-Fluoro-5-[(Z)-2-(4-fluorophenyl)-vinyl]-2-methyl-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
Show/Hide
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C20H18F2N2
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1
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| 1 |
IC50 = 2950 nM
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CP0379361
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N,N-dimethyl-N'-[(E)-(1-naphthalen-1-ylsulfonyl-4-nitroindol-3-yl)methylideneamino]methanimidamide
Show/Hide
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C22H19N5O4S
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1
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| 1 |
IC50 = 2960 nM
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CP0378181
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8-fluoro-2-methyl-5-(2-(pyridin-2-yl)ethyl)-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
Show/Hide
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C19H20FN3
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1
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| 1 |
IC50 = 2980 nM
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CP0478590
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8-fluoro-2-methyl-5-(2-(pyridin-4-yl)ethyl)-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
Show/Hide
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C19H20FN3
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1
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| 1 |
IC50 = 3240 nM
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CP0944161
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2-Methyl-8-(pyridin-3-ylsulfonyl)-2,3,4,5-tetrahydro-1Hpyrido[4,3-b]indole hydrochloride
Show/Hide
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C17H18ClN3O2S
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1
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| 1 |
IC50 = 3400 nM
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CP0404071
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(E)-1-[1-(1-methylimidazol-2-yl)sulfonyl-2-phenylindol-3-yl]-N-(4-methylpiperazin-1-yl)methanimine
Show/Hide
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C24H26N6O2S
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1
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| 1 |
IC50 = 3600 nM
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CP0453881
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8-Fluoro-5-[(Z)-1-methyl-2-phenylvinyl]-2-methyl-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
Show/Hide
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C21H21FN2
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1
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| 1 |
IC50 = 3720 nM
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CP0396037
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(E)-1-[1-(2,3-dihydro-1,4-benzodioxin-5-ylsulfonyl)-2-phenylindol-3-yl]-N-(4-methylpiperazin-1-yl)methanimine
Show/Hide
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C28H28N4O4S
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1
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| 1 |
IC50 = 3800 nM
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CP0523847
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N-(3-fluorophenyl)-10-(4-methylphenyl)sulfonyl-5-thia-1,8,11,12-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaen-7-amine
Show/Hide
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C20H14FN5O2S2
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1
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| 1 |
IC50 = 3810 nM
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CP0374343
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2-Benzyl-N-(3-fluorophenyl)-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole-8-sulfonamide
Show/Hide
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C24H22FN3O2S
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1
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| 1 |
IC50 = 3900 nM
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CP0386768
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N-[2-(4-methylpiperazin-1-yl)-1,3-benzothiazol-6-yl]naphthalene-1-sulfonamide
Show/Hide
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C22H22N4O2S2
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1
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| 1 |
IC50 = 3900 nM
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CP0453872
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2,8-Dimethyl-5-[2-(4-trifluoromethylphenyl)ethyl]-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
Show/Hide
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C22H23F3N2
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1
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| 1 |
IC50 = 4070 nM
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CP0524739
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8-methoxy-2-methyl-5-(2-(pyridin-4-yl)ethyl)-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
Show/Hide
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C20H23N3O
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1
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| 1 |
IC50 = 4340 nM
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CP0376018
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(E)-1-[1-(4-fluorophenyl)sulfonyl-2-methylindol-3-yl]-N-(4-methylpiperazin-1-yl)methanimine
Show/Hide
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C21H23FN4O2S
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1
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| 1 |
IC50 = 4740 nM
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CP0480574
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N'-[(E)-[1-(4-fluorophenyl)sulfonyl-4-nitroindol-3-yl]methylideneamino]-N,N-dimethylmethanimidamide
Show/Hide
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C18H16FN5O4S
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1
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| 1 |
IC50 = 4970 nM
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CP0489489
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10-(benzenesulfonyl)-N-phenyl-5-thia-1,8,11,12-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaen-7-amine
Show/Hide
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C19H13N5O2S2
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1
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| 1 |
IC50 = 5000 nM
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CP0484904
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3-(benzenesulfonyl)-2-methylsulfanylpyrazolo[1,5-a]pyrimidine
Show/Hide
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C13H11N3O2S2
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2
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| 1 |
IC50 = 5200 nM
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| 2 |
Ki = 114.82 nM
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CP0509337
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N-(3-methylphenyl)-10-(4-methylphenyl)sulfonyl-5-thia-1,8,11,12-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaen-7-amine
Show/Hide
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C21H17N5O2S2
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1
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| 1 |
IC50 = 5220 nM
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CP0430387
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8-Fluoro-2-methyl-5-[(Z)-2-(4-trifluoromethyl-phenyl)-vinyl]-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
Show/Hide
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C21H18F4N2
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1
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| 1 |
IC50 = 5580 nM
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CP0498731
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2-Methyl-5-((Z)-styryl)-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
Show/Hide
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C20H20N2
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1
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| 1 |
IC50 = 5730 nM
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CP0390107
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2-methyl-5-(2-(pyridin-3-yl)ethyl)-8-(trifluoromethyl)-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
Show/Hide
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C20H20F3N3
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1
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| 1 |
IC50 = 5800 nM
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CP0424945
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2-methyl-5-(2-(pyridin-3-yl)ethyl)-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
Show/Hide
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C19H21N3
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1
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| 1 |
IC50 = 5990 nM
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CP0563372
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US8618114, 1.2.19(4).HCl
Show/Hide
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C23H30N6O3S
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1
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| 1 |
IC50 = 6059 nM
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CP0398560
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N'-[(E)-[1-(4-iodophenyl)sulfonyl-4-nitroindol-3-yl]methylideneamino]-N,N-dimethylmethanimidamide
Show/Hide
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C18H16IN5O4S
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1
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| 1 |
IC50 = 6340 nM
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CP0390108
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2-methyl-5-(2-(pyridin-4-yl)ethyl)-8-(trifluoromethyl)-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
Show/Hide
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C20H20F3N3
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1
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| 1 |
IC50 = 6400 nM
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CP0396036
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(E)-N-(4-methylpiperazin-1-yl)-1-(1-naphthalen-1-ylsulfonyl-2-phenylindol-3-yl)methanimine
Show/Hide
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C30H28N4O2S
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1
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| 1 |
IC50 = 6600 nM
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CP0397525
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(E)-1-[1-(5-chloro-2-methoxy-4-methylphenyl)sulfonyl-2-phenylindol-3-yl]-N-(4-methylpiperazin-1-yl)methanimine
Show/Hide
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C28H29ClN4O3S
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1
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| 1 |
IC50 = 7400 nM
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CP0524747
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2-methyl-5-(2-(pyridin-2-yl)ethyl)-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole-8-carbonitrile
Show/Hide
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C20H20N4
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1
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| 1 |
IC50 = 7470 nM
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CP0524501
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8-methoxy-2-methyl-5-(2-(pyridin-2-yl)ethyl)-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
Show/Hide
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C20H23N3O
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1
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| 1 |
IC50 = 8360 nM
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CP0465478
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US8618114, 1.1(5)
Show/Hide
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C15H14BrN3O2S2
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1
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| 1 |
IC50 = 8400 nM
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CP0378179
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2-methyl-5-(2-(pyridin-4-yl)ethyl)-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
Show/Hide
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C19H21N3
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1
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| 1 |
IC50 = 8910 nM
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CP0377932
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2-methyl-5-(2-(pyridin-4-yl)ethyl)-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole-8-carboxylic acid
Show/Hide
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C20H21N3O2
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1
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| 1 |
IC50 > 10000 nM
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CP0389115
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8-fluoro-2-methyl-5-(2-(pyridin-3-yl)ethyl)-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
Show/Hide
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C19H20FN3
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1
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| 1 |
IC50 > 10000 nM
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CP0560638
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US8618114, 1.1(6)
Show/Hide
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C21H19N3O3S2
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1
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| 1 |
IC50 > 10000 nM
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CP0390109
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8-fluoro-2-methyl-5-(2-(6-methylpyridin-3-yl)ethyl)-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
Show/Hide
|
C20H22FN3
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1
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| 1 |
IC50 = 10690 nM
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CP0377931
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2-methyl-5-(2-(pyridin-2-yl)ethyl)-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
Show/Hide
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C19H21N3
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1
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| 1 |
IC50 = 15750 nM
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CP0436736
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8-Fluoro-2-methyl-5-[2-(4-trifluoromethylphenyl)ethyl]-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
Show/Hide
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C21H20F4N2
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1
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| 1 |
IC50 = 20700 nM
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CP0473482
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N,N,2-trimethyl-1,3,4,5-tetrahydropyrido[4,3-b]indole-8-sulfonamide
Show/Hide
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C14H19N3O2S
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1
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| 1 |
IC50 = 26000 nM
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CP0918848
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2-Methyl-5-[(4-methylphenyl)sulfonyl]-8-(phenylsulfonyl)-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole hydrochloride
Show/Hide
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C25H25ClN2O4S2
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1
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| 1 |
IC50 = 28000 nM
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CP0539527
|
US8618114, 1.1.8(2)
Show/Hide
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C19H16N4O3S2
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1
|
| 1 |
IC50 = 30100 nM
|
|
|
|
CP0377930
|
2-methyl-8-pyridin-3-yl-5-(2-pyridin-2-ylethyl)-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
Show/Hide
|
C24H24N4
|
1
|
| 1 |
IC50 = 43200 nM
|
|
|
|
CP0488719
|
2-Methyl-8-[(4-methylpiperazin-1-yl)sulfonyl]-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
Show/Hide
|
C17H24N4O2S
|
1
|
| 1 |
IC50 = 62000 nM
|
|
|
|
CP0504476
|
3-Phenylsulfonyl-N,N-dimethylthieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-amine
Show/Hide
|
C15H13N5O2S2
|
2
|
| 1 |
IC50 > 30 nM
|
|
|
| 2 |
IC50 > 300 nM
|
|
|
|
CP0377176
|
N-[10-(benzenesulfonyl)-5-thia-1,8,11,12-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaen-7-yl]-N',N'-dimethylethane-1,2-diamine
Show/Hide
|
C17H18N6O2S2
|
1
|
| 1 |
IC50 > 300 nM
|
|
|
|
CP0359336
|
3-(4-ethylphenylsulfonyl)-N-(3-methoxypropyl)thieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-amine
Show/Hide
|
C19H21N5O3S2
|
1
|
| 1 |
IC50 > 5000 nM
|
|
|
|
CP0454583
|
3-(4-bromophenylsulfonyl)-N-(3-methoxypropyl)thieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-amine
Show/Hide
|
C17H16BrN5O3S2
|
1
|
| 1 |
IC50 > 5000 nM
|
|
|
|
CP0475423
|
3-(4-chlorophenylsulfonyl)-N-(3-methoxypropyl)thieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-amine
Show/Hide
|
C17H16ClN5O3S2
|
1
|
| 1 |
IC50 > 5000 nM
|
|
|
|
CP0496040
|
10-(benzenesulfonyl)-N-(1,3-benzothiazol-2-yl)-5-thia-1,8,11,12-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaen-7-amine
Show/Hide
|
C20H12N6O2S3
|
1
|
| 1 |
IC50 > 5000 nM
|
|
|
|
CP0506202
|
3-(4-ethylphenylsulfonyl)-N-isopentylthieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-amine
Show/Hide
|
C20H23N5O2S2
|
1
|
| 1 |
IC50 > 5000 nM
|
|
|
|
CP0509320
|
N-butyl-10-(4-propan-2-ylphenyl)sulfonyl-5-thia-1,8,11,12-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaen-7-amine
Show/Hide
|
C20H23N5O2S2
|
1
|
| 1 |
IC50 > 5000 nM
|
|
|
|
CP0509321
|
3-(4-isopropylphenylsulfonyl)-N-(2-methoxyethyl)thieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidin-5-amine
Show/Hide
|
C19H21N5O3S2
|
1
|
| 1 |
IC50 > 5000 nM
|
|
|
|
CP0509721
|
N-(3-methylbutyl)-10-(4-propan-2-ylphenyl)sulfonyl-5-thia-1,8,11,12-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaen-7-amine
Show/Hide
|
C21H25N5O2S2
|
1
|
| 1 |
IC50 > 5000 nM
|
|
|
|
CP0370117
|
4-(2-Bromo-6-pyrrolidin-1-yl-pyridine-4-sulfonyl)-phenylamine
Show/Hide
|
C15H16BrN3O2S
|
2
|
| 1 |
Kd = 3.162 nM
|
|
|
| 2 |
Ki = 1 nM
|
|
|
|
CP0853831
|
[7-(2-amino-ethyl)-3-benzenesulfonyl-5-methyl-pyrazolo-[1,5-a]pyrimidin-2-yl]-methyl-amine
Show/Hide
|
C16H19N5O2S
|
2
|
| 1 |
Kd = 3.981 nM
|
|
|
| 2 |
Ki = 3.09 nM
|
|
|
|
CP0467208
|
4-(2,6-dichlorophenyl)sulfonyl-8-piperazin-1-yl-2,3-dihydro-1,4-benzoxazine
Show/Hide
|
C18H19Cl2N3O3S
|
1
|
| 1 |
Ki = 0.0631 nM
|
|
|
|
CP0445699
|
5-Chloro-3-methyl-benzo[b]thiophene-2-sulfonic acid [3-(2-dimethylamino-ethyl)-1H-indol-5-yl]-amide
Show/Hide
|
C21H22ClN3O2S2
|
1
|
| 1 |
Ki = 0.1 nM
|
|
|
|
CP0515013
|
4-(2-fluorophenyl)sulfonyl-6-methoxy-8-piperazin-1-yl-2,3-dihydro-1,4-benzoxazine
Show/Hide
|
C19H22FN3O4S
|
1
|
| 1 |
Ki = 0.1585 nM
|
|
|
|
CP0860287
|
N-Methyl-2-(phenylsulfonyl)-5-(piperazin-1-yl)aniline hydrochloride
Show/Hide
|
C17H22ClN3O2S
|
1
|
| 1 |
Ki = 0.16 nM
|
|
|
|
CP0037941
|
2-[1-(Naphthalene-1-sulfonyl)-1H-indol-6-yl]-octahydro-pyrrolo[1,2-a]pyrazine
Show/Hide
|
C25H25N3O2S
|
1
|
| 1 |
Ki = 0.2 nM
|
|
|
|
CP0309013
|
5-chloro-N-[3-[2-(dimethylamino)ethyl]-1H-indol-5-yl]naphthalene-2-sulfonamide
Show/Hide
|
C22H22ClN3O2S
|
2
|
| 1 |
Ki = 0.2 nM
|
|
|
| 2 |
Ki = 0.7 nM
|
|
|
|
CP0404170
|
4-(2-chlorophenyl)sulfonyl-6-methyl-8-piperazin-1-yl-2,3-dihydro-1,4-benzoxazine
Show/Hide
|
C19H22ClN3O3S
|
1
|
| 1 |
Ki = 0.2 nM
|
|
|
|
CP0756875
|
N2,N6,N6,5,7-pentamethyl-3-(phenylsulfonyl)pyrazolo[1,5-a]pyrimidine-2,6-diamine
Show/Hide
|
C17H21N5O2S
|
1
|
| 1 |
Ki = 0.2089 nM
|
|
|
|
CP0904735
|
N2,5-dimethyl-3-(3-chlorophenylsulfonyl)pyrazolo[1,5-a]pyrimidine-2,7-diamine
Show/Hide
|
C14H14ClN5O2S
|
1
|
| 1 |
Ki = 0.2188 nM
|
|
|
|
CP0438807
|
3-(benzenesulfonyl)-N-methyl-6,7,8,9-tetrahydropyrazolo[1,5-a]quinazolin-2-amine
Show/Hide
|
C17H18N4O2S
|
1
|
| 1 |
Ki = 0.259 nM
|
|
|
|
CP0929210
|
1-Benzenesulfonyl-3-((R)-1-methyl-pyrrolidin-2-ylmethyl)-1H-indole oxalic acid
Show/Hide
|
C22H24N2O6S
|
1
|
| 1 |
Ki = 0.3 nM
|
|
|
|
CP0456508
|
1-Benzenesulfonyl-3-((R)-1-methyl-pyrrolidin-2-ylmethyl)-1H-indole; oxalic acid
Show/Hide
|
C20H22N2O2S
|
1
|
| 1 |
Ki = 0.3 nM
|
|
|
|
CP0445700
|
5-Chloro-3-methyl-benzo[b]thiophene-2-sulfonic acid [3-(2-diethylamino-ethyl)-1H-indol-5-yl]-amide
Show/Hide
|
C23H26ClN3O2S2
|
1
|
| 1 |
Ki = 0.3 nM
|
|
|
|
CP0144979
|
1-(phenylsulfonyl)-4-(piperazin-1-yl)-1H-indole
Show/Hide
|
C18H19N3O2S
|
2
|
| 1 |
Ki = 0.3 nM
|
|
|
| 2 |
Ki = 1 nM
|
|
|
|
CP0485158
|
4-(2-fluorophenyl)sulfonyl-2,2-dimethyl-8-piperazin-1-yl-3H-1,4-benzoxazine
Show/Hide
|
C20H24FN3O3S
|
1
|
| 1 |
Ki = 0.3162 nM
|
|
|
|
CP0506507
|
10-(benzenesulfonyl)-N-methyl-1,8,12-triazatricyclo[7.3.0.02,6]dodeca-2(6),7,9,11-tetraen-11-amine
Show/Hide
|
C16H16N4O2S
|
1
|
| 1 |
Ki = 0.375 nM
|
|
|
|
CP0492794
|
4-(2-fluorophenyl)sulfonyl-6-methyl-8-piperazin-1-yl-2,3-dihydro-1,4-benzoxazine
Show/Hide
|
C19H22FN3O3S
|
1
|
| 1 |
Ki = 0.3981 nM
|
|
|
|
CP0513752
|
4-(benzenesulfonyl)-6-methoxy-8-piperazin-1-yl-2,3-dihydro-1,4-benzoxazine
Show/Hide
|
C19H23N3O4S
|
1
|
| 1 |
Ki = 0.3981 nM
|
|
|
|
CP0559980
|
6-chloro-4-(2-fluorophenyl)sulfonyl-8-piperazin-1-yl-2,3-dihydro-1,4-benzoxazine
Show/Hide
|
C18H19ClFN3O3S
|
1
|
| 1 |
Ki = 0.3981 nM
|
|
|
|
CP0490739
|
4-(4-(piperazin-1-yl)-1H-indol-1-ylsulfonyl)benzenamine
Show/Hide
|
C18H20N4O2S
|
1
|
| 1 |
Ki = 0.4 nM
|
|
|
|
CP0431328
|
Biphenyl-4-sulfonic acid [3-(2-dimethylamino-ethyl)-1H-indol-5-yl]-amide
Show/Hide
|
C24H25N3O2S
|
1
|
| 1 |
Ki = 0.4 nM
|
|
|
|
CP0398684
|
7-[4-[4-[1-(benzenesulfonyl)indol-4-yl]piperazin-1-yl]butoxy]-3,4-dihydro-1H-quinolin-2-one
Show/Hide
|
C31H34N4O4S
|
1
|
| 1 |
Ki = 0.4 nM
|
|
|
|
CP0374246
|
10-(benzenesulfonyl)-N,7-dimethyl-1,8,12-triazatricyclo[7.3.0.02,6]dodeca-2(6),7,9,11-tetraen-11-amine
Show/Hide
|
C17H18N4O2S
|
1
|
| 1 |
Ki = 0.413 nM
|
|
|
|
CP0875123
|
[6-Dimethylaminomethyl)-5,7-dimethyl-3-(3-chlorophenylsulfonyl)-pyrazolo[1,5-a]pyrimidin-2-yl]-methylamine
Show/Hide
|
C18H22ClN5O2S
|
1
|
| 1 |
Ki = 0.4169 nM
|
|
|
|
CP0375939
|
5-Chloro-3-methyl-benzo[b]thiophene-2-sulfonic acid [3-(2-dipropylamino-ethyl)-1H-indol-5-yl]-amide
Show/Hide
|
C25H30ClN3O2S2
|
1
|
| 1 |
Ki = 0.5 nM
|
|
|
|
CP0510012
|
4-(2,1,3-benzoxadiazol-4-ylsulfonyl)-6-chloro-8-piperazin-1-yl-2,3-dihydro-1,4-benzoxazine
Show/Hide
|
C18H18ClN5O4S
|
1
|
| 1 |
Ki = 0.5012 nM
|
|
|
|
CP0430801
|
3-(benzenesulfonyl)-N-methyl-5,6,7,8-tetrahydropyrazolo[5,1-b]quinazolin-2-amine
Show/Hide
|
C17H18N4O2S
|
1
|
| 1 |
Ki = 0.542 nM
|
|
|
|
CP0434253
|
4-(2-fluorophenyl)sulfonyl-8-piperazin-1-ylspiro[3H-1,4-benzoxazine-2,1'-cyclobutane]
Show/Hide
|
C21H24FN3O3S
|
1
|
| 1 |
Ki = 0.631 nM
|
|
|
|
CP0485155
|
6-fluoro-4-(2-fluorophenyl)sulfonyl-8-piperazin-1-yl-2,3-dihydro-1,4-benzoxazine
Show/Hide
|
C18H19F2N3O3S
|
1
|
| 1 |
Ki = 0.631 nM
|
|
|
|
CP0485333
|
6-chloro-8-piperazin-1-yl-4-quinolin-8-ylsulfonyl-2,3-dihydro-1,4-benzoxazine
Show/Hide
|
C21H21ClN4O3S
|
1
|
| 1 |
Ki = 0.631 nM
|
|
|
|
CP0126985
|
3-(3-chlorophenyl)sulfonyl-5,7-dimethyl-2-methylsulfanylpyrazolo[1,5-a]pyrimidine
Show/Hide
|
C15H14ClN3O2S2
|
1
|
| 1 |
Ki = 0.7586 nM
|
|
|
|
CP0538535
|
6-chloro-4-naphthalen-1-ylsulfonyl-8-piperazin-1-yl-2,3-dihydro-1,4-benzoxazine
Show/Hide
|
C22H22ClN3O3S
|
1
|
| 1 |
Ki = 0.7943 nM
|
|
|
|
CP0258948
|
4-(3-(2-(dimethylamino)ethyl)-1H-indol-1-ylsulfonyl)benzenamine
Show/Hide
|
C18H21N3O2S
|
1
|
| 1 |
Ki = 0.8 nM
|
|
|
|
CP0041243
|
5-chloro-N-[4-methoxy-3-(piperazin-1-yl)phenyl]-3-methyl-1-benzothiophene-2-sulfonamide hydrochloride
Show/Hide
|
C20H22ClN3O3S2
|
4
|
| 1 |
Ki = 0.8 nM
|
|
|
| 2 |
Ki = 1 nM
|
|
|
| 3 |
Ki = 1.3 nM
|
|
|
| 4 |
Ki = 13 nM
|
|
|
|
CP0442268
|
N-[3-[2-(dimethylamino)ethyl]-1H-indol-5-yl]naphthalene-1-sulfonamide
Show/Hide
|
C22H23N3O2S
|
1
|
| 1 |
Ki = 0.8 nM
|
|
|
|
CP0276427
|
10-(benzenesulfonyl)-11-methylsulfanyl-2-piperazin-1-yl-1,8,12-triazatricyclo[7.3.0.03,7]dodeca-2,7,9,11-tetraene
Show/Hide
|
C20H23N5O2S2
|
1
|
| 1 |
Ki = 0.85 nM
|
|
|
|
CP0853830
|
[6-(Dimethylaminomethyl)-5,7-dimethyl-3(3-fluorophenylsulfonyl)-pyrazolo[1,5-a]pyrimidin-2-yl]-methylamine
Show/Hide
|
C18H22FN5O2S
|
1
|
| 1 |
Ki = 0.8913 nM
|
|
|
|
CP0279831
|
2-(5-methoxy-1-naphthalen-1-ylsulfonylindol-3-yl)-N,N-dimethylethanamine
Show/Hide
|
C23H24N2O3S
|
1
|
| 1 |
Ki = 0.9 nM
|
|
|
|
CP0834162
|
(5-Aminomethyl-7-methyl-3-phenylsulfonyl-pyrazolo[1,5-a]pyrimidin-2-yl)-methylamine
Show/Hide
|
C15H17N5O2S
|
1
|
| 1 |
Ki = 0.9772 nM
|
|
|
|
CP0375936
|
Biphenyl-4-sulfonic acid [3-(2-diethylamino-ethyl)-1H-indol-5-yl]-amide
Show/Hide
|
C26H29N3O2S
|
1
|
| 1 |
Ki = 1 nM
|
|
|
|
CP0445712
|
5-Chloro-3-methyl-benzo[b]thiophene-2-sulfonic acid [3-(1-methyl-piperidin-4-yl)-1H-indol-5-yl]-amide
Show/Hide
|
C23H24ClN3O2S2
|
1
|
| 1 |
Ki = 1 nM
|
|
|
|
CP0379280
|
2-[3-[4-[1-(benzenesulfonyl)indol-4-yl]piperazin-1-yl]propoxy]benzamide
Show/Hide
|
C28H30N4O4S
|
1
|
| 1 |
Ki = 1 nM
|
|
|
|
CP0126984
|
3-(3-fluorophenyl)sulfonyl-5,7-dimethyl-2-methylsulfanylpyrazolo[1,5-a]pyrimidine
Show/Hide
|
C15H14FN3O2S2
|
1
|
| 1 |
Ki = 1.072 nM
|
|
|
|
CP0523219
|
4-(3-benzenesulfonylphenyl)piperazine
Show/Hide
|
C16H18N2O2S
|
1
|
| 1 |
Ki = 1.2 nM
|
|
|
|
CP0725538
|
2-(6-{[(6-Chloroimidazo[2,1-b][1,3]thiazol-5-yl)sulfonyl]amino}-2,3-dihydro-1H-inden-1-ylidene)hydrazinecarboximidamide hydrochloride
Show/Hide
|
C15H15Cl2N7O2S2
|
1
|
| 1 |
Ki = 1.2 nM
|
|
|
|
CP0219258
|
5,7-dimethyl-2-(methylthio)-3-(phenylsulfonyl)pyrazolo[1,5-a]pyrimidine
Show/Hide
|
C15H15N3O2S2
|
2
|
| 1 |
Ki = 1.2 nM
|
|
|
| 2 |
Ki = 1.202 nM
|
|
|
|
CP0490322
|
4-[(6-fluoro-8-piperazin-1-yl-2,3-dihydro-1,4-benzoxazin-4-yl)sulfonyl]aniline
Show/Hide
|
C18H21FN4O3S
|
1
|
| 1 |
Ki = 1.259 nM
|
|
|
|
CP0527983
|
4-(2-fluorophenyl)sulfonyl-8-piperazin-1-yl-2,3-dihydro-1,4-benzoxazine
Show/Hide
|
C18H20FN3O3S
|
1
|
| 1 |
Ki = 1.259 nM
|
|
|
|
CP0403818
|
2-[1-(2,5-dimethoxyphenyl)sulfonyl-5-methoxyindol-3-yl]-N,N-dimethylethanamine
Show/Hide
|
C21H26N2O5S
|
1
|
| 1 |
Ki = 1.3 nM
|
|
|
|
CP0281706
|
6-(1,2,3,5,8,8a-Hexahydro-indolizin-7-yl)-1-(naphthalene-1-sulfonyl)-1H-indole
Show/Hide
|
C26H24N2O2S
|
1
|
| 1 |
Ki = 1.3 nM
|
|
|
|
CP0929038
|
1-[(2-Bromophenyl)sulfonyl]-5-methoxy-3-[(1-piperazinyl)-methyl]-1H-indole Dimesylate Dihydrate
Show/Hide
|
C22H34BrN3O11S3
|
1
|
| 1 |
Ki = 1.3 nM
|
|
|
|
CP0318500
|
5-(1,4-diazepan-1-yl)-2-(4-fluorophenylsulfonyl)-N-methylbenzenamine
Show/Hide
|
C18H22FN3O2S
|
1
|
| 1 |
Ki = 1.4 nM
|
|
|
|
CP0533233
|
5-(1,4-diazepan-1-yl)-2-(3-fluorophenyl)sulfonyl-N-methylaniline
Show/Hide
|
C18H22FN3O2S
|
1
|
| 1 |
Ki = 1.4 nM
|
|
|
|
CP0073333
|
3-benzenesulfonyl-8-piperazin-1-ylquinoline
Show/Hide
|
C19H19N3O2S
|
1
|
| 1 |
Ki = 1.4 nM
|
|
|
|
CP0046912
|
(1R)-N-(prop-2-yn-1-yl)-2,3-dihydro-1H-inden-1-amine
Show/Hide
|
C12H13N
|
1
|
| 1 |
Ki = 1.4 nM
|
|
|
|
CP0078746
|
1-(2-bromophenyl)sulfonyl-4-[(4-methylpiperazin-1-yl)methyl]indole
Show/Hide
|
C20H22BrN3O2S
|
1
|
| 1 |
Ki = 1.43 nM
|
|
|
|
CP0533097
|
1-[9-(benzenesulfonyl)-1,2,3,4-tetrahydrocarbazol-4-yl]-N,N-dimethylmethanamine
Show/Hide
|
C21H24N2O2S
|
1
|
| 1 |
Ki = 1.5 nM
|
|
|
|
CP0152148
|
2-(5-methoxy-1-naphthalen-2-ylsulfonylindol-3-yl)-N,N-dimethylethanamine
Show/Hide
|
C23H24N2O3S
|
1
|
| 1 |
Ki = 1.6 nM
|
|
|
|
CP0725536
|
(+/-)-2-(6-{[(6-Chloroimidazo[2,1-b][1,3]thiazol-5-yl)sulfonyl]amino}-2-methyl-2,3-dihydro-1H-inden-1-ylidene)hydrazinecarboximidamide hydrochloride
Show/Hide
|
C16H17Cl2N7O2S2
|
1
|
| 1 |
Ki = 1.6 nM
|
|
|
|
CP0440757
|
3-chloro-4-fluoro-N-[3-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]propyl]benzenesulfonamide
Show/Hide
|
C21H22ClF2N3O3S
|
1
|
| 1 |
Ki = 1.6 nM
|
|
|
|
CP0854696
|
1-[(4-Isopropylphenyl)sulfonyl]-5-methoxy-3-[(4-methyl-1-piperazinyl)methyl]-1H-indole Dimesylate
Show/Hide
|
C26H39N3O9S3
|
1
|
| 1 |
Ki = 1.63 nM
|
|
|
|
CP0860288
|
5-(Piperazine-1-yl)-2-(phenylsulfonyl)aniline hydrochloride
Show/Hide
|
C16H20ClN3O2S
|
1
|
| 1 |
Ki = 1.65 nM
|
|
|
|
CP0530962
|
2-[1-(Naphthalene-1-sulfonyl)-1H-indol-6-yl]-octahydro-pyrido[1,2-a]pyrazine
Show/Hide
|
C26H27N3O2S
|
1
|
| 1 |
Ki = 1.7 nM
|
|
|
|
CP0921637
|
1-Benzenesulfonyl-3-((S)-1-methyl-pyrrolidin-2-ylmethyl)-1H-indole oxalic acid
Show/Hide
|
C22H24N2O6S
|
1
|
| 1 |
Ki = 1.7 nM
|
|
|
|
CP0457934
|
1-Benzenesulfonyl-3-((S)-1-methyl-pyrrolidin-2-ylmethyl)-1H-indole; oxalic acid
Show/Hide
|
C20H22N2O2S
|
1
|
| 1 |
Ki = 1.7 nM
|
|
|
|
CP0379282
|
1-(benzenesulfonyl)-4-[4-[3-(2-propan-2-yloxyphenoxy)propyl]piperazin-1-yl]indole
Show/Hide
|
C30H35N3O4S
|
1
|
| 1 |
Ki = 1.7 nM
|
|
|
|
CP0517964
|
3-[(4-ethylpiperazin-1-yl)methyl]-5-methoxy-1-(4-propan-2-ylphenyl)sulfonylindole
Show/Hide
|
C25H33N3O3S
|
1
|
| 1 |
Ki = 1.7 nM
|
|
|
|
CP0457932
|
2-ethyl-5-methoxy-3-[[(2R)-1-methylpyrrolidin-2-yl]methyl]-1H-indole
Show/Hide
|
C17H24N2O
|
1
|
| 1 |
Ki = 1.8 nM
|
|
|
|
CP0175237
|
5-(benzenesulfonyl)-N,11-dimethyl-2,3,7,11-tetrazatricyclo[7.4.0.02,6]trideca-1(9),3,5,7-tetraen-4-amine
Show/Hide
|
C17H19N5O2S
|
1
|
| 1 |
Ki = 1.8 nM
|
|
|
|
CP0440753
|
5-chloro-N-[4-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]butyl]-3-methyl-1-benzothiophene-2-sulfonamide
Show/Hide
|
C25H27ClFN3O3S2
|
1
|
| 1 |
Ki = 1.8 nM
|
|
|
|
CP0915687
|
[7-Dimethylaminomethyl-5-methyl-3-phenylsulfonylpyrazolo[1,5-a]pyrimidin-2-yl]-methyl-amine
Show/Hide
|
C17H21N5O2S
|
1
|
| 1 |
Ki = 1.82 nM
|
|
|
|
CP0148433
|
9-(benzenesulfonyl)-6-bromo-N,N-dimethyl-1,2,3,4-tetrahydrocarbazol-3-amine
Show/Hide
|
C20H21BrN2O2S
|
1
|
| 1 |
Ki = 1.83 nM
|
|
|
|
CP0915998
|
(7-aminomethyl-3-benzenesulfonyl-5-methyl-pyrazolo[1,5-a]pyrimidin-2-yl)-methyl-amine
Show/Hide
|
C15H17N5O2S
|
1
|
| 1 |
Ki = 1.862 nM
|
|
|
|
CP0427892
|
N,N-dimethyl-2-[1-[4-(trifluoromethyl)phenyl]sulfonylindol-3-yl]ethanamine
Show/Hide
|
C19H19F3N2O2S
|
1
|
| 1 |
Ki = 1.9 nM
|
|
|
|
CP0528331
|
1-(4-aminophenylsulfonyl)-N4,N6-dimethyl-1H-indole-4,6-diamine
Show/Hide
|
C16H18N4O2S
|
1
|
| 1 |
Ki = 1.9 nM
|
|
|
|
CP0310111
|
6-Chloro-imidazo[2,1-b]thiazole-5-sulfonic acid [1-(2-dimethylamino-ethyl)-1H-indol-5-yl]-amide
Show/Hide
|
C17H18ClN5O2S2
|
1
|
| 1 |
Ki = 1.9 nM
|
|
|
|
CP0516219
|
5-(benzenesulfonyl)-N-methyl-2,3,7,11-tetrazatricyclo[7.4.0.02,6]trideca-1(9),3,5,7-tetraen-4-amine
Show/Hide
|
C16H17N5O2S
|
1
|
| 1 |
Ki = 1.9 nM
|
|
|
|
CP0175239
|
5,7-Dimethyl-2-(ethylthio)-3-phenylsulfonyl-pyrazolo[1,5-a]pyrimidine
Show/Hide
|
C16H17N3O2S2
|
1
|
| 1 |
Ki = 1.91 nM
|
|
|
|
CP0148435
|
N,N-dimethyl-9-[3-(trifluoromethyl)phenyl]sulfonyl-1,2,3,4-tetrahydrocarbazol-3-amine
Show/Hide
|
C21H21F3N2O2S
|
1
|
| 1 |
Ki = 1.92 nM
|
|
|
|
CP0471151
|
4-(3-chlorophenyl)sulfonyl-8-piperazin-1-yl-2,3-dihydro-1,4-benzoxazine
Show/Hide
|
C18H20ClN3O3S
|
1
|
| 1 |
Ki = 1.995 nM
|
|
|
|
CP0485156
|
2-[(6-methyl-8-piperazin-1-yl-2,3-dihydro-1,4-benzoxazin-4-yl)sulfonyl]benzonitrile
Show/Hide
|
C20H22N4O3S
|
1
|
| 1 |
Ki = 1.995 nM
|
|
|
|
CP0505563
|
4-[5,7-dimethyl-2-(methylamino)pyrazolo[1,5-a]pyrimidin-3-yl]sulfonylphenol
Show/Hide
|
C15H16N4O3S
|
1
|
| 1 |
Ki = 1.995 nM
|
|
|
|
CP0045069
|
2-[1-(benzenesulfonyl)-5-methoxyindol-3-yl]-N,N-dimethylethanamine
Show/Hide
|
C19H22N2O3S
|
3
|
| 1 |
Ki = 2 nM
|
|
|
| 2 |
Ki = 2.1 nM
|
|
|
| 3 |
Ki = 2.3 nM
|
|
|
|
CP0144949
|
2-[1-({6-chloroimidazo[2,1-b][1,3]thiazole-5-}sulfonyl)-1H-indol-3-yl]ethan-1-amine
Show/Hide
|
C15H13ClN4O2S2
|
1
|
| 1 |
Ki = 2 nM
|
|
|
|
CP0407460
|
4-(4-methoxyphenyl)-6-(4-methylpiperazin-1-yl)-1-(2-methylpropylsulfonyl)pyrrolo[2,3-b]pyridine
Show/Hide
|
C23H30N4O3S
|
1
|
| 1 |
Ki = 2 nM
|
|
|
|
CP0854701
|
1-[(2-Bromophenyl)sulfonyl]-5-methoxy-3-[(4-methyl-1-piperazinyl)methyl]-1H-indole Dimesylate Monohydrate
Show/Hide
|
C22H30BrN3O7S2
|
1
|
| 1 |
Ki = 2 nM
|
|
|
|
CP0894863
|
1-(4-Isopropylbenzenesulfonyl)-5-methoxy-3-(4-methyl-[1,4]-diazepan-1-ylmethyl)-1H-indole Dihydrochloride
Show/Hide
|
C25H35Cl2N3O3S
|
1
|
| 1 |
Ki = 2 nM
|
|
|
|
CP0249646
|
4-[5-[[2-(5-fluoro-1H-indol-3-yl)ethylamino]methyl]furan-2-yl]phenol
Show/Hide
|
C21H19FN2O2
|
1
|
| 1 |
Ki = 2 nM
|
|
|
|
CP0466465
|
4-[5-[[2-(6-fluoro-1H-indol-3-yl)ethylamino]methyl]furan-2-yl]phenol
Show/Hide
|
C21H19FN2O2
|
1
|
| 1 |
Ki = 2 nM
|
|
|
|
CP0159204
|
5-[1-(benzenesulfonyl)-5-methoxyindol-3-yl]-1H-imidazol-2-amine;hydrochloride
Show/Hide
|
C18H17ClN4O3S
|
1
|
| 1 |
Ki = 2 nM
|
|
|
|
CP0430225
|
7-[5-methoxy-3-(1,2,3,6-tetrahydropyridin-4-yl)indol-1-yl]sulfonylquinoline
Show/Hide
|
C23H21N3O3S
|
1
|
| 1 |
Ki = 2 nM
|
|
|
|
CP0916029
|
[6-(2-Dimethylaminoethyl)-5,7-dimethyl-3-phenylsulfonylpyrazolo[1,5-a]pyrimidin-2-yl]-methylamine
Show/Hide
|
C19H25N5O2S
|
1
|
| 1 |
Ki = 2.089 nM
|
|
|
|
CP0542305
|
4-(benzenesulfonyl)-N-methyl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1,3,5,8-tetraen-5-amine
Show/Hide
|
C16H17N5O2S
|
1
|
| 1 |
Ki = 2.1 nM
|
|
|
|
CP0543199
|
1-(4-bromophenyl)sulfonyl-3-[(4-methylpiperazin-1-yl)methyl]indole
Show/Hide
|
C20H22BrN3O2S
|
1
|
| 1 |
Ki = 2.13 nM
|
|
|
|
CP0265775
|
6-chloro-N-[3-[2-(dimethylamino)ethyl]-1H-indol-5-yl]imidazo[2,1-b][1,3]thiazole-5-sulfonamide
Show/Hide
|
C17H18ClN5O2S2
|
1
|
| 1 |
Ki = 2.2 nM
|
|
|
|
CP0355993
|
6-chloro-N-[3-(4,5-dihydro-1H-imidazol-2-ylhydrazono)-2,3-dihydro-1H-inden-5-yl]imidazo[2,1-b][1,3]thiazole-5-sulfonamide
Show/Hide
|
C17H16ClN7O2S2
|
1
|
| 1 |
Ki = 2.2 nM
|
|
|
|
CP0411522
|
7-[3-[4-[1-(benzenesulfonyl)indol-4-yl]piperazin-1-yl]propoxy]-3,4-dihydro-1H-quinolin-2-one
Show/Hide
|
C30H32N4O4S
|
1
|
| 1 |
Ki = 2.3 nM
|
|
|
|
CP0399032
|
6-chloro-N-[4-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]butyl]naphthalene-2-sulfonamide
Show/Hide
|
C26H27ClFN3O3S
|
1
|
| 1 |
Ki = 2.4 nM
|
|
|
|
CP0440755
|
N-[4-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]butyl]naphthalene-2-sulfonamide
Show/Hide
|
C26H28FN3O3S
|
1
|
| 1 |
Ki = 2.4 nM
|
|
|
|
CP0553072
|
N,N-dimethyl-2-[1-(4-methylphenyl)sulfonylindol-3-yl]ethanamine
Show/Hide
|
C19H22N2O2S
|
1
|
| 1 |
Ki = 2.5 nM
|
|
|
|
CP0477815
|
4-(benzenesulfonyl)-6-methyl-8-piperazin-1-yl-2,3-dihydro-1,4-benzoxazine
Show/Hide
|
C19H23N3O3S
|
1
|
| 1 |
Ki = 2.512 nM
|
|
|
|
CP0441383
|
1-(Benzenesulfonyl)-5-(piperazin-1-yl-methyl)-1H-indole
Show/Hide
|
C19H21N3O2S
|
1
|
| 1 |
Ki = 2.52 nM
|
|
|
|
CP0212171
|
1-(2-Bromo benzenesulfonyl)-5-(4-ethylpiperazin-1-yl-methyl)-1H-indole
Show/Hide
|
C21H24BrN3O2S
|
1
|
| 1 |
Ki = 2.56 nM
|
|
|
|
CP0505259
|
3-chloro-1-(4-fluoro benzenesulfonyl)-5-(piperazin-1-yl-methyl)-1H-indole
Show/Hide
|
C19H19ClFN3O2S
|
1
|
| 1 |
Ki = 2.58 nM
|
|
|
|
CP0677880
|
2-(5-{[(6-Chloroimidazo[2,1-b][1,3]thiazol-5-yl)sulfonyl]amino}-2,3-dihydro-1H-inden-1-ylidene)hydrazinecarboximidamide hydrochloride
Show/Hide
|
C15H15Cl2N7O2S2
|
1
|
| 1 |
Ki = 2.6 nM
|
|
|
|
CP0456750
|
9-(3-chlorophenyl)sulfonyl-N,N-dimethyl-6-methylsulfanyl-1,2,3,4-tetrahydrocarbazol-3-amine
Show/Hide
|
C21H23ClN2O2S2
|
1
|
| 1 |
Ki = 2.68 nM
|
|
|
|
CP0304087
|
2-(benzenesulfonyl)-N-ethyl-5-piperazin-1-ylaniline
Show/Hide
|
C18H23N3O2S
|
1
|
| 1 |
Ki = 2.7 nM
|
|
|
|
CP0488217
|
2-[4-[4-[1-(benzenesulfonyl)indol-4-yl]piperazin-1-yl]butoxy]benzamide
Show/Hide
|
C29H32N4O4S
|
1
|
| 1 |
Ki = 2.8 nM
|
|
|
|
CP0652571
|
2-Bromobenzenesulfonyl-4-(piperazin-1-ylmethyl)-1H-indole dihydrochloride
Show/Hide
|
C19H22BrCl2N3O2S
|
1
|
| 1 |
Ki = 2.82 nM
|
|
|
|
CP0429488
|
9-(2-bromophenyl)sulfonyl-N,N-dimethyl-1,2,3,4-tetrahydrocarbazol-3-amine
Show/Hide
|
C20H21BrN2O2S
|
1
|
| 1 |
Ki = 2.85 nM
|
|
|
|
CP0170456
|
3-chloro-1-(4-fluoro benzenesulfonyl)-5-(4-methylpiperazin-1-yl-methyl)-1H-indole
Show/Hide
|
C20H21ClFN3O2S
|
1
|
| 1 |
Ki = 2.97 nM
|
|
|
|
CP0524175
|
2-[1-(Naphthalene-2-sulfonyl)-1H-indol-6-yl]-octahydro-pyrido[1,2-a]pyrazine
Show/Hide
|
C26H27N3O2S
|
1
|
| 1 |
Ki = 3 nM
|
|
|
|
CP0099906
|
N-(2,5-dibromo-3-fluorophenyl)-4-methoxy-3-piperazin-1-ylbenzenesulfonamide
Show/Hide
|
C17H18Br2FN3O3S
|
1
|
| 1 |
Ki = 3 nM
|
|
|
|
CP0255950
|
2-[1-(benzenesulfonyl)indol-3-yl]-N,N-dimethylethanamine
Show/Hide
|
C18H20N2O2S
|
3
|
| 1 |
Ki = 3 nM
|
|
|
| 2 |
Ki = 4 nM
|
|
|
| 3 |
Ki = 4.1 nM
|
|
|
|
CP0285245
|
2-(1-benzyl-1H-inden-3-yl)-N,N-dimethylethanamine
Show/Hide
|
C20H23N
|
1
|
| 1 |
Ki = 3 nM
|
|
|
|
CP0435522
|
2-(3-benzyl-3H-inden-1-yl)-N-methylethanamine
Show/Hide
|
C19H21N
|
1
|
| 1 |
Ki = 3 nM
|
|
|
|
CP0401918
|
indenylsulfonamide, 28
Show/Hide
|
C19H19ClN4O2S2
|
1
|
| 1 |
Ki = 3 nM
|
|
|
|
CP0690827
|
1-[1-(2-methylpropanesulfonyl)-4-[4-(trifluoromethyl)phenyl]-1H-pyrrolo[2,3-b]pyridin-6-yl]piperazine
Show/Hide
|
C22H25F3N4O2S
|
1
|
| 1 |
Ki = 3 nM
|
|
|
|
CP0455170
|
1-(3-chlorophenyl)sulfonyl-N-[(3S)-pyrrolidin-3-yl]pyrrolo[3,2-c]quinolin-4-amine
Show/Hide
|
C21H19ClN4O2S
|
1
|
| 1 |
Ki = 3 nM
|
|
|
|
CP0426435
|
4-[5-[[2-(5-methoxy-1H-indol-3-yl)ethylamino]methyl]furan-2-yl]phenol
Show/Hide
|
C22H22N2O3
|
1
|
| 1 |
Ki = 3 nM
|
|
|
|
CP0435398
|
N-[4-[1-(benzenesulfonyl)-5-methoxyindol-3-yl]-5-methyl-1H-imidazol-2-yl]-2-phenylacetamide
Show/Hide
|
C27H24N4O4S
|
1
|
| 1 |
Ki = 3 nM
|
|
|
|
CP0489725
|
4-[1-(benzenesulfonyl)-5-methoxyindol-3-yl]-5-methyl-1H-imidazol-2-amine;hydrochloride
Show/Hide
|
C19H19ClN4O3S
|
1
|
| 1 |
Ki = 3 nM
|
|
|
|
CP0430226
|
4-[5-methoxy-3-(1,2,3,6-tetrahydropyridin-4-yl)indol-1-yl]sulfonylisoquinoline
Show/Hide
|
C23H21N3O3S
|
1
|
| 1 |
Ki = 3 nM
|
|
|
|
CP0441384
|
1-(4-Chloro benzenesulfonyl)-5-(4-methylpiperazin-1-yl-methyl)-1H-indole
Show/Hide
|
C20H22ClN3O2S
|
1
|
| 1 |
Ki = 3.02 nM
|
|
|
|
CP0393102
|
2-[1-(4-chlorophenyl)sulfonyl-5-methoxyindol-3-yl]-N,N-dimethylethanamine
Show/Hide
|
C19H21ClN2O3S
|
1
|
| 1 |
Ki = 3.1 nM
|
|
|
|
CP0487326
|
1-(3-trifluoromethyl benzenesulfonyl)-5-(4-methylpiperazin-1-yl-methyl)-1H-indole
Show/Hide
|
C21H22F3N3O2S
|
1
|
| 1 |
Ki = 3.15 nM
|
|
|
|
CP0553064
|
4-(2-chlorophenyl)sulfonyl-8-piperazin-1-yl-2,3-dihydro-1,4-benzoxazine
Show/Hide
|
C18H20ClN3O3S
|
1
|
| 1 |
Ki = 3.162 nM
|
|
|
|
CP0172992
|
3-(4-chlorophenyl)sulfonyl-5,7-dimethyl-2-methylsulfanylpyrazolo[1,5-a]pyrimidine
Show/Hide
|
C15H14ClN3O2S2
|
1
|
| 1 |
Ki = 3.162 nM
|
|
|
|
CP0212172
|
1-(4-Fluoro benzenesulfonyl)-5-(4-ethylpiperazin-1-yl-methyl)-1H-indole
Show/Hide
|
C21H24FN3O2S
|
1
|
| 1 |
Ki = 3.21 nM
|
|
|
|
CP0058302
|
1-(benzenesulfonyl)-4-[(4-methylpiperazin-1-yl)methyl]indole
Show/Hide
|
C20H23N3O2S
|
1
|
| 1 |
Ki = 3.24 nM
|
|
|
|
CP0527480
|
2-[1-(Toluene-4-sulfonyl)-1H-indol-6-yl]-octahydro-pyrrolo[1,2-a]pyrazine
Show/Hide
|
C22H25N3O2S
|
1
|
| 1 |
Ki = 3.3 nM
|
|
|
|
CP0490061
|
5-Chloro-naphthalene-1-sulfonic acid [3-(2-diethylamino-ethyl)-1H-indol-5-yl]-amide
Show/Hide
|
C24H26ClN3O2S
|
1
|
| 1 |
Ki = 3.3 nM
|
|
|
|
CP0447245
|
6-chloro-N-[4-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]butyl]-1-benzothiophene-2-sulfonamide
Show/Hide
|
C24H25ClFN3O3S2
|
1
|
| 1 |
Ki = 3.3 nM
|
|
|
|
CP0524497
|
3-Chloro-1-(2,4-difluorobenzenesulfonyl)-5-(4-methylpiperazin-1-yl-methyl)-1H-indole
Show/Hide
|
C20H20ClF2N3O2S
|
1
|
| 1 |
Ki = 3.36 nM
|
|
|
|
CP0443093
|
5-fluoro-N-[4-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]butyl]-3-methyl-1-benzothiophene-2-sulfonamide
Show/Hide
|
C25H27F2N3O3S2
|
1
|
| 1 |
Ki = 3.4 nM
|
|
|
|
CP0431329
|
N-[3-[2-(diethylamino)ethyl]-1H-indol-5-yl]naphthalene-1-sulfonamide
Show/Hide
|
C24H27N3O2S
|
1
|
| 1 |
Ki = 3.5 nM
|
|
|
|
CP0217150
|
IDALOPIRDINE
Show/Hide
|
C20H19F5N2O
|
1
|
| 1 |
Ki = 3.54 nM
|
|
|
|
CP0455332
|
2-[1-(2,4-Difluoro-benzenesulfonyl)-1H-indol-6-yl]-octahydro-pyrido[1,2-a]pyrazine
Show/Hide
|
C22H23F2N3O2S
|
1
|
| 1 |
Ki = 3.6 nM
|
|
|
|
CP0488666
|
9-(2-fluorophenyl)sulfonyl-6-methoxy-N,N-dimethyl-1,2,3,4-tetrahydrocarbazol-3-amine
Show/Hide
|
C21H23FN2O3S
|
1
|
| 1 |
Ki = 3.63 nM
|
|
|
|
CP0526067
|
6-methoxy-N,N-dimethyl-9-[3-(trifluoromethyl)phenyl]sulfonyl-1,2,3,4-tetrahydrocarbazol-3-amine
Show/Hide
|
C22H23F3N2O3S
|
1
|
| 1 |
Ki = 3.71 nM
|
|
|
|
CP0523325
|
1-(benzenesulfonyl)-4-[4-[3-(1-benzofuran-6-yloxy)propyl]piperazin-1-yl]indole
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C29H29N3O4S
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1
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| 1 |
Ki = 3.8 nM
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CP0126986
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3-(3-chloro-4-fluorophenyl)sulfonyl-5,7-dimethyl-2-methylsulfanylpyrazolo[1,5-a]pyrimidine
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C15H13ClFN3O2S2
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1
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| 1 |
Ki = 3.802 nM
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CP0170320
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1-Benzenesulfonyl-5-(4-methylpiperazin-1-yl-methyl)-1H-indole
Show/Hide
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C20H23N3O2S
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1
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| 1 |
Ki = 3.83 nM
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CP0375940
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N-[3-[2-(dipropylamino)ethyl]-1H-indol-5-yl]naphthalene-2-sulfonamide
Show/Hide
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C26H31N3O2S
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1
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| 1 |
Ki = 3.9 nM
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CP0483780
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4-(benzenesulfonyl)-6-chloro-8-(1,4-diazepan-1-yl)-2,3-dihydro-1,4-benzoxazine
Show/Hide
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C19H22ClN3O3S
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1
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| 1 |
Ki = 3.981 nM
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CP0502066
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4-(benzenesulfonyl)-6-fluoro-2,2-dimethyl-8-piperidin-4-yl-3H-1,4-benzoxazine
Show/Hide
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C21H25FN2O3S
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1
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| 1 |
Ki = 3.981 nM
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CP0487316
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4-(5,7-dimethyl-2-methylsulfanylpyrazolo[1,5-a]pyrimidin-3-yl)sulfonylphenol
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C15H15N3O3S2
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1
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| 1 |
Ki = 3.981 nM
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CP0446545
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5-Chloro-3-methyl-benzo[b]thiophene-2-sulfonic acid [3-(2-pyrrolidin-1-yl-ethyl)-1H-indol-5-yl]-amide
Show/Hide
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C23H24ClN3O2S2
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1
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| 1 |
Ki = 4 nM
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CP0121807
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6-(4-methylpiperazin-1-yl)-1-(2-methylpropylsulfonyl)-4-[4-(trifluoromethyl)phenyl]pyrrolo[2,3-b]pyridine
Show/Hide
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C23H27F3N4O2S
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1
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| 1 |
Ki = 4 nM
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CP0877966
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5-Fluoro-1-[(4-isopropylphenyl)sulfonyl]-3-[(4-methyl-1-piperazinyl)methyl]-1H-indole Dihydrochloride
Show/Hide
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C23H30Cl2FN3O2S
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1
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| 1 |
Ki = 4 nM
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CP0438428
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4-[1-(benzenesulfonyl)indol-6-yl]-5-methyl-1H-imidazol-2-amine;hydrochloride
Show/Hide
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C18H17ClN4O2S
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1
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| 1 |
Ki = 4 nM
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CP0430227
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5-[5-methoxy-3-(1,2,3,6-tetrahydropyridin-4-yl)indol-1-yl]sulfonylquinoline
Show/Hide
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C23H21N3O3S
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1
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| 1 |
Ki = 4 nM
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CP0673870
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2-(6-{[(6-chloroimidazo[2,1-b][1,3]thiazol-5-yl)sulfonyl](methyl)amino}-2,3-dihydro-1H-inden-1-ylidene)hydrazinecarboximidamide hydrochloride
Show/Hide
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C16H17Cl2N7O2S2
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1
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| 1 |
Ki = 4.1 nM
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CP0037955
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METHIOTHEPIN
Show/Hide
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C20H24N2S2
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1
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| 1 |
Ki = 4.1 nM
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CP0505290
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1-(2-Chloro-5-trifluoromethyl benzenesulfonyl)-3-chloro-5-(4-methylpiperazin-1-yl-methyl)-1H-indole
Show/Hide
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C21H20Cl2F3N3O2S
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1
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| 1 |
Ki = 4.16 nM
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CP0148432
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9-(3-chlorophenyl)sulfonyl-N,N-dimethyl-1,2,3,4-tetrahydrocarbazol-3-amine
Show/Hide
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C20H21ClN2O2S
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1
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| 1 |
Ki = 4.21 nM
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CP0442278
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N-[3-(2-pyrrolidin-1-ylethyl)-1H-indol-5-yl]naphthalene-2-sulfonamide
Show/Hide
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C24H25N3O2S
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1
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| 1 |
Ki = 4.3 nM
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CP0523304
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9-(2-bromophenyl)sulfonyl-6-methoxy-N,N-dimethyl-1,2,3,4-tetrahydrocarbazol-3-amine
Show/Hide
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C21H23BrN2O3S
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1
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| 1 |
Ki = 4.3 nM
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CP0469996
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1-(benzenesulfonyl)-5-methoxy-3-[(4-methylpiperazin-1-yl)methyl]indole
Show/Hide
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C21H25N3O3S
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1
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| 1 |
Ki = 4.3 nM
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CP0039675
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6-chloro-N-[3-[2-(dimethylamino)ethyl]-2-methyl-1H-inden-5-yl]imidazo[2,1-b][1,3]thiazole-5-sulfonamide
Show/Hide
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C19H21ClN4O2S2
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1
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| 1 |
Ki = 4.5 nM
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CP0486155
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N-[3-(2-pyrrolidin-1-ylethyl)-1H-indol-5-yl]naphthalene-1-sulfonamide
Show/Hide
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C24H25N3O2S
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1
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| 1 |
Ki = 4.5 nM
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CP0953941
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1-[(2-Bromophenyl)sulfonyl]-3-[(1-piperazinyl)methyl]-1H-indole Dihydrochloride
Show/Hide
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C19H22BrCl2N3O2S
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1
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| 1 |
Ki = 4.5 nM
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CP0516155
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9-(benzenesulfonyl)-N,N-dimethyl-6-methylsulfanyl-1,2,3,4-tetrahydrocarbazol-3-amine
Show/Hide
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C21H24N2O2S2
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1
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| 1 |
Ki = 4.57 nM
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CP0885043
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N-(5,7-dimethyl-2-(methylamino)-3-(phenylsulfonyl)pyrazolo[1,5-a]pyrimidin-6-yl)acetamide
Show/Hide
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C17H19N5O3S
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1
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| 1 |
Ki = 4.677 nM
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CP0553634
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9-(2-chlorophenyl)sulfonyl-6-methoxy-N,N-dimethyl-1,2,3,4-tetrahydrocarbazol-3-amine
Show/Hide
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C21H23ClN2O3S
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1
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| 1 |
Ki = 4.68 nM
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CP0461878
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7-[1-(Naphthalene-1-sulfonyl)-1H-indol-6-yl]-octahydro-indolizin-7-ol
Show/Hide
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C26H26N2O3S
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1
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| 1 |
Ki = 4.7 nM
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CP0437056
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N-[3-(1-methylpiperidin-4-yl)-1H-indol-5-yl]naphthalene-1-sulfonamide
Show/Hide
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C24H25N3O2S
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1
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| 1 |
Ki = 4.7 nM
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CP0500050
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4-[(4-methylpiperazin-1-yl)methyl]-1-naphthalen-1-ylsulfonylindole
Show/Hide
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C24H25N3O2S
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1
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| 1 |
Ki = 4.82 nM
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CP0461850
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2-[1-(Toluene-4-sulfonyl)-1H-indol-6-yl]-octahydro-pyrido[1,2-a]pyrazine
Show/Hide
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C23H27N3O2S
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1
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| 1 |
Ki = 4.9 nM
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CP0285020
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2-(7-methoxy-1-naphthalen-2-ylsulfonylindol-3-yl)-N,N-dimethylethanamine
Show/Hide
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C23H24N2O3S
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1
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| 1 |
Ki = 5 nM
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CP0045063
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2-methyl-4-(4-methylpiperazin-1-yl)-10H-thieno[2,3-b][1,5]benzodiazepine
Show/Hide
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C17H20N4S
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5
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| 1 |
Ki = 5 nM
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| 2 |
Ki = 7 nM
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| 3 |
Ki = 7.943 nM
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| 4 |
Ki = 8.8 nM
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| 5 |
Ki = 10.7 nM
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CP0461293
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N-[4-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]butyl]naphthalene-2-sulfonamide
Show/Hide
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C25H28N4O2S2
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1
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| 1 |
Ki = 5 nM
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CP0549220
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4-(1H-indol-5-yl)-6-(4-methylpiperazin-1-yl)-1-(2-methylpropylsulfonyl)pyrrolo[2,3-b]pyridine
Show/Hide
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C24H29N5O2S
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1
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| 1 |
Ki = 5 nM
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CP0854694
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1-[(4-Fluorophenyl)sulfonyl]-5-methoxy-3-[(4-methyl-1-piperazinyl)methyl]-1H-indole Dimesylate
Show/Hide
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C23H32FN3O9S3
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1
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| 1 |
Ki = 5 nM
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CP0426434
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4-[5-[[2-(5-methyl-1H-indol-3-yl)ethylamino]methyl]furan-2-yl]phenol
Show/Hide
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C22H22N2O2
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1
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| 1 |
Ki = 5 nM
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CP0554277
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4-[3-(1,2,3,6-tetrahydropyridin-4-yl)indol-1-yl]sulfonylisoquinoline
Show/Hide
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C22H19N3O2S
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1
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| 1 |
Ki = 5 nM
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CP0449693
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9-(3-chlorophenyl)sulfonyl-6-fluoro-N,N-dimethyl-1,2,3,4-tetrahydrocarbazol-3-amine
Show/Hide
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C20H20ClFN2O2S
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1
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| 1 |
Ki = 5.01 nM
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CP0553066
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6-fluoro-4-(3-fluorophenyl)sulfonyl-2,2-dimethyl-8-piperidin-4-yl-3H-1,4-benzoxazine
Show/Hide
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C21H24F2N2O3S
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1
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| 1 |
Ki = 5.012 nM
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CP0526066
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9-(2-bromophenyl)sulfonyl-6-fluoro-N,N-dimethyl-1,2,3,4-tetrahydrocarbazol-3-amine
Show/Hide
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C20H20BrFN2O2S
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1
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| 1 |
Ki = 5.02 nM
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CP0506619
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N-[3-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]propyl]-3-chloro-4-fluorobenzenesulfonamide
Show/Hide
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C20H22ClFN4O2S2
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1
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| 1 |
Ki = 5.1 nM
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CP0754497
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2-(6-{[(6-chloroimidazo[2,1-b][1,3]thiazol-5-yl)sulfonyl]amino}-3,3-dimethyl-2,3-dihydro-1H-inden-1-ylidene)hydrazinecarboximidamide hydrochloride
Show/Hide
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C17H19Cl2N7O2S2
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1
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| 1 |
Ki = 5.2 nM
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CP0410412
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5-Chloro-3-methyl-benzo[b]thiophene-2-sulfonic acid (3-dimethylaminomethyl-1H-indol-5-yl)-amide
Show/Hide
|
C20H20ClN3O2S2
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1
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| 1 |
Ki = 5.3 nM
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CP0488653
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1-(benzenesulfonyl)-4-[4-[3-(4-fluorophenoxy)propyl]piperazin-1-yl]indole
Show/Hide
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C27H28FN3O3S
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1
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| 1 |
Ki = 5.4 nM
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CP0076180
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9-(benzenesulfonyl)-6-methoxy-N,N-dimethyl-1,2,3,4-tetrahydrocarbazol-3-amine
Show/Hide
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C21H24N2O3S
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1
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| 1 |
Ki = 5.44 nM
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CP0526068
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6-bromo-N,N-dimethyl-9-[3-(trifluoromethyl)phenyl]sulfonyl-1,2,3,4-tetrahydrocarbazol-3-amine
Show/Hide
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C21H20BrF3N2O2S
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1
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| 1 |
Ki = 5.5 nM
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CP0499034
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1-(2,3-Dichlorobenzenesulfonyl)-5-(4-ethylpiperazin-1-yl-methyl)-1H-indole
Show/Hide
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C21H23Cl2N3O2S
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1
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| 1 |
Ki = 5.52 nM
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CP0170455
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3-Chloro-1-(2,4-difluoro benzenesulfonyl)-5-(piperazin-1-yl-methyl)-1H-indole
Show/Hide
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C19H18ClF2N3O2S
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1
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| 1 |
Ki = 5.57 nM
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CP0453210
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2-(1-Benzenesulfonyl-1H-indol-6-yl)-octahydro-pyrido[1,2-a]pyrazine
Show/Hide
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C22H25N3O2S
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1
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| 1 |
Ki = 5.7 nM
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CP0546256
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1-(2-bromophenyl)sulfonyl-5-methoxy-3-[(4-methyl-1,4-diazepan-1-yl)methyl]indole
Show/Hide
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C22H26BrN3O3S
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1
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| 1 |
Ki = 5.7 nM
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CP0963614
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1-[(4-Isopropylphenyl)sulfonyl]-5-methoxy-3-[(1-piperazinyl)methyl]-1H-indole Dihydrochloride
Show/Hide
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C23H31Cl2N3O3S
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1
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| 1 |
Ki = 5.7 nM
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CP0479257
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1-(3-trifluoromethyl benzenesulfonyl)-5-(4-ethylpiperazin-1-yl-methyl)-1H-indole
Show/Hide
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C22H24F3N3O2S
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1
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| 1 |
Ki = 5.72 nM
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CP0185708
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1-(4-Isopropyl benzenesulfonyl)-5-(4-ethylpiperazin-1-yl-methyl)-1H-indole
Show/Hide
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C24H31N3O2S
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1
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| 1 |
Ki = 5.81 nM
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CP0523303
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6-methoxy-N,N-dimethyl-9-(4-methylphenyl)sulfonyl-1,2,3,4-tetrahydrocarbazol-3-amine
Show/Hide
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C22H26N2O3S
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1
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| 1 |
Ki = 5.89 nM
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CP0149650
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2-(1-benzyl-1H-indol-3-yl)-N,N-dimethylethanamine
Show/Hide
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C19H22N2
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1
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| 1 |
Ki = 6 nM
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CP0481336
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6-(4-methylpiperazin-1-yl)-1-propan-2-ylsulfonyl-4-[4-(trifluoromethyl)phenyl]pyrrolo[2,3-b]pyridine
Show/Hide
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C22H25F3N4O2S
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1
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| 1 |
Ki = 6 nM
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CP0566558
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3-[(4-methylpiperazin-1-yl)methyl]-1-(4-propan-2-ylphenyl)sulfonylindole
Show/Hide
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C23H29N3O2S
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1
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| 1 |
Ki = 6 nM
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CP0854698
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1-(Phenylsulfonyl)-3-[(4-methyl-1-piperazinyl)methyl]-1H-indole Dihydrochloride
Show/Hide
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C20H25Cl2N3O2S
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1
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| 1 |
Ki = 6 nM
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CP0073332
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2-ethyl-3-[(3-fluorophenyl)methyl]-7-piperazin-1-ylimidazo[4,5-b]pyridine
Show/Hide
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C19H22FN5
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1
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| 1 |
Ki = 6 nM
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CP0430229
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3-[5-methoxy-3-(1,2,3,6-tetrahydropyridin-4-yl)indol-1-yl]sulfonylisoquinoline
Show/Hide
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C23H21N3O3S
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1
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| 1 |
Ki = 6 nM
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CP0517109
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4-[1-(2,5-dichlorophenoxy)propyl]-6-(4-methylpiperazin-1-yl)-1,3,5-triazin-2-amine
Show/Hide
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C17H22Cl2N6O
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2
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| 1 |
Ki = 6 nM
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| 2 |
Ki = 6.026 nM
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CP0517110
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4-[1-(2,3-dichlorophenoxy)propyl]-6-(4-methylpiperazin-1-yl)-1,3,5-triazin-2-amine
Show/Hide
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C17H22Cl2N6O
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1
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| 1 |
Ki = 6 nM
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CP0440756
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N-[4-[4-(1,2-benzoxazol-3-yl)piperazin-1-yl]butyl]naphthalene-2-sulfonamide
Show/Hide
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C25H28N4O3S
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1
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| 1 |
Ki = 6.2 nM
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CP0307921
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N-[4-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]butyl]-1-benzothiophene-2-sulfonamide
Show/Hide
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C24H26FN3O3S2
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1
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| 1 |
Ki = 6.5 nM
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CP0543203
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1-(2-bromophenyl)sulfonyl-3-[(4-ethylpiperazin-1-yl)methyl]-5-methoxyindole
Show/Hide
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C22H26BrN3O3S
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1
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| 1 |
Ki = 6.7 nM
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CP0326089
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3-(4-fluorophenyl)sulfonyl-5,7-dimethyl-2-methylsulfanylpyrazolo[1,5-a]pyrimidine
Show/Hide
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C15H14FN3O2S2
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1
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| 1 |
Ki = 6.761 nM
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CP0486926
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Biphenyl-4-sulfonic acid [3-(1-methyl-piperidin-4-yl)-1H-indol-5-yl]-amide
Show/Hide
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C26H27N3O2S
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1
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| 1 |
Ki = 6.8 nM
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CP0499884
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9-(4-methoxyphenyl)sulfonyl-N,N-dimethyl-6-methylsulfanyl-1,2,3,4-tetrahydrocarbazol-3-amine
Show/Hide
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C22H26N2O3S2
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1
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| 1 |
Ki = 6.89 nM
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CP0376131
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4-(4-benzenesulfonylphenyl)piperazine
Show/Hide
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C16H18N2O2S
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2
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| 1 |
Ki = 6.9 nM
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| 2 |
Ki = 10.8 nM
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CP0389008
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1-(benzenesulfonyl)-4-[4-[4-(4-fluorophenoxy)butyl]piperazin-1-yl]indole
Show/Hide
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C28H30FN3O3S
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1
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| 1 |
Ki = 6.9 nM
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CP0860732
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1-[(4-Fluorophenyl)sulfonyl]-5-methoxy-3-[(1-piperazinyl)methyl]-1H-indole Dimesylate
Show/Hide
|
C22H30FN3O9S3
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1
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| 1 |
Ki = 6.9 nM
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CP0559656
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1-(4-aminophenylsulfonyl)-N-methyl-1H-indol-6-amine
Show/Hide
|
C15H15N3O2S
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1
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| 1 |
Ki = 7 nM
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CP0407461
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4-[6-(4-methylpiperazin-1-yl)-1-(2-methylpropylsulfonyl)pyrrolo[2,3-b]pyridin-4-yl]benzonitrile
Show/Hide
|
C23H27N5O2S
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1
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| 1 |
Ki = 7 nM
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CP0848183
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1-methyl-4-[1-(oxane-4-sulfonyl)-4-[4-(trifluoromethyl)phenyl]-1H-pyrrolo[2,3-b]pyridin-6-yl]piperazine
Show/Hide
|
C24H27F3N4O3S
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1
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| 1 |
Ki = 7 nM
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CP0417452
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3-[(3-chlorophenyl)methyl]-2-ethyl-7-piperazin-1-ylimidazo[4,5-b]pyridine
Show/Hide
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C19H22ClN5
|
1
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| 1 |
Ki = 7 nM
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CP0457522
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4-[5-[[2-(1H-indol-3-yl)ethylamino]methyl]furan-2-yl]phenol
Show/Hide
|
C21H20N2O2
|
1
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| 1 |
Ki = 7 nM
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CP0540657
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7-[3-(1,2,3,6-tetrahydropyridin-4-yl)indol-1-yl]sulfonylquinoline
Show/Hide
|
C22H19N3O2S
|
1
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| 1 |
Ki = 7 nM
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CP0451728
|
1-[(3-chlorophenyl)methyl]-4-piperazin-1-ylindole
Show/Hide
|
C19H20ClN3
|
1
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| 1 |
Ki = 7 nM
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CP0395881
|
3,4-dichloro-N-[3-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]propyl]benzenesulfonamide
Show/Hide
|
C21H22Cl2FN3O3S
|
1
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| 1 |
Ki = 7.1 nM
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CP0442277
|
N-[3-[2-(dibutylamino)ethyl]-1H-indol-5-yl]naphthalene-1-sulfonamide
Show/Hide
|
C28H35N3O2S
|
1
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| 1 |
Ki = 7.2 nM
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CP0337657
|
7-[4-[4-[1-[(3-chlorophenyl)methyl]indol-4-yl]piperazin-1-yl]butoxy]-3,4-dihydro-1H-quinolin-2-one
Show/Hide
|
C32H35ClN4O2
|
1
|
| 1 |
Ki = 7.3 nM
|
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|
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CP0460863
|
2-[1-(2,5-dimethoxyphenyl)sulfonyl-4-methoxyindol-3-yl]-N,N-dimethylethanamine
Show/Hide
|
C21H26N2O5S
|
1
|
| 1 |
Ki = 7.4 nM
|
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CP0526064
|
6-bromo-N,N-dimethyl-9-(4-propan-2-ylphenyl)sulfonyl-1,2,3,4-tetrahydrocarbazol-3-amine
Show/Hide
|
C23H27BrN2O2S
|
1
|
| 1 |
Ki = 7.5 nM
|
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CP0548818
|
1-(benzenesulfonyl)-3-(piperazin-1-ylmethyl)indole
Show/Hide
|
C19H21N3O2S
|
1
|
| 1 |
Ki = 7.5 nM
|
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CP0429443
|
1-(benzenesulfonyl)-4-[4-(3-phenoxypropyl)piperazin-1-yl]indole
Show/Hide
|
C27H29N3O3S
|
1
|
| 1 |
Ki = 7.6 nM
|
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CP0524498
|
1-(2-Bromo benzenesulfonyl)-5-(piperazin-1-yl-methyl)-1H-indole
Show/Hide
|
C19H20BrN3O2S
|
1
|
| 1 |
Ki = 7.77 nM
|
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CP0904273
|
1-(4-Fluoro benzenesulfonyl)-5-methoxy-3-(4-methyl-[1,4]diazepane-1-yl methyl)-1H-indole Dihydrochloride
Show/Hide
|
C22H28Cl2FN3O3S
|
1
|
| 1 |
Ki = 7.79 nM
|
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CP0915708
|
1-Benzenesulfonyl-3-(R)-1-pyrrolidin-2-ylmethyl-1H-indole oxalic acid
Show/Hide
|
C21H22N2O6S
|
1
|
| 1 |
Ki = 7.8 nM
|
|
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CP0394458
|
5-methoxy-3-[(4-methylpiperazin-1-yl)methyl]-1-naphthalen-1-ylsulfonylindole
Show/Hide
|
C25H27N3O3S
|
1
|
| 1 |
Ki = 7.8 nM
|
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CP0543200
|
1-(2-fluorophenyl)sulfonyl-3-[(4-methylpiperazin-1-yl)methyl]indole
Show/Hide
|
C20H22FN3O2S
|
1
|
| 1 |
Ki = 7.8 nM
|
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CP0948409
|
1-Benzenesulfonyl-(4-piperazin-1-ylmethyl)-1H-indole dihydrochloride
Show/Hide
|
C19H23Cl2N3O2S
|
1
|
| 1 |
Ki = 7.84 nM
|
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CP0523523
|
1-(4-methylphenyl)sulfonyl-4-[(4-methylpiperazin-1-yl)methyl]indole
Show/Hide
|
C21H25N3O2S
|
1
|
| 1 |
Ki = 7.92 nM
|
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CP0490323
|
6-tert-butyl-4-(2-fluorophenyl)sulfonyl-8-piperazin-1-yl-2,3-dihydro-1,4-benzoxazine
Show/Hide
|
C22H28FN3O3S
|
1
|
| 1 |
Ki = 7.943 nM
|
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CP0488180
|
9-(benzenesulfonyl)-6,8-difluoro-N,N-dimethyl-1,2,3,4-tetrahydrocarbazol-3-amine
Show/Hide
|
C20H20F2N2O2S
|
1
|
| 1 |
Ki = 7.95 nM
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CP0397846
|
2-[5-methoxy-1-(4-methoxyphenyl)sulfonylindol-3-yl]-N,N-dimethylethanamine
Show/Hide
|
C20H24N2O4S
|
1
|
| 1 |
Ki = 8 nM
|
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CP0485371
|
N-[(4-chlorophenyl)methyl]-2-nitro-5-piperazin-1-ylaniline
Show/Hide
|
C17H19ClN4O2
|
1
|
| 1 |
Ki = 8 nM
|
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CP0374729
|
5-(Dimethylamino)-N-(4-methoxy-3-piperazin-1-ylphenyl)naphthalene-1-sulfonamide
Show/Hide
|
C23H28N4O3S
|
1
|
| 1 |
Ki = 8 nM
|
|
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CP0847305
|
1-[1-(2-methoxyethanesulfonyl)-4-[4-(trifluoromethyl)phenyl]-1H-pyrrolo[2,3-b]pyridin-6-yl]-4-methylpiperazine
Show/Hide
|
C22H25F3N4O3S
|
1
|
| 1 |
Ki = 8 nM
|
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|
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CP0159262
|
5-methyl-4-(1-naphthalen-1-ylsulfonylindol-3-yl)-1H-imidazol-2-amine;hydrochloride
Show/Hide
|
C22H19ClN4O2S
|
1
|
| 1 |
Ki = 8 nM
|
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CP0576836
|
3-[5-methoxy-3-(1,2,3,6-tetrahydropyridin-4-yl)indol-1-yl]sulfonylquinoline
Show/Hide
|
C23H21N3O3S
|
1
|
| 1 |
Ki = 8 nM
|
|
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CP0499461
|
9-(2-bromophenyl)sulfonyl-6-chloro-N,N-dimethyl-1,2,3,4-tetrahydrocarbazol-3-amine
Show/Hide
|
C20H20BrClN2O2S
|
1
|
| 1 |
Ki = 8.13 nM
|
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|
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CP0429485
|
N,N-dimethyl-9-(4-methylphenyl)sulfonyl-1,2,3,4-tetrahydrocarbazol-3-amine
Show/Hide
|
C21H24N2O2S
|
1
|
| 1 |
Ki = 8.28 nM
|
|
|
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CP0511342
|
1-(2-Bromo benzenesulfonyl)-5-(4-methylpiperazin-1-yl-methyl)-1H-indole
Show/Hide
|
C20H22BrN3O2S
|
1
|
| 1 |
Ki = 8.3 nM
|
|
|
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CP0913136
|
N-Acetyl-2-(phenylsulfonyl)-5-(piperazin-1-yl)aniline hydrochloride
Show/Hide
|
C18H22ClN3O3S
|
1
|
| 1 |
Ki = 8.3 nM
|
|
|
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CP0443754
|
1-(2-bromo-4-methoxyphenyl)sulfonyl-4-[(4-methylpiperazin-1-yl)methyl]indole
Show/Hide
|
C21H24BrN3O3S
|
1
|
| 1 |
Ki = 8.58 nM
|
|
|
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CP0393704
|
1-(4-fluorophenyl)sulfonyl-3-[(4-methylpiperazin-1-yl)methyl]indole
Show/Hide
|
C20H22FN3O2S
|
1
|
| 1 |
Ki = 8.76 nM
|
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|
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CP0447214
|
N-[4-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]butyl]naphthalene-1-sulfonamide
Show/Hide
|
C26H28FN3O3S
|
1
|
| 1 |
Ki = 8.8 nM
|
|
|
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CP0566559
|
1-(benzenesulfonyl)-3-[(4-ethylpiperazin-1-yl)methyl]-5-methoxyindole
Show/Hide
|
C22H27N3O3S
|
1
|
| 1 |
Ki = 8.8 nM
|
|
|
|
CP0526069
|
9-(benzenesulfonyl)-N,N-dimethyl-1,2,3,4-tetrahydrocarbazol-3-amine
Show/Hide
|
C20H22N2O2S
|
1
|
| 1 |
Ki = 8.82 nM
|
|
|
|
CP0450842
|
5-[(2R)-2-[2-[4-(1-benzothiophen-4-yl)piperazin-1-yl]ethyl]pyrrolidin-1-yl]sulfonylisoquinoline
Show/Hide
|
C27H30N4O2S2
|
1
|
| 1 |
Ki = 9 nM
|
|
|
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CP0420831
|
4-[1-(3-fluorophenyl)sulfonyl-5-methoxyindol-3-yl]-5-methyl-1H-imidazol-2-amine;hydrochloride
Show/Hide
|
C19H18ClFN4O3S
|
1
|
| 1 |
Ki = 9 nM
|
|
|
|
CP0424449
|
N-[4-[1-(3-fluorophenyl)sulfonyl-5-methoxyindol-3-yl]-5-methyl-1H-imidazol-2-yl]propanamide
Show/Hide
|
C22H21FN4O4S
|
1
|
| 1 |
Ki = 9 nM
|
|
|
|
CP0440884
|
5-[1-(3-fluorophenyl)sulfonyl-5-methoxyindol-3-yl]-1H-imidazol-2-amine;hydrochloride
Show/Hide
|
C18H16ClFN4O3S
|
1
|
| 1 |
Ki = 9 nM
|
|
|
|
CP0566208
|
4-(5-methoxy-1-naphthalen-2-ylsulfonylindol-3-yl)-5-methyl-1H-imidazol-2-amine;hydrochloride
Show/Hide
|
C23H21ClN4O3S
|
1
|
| 1 |
Ki = 9 nM
|
|
|
|
CP0554271
|
7-[5-chloro-3-(1,2,3,6-tetrahydropyridin-4-yl)indol-1-yl]sulfonylquinoline
Show/Hide
|
C22H18ClN3O2S
|
1
|
| 1 |
Ki = 9 nM
|
|
|
|
CP0932598
|
3-((S)-1-Methyl-pyrrolidin-2-ylmethyl)-1H-indole hydrochloride
Show/Hide
|
C14H19ClN2
|
1
|
| 1 |
Ki = 9.1 nM
|
|
|
|
CP0565986
|
9-(2-chlorophenyl)sulfonyl-N,N-dimethyl-1,2,3,4-tetrahydrocarbazol-3-amine
Show/Hide
|
C20H21ClN2O2S
|
1
|
| 1 |
Ki = 9.15 nM
|
|
|
|
CP0405051
|
5,7-dichloro-3-(4-(diethylamino)phenyl)-3-methylquinoline-2,4(1H,3H)-dione
Show/Hide
|
C20H20Cl2N2O2
|
1
|
| 1 |
Ki = 9.2 nM
|
|
|
|
CP0394461
|
1-(4-bromophenyl)sulfonyl-5-fluoro-3-[(4-methylpiperazin-1-yl)methyl]indole
Show/Hide
|
C20H21BrFN3O2S
|
1
|
| 1 |
Ki = 9.2 nM
|
|
|
|
CP0566565
|
4-chloro-3-[(4-methylpiperazin-1-yl)methyl]-1-(4-propan-2-ylphenyl)sulfonylindole
Show/Hide
|
C23H28ClN3O2S
|
1
|
| 1 |
Ki = 9.2 nM
|
|
|
|
CP0469211
|
3,5-Dichloro-N-[3-(2-diethylamino-ethyl)-1H-indol-5-yl]-benzenesulfonamide
Show/Hide
|
C20H23Cl2N3O2S
|
1
|
| 1 |
Ki = 9.3 nM
|
|
|
|
CP0462735
|
1-(4-Chlorobenzenesulfonyl)-3-chloro-5-(4-methyl piperazin-1-yl-methyl)-1H-indole
Show/Hide
|
C20H21Cl2N3O2S
|
1
|
| 1 |
Ki = 9.33 nM
|
|
|
|
CP0479921
|
2-[1-(2,5-dimethoxyphenyl)sulfonyl-6-methoxyindol-3-yl]-N,N-dimethylethanamine
Show/Hide
|
C21H26N2O5S
|
1
|
| 1 |
Ki = 9.5 nM
|
|
|
|
CP0475987
|
3-(4-methoxyphenyl)sulfonyl-N,5,7-trimethylpyrazolo[1,5-a]pyrimidin-2-amine
Show/Hide
|
C16H18N4O3S
|
1
|
| 1 |
Ki = 9.55 nM
|
|
|
|
CP0375963
|
5-Chloro-naphthalene-1-sulfonic acid [3-(1-methyl-piperidin-4-yl)-1H-indol-5-yl]-amide
Show/Hide
|
C24H24ClN3O2S
|
1
|
| 1 |
Ki = 9.6 nM
|
|
|
|
CP0574460
|
1-(4-methylphenyl)sulfonyl-3-[(4-methylpiperazin-1-yl)methyl]indole
Show/Hide
|
C21H25N3O2S
|
1
|
| 1 |
Ki = 9.6 nM
|
|
|
|
CP0381429
|
6-Chloro-imidazo[2,1-b]thiazole-5-sulfonic acid [1-(2-pyrrolidin-1-yl-ethyl)-1H-indol-5-yl]-amide
Show/Hide
|
C19H20ClN5O2S2
|
1
|
| 1 |
Ki = 9.8 nM
|
|
|
|
CP0570515
|
1-(4-fluorophenyl)sulfonyl-4-[(4-methylpiperazin-1-yl)methyl]indole
Show/Hide
|
C20H22FN3O2S
|
1
|
| 1 |
Ki = 9.89 nM
|
|
|
|
CP0921245
|
3-Benzyl-1-((R)-1-methyl-pyrrolidin-2-ylmethyl)-1H-indole oxalic acid
Show/Hide
|
C23H26N2O4
|
1
|
| 1 |
Ki = 9.9 nM
|
|
|
|
CP0445063
|
2-[3-[4-[1-[(3-fluorophenyl)methyl]indol-4-yl]piperazin-1-yl]propoxy]benzamide
Show/Hide
|
C29H31FN4O2
|
1
|
| 1 |
Ki = 9.9 nM
|
|
|
|
CP0467210
|
4-(3-fluorophenyl)sulfonyl-8-piperazin-1-yl-2,3-dihydro-1,4-benzoxazine
Show/Hide
|
C18H20FN3O3S
|
1
|
| 1 |
Ki = 10 nM
|
|
|
|
CP0039676
|
4-indol-1-ylsulfonylaniline
Show/Hide
|
C14H12N2O2S
|
1
|
| 1 |
Ki = 10 nM
|
|
|
|
CP0174706
|
6-chloro-N-[3-[2-(dimethylamino)ethyl]-1H-inden-5-yl]imidazo[2,1-b][1,3]thiazole-5-sulfonamide
Show/Hide
|
C18H19ClN4O2S2
|
1
|
| 1 |
Ki = 10 nM
|
|
|
|
CP0435386
|
N-[4-[1-(benzenesulfonyl)-5-methoxyindol-3-yl]-5-methyl-1H-imidazol-2-yl]acetamide
Show/Hide
|
C21H20N4O4S
|
1
|
| 1 |
Ki = 10 nM
|
|
|
|
CP0435403
|
4-(5-methoxy-1-naphthalen-1-ylsulfonylindol-3-yl)-5-methyl-1H-imidazol-2-amine;hydrochloride
Show/Hide
|
C23H21ClN4O3S
|
1
|
| 1 |
Ki = 10 nM
|
|
|
|
CP0435406
|
N-[4-(5-methoxy-1-naphthalen-1-ylsulfonylindol-3-yl)-5-methyl-1H-imidazol-2-yl]acetamide
Show/Hide
|
C25H22N4O4S
|
1
|
| 1 |
Ki = 10 nM
|
|
|
|
CP0519609
|
5-[1-(benzenesulfonyl)indol-3-yl]-1H-imidazol-2-amine;hydrochloride
Show/Hide
|
C17H15ClN4O2S
|
1
|
| 1 |
Ki = 10 nM
|
|
|
|
CP0521247
|
N-[4-(5-methoxy-1-naphthalen-1-ylsulfonylindol-3-yl)-5-methyl-1H-imidazol-2-yl]propanamide
Show/Hide
|
C26H24N4O4S
|
1
|
| 1 |
Ki = 10 nM
|
|
|
|
CP0546255
|
1-(2-bromophenyl)sulfonyl-3-[(4-methylpiperazin-1-yl)methyl]indole
Show/Hide
|
C20H22BrN3O2S
|
1
|
| 1 |
Ki = 10.2 nM
|
|
|
|
CP0543205
|
1-(4-bromophenyl)sulfonyl-5-methoxy-3-[(4-methylpiperazin-1-yl)methyl]indole
Show/Hide
|
C21H24BrN3O3S
|
1
|
| 1 |
Ki = 10.3 nM
|
|
|
|
CP0429486
|
9-(2-fluorophenyl)sulfonyl-N,N-dimethyl-1,2,3,4-tetrahydrocarbazol-3-amine
Show/Hide
|
C20H21FN2O2S
|
1
|
| 1 |
Ki = 10.4 nM
|
|
|
|
CP0932400
|
1-(4-Methylbenzenesulfonyl)-4-(piperazin-1-ylmethyl)-1H-indole dihydrochloride
Show/Hide
|
C20H25Cl2N3O2S
|
1
|
| 1 |
Ki = 10.72 nM
|
|
|
|
CP0538194
|
2-(4-methoxy-1-(phenylsulfonyl)-1H-indol-3-yl)-N,N-dimethylethanamine
Show/Hide
|
C19H22N2O3S
|
1
|
| 1 |
Ki = 11 nM
|
|
|
|
CP0462736
|
1-(4-Methyl benzenesulfonyl)-5-(4-ethylpiperazin-1-yl-methyl)-1H-indole
Show/Hide
|
C22H27N3O2S
|
1
|
| 1 |
Ki = 11 nM
|
|
|
|
CP0389009
|
1-(benzenesulfonyl)-4-[4-[4-(2-propan-2-yloxyphenoxy)butyl]piperazin-1-yl]indole
Show/Hide
|
C31H37N3O4S
|
1
|
| 1 |
Ki = 11 nM
|
|
|
|
CP0377152
|
4-(4-ethylphenyl)-6-(4-methylpiperazin-1-yl)-1-(2-methylpropylsulfonyl)pyrrolo[2,3-b]pyridine
Show/Hide
|
C24H32N4O2S
|
1
|
| 1 |
Ki = 11 nM
|
|
|
|
CP0415732
|
4-[(2R)-2-[2-[4-(1-benzothiophen-4-yl)piperazin-1-yl]ethyl]pyrrolidin-1-yl]sulfonylisoquinoline
Show/Hide
|
C27H30N4O2S2
|
1
|
| 1 |
Ki = 11 nM
|
|
|
|
CP0402158
|
4-(4-methylpiperazin-1-yl)-6-[(5-methyl-2-propan-2-ylphenoxy)methyl]-1,3,5-triazin-2-amine
Show/Hide
|
C19H28N6O
|
1
|
| 1 |
Ki = 11 nM
|
|
|
|
CP0430231
|
5-[5-chloro-3-(1,2,3,6-tetrahydropyridin-4-yl)indol-1-yl]sulfonylquinoline
Show/Hide
|
C22H18ClN3O2S
|
1
|
| 1 |
Ki = 11 nM
|
|
|
|
CP0554276
|
3-[5-chloro-3-(1,2,3,6-tetrahydropyridin-4-yl)indol-1-yl]sulfonylquinoline
Show/Hide
|
C22H18ClN3O2S
|
1
|
| 1 |
Ki = 11 nM
|
|
|
|
CP0471354
|
4-[1-(3,5-dichlorophenoxy)propyl]-6-(4-methylpiperazin-1-yl)-1,3,5-triazin-2-amine
Show/Hide
|
C17H22Cl2N6O
|
1
|
| 1 |
Ki = 11 nM
|
|
|
|
CP0443753
|
4-[(4-methylpiperazin-1-yl)methyl]-1-(4-propan-2-ylphenyl)sulfonylindole
Show/Hide
|
C23H29N3O2S
|
1
|
| 1 |
Ki = 11.13 nM
|
|
|
|
CP0499166
|
1-(2-Chloro-5-trifluoromethyl benzenesulfonyl)-5-(4-methylpiperazin-1-yl-methyl)-1H-indole
Show/Hide
|
C21H21ClF3N3O2S
|
1
|
| 1 |
Ki = 11.3 nM
|
|
|
|
CP0521045
|
3-[(4-methylpiperazin-1-yl)methyl]-1-naphthalen-1-ylsulfonylindole
Show/Hide
|
C24H25N3O2S
|
1
|
| 1 |
Ki = 11.5 nM
|
|
|
|
CP0854700
|
1-[(4-Isopropylphenyl)sulfonyl]-4-methoxy-3-[(4-methyl-1-piperazinyl)methyl]-1H-indole Dihydrochloride
Show/Hide
|
C24H33Cl2N3O3S
|
1
|
| 1 |
Ki = 11.6 nM
|
|
|
|
CP0485370
|
5-(4-methylpiperazin-1-yl)-2-nitro-N-(1-phenylethyl)benzenamine
Show/Hide
|
C19H24N4O2
|
1
|
| 1 |
Ki = 12 nM
|
|
|
|
CP0499883
|
N,N-dimethyl-2-[1-(2-phenylethyl)indol-3-yl]ethanamine
Show/Hide
|
C20H24N2
|
1
|
| 1 |
Ki = 12 nM
|
|
|
|
CP0469585
|
4-(2,5-dimethylthiophen-3-yl)-6-(4-methylpiperazin-1-yl)-1-(2-methylpropylsulfonyl)pyrrolo[2,3-b]pyridine
Show/Hide
|
C22H30N4O2S2
|
1
|
| 1 |
Ki = 12 nM
|
|
|
|
CP0558334
|
1-(2-bromophenyl)sulfonyl-5-fluoro-3-[(4-methylpiperazin-1-yl)methyl]indole
Show/Hide
|
C20H21BrFN3O2S
|
1
|
| 1 |
Ki = 12 nM
|
|
|
|
CP0554278
|
3-[3-(1,2,3,6-tetrahydropyridin-4-yl)indol-1-yl]sulfonylisoquinoline
Show/Hide
|
C22H19N3O2S
|
1
|
| 1 |
Ki = 12 nM
|
|
|
|
CP0451281
|
4-[1-(2,5-dichlorophenoxy)butyl]-6-(4-methylpiperazin-1-yl)-1,3,5-triazin-2-amine
Show/Hide
|
C18H24Cl2N6O
|
1
|
| 1 |
Ki = 12 nM
|
|
|
|
CP0486973
|
6-chloro-N,N-dimethyl-9-[3-(trifluoromethyl)phenyl]sulfonyl-1,2,3,4-tetrahydrocarbazol-3-amine
Show/Hide
|
C21H20ClF3N2O2S
|
1
|
| 1 |
Ki = 12.2 nM
|
|
|
|
CP0176560
|
5,7-dichloro-3-(4-hydroxyphenyl)-3-methylquinoline-2,4(1H,3H)-dione
Show/Hide
|
C16H11Cl2NO3
|
1
|
| 1 |
Ki = 12.3 nM
|
|
|
|
CP0487328
|
1-(2,4-Difluoro benzenesulfonyl)-5-(4-ethylpiperazin-1-yl-methyl)-1H-indole
Show/Hide
|
C21H23F2N3O2S
|
1
|
| 1 |
Ki = 12.4 nM
|
|
|
|
CP0874093
|
rac-N,N-Dimethyl[9-(4-fluorobenzenesulfonyl)-2,3,4,9-tetrahydro-1H-carbazol-3-yl]amine hydrochloride
Show/Hide
|
C20H22ClFN2O2S
|
1
|
| 1 |
Ki = 12.5 nM
|
|
|
|
CP0453999
|
4-(benzenesulfonyl)-8-piperazin-1-yl-2,3-dihydro-1,4-benzoxazine
Show/Hide
|
C18H21N3O3S
|
1
|
| 1 |
Ki = 12.59 nM
|
|
|
|
CP0080436
|
4-Amino-N-(2,6-bis-methylamino-pyridin-4-yl)-benzenesulfonamide
Show/Hide
|
C13H17N5O2S
|
3
|
| 1 |
Ki = 12.6 nM
|
|
|
| 2 |
Ki = 14.8 nM
|
|
|
| 3 |
Ki = 512 nM
|
|
|
|
CP0445066
|
2-[3-[4-[1-[(3-chlorophenyl)methyl]indol-4-yl]piperazin-1-yl]propoxy]benzamide
Show/Hide
|
C29H31ClN4O2
|
1
|
| 1 |
Ki = 12.6 nM
|
|
|
|
CP0549040
|
4-[1-(2,5-dichlorophenoxy)ethyl]-6-(4-methylpiperazin-1-yl)-1,3,5-triazin-2-amine
Show/Hide
|
C16H20Cl2N6O
|
2
|
| 1 |
Ki = 12.88 nM
|
|
|
| 2 |
Ki = 13 nM
|
|
|
|
CP0528041
|
2-(1-(4-methoxyphenylsulfonyl)-1H-indol-3-yl)-N,N-dimethylethanamine
Show/Hide
|
C19H22N2O3S
|
1
|
| 1 |
Ki = 13 nM
|
|
|
|
CP0071154
|
2-(5-methoxy-1H-indol-3-yl)-N,N-dimethyl-ethanamine
Show/Hide
|
C13H18N2O
|
3
|
| 1 |
Ki = 13 nM
|
|
|
| 2 |
Ki = 16 nM
|
|
|
| 3 |
Ki = 78 nM
|
|
|
|
CP0496954
|
1-Naphthyl(4-piperazin-1-yl-1H-benzimidazol-2-yl)methanone
Show/Hide
|
C22H20N4O
|
1
|
| 1 |
Ki = 13 nM
|
|
|
|
CP0447122
|
N-[3-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]propyl]-3-methylbenzenesulfonamide
Show/Hide
|
C22H26FN3O3S
|
1
|
| 1 |
Ki = 13 nM
|
|
|
|
CP0447218
|
N-[4-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]butyl]-1-benzothiophene-3-sulfonamide
Show/Hide
|
C24H26FN3O3S2
|
1
|
| 1 |
Ki = 13 nM
|
|
|
|
CP0489949
|
N-[3-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]propyl]-1-benzothiophene-3-sulfonamide
Show/Hide
|
C23H24FN3O3S2
|
1
|
| 1 |
Ki = 13 nM
|
|
|
|
CP0379281
|
7-[4-[4-(1-benzylindol-4-yl)piperazin-1-yl]butoxy]-3,4-dihydro-1H-quinolin-2-one
Show/Hide
|
C32H36N4O2
|
1
|
| 1 |
Ki = 13 nM
|
|
|
|
CP0389653
|
3-[(3-fluorophenyl)methyl]-7-piperazin-1-yl-2-propan-2-ylimidazo[4,5-b]pyridine
Show/Hide
|
C20H24FN5
|
1
|
| 1 |
Ki = 13 nM
|
|
|
|
CP0396080
|
5-[(2R)-2-[2-[4-(1-benzothiophen-4-yl)piperazin-1-yl]ethyl]pyrrolidin-1-yl]sulfonylquinoline
Show/Hide
|
C27H30N4O2S2
|
1
|
| 1 |
Ki = 13 nM
|
|
|
|
CP0519611
|
N-[5-methyl-4-(1-naphthalen-1-ylsulfonylindol-3-yl)-1H-imidazol-2-yl]acetamide
Show/Hide
|
C24H20N4O3S
|
1
|
| 1 |
Ki = 13 nM
|
|
|
|
CP0494155
|
3-[3-(1,2,3,6-tetrahydropyridin-4-yl)indol-1-yl]sulfonylquinoline
Show/Hide
|
C22H19N3O2S
|
1
|
| 1 |
Ki = 13 nM
|
|
|
|
CP0917676
|
rac-N-Methyl[6-methoxy-9-(3-trifluoromethylphenylsulfonyl)-2,3,4,9-tetrahydro-1H-carbazol-3-yl]amine hydrochloride
Show/Hide
|
C21H22ClF3N2O3S
|
1
|
| 1 |
Ki = 13.1 nM
|
|
|
|
CP0570514
|
1-(3-chlorophenyl)sulfonyl-4-[(4-methylpiperazin-1-yl)methyl]indole
Show/Hide
|
C20H22ClN3O2S
|
1
|
| 1 |
Ki = 13.17 nM
|
|
|
|
CP0499460
|
N,N-dimethyl-9-(4-methylphenyl)sulfonyl-6-methylsulfanyl-1,2,3,4-tetrahydrocarbazol-3-amine
Show/Hide
|
C22H26N2O2S2
|
1
|
| 1 |
Ki = 13.8 nM
|
|
|
|
CP0486890
|
2-[1-(benzenesulfonyl)indol-3-yl]-N,N-diethylethanamine
Show/Hide
|
C20H24N2O2S
|
1
|
| 1 |
Ki = 14 nM
|
|
|
|
CP0421348
|
4-[5-[[2-(4-methoxy-1H-indol-3-yl)ethylamino]methyl]furan-2-yl]phenol
Show/Hide
|
C22H22N2O3
|
1
|
| 1 |
Ki = 14 nM
|
|
|
|
CP0144741
|
4-[1-(benzenesulfonyl)indol-3-yl]-5-methyl-1H-imidazol-2-amine;hydrochloride
Show/Hide
|
C18H17ClN4O2S
|
1
|
| 1 |
Ki = 14 nM
|
|
|
|
CP0438431
|
N-[4-[1-(benzenesulfonyl)-5-methoxyindol-3-yl]-5-methyl-1H-imidazol-2-yl]propanamide
Show/Hide
|
C22H22N4O4S
|
1
|
| 1 |
Ki = 14 nM
|
|
|
|
CP0519613
|
N-[4-[1-(3-fluorophenyl)sulfonyl-5-methoxyindol-3-yl]-5-methyl-1H-imidazol-2-yl]acetamide
Show/Hide
|
C21H19FN4O4S
|
1
|
| 1 |
Ki = 14 nM
|
|
|
|
CP0555129
|
6-[5-methoxy-3-(1,2,3,6-tetrahydropyridin-4-yl)indol-1-yl]sulfonylquinoline
Show/Hide
|
C23H21N3O3S
|
1
|
| 1 |
Ki = 14 nM
|
|
|
|
CP0016259
|
4-(benzenesulfonyl)-N,11-dimethyl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1,3,5,8-tetraen-5-amine
Show/Hide
|
C17H19N5O2S
|
1
|
| 1 |
Ki = 14.3 nM
|
|
|
|
CP0860733
|
1-[(2-Bromophenyl)sulfonyl]-4-methoxy-3-[(4-methyl-1-piperazinyl)methyl]-1H-indole Dihydrochloride
Show/Hide
|
C21H26BrCl2N3O3S
|
1
|
| 1 |
Ki = 14.3 nM
|
|
|
|
CP0493948
|
1-(4-Fluoro benzenesulfonyl)-5-(4-methylpiperazin-1-yl-methyl)-1H-indole
Show/Hide
|
C20H22FN3O2S
|
1
|
| 1 |
Ki = 14.6 nM
|
|
|
|
CP0293425
|
5-(benzenesulfonyl)-11-methyl-4-methylsulfanyl-2,3,7,11-tetrazatricyclo[7.4.0.02,6]trideca-1(9),3,5,7-tetraene
Show/Hide
|
C17H18N4O2S2
|
1
|
| 1 |
Ki = 14.8 nM
|
|
|
|
CP0376127
|
N-[1-[2-(dimethylamino)ethyl]indol-4-yl]naphthalene-2-sulfonamide
Show/Hide
|
C22H23N3O2S
|
1
|
| 1 |
Ki = 14.9 nM
|
|
|
|
CP0511341
|
1-(4-Isopropyl benzenesulfonyl)-5-(piperazin-1-yl-methyl)-1H-indole
Show/Hide
|
C22H27N3O2S
|
1
|
| 1 |
Ki = 14.9 nM
|
|
|
|
CP0496006
|
2-(6-methoxy-1-(phenylsulfonyl)-1H-indol-3-yl)-N,N-dimethylethanamine
Show/Hide
|
C19H22N2O3S
|
1
|
| 1 |
Ki = 15 nM
|
|
|
|
CP0444937
|
2-[1-(benzenesulfonyl)pyrrol-3-yl]-N,N-dimethylethanamine
Show/Hide
|
C14H18N2O2S
|
1
|
| 1 |
Ki = 15 nM
|
|
|
|
CP0483771
|
N-[3-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]propyl]-3,4-dichlorobenzenesulfonamide
Show/Hide
|
C20H22Cl2N4O2S2
|
1
|
| 1 |
Ki = 15 nM
|
|
|
|
CP0473914
|
1-cyclohexylsulfonyl-6-(4-methylpiperazin-1-yl)-4-[4-(trifluoromethyl)phenyl]pyrrolo[2,3-b]pyridine
Show/Hide
|
C25H29F3N4O2S
|
1
|
| 1 |
Ki = 15 nM
|
|
|
|
CP0438422
|
N-[5-methyl-4-(1-naphthalen-1-ylsulfonylindol-3-yl)-1H-imidazol-2-yl]propanamide
Show/Hide
|
C25H22N4O3S
|
1
|
| 1 |
Ki = 15 nM
|
|
|
|
CP0521240
|
N-[4-[1-(benzenesulfonyl)indol-6-yl]-5-methyl-1H-imidazol-2-yl]acetamide
Show/Hide
|
C20H18N4O3S
|
1
|
| 1 |
Ki = 15 nM
|
|
|
|
CP0392353
|
5-Chloro-3-methyl-benzo[b]thiophene-2-sulfonic acid [3-(2-morpholin-4-yl-ethyl)-1H-indol-5-yl]-amide
Show/Hide
|
C23H24ClN3O3S2
|
1
|
| 1 |
Ki = 15.1 nM
|
|
|
|
CP0488179
|
9-(4-bromophenyl)sulfonyl-6-methoxy-N,N-dimethyl-1,2,3,4-tetrahydrocarbazol-3-amine
Show/Hide
|
C21H23BrN2O3S
|
1
|
| 1 |
Ki = 15.1 nM
|
|
|
|
CP0429490
|
9-(4-bromophenyl)sulfonyl-N,N-dimethyl-1,2,3,4-tetrahydrocarbazol-3-amine
Show/Hide
|
C20H21BrN2O2S
|
1
|
| 1 |
Ki = 15.5 nM
|
|
|
|
CP0517741
|
6-fluoro-N,N-dimethyl-9-(4-propan-2-ylphenyl)sulfonyl-1,2,3,4-tetrahydrocarbazol-3-amine
Show/Hide
|
C23H27FN2O2S
|
1
|
| 1 |
Ki = 15.5 nM
|
|
|
|
CP0569573
|
5-methoxy-1-(4-methylphenyl)sulfonyl-3-[(4-methylpiperazin-1-yl)methyl]indole
Show/Hide
|
C22H27N3O3S
|
1
|
| 1 |
Ki = 15.5 nM
|
|
|
|
CP0449694
|
9-(benzenesulfonyl)-6-fluoro-N,N-dimethyl-1,2,3,4-tetrahydrocarbazol-3-amine
Show/Hide
|
C20H21FN2O2S
|
1
|
| 1 |
Ki = 15.7 nM
|
|
|
|
CP0444753
|
4-[1-(2,3-dichlorophenoxy)ethyl]-6-(4-methylpiperazin-1-yl)-1,3,5-triazin-2-amine
Show/Hide
|
C16H20Cl2N6O
|
2
|
| 1 |
Ki = 15.85 nM
|
|
|
| 2 |
Ki = 16 nM
|
|
|
|
CP0509785
|
2-(1-Naphthylmethyl)-4-piperazin-1-yl-1H-benzimidazole
Show/Hide
|
C22H22N4
|
1
|
| 1 |
Ki = 16 nM
|
|
|
|
CP0429322
|
1-(benzenesulfonyl)-4-[4-(4-phenoxybutyl)piperazin-1-yl]indole
Show/Hide
|
C28H31N3O3S
|
1
|
| 1 |
Ki = 16 nM
|
|
|
|
CP0420134
|
6-(4-methylpiperazin-1-yl)-1-(2-methylpropylsulfonyl)-4-phenylpyrrolo[2,3-b]pyridine
Show/Hide
|
C22H28N4O2S
|
1
|
| 1 |
Ki = 16 nM
|
|
|
|
CP0440882
|
N-[4-[1-(benzenesulfonyl)-5-methoxyindol-3-yl]-5-ethyl-1H-imidazol-2-yl]propanamide
Show/Hide
|
C23H24N4O4S
|
1
|
| 1 |
Ki = 16 nM
|
|
|
|
CP0498135
|
9-(benzenesulfonyl)-6-chloro-N,N-dimethyl-1,2,3,4-tetrahydrocarbazol-3-amine
Show/Hide
|
C20H21ClN2O2S
|
1
|
| 1 |
Ki = 16.1 nM
|
|
|
|
CP0540716
|
1-(3-chlorophenyl)sulfonyl-3-[(4-methylpiperazin-1-yl)methyl]indole
Show/Hide
|
C20H22ClN3O2S
|
1
|
| 1 |
Ki = 16.3 nM
|
|
|
|
CP0485627
|
4-[1-(2,5-dichlorophenoxy)pentyl]-6-(4-methylpiperazin-1-yl)-1,3,5-triazin-2-amine
Show/Hide
|
C19H26Cl2N6O
|
2
|
| 1 |
Ki = 16.98 nM
|
|
|
| 2 |
Ki = 17 nM
|
|
|
|
CP0509160
|
6-Chloro-N-[2-methyl-3-(2-pyrrolidin-1-ylethyl)-1H-inden-5-yl]imidazo[2,1-b][1,3]thiazole-5-sulfonamide
Show/Hide
|
C21H23ClN4O2S2
|
1
|
| 1 |
Ki = 17 nM
|
|
|
|
CP0500575
|
N-[3-(2-aminoethyl)-4-methoxyphenyl]benzenesulfonamide
Show/Hide
|
C15H18N2O3S
|
1
|
| 1 |
Ki = 17 nM
|
|
|
|
CP0440922
|
N-[4-[4-(1,2-benzoxazol-3-yl)piperazin-1-yl]butyl]-5-fluoro-3-methyl-1-benzothiophene-2-sulfonamide
Show/Hide
|
C24H27FN4O3S2
|
1
|
| 1 |
Ki = 17 nM
|
|
|
|
CP0548761
|
5-bromo-1-(4-fluorophenyl)sulfonyl-3-[(4-methylpiperazin-1-yl)methyl]indole
Show/Hide
|
C20H21BrFN3O2S
|
1
|
| 1 |
Ki = 17 nM
|
|
|
|
CP0493761
|
N-[4-[1-(benzenesulfonyl)indol-6-yl]-5-methyl-1H-imidazol-2-yl]propanamide
Show/Hide
|
C21H20N4O3S
|
1
|
| 1 |
Ki = 17 nM
|
|
|
|
CP0925352
|
rac-N-Methyl[9-(3-trifluoromethylphenylsulfonyl)-2,3,4,9-tetrahydro-1H-carbazol-3-yl]amine hydrochloride
Show/Hide
|
C20H20ClF3N2O2S
|
1
|
| 1 |
Ki = 17.12 nM
|
|
|
|
CP0543206
|
5-chloro-1-(4-fluorophenyl)sulfonyl-3-[(4-methylpiperazin-1-yl)methyl]indole
Show/Hide
|
C20H21ClFN3O2S
|
1
|
| 1 |
Ki = 17.5 nM
|
|
|
|
CP0479256
|
1-[4-(Isopropyl benzenesulfonyl)]-5-(4-methylpiperazin-1-yl-methyl)-1H-indole
Show/Hide
|
C23H29N3O2S
|
1
|
| 1 |
Ki = 17.9 nM
|
|
|
|
CP0441385
|
1-(2,3-Dichloro benzenesulfonyl)-5-(4-methylpiperazin-1-yl-methyl)-1H-indole
Show/Hide
|
C20H21Cl2N3O2S
|
1
|
| 1 |
Ki = 18 nM
|
|
|
|
CP0395872
|
N-[4-[4-(1,2-benzoxazol-3-yl)piperazin-1-yl]butyl]-6-chloronaphthalene-2-sulfonamide
Show/Hide
|
C25H27ClN4O3S
|
1
|
| 1 |
Ki = 18 nM
|
|
|
|
CP0476721
|
5-[(2R)-2-[2-[4-(5-chloro-1H-indol-3-yl)-3,6-dihydro-2H-pyridin-1-yl]ethyl]pyrrolidin-1-yl]sulfonylquinoline
Show/Hide
|
C28H29ClN4O2S
|
1
|
| 1 |
Ki = 18 nM
|
|
|
|
CP0489683
|
N-[5-[1-(benzenesulfonyl)-5-methoxyindol-3-yl]-1H-imidazol-2-yl]acetamide
Show/Hide
|
C20H18N4O4S
|
1
|
| 1 |
Ki = 18 nM
|
|
|
|
CP0430230
|
4-[5-chloro-3-(1,2,3,6-tetrahydropyridin-4-yl)indol-1-yl]sulfonylisoquinoline
Show/Hide
|
C22H18ClN3O2S
|
1
|
| 1 |
Ki = 18 nM
|
|
|
|
CP0494154
|
7-[2-methyl-3-(1,2,3,6-tetrahydropyridin-4-yl)indol-1-yl]sulfonylquinoline
Show/Hide
|
C23H21N3O2S
|
1
|
| 1 |
Ki = 18 nM
|
|
|
|
CP0526065
|
6-chloro-N,N-dimethyl-9-(4-methylphenyl)sulfonyl-1,2,3,4-tetrahydrocarbazol-3-amine
Show/Hide
|
C21H23ClN2O2S
|
1
|
| 1 |
Ki = 18.09 nM
|
|
|
|
CP0472389
|
5-methoxy-1-(4-methoxyphenyl)sulfonyl-3-[(4-methylpiperazin-1-yl)methyl]indole
Show/Hide
|
C22H27N3O4S
|
1
|
| 1 |
Ki = 18.3 nM
|
|
|
|
CP0392445
|
2-[5-(6-Chloro-imidazo[2,1-b]thiazole-5-sulfonylamino)-1H-indol-3-yl]-N,N-dimethyl-2-oxo-acetamide
Show/Hide
|
C17H14ClN5O4S2
|
1
|
| 1 |
Ki = 18.4 nM
|
|
|
|
CP0574464
|
1-(4-fluorophenyl)sulfonyl-4-methoxy-3-[(4-methylpiperazin-1-yl)methyl]indole
Show/Hide
|
C21H24FN3O3S
|
1
|
| 1 |
Ki = 18.4 nM
|
|
|
|
CP0442265
|
N-[1-(2-pyrrolidin-1-ylethyl)indol-6-yl]naphthalene-1-sulfonamide
Show/Hide
|
C24H25N3O2S
|
1
|
| 1 |
Ki = 18.6 nM
|
|
|
|
CP0853829
|
6-chloro-3-(3-chlorophenylsulfonyl)-N2,5-dimethylpyrazolo[1,5-a]pyrimidine-2,7-diamine
Show/Hide
|
C14H13Cl2N5O2S
|
1
|
| 1 |
Ki = 18.62 nM
|
|
|
|
CP0558333
|
1-(2-bromophenyl)sulfonyl-3-[(4-methylpiperazin-1-yl)methyl]indol-5-ol
Show/Hide
|
C20H22BrN3O3S
|
1
|
| 1 |
Ki = 18.7 nM
|
|
|
|
CP0428022
|
N-[2-(2-methoxyphenoxy)ethyl]-5-(4-methylpiperazin-1-yl)-2-nitroaniline
Show/Hide
|
C20H26N4O4
|
1
|
| 1 |
Ki = 19 nM
|
|
|
|
CP0405273
|
1-(3-bromophenyl)sulfonyl-3-[(4-methylpiperazin-1-yl)methyl]indole
Show/Hide
|
C20H22BrN3O2S
|
1
|
| 1 |
Ki = 19 nM
|
|
|
|
CP0424446
|
4-[1-(benzenesulfonyl)-5-methoxyindol-3-yl]-5-ethyl-1H-imidazol-2-amine;hydrochloride
Show/Hide
|
C20H21ClN4O3S
|
1
|
| 1 |
Ki = 19 nM
|
|
|
|
CP0402157
|
4-[1-(2-chlorophenyl)sulfanylethyl]-6-(4-methylpiperazin-1-yl)-1,3,5-triazin-2-amine
Show/Hide
|
C16H21ClN6S
|
1
|
| 1 |
Ki = 19 nM
|
|
|
|
CP0436439
|
5-Methoxy-1-(naphthalene-2-sulfonyl)-3-(1,2,3,6-tetrahydro-pyridin-4-yl)-1H-indole
Show/Hide
|
C24H22N2O3S
|
1
|
| 1 |
Ki = 19 nM
|
|
|
|
CP0456324
|
N-[1-[2-(dimethylamino)ethyl]indol-6-yl]naphthalene-1-sulfonamide
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C22H23N3O2S
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1
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| 1 |
Ki = 19.8 nM
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CP0526063
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6-methoxy-9-(4-methoxyphenyl)sulfonyl-N,N-dimethyl-1,2,3,4-tetrahydrocarbazol-3-amine
Show/Hide
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C22H26N2O4S
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1
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| 1 |
Ki = 19.8 nM
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CP0533095
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2-(1-(4-chlorobenzyl)-1H-indol-3-yl)-N,N-dimethylethanamine
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C19H21ClN2
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1
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| 1 |
Ki = 20 nM
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CP0443351
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5-chloro-3-methyl-N-(2-methyl-3-(2-(pyrrolidin-1-yl)ethyl)-1H-inden-5-yl)benzo[b]thiophene-2-sulfonamide
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C25H27ClN2O2S2
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1
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| 1 |
Ki = 20 nM
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CP0260687
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7-[4-[4-[1-[(3-fluorophenyl)methyl]indol-4-yl]piperazin-1-yl]butoxy]-3,4-dihydro-1H-quinolin-2-one
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C32H35FN4O2
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1
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| 1 |
Ki = 20 nM
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CP0566560
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3-[(4-ethylpiperazin-1-yl)methyl]-1-(4-fluorophenyl)sulfonyl-5-methoxyindole
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C22H26FN3O3S
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1
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| 1 |
Ki = 20 nM
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CP0461825
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4-(4-Methylpiperazin-1-yl)-6-(naphthalen-1-ylmethyl)-1,3,5-triazin-2-amine (12)
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C19H22N6
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1
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| 1 |
Ki = 20 nM
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CP0417454
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3-[(3-chlorophenyl)methyl]-7-piperazin-1-yl-2-propan-2-ylimidazo[4,5-b]pyridine
Show/Hide
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C20H24ClN5
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1
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| 1 |
Ki = 20 nM
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CP0056386
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5-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-6-chloroindolin-2-one
Show/Hide
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C21H21ClN4OS
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2
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| 1 |
Ki = 20 nM
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| 2 |
Ki = 63.1 nM
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CP0530224
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6-[3-(1,2,3,6-tetrahydropyridin-4-yl)indol-1-yl]sulfonylquinoline
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C22H19N3O2S
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1
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| 1 |
Ki = 20 nM
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CP0554273
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3-[2-methyl-3-(1,2,3,6-tetrahydropyridin-4-yl)indol-1-yl]sulfonylisoquinoline
Show/Hide
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C23H21N3O2S
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1
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| 1 |
Ki = 20 nM
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CP0523302
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9-(4-methoxyphenyl)sulfonyl-N,N-dimethyl-1,2,3,4-tetrahydrocarbazol-3-amine
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C21H24N2O3S
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1
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| 1 |
Ki = 20.4 nM
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CP0490740
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1-(4-aminophenylsulfonyl)-N-methyl-1H-indol-4-amine
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C15H15N3O2S
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1
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| 1 |
Ki = 21 nM
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CP0416927
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N-[3-(2-aminoethyl)phenyl]benzenesulfonamide
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C14H16N2O2S
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1
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| 1 |
Ki = 21 nM
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CP0457581
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3-[(3-chlorophenyl)methyl]-2-methyl-7-piperazin-1-ylimidazo[4,5-b]pyridine
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C18H20ClN5
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1
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| 1 |
Ki = 21 nM
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CP0457523
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4-[5-[[2-(5-methoxy-2-methyl-1H-indol-3-yl)ethylamino]methyl]furan-2-yl]phenol
Show/Hide
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C23H24N2O3
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1
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| 1 |
Ki = 21 nM
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CP0144745
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4-[1-(benzenesulfonyl)-5-methoxyindol-3-yl]-N-(2,2-difluoroethyl)-5-methyl-1H-imidazol-2-amine
Show/Hide
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C21H20F2N4O3S
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1
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| 1 |
Ki = 21 nM
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CP0519612
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4-[1-(benzenesulfonyl)-5-methoxyindol-3-yl]-N-benzyl-5-methyl-1H-imidazol-2-amine
Show/Hide
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C26H24N4O3S
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1
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| 1 |
Ki = 21 nM
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CP0537415
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4-(4-methylpiperazin-1-yl)-6-(1-phenoxypropyl)-1,3,5-triazin-2-amine
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C17H24N6O
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1
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| 1 |
Ki = 21 nM
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CP0378291
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N-[3-(1-methylpiperidin-4-yl)-1H-indol-5-yl]quinoline-8-sulfonamide
Show/Hide
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C23H24N4O2S
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1
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| 1 |
Ki = 21.2 nM
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CP0468503
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N-[3-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]propyl]-3-methylbenzenesulfonamide
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C21H26N4O2S2
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1
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| 1 |
Ki = 22 nM
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CP0398682
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7-[4-[4-(1-benzylindol-3-yl)-3,6-dihydro-2H-pyridin-1-yl]butoxy]-3,4-dihydro-1H-quinolin-2-one
Show/Hide
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C33H35N3O2
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1
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| 1 |
Ki = 22 nM
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CP0559558
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4-[6-(4-methylpiperazin-1-yl)-1-(2-methylpropylsulfonyl)pyrrolo[2,3-b]pyridin-4-yl]phenol
Show/Hide
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C22H28N4O3S
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1
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| 1 |
Ki = 22 nM
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CP0548789
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4-(1H-indol-3-ylmethyl)-6-(4-methylpiperazin-1-yl)-1,3,5-triazin-2-amine
Show/Hide
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C17H21N7
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1
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| 1 |
Ki = 22 nM
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CP0430228
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7-[6-chloro-3-(1,2,3,6-tetrahydropyridin-4-yl)indol-1-yl]sulfonylquinoline
Show/Hide
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C22H18ClN3O2S
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1
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| 1 |
Ki = 22 nM
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CP0392082
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US8618114, 1.2.12(11)
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C19H26N6O2S
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1
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| 1 |
Ki = 22.39 nM
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CP0443105
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N-[3-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]propyl]-1,3-benzothiazole-4-sulfonamide
Show/Hide
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C22H23FN4O3S2
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1
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| 1 |
Ki = 23 nM
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CP0481184
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N-[4-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]butyl]-4-(trifluoromethoxy)benzenesulfonamide
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C23H25F4N3O4S
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1
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| 1 |
Ki = 23 nM
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CP0411521
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2-[3-[4-[1-[(2-fluorophenyl)methyl]indol-4-yl]piperazin-1-yl]propoxy]benzamide
Show/Hide
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C29H31FN4O2
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1
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| 1 |
Ki = 23 nM
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CP0396618
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4-[(2R)-2-[2-[4-(5-chloro-1H-indol-3-yl)-3,6-dihydro-2H-pyridin-1-yl]ethyl]pyrrolidin-1-yl]sulfonylisoquinoline
Show/Hide
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C28H29ClN4O2S
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1
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| 1 |
Ki = 23 nM
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CP0438427
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N-[4-(5-methoxy-1-naphthalen-2-ylsulfonylindol-3-yl)-5-methyl-1H-imidazol-2-yl]acetamide
Show/Hide
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C25H22N4O4S
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1
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| 1 |
Ki = 23 nM
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CP0402156
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4-[1-(2-chlorophenoxy)ethyl]-6-(4-methylpiperazin-1-yl)-1,3,5-triazin-2-amine
Show/Hide
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C16H21ClN6O
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1
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| 1 |
Ki = 23 nM
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CP0567761
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4-[1-(2,3-dichlorophenoxy)butyl]-6-(4-methylpiperazin-1-yl)-1,3,5-triazin-2-amine
Show/Hide
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C18H24Cl2N6O
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1
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| 1 |
Ki = 23 nM
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CP0381775
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1-(4-bromophenyl)sulfonyl-4-[(4-methylpiperazin-1-yl)methyl]indole
Show/Hide
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C20H22BrN3O2S
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1
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| 1 |
Ki = 23.41 nM
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CP0565527
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1-(2-bromophenyl)sulfonyl-4-chloro-3-[(4-methylpiperazin-1-yl)methyl]indole
Show/Hide
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C20H21BrClN3O2S
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1
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| 1 |
Ki = 23.5 nM
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CP0441724
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2-[3-[4-(1-benzylindol-4-yl)piperazin-1-yl]propoxy]benzamide
Show/Hide
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C29H32N4O2
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1
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| 1 |
Ki = 24 nM
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CP0472072
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6-(4-methylpiperazin-1-yl)-1-(2-methylpropylsulfonyl)-4-[2-(trifluoromethyl)phenyl]pyrrolo[2,3-b]pyridine
Show/Hide
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C23H27F3N4O2S
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1
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| 1 |
Ki = 24 nM
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CP0540669
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4-(5-methoxy-3-piperidin-4-ylindol-1-yl)sulfonylisoquinoline
Show/Hide
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C23H23N3O3S
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1
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| 1 |
Ki = 24 nM
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CP0551733
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5-Chloro-thiophene-2-sulfonic acid [3-(1-methyl-piperidin-4-yl)-1H-indol-5-yl]-amide
Show/Hide
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C18H20ClN3O2S2
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1
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| 1 |
Ki = 24.3 nM
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CP0517744
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9-(4-fluorophenyl)sulfonyl-6-methoxy-N,N-dimethyl-1,2,3,4-tetrahydrocarbazol-3-amine
Show/Hide
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C21H23FN2O3S
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1
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| 1 |
Ki = 24.3 nM
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CP0508846
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2-(benzenesulfonyl)-N-methylaniline
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C13H13NO2S
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1
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| 1 |
Ki = 24.3 nM
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CP0488668
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9-(4-fluorophenyl)sulfonyl-N,N-dimethyl-6-methylsulfanyl-1,2,3,4-tetrahydrocarbazol-3-amine
Show/Hide
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C21H23FN2O2S2
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1
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| 1 |
Ki = 24.9 nM
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CP0196335
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N-(furan-2-ylmethyl)-2-nitro-5-piperazin-1-ylaniline
Show/Hide
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C15H18N4O3
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1
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| 1 |
Ki = 25 nM
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CP0461307
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5-fluoro-N-[3-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]propyl]-3-methyl-1-benzothiophene-2-sulfonamide
Show/Hide
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C24H25F2N3O3S2
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1
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| 1 |
Ki = 25 nM
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CP0135185
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4-[5-[[2-(5-fluoro-1H-pyrrolo[2,3-b]pyridin-3-yl)ethylamino]methyl]furan-2-yl]phenol
Show/Hide
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C20H18FN3O2
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1
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| 1 |
Ki = 25 nM
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CP0423253
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N-[4-[1-(benzenesulfonyl)indol-3-yl]-5-methyl-1H-imidazol-2-yl]acetamide
Show/Hide
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C20H18N4O3S
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1
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| 1 |
Ki = 25 nM
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CP0548531
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1-(4-methoxyphenyl)sulfonyl-3-[(4-methylpiperazin-1-yl)methyl]indole
Show/Hide
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C21H25N3O3S
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1
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| 1 |
Ki = 25.1 nM
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CP0508301
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10-(benzenesulfonyl)-N,N,7-trimethyl-1,8,12-triazatricyclo[7.3.0.02,6]dodeca-2(6),7,9,11-tetraen-11-amine
Show/Hide
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C18H20N4O2S
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1
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| 1 |
Ki = 25.5 nM
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CP0471362
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5-(4-methylpiperazin-1-yl)-2-nitro-N-(2-(o-tolyloxy)ethyl)benzenamine
Show/Hide
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C20H26N4O3
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1
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| 1 |
Ki = 26 nM
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CP0381488
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1-(benzenesulfonyl)-4-N,6-N-dimethylindole-4,6-diamine
Show/Hide
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C16H17N3O2S
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1
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| 1 |
Ki = 26 nM
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CP0839170
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2-(6-{[(4-methyl-3,4-dihydro-2H-1,4-benzoxazine-7-yl)sulfonyl]amino}-2,3-dihydro-1H-inden-1-ylidene)hydrazinecarboximidamide hydrochloride
Show/Hide
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C19H23ClN6O3S
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1
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| 1 |
Ki = 26 nM
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CP0468502
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6-chloro-N-[3-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]propyl]naphthalene-2-sulfonamide
Show/Hide
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C25H25ClFN3O3S
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1
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| 1 |
Ki = 26 nM
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CP0499522
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3,4-dichloro-N-[4-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]butyl]benzenesulfonamide
Show/Hide
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C22H24Cl2FN3O3S
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1
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| 1 |
Ki = 26 nM
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CP0541474
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2-methyl-3-[(3-methylphenyl)methyl]-7-piperazin-1-ylimidazo[4,5-b]pyridine
Show/Hide
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C19H23N5
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1
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| 1 |
Ki = 26 nM
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CP0382741
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4-(4-methylpiperazin-1-yl)-6-(phenylsulfanylmethyl)-1,3,5-triazin-2-amine
Show/Hide
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C15H20N6S
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1
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| 1 |
Ki = 26 nM
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CP0451283
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4-[1-(3,5-dichlorophenoxy)butyl]-6-(4-methylpiperazin-1-yl)-1,3,5-triazin-2-amine
Show/Hide
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C18H24Cl2N6O
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1
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| 1 |
Ki = 26 nM
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CP0480089
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4-[1-(3,5-dichlorophenoxy)ethyl]-6-(4-methylpiperazin-1-yl)-1,3,5-triazin-2-amine
Show/Hide
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C16H20Cl2N6O
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2
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| 1 |
Ki = 26.92 nM
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| 2 |
Ki = 27 nM
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CP0471363
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1-methyl-4-(4-nitro-3-phenoxyphenyl)piperazine
Show/Hide
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C17H19N3O3
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1
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| 1 |
Ki = 27 nM
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CP0472698
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5-Chloro-N-{[5-(dimethylamino)-1-naphthyl]sulfonyl}-N-(4-methoxy-3-piperazin-1-ylphenyl)-3-methyl-1-benzothiophene-2-sulfonamide
Show/Hide
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C32H33ClN4O5S3
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1
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| 1 |
Ki = 27 nM
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CP0447211
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N-[4-[4-(1,2-benzoxazol-3-yl)piperazin-1-yl]butyl]-3-chloro-4-fluorobenzenesulfonamide
Show/Hide
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C21H24ClFN4O3S
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1
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| 1 |
Ki = 27 nM
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CP0482709
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N-[3-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]propyl]-1,3-benzothiazole-4-sulfonamide
Show/Hide
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C21H23N5O2S3
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1
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| 1 |
Ki = 27 nM
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CP0500522
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1-(Naphthalene-2-sulfonyl)-3-(1,2,3,6-tetrahydro-pyridin-4-yl)-1H-indole
Show/Hide
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C23H20N2O2S
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1
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| 1 |
Ki = 27 nM
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CP0046242
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3-chloro-1-(3-chlorophenyl)sulfonyl-4-[(4-methylpiperazin-1-yl)methyl]indole
Show/Hide
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C20H21Cl2N3O2S
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1
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| 1 |
Ki = 27.19 nM
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CP0546257
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5-bromo-3-[(4-methylpiperazin-1-yl)methyl]-1-(4-propan-2-ylphenyl)sulfonylindole
Show/Hide
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C23H28BrN3O2S
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1
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| 1 |
Ki = 27.6 nM
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CP0543507
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N-benzyl-2-nitro-5-piperazin-1-ylaniline
Show/Hide
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C17H20N4O2
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1
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| 1 |
Ki = 28 nM
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CP0549604
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4-[(3-chlorophenyl)methyl]-6-(4-methylpiperazin-1-yl)-1,3,5-triazin-2-amine
Show/Hide
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C15H19ClN6
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1
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| 1 |
Ki = 28 nM
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CP0521765
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1-(4-Chloro benzenesulfonyl)-5-(4-ethylpiperazin-1-yl-methyl)-1H-indole
Show/Hide
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C21H24ClN3O2S
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1
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| 1 |
Ki = 28.2 nM
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CP0436407
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1-(2,4-dichlorophenyl)sulfonyl-3-[(4-methylpiperazin-1-yl)methyl]indole
Show/Hide
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C20H21Cl2N3O2S
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1
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| 1 |
Ki = 28.2 nM
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CP0535837
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5,7-dichloro-3-(4-(ethylamino)phenyl)-3-methylquinoline-2,4(1H,3H)-dione
Show/Hide
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C18H16Cl2N2O2
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1
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| 1 |
Ki = 28.3 nM
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CP0446624
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10-(benzenesulfonyl)-N,N-dimethyl-1,8,12-triazatricyclo[7.3.0.02,6]dodeca-2(6),7,9,11-tetraen-11-amine
Show/Hide
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C17H18N4O2S
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1
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| 1 |
Ki = 28.8 nM
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CP0488178
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6-bromo-9-(4-methoxyphenyl)sulfonyl-N,N-dimethyl-1,2,3,4-tetrahydrocarbazol-3-amine
Show/Hide
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C21H23BrN2O3S
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1
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| 1 |
Ki = 28.99 nM
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CP0268549
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4-(1,2,3,4-Tetrahydro-carbazole-9-sulfonyl)-phenylamine
Show/Hide
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C18H18N2O2S
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1
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| 1 |
Ki = 29 nM
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CP0504961
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N,N-dimethyl-2-[1-[(4-methylphenyl)methyl]indol-3-yl]ethanamine
Show/Hide
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C20H24N2
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1
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| 1 |
Ki = 29 nM
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CP0921628
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3-Benzyl-1-((S)-1-methyl-pyrrolidin-2-ylmethyl)-1H-indole oxalic acid
Show/Hide
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C23H26N2O4
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1
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| 1 |
Ki = 29 nM
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CP0440055
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N-[4-[4-(1,2-benzoxazol-3-yl)piperazin-1-yl]butyl]-3,4-dichlorobenzenesulfonamide
Show/Hide
|
C21H24Cl2N4O3S
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1
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| 1 |
Ki = 29 nM
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CP0548030
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1-(2-chloro-4-fluorophenyl)sulfonyl-3-[(4-methylpiperazin-1-yl)methyl]indole
Show/Hide
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C20H21ClFN3O2S
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1
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| 1 |
Ki = 29 nM
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CP0416278
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3-(5-fluoro-1H-indol-3-yl)-1-[4-[4-(1H-indol-3-yl)piperidin-1-yl]butyl]pyrrolidine-2,5-dione
Show/Hide
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C29H31FN4O2
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1
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| 1 |
Ki = 29 nM
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CP0552643
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4-[1-(benzenesulfonyl)indol-3-yl]-5-ethyl-1H-imidazol-2-amine;hydrochloride
Show/Hide
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C19H19ClN4O2S
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1
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| 1 |
Ki = 29 nM
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CP0481359
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6-bromo-9-(3,4-difluorophenyl)sulfonyl-N,N-dimethyl-1,2,3,4-tetrahydrocarbazol-3-amine
Show/Hide
|
C20H19BrF2N2O2S
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1
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| 1 |
Ki = 29.01 nM
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CP0392542
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1-(4-methoxyphenyl)sulfonyl-4-[(4-methylpiperazin-1-yl)methyl]indole
Show/Hide
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C21H25N3O3S
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1
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| 1 |
Ki = 29.15 nM
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CP0393701
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1-(3-methoxyphenyl)sulfonyl-3-[(4-methylpiperazin-1-yl)methyl]indole
Show/Hide
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C21H25N3O3S
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1
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| 1 |
Ki = 29.4 nM
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CP0474330
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2-chloro-5-methoxy-3-[(4-methylpiperazin-1-yl)methyl]-1-(4-propan-2-ylphenyl)sulfonylindole
Show/Hide
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C24H30ClN3O3S
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1
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| 1 |
Ki = 29.6 nM
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CP0559068
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1-(2,4-difluorophenyl)sulfonyl-3-[(4-methylpiperazin-1-yl)methyl]indole
Show/Hide
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C20H21F2N3O2S
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1
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| 1 |
Ki = 30 nM
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CP0548792
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4-[(3-methylphenyl)methyl]-6-(4-methylpiperazin-1-yl)-1,3,5-triazin-2-amine
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C16H22N6
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1
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| 1 |
Ki = 30 nM
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CP0549093
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3-[(3-chlorophenyl)methyl]-2-pentan-3-yl-7-piperazin-1-ylimidazo[4,5-b]pyridine
Show/Hide
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C22H28ClN5
|
1
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| 1 |
Ki = 30 nM
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CP0530226
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7-(5-methoxy-3-piperidin-4-ylindol-1-yl)sulfonylquinoline
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C23H23N3O3S
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1
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| 1 |
Ki = 30 nM
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CP0103199
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5,7-dichloro-3-(3-hydroxyphenyl)-3-methylquinoline-2,4(1H,3H)-dione
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C16H11Cl2NO3
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1
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| 1 |
Ki = 30.1 nM
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CP0876596
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N,N-Dimethyl-2-(phenylsulfonyl)-5-(piperazin-1-yl)aniline hydrochloride
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C18H24ClN3O2S
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1
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| 1 |
Ki = 30.1 nM
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CP0058304
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1-(benzenesulfonyl)-3-bromo-4-[(4-methylpiperazin-1-yl)methyl]indole
Show/Hide
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C20H22BrN3O2S
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1
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| 1 |
Ki = 30.28 nM
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CP0418494
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6-Chloro-N-[3-(2-piperidin-1-ylethyl)-1H-inden-5-yl]imidazo[2,1-b][1,3]thiazole-5-sulfonamide
Show/Hide
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C21H23ClN4O2S2
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1
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| 1 |
Ki = 31 nM
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CP0489684
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N-[4-[1-(benzenesulfonyl)-5-methoxyindol-3-yl]-5-ethyl-1H-imidazol-2-yl]acetamide
Show/Hide
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C22H22N4O4S
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1
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| 1 |
Ki = 31 nM
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CP0508353
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4-chloro-1-(4-fluorophenyl)sulfonyl-3-[(4-methylpiperazin-1-yl)methyl]indole
Show/Hide
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C20H21ClFN3O2S
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1
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| 1 |
Ki = 31.2 nM
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CP0498582
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6-Chloro-imidazo[2,1-b]thiazole-5-sulfonic acid [1-(2-piperidin-1-yl-ethyl)-1H-indol-5-yl]-amide
Show/Hide
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C20H22ClN5O2S2
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1
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| 1 |
Ki = 31.4 nM
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CP0391889
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2-(3-benzylindol-1-yl)-N,N-dimethylethanamine
Show/Hide
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C19H22N2
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1
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| 1 |
Ki = 32 nM
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CP0395875
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N-[3-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]propyl]naphthalene-2-sulfonamide
Show/Hide
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C25H26FN3O3S
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1
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| 1 |
Ki = 32 nM
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CP0548694
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4-[(3,4-dichlorophenyl)methyl]-6-(4-methylpiperazin-1-yl)-1,3,5-triazin-2-amine
Show/Hide
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C15H18Cl2N6
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1
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| 1 |
Ki = 32 nM
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CP0486972
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6-fluoro-N,N-dimethyl-9-(4-methylphenyl)sulfonyl-1,2,3,4-tetrahydrocarbazol-3-amine
Show/Hide
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C21H23FN2O2S
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1
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| 1 |
Ki = 32.4 nM
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CP0517745
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6-fluoro-9-(4-fluorophenyl)sulfonyl-N,N-dimethyl-1,2,3,4-tetrahydrocarbazol-3-amine
Show/Hide
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C20H20F2N2O2S
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1
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| 1 |
Ki = 32.8 nM
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CP0371741
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2-nitro-N-phenethyl-5-(piperazin-1-yl)benzenamine
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C18H22N4O2
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1
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| 1 |
Ki = 33 nM
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CP0466976
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N-[4-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]butyl]-1-benzothiophene-2-sulfonamide
Show/Hide
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C23H26N4O2S3
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1
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| 1 |
Ki = 33 nM
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CP0412625
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2-[3-[4-[1-(benzenesulfonyl)indol-3-yl]-3,6-dihydro-2H-pyridin-1-yl]propoxy]benzamide
Show/Hide
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C29H29N3O4S
|
1
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| 1 |
Ki = 33 nM
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CP0427416
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3-[(3-chlorophenyl)methyl]-7-piperazin-1-ylimidazo[4,5-b]pyridine
Show/Hide
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C17H18ClN5
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1
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| 1 |
Ki = 33 nM
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CP0853828
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[7-(2-Dimethylamino-ethyl)-5-methyl-3-phenylsulfonylpyrazolo[1,5-a]pyrimidin-2-yl]-methyl-amine
Show/Hide
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C18H23N5O2S
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1
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| 1 |
Ki = 33.88 nM
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CP0439120
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[4-(4-methylpiperazin-1-yl)-1H-benzimidazol-2-yl]-naphthalen-1-ylmethanone
Show/Hide
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C23H22N4O
|
1
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| 1 |
Ki = 34 nM
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CP0435404
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5-[1-(benzenesulfonyl)indol-4-yl]-1H-imidazol-2-amine;hydrochloride
Show/Hide
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C17H15ClN4O2S
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1
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| 1 |
Ki = 34 nM
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CP0945735
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1-[(2-Fluorophenyl)sulfonyl]-5-hydroxy-3-[(4-methyl-1-piperazinyl)methyl]-1H-indole Dihydrochloride
Show/Hide
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C20H24Cl2FN3O3S
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1
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| 1 |
Ki = 34.9 nM
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CP0468501
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N-[3-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]propyl]-4-(trifluoromethoxy)benzenesulfonamide
Show/Hide
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C22H23F4N3O4S
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1
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| 1 |
Ki = 35 nM
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CP0486987
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N-[3-[4-(1,2-benzoxazol-3-yl)piperazin-1-yl]propyl]-1-benzothiophene-2-sulfonamide
Show/Hide
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C22H24N4O3S2
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1
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| 1 |
Ki = 35 nM
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CP0432054
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1-(benzenesulfonyl)-6-chloro-3-[(4-methylpiperazin-1-yl)methyl]indole
Show/Hide
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C20H22ClN3O2S
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1
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| 1 |
Ki = 35.7 nM
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CP0549219
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6-(4-methylpiperazin-1-yl)-1-(2-methylpropylsulfonyl)-4-pyridin-3-ylpyrrolo[2,3-b]pyridine
Show/Hide
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C21H27N5O2S
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1
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| 1 |
Ki = 36 nM
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CP0541475
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3-benzyl-2-ethyl-7-piperazin-1-ylimidazo[4,5-b]pyridine
Show/Hide
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C19H23N5
|
1
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| 1 |
Ki = 36 nM
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CP0432053
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6-methoxy-3-[(4-methylpiperazin-1-yl)methyl]-1-(4-propan-2-ylphenyl)sulfonylindole
Show/Hide
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C24H31N3O3S
|
1
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| 1 |
Ki = 36.1 nM
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CP0484614
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4-(4-Methylpiperazin-1-yl)-2-(1-naphthylmethyl)-1H-benzimidazole
Show/Hide
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C23H24N4
|
1
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| 1 |
Ki = 36.22 nM
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CP0566564
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1-(2-bromophenyl)sulfonyl-3-[(4-methylpiperazin-1-yl)methyl]-5-propan-2-yloxyindole
Show/Hide
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C23H28BrN3O3S
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1
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| 1 |
Ki = 36.3 nM
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CP0531988
|
2-(4-(benzenesulfonyl)phenyl)-1-aminoethane
Show/Hide
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C14H15NO2S
|
1
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| 1 |
Ki = 37 nM
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CP0544508
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3-[6-chloro-3-(1,2,3,6-tetrahydropyridin-4-yl)indol-1-yl]sulfonylquinoline
Show/Hide
|
C22H18ClN3O2S
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1
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| 1 |
Ki = 37 nM
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CP0293306
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3-(4-methoxyphenyl)sulfonyl-5,7-dimethyl-2-methylsulfanylpyrazolo[1,5-a]pyrimidine
Show/Hide
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C16H17N3O3S2
|
1
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| 1 |
Ki = 37.15 nM
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CP0475985
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4-(5,7-dimethyl-2-methylsulfanylpyrazolo[1,5-a]pyrimidin-3-yl)sulfonyl-N,N-dimethylaniline
Show/Hide
|
C17H20N4O2S2
|
1
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| 1 |
Ki = 37.15 nM
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CP0569572
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5-methoxy-3-[(4-methylpiperazin-1-yl)methyl]-1-[4-(trifluoromethoxy)phenyl]sulfonylindole
Show/Hide
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C22H24F3N3O4S
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1
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| 1 |
Ki = 37.8 nM
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CP0376266
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N-[3-[2-(methylamino)ethyl]phenyl]benzenesulfonamide
Show/Hide
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C15H18N2O2S
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1
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| 1 |
Ki = 38 nM
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CP0500574
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N-[4-(2-aminoethyl)phenyl]benzenesulfonamide
Show/Hide
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C14H16N2O2S
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1
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| 1 |
Ki = 38 nM
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CP0450839
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3-[4-[2-[(2R)-1-quinolin-5-ylsulfonylpyrrolidin-2-yl]ethyl]piperazin-1-yl]-1,2-benzothiazole
Show/Hide
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C26H29N5O2S2
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1
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| 1 |
Ki = 38 nM
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CP0301336
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N-[[4-[5-[4-[1-(benzenesulfonyl)indol-4-yl]piperazin-1-yl]pentoxy]phenyl]methyl]-N-methylprop-2-yn-1-amine
Show/Hide
|
C34H40N4O3S
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1
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| 1 |
Ki = 38 nM
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CP0917435
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rac-6-methoxy-9-(3-(trifluoromethyl)phenylsulfonyl)-2,3,4,9-tetrahydro-1H-carbazol-3-amine hydrochloride
Show/Hide
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C20H20ClF3N2O3S
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1
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| 1 |
Ki = 39.1 nM
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CP0471152
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4-(4-chlorophenyl)sulfonyl-8-(3,5-dimethylpiperazin-1-yl)-6-methyl-2,3-dihydro-1,4-benzoxazine
Show/Hide
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C21H26ClN3O3S
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1
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| 1 |
Ki = 39.81 nM
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CP0461294
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N-[3-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]propyl]naphthalene-2-sulfonamide
Show/Hide
|
C24H26N4O2S2
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1
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| 1 |
Ki = 40 nM
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CP0461312
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N-[3-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]propyl]-1-benzothiophene-2-sulfonamide
Show/Hide
|
C23H24FN3O3S2
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1
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| 1 |
Ki = 40 nM
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CP0396077
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3-[4-[2-[(2R)-1-isoquinolin-5-ylsulfonylpyrrolidin-2-yl]ethyl]piperazin-1-yl]-1,2-benzothiazole
Show/Hide
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C26H29N5O2S2
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1
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| 1 |
Ki = 40 nM
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CP0445918
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3-[4-[2-[(2R)-1-isoquinolin-4-ylsulfonylpyrrolidin-2-yl]ethyl]piperazin-1-yl]-1,2-benzothiazole
Show/Hide
|
C26H29N5O2S2
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1
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| 1 |
Ki = 40 nM
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CP0480619
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4-{3-methyl-1H-pyrrolo[3,2-c]pyridine-1-sulfonyl}aniline, 18
Show/Hide
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C14H13N3O2S
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1
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| 1 |
Ki = 41 nM
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CP0499462
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9-(4-bromophenyl)sulfonyl-6-chloro-N,N-dimethyl-1,2,3,4-tetrahydrocarbazol-3-amine
Show/Hide
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C20H20BrClN2O2S
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1
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| 1 |
Ki = 41.1 nM
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CP0469207
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N-[1-[2-(dimethylamino)ethyl]indol-6-yl]naphthalene-2-sulfonamide
Show/Hide
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C22H23N3O2S
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1
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| 1 |
Ki = 41.2 nM
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CP0395870
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N-[4-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]butyl]thiophene-2-sulfonamide
Show/Hide
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C19H24N4O2S3
|
1
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| 1 |
Ki = 42 nM
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CP0427391
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3-[2-(3-chlorophenyl)ethyl]-2-ethyl-7-piperazin-1-ylimidazo[4,5-b]pyridine
Show/Hide
|
C20H24ClN5
|
1
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| 1 |
Ki = 42 nM
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CP0533346
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3-[(3-methylphenyl)methyl]-2-pentan-3-yl-7-piperazin-1-ylimidazo[4,5-b]pyridine
Show/Hide
|
C23H31N5
|
1
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| 1 |
Ki = 42 nM
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CP0514093
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9-(4-bromophenyl)sulfonyl-6-fluoro-N,N-dimethyl-1,2,3,4-tetrahydrocarbazol-3-amine
Show/Hide
|
C20H20BrFN2O2S
|
1
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| 1 |
Ki = 43.5 nM
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CP0464103
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4-((3-(2-(dimethylamino)ethyl)-1H-indol-1-yl)methyl)benzenamine
Show/Hide
|
C19H23N3
|
1
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| 1 |
Ki = 44 nM
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CP0473172
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6-chloro-N-[3-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]propyl]-1-benzothiophene-2-sulfonamide
Show/Hide
|
C23H23ClFN3O3S2
|
1
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| 1 |
Ki = 44 nM
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CP0547882
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4-(5-methoxy-1-naphthalen-1-ylsulfonylindol-3-yl)-5-methyl-1,3-thiazol-2-amine
Show/Hide
|
C23H19N3O3S2
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1
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| 1 |
Ki = 44 nM
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CP0118951
|
4-Amino-N-(2,6-bis-dimethylamino-pyrimidin-4-yl)-benzenesulfonamide
Show/Hide
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C12H16N6O2S
|
4
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| 1 |
Ki = 44.7 nM
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| 2 |
Ki = 47 nM
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| 3 |
Ki = 50 nM
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| 4 |
Ki = 55 nM
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CP0449172
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2-[1-(4-chlorophenyl)sulfonyl-7-methoxyindol-3-yl]-N,N-dimethylethanamine
Show/Hide
|
C19H21ClN2O3S
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1
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| 1 |
Ki = 45 nM
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CP0447124
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N-[4-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]butyl]-6-chloro-1-benzothiophene-2-sulfonamide
Show/Hide
|
C23H25ClN4O2S3
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1
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| 1 |
Ki = 45 nM
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CP0412626
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7-[4-[4-[1-[(2-fluorophenyl)methyl]indol-4-yl]piperazin-1-yl]butoxy]-3,4-dihydro-1H-quinolin-2-one
Show/Hide
|
C32H35FN4O2
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1
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| 1 |
Ki = 45 nM
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CP0123095
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6-[5-[4-(4-chlorophenyl)piperazin-1-yl]pentyl]-2,4-dimethyl-7-phenylpurino[7,8-a]imidazole-1,3-dione
Show/Hide
|
C30H34ClN7O2
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1
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| 1 |
Ki = 45 nM
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CP0562582
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1-(3-fluorophenyl)sulfonyl-3-(1,2,3,6-tetrahydropyridin-4-yl)pyrrolo[3,2-h]quinoline
Show/Hide
|
C22H18FN3O2S
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1
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| 1 |
Ki = 45 nM
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CP0389125
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6-fluoro-3-[1-[2-[(2R)-1-quinolin-5-ylsulfonylpyrrolidin-2-yl]ethyl]piperidin-4-yl]-1,2-benzoxazole
Show/Hide
|
C27H29FN4O3S
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1
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| 1 |
Ki = 45 nM
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CP0022455
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2-Me 5-HT
Show/Hide
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C11H14N2O
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1
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| 1 |
Ki = 46 nM
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CP0877470
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1-Benzenesulfonyl-3-(S)-1-pyrrolidin-2-ylmethyl-1H-indole oxalic acid
Show/Hide
|
C21H22N2O6S
|
1
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| 1 |
Ki = 46 nM
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CP0395873
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N-[4-[4-(1,2-benzoxazol-3-yl)piperazin-1-yl]butyl]-6-chloro-1-benzothiophene-2-sulfonamide
Show/Hide
|
C23H25ClN4O3S2
|
1
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| 1 |
Ki = 46 nM
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CP0447121
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N-[4-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]butyl]-4-(trifluoromethoxy)benzenesulfonamide
Show/Hide
|
C22H25F3N4O3S2
|
1
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| 1 |
Ki = 47 nM
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CP0447213
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3-chloro-4-fluoro-N-[4-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]butyl]benzenesulfonamide
Show/Hide
|
C22H24ClF2N3O3S
|
1
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| 1 |
Ki = 48 nM
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CP0377151
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6-(4-methylpiperazin-1-yl)-1-(2-methylpropylsulfonyl)-4-[3-(trifluoromethyl)phenyl]pyrrolo[2,3-b]pyridine
Show/Hide
|
C23H27F3N4O2S
|
1
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| 1 |
Ki = 48 nM
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CP0434153
|
2-(benzenesulfonyl)-N-methyl-5-pyridin-3-ylaniline
Show/Hide
|
C18H16N2O2S
|
1
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| 1 |
Ki = 48.3 nM
|
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CP0427904
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N-[(6R)-6-(dimethylamino)-5,6,7,8-tetrahydronaphthalen-1-yl]benzenesulfonamide
Show/Hide
|
C18H22N2O2S
|
1
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| 1 |
Ki = 49 nM
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CP0430918
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4-(4-Methylpiperazin-1-yl)-2-(2-naphthylmethyl)-1H-benzimidazole
Show/Hide
|
C22H22N4
|
1
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| 1 |
Ki = 49 nM
|
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CP0488987
|
1-(3-chlorophenyl)sulfonyl-3-(1,2,3,6-tetrahydropyridin-4-yl)pyrrolo[3,2-h]quinoline
Show/Hide
|
C22H18ClN3O2S
|
1
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| 1 |
Ki = 49 nM
|
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CP0374389
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4-[1-(2-Dimethylamino-ethyl)-1H-indol-3-ylmethyl]-phenylamine
Show/Hide
|
C19H23N3
|
1
|
| 1 |
Ki = 50 nM
|
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CP0512383
|
2-(3-benzenesulfonyl)phenyl-1-aminoethane
Show/Hide
|
C14H15NO2S
|
1
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| 1 |
Ki = 50 nM
|
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CP0965119
|
1-[(4-Isopropylphenyl)sulfonyl]-5-hydroxy-3-[(4-methyl-1-piperazinyl)methyl]-1H-indole Dihydrochloride
Show/Hide
|
C23H31Cl2N3O3S
|
1
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| 1 |
Ki = 50 nM
|
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CP0440888
|
2-[1-(benzenesulfonyl)indol-3-yl]-1H-imidazo[1,2-a]pyrimidin-4-ium;bromide
Show/Hide
|
C20H15BrN4O2S
|
1
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| 1 |
Ki = 50 nM
|
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CP0489726
|
N-[5-[1-(3-fluorophenyl)sulfonyl-5-methoxyindol-3-yl]-1H-imidazol-2-yl]acetamide
Show/Hide
|
C20H17FN4O4S
|
1
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| 1 |
Ki = 50 nM
|
|
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CP0567554
|
4-[4-[4-[1-(benzenesulfonyl)indol-4-yl]piperazin-1-yl]butoxy]-N-prop-2-ynyl-2,3-dihydro-1H-inden-1-amine
Show/Hide
|
C34H38N4O3S
|
1
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| 1 |
Ki = 50 nM
|
|
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CP0033479
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(chloropromazine) [3-(2-Chloro-phenothiazin-10-yl)-propyl]-dimethyl-amine
Show/Hide
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C17H19ClN2S
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1
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| 1 |
Ki = 50.12 nM
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CP0129680
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N-[3-[2-(dimethylamino)ethyl]-2-methyl-1H-inden-5-yl]naphthalene-2-sulfonamide
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C24H26N2O2S
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1
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| 1 |
Ki = 51 nM
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CP0483720
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4-[5-[4-[1-(benzenesulfonyl)indol-4-yl]piperazin-1-yl]pentoxy]-N-prop-2-ynyl-2,3-dihydro-1H-inden-1-amine
Show/Hide
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C35H40N4O3S
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1
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| 1 |
Ki = 51 nM
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CP0451282
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4-[1-(3,5-dichlorophenoxy)pentyl]-6-(4-methylpiperazin-1-yl)-1,3,5-triazin-2-amine
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C19H26Cl2N6O
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1
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| 1 |
Ki = 51 nM
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CP0381424
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1-[1-(Naphthalene-1-sulfonyl)-piperidin-4-yl]-1,4-dihydro-benzo[d][1,3]oxazin-2-one
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C23H22N2O4S
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1
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| 1 |
Ki = 51.7 nM
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CP0443071
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N-[3-[2-(dimethylamino)ethyl]phenyl]benzenesulfonamide
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C16H20N2O2S
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1
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| 1 |
Ki = 52 nM
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CP0398681
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7-[4-[4-[1-(benzenesulfonyl)indol-3-yl]-3,6-dihydro-2H-pyridin-1-yl]butoxy]-3,4-dihydro-1H-quinolin-2-one
Show/Hide
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C32H33N3O4S
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1
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| 1 |
Ki = 52 nM
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CP0519883
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7-[4-[2-[1-(benzenesulfonyl)indol-3-yl]ethylamino]butoxy]-3,4-dihydro-1H-quinolin-2-one
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C29H31N3O4S
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1
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| 1 |
Ki = 52 nM
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CP0548695
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4-[(4-chlorophenyl)methyl]-6-(4-methylpiperazin-1-yl)-1,3,5-triazin-2-amine
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C15H19ClN6
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1
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| 1 |
Ki = 52 nM
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CP0317610
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1,1-dioxo-2-[6-[4-[3-(trifluoromethyl)phenyl]piperazin-1-yl]hexyl]-1,2-benzothiazol-3-one
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C24H28F3N3O3S
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1
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| 1 |
Ki = 52 nM
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CP0478914
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N-[6-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]hexyl]naphthalene-1-sulfonamide
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C27H32N4O2S2
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1
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| 1 |
Ki = 52 nM
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CP0099907
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6-Chloro-imidazo[2,1-b]thiazole-5-sulfonic acid [1-(2-pyrrolidin-1-yl-ethyl)-1H-indol-6-yl]-amide
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C19H20ClN5O2S2
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1
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| 1 |
Ki = 52.2 nM
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CP0235339
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N-[3-[2-(dimethylamino)ethyl]-2-methyl-1H-inden-5-yl]-1-benzothiophene-3-sulfonamide
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C22H24N2O2S2
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1
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| 1 |
Ki = 53 nM
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CP0510212
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N-[4-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]butyl]-3-chloro-4-fluorobenzenesulfonamide
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C21H24ClFN4O2S2
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1
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| 1 |
Ki = 53 nM
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CP0500049
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1-(benzenesulfonyl)-3-chloro-4-[(4-methylpiperazin-1-yl)methyl]indole
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C20H22ClN3O2S
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1
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| 1 |
Ki = 53.62 nM
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CP0135451
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2-(5-methoxy-2-phenyl-1H-indol-3-yl)-N,N-dimethylethanamine
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C19H22N2O
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1
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| 1 |
Ki = 54 nM
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CP0468506
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N-[4-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]butyl]-5-fluoro-3-methyl-1-benzothiophene-2-sulfonamide
Show/Hide
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C24H27FN4O2S3
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1
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| 1 |
Ki = 54 nM
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CP0475566
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6-(4-methylpiperazin-1-yl)-1-methylsulfonyl-4-[4-(trifluoromethyl)phenyl]pyrrolo[2,3-b]pyridine
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C20H21F3N4O2S
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1
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| 1 |
Ki = 54 nM
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CP0451727
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N-[[4-[4-[4-[1-(benzenesulfonyl)indol-4-yl]piperazin-1-yl]butoxy]phenyl]methyl]-N-methylprop-2-yn-1-amine
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C33H38N4O3S
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1
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| 1 |
Ki = 54 nM
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CP0202356
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(+/-)-5,7-dichloro-3-phenyl-3-methylquinoline-2,4-dione
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C16H11Cl2NO2
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1
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| 1 |
Ki = 54.7 nM
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CP0557796
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3-[5-[[2-(5-methoxy-1H-indol-3-yl)ethylamino]methyl]furan-2-yl]phenol
Show/Hide
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C22H22N2O3
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1
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| 1 |
Ki = 55 nM
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CP0486128
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6-Chloro-imidazo[2,1-b]thiazole-5-sulfonic acid [1-(2-dimethylamino-ethyl)-1H-indol-6-yl]-amide
Show/Hide
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C17H18ClN5O2S2
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1
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| 1 |
Ki = 55.2 nM
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CP0566561
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1-(4-fluorophenyl)sulfonyl-2-methyl-3-[(4-methylpiperazin-1-yl)methyl]indole
Show/Hide
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C21H24FN3O2S
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1
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| 1 |
Ki = 55.6 nM
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CP0468504
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N-[3-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]propyl]-4-(trifluoromethoxy)benzenesulfonamide
Show/Hide
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C21H23F3N4O3S2
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1
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| 1 |
Ki = 56 nM
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CP0566567
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4-[(2-chlorophenyl)methyl]-6-(4-methylpiperazin-1-yl)-1,3,5-triazin-2-amine
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C15H19ClN6
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1
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| 1 |
Ki = 56 nM
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CP0549596
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2-ethyl-3-[2-(3-fluorophenyl)ethyl]-7-piperazin-1-ylimidazo[4,5-b]pyridine
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C20H24FN5
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1
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| 1 |
Ki = 56 nM
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CP0495322
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2-[(3E)-3-benzylideneinden-1-yl]-N,N-dimethylethanamine
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C20H21N
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1
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| 1 |
Ki = 57 nM
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CP0411523
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2-[3-[4-[1-(benzenesulfonyl)indol-3-yl]piperidin-1-yl]propoxy]benzamide
Show/Hide
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C29H31N3O4S
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1
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| 1 |
Ki = 57 nM
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CP0466603
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3-[(2,5-difluorophenyl)methyl]-2-ethyl-7-piperazin-1-ylimidazo[4,5-b]pyridine
Show/Hide
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C19H21F2N5
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1
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| 1 |
Ki = 57 nM
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CP0526778
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N-[6-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]hexyl]naphthalene-2-sulfonamide
Show/Hide
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C27H32N4O2S2
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1
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| 1 |
Ki = 57 nM
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CP0442214
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N-[1-[2-(dimethylamino)ethyl]indol-5-yl]naphthalene-2-sulfonamide
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C22H23N3O2S
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1
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| 1 |
Ki = 57.7 nM
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CP0469197
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5-Chloro-3-methyl-benzo[b]thiophene-2-sulfonic acid [1-(2-dimethylamino-ethyl)-2-methyl-1H-indol-4-yl]-amide
Show/Hide
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C22H24ClN3O2S2
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1
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| 1 |
Ki = 57.7 nM
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CP0439117
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2-Benzyl-4-piperazin-1-yl-1H-benzimidazole
Show/Hide
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C18H20N4
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1
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| 1 |
Ki = 58 nM
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CP0511763
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1-(3-fluorophenyl)sulfonyl-3-[(4-methylpiperazin-1-yl)methyl]indole
Show/Hide
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C20H22FN3O2S
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1
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| 1 |
Ki = 58 nM
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CP0429637
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2-[6-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]hexyl]-1,1-dioxo-1,2-benzothiazol-3-one
Show/Hide
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C24H28N4O3S2
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1
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| 1 |
Ki = 58 nM
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CP0560087
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N-[(4-chlorophenyl)methyl]-5-(4-methylpiperazin-1-yl)-2-nitroaniline
Show/Hide
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C18H21ClN4O2
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1
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| 1 |
Ki = 59 nM
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CP0546258
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1-(4-bromophenyl)sulfonyl-6-chloro-3-[(4-methylpiperazin-1-yl)methyl]indole
Show/Hide
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C20H21BrClN3O2S
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1
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| 1 |
Ki = 59.7 nM
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CP0907824
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3-(R)-1-Pyrrolidin-2-ylmethyl-1H-indole hydrochloride
Show/Hide
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C13H17ClN2
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1
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| 1 |
Ki = 60 nM
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CP0391303
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4-[(2S)-2-[2-[4-(5-chloro-1H-indol-3-yl)-3,6-dihydro-2H-pyridin-1-yl]ethyl]pyrrolidin-1-yl]sulfonylisoquinoline
Show/Hide
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C28H29ClN4O2S
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1
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| 1 |
Ki = 60 nM
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CP0478896
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4-[5-[[2-(5-chloro-1H-indol-3-yl)ethylamino]methyl]furan-2-yl]phenol
Show/Hide
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C21H19ClN2O2
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1
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| 1 |
Ki = 60 nM
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CP0126804
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N-(furan-2-ylmethyl)-5-(4-methylpiperazin-1-yl)-2-nitroaniline
Show/Hide
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C16H20N4O3
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1
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| 1 |
Ki = 61 nM
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CP0447107
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N-[4-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]butyl]-6-chloronaphthalene-2-sulfonamide
Show/Hide
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C25H27ClN4O2S2
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1
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| 1 |
Ki = 61 nM
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CP0545966
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1-(3-bromophenyl)sulfonyl-3-(1,2,3,6-tetrahydropyridin-4-yl)pyrrolo[3,2-h]quinoline
Show/Hide
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C22H18BrN3O2S
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1
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| 1 |
Ki = 61 nM
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CP0417453
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3-[(2-fluorophenyl)methyl]-7-piperazin-1-yl-2-propan-2-ylimidazo[4,5-b]pyridine
Show/Hide
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C20H24FN5
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1
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| 1 |
Ki = 61 nM
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CP0443918
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2-(1H-indol-3-yl)-N-methyl-N-[(5-phenylfuran-2-yl)methyl]ethanamine
Show/Hide
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C22H22N2O
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1
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| 1 |
Ki = 61 nM
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CP0500309
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6-bromo-N,N-dimethyl-9-(2,3,4-trifluorophenyl)sulfonyl-1,2,3,4-tetrahydrocarbazol-3-amine
Show/Hide
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C20H18BrF3N2O2S
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1
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| 1 |
Ki = 61.21 nM
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CP0376265
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4-(3-benzenesulfonamidophenyl)piperazine
Show/Hide
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C16H19N3O2S
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1
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| 1 |
Ki = 62 nM
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CP0772880
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2-{6-[(2-Naphthylsulfonyl)amino]-2,3-dihydro-1H-inden-1-ylidene}hydrazinecarboximidamide hydrochloride
Show/Hide
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C20H20ClN5O2S
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1
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| 1 |
Ki = 62 nM
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CP0523324
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2-[3-[2-[1-(benzenesulfonyl)indol-3-yl]ethylamino]propoxy]benzamide
Show/Hide
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C26H27N3O4S
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1
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| 1 |
Ki = 62 nM
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CP0513852
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2-methyl-7-piperazin-1-yl-3-[[3-(trifluoromethyl)phenyl]methyl]imidazo[4,5-b]pyridine
Show/Hide
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C19H20F3N5
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1
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| 1 |
Ki = 62 nM
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CP0461314
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N-[3-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]propyl]-1-benzothiophene-2-sulfonamide
Show/Hide
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C22H24N4O2S3
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1
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| 1 |
Ki = 63 nM
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CP0230643
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1-[4-[4-(5-fluoro-1H-indol-3-yl)piperidin-1-yl]butyl]-3-(1H-indol-3-yl)pyrrolidine-2,5-dione
Show/Hide
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C29H31FN4O2
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1
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| 1 |
Ki = 63 nM
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CP0480620
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2-{1H-pyrrolo[3,2-c]pyridin-3-yl}ethan-1-amine, 9
Show/Hide
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C9H11N3
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1
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| 1 |
Ki = 64 nM
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CP0470547
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1-(2,5-dimethylphenyl)sulfonyl-3-[(4-methylpiperazin-1-yl)methyl]indole
Show/Hide
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C22H27N3O2S
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1
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| 1 |
Ki = 64 nM
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CP0548031
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1-(2,6-difluorophenyl)sulfonyl-3-[(4-methylpiperazin-1-yl)methyl]indole
Show/Hide
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C20H21F2N3O2S
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1
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| 1 |
Ki = 64 nM
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CP0478504
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4-[(4-methylphenyl)methyl]-6-(4-methylpiperazin-1-yl)-1,3,5-triazin-2-amine
Show/Hide
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C16H22N6
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1
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| 1 |
Ki = 64 nM
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CP0517794
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4-[(3-fluorophenyl)methyl]-6-(4-methylpiperazin-1-yl)-1,3,5-triazin-2-amine
Show/Hide
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C15H19FN6
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1
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| 1 |
Ki = 64 nM
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CP0431319
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N-[1-[2-(dimethylamino)ethyl]indol-4-yl]naphthalene-1-sulfonamide
Show/Hide
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C22H23N3O2S
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1
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| 1 |
Ki = 64.7 nM
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CP0440889
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4-(5-methoxy-1-naphthalen-2-ylsulfonylindol-3-yl)-5-methyl-1,3-thiazol-2-amine
Show/Hide
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C23H19N3O3S2
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1
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| 1 |
Ki = 65 nM
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CP0490641
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(2S)-2-[[4-[5-[4-[1-(benzenesulfonyl)indol-4-yl]piperazin-1-yl]pentoxy]phenyl]methylamino]propanamide
Show/Hide
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C33H41N5O4S
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1
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| 1 |
Ki = 65 nM
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CP0443102
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N-[3-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]propyl]thiophene-2-sulfonamide
Show/Hide
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C19H22FN3O3S2
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1
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| 1 |
Ki = 66 nM
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CP0439121
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2-Benzyl-4-(4-methylpiperazin-1-yl)-1H-benzimidazole
Show/Hide
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C19H22N4
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1
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| 1 |
Ki = 66.8 nM
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CP0443914
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N-[[5-(4-chlorophenyl)furan-2-yl]methyl]-2-(5-methoxy-1H-indol-3-yl)ethanamine
Show/Hide
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C22H21ClN2O2
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1
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| 1 |
Ki = 67 nM
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CP0398056
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7-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butyl]-1,3-dimethylpurine-2,6-dione;hydrochloride
Show/Hide
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C21H26Cl2N6O2
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1
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| 1 |
Ki = 68 nM
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CP0483673
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(2S)-2-[[4-[4-[4-[1-(benzenesulfonyl)indol-4-yl]piperazin-1-yl]butoxy]phenyl]methylamino]propanamide
Show/Hide
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C32H39N5O4S
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1
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| 1 |
Ki = 68 nM
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CP0558560
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5-methyl-4-(1-naphthalen-1-ylsulfonylindol-3-yl)-1,3-thiazol-2-amine
Show/Hide
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C22H17N3O2S2
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1
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| 1 |
Ki = 69 nM
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CP0449440
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3-(2-aminoethyl)-N-phenylbenzenesulfonamide
Show/Hide
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C14H16N2O2S
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1
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| 1 |
Ki = 70 nM
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CP0877506
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N-[3-(4,5-dihydro-1H-imidazol-2-ylhydrazono-2,3-dihydro-1H-inden-5-yl)-4-methyl-3,4-dihydro-2H-1,4-benzoxazine-7-sulfonamide
Show/Hide
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C21H24N6O3S
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1
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| 1 |
Ki = 70 nM
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CP0443106
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N-[4-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]butyl]-1,3-benzothiazole-4-sulfonamide
Show/Hide
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C23H25FN4O3S2
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1
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| 1 |
Ki = 70 nM
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CP0488665
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6-bromo-9-[2-chloro-5-(trifluoromethyl)phenyl]sulfonyl-N,N-dimethyl-1,2,3,4-tetrahydrocarbazol-3-amine
Show/Hide
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C21H19BrClF3N2O2S
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1
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| 1 |
Ki = 70.6 nM
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CP0447123
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N-[4-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]butyl]-3,4-dichlorobenzenesulfonamide
Show/Hide
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C21H24Cl2N4O2S2
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1
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| 1 |
Ki = 71 nM
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CP0394123
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3-(5-fluoro-1H-indol-3-yl)-1-[4-[4-(5-methoxy-1H-indol-3-yl)piperidin-1-yl]butyl]pyrrolidine-2,5-dione
Show/Hide
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C30H33FN4O3
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1
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| 1 |
Ki = 71 nM
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CP0416050
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5-[(2S)-2-[2-[4-(1-benzothiophen-4-yl)piperazin-1-yl]ethyl]pyrrolidin-1-yl]sulfonylisoquinoline
Show/Hide
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C27H30N4O2S2
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1
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| 1 |
Ki = 72 nM
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CP0416728
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2-[6-[4-(4-chlorophenyl)piperazin-1-yl]hexyl]-1,1-dioxo-1,2-benzothiazol-3-one
Show/Hide
|
C23H28ClN3O3S
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1
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| 1 |
Ki = 72 nM
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CP0416732
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2-[6-[4-(2,3-dichlorophenyl)piperazin-1-yl]hexyl]-1,1-dioxo-1,2-benzothiazol-3-one
Show/Hide
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C23H27Cl2N3O3S
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2
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| 1 |
Ki = 72 nM
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| 2 |
Ki = 920 nM
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CP0517111
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4-[1-(2,3-dichlorophenoxy)pentyl]-6-(4-methylpiperazin-1-yl)-1,3,5-triazin-2-amine
Show/Hide
|
C19H26Cl2N6O
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1
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| 1 |
Ki = 73 nM
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CP0578375
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1-(3-chlorophenyl)sulfonyl-N-[(3S)-oxolan-3-yl]pyrrolo[3,2-c]quinolin-4-amine
Show/Hide
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C21H18ClN3O3S
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1
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| 1 |
Ki = 73 nM
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CP0454144
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5-bromo-7-methoxy-3-methyl-3-phenylquinoline-2,4(1H,3H)-dione
Show/Hide
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C17H14BrNO3
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1
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| 1 |
Ki = 73.2 nM
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CP0853514
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rac-[9-(3-trifluoromethylphenylsulfonyl)-2,3,4,9-tetrahydro-1H-carbazol-3-yl]amine hydrochloride
Show/Hide
|
C19H18ClF3N2O2S
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1
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| 1 |
Ki = 73.4 nM
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CP0442264
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2-Naphthalen-1-yl-ethanesulfonic acid [1-(2-dimethylamino-ethyl)-1H-indol-6-yl]-amide
Show/Hide
|
C24H27N3O2S
|
1
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| 1 |
Ki = 74.5 nM
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CP0475996
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6-Chloro-imidazo[2,1-b]thiazole-5-sulfonic acid [1-(2-dimethylamino-ethyl)-2-methyl-1H-indol-5-yl]-amide
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C18H20ClN5O2S2
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1
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| 1 |
Ki = 74.6 nM
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CP0488895
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3-bromo-1-(3-chlorophenyl)sulfonyl-4-[(4-methylpiperazin-1-yl)methyl]indole
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C20H21BrClN3O2S
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1
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| 1 |
Ki = 75.3 nM
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CP0426437
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2-(5-methoxy-1H-indol-3-yl)-N-[[5-(3-methoxyphenyl)furan-2-yl]methyl]ethanamine
Show/Hide
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C23H24N2O3
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1
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| 1 |
Ki = 76 nM
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CP0396072
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5-[(2S)-2-[2-[4-(5-chloro-1H-indol-3-yl)-3,6-dihydro-2H-pyridin-1-yl]ethyl]pyrrolidin-1-yl]sulfonylquinoline
Show/Hide
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C28H29ClN4O2S
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1
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| 1 |
Ki = 77 nM
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CP0548569
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4-[3-[4-[1-[(3-chlorophenyl)methyl]indol-4-yl]piperazin-1-yl]propoxy]-N-prop-2-ynyl-2,3-dihydro-1H-inden-1-amine
Show/Hide
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C34H37ClN4O
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1
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| 1 |
Ki = 77 nM
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CP0525633
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3-(3-bromo-4-hydroxyphenyl)-5,7-dichloro-3-methylquinoline-2,4(1H,3H)-dione
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C16H10BrCl2NO3
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1
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| 1 |
Ki = 77.5 nM
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CP0519614
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2-[1-(benzenesulfonyl)-5-methoxyindol-3-yl]-3-methyl-1H-imidazo[1,2-a]pyridin-4-ium;bromide
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C23H20BrN3O3S
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1
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| 1 |
Ki = 78 nM
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CP0489682
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N-[5-[1-(benzenesulfonyl)indol-3-yl]-1H-imidazol-2-yl]acetamide
Show/Hide
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C19H16N4O3S
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1
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| 1 |
Ki = 79 nM
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CP0036840
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2-(5-methoxy-2-methyl-1H-indol-3-yl)-N,N-dimethylethanamine
Show/Hide
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C14H20N2O
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1
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| 1 |
Ki = 80 nM
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CP0526506
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N-[2-(4-tert-butylphenoxy)ethyl]-5-(4-methylpiperazin-1-yl)-2-nitroaniline
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C23H32N4O3
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1
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| 1 |
Ki = 80 nM
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CP0513736
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4-[(2-methylphenyl)methyl]-6-(4-methylpiperazin-1-yl)-1,3,5-triazin-2-amine
Show/Hide
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C16H22N6
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1
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| 1 |
Ki = 80 nM
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CP0427390
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3-[(4-fluorophenyl)methyl]-7-piperazin-1-yl-2-propan-2-ylimidazo[4,5-b]pyridine
Show/Hide
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C20H24FN5
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1
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| 1 |
Ki = 80 nM
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CP0518984
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3-[2-(3-chlorophenyl)ethyl]-7-piperazin-1-yl-2-propan-2-ylimidazo[4,5-b]pyridine
Show/Hide
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C21H26ClN5
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1
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| 1 |
Ki = 80 nM
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CP0422317
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1-[4-[4-(1H-indol-3-yl)piperidin-1-yl]butyl]-3-(5-methoxy-1H-indol-3-yl)pyrrolidine-2,5-dione
Show/Hide
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C30H34N4O3
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1
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| 1 |
Ki = 81 nM
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CP0396076
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5-[(2S)-2-[2-[4-(1-benzothiophen-4-yl)piperazin-1-yl]ethyl]pyrrolidin-1-yl]sulfonylquinoline
Show/Hide
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C27H30N4O2S2
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1
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| 1 |
Ki = 82 nM
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CP0555127
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7-[5-methoxy-3-(1-methyl-3,6-dihydro-2H-pyridin-4-yl)indol-1-yl]sulfonylquinoline
Show/Hide
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C24H23N3O3S
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1
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| 1 |
Ki = 82 nM
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CP0103198
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3-(3-(benzyloxy)phenyl)-5,7-dichloro-3-methylquinoline-2,4(1H,3H)-dione
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C23H17Cl2NO3
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1
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| 1 |
Ki = 82.4 nM
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CP0486995
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N-[3-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]propyl]naphthalene-1-sulfonamide
Show/Hide
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C25H26FN3O3S
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1
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| 1 |
Ki = 83 nM
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CP0441717
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2-[3-[4-[1-[(4-fluorophenyl)methyl]indol-4-yl]piperazin-1-yl]propoxy]benzamide
Show/Hide
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C29H31FN4O2
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1
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| 1 |
Ki = 83 nM
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CP0435387
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N-[4-[1-(benzenesulfonyl)-2-methylindol-3-yl]-5-methyl-1H-imidazol-2-yl]acetamide
Show/Hide
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C21H20N4O3S
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1
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| 1 |
Ki = 83 nM
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CP0519608
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4-[1-(benzenesulfonyl)-5-methoxyindol-3-yl]-5-methyl-N-(2-phenylethyl)-1H-imidazol-2-amine
Show/Hide
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C27H26N4O3S
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1
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| 1 |
Ki = 83 nM
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CP0499979
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{2-[1-(benzenesulfonyl)-1H-pyrrolo[3,2-c]pyridin-3-yl]ethyl}dimethylamine, 15
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C17H19N3O2S
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1
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| 1 |
Ki = 84 nM
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CP0461305
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N-[3-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]propyl]imidazo[1,2-a]pyridine-3-sulfonamide
Show/Hide
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C21H24N6O2S2
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1
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| 1 |
Ki = 84 nM
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CP0528128
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4-(4-benzenesulfonamidophenyl)piperazine
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C16H19N3O2S
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1
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| 1 |
Ki = 85 nM
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CP0387086
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1-[4-[4-(5-fluoro-1H-indol-3-yl)piperidin-1-yl]butyl]-3-(5-methoxy-1H-indol-3-yl)pyrrolidine-2,5-dione
Show/Hide
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C30H33FN4O3
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1
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| 1 |
Ki = 85 nM
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CP0486127
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N-[1-[2-(dimethylamino)ethyl]-2-methylindol-5-yl]naphthalene-2-sulfonamide
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C23H25N3O2S
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1
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| 1 |
Ki = 85.8 nM
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CP0188400
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9-[4-[4-(4-chlorophenyl)piperazin-1-yl]butyl]-1,3-dimethylpurino[7,8-a]pyrimidine-2,4,8-trione
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C24H28ClN7O3
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1
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| 1 |
Ki = 86 nM
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CP0339662
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N-(1,2-dimethoxy-6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-10-yl)methanesulfonamide
Show/Hide
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C20H24N2O4S
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1
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| 1 |
Ki = 86 nM
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CP0551590
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4-[1-(3,4-dichlorophenoxy)propyl]-6-(4-methylpiperazin-1-yl)-1,3,5-triazin-2-amine
Show/Hide
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C17H22Cl2N6O
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1
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| 1 |
Ki = 86 nM
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CP0473171
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N-[4-[4-(1,2-benzoxazol-3-yl)piperazin-1-yl]butyl]-3-methylbenzenesulfonamide
Show/Hide
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C22H28N4O3S
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1
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| 1 |
Ki = 87 nM
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CP0448037
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6-(4-methylpiperazin-1-yl)-1-(2-methylpropylsulfonyl)-4-(1-methylpyrazol-4-yl)pyrrolo[2,3-b]pyridine
Show/Hide
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C20H28N6O2S
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1
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| 1 |
Ki = 87 nM
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CP0382743
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4-[(2-methylphenoxy)methyl]-6-(4-methylpiperazin-1-yl)-1,3,5-triazin-2-amine
Show/Hide
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C16H22N6O
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1
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| 1 |
Ki = 87 nM
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CP0034894
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2-(5-methoxy-1H-indol-3-yl)ethanamine
Show/Hide
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C11H14N2O
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1
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| 1 |
Ki = 88 nM
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CP0548693
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4-[(2-fluorophenyl)methyl]-6-(4-methylpiperazin-1-yl)-1,3,5-triazin-2-amine
Show/Hide
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C15H19FN6
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1
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| 1 |
Ki = 88 nM
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CP0172993
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2,5,7-Triimethyl-phenylsulfonyl-pyrazolo[1,5-a]pyrimidine
Show/Hide
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C15H15N3O2S
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1
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| 1 |
Ki = 88.8 nM
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CP0042927
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7-{4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butoxy}-3,4-dihydroquinolin-2(1H)-one
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C23H27Cl2N3O2
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3
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| 1 |
Ki = 89 nM
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| 2 |
Ki = 90 nM
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| 3 |
Ki = 199.53 nM
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CP0427903
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1-phenylthio-N,N-dimethyltryptamine
Show/Hide
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C18H20N2S
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1
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| 1 |
Ki = 90 nM
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CP0457933
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N-[(6S)-6-(dimethylamino)-5,6,7,8-tetrahydronaphthalen-1-yl]benzenesulfonamide
Show/Hide
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C18H22N2O2S
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1
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| 1 |
Ki = 90 nM
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CP0373611
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5-[(3aS,6aR)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[6-[4-[5-[(5-chloro-3-methyl-1-benzothiophen-2-yl)sulfonylamino]-2-methoxyphenyl]piperazin-1-yl]hexyl]pentanamide
Show/Hide
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C36H49ClN6O5S3
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1
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| 1 |
Ki = 90 nM
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CP0421349
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2-(5-methoxy-1H-indol-3-yl)-N-[[5-(4-methoxyphenyl)furan-2-yl]methyl]ethanamine
Show/Hide
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C23H24N2O3
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1
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| 1 |
Ki = 90 nM
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CP0874539
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5-Chloro-3-methyl-benzo[b]thiophene-2-sulfonic acid [1-(2-dimethylamino-ethyl)-2,3-dihydro-1H-indol-6-yl]-amide
Show/Hide
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C21H22ClN3O2S2
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1
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| 1 |
Ki = 90.2 nM
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CP0460482
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4-[3-[(4-methylpiperazin-1-yl)methyl]indol-1-yl]sulfonylbenzonitrile
Show/Hide
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C21H22N4O2S
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1
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| 1 |
Ki = 90.5 nM
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CP0571804
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1-(2-bromophenyl)sulfonyl-3-chloro-4-[(4-methylpiperazin-1-yl)methyl]indole
Show/Hide
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C20H21BrClN3O2S
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1
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| 1 |
Ki = 90.71 nM
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CP0381395
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5-chloro-N-[1-[2-(2,3-dichlorophenoxy)ethyl]pyrrolidin-3-yl]thiophene-2-sulfonamide
Show/Hide
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C16H17Cl3N2O3S2
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1
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| 1 |
Ki = 91 nM
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CP0548529
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1-(2,5-dimethoxyphenyl)sulfonyl-3-[(4-methylpiperazin-1-yl)methyl]indole
Show/Hide
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C22H27N3O4S
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1
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| 1 |
Ki = 91 nM
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CP0443912
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2-(1H-indol-3-yl)-N-[(5-phenylfuran-2-yl)methyl]ethanamine
Show/Hide
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C21H20N2O
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1
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| 1 |
Ki = 91 nM
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CP0475614
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3-[(3-methoxyphenyl)methyl]-7-piperazin-1-yl-2-propan-2-ylimidazo[4,5-b]pyridine
Show/Hide
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C21H27N5O
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1
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| 1 |
Ki = 92 nM
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CP0529086
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3-[4-[2-[(2S)-1-isoquinolin-5-ylsulfonylpyrrolidin-2-yl]ethyl]piperazin-1-yl]-1,2-benzoxazole
Show/Hide
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C26H29N5O3S
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1
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| 1 |
Ki = 92 nM
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CP0378288
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2-[7-methoxy-1-(4-methoxyphenyl)sulfonylindol-3-yl]-N,N-dimethylethanamine
Show/Hide
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C20H24N2O4S
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1
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| 1 |
Ki = 93 nM
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CP0438423
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2-[1-(benzenesulfonyl)-5-methoxyindol-3-yl]-3-methyl-5,6,7,8-tetrahydroimidazo[1,2-a]pyrimidine;hydrochloride
Show/Hide
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C22H23ClN4O3S
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1
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| 1 |
Ki = 93 nM
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CP0485172
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2-(1-(4-chlorophenylsulfonyl)-1H-indol-3-yl)-N,N-dimethylethanamine
Show/Hide
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C18H19ClN2O2S
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1
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| 1 |
Ki = 94 nM
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CP0501216
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N-[1-[2-(dimethylamino)ethyl]indol-5-yl]naphthalene-1-sulfonamide
Show/Hide
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C22H23N3O2S
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1
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| 1 |
Ki = 94.2 nM
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CP0447262
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N-[4-[4-(1,2-benzoxazol-3-yl)piperazin-1-yl]butyl]imidazo[1,2-a]pyridine-3-sulfonamide
Show/Hide
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C22H26N6O3S
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1
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| 1 |
Ki = 95 nM
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CP0958894
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1-(2-Bromo benzenesulfonyl)-3-(piperazin-1-ylmethyl)-1H-pyrrolo[3,2-b]pyridine Dihydrochloride
Show/Hide
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C18H21BrCl2N4O2S
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1
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| 1 |
Ki = 95 nM
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CP0468977
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4-Benzyl-6-(4-methylpiperazin-1-yl)-1,3,5-triazin-2-amine (13)
Show/Hide
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C15H20N6
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1
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| 1 |
Ki = 95 nM
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CP0537421
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4-[1-(3,4-dichlorophenoxy)ethyl]-6-(4-methylpiperazin-1-yl)-1,3,5-triazin-2-amine
Show/Hide
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C16H20Cl2N6O
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1
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| 1 |
Ki = 95 nM
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CP0445256
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4-fluoro-N-[1-[2-(5,6,7,8-tetrahydronaphthalen-1-yloxy)ethyl]pyrrolidin-3-yl]benzenesulfonamide
Show/Hide
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C22H27FN2O3S
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1
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| 1 |
Ki = 96 nM
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CP0574463
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1-(4-bromophenyl)sulfonyl-3-[(4-methylpiperazin-1-yl)methyl]-5-(2,2,2-trifluoroethoxy)indole
Show/Hide
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C22H23BrF3N3O3S
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1
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| 1 |
Ki = 96.3 nM
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CP0875120
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6-Chloro-imidazo[2,1-b]thiazole-5-sulfonic acid [1-(2-diethylamino-ethyl)-2,3-dihydro-1H-indol-5-yl]-amide
Show/Hide
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C19H22ClN5O2S2
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1
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| 1 |
Ki = 97.3 nM
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CP0376680
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3-bromo-4-[(4-methylpiperazin-1-yl)methyl]-1-naphthalen-1-ylsulfonylindole
Show/Hide
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C24H24BrN3O2S
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1
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| 1 |
Ki = 97.61 nM
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CP0087385
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2-(5-Methoxy-2-methyl-1H-indol-3-yl)-ethylamine
Show/Hide
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C12H16N2O
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1
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| 1 |
Ki = 98 nM
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CP0520603
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3-chloro-4-[(4-methylpiperazin-1-yl)methyl]-1-(4-propan-2-ylphenyl)sulfonylindole
Show/Hide
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C23H28ClN3O2S
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1
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| 1 |
Ki = 99.7 nM
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CP0431024
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N-methyl-2-[3-(2-phenylethyl)-3H-inden-1-yl]ethanamine
Show/Hide
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C20H23N
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1
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| 1 |
Ki = 100 nM
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CP0480621
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dimethyl(2-{1H-pyrrolo[3,2-c]pyridin-3-yl}ethyl)amine, 14
Show/Hide
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C11H15N3
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1
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| 1 |
Ki = 100 nM
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CP0395869
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N-[4-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]butyl]-3-methylbenzenesulfonamide
Show/Hide
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C22H28N4O2S2
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1
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| 1 |
Ki = 100 nM
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CP0447097
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N-[3-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]propyl]imidazo[1,2-a]pyridine-3-sulfonamide
Show/Hide
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C22H24FN5O3S
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1
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| 1 |
Ki = 100 nM
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CP0468505
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N-[3-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]propyl]-6-chloronaphthalene-2-sulfonamide
Show/Hide
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C24H25ClN4O2S2
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1
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| 1 |
Ki = 100 nM
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CP0489950
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N-[4-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]butyl]imidazo[1,2-a]pyridine-3-sulfonamide
Show/Hide
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C23H26FN5O3S
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1
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| 1 |
Ki = 100 nM
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CP0471904
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7-[4-[4-[1-[(4-fluorophenyl)methyl]indol-4-yl]piperazin-1-yl]butoxy]-3,4-dihydro-1H-quinolin-2-one
Show/Hide
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C32H35FN4O2
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1
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| 1 |
Ki = 100 nM
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CP0559067
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1-(2,6-dichlorophenyl)sulfonyl-3-[(4-methylpiperazin-1-yl)methyl]indole
Show/Hide
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C20H21Cl2N3O2S
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1
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| 1 |
Ki = 100 nM
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CP0566566
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4-[(4-fluorophenyl)methyl]-6-(4-methylpiperazin-1-yl)-1,3,5-triazin-2-amine
Show/Hide
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C15H19FN6
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1
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| 1 |
Ki = 100 nM
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CP0121280
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7-[2-[2-(3-chlorophenyl)ethylamino]ethyl]quinolin-2-amine
Show/Hide
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C19H20ClN3
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1
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| 1 |
Ki < 100 nM
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CP0476602
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4-[1-(benzenesulfonyl)indol-3-yl]-5-methyl-1,3-thiazol-2-amine
Show/Hide
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C18H15N3O2S2
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1
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| 1 |
Ki = 100 nM
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CP0466077
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4-[2-[4-[1-[(3-chlorophenyl)methyl]indol-4-yl]piperazin-1-yl]ethoxy]-N-prop-2-ynyl-2,3-dihydro-1H-inden-1-amine
Show/Hide
|
C33H35ClN4O
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1
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| 1 |
Ki = 100 nM
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CP0469208
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N-[1-(2-pyrrolidin-1-ylethyl)indol-6-yl]naphthalene-2-sulfonamide
Show/Hide
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C24H25N3O2S
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1
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| 1 |
Ki = 100.8 nM
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CP0513851
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3-benzyl-2-methyl-7-piperazin-1-ylimidazo[4,5-b]pyridine
Show/Hide
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C18H21N5
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1
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| 1 |
Ki = 101 nM
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CP0478897
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2-(5-methoxy-1H-indol-3-yl)-N-[(5-quinolin-3-ylfuran-2-yl)methyl]ethanamine
Show/Hide
|
C25H23N3O2
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1
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| 1 |
Ki = 101 nM
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CP0548407
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2-[5-(4-naphthalen-1-ylpiperazin-1-yl)pentyl]-1,1-dioxo-1,2-benzothiazol-3-one
Show/Hide
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C26H29N3O3S
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1
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| 1 |
Ki = 101 nM
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CP0453914
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N-[1-[2-(5,6,7,8-tetrahydronaphthalen-1-yloxy)ethyl]pyrrolidin-3-yl]thiophene-2-sulfonamide
Show/Hide
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C20H26N2O3S2
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1
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| 1 |
Ki = 102 nM
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CP0486998
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4-fluoro-N-[(3R)-1-[2-(2-phenylphenoxy)ethyl]pyrrolidin-3-yl]benzenesulfonamide
Show/Hide
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C24H25FN2O3S
|
1
|
| 1 |
Ki = 102 nM
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CP0554274
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3-[6-chloro-3-(1,2,3,6-tetrahydropyridin-4-yl)indol-1-yl]sulfonylisoquinoline
Show/Hide
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C22H18ClN3O2S
|
1
|
| 1 |
Ki = 102 nM
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CP0341634
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2-methoxy-N,N,6-trimethyl-1-prop-2-enoxy-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-10-amine
Show/Hide
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C23H28N2O2
|
1
|
| 1 |
Ki = 102 nM
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CP0466254
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4-[(2S)-2-[2-[4-(1-benzothiophen-4-yl)piperazin-1-yl]ethyl]azetidin-1-yl]sulfonylisoquinoline
Show/Hide
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C26H28N4O2S2
|
1
|
| 1 |
Ki = 104 nM
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CP0391600
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1,1-dioxo-2-[6-(4-pyrimidin-2-ylpiperazin-1-yl)hexyl]-1,2-benzothiazol-3-one
Show/Hide
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C21H27N5O3S
|
2
|
| 1 |
Ki = 104 nM
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| 2 |
Ki = 5708 nM
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CP0650232
|
Doxepin
Show/Hide
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C19H21NO
|
1
|
| 1 |
Ki = 105 nM
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CP0547877
|
4-[1-(benzenesulfonyl)-5-methoxyindol-3-yl]-5-methyl-1,3-thiazol-2-amine
Show/Hide
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C19H17N3O3S2
|
1
|
| 1 |
Ki = 105 nM
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CP0496005
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N-benzyl-2-(5-methoxy-1H-indol-3-yl)-N-methylethanamine
Show/Hide
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C19H22N2O
|
1
|
| 1 |
Ki = 106 nM
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CP0549595
|
3-[(4-chlorophenyl)methyl]-7-piperazin-1-yl-2-propan-2-ylimidazo[4,5-b]pyridine
Show/Hide
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C20H24ClN5
|
1
|
| 1 |
Ki = 107 nM
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CP0435405
|
N-[4-[1-(benzenesulfonyl)-5-fluoroindol-3-yl]-5-methyl-1H-imidazol-2-yl]propanamide
Show/Hide
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C21H19FN4O3S
|
1
|
| 1 |
Ki = 107 nM
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CP0490062
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1-[1-(5-Chloro-3-methyl-benzo[b]thiophene-2-sulfonyl)-piperidin-4-yl]-1,4-dihydro-benzo[d][1,3]oxazin-2-one
Show/Hide
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C22H21ClN2O4S2
|
1
|
| 1 |
Ki = 107.4 nM
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CP0264050
|
2-(benzylamino)-4-(4-methylpiperazin-1-yl)benzonitrile
Show/Hide
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C19H22N4
|
1
|
| 1 |
Ki = 108 nM
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CP0389650
|
3-[(2-chlorophenyl)methyl]-2-pentan-3-yl-7-piperazin-1-ylimidazo[4,5-b]pyridine
Show/Hide
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C22H28ClN5
|
1
|
| 1 |
Ki = 108 nM
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CP0497449
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5-Chloro-3-methyl-benzo[b]thiophene-2-sulfonic acid [1-(2-pyrrolidin-1-yl-ethyl)-1H-indol-6-yl]-amide
Show/Hide
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C23H24ClN3O2S2
|
1
|
| 1 |
Ki = 108.8 nM
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CP0391904
|
3-(4-methylphenyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine
Show/Hide
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C14H17N3
|
1
|
| 1 |
Ki = 109 nM
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CP0487394
|
2-(4-methoxy-1H-indol-3-yl)-N-[(5-phenylfuran-2-yl)methyl]ethanamine
Show/Hide
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C22H22N2O2
|
1
|
| 1 |
Ki = 109 nM
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CP0542763
|
4-N-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butyl]-2-N-[2-(1H-indol-3-yl)ethyl]-1,3,5-triazine-2,4,6-triamine
Show/Hide
|
C27H33Cl2N9
|
1
|
| 1 |
Ki = 109 nM
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CP0482708
|
N-[3-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]propyl]-6-chloro-1-benzothiophene-2-sulfonamide
Show/Hide
|
C22H23ClN4O2S3
|
1
|
| 1 |
Ki = 110 nM
|
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CP0569024
|
3-benzyl-7-piperazin-1-ylimidazo[4,5-b]pyridine
Show/Hide
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C17H19N5
|
1
|
| 1 |
Ki = 110 nM
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CP0532785
|
2-[6-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]hexyl]benzo[de]isoquinoline-1,3-dione
Show/Hide
|
C29H30N4O2S
|
1
|
| 1 |
Ki = 110 nM
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|
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CP0402058
|
4-(4-methylpiperazin-1-yl)-6-(1-phenylselanylethyl)-1,3,5-triazin-2-amine
Show/Hide
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C16H22N6Se
|
1
|
| 1 |
Ki = 111 nM
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CP0066127
|
3-(2-chloranyl-5,6-dihydrobenzo[b][1]benzazepin-11-yl)-N,N-dimethyl-propan-1-amine;hydrochloride
Show/Hide
|
C19H23ClN2
|
1
|
| 1 |
Ki = 112 nM
|
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CP0555128
|
6-[6-chloro-3-(1,2,3,6-tetrahydropyridin-4-yl)indol-1-yl]sulfonylquinoline
Show/Hide
|
C22H18ClN3O2S
|
1
|
| 1 |
Ki = 112 nM
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CP0548680
|
4-[4-[4-[1-[(3-chlorophenyl)methyl]indol-4-yl]piperazin-1-yl]butoxy]-N-prop-2-ynyl-2,3-dihydro-1H-inden-1-amine
Show/Hide
|
C35H39ClN4O
|
1
|
| 1 |
Ki = 113 nM
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CP0371740
|
2-nitro-N-(2-phenoxyethyl)-5-(piperazin-1-yl)benzenamine
Show/Hide
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C18H22N4O3
|
1
|
| 1 |
Ki = 114 nM
|
|
|
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CP0499584
|
2-(3-phenylthio)phenyl)-1-aminoethane
Show/Hide
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C14H15NS
|
1
|
| 1 |
Ki = 115 nM
|
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|
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CP0086335
|
4-[(2S)-2-[2-[4-(1-benzothiophen-4-yl)piperazin-1-yl]ethyl]pyrrolidin-1-yl]sulfonylisoquinoline
Show/Hide
|
C27H30N4O2S2
|
1
|
| 1 |
Ki = 116 nM
|
|
|
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CP0442216
|
N-[1-[2-(diethylamino)ethyl]indol-5-yl]naphthalene-1-sulfonamide
Show/Hide
|
C24H27N3O2S
|
1
|
| 1 |
Ki = 116.2 nM
|
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CP0381423
|
N-[3-(2-morpholin-4-ylethyl)-1H-indol-5-yl]quinoline-2-sulfonamide
Show/Hide
|
C23H24N4O3S
|
1
|
| 1 |
Ki = 117 nM
|
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CP0382746
|
4-[1-(3-chlorophenoxy)ethyl]-6-(4-methylpiperazin-1-yl)-1,3,5-triazin-2-amine
Show/Hide
|
C16H21ClN6O
|
1
|
| 1 |
Ki = 118 nM
|
|
|
|
CP0384339
|
5-(4-methylpiperazin-1-yl)-2-nitro-N-phenethylbenzenamine
Show/Hide
|
C19H24N4O2
|
1
|
| 1 |
Ki = 119 nM
|
|
|
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CP0378964
|
4-(4-chlorophenyl)sulfonyl-5-(3,4-dihydro-1H-isoquinolin-2-yl)-2-ethylsulfonyl-1,3-thiazole
Show/Hide
|
C20H19ClN2O4S3
|
2
|
| 1 |
Ki = 119 nM
|
|
|
| 2 |
Ki = 150 nM
|
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|
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CP0548530
|
1-(3,4-difluorophenyl)sulfonyl-3-[(4-methylpiperazin-1-yl)methyl]indole
Show/Hide
|
C20H21F2N3O2S
|
1
|
| 1 |
Ki = 119 nM
|
|
|
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CP0395871
|
N-[3-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]propyl]-5-fluoro-3-methyl-1-benzothiophene-2-sulfonamide
Show/Hide
|
C23H25FN4O2S3
|
1
|
| 1 |
Ki = 120 nM
|
|
|
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CP0395876
|
N-[4-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]butyl]-1,3-benzothiazole-4-sulfonamide
Show/Hide
|
C22H25N5O2S3
|
1
|
| 1 |
Ki = 120 nM
|
|
|
|
CP0443917
|
2-(5-methoxy-1H-indol-3-yl)-N-[[5-(1H-pyrazol-4-yl)furan-2-yl]methyl]ethanamine
Show/Hide
|
C19H20N4O2
|
1
|
| 1 |
Ki = 121 nM
|
|
|
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CP0443749
|
3-bromo-1-(4-fluorophenyl)sulfonyl-4-[(4-methylpiperazin-1-yl)methyl]indole
Show/Hide
|
C20H21BrFN3O2S
|
1
|
| 1 |
Ki = 122 nM
|
|
|
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CP0431324
|
N-[1-[2-(dimethylamino)ethyl]-2-methylindol-5-yl]naphthalene-1-sulfonamide
Show/Hide
|
C23H25N3O2S
|
1
|
| 1 |
Ki = 123.6 nM
|
|
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CP0378289
|
1-[1-(Benzo[b]thiophene-3-sulfonyl)-piperidin-4-yl]-8-methyl-1,4-dihydro-benzo[d][1,3]oxazin-2-one
Show/Hide
|
C22H22N2O4S2
|
1
|
| 1 |
Ki = 124.5 nM
|
|
|
|
CP0392443
|
1-[1-(Benzo[b]thiophene-3-sulfonyl)-piperidin-4-yl]-1,4-dihydro-benzo[d][1,3]oxazin-2-one
Show/Hide
|
C21H20N2O4S2
|
1
|
| 1 |
Ki = 125.8 nM
|
|
|
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CP0553065
|
N-[4-(3-fluorophenyl)sulfonyl-2,2-dimethyl-3H-1,4-benzoxazin-8-yl]-N',N'-dimethylethane-1,2-diamine
Show/Hide
|
C20H26FN3O3S
|
1
|
| 1 |
Ki = 125.89 nM
|
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CP0457580
|
1-[(3-chlorophenyl)methyl]-4-piperazin-1-yl-2-propan-2-ylimidazo[4,5-c]pyridine
Show/Hide
|
C20H24ClN5
|
1
|
| 1 |
Ki = 126 nM
|
|
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CP0438623
|
4-[(2-chlorophenyl)sulfanylmethyl]-6-(4-methylpiperazin-1-yl)-1,3,5-triazin-2-amine
Show/Hide
|
C15H19ClN6S
|
1
|
| 1 |
Ki = 126 nM
|
|
|
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CP0893595
|
N-(4-(4-(3-chlorophenyl)piperazin-1-yl)butyl)naphthalene-1-sulfonamide hydrochloride
Show/Hide
|
C24H29Cl2N3O2S
|
1
|
| 1 |
Ki = 127 nM
|
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CP0414434
|
1,2-dimethoxy-N,N,6-trimethyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-10-amine
Show/Hide
|
C21H26N2O2
|
1
|
| 1 |
Ki = 127 nM
|
|
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CP0382742
|
4-[(2,4-dichlorophenoxy)methyl]-6-(4-methylpiperazin-1-yl)-1,3,5-triazin-2-amine
Show/Hide
|
C15H18Cl2N6O
|
1
|
| 1 |
Ki = 128 nM
|
|
|
|
CP0443487
|
3,5-dimethyl-4-[6-(4-methylpiperazin-1-yl)-1-(2-methylpropylsulfonyl)pyrrolo[2,3-b]pyridin-4-yl]-1,2-oxazole
Show/Hide
|
C21H29N5O3S
|
1
|
| 1 |
Ki = 129 nM
|
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CP0382744
|
4-[(2-chlorophenoxy)methyl]-6-(4-methylpiperazin-1-yl)-1,3,5-triazin-2-amine
Show/Hide
|
C15H19ClN6O
|
1
|
| 1 |
Ki = 129 nM
|
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CP0460929
|
2-(5-methoxy-1-propan-2-ylindol-3-yl)-N,N-dimethylethanamine
Show/Hide
|
C16H24N2O
|
1
|
| 1 |
Ki = 130 nM
|
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|
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CP0447217
|
N-[4-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]butyl]thiophene-2-sulfonamide
Show/Hide
|
C20H24FN3O3S2
|
1
|
| 1 |
Ki = 130 nM
|
|
|
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CP0396074
|
5-[(2S)-2-[2-[4-(1-benzothiophen-4-yl)piperazin-1-yl]ethyl]azetidin-1-yl]sulfonylquinoline
Show/Hide
|
C26H28N4O2S2
|
1
|
| 1 |
Ki = 130 nM
|
|
|
|
CP0488988
|
1-(benzenesulfonyl)-3-(1,2,3,6-tetrahydropyridin-4-yl)pyrrolo[3,2-h]quinoline
Show/Hide
|
C22H19N3O2S
|
1
|
| 1 |
Ki = 131 nM
|
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CP0501158
|
1-[1-(2,5-Dimethoxy-benzenesulfonyl)-piperidin-4-yl]-8-methyl-1,4-dihydro-benzo[d][1,3]oxazin-2-one
Show/Hide
|
C22H26N2O6S
|
1
|
| 1 |
Ki = 131.3 nM
|
|
|
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CP0553071
|
2-(1-(4-methoxybenzyl)-1H-indol-3-yl)-N,N-dimethylethanamine
Show/Hide
|
C20H24N2O
|
1
|
| 1 |
Ki = 132 nM
|
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|
|
CP0376095
|
N-[3-(2-morpholin-4-ylethyl)-1H-indol-5-yl]naphthalene-2-sulfonamide
Show/Hide
|
C24H25N3O3S
|
1
|
| 1 |
Ki = 132 nM
|
|
|
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CP0471830
|
2-[6-[4-(3,4-dichlorophenyl)piperazin-1-yl]hexyl]-1,1-dioxo-1,2-benzothiazol-3-one
Show/Hide
|
C23H27Cl2N3O3S
|
1
|
| 1 |
Ki = 132 nM
|
|
|
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CP0478895
|
N-[[5-(4-fluorophenyl)furan-2-yl]methyl]-2-(4-methoxy-1H-indol-3-yl)ethanamine
Show/Hide
|
C22H21FN2O2
|
1
|
| 1 |
Ki = 132 nM
|
|
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CP0233038
|
1-(cyclopropylmethoxy)-2-methoxy-6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-10-amine
Show/Hide
|
C22H26N2O2
|
1
|
| 1 |
Ki = 132 nM
|
|
|
|
CP0510211
|
N-[2-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]ethyl]naphthalene-2-sulfonamide
Show/Hide
|
C24H24FN3O3S
|
1
|
| 1 |
Ki = 133 nM
|
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CP0436409
|
3-[(4-benzylpiperazin-1-yl)methyl]-1-(2-bromophenyl)sulfonylindole
Show/Hide
|
C26H26BrN3O2S
|
1
|
| 1 |
Ki = 133 nM
|
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|
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CP0524251
|
2-(1-(butylsulfonyl)-1H-indol-3-yl)-N,N-dimethylethanamine
Show/Hide
|
C16H24N2O2S
|
1
|
| 1 |
Ki = 135 nM
|
|
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CP0373612
|
5-(Dimethylamino)-N-(5-(dimethylamino)naphthalen-1-ylsulfonyl)-N-(4-methoxy-3-(piperazin-1-yl)phenyl)naphthalene-1-sulfonamide
Show/Hide
|
C35H39N5O5S2
|
1
|
| 1 |
Ki = 135 nM
|
|
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CP0490397
|
(9-Benzyl-2,3,4,9-tetrahydro-1H-carbazol-4-ylmethyl)-dimethyl-amine
Show/Hide
|
C22H26N2
|
1
|
| 1 |
Ki = 136 nM
|
|
|
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CP0562769
|
2-N-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butyl]-1,3,5-triazine-2,4,6-triamine
Show/Hide
|
C17H24Cl2N8
|
1
|
| 1 |
Ki = 136 nM
|
|
|
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CP0386967
|
1-(3-bromophenyl)sulfonyl-3-(1,2,3,6-tetrahydropyridin-4-yl)pyrrolo[2,3-f]quinoline
Show/Hide
|
C22H18BrN3O2S
|
1
|
| 1 |
Ki = 137 nM
|
|
|
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CP0396617
|
6-fluoro-3-[1-[2-[(2S)-1-isoquinolin-4-ylsulfonylpyrrolidin-2-yl]ethyl]piperidin-4-yl]-1,2-benzoxazole
Show/Hide
|
C27H29FN4O3S
|
1
|
| 1 |
Ki = 137 nM
|
|
|
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CP0548570
|
N-[[4-[6-[4-[1-[(3-chlorophenyl)methyl]indol-4-yl]piperazin-1-yl]hexoxy]phenyl]methyl]-N-methylprop-2-yn-1-amine
Show/Hide
|
C36H43ClN4O
|
1
|
| 1 |
Ki = 137 nM
|
|
|
|
CP0776667
|
N-{4-[4-(3-Chlorophenyl)-piperazin-1-yl]-butyl}-3-quinolinesulfonamide hydrochloride
Show/Hide
|
C23H28Cl2N4O2S
|
1
|
| 1 |
Ki = 139 nM
|
|
|
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CP0389649
|
3-[(3,4-difluorophenyl)methyl]-2-ethyl-7-piperazin-1-ylimidazo[4,5-b]pyridine
Show/Hide
|
C19H21F2N5
|
1
|
| 1 |
Ki = 139 nM
|
|
|
|
CP0395874
|
N-[4-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]butyl]-3-methylbenzenesulfonamide
Show/Hide
|
C23H28FN3O3S
|
1
|
| 1 |
Ki = 140 nM
|
|
|
|
CP0481185
|
N-[4-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]butyl]imidazo[1,2-a]pyridine-3-sulfonamide
Show/Hide
|
C22H26N6O2S2
|
1
|
| 1 |
Ki = 140 nM
|
|
|
|
CP0506649
|
N-[3-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]propyl]thiophene-2-sulfonamide
Show/Hide
|
C18H22N4O2S3
|
1
|
| 1 |
Ki = 140 nM
|
|
|
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CP0398680
|
7-[4-[4-[1-(benzenesulfonyl)indol-3-yl]piperidin-1-yl]butoxy]-3,4-dihydro-1H-quinolin-2-one
Show/Hide
|
C32H35N3O4S
|
1
|
| 1 |
Ki = 140 nM
|
|
|
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CP0507403
|
N-[[4-[5-[4-[1-[(3-chlorophenyl)methyl]indol-4-yl]piperazin-1-yl]pentoxy]phenyl]methyl]-N-methylprop-2-yn-1-amine
Show/Hide
|
C35H41ClN4O
|
1
|
| 1 |
Ki = 140 nM
|
|
|
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CP0574437
|
4-amino-N-[2-[4-[3-(4-amino-5-chloro-2-methoxyphenyl)-3-oxopropyl]piperidin-1-yl]ethyl]-3,5-dibromobenzenesulfonamide
Show/Hide
|
C23H29Br2ClN4O4S
|
1
|
| 1 |
Ki = 140 nM
|
|
|
|
CP0475997
|
N-[1-[2-(diethylamino)ethyl]indol-5-yl]naphthalene-2-sulfonamide
Show/Hide
|
C24H27N3O2S
|
1
|
| 1 |
Ki = 140.5 nM
|
|
|
|
CP0389651
|
2-(2,2-dimethylpropyl)-3-[(3-methylphenyl)methyl]-7-piperazin-1-ylimidazo[4,5-b]pyridine
Show/Hide
|
C23H31N5
|
1
|
| 1 |
Ki = 142 nM
|
|
|
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CP0500282
|
2-(5,5-dioxoindolo[1,2-b][1,2]benzothiazol-11-yl)-N,N-dimethylethanamine
Show/Hide
|
C18H18N2O2S
|
1
|
| 1 |
Ki = 143 nM
|
|
|
|
CP0513729
|
5,7-dichloro-3-(4-methoxyphenyl)-3-methylquinoline-2,4(1H,3H)-dione
Show/Hide
|
C17H13Cl2NO3
|
1
|
| 1 |
Ki = 147 nM
|
|
|
|
CP0854353
|
N-(4-(4-(3-chlorophenyl)piperazin-1-yl)butyl)naphthalene-2-sulfonamide hydrochloride
Show/Hide
|
C24H29Cl2N3O2S
|
1
|
| 1 |
Ki = 147 nM
|
|
|
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CP0381348
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3-chloro-N-[[1-[2-(2-methylsulfanylphenoxy)ethyl]piperidin-4-yl]methyl]benzenesulfonamide
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C21H27ClN2O3S2
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1
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| 1 |
Ki = 147 nM
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CP0517220
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N-[2-[4-[3-(4-amino-5-chloro-2-methoxyphenyl)-3-oxopropyl]piperidin-1-yl]ethyl]-3-bromo-4-methoxybenzenesulfonamide
Show/Hide
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C24H31BrClN3O5S
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1
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| 1 |
Ki = 147 nM
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CP0507070
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N-[(4-cyanophenyl)methyl]-3-[2-[4-(2-phenylphenyl)piperazin-1-yl]ethoxy]propanamide
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C29H32N4O2
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1
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| 1 |
Ki = 148 nM
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CP0438624
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4-[(3-chlorophenoxy)methyl]-6-(4-methylpiperazin-1-yl)-1,3,5-triazin-2-amine
Show/Hide
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C15H19ClN6O
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1
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| 1 |
Ki = 148 nM
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CP0380664
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7-[4-[2-(1-benzylindol-3-yl)ethylamino]butoxy]-3,4-dihydro-1H-quinolin-2-one
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C30H33N3O2
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1
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| 1 |
Ki = 150 nM
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CP0412623
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7-[4-[4-(1-benzylindol-3-yl)piperidin-1-yl]butoxy]-3,4-dihydro-1H-quinolin-2-one
Show/Hide
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C33H37N3O2
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1
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| 1 |
Ki = 150 nM
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CP0393700
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3-[(4-methylpiperazin-1-yl)methyl]-1-[4-(trifluoromethoxy)phenyl]sulfonylindole
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C21H22F3N3O3S
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1
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| 1 |
Ki = 150 nM
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CP0375962
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1-[1-(Quinoline-8-sulfonyl)-piperidin-4-yl]-1,4-dihydro-benzo[d][1,3]oxazin-2-one
Show/Hide
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C22H21N3O4S
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1
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| 1 |
Ki = 151.9 nM
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CP0562342
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2-(1H-indol-3-yl)-N-[(5-phenylthiophen-2-yl)methyl]ethanamine
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C21H20N2S
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1
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| 1 |
Ki = 152 nM
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CP0508845
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2-(benzenesulfonyl)-N-methyl-5-phenylaniline
Show/Hide
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C19H17NO2S
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1
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| 1 |
Ki = 153 nM
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CP0533188
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3-(benzenesulfonyl)-7-(methoxymethyl)-5-methyl-2-methylsulfanylpyrazolo[1,5-a]pyrimidine
Show/Hide
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C16H17N3O3S2
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1
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| 1 |
Ki = 154.88 nM
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CP0896648
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N-{4-[4-(3-Chlorophenyl)-piperazin-1-yl]-butyl}-6-chloro-3-quinolinesulfonamide hydrochloride
Show/Hide
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C23H27Cl3N4O2S
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1
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| 1 |
Ki = 155 nM
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CP0535838
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3-(4-aminophenyl)-5,7-dichloro-3-methylquinoline-2,4(1H,3H)-dione
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C16H12Cl2N2O2
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1
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| 1 |
Ki = 156 nM
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CP0486997
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2,5-difluoro-N-[1-[2-(5,6,7,8-tetrahydronaphthalen-1-yloxy)ethyl]pyrrolidin-3-yl]benzenesulfonamide
Show/Hide
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C22H26F2N2O3S
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1
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| 1 |
Ki = 156 nM
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CP0429636
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2-[6-(4-naphthalen-1-ylpiperazin-1-yl)hexyl]-1,1-dioxo-1,2-benzothiazol-3-one
Show/Hide
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C27H31N3O3S
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1
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| 1 |
Ki = 157 nM
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CP0476616
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5-[1-(benzenesulfonyl)-5-methoxyindol-3-yl]-1-(2,2-difluoroethyl)-4-methylimidazol-2-amine
Show/Hide
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C21H20F2N4O3S
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1
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| 1 |
Ki = 157 nM
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CP0548791
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4-[(3-methoxyphenyl)methyl]-6-(4-methylpiperazin-1-yl)-1,3,5-triazin-2-amine
Show/Hide
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C16H22N6O
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1
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| 1 |
Ki = 158 nM
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CP0526780
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3-[6-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]hexyl]-2lambda6-thia-3-azatricyclo[6.3.1.04,12]dodeca-1(11),4,6,8(12),9-pentaene 2,2-dioxide
Show/Hide
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C27H30N4O2S2
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1
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| 1 |
Ki = 158 nM
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CP0483664
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(2S)-2-[[4-[3-[4-[1-[(3-chlorophenyl)methyl]indol-4-yl]piperazin-1-yl]propoxy]phenyl]methylamino]propanamide
Show/Hide
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C32H38ClN5O2
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1
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| 1 |
Ki = 158 nM
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CP0472552
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N-[2-[4-[3-(4-amino-5-chloro-2-methoxyphenyl)-3-oxopropyl]piperidin-1-yl]ethyl]-3-chloro-4-methoxybenzenesulfonamide
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C24H31Cl2N3O5S
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1
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| 1 |
Ki = 158 nM
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CP0380583
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3-(1H-indol-3-yl)-1-[4-[4-(5-methoxy-1H-indol-3-yl)piperidin-1-yl]butyl]pyrrolidine-2,5-dione
Show/Hide
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C30H34N4O3
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1
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| 1 |
Ki = 159 nM
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CP0348615
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2-[6-(4-Benzo[d]isothiazol-3-yl-piperazin-1-yl)-hexyl]-isoindole-1,3-dione
Show/Hide
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C25H28N4O2S
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1
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| 1 |
Ki = 160 nM
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CP0389652
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2-(4-fluorophenyl)-3-[(3-fluorophenyl)methyl]-7-piperazin-1-ylimidazo[4,5-b]pyridine
Show/Hide
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C23H21F2N5
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1
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| 1 |
Ki = 162 nM
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CP0451726
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(2S)-2-[[4-[4-[4-[1-[(3-chlorophenyl)methyl]indol-4-yl]piperazin-1-yl]butoxy]phenyl]methylamino]propanamide
Show/Hide
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C33H40ClN5O2
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1
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| 1 |
Ki = 162 nM
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CP0343719
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2-nitro-5-(piperazin-1-yl)-N-(2-(o-tolyloxy)ethyl)benzenamine
Show/Hide
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C19H24N4O3
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1
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| 1 |
Ki = 163 nM
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CP0375938
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N-[3-[3-(diethylamino)propyl]-1H-indol-5-yl]naphthalene-2-sulfonamide
Show/Hide
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C25H29N3O2S
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1
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| 1 |
Ki = 163 nM
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CP0375942
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N-[3-(2-morpholin-4-ylethyl)-1H-indol-5-yl]naphthalene-1-sulfonamide
Show/Hide
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C24H25N3O3S
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1
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| 1 |
Ki = 163.5 nM
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CP0485360
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N-[2-amino-4-(4-methylpiperazin-1-yl)phenyl]-N-benzylacetamide
Show/Hide
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C20H26N4O
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1
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| 1 |
Ki = 164 nM
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CP0479117
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5-Chloro-N-[3-(4-{[5-(dimethylamino)-1-naphthyl]sulfonyl}-piperazin-1-yl)-4-methoxyphenyl]-3-methyl-1-benzothiophene-2-sulfonamide
Show/Hide
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C32H33ClN4O5S3
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1
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| 1 |
Ki = 165 nM
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CP0443750
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3-chloro-4-[(4-methylpiperazin-1-yl)methyl]-1-naphthalen-1-ylsulfonylindole
Show/Hide
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C24H24ClN3O2S
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1
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| 1 |
Ki = 165 nM
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CP0457617
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2-(2,2-dimethylpropyl)-3-[(3-methoxyphenyl)methyl]-7-piperazin-1-ylimidazo[4,5-b]pyridine
Show/Hide
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C23H31N5O
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1
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| 1 |
Ki = 165 nM
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CP0518982
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3-[(3-chlorophenyl)methyl]-7-piperazin-1-yl-2-thiophen-2-ylimidazo[4,5-b]pyridine
Show/Hide
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C21H20ClN5S
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1
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| 1 |
Ki = 165 nM
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CP0432872
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8-Methyl-1-[1-(quinoline-8-sulfonyl)-piperidin-4-yl]-1,4-dihydro-benzo[d][1,3]oxazin-2-one
Show/Hide
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C23H23N3O4S
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1
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| 1 |
Ki = 165.9 nM
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CP0228753
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(6-Methoxy-2,3,4,9-tetrahydro-1H-carbazol-4-ylmethyl)-dimethyl-amine
Show/Hide
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C16H22N2O
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1
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| 1 |
Ki = 168 nM
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CP0152345
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2-[4-[(3Z)-3-(2-chloranylthioxanthen-9-ylidene)propyl]piperazin-1-yl]ethanol;hydrochloride
Show/Hide
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C22H25ClN2OS
|
1
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| 1 |
Ki = 169 nM
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CP0390939
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6-fluoro-3-[1-[2-[(2S)-1-quinolin-5-ylsulfonylpyrrolidin-2-yl]ethyl]piperidin-4-yl]-1,2-benzoxazole
Show/Hide
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C27H29FN4O3S
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1
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| 1 |
Ki = 169 nM
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CP0533144
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N-[(4-fluorophenyl)methyl]-5-(4-methylpiperazin-1-yl)-2-nitroaniline
Show/Hide
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C18H21FN4O2
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1
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| 1 |
Ki = 172 nM
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CP0373613
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5-(Dimethylamino)-N-(3-{4-[4-({[5-(dimethylamino)-1-naphthyl]-sulfonyl}amino)butyl]piperazin-1-yl}-4-methoxyphenyl)naphthalene-1-sulfonamide
Show/Hide
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C39H48N6O5S2
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1
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| 1 |
Ki = 175 nM
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CP0390936
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5-[(2S)-2-[2-[4-(1-benzothiophen-4-yl)piperazin-1-yl]ethyl]azepan-1-yl]sulfonylquinoline
Show/Hide
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C29H34N4O2S2
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1
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| 1 |
Ki = 176 nM
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CP0486994
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3-chloro-N-[[1-[2-(2-propan-2-ylphenoxy)ethyl]piperidin-4-yl]methyl]benzenesulfonamide
Show/Hide
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C23H31ClN2O3S
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1
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| 1 |
Ki = 177 nM
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CP0513853
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3-[(2-chlorophenyl)methyl]-2-ethyl-7-piperazin-1-ylimidazo[4,5-b]pyridine
Show/Hide
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C19H22ClN5
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1
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| 1 |
Ki = 177 nM
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CP0069200
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1H-indole-3-ethanamine
Show/Hide
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C10H12N2
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1
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| 1 |
Ki = 180 nM
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CP0417065
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3-[6-(4-pyridin-2-ylpiperazin-1-yl)hexyl]-2lambda6-thia-3-azatricyclo[6.3.1.04,12]dodeca-1(11),4,6,8(12),9-pentaene 2,2-dioxide
Show/Hide
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C25H30N4O2S
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1
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| 1 |
Ki = 182 nM
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CP0441758
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2-[1-(2,5-dimethoxyphenyl)sulfonyl-7-methoxyindol-3-yl]-N,N-dimethylethanamine
Show/Hide
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C21H26N2O5S
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1
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| 1 |
Ki = 183 nM
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CP0116953
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1,1'-sulfonylbis(4-aminobenzene)
Show/Hide
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C12H12N2O2S
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1
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| 1 |
Ki = 183 nM
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CP0076852
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2-(5-methoxy-2-propyl-1H-indol-3-yl)-N,N-dimethylethanamine
Show/Hide
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C16H24N2O
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1
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| 1 |
Ki = 185 nM
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CP0513237
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3-chloro-N-[1-[2-(2-methylsulfanylphenoxy)ethyl]pyrrolidin-3-yl]benzenesulfonamide
Show/Hide
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C19H23ClN2O3S2
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1
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| 1 |
Ki = 185 nM
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CP0542457
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N-[[5-(3-chlorophenyl)furan-2-yl]methyl]-2-(1H-indol-3-yl)ethanamine
Show/Hide
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C21H19ClN2O
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1
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| 1 |
Ki = 185 nM
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CP0473056
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3-[6-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]hexyl]-1,3-benzoxazol-2-one
Show/Hide
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C24H28N4O2S
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1
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| 1 |
Ki = 189 nM
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CP0484413
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3-[6-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]hexyl]-1H-benzimidazol-2-one
Show/Hide
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C24H29N5OS
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1
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| 1 |
Ki = 189 nM
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CP0408251
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4-[(2S)-2-[2-[4-(1-benzothiophen-4-yl)piperazin-1-yl]ethyl]azepan-1-yl]sulfonylisoquinoline
Show/Hide
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C29H34N4O2S2
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1
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| 1 |
Ki = 190 nM
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CP0534784
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4-[(2-methoxyphenyl)methyl]-6-(4-methylpiperazin-1-yl)-1,3,5-triazin-2-amine
Show/Hide
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C16H22N6O
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1
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| 1 |
Ki = 193 nM
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CP0402605
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5-(Dimethylamino)-N-(8-{4-[5-({[5-(dimethylamino)-1-naphthyl]-sulfonyl}amino)-2-methoxyphenyl]piperazin-1-yl}octyl)naphthalene-1-sulfonamide
Show/Hide
|
C43H56N6O5S2
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1
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| 1 |
Ki = 194 nM
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CP0566562
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1-(2-bromophenyl)sulfonyl-3-[(4-methylpiperazin-1-yl)methyl]-5-methylsulfanylindole
Show/Hide
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C21H24BrN3O2S2
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1
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| 1 |
Ki = 194 nM
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CP0442266
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2-Naphthalen-1-yl-ethanesulfonic acid [1-(2-pyrrolidin-1-yl-ethyl)-1H-indol-6-yl]-amide
Show/Hide
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C26H29N3O2S
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1
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| 1 |
Ki = 194.8 nM
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CP0490622
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N-[[4-[4-[4-[1-[(3-chlorophenyl)methyl]indol-4-yl]piperazin-1-yl]butoxy]phenyl]methyl]-N-methylprop-2-yn-1-amine
Show/Hide
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C34H39ClN4O
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1
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| 1 |
Ki = 195 nM
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CP0501993
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5,7-dibromo-3-methyl-3-phenylquinoline-2,4(1H,3H)-dione
Show/Hide
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C16H11Br2NO2
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1
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| 1 |
Ki = 196.9 nM
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CP0548405
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2-[5-[4-(2,3-dichlorophenyl)piperazin-1-yl]pentyl]-1,1-dioxo-1,2-benzothiazol-3-one
Show/Hide
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C22H25Cl2N3O3S
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1
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| 1 |
Ki = 197 nM
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CP0414432
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N-(2-methoxy-6-methyl-1-prop-2-enoxy-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-10-yl)butanamide
Show/Hide
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C25H30N2O3
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1
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| 1 |
Ki = 198 nM
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CP0381352
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3,4-difluoro-N-[1-[2-(2-phenylphenoxy)ethyl]piperidin-4-yl]benzenesulfonamide
Show/Hide
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C25H26F2N2O3S
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1
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| 1 |
Ki = 199 nM
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CP0562345
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4-[5-[[2-(5-methoxy-1H-indol-3-yl)ethyl-methylamino]methyl]furan-2-yl]phenol
Show/Hide
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C23H24N2O3
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1
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| 1 |
Ki = 199 nM
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CP0542173
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N-[3-[(8-piperazin-1-yl-2,3-dihydro-1,4-benzoxazin-4-yl)sulfonyl]phenyl]methanesulfonamide
Show/Hide
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C19H24N4O5S2
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1
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| 1 |
Ki = 199.53 nM
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CP0521897
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2-(5-methoxy-1-propylindol-3-yl)-N,N-dimethylethanamine
Show/Hide
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C16H24N2O
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1
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| 1 |
Ki = 200 nM
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CP0445257
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5-chloro-N-[(3R)-1-[2-(2-propan-2-ylphenoxy)ethyl]pyrrolidin-3-yl]thiophene-2-sulfonamide
Show/Hide
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C19H25ClN2O3S2
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1
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| 1 |
Ki = 200 nM
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CP0566563
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1-(2-bromophenyl)sulfonyl-3-[(4-methylpiperazin-1-yl)methyl]-5-nitroindole
Show/Hide
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C20H21BrN4O4S
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1
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| 1 |
Ki = 200 nM
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CP0487392
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2-(1H-indol-3-yl)-N-[(5-naphthalen-1-ylfuran-2-yl)methyl]ethanamine
Show/Hide
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C25H22N2O
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1
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| 1 |
Ki = 201 nM
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CP0445258
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5-chloro-N-[(3R)-1-[2-(2-phenylphenoxy)ethyl]pyrrolidin-3-yl]thiophene-2-sulfonamide
Show/Hide
|
C22H23ClN2O3S2
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1
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| 1 |
Ki = 202 nM
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CP0398058
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7-[4-[4-(3-chlorophenyl)piperazin-1-yl]butyl]-1,3-dimethyl-8-morpholin-4-ylpurine-2,6-dione
Show/Hide
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C25H34ClN7O3
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1
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| 1 |
Ki = 207 nM
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CP0402155
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4-[(3-methylphenoxy)methyl]-6-(4-methylpiperazin-1-yl)-1,3,5-triazin-2-amine
Show/Hide
|
C16H22N6O
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1
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| 1 |
Ki = 207 nM
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CP0464104
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2-(1-(cyclohexylsulfonyl)-1H-indol-3-yl)-N,N-dimethylethanamine
Show/Hide
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C18H26N2O2S
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1
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| 1 |
Ki = 210 nM
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CP0440062
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N-[2-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]ethyl]-3-methylbenzenesulfonamide
Show/Hide
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C21H24FN3O3S
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1
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| 1 |
Ki = 210 nM
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CP0520069
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N-[[5-(3,5-dichlorophenyl)furan-2-yl]methyl]-2-(5-methoxy-1H-indol-3-yl)ethanamine
Show/Hide
|
C22H20Cl2N2O2
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1
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| 1 |
Ki = 210 nM
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CP0072206
|
NORTRIPTYLINE
Show/Hide
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C19H21N
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1
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| 1 |
Ki = 214 nM
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CP0475765
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5-Chloro-N-[8-({[5-(dimethylamino)-1-naphthyl]sulfonyl}amino)-octyl]-N-(4-methoxy-3-piperazin-1-ylphenyl)-3-methyl-1-benzothiophene-2-sulfonamide
Show/Hide
|
C40H50ClN5O5S3
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1
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| 1 |
Ki = 215 nM
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CP0434001
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N-[(1Z)-1-benzylidene-3-[2-(dimethylamino)ethyl]-2-methylinden-5-yl]naphthalene-2-sulfonamide
Show/Hide
|
C31H30N2O2S
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1
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| 1 |
Ki = 216 nM
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CP0414433
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N-(2-methoxy-6-methyl-1-prop-2-ynoxy-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-10-yl)methanesulfonamide
Show/Hide
|
C22H24N2O4S
|
1
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| 1 |
Ki = 218 nM
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CP0530225
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7-[3-(1-butyl-3,6-dihydro-2H-pyridin-4-yl)-5-methoxyindol-1-yl]sulfonylquinoline
Show/Hide
|
C27H29N3O3S
|
1
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| 1 |
Ki = 219 nM
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CP0231658
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4-amino-N-[2-[4-[3-(4-amino-5-chloro-2-methoxyphenyl)-3-oxopropyl]piperidin-1-yl]ethyl]-3-bromobenzenesulfonamide
Show/Hide
|
C23H30BrClN4O4S
|
1
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| 1 |
Ki = 219 nM
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CP0464770
|
N,N-dimethyl-2-(1-pentylsulfonylindol-3-yl)ethanamine
Show/Hide
|
C17H26N2O2S
|
1
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| 1 |
Ki = 220 nM
|
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CP0510654
|
2-ethyl-5-methoxy-3-[[(2S)-1-methylpyrrolidin-2-yl]methyl]-1H-indole
Show/Hide
|
C17H24N2O
|
1
|
| 1 |
Ki = 220 nM
|
|
|
|
CP0418453
|
N-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butyl]isoquinoline-4-sulfonamide
Show/Hide
|
C23H26Cl2N4O2S
|
1
|
| 1 |
Ki = 220 nM
|
|
|
|
CP0551437
|
N-[[5-(1,3-benzodioxol-5-yl)furan-2-yl]methyl]-2-(1H-indol-3-yl)ethanamine
Show/Hide
|
C22H20N2O3
|
1
|
| 1 |
Ki = 220 nM
|
|
|
|
CP0472430
|
4-[(2R)-2-[2-[4-(1-benzothiophen-4-yl)piperazin-1-yl]ethyl]piperidin-1-yl]sulfonylisoquinoline
Show/Hide
|
C28H32N4O2S2
|
1
|
| 1 |
Ki = 221 nM
|
|
|
|
CP0525896
|
N-[6-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]hexyl]benzamide
Show/Hide
|
C24H30N4OS
|
1
|
| 1 |
Ki = 221 nM
|
|
|
|
CP0500053
|
3-chloro-1-(4-methylphenyl)sulfonyl-4-[(4-methylpiperazin-1-yl)methyl]indole
Show/Hide
|
C21H24ClN3O2S
|
1
|
| 1 |
Ki = 222 nM
|
|
|
|
CP0554895
|
4-[5-[4-[1-[(3-chlorophenyl)methyl]indol-4-yl]piperazin-1-yl]pentoxy]-N-prop-2-ynyl-2,3-dihydro-1H-inden-1-amine
Show/Hide
|
C36H41ClN4O
|
1
|
| 1 |
Ki = 223 nM
|
|
|
|
CP0376238
|
2-[5-(6-Chloro-imidazo[2,1-b]thiazole-5-sulfonylamino)-1H-indol-3-yl]-N,N-diethyl-2-oxo-acetamide
Show/Hide
|
C19H18ClN5O4S2
|
1
|
| 1 |
Ki = 224.4 nM
|
|
|
|
CP0426092
|
5-chloro-N-[1-[2-(2,5-dichlorophenoxy)ethyl]pyrrolidin-3-yl]thiophene-2-sulfonamide
Show/Hide
|
C16H17Cl3N2O3S2
|
1
|
| 1 |
Ki = 225 nM
|
|
|
|
CP0483352
|
3-[6-[4-(3,4-dichlorophenyl)piperazin-1-yl]hexyl]-2lambda6-thia-3-azatricyclo[6.3.1.04,12]dodeca-1(11),4,6,8(12),9-pentaene 2,2-dioxide;hydrochloride
Show/Hide
|
C26H30Cl3N3O2S
|
1
|
| 1 |
Ki = 225 nM
|
|
|
|
CP0505676
|
N-[3-(3-aminopropyl)phenyl]benzenesulfonamide
Show/Hide
|
C15H18N2O2S
|
1
|
| 1 |
Ki = 230 nM
|
|
|
|
CP0488996
|
5-[6-(4-methylpiperazin-1-yl)-1-(2-methylpropylsulfonyl)pyrrolo[2,3-b]pyridin-4-yl]-1H-pyridin-2-one
Show/Hide
|
C21H27N5O3S
|
1
|
| 1 |
Ki = 231 nM
|
|
|
|
CP0466078
|
(2S)-2-[[4-[5-[4-[1-[(3-chlorophenyl)methyl]indol-4-yl]piperazin-1-yl]pentoxy]phenyl]methylamino]propanamide
Show/Hide
|
C34H42ClN5O2
|
1
|
| 1 |
Ki = 232 nM
|
|
|
|
CP0850796
|
5-N-(1-{2-[(Propan-2-yl)phenoxy]ethyl}piperidin-4-yl)-quinolinesulfonamide
Show/Hide
|
C25H31N3O3S
|
1
|
| 1 |
Ki = 233 nM
|
|
|
|
CP0431614
|
4-[(4-methylphenoxy)methyl]-6-(4-methylpiperazin-1-yl)-1,3,5-triazin-2-amine
Show/Hide
|
C16H22N6O
|
1
|
| 1 |
Ki = 235 nM
|
|
|
|
CP0483144
|
3-[6-[4-(2,3-dichlorophenyl)piperazin-1-yl]hexyl]-2lambda6-thia-3-azatricyclo[6.3.1.04,12]dodeca-1(11),4,6,8(12),9-pentaene 2,2-dioxide;hydrochloride
Show/Hide
|
C26H30Cl3N3O2S
|
1
|
| 1 |
Ki = 237 nM
|
|
|
|
CP0574462
|
1-(4-fluorophenyl)sulfonyl-6-methoxy-3-[(4-methylpiperazin-1-yl)methyl]indole
Show/Hide
|
C21H24FN3O3S
|
1
|
| 1 |
Ki = 239 nM
|
|
|
|
CP0447417
|
2-(1-ethyl-5-methoxyindol-3-yl)-N,N-dimethylethanamine
Show/Hide
|
C15H22N2O
|
1
|
| 1 |
Ki = 240 nM
|
|
|
|
CP0486999
|
4-fluoro-N-[1-[2-(2-propan-2-ylphenoxy)ethyl]piperidin-4-yl]benzenesulfonamide
Show/Hide
|
C22H29FN2O3S
|
1
|
| 1 |
Ki = 240 nM
|
|
|
|
CP0683568
|
2-fluoro-N-(1-(2-(2-isopropylphenoxy)ethyl)piperidin-4-yl)benzenesulfonamide
Show/Hide
|
C22H29FN2O3S
|
1
|
| 1 |
Ki = 240 nM
|
|
|
|
CP0382740
|
4-(4-methylpiperazin-1-yl)-6-(phenylselanylmethyl)-1,3,5-triazin-2-amine
Show/Hide
|
C15H20N6Se
|
1
|
| 1 |
Ki = 242 nM
|
|
|
|
CP0485358
|
N-[2-(4-methoxyphenoxy)ethyl]-5-(4-methylpiperazin-1-yl)-2-nitroaniline
Show/Hide
|
C20H26N4O4
|
1
|
| 1 |
Ki = 245 nM
|
|
|
|
CP0453916
|
3-chloro-N-[1-[2-(2-propan-2-ylphenoxy)ethyl]pyrrolidin-3-yl]benzenesulfonamide
Show/Hide
|
C21H27ClN2O3S
|
1
|
| 1 |
Ki = 245 nM
|
|
|
|
CP0421835
|
5-bromo-3-(3-methylimidazol-4-yl)-1H-indole
Show/Hide
|
C12H10BrN3
|
1
|
| 1 |
Ki = 245 nM
|
|
|
|
CP0384574
|
2-[6-[4-(2-ethoxyphenyl)piperazin-1-yl]hexyl]benzo[de]isoquinoline-1,3-dione
Show/Hide
|
C30H35N3O3
|
1
|
| 1 |
Ki = 246 nM
|
|
|
|
CP0486925
|
8-Methyl-1-[1-(naphthalene-1-sulfonyl)-piperidin-4-yl]-1,4-dihydro-benzo[d][1,3]oxazin-2-one
Show/Hide
|
C24H24N2O4S
|
1
|
| 1 |
Ki = 246.2 nM
|
|
|
|
CP0519024
|
2-(4-methoxy-1H-indol-3-yl)-N-[[5-(3-methoxyphenyl)furan-2-yl]methyl]ethanamine
Show/Hide
|
C23H24N2O3
|
1
|
| 1 |
Ki = 247 nM
|
|
|
|
CP0544507
|
7-[5-methoxy-3-(1-propyl-3,6-dihydro-2H-pyridin-4-yl)indol-1-yl]sulfonylquinoline
Show/Hide
|
C26H27N3O3S
|
1
|
| 1 |
Ki = 247 nM
|
|
|
|
CP0445255
|
4-fluoro-N-[1-(2-phenoxyethyl)pyrrolidin-3-yl]benzenesulfonamide
Show/Hide
|
C18H21FN2O3S
|
1
|
| 1 |
Ki = 248 nM
|
|
|
|
CP0391901
|
3-(4-chlorophenyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine
Show/Hide
|
C13H14ClN3
|
1
|
| 1 |
Ki = 248 nM
|
|
|
|
CP0533167
|
1-(3-(3,5-dimethyl-1H-pyrazol-1-yl)-4-nitrophenyl)-4-methylpiperazine
Show/Hide
|
C16H21N5O2
|
1
|
| 1 |
Ki = 250 nM
|
|
|
|
CP0443103
|
N-[2-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]ethyl]naphthalene-1-sulfonamide
Show/Hide
|
C24H24FN3O3S
|
1
|
| 1 |
Ki = 250 nM
|
|
|
|
CP0435391
|
2-[1-(benzenesulfonyl)-5-methoxyindol-3-yl]-3-methyl-1H-imidazo[1,2-a]pyrimidin-4-ium;bromide
Show/Hide
|
C22H19BrN4O3S
|
1
|
| 1 |
Ki = 250 nM
|
|
|
|
CP0491001
|
2-[6-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]hexyl]-[1,2,4]triazolo[4,3-a]pyridin-3-one
Show/Hide
|
C23H28N6OS
|
1
|
| 1 |
Ki = 252 nM
|
|
|
|
CP0427415
|
1-[(3-chlorophenyl)methyl]-2-methyl-4-piperazin-1-ylimidazo[4,5-c]pyridine
Show/Hide
|
C18H20ClN5
|
1
|
| 1 |
Ki = 254 nM
|
|
|
|
CP0511650
|
5,7-dichloro-3-methyl-3-(4-(methylamino)phenyl)quinoline-2,4(1H,3H)-dione
Show/Hide
|
C17H14Cl2N2O2
|
1
|
| 1 |
Ki = 257 nM
|
|
|
|
CP0418456
|
N-[3-[4-(2,3-dichlorophenyl)piperazin-1-yl]propyl]quinoline-7-sulfonamide
Show/Hide
|
C22H24Cl2N4O2S
|
1
|
| 1 |
Ki = 257 nM
|
|
|
|
CP0486996
|
N-[1-[2-(2-propan-2-ylphenoxy)ethyl]pyrrolidin-3-yl]thiophene-2-sulfonamide
Show/Hide
|
C19H26N2O3S2
|
1
|
| 1 |
Ki = 258 nM
|
|
|
|
CP0490640
|
4-[6-[4-[1-[(3-chlorophenyl)methyl]indol-4-yl]piperazin-1-yl]hexoxy]-N-prop-2-ynyl-2,3-dihydro-1H-inden-1-amine
Show/Hide
|
C37H43ClN4O
|
1
|
| 1 |
Ki = 259 nM
|
|
|
|
CP0424448
|
N-[4-[1-(benzenesulfonyl)indol-3-yl]-5-ethyl-1H-imidazol-2-yl]acetamide
Show/Hide
|
C21H20N4O3S
|
1
|
| 1 |
Ki = 263 nM
|
|
|
|
CP0519020
|
2-(1H-indol-3-yl)-N-[(5-phenyl-1H-pyrrol-2-yl)methyl]ethanamine
Show/Hide
|
C21H21N3
|
1
|
| 1 |
Ki = 264 nM
|
|
|
|
CP0500037
|
5-Chloro-N-(3-{4-[6-({[5-(dimethylamino)-1-naphthyl]sulfonyl}-amino)hexyl]piperazin-1-yl}-4-methoxyphenyl)-3-methyl-1-benzothiophene-2-sulfonamide
Show/Hide
|
C38H46ClN5O5S3
|
1
|
| 1 |
Ki = 266 nM
|
|
|
|
CP0519023
|
N-[[5-(3,5-dichlorophenyl)furan-2-yl]methyl]-2-(1H-indol-3-yl)ethanamine
Show/Hide
|
C21H18Cl2N2O
|
1
|
| 1 |
Ki = 266 nM
|
|
|
|
CP0508203
|
N-[1-[2-(2-phenylphenoxy)ethyl]pyrrolidin-3-yl]thiophene-2-sulfonamide
Show/Hide
|
C22H24N2O3S2
|
1
|
| 1 |
Ki = 267 nM
|
|
|
|
CP0386966
|
1-[(3-chlorophenyl)methyl]-3-(1,2,3,6-tetrahydropyridin-4-yl)pyrrolo[3,2-h]quinoline
Show/Hide
|
C23H20ClN3
|
1
|
| 1 |
Ki = 269 nM
|
|
|
|
CP0499321
|
dimethyl(2-{2-phenyl-1H-pyrrolo[3,2-c]pyridin-3-yl}ethyl)amine, 21
Show/Hide
|
C17H19N3
|
1
|
| 1 |
Ki = 270 nM
|
|
|
|
CP0433625
|
4-fluoro-N-[(3S)-1-[2-(2-phenylphenoxy)ethyl]pyrrolidin-3-yl]benzenesulfonamide
Show/Hide
|
C24H25FN2O3S
|
1
|
| 1 |
Ki = 271 nM
|
|
|
|
CP0537420
|
4-[3-(2,3-dichlorophenoxy)propyl]-6-(4-methylpiperazin-1-yl)-1,3,5-triazin-2-amine
Show/Hide
|
C17H22Cl2N6O
|
1
|
| 1 |
Ki = 274 nM
|
|
|
|
CP0494564
|
N-[3-[2-(dimethylamino)ethyl]-2-methyl-1H-inden-5-yl]naphthalene-1-sulfonamide
Show/Hide
|
C24H26N2O2S
|
1
|
| 1 |
Ki = 276 nM
|
|
|
|
CP0849204
|
3-Chloro-N-{1-[2-(biphenyl-2-yloxy)ethyl]piperidin-4-yl}-benzenesulfonamide
Show/Hide
|
C25H27ClN2O3S
|
1
|
| 1 |
Ki = 276 nM
|
|
|
|
CP0548032
|
1-(benzenesulfonyl)-3-[(4-methylpiperazin-1-yl)methyl]pyrrolo[2,3-b]pyridine
Show/Hide
|
C19H22N4O2S
|
1
|
| 1 |
Ki = 277 nM
|
|
|
|
CP0568683
|
4-N-[2-(1H-indol-3-yl)ethyl]-2-N-[2-(4-phenylpiperazin-1-yl)ethyl]-1,3,5-triazine-2,4,6-triamine
Show/Hide
|
C25H31N9
|
1
|
| 1 |
Ki = 277 nM
|
|
|
|
CP0443747
|
3-bromo-4-[(4-methylpiperazin-1-yl)methyl]-1-(4-propan-2-ylphenyl)sulfonylindole
Show/Hide
|
C23H28BrN3O2S
|
1
|
| 1 |
Ki = 278 nM
|
|
|
|
CP0553073
|
N,N-dimethyl-2-(1-propylsulfonylindol-3-yl)ethanamine
Show/Hide
|
C15H22N2O2S
|
1
|
| 1 |
Ki = 280 nM
|
|
|
|
CP0440887
|
1-[3-[1-(benzenesulfonyl)indol-3-yl]-2-methyl-6,7-dihydro-5H-imidazo[1,2-a]pyrimidin-8-yl]ethanone
Show/Hide
|
C23H22N4O3S
|
1
|
| 1 |
Ki = 280 nM
|
|
|
|
CP0413781
|
N-[1-[2-(2-cyclopentylphenoxy)ethyl]piperidin-4-yl]-3-fluorobenzenesulfonamide
Show/Hide
|
C24H31FN2O3S
|
1
|
| 1 |
Ki = 281 nM
|
|
|
|
CP0399644
|
(3S)-2-[6-[4-(2-methylsulfanylphenyl)piperazin-1-yl]hexanoyl]-3,4-dihydro-1H-isoquinoline-3-carboxamide
Show/Hide
|
C27H36N4O2S
|
1
|
| 1 |
Ki = 282 nM
|
|
|
|
CP0571683
|
2-N-[5-[4-(2,3-dichlorophenyl)piperazin-1-yl]pentyl]-1,3,5-triazine-2,4,6-triamine
Show/Hide
|
C18H26Cl2N8
|
1
|
| 1 |
Ki = 282 nM
|
|
|
|
CP0223269
|
2-{[5,7-Dimethyl-3-(phenylsulfonyl)pyrazolo[1,5-a]pyrimidin-2-yl]oxy}ethanol
Show/Hide
|
C16H17N3O4S
|
1
|
| 1 |
Ki = 283 nM
|
|
|
|
CP0545014
|
2-[6-(4-naphthalen-1-ylpiperazin-1-yl)hexyl]-[1,2,4]triazolo[4,3-a]pyridin-3-one
Show/Hide
|
C26H31N5O
|
1
|
| 1 |
Ki = 285 nM
|
|
|
|
CP0953786
|
5-Bromo-1-(3-bromo benzenesulfonyl)-3-[2-(4-methyl piperazin-1-yl)ethyl]-1H-indole Dihydrochloride
Show/Hide
|
C21H25Br2Cl2N3O2S
|
1
|
| 1 |
Ki = 289 nM
|
|
|
|
CP0485369
|
N-[2-(4-chlorophenoxy)ethyl]-2-nitro-5-piperazin-1-ylaniline
Show/Hide
|
C18H21ClN4O3
|
1
|
| 1 |
Ki = 290 nM
|
|
|
|
CP0376267
|
N-[3-(aminomethyl)phenyl]benzenesulfonamide
Show/Hide
|
C13H14N2O2S
|
1
|
| 1 |
Ki = 290 nM
|
|
|
|
CP0462437
|
6-(4-methylpiperazin-1-yl)-1-(2-methylpropylsulfonyl)-4-(4-phenylmethoxyphenyl)pyrrolo[2,3-b]pyridine
Show/Hide
|
C29H34N4O3S
|
1
|
| 1 |
Ki = 290 nM
|
|
|
|
CP0391298
|
3-[4-[2-[(2S)-1-quinolin-5-ylsulfonylpyrrolidin-2-yl]ethyl]piperazin-1-yl]-1,2-benzoxazole
Show/Hide
|
C26H29N5O3S
|
1
|
| 1 |
Ki = 291 nM
|
|
|
|
CP0501995
|
(S)-5,7-dichloro-3-(4-methoxyphenyl)-3-methylquinoline-2,4(1H,3H)-dione
Show/Hide
|
C17H13Cl2NO3
|
1
|
| 1 |
Ki = 293 nM
|
|
|
|
CP0568318
|
2-[6-[4-(2,3-dichlorophenyl)piperazin-1-yl]hexyl]-[1,2,4]triazolo[4,3-a]pyridin-3-one
Show/Hide
|
C22H27Cl2N5O
|
1
|
| 1 |
Ki = 299 nM
|
|
|
|
CP0498747
|
N,N-dimethyl-2-(2-methyl-1H-indol-3-yl)ethanamine
Show/Hide
|
C13H18N2
|
1
|
| 1 |
Ki = 300 nM
|
|
|
|
CP0418454
|
N-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butyl]quinoline-7-sulfonamide
Show/Hide
|
C23H26Cl2N4O2S
|
1
|
| 1 |
Ki = 301 nM
|
|
|
|
CP0394125
|
3-(5-fluoro-1H-indol-3-yl)-1-[4-[4-(5-fluoro-1H-indol-3-yl)piperidin-1-yl]butyl]pyrrolidine-2,5-dione
Show/Hide
|
C29H30F2N4O2
|
1
|
| 1 |
Ki = 301 nM
|
|
|
|
CP0538566
|
2-[6-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]hexylsulfanyl]-1,3-benzoxazole
Show/Hide
|
C24H28N4OS2
|
1
|
| 1 |
Ki = 302 nM
|
|
|
|
CP0562343
|
2-(1-methylindol-3-yl)-N-[(5-phenylfuran-2-yl)methyl]ethanamine
Show/Hide
|
C22H22N2O
|
1
|
| 1 |
Ki = 303 nM
|
|
|
|
CP0444376
|
3-(4-bromophenyl)-5,7-dichloro-3-methylquinoline-2,4(1H,3H)-dione
Show/Hide
|
C16H10BrCl2NO2
|
1
|
| 1 |
Ki = 304 nM
|
|
|
|
CP0533916
|
4-(4-methylpiperazin-1-yl)-6-(thiophen-2-ylmethyl)-1,3,5-triazin-2-amine
Show/Hide
|
C13H18N6S
|
1
|
| 1 |
Ki = 305 nM
|
|
|
|
CP0156479
|
(+)-N-methyl-laurotetanine
Show/Hide
|
C20H23NO4
|
1
|
| 1 |
Ki = 306 nM
|
|
|
|
CP0448728
|
4-[4-[2-[4-(2,3-dichlorophenyl)piperazin-1-yl]ethyl]piperidin-1-yl]sulfonylisoquinoline
Show/Hide
|
C26H30Cl2N4O2S
|
1
|
| 1 |
Ki = 309 nM
|
|
|
|
CP0416051
|
3-[4-[2-[(2S)-1-quinolin-5-ylsulfonylpyrrolidin-2-yl]ethyl]piperazin-1-yl]-1,2-benzothiazole
Show/Hide
|
C26H29N5O2S2
|
1
|
| 1 |
Ki = 311 nM
|
|
|
|
CP0569761
|
1-[(2-bromophenyl)methyl]-3-[(4-methylpiperazin-1-yl)methyl]indole
Show/Hide
|
C21H24BrN3
|
1
|
| 1 |
Ki = 312 nM
|
|
|
|
CP0518983
|
3-[2-(3-chlorophenyl)ethyl]-2-methyl-7-piperazin-1-ylimidazo[4,5-b]pyridine
Show/Hide
|
C19H22ClN5
|
1
|
| 1 |
Ki = 312 nM
|
|
|
|
CP0413769
|
4-fluoro-N-[[1-[2-(2-propan-2-ylphenoxy)ethyl]piperidin-4-yl]methyl]benzenesulfonamide
Show/Hide
|
C23H31FN2O3S
|
1
|
| 1 |
Ki = 313 nM
|
|
|
|
CP0219574
|
3-[4-[2-[(2S)-1-isoquinolin-4-ylsulfonylpyrrolidin-2-yl]ethyl]piperazin-1-yl]-1,2-benzothiazole
Show/Hide
|
C26H29N5O2S2
|
1
|
| 1 |
Ki = 313 nM
|
|
|
|
CP0382802
|
3-[(2,4-dichlorophenyl)methyl]-1-[5-[4-(3,4-dichlorophenyl)piperazin-1-yl]pentyl]-5,5-dimethylimidazolidine-2,4-dione;hydrochloride
Show/Hide
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C27H32Cl4N4O2
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1
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| 1 |
Ki = 314 nM
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CP0484860
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4-fluoro-N-[[1-[2-(2-phenylphenoxy)ethyl]piperidin-4-yl]methyl]benzenesulfonamide
Show/Hide
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C26H29FN2O3S
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1
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| 1 |
Ki = 315 nM
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CP0538536
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4-(2-methylsulfonylphenyl)sulfonyl-8-piperazin-1-yl-2,3-dihydro-1,4-benzoxazine
Show/Hide
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C19H23N3O5S2
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1
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| 1 |
Ki = 316.23 nM
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CP0427389
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3-[(4-fluorophenyl)methyl]-2-methyl-7-piperazin-1-ylimidazo[4,5-b]pyridine
Show/Hide
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C18H20FN5
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1
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| 1 |
Ki = 317 nM
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CP0414548
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N-[6-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]hexyl]benzenesulfonamide
Show/Hide
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C23H30N4O2S2
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1
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| 1 |
Ki = 317 nM
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CP0513850
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1-[(3-chlorophenyl)methyl]-4-piperazin-1-ylimidazo[4,5-c]pyridine
Show/Hide
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C17H18ClN5
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1
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| 1 |
Ki = 320 nM
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CP0520823
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N-[1-(cyclopropylmethoxy)-2-methoxy-6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-10-yl]butanamide
Show/Hide
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C26H32N2O3
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1
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| 1 |
Ki = 322 nM
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CP0860096
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2,5-Difluoro-N-(1-{2-[(propan-2-yl)phenoxy]ethyl}piperidin-4-yl)-benzenesulfonamide
Show/Hide
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C22H28F2N2O3S
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1
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| 1 |
Ki = 324 nM
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CP0407076
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3-chloro-N-[8-[2-(3-phenylphenoxy)ethyl]-8-azabicyclo[3.2.1]octan-3-yl]benzenesulfonamide
Show/Hide
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C27H29ClN2O3S
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1
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| 1 |
Ki = 325 nM
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CP0453618
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N-[3-[4-(2,3-dichlorophenyl)piperazin-1-yl]propyl]quinoline-6-sulfonamide
Show/Hide
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C22H24Cl2N4O2S
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1
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| 1 |
Ki = 326 nM
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CP0574461
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(2-bromophenyl)-[5-fluoro-3-[(4-methylpiperazin-1-yl)methyl]indol-1-yl]methanone
Show/Hide
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C21H21BrFN3O
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1
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| 1 |
Ki = 326 nM
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CP0481685
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3,4-difluoro-N-[1-[2-(2-phenylphenoxy)ethyl]pyrrolidin-3-yl]benzenesulfonamide
Show/Hide
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C24H24F2N2O3S
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1
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| 1 |
Ki = 327 nM
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CP0531462
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1-(cyclopropylmethoxy)-2-methoxy-N,N,6-trimethyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-10-amine
Show/Hide
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C24H30N2O2
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1
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| 1 |
Ki = 329 nM
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CP0510213
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N-[3-[4-(1,2-benzoxazol-3-yl)piperazin-1-yl]propyl]-3-chloro-4-fluorobenzenesulfonamide
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C20H22ClFN4O3S
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1
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| 1 |
Ki = 330 nM
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CP0562344
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N-[2-(1H-indol-3-yl)ethyl]-N-[(5-phenylfuran-2-yl)methyl]propan-1-amine
Show/Hide
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C24H26N2O
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1
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| 1 |
Ki = 334 nM
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CP0490063
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1-[1-(5-Dimethylamino-naphthalene-1-sulfonyl)-piperidin-4-yl]-8-methyl-1,4-dihydro-benzo[d][1,3]oxazin-2-one
Show/Hide
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C26H29N3O4S
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1
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| 1 |
Ki = 336 nM
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CP0482614
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3-[(2-methoxyphenyl)methyl]-2-methyl-7-piperazin-1-ylimidazo[4,5-b]pyridine
Show/Hide
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C19H23N5O
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1
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| 1 |
Ki = 337 nM
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CP0445915
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5-[(2R)-2-[2-[4-(1-benzothiophen-4-yl)piperazin-1-yl]ethyl]piperidin-1-yl]sulfonylquinoline
Show/Hide
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C28H32N4O2S2
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1
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| 1 |
Ki = 337 nM
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CP0734688
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N-{4-[4-(4-Chlorophenyl)-piperazin-1-yl]-butyl}-3-quinolinesulfonamide hydrochloride
Show/Hide
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C23H28Cl2N4O2S
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1
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| 1 |
Ki = 339 nM
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CP0466079
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(2S)-2-[[4-[6-[4-[1-[(3-chlorophenyl)methyl]indol-4-yl]piperazin-1-yl]hexoxy]phenyl]methylamino]propanamide
Show/Hide
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C35H44ClN5O2
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1
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| 1 |
Ki = 340 nM
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CP0415694
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3-[4-[2-[(2S)-1-quinolin-5-ylsulfonylazetidin-2-yl]ethyl]piperazin-1-yl]-1,2-benzothiazole
Show/Hide
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C25H27N5O2S2
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1
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| 1 |
Ki = 344 nM
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CP0501994
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5-chloro-7-methoxy-3-methyl-3-phenylquinoline-2,4(1H,3H)-dione
Show/Hide
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C17H14ClNO3
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1
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| 1 |
Ki = 344.6 nM
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CP0564428
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4-[5-[[1-(5-methoxy-1H-indol-3-yl)propan-2-ylamino]methyl]furan-2-yl]phenol
Show/Hide
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C23H24N2O3
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1
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| 1 |
Ki = 345 nM
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CP0511649
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5,7-dichloro-3-(4-(dimethylamino)phenyl)-3-methylquinoline-2,4(1H,3H)-dione
Show/Hide
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C18H16Cl2N2O2
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1
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| 1 |
Ki = 346 nM
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CP0417067
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2-[6-[4-(3-methoxyphenyl)piperazin-1-yl]hexyl]benzo[de]isoquinoline-1,3-dione
Show/Hide
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C29H33N3O3
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1
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| 1 |
Ki = 347 nM
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CP0393702
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1-(2-bromophenyl)sulfonyl-5-methoxy-3-[(4-methylpiperazin-1-yl)methyl]indazole
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C20H23BrN4O3S
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1
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| 1 |
Ki = 348 nM
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CP0460483
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1-(2-bromophenyl)sulfonyl-3-[[4-(2-fluoroethyl)piperazin-1-yl]methyl]-5-methoxyindole
Show/Hide
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C22H25BrFN3O3S
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1
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| 1 |
Ki = 348 nM
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CP0390938
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3-[4-[2-[(2S)-1-isoquinolin-4-ylsulfonylazetidin-2-yl]ethyl]piperazin-1-yl]-1,2-benzothiazole
Show/Hide
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C25H27N5O2S2
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1
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| 1 |
Ki = 348 nM
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CP0568393
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1-[(3-chlorophenyl)methyl]-4-(3-methoxypiperidin-1-yl)pyrrolo[3,2-c]quinoline
Show/Hide
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C24H24ClN3O
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1
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| 1 |
Ki = 350 nM
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CP0531632
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N-(2-methoxy-6-methyl-1-prop-2-ynoxy-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-10-yl)butanamide
Show/Hide
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C25H28N2O3
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1
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| 1 |
Ki = 354 nM
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CP0431612
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4-[(4-chloro-3-methylphenoxy)methyl]-6-(4-methylpiperazin-1-yl)-1,3,5-triazin-2-amine
Show/Hide
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C16H21ClN6O
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1
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| 1 |
Ki = 355 nM
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CP0531466
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N-(1,2-dimethoxy-6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-10-yl)butanamide
Show/Hide
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C23H28N2O3
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1
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| 1 |
Ki = 356 nM
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CP0453912
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4-fluoro-N-[1-[2-(2-methylsulfanylphenoxy)ethyl]pyrrolidin-3-yl]benzenesulfonamide
Show/Hide
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C19H23FN2O3S2
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1
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| 1 |
Ki = 357 nM
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CP0391907
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3-(4-chlorophenyl)-5,6,7,8-tetrahydro-4H-[1,2]oxazolo[4,5-d]azepine
Show/Hide
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C13H13ClN2O
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1
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| 1 |
Ki = 360 nM
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CP0487359
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3-[4-[2-[(2S)-1-isoquinolin-5-ylsulfonylpyrrolidin-2-yl]ethyl]piperazin-1-yl]-1,2-benzothiazole
Show/Hide
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C26H29N5O2S2
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1
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| 1 |
Ki = 360 nM
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CP0948273
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{4-[1-(2-Bromobenzenesulfonyl)-1H-indol-3-ylmethyl]piperazin-1-yl}phenylmethanone Hydrochloride
Show/Hide
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C26H25BrClN3O3S
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1
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| 1 |
Ki = 365 nM
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CP0563987
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1-(3-fluorophenyl)sulfonyl-3-(1,2,3,6-tetrahydropyridin-4-yl)pyrrolo[2,3-f]quinoline
Show/Hide
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C22H18FN3O2S
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1
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| 1 |
Ki = 365 nM
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CP0432719
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2-[6-[4-(3-chlorophenyl)piperazin-1-yl]hexyl]-1,1-dioxo-1,2-benzothiazol-3-one
Show/Hide
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C23H28ClN3O3S
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1
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| 1 |
Ki = 372 nM
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CP0569023
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1-benzyl-2-methyl-4-piperazin-1-ylimidazo[4,5-c]pyridine
Show/Hide
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C18H21N5
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1
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| 1 |
Ki = 374 nM
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CP0478413
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3-[6-[4-[3-(trifluoromethyl)phenyl]piperazin-1-yl]hexyl]-2lambda6-thia-3-azatricyclo[6.3.1.04,12]dodeca-1(11),4,6,8(12),9-pentaene 2,2-dioxide;hydrochloride
Show/Hide
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C27H31ClF3N3O2S
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1
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| 1 |
Ki = 374 nM
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CP0399640
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5-[4-(2-phenylphenyl)piperazin-1-yl]-1-[(2S)-2-(piperidine-1-carbonyl)pyrrolidin-1-yl]pentan-1-one
Show/Hide
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C31H42N4O2
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1
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| 1 |
Ki = 376 nM
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CP0414533
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3-[6-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]hexyl]-1,3-diazatricyclo[6.3.1.04,12]dodeca-4,6,8(12)-trien-2-one
Show/Hide
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C27H33N5OS
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1
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| 1 |
Ki = 379 nM
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CP0543201
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1-[4-[[1-(2-bromophenyl)sulfonylindol-3-yl]methyl]piperazin-1-yl]ethanone
Show/Hide
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C21H22BrN3O3S
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1
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| 1 |
Ki = 385 nM
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CP0542762
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2-N-[6-[4-(2,3-dichlorophenyl)piperazin-1-yl]hexyl]-1,3,5-triazine-2,4,6-triamine
Show/Hide
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C19H28Cl2N8
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1
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| 1 |
Ki = 389 nM
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CP0401242
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3-[(2,4-dichlorophenyl)methyl]-1-[5-[4-(2,3-dichlorophenyl)piperazin-1-yl]pentyl]-5,5-dimethylimidazolidine-2,4-dione;hydrochloride
Show/Hide
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C27H32Cl4N4O2
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1
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| 1 |
Ki = 395 nM
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CP0476100
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N-benzyl-6-[(2S)-2-methyl-4-(2-phenylphenyl)piperazin-1-yl]hexanamide
Show/Hide
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C30H37N3O
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1
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| 1 |
Ki = 395 nM
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CP0892860
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N-{4-[4-(3-Chlorophenyl)-piperazin-1-yl]-butyl}-6-quinolinesulfonamide hydrochloride
Show/Hide
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C23H28Cl2N4O2S
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1
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| 1 |
Ki = 397 nM
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CP0877964
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1-(2-Bromobenzenesulfonyl)-5-bromo-3-[(4-methylpiperazin-1-yl)ethyl]-1H-indole Dihydrochloride
Show/Hide
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C21H25Br2Cl2N3O2S
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1
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| 1 |
Ki = 398 nM
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CP0466838
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2-(4-(4-(5-fluoro-1H-indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)butyl)isoindoline-1,3-dione
Show/Hide
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C25H24FN3O2
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1
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| 1 |
Ki = 398.11 nM
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CP0417575
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5-[4-[2-[4-(2,3-dichlorophenyl)piperazin-1-yl]ethyl]piperidin-1-yl]sulfonylquinoline
Show/Hide
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C26H30Cl2N4O2S
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1
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| 1 |
Ki = 401 nM
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CP0428023
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2-(benzyloxy)-N-(furan-2-ylmethyl)-5-(4-methylpiperazin-1-yl)benzenamine
Show/Hide
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C23H27N3O2
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1
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| 1 |
Ki = 402 nM
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CP0568317
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2-[6-[4-[3-(trifluoromethyl)phenyl]piperazin-1-yl]hexyl]-[1,2,4]triazolo[4,3-a]pyridin-3-one
Show/Hide
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C23H28F3N5O
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1
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| 1 |
Ki = 404 nM
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CP0389596
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6-[5-[4-(3,4-dichlorophenyl)piperazin-1-yl]pentyl]-2,4,7-trimethylpurino[7,8-a]imidazole-1,3-dione
Show/Hide
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C25H31Cl2N7O2
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1
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| 1 |
Ki = 405 nM
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CP0440392
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5-iodo-3-(3-methylimidazol-4-yl)-1H-indole
Show/Hide
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C12H10IN3
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1
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| 1 |
Ki = 407 nM
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CP0526507
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N-benzyl-2-methoxy-5-(4-methylpiperazin-1-yl)aniline
Show/Hide
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C19H25N3O
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1
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| 1 |
Ki = 409 nM
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CP0525831
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5-chloro-N-[[1-[2-(2-phenylphenoxy)ethyl]piperidin-4-yl]methyl]thiophene-2-sulfonamide
Show/Hide
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C24H27ClN2O3S2
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1
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| 1 |
Ki = 410 nM
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CP0367684
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(2-methoxy-6-methyl-1-prop-2-ynoxy-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-10-yl)urea
Show/Hide
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C22H23N3O3
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1
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| 1 |
Ki = 410 nM
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CP0382642
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N-[[4-(methoxymethoxy)phenyl]methyl]-6-[4-(2-phenylphenyl)piperazin-1-yl]hexanamide
Show/Hide
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C31H39N3O3
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1
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| 1 |
Ki = 413 nM
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CP0352456
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(1,2-dimethoxy-6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-10-yl)urea
Show/Hide
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C20H23N3O3
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1
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| 1 |
Ki = 415 nM
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CP0391906
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3-(4-fluorophenyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine
Show/Hide
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C13H14FN3
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1
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| 1 |
Ki = 416 nM
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CP0478894
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2-(1H-indol-3-yl)-N-[(5-naphthalen-1-ylthiophen-2-yl)methyl]ethanamine
Show/Hide
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C25H22N2S
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1
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| 1 |
Ki = 418 nM
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CP0542456
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N-[[5-(furan-2-yl)furan-2-yl]methyl]-2-(1H-indol-3-yl)ethanamine
Show/Hide
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C19H18N2O2
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1
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| 1 |
Ki = 419 nM
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CP0548631
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1-(3-chlorophenyl)sulfonyl-3-(1,2,3,6-tetrahydropyridin-4-yl)pyrrolo[2,3-f]quinoline
Show/Hide
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C22H18ClN3O2S
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1
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| 1 |
Ki = 427 nM
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CP0416279
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3-(5-methoxy-1H-indol-3-yl)-1-[4-[4-(5-methoxy-1H-indol-3-yl)piperidin-1-yl]butyl]pyrrolidine-2,5-dione
Show/Hide
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C31H36N4O4
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1
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| 1 |
Ki = 427 nM
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CP0458499
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N-[2-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]ethyl]-3-methylbenzenesulfonamide
Show/Hide
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C20H24N4O2S2
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1
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| 1 |
Ki = 430 nM
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CP0495706
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3-[6-[4-(4-chlorophenyl)piperazin-1-yl]hexyl]-2lambda6-thia-3-azatricyclo[6.3.1.04,12]dodeca-1(11),4,6,8(12),9-pentaene 2,2-dioxide;hydrochloride
Show/Hide
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C26H31Cl2N3O2S
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1
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| 1 |
Ki = 433 nM
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CP0445704
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N-benzyl-6-[(2R)-2-methyl-4-(2-phenylphenyl)piperazin-1-yl]hexanamide
Show/Hide
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C30H37N3O
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1
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| 1 |
Ki = 434 nM
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CP0444016
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2-[4-[3-(1H-indol-3-yl)piperidin-1-yl]butyl]-4-phenylpyrido[1,2-c]pyrimidine-1,3-dione
Show/Hide
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C31H32N4O2
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1
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| 1 |
Ki = 435 nM
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CP0434049
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N,N-dimethyl-2-(1-octylsulfonylindol-3-yl)ethanamine
Show/Hide
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C20H32N2O2S
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1
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| 1 |
Ki = 440 nM
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CP0507100
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4-[(4-methoxyphenyl)methyl]-6-(4-methylpiperazin-1-yl)-1,3,5-triazin-2-amine
Show/Hide
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C16H22N6O
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1
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| 1 |
Ki = 440 nM
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CP0444713
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2-(1-(4-(trifluoromethyl)benzyl)-1H-indol-3-yl)-N,N-dimethylethanamine
Show/Hide
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C20H21F3N2
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1
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| 1 |
Ki = 445 nM
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CP0472682
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5-[4-[2-[4-(3-chlorophenyl)piperazin-1-yl]ethyl]piperidin-1-yl]sulfonylquinoline
Show/Hide
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C26H31ClN4O2S
|
1
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| 1 |
Ki = 445 nM
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CP0388194
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5-Chloro-N-(3-{4-[8-({[5-(dimethylamino)-1-naphthyl]sulfonyl}-amino)octyl]piperazin-1-yl}-4-methoxyphenyl)-3-methyl-1-benzothiophene-2-sulfonamide
Show/Hide
|
C40H50ClN5O5S3
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1
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| 1 |
Ki = 447 nM
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CP0282007
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6-[4-[4-(4-chlorophenyl)piperazin-1-yl]butyl]-2,4-dimethyl-7-phenylpurino[7,8-a]imidazole-1,3-dione
Show/Hide
|
C29H32ClN7O2
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1
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| 1 |
Ki = 447 nM
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CP0569022
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1-benzyl-4-piperazin-1-ylimidazo[4,5-c]pyridine
Show/Hide
|
C17H19N5
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1
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| 1 |
Ki = 450 nM
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CP0459430
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2-[4-[3-(5-methoxy-1H-indol-3-yl)piperidin-1-yl]butyl]-4-(4-methoxyphenyl)-5,6,7,8-tetrahydropyrido[1,2-c]pyrimidine-1,3-dione
Show/Hide
|
C33H40N4O4
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1
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| 1 |
Ki = 452 nM
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CP0418455
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N-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butyl]isoquinoline-3-sulfonamide
Show/Hide
|
C23H26Cl2N4O2S
|
1
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| 1 |
Ki = 454 nM
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CP0538216
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N-[4-(5-methoxy-1-naphthalen-2-ylsulfonylindol-3-yl)-5-methyl-1H-imidazol-2-yl]propanamide
Show/Hide
|
C26H24N4O4S
|
1
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| 1 |
Ki = 455 nM
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CP0476720
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3-[4-[2-[(2S)-1-quinolin-5-ylsulfonylazepan-2-yl]ethyl]piperazin-1-yl]-1,2-benzothiazole
Show/Hide
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C28H33N5O2S2
|
1
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| 1 |
Ki = 457 nM
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CP0482089
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2-[6-[4-(2-chlorophenyl)piperazin-1-yl]hexyl]-1,1-dioxo-1,2-benzothiazol-3-one
Show/Hide
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C23H28ClN3O3S
|
1
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| 1 |
Ki = 459 nM
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CP0471364
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methyl 4-(4-methylpiperazin-1-yl)-2-(2-phenylethylamino)benzoate
Show/Hide
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C21H27N3O2
|
1
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| 1 |
Ki = 462 nM
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CP0444754
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4-[3-(2,5-dichlorophenoxy)propyl]-6-(4-methylpiperazin-1-yl)-1,3,5-triazin-2-amine
Show/Hide
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C17H22Cl2N6O
|
1
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| 1 |
Ki = 470 nM
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CP0107214
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3-fluoro-N-[1-[2-(2-propan-2-ylphenoxy)ethyl]piperidin-4-yl]benzenesulfonamide
Show/Hide
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C22H29FN2O3S
|
1
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| 1 |
Ki = 471 nM
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CP0443915
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4-[5-[[1-(1H-indol-3-yl)propan-2-ylamino]methyl]furan-2-yl]phenol
Show/Hide
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C22H22N2O2
|
1
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| 1 |
Ki = 475 nM
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CP0544199
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2-N-[2-(2,3-dichloroanilino)ethyl]-4-N-[2-(1H-indol-3-yl)ethyl]-1,3,5-triazine-2,4,6-triamine
Show/Hide
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C21H22Cl2N8
|
1
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| 1 |
Ki = 475 nM
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CP0483351
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3-[6-[4-(2-ethoxyphenyl)piperazin-1-yl]hexyl]-2lambda6-thia-3-azatricyclo[6.3.1.04,12]dodeca-1(11),4,6,8(12),9-pentaene 2,2-dioxide
Show/Hide
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C28H35N3O3S
|
1
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| 1 |
Ki = 476 nM
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CP0382643
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N-[(1S)-1-phenylethyl]-6-[4-(2-phenylphenyl)piperazin-1-yl]hexanamide
Show/Hide
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C30H37N3O
|
1
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| 1 |
Ki = 480 nM
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CP0478414
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1-[6-[4-(3-chlorophenyl)piperazin-1-yl]hexyl]benzo[cd]indol-2-one;hydrochloride
Show/Hide
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C27H31Cl2N3O
|
1
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| 1 |
Ki = 480 nM
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CP0503891
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N-[5-(4-methylpiperazin-1-yl)-2-nitrophenyl]pyrrol-1-amine
Show/Hide
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C15H19N5O2
|
1
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| 1 |
Ki = 481 nM
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CP0371742
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1-(3-(3,5-dimethyl-1H-pyrazol-1-yl)-4-nitrophenyl)piperazine
Show/Hide
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C15H19N5O2
|
1
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| 1 |
Ki = 482 nM
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CP0405275
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3-[(4-methylpiperazin-1-yl)methyl]-1H-indole
Show/Hide
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C14H19N3
|
1
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| 1 |
Ki = 482 nM
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CP0449729
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N-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butyl]quinoline-6-sulfonamide
Show/Hide
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C23H26Cl2N4O2S
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1
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| 1 |
Ki = 484 nM
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CP0457692
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2-(1H-indol-3-yl)-N-[[5-(3-propan-2-yloxyphenyl)furan-2-yl]methyl]ethanamine
Show/Hide
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C24H26N2O2
|
1
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| 1 |
Ki = 486 nM
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CP0530031
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(1R,2S,6R,7S)-4-[6-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]hexyl]-4-azatricyclo[5.2.1.02,6]decane-3,5-dione
Show/Hide
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C26H34N4O2S
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1
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| 1 |
Ki = 486 nM
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CP0513115
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N'-[3-(benzenesulfonyl)-5,7-dimethylpyrazolo[1,5-a]pyrimidin-2-yl]-N,N,N'-trimethylethane-1,2-diamine
Show/Hide
|
C19H25N5O2S
|
1
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| 1 |
Ki = 489 nM
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CP0429321
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2-[3-[4-(1-benzylindol-3-yl)piperidin-1-yl]propoxy]benzamide
Show/Hide
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C30H33N3O2
|
1
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| 1 |
Ki = 490 nM
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CP0468442
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2-(benzenesulfonyl)aniline
Show/Hide
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C12H11NO2S
|
1
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| 1 |
Ki = 491 nM
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CP0321822
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4-(benzenesulfonyl)-11-methyl-5-methylsulfanyl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1,3,5,8-tetraene
Show/Hide
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C17H18N4O2S2
|
1
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| 1 |
Ki = 492 nM
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CP0456120
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3-(4-methylphenyl)-5,6,7,8-tetrahydro-4H-[1,2]oxazolo[4,5-d]azepine
Show/Hide
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C14H16N2O
|
1
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| 1 |
Ki = 492 nM
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CP0417091
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3-[6-[4-(2-nitrophenyl)piperazin-1-yl]hexyl]-2lambda6-thia-3-azatricyclo[6.3.1.04,12]dodeca-1(11),4,6,8(12),9-pentaene 2,2-dioxide
Show/Hide
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C26H30N4O4S
|
1
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| 1 |
Ki = 494 nM
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CP0391297
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3-[4-[2-[(2S)-1-isoquinolin-4-ylsulfonylpyrrolidin-2-yl]ethyl]piperazin-1-yl]-1,2-benzoxazole
Show/Hide
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C26H29N5O3S
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1
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| 1 |
Ki = 497 nM
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CP0521248
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N-[4-[1-(benzenesulfonyl)indol-4-yl]-5-methyl-1H-imidazol-2-yl]propanamide
Show/Hide
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C21H20N4O3S
|
1
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| 1 |
Ki = 501 nM
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CP0426093
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N-[1-[2-(2-propan-2-ylphenoxy)ethyl]pyrrolidin-3-yl]quinoline-8-sulfonamide
Show/Hide
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C24H29N3O3S
|
1
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| 1 |
Ki = 504 nM
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CP0520838
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N-[1-(cyclopropylmethoxy)-2-methoxy-6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-10-yl]methanesulfonamide
Show/Hide
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C23H28N2O4S
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1
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| 1 |
Ki = 505 nM
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CP0542766
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2-N-[2-(1H-indol-3-yl)ethyl]-4-N-[4-(4-phenylpiperazin-1-yl)butyl]-1,3,5-triazine-2,4,6-triamine
Show/Hide
|
C27H35N9
|
1
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| 1 |
Ki = 506 nM
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CP0382745
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4-(4-methylpiperazin-1-yl)-6-(phenoxymethyl)-1,3,5-triazin-2-amine
Show/Hide
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C15H20N6O
|
1
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| 1 |
Ki = 507 nM
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CP0495707
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3-[6-[4-(2-chlorophenyl)piperazin-1-yl]hexyl]-2lambda6-thia-3-azatricyclo[6.3.1.04,12]dodeca-1(11),4,6,8(12),9-pentaene 2,2-dioxide;hydrochloride
Show/Hide
|
C26H31Cl2N3O2S
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1
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| 1 |
Ki = 507 nM
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CP0438561
|
2-(5-methoxy-1-methylindol-3-yl)-N,N-dimethylethanamine
Show/Hide
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C14H20N2O
|
1
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| 1 |
Ki = 510 nM
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CP0121966
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6-[4-[4-(2,3-dimethylphenyl)piperazin-1-yl]butyl]-2,4,7-trimethylpurino[7,8-a]imidazole-1,3-dione
Show/Hide
|
C26H35N7O2
|
1
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| 1 |
Ki = 510 nM
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CP0381351
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2,5-difluoro-N-[1-[2-(2-phenylphenoxy)ethyl]pyrrolidin-3-yl]benzenesulfonamide
Show/Hide
|
C24H24F2N2O3S
|
1
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| 1 |
Ki = 515 nM
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CP0443916
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4-[5-[[2-(5-fluoro-1-benzofuran-3-yl)ethylamino]methyl]furan-2-yl]phenol
Show/Hide
|
C21H18FNO3
|
1
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| 1 |
Ki = 522 nM
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CP0402603
|
4-{5-[4-(Dimethylamino)phenyl]-1,3-oxazol-2-yl}-N-(4-methoxy-3-piperazin-1-ylphenyl)benzenesulfonamide
Show/Hide
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C28H31N5O4S
|
1
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| 1 |
Ki = 523 nM
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CP0540236
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[1-(cyclopropylmethoxy)-2-methoxy-6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-10-yl]urea
Show/Hide
|
C23H27N3O3
|
1
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| 1 |
Ki = 527 nM
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CP0578854
|
4-[5-[[2-(1H-pyrrolo[2,3-b]pyridin-3-yl)ethylamino]methyl]furan-2-yl]phenol
Show/Hide
|
C20H19N3O2
|
1
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| 1 |
Ki = 531 nM
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CP0530033
|
(1R,2S,6R,7S)-4-[6-[4-(2,3-dichlorophenyl)piperazin-1-yl]hexyl]-4-azatricyclo[5.2.1.02,6]decane-3,5-dione
Show/Hide
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C25H33Cl2N3O2
|
1
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| 1 |
Ki = 536 nM
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CP0453913
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5-chloro-N-[(3S)-1-[2-(2-propan-2-ylphenoxy)ethyl]pyrrolidin-3-yl]thiophene-2-sulfonamide
Show/Hide
|
C19H25ClN2O3S2
|
1
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| 1 |
Ki = 537 nM
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CP0390348
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3-fluoro-N-[8-[2-(3-propan-2-ylphenoxy)ethyl]-8-azabicyclo[3.2.1]octan-3-yl]benzenesulfonamide
Show/Hide
|
C24H31FN2O3S
|
1
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| 1 |
Ki = 539 nM
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CP0915709
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1-((R)-1-Methyl-pyrrolidin-2-ylmethyl)-1H-indole hydrochloride
Show/Hide
|
C14H19ClN2
|
1
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| 1 |
Ki = 550 nM
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CP0541120
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5-chloro-4-fluoro-3-(3-methylimidazol-4-yl)-1H-indole
Show/Hide
|
C12H9ClFN3
|
1
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| 1 |
Ki = 550 nM
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CP0433627
|
5-chloro-N-[(3S)-1-[2-(2-phenylphenoxy)ethyl]pyrrolidin-3-yl]thiophene-2-sulfonamide
Show/Hide
|
C22H23ClN2O3S2
|
1
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| 1 |
Ki = 551 nM
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CP0454528
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5-(Dimethylamino)-N-(3-{4-[6-({[5-(dimethylamino)-1-naphthyl]-sulfonyl}amino)hexyl]piperazin-1-yl}-4-methoxyphenyl)naphthalene-1-sulfonamide
Show/Hide
|
C41H52N6O5S2
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1
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| 1 |
Ki = 554 nM
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CP0482397
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6-chloro-N-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butyl]quinoline-3-sulfonamide
Show/Hide
|
C23H25Cl3N4O2S
|
1
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| 1 |
Ki = 555 nM
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CP0487393
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N-[[5-(3-methoxyphenyl)furan-2-yl]methyl]-2-(1-methylindol-3-yl)ethanamine
Show/Hide
|
C23H24N2O2
|
1
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| 1 |
Ki = 556 nM
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CP0402811
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4-fluoro-N-[8-[2-(3-propan-2-ylphenoxy)ethyl]-8-azabicyclo[3.2.1]octan-3-yl]benzenesulfonamide
Show/Hide
|
C24H31FN2O3S
|
1
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| 1 |
Ki = 559 nM
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CP0486993
|
N-[3-[4-(1,2-benzoxazol-3-yl)piperazin-1-yl]propyl]-6-chloro-1-benzothiophene-2-sulfonamide
Show/Hide
|
C22H23ClN4O3S2
|
1
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| 1 |
Ki = 560 nM
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CP0211753
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5,7-Dimethyl-3-phenylsulfonyl-pyrazolo[1,5-a]pyrimidine
Show/Hide
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C14H13N3O2S
|
1
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| 1 |
Ki = 561 nM
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CP0376752
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N-[(1R)-1-phenylethyl]-6-[4-(2-phenylphenyl)piperazin-1-yl]hexanamide
Show/Hide
|
C30H37N3O
|
1
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| 1 |
Ki = 561 nM
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CP0555842
|
4-(4-aminophenyl)sulfonylbenzene-1,2-diamine
Show/Hide
|
C12H13N3O2S
|
1
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| 1 |
Ki = 564 nM
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CP0414547
|
1-[6-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]hexyl]benzo[cd]indol-2-one
Show/Hide
|
C28H30N4OS
|
1
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| 1 |
Ki = 568 nM
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CP0088232
|
N,N-diethyl-2-(1H-indol-3-yl)ethanamine
Show/Hide
|
C14H20N2
|
1
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| 1 |
Ki = 575 nM
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CP0544200
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4-N-[2-(2,3-dichlorophenyl)ethyl]-2-N-[2-(1H-indol-3-yl)ethyl]-1,3,5-triazine-2,4,6-triamine
Show/Hide
|
C21H21Cl2N7
|
1
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| 1 |
Ki = 575 nM
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CP0545007
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3-[6-[4-(3-chlorophenyl)piperazin-1-yl]hexyl]-1,3-diazatricyclo[6.3.1.04,12]dodeca-4,6,8(12)-triene-2-thione
Show/Hide
|
C26H33ClN4S
|
1
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| 1 |
Ki = 582 nM
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CP0476615
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1-[5-[1-(benzenesulfonyl)indol-3-yl]-6-methyl-2,3-dihydroimidazo[1,2-a]imidazol-1-yl]ethanone
Show/Hide
|
C22H20N4O3S
|
1
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| 1 |
Ki = 585 nM
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CP0542760
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2-N-[2-(1H-indol-3-yl)ethyl]-4-N-[2-(2-methoxyphenyl)ethyl]-1,3,5-triazine-2,4,6-triamine
Show/Hide
|
C22H25N7O
|
1
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| 1 |
Ki = 585 nM
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CP0505620
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2-(1-(isopropylsulfonyl)-1H-indol-3-yl)-N,N-dimethylethanamine
Show/Hide
|
C15H22N2O2S
|
1
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| 1 |
Ki = 590 nM
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CP0390722
|
N-[4-(3,4-dihydro-1H-isoquinolin-2-yl)butyl]quinoline-3-sulfonamide
Show/Hide
|
C22H25N3O2S
|
1
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| 1 |
Ki = 590 nM
|
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CP0398683
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2-[3-[4-(1-benzylindol-3-yl)-3,6-dihydro-2H-pyridin-1-yl]propoxy]benzamide
Show/Hide
|
C30H31N3O2
|
1
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| 1 |
Ki = 590 nM
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CP0562205
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N-(2-methoxy-6-methyl-1-prop-2-enoxy-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-10-yl)methanesulfonamide
Show/Hide
|
C22H26N2O4S
|
1
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| 1 |
Ki = 590 nM
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CP0399643
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(3S)-2-[5-[4-(2-phenylphenyl)piperazin-1-yl]pentanoyl]-3,4-dihydro-1H-isoquinoline-3-carboxamide
Show/Hide
|
C31H36N4O2
|
1
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| 1 |
Ki = 594 nM
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CP0449784
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N-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butyl]quinoline-8-sulfonamide
Show/Hide
|
C23H26Cl2N4O2S
|
1
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| 1 |
Ki = 598 nM
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CP0400693
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1-[(2S)-2-(piperidine-1-carbonyl)pyrrolidin-1-yl]-7-[4-(2-propan-2-ylphenyl)piperazin-1-yl]heptan-1-one
Show/Hide
|
C30H48N4O2
|
1
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| 1 |
Ki = 603 nM
|
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CP0426679
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4,5-difluoro-3-(3-methylimidazol-4-yl)-1H-indole
Show/Hide
|
C12H9F2N3
|
1
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| 1 |
Ki = 603 nM
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CP0046432
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N-[(4-cyanophenyl)methyl]-6-[4-[4-fluoro-2-(4-methoxyphenyl)phenyl]piperazin-1-yl]hexanamide
Show/Hide
|
C31H35FN4O2
|
1
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| 1 |
Ki = 614 nM
|
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CP0390937
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3-[4-[2-[(2S)-1-quinolin-4-ylsulfonylazepan-2-yl]ethyl]piperazin-1-yl]-1,2-benzothiazole
Show/Hide
|
C28H33N5O2S2
|
1
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| 1 |
Ki = 623 nM
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CP0416668
|
3-[6-[4-(3-chlorophenyl)piperazin-1-yl]hexyl]-2lambda6-thia-3-azatricyclo[6.3.1.04,12]dodeca-1(11),4,6,8(12),9-pentaene 2,2-dioxide;hydrochloride
Show/Hide
|
C26H31Cl2N3O2S
|
1
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| 1 |
Ki = 624 nM
|
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CP0492795
|
4-(2-fluorophenyl)sulfonyl-2,3-dihydro-1,4-benzoxazin-8-amine
Show/Hide
|
C14H13FN2O3S
|
1
|
| 1 |
Ki = 630.96 nM
|
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CP0853816
|
3-((R)-1-Methyl-pyrrolidin-2-ylmethyl)-1H-indole hydrochloride
Show/Hide
|
C14H19ClN2
|
1
|
| 1 |
Ki = 640 nM
|
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CP0408597
|
4-Inden-(1E)-ylidenemethyl-phenylamine
Show/Hide
|
C16H13N
|
1
|
| 1 |
Ki = 640 nM
|
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CP0376759
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N-[[4-(methoxymethoxy)phenyl]methyl]-6-[4-[2-(4-methoxyphenyl)phenyl]piperazin-1-yl]hexanamide
Show/Hide
|
C32H41N3O4
|
1
|
| 1 |
Ki = 640 nM
|
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CP0475050
|
5-[4-[2-[4-[3-(trifluoromethyl)phenyl]piperazin-1-yl]ethyl]piperidin-1-yl]sulfonylquinoline
Show/Hide
|
C27H31F3N4O2S
|
1
|
| 1 |
Ki = 640 nM
|
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CP0853601
|
1-Methyl-N-(1-{2-[(propan-2-yl)phenoxy]ethyl}piperidin-4-yl)-1H-pyrazole-4-sulfonamide
Show/Hide
|
C20H30N4O3S
|
1
|
| 1 |
Ki = 641 nM
|
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CP0445925
|
5-[(2R)-2-[2-[4-(1H-indol-4-yl)piperazin-1-yl]ethyl]pyrrolidin-1-yl]sulfonylquinoline
Show/Hide
|
C27H31N5O2S
|
1
|
| 1 |
Ki = 641 nM
|
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CP0538554
|
6-[4-[2-(4-methoxyphenyl)phenyl]piperazin-1-yl]-N-[(1S)-1-phenylethyl]hexanamide
Show/Hide
|
C31H39N3O2
|
1
|
| 1 |
Ki = 652 nM
|
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CP0400394
|
5'-Chloro-1H,1''H-[3,3':3',3''-terindol]-2'(1'H)-one (4c)
Show/Hide
|
C24H16ClN3O
|
2
|
| 1 |
Ki = 670 nM
|
|
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| 2 |
Ki = 720 nM
|
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CP0417090
|
2-[6-[4-(2-methoxyphenyl)piperazin-1-yl]hexyl]benzo[de]isoquinoline-1,3-dione
Show/Hide
|
C29H33N3O3
|
1
|
| 1 |
Ki = 671 nM
|
|
|
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CP0486986
|
N-[2-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]ethyl]naphthalene-2-sulfonamide
Show/Hide
|
C23H24N4O2S2
|
1
|
| 1 |
Ki = 680 nM
|
|
|
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CP0445064
|
2-[3-[2-(1-benzylindol-3-yl)ethylamino]propoxy]benzamide
Show/Hide
|
C27H29N3O2
|
1
|
| 1 |
Ki = 680 nM
|
|
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CP0483353
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1-[6-[4-(4-chlorophenyl)piperazin-1-yl]hexyl]benzo[cd]indol-2-one;hydrochloride
Show/Hide
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C27H31Cl2N3O
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1
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| 1 |
Ki = 689 nM
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CP0530348
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2-[4-[3-(5-methoxy-1H-indol-3-yl)piperidin-1-yl]butyl]-4-(4-methoxyphenyl)pyrido[1,2-c]pyrimidine-1,3-dione
Show/Hide
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C33H36N4O4
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1
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| 1 |
Ki = 690 nM
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CP0519021
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N-[[5-(3,4-dimethoxyphenyl)furan-2-yl]methyl]-2-(1H-indol-3-yl)ethanamine
Show/Hide
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C23H24N2O3
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1
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| 1 |
Ki = 693 nM
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CP0543753
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1-[(3-chlorophenyl)methyl]-N-(oxolan-2-ylmethyl)pyrrolo[3,2-c]quinolin-4-amine
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C23H22ClN3O
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1
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| 1 |
Ki = 696 nM
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CP0463475
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4-(4-fluorophenyl)-2-[4-[3-(1H-indol-3-yl)piperidin-1-yl]butyl]pyrido[1,2-c]pyrimidine-1,3-dione
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C31H31FN4O2
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1
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| 1 |
Ki = 697 nM
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CP0377051
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N-[(1S)-1-(4-cyanophenyl)ethyl]-6-[4-[2-(4-methoxyphenyl)phenyl]piperazin-1-yl]hexanamide
Show/Hide
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C32H38N4O2
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1
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| 1 |
Ki = 700 nM
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CP0514793
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2-[5-[4-(4-chlorophenyl)piperazin-1-yl]pentyl]-1,1-dioxo-1,2-benzothiazol-3-one
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C22H26ClN3O3S
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1
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| 1 |
Ki = 703 nM
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CP0384693
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3-[6-[4-(2-fluorophenyl)piperazin-1-yl]hexyl]-2lambda6-thia-3-azatricyclo[6.3.1.04,12]dodeca-1(11),4,6,8(12),9-pentaene 2,2-dioxide;hydrochloride
Show/Hide
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C26H31ClFN3O2S
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1
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| 1 |
Ki = 710 nM
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CP0386364
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1-(benzenesulfonyl)-3-(1,2,3,6-tetrahydropyridin-4-yl)pyrrolo[2,3-f]quinoline
Show/Hide
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C22H19N3O2S
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1
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| 1 |
Ki = 711 nM
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CP0535835
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5-chloro-7-(dimethylamino)-3-methyl-3-phenylquinoline-2,4(1H,3H)-dione
Show/Hide
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C18H17ClN2O2
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1
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| 1 |
Ki = 715 nM
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CP0507071
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6-[4-[2-(4-methoxyphenyl)phenyl]piperazin-1-yl]-N-[(1R)-1-phenylethyl]hexanamide
Show/Hide
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C31H39N3O2
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1
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| 1 |
Ki = 721 nM
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CP0471140
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5,7-dimethoxy-3-methyl-3-phenylquinoline-2,4(1H,3H)-dione
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C18H17NO4
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1
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| 1 |
Ki = 728 nM
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CP0435657
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2-[4-[3-(5-fluoro-1H-indol-3-yl)piperidin-1-yl]butyl]-4-(4-fluorophenyl)-5,6,7,8-tetrahydropyrido[1,2-c]pyrimidine-1,3-dione
Show/Hide
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C31H34F2N4O2
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1
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| 1 |
Ki = 728 nM
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CP0408780
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4-(Indane-1-sulfonyl)-phenylamine
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C15H15NO2S
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1
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| 1 |
Ki = 740 nM
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CP0576381
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1-[(3-methoxyphenyl)methyl]-4-(4-methoxypiperidin-1-yl)pyrrolo[3,2-c]quinoline
Show/Hide
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C25H27N3O2
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1
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| 1 |
Ki = 740 nM
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CP0526476
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5-Chloro-N-(4-{[8-({[5-(dimethylamino)-1-naphthyl]sulfonyl}-amino)octyl]oxy}-3-piperazin-1-ylphenyl)-3-methyl-1-benzothiophene-2-sulfonamide
Show/Hide
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C39H48ClN5O5S3
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1
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| 1 |
Ki = 741 nM
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CP0848197
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(E)-5-((5-bromo-1H-indol-3-yl)methylene)-2-iminoimidazolidin-4-one
Show/Hide
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C12H9BrN4O
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1
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| 1 |
Ki = 742 nM
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CP0445706
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N-[(4-cyanophenyl)methyl]-6-[4-[2-(4-methoxyphenyl)phenyl]piperazin-1-yl]hexanamide
Show/Hide
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C31H36N4O2
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1
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| 1 |
Ki = 745 nM
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CP0388195
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5-Chloro-N-[4-({[5-(dimethylamino)-1-naphthyl]sulfonyl}amino)-butyl]-N-(4-methoxy-3-piperazin-1-ylphenyl)-3-methyl-1-benzothiophene-2-sulfonamide
Show/Hide
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C36H42ClN5O5S3
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1
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| 1 |
Ki = 747 nM
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CP0904743
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N-{4-[4-(4-Chlorophenyl)-piperazin-1-yl]-butyl}-4-isoquinolinesulfonamide hydrochloride
Show/Hide
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C23H28Cl2N4O2S
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1
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| 1 |
Ki = 750 nM
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CP0041761
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2-(4-hydroxyphenyl)-3-({4-[2-(piperidin-1-yl)ethoxy]phenyl}carbonyl)-1-benzothiophen-6-ol
Show/Hide
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C28H27NO4S
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1
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| 1 |
Ki = 750 nM
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CP0435400
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N-[4-[1-(benzenesulfonyl)-5-fluoroindol-3-yl]-5-methyl-1H-imidazol-2-yl]acetamide
Show/Hide
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C20H17FN4O3S
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1
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| 1 |
Ki = 759 nM
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CP0476750
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N-[3-(benzenesulfonyl)-5,7-dimethylpyrazolo[1,5-a]pyrimidin-2-yl]-N',N'-dimethylpropane-1,3-diamine
Show/Hide
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C19H25N5O2S
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1
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| 1 |
Ki = 764 nM
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CP0466249
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4-[(2R)-2-[2-[4-(1H-indol-4-yl)piperazin-1-yl]ethyl]pyrrolidin-1-yl]sulfonylisoquinoline
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C27H31N5O2S
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1
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| 1 |
Ki = 766 nM
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CP0575067
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2-N-[2-(2,3-dichlorophenoxy)ethyl]-4-N-[2-(1H-indol-3-yl)ethyl]-1,3,5-triazine-2,4,6-triamine
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C21H21Cl2N7O
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1
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| 1 |
Ki = 771 nM
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CP0532783
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N-[6-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]hexyl]-4-methyl-N-phenylbenzenesulfonamide
Show/Hide
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C30H36N4O2S2
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1
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| 1 |
Ki = 772 nM
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CP0421347
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2-(1H-indol-3-yl)-N-[[5-(4-nitrophenyl)furan-2-yl]methyl]ethanamine
Show/Hide
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C21H19N3O3
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1
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| 1 |
Ki = 774 nM
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CP0467727
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2-[6-[4-(2-methoxyphenyl)piperazin-1-yl]hexyl]-1,1-dioxo-1,2-benzothiazol-3-one
Show/Hide
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C24H31N3O4S
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1
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| 1 |
Ki = 779 nM
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CP0417576
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5-[4-[2-[4-(3,4-dichlorophenyl)piperazin-1-yl]ethyl]piperidin-1-yl]sulfonylquinoline
Show/Hide
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C26H30Cl2N4O2S
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1
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| 1 |
Ki = 791 nM
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CP0421839
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3-(3-ethylimidazol-4-yl)-4,5-difluoro-1H-indole
Show/Hide
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C13H11F2N3
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1
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| 1 |
Ki = 794 nM
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CP0528449
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5-bromo-4-fluoro-3-(3-methylimidazol-4-yl)-1H-indole
Show/Hide
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C12H9BrFN3
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1
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| 1 |
Ki = 794 nM
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CP0578376
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1-[(3-chlorophenyl)methyl]-4-(4-methoxypiperidin-1-yl)pyrrolo[3,2-c]quinoline
Show/Hide
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C24H24ClN3O
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1
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| 1 |
Ki = 799 nM
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CP0526779
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6-[6-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]hexoxy]-3,4-dihydro-1H-quinolin-2-one
Show/Hide
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C26H32N4O2S
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1
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| 1 |
Ki = 805 nM
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CP0459263
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N-[3-[4-(2-methoxyphenyl)piperazin-1-yl]propyl]quinoline-6-sulfonamide
Show/Hide
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C23H28N4O3S
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1
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| 1 |
Ki = 825 nM
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CP0569025
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3-[(2-chlorophenyl)methyl]-2-methyl-7-piperazin-1-ylimidazo[4,5-b]pyridine
Show/Hide
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C18H20ClN5
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1
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| 1 |
Ki = 829 nM
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CP0376742
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3-[2-[4-(2-phenylphenyl)piperazin-1-yl]ethoxy]-N-[[4-(trifluoromethyl)phenyl]methyl]propanamide
Show/Hide
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C29H32F3N3O2
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1
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| 1 |
Ki = 830 nM
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CP0455245
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3-chloro-N-[[1-[2-(3-fluorophenoxy)ethyl]piperidin-4-yl]methyl]benzenesulfonamide
Show/Hide
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C20H24ClFN2O3S
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1
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| 1 |
Ki = 831 nM
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CP0469237
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N-[4-[2-[4-[3-(4-amino-5-chloro-2-methoxyphenyl)-3-oxopropyl]piperidin-1-yl]ethylsulfamoyl]phenyl]acetamide
Show/Hide
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C25H33ClN4O5S
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1
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| 1 |
Ki = 834 nM
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CP0519720
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6-[5-[4-(4-chlorophenyl)piperazin-1-yl]pentyl]-2,4,7-trimethylpurino[7,8-a]imidazole-1,3-dione
Show/Hide
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C25H32ClN7O2
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1
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| 1 |
Ki = 837 nM
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CP0543754
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1-[(3-chlorophenyl)methyl]-N-(oxolan-3-ylmethyl)pyrrolo[3,2-c]quinolin-4-amine
Show/Hide
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C23H22ClN3O
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1
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| 1 |
Ki = 838 nM
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CP0113424
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9-[5-[4-(4-chlorophenyl)piperazin-1-yl]pentyl]-1,3-dimethylpurino[7,8-a]pyrimidine-2,4,8-trione
Show/Hide
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C25H30ClN7O3
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1
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| 1 |
Ki = 839 nM
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CP0445710
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N-[(1R)-1-(4-cyanophenyl)ethyl]-6-[4-[2-(4-methoxyphenyl)phenyl]piperazin-1-yl]hexanamide
Show/Hide
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C32H38N4O2
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1
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| 1 |
Ki = 843 nM
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CP0683995
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(5Z)-5-((5-bromo-1H-indol-3-yl)methylene)-2-(methylimino)imidazolidin-4-one
Show/Hide
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C13H11BrN4O
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1
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| 1 |
Ki = 860 nM
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CP0381350
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N-[1-(2-phenoxyethyl)piperidin-4-yl]thiophene-2-sulfonamide
Show/Hide
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C17H22N2O3S2
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1
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| 1 |
Ki = 862 nM
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CP0466796
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1-(benzenesulfonyl)-2-methoxybenzene
Show/Hide
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C13H12O3S
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1
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| 1 |
Ki = 866 nM
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CP0508302
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5-Methyl-3-(phenylsulfonyl)-2-piperazin-1-yl-7,8-dihydro-6Hcyclopenta[e]pyrazolo[1,5-a]pyrimidine
Show/Hide
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C20H23N5O2S
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1
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| 1 |
Ki = 869 nM
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CP0490399
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5,7-dichloro-3-(4-chlorophenyl)-3-methylquinoline-2,4(1H,3H)-dione
Show/Hide
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C16H10Cl3NO2
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1
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| 1 |
Ki = 877 nM
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CP0535836
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(R)-5,7-dichloro-3-(4-methoxyphenyl)-3-methylquinoline-2,4(1H,3H)-dione
Show/Hide
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C17H13Cl2NO3
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1
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| 1 |
Ki = 893 nM
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CP0434356
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6-chloro-N-[3-[4-(2,3-dichlorophenyl)piperazin-1-yl]propyl]quinoline-3-sulfonamide
Show/Hide
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C22H23Cl3N4O2S
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1
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| 1 |
Ki = 901 nM
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CP0431613
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4-[(4-chloro-2-methylphenoxy)methyl]-6-(4-methylpiperazin-1-yl)-1,3,5-triazin-2-amine
Show/Hide
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C16H21ClN6O
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1
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| 1 |
Ki = 911 nM
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CP0417077
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1-[6-[4-(2,3-dichlorophenyl)piperazin-1-yl]hexyl]benzo[cd]indol-2-one;hydrochloride
Show/Hide
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C27H30Cl3N3O
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1
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| 1 |
Ki = 918 nM
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CP0459145
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2-[6-[4-(3-methoxyphenyl)piperazin-1-yl]hexyl]-1,1-dioxo-1,2-benzothiazol-3-one
Show/Hide
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C24H31N3O4S
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1
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| 1 |
Ki = 921 nM
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CP0376748
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6-[4-[2-(4-cyanophenyl)-4-fluorophenyl]piperazin-1-yl]-N-[(4-cyanophenyl)methyl]hexanamide
Show/Hide
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C31H32FN5O
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1
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| 1 |
Ki = 927 nM
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CP0471365
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N-benzyl-5-(4-methylpiperazin-1-yl)-2-phenylmethoxyaniline
Show/Hide
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C25H29N3O
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1
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| 1 |
Ki = 928 nM
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CP0417076
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3-[6-[4-[4-(trifluoromethyl)phenyl]piperazin-1-yl]hexyl]-2lambda6-thia-3-azatricyclo[6.3.1.04,12]dodeca-1(11),4,6,8(12),9-pentaene 2,2-dioxide;hydrochloride
Show/Hide
|
C27H31ClF3N3O2S
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1
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| 1 |
Ki = 937 nM
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CP0396615
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3-[4-[2-[(2R)-1-quinolin-5-ylsulfonylpiperidin-2-yl]ethyl]piperazin-1-yl]-1,2-benzothiazole
Show/Hide
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C27H31N5O2S2
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1
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| 1 |
Ki = 949 nM
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CP0484847
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3,4-difluoro-N-[1-[2-(3-fluorophenoxy)ethyl]pyrrolidin-3-yl]benzenesulfonamide
Show/Hide
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C18H19F3N2O3S
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1
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| 1 |
Ki = 951 nM
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CP0454146
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5,7-dichloro-3-(4-iodophenyl)-3-methylquinoline-2,4(1H,3H)-dione
Show/Hide
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C16H10Cl2INO2
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1
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| 1 |
Ki = 952 nM
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CP0417066
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1-[6-[4-(2-nitrophenyl)piperazin-1-yl]hexyl]benzo[cd]indol-2-one
Show/Hide
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C27H30N4O3
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1
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| 1 |
Ki = 952 nM
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CP0462945
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5-chloro-N-[1-(2-phenoxyethyl)pyrrolidin-3-yl]thiophene-2-sulfonamide
Show/Hide
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C16H19ClN2O3S2
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1
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| 1 |
Ki = 957 nM
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CP0311502
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1,1-dioxo-2-[6-(4-phenylpiperazin-1-yl)hexyl]-1,2-benzothiazol-3-one
Show/Hide
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C23H29N3O3S
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1
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| 1 |
Ki = 971 nM
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CP0502595
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4-(4,6-dinitro-1H-indol-1-ylsulfonyl)benzenamine
Show/Hide
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C14H10N4O6S
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1
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| 1 |
Ki = 980 nM
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CP0568369
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7-(1-benzylpyrrolo[3,2-c]quinolin-4-yl)-2-oxa-7-azaspiro[3.4]octane
Show/Hide
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C24H23N3O
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1
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| 1 |
Ki = 992 nM
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CP0408250
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5-[(2R)-2-[2-[4-(2,3-dihydro-1,4-benzodioxin-5-yl)piperazin-1-yl]ethyl]pyrrolidin-1-yl]sulfonylquinoline
Show/Hide
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C27H32N4O4S
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1
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| 1 |
Ki = 996 nM
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CP0384573
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1-[6-(4-quinolin-8-ylpiperazin-1-yl)hexyl]benzo[cd]indol-2-one
Show/Hide
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C30H32N4O
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1
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| 1 |
Ki = 999 nM
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CP0485091
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4-[3-(2,4-dichlorophenoxy)propyl]-6-(4-methylpiperazin-1-yl)-1,3,5-triazin-2-amine
Show/Hide
|
C17H22Cl2N6O
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1
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| 1 |
Ki = 999 nM
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CP0168317
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1-(4,4-bis(4-fluorophenyl)butyl)-4-(4-chloro-3-(trifluoromethyl)phenyl)piperidin-4-ol
Show/Hide
|
C28H27ClF5NO
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1
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| 1 |
Ki = 1000 nM
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CP0412880
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2-methoxy-5-(4-methylpiperazin-1-yl)-N-phenethylbenzenamine
Show/Hide
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C20H27N3O
|
1
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| 1 |
Ki = 1013 nM
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CP0475051
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4-[4-[2-[4-[3-(trifluoromethyl)phenyl]piperazin-1-yl]ethyl]piperidin-1-yl]sulfonylisoquinoline
Show/Hide
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C27H31F3N4O2S
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1
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| 1 |
Ki = 1016 nM
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CP0448726
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5-[4-[2-[4-(4-chlorophenyl)piperazin-1-yl]ethyl]piperidin-1-yl]sulfonylquinoline
Show/Hide
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C26H31ClN4O2S
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1
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| 1 |
Ki = 1020 nM
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CP0454693
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2-(2-methoxy-6,7,8,9-tetrahydropyrido[1,2-a]indol-10-yl)-N,N-dimethylethanamine
Show/Hide
|
C17H24N2O
|
1
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| 1 |
Ki = 1030 nM
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CP0423149
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4-(2-fluorophenyl)-2-[4-[3-(1H-indol-3-yl)piperidin-1-yl]butyl]-5,6,7,8-tetrahydropyrido[1,2-c]pyrimidine-1,3-dione
Show/Hide
|
C31H35FN4O2
|
1
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| 1 |
Ki = 1030 nM
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CP0459429
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4-(2-chlorophenyl)-2-[4-[3-(1H-indol-3-yl)piperidin-1-yl]butyl]-5,6,7,8-tetrahydropyrido[1,2-c]pyrimidine-1,3-dione
Show/Hide
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C31H35ClN4O2
|
1
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| 1 |
Ki = 1030 nM
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CP0564427
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N-[[5-(3-methoxyphenyl)furan-2-yl]methyl]-1-(1-methylindol-3-yl)propan-2-amine
Show/Hide
|
C24H26N2O2
|
1
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| 1 |
Ki = 1032 nM
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CP0470858
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3-[2-[4-(3-phenylpyridin-2-yl)piperazin-1-yl]ethoxy]-N-[[4-(trifluoromethyl)phenyl]methyl]propanamide
Show/Hide
|
C28H31F3N4O2
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1
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| 1 |
Ki = 1039 nM
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CP0003923
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(2-{4-[(1Z)-1,2-diphenylbut-1-en-1-yl]phenoxy}ethyl)dimethylamine
Show/Hide
|
C26H29NO
|
1
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| 1 |
Ki = 1041 nM
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CP0448742
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4-[4-[2-[4-(3,4-dichlorophenyl)piperazin-1-yl]ethyl]piperidin-1-yl]sulfonylisoquinoline
Show/Hide
|
C26H30Cl2N4O2S
|
1
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| 1 |
Ki = 1041 nM
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CP0551591
|
4-[3-(3,4-dichlorophenoxy)propyl]-6-(4-methylpiperazin-1-yl)-1,3,5-triazin-2-amine
Show/Hide
|
C17H22Cl2N6O
|
1
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| 1 |
Ki = 1061 nM
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CP0377050
|
3-[2-[4-[3-(4-fluorophenyl)pyridin-2-yl]piperazin-1-yl]ethoxy]-N-[[4-(trifluoromethyl)phenyl]methyl]propanamide
Show/Hide
|
C28H30F4N4O2
|
1
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| 1 |
Ki = 1074 nM
|
|
|
|
CP0476619
|
N-[4-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)butyl]quinoline-3-sulfonamide
Show/Hide
|
C20H23N3O2S2
|
1
|
| 1 |
Ki = 1082 nM
|
|
|
|
CP0008601
|
4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1-(4-fluoro-phenyl)-butan-1-one;propionate(HCl)
Show/Hide
|
C21H23ClFNO2
|
1
|
| 1 |
Ki = 1083 nM
|
|
|
|
CP0395877
|
N-[3-[4-(1,2-benzoxazol-3-yl)piperazin-1-yl]propyl]-3,4-dichlorobenzenesulfonamide
Show/Hide
|
C20H22Cl2N4O3S
|
1
|
| 1 |
Ki = 1100 nM
|
|
|
|
CP0443099
|
N-[4-[4-(1,2-benzoxazol-3-yl)piperazin-1-yl]butyl]-1-benzothiophene-2-sulfonamide
Show/Hide
|
C23H26N4O3S2
|
1
|
| 1 |
Ki = 1100 nM
|
|
|
|
CP0527898
|
N-[6-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]hexyl]-N-[3-(trifluoromethyl)phenyl]benzenesulfonamide
Show/Hide
|
C30H33F3N4O2S2
|
1
|
| 1 |
Ki = 1103 nM
|
|
|
|
CP0039958
|
(risperidone)3-{2-[4-(6-Fluoro-benzo[d]isoxazol-3-yl)-piperidin-1-yl]-ethyl}-2-methyl-6,7,8,9-tetrahydro-pyrido[1,2-a]pyrimidin-4-one
Show/Hide
|
C23H27FN4O2
|
1
|
| 1 |
Ki = 1107 nM
|
|
|
|
CP0417075
|
1-[6-[4-[2-(trifluoromethyl)phenyl]piperazin-1-yl]hexyl]benzo[cd]indol-2-one;hydrochloride
Show/Hide
|
C28H31ClF3N3O
|
1
|
| 1 |
Ki = 1128 nM
|
|
|
|
CP0412404
|
1'-[2-[4-(3,4-dichlorophenyl)piperazin-1-yl]ethyl]spiro[1H-indole-3,3'-pyrrolidine]-2-one
Show/Hide
|
C23H26Cl2N4O
|
1
|
| 1 |
Ki = 1131 nM
|
|
|
|
CP0545006
|
3-[6-[4-(3-chlorophenyl)piperazin-1-yl]hexyl]-1,3-diazatricyclo[6.3.1.04,12]dodeca-4,6,8(12)-trien-2-one
Show/Hide
|
C26H33ClN4O
|
1
|
| 1 |
Ki = 1139 nM
|
|
|
|
CP0530032
|
(1S,2R,6S,7R)-4-[6-[4-(3-chlorophenyl)piperazin-1-yl]hexyl]-4-azatricyclo[5.2.1.02,6]decane-3,5-dione
Show/Hide
|
C25H34ClN3O2
|
1
|
| 1 |
Ki = 1142 nM
|
|
|
|
CP0423146
|
2-[4-[3-(1H-indol-3-yl)piperidin-1-yl]butyl]-4-phenyl-5,6,7,8-tetrahydropyrido[1,2-c]pyrimidine-1,3-dione
Show/Hide
|
C31H36N4O2
|
1
|
| 1 |
Ki = 1146 nM
|
|
|
|
CP0376749
|
N-[[4-(3-morpholin-4-ylpropoxy)phenyl]methyl]-6-[4-(2-phenylphenyl)piperazin-1-yl]hexanamide
Show/Hide
|
C36H48N4O3
|
1
|
| 1 |
Ki = 1152 nM
|
|
|
|
CP0513899
|
4-(4-fluorophenyl)sulfonyl-11-methyl-5-methylsulfanyl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1,3,5,8-tetraene
Show/Hide
|
C17H17FN4O2S2
|
1
|
| 1 |
Ki = 1155 nM
|
|
|
|
CP0545010
|
2-[[4-[[4-(3-chlorophenyl)piperazin-1-yl]methyl]phenyl]methyl]-[1,2,4]triazolo[4,3-a]pyridin-3-one
Show/Hide
|
C24H24ClN5O
|
1
|
| 1 |
Ki = 1160 nM
|
|
|
|
CP0400005
|
5-chloro-2-(3,4-dihydro-1H-isoquinolin-2-yl)-4-(4-methylphenyl)sulfonyl-1,3-thiazole
Show/Hide
|
C19H17ClN2O2S2
|
1
|
| 1 |
Ki = 1174 nM
|
|
|
|
CP0568664
|
4-N-[2-(1H-indol-3-yl)ethyl]-2-N-[2-(2-methoxyphenoxy)ethyl]-1,3,5-triazine-2,4,6-triamine
Show/Hide
|
C22H25N7O2
|
1
|
| 1 |
Ki = 1183 nM
|
|
|
|
CP0448727
|
4-[4-[2-[4-(3-chlorophenyl)piperazin-1-yl]ethyl]piperidin-1-yl]sulfonylisoquinoline
Show/Hide
|
C26H31ClN4O2S
|
1
|
| 1 |
Ki = 1185 nM
|
|
|
|
CP0053492
|
8-[4,4-bis(4-fluorophenyl)butyl]-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one
Show/Hide
|
C29H31F2N3O
|
1
|
| 1 |
Ki = 1188 nM
|
|
|
|
CP0475928
|
7-[5-[4-(3-chlorophenyl)piperazin-1-yl]pentyl]-1,3-dimethylpurine-2,6-dione;hydrochloride
Show/Hide
|
C22H29ClN6O2
|
1
|
| 1 |
Ki = 1195 nM
|
|
|
|
CP0236186
|
2-(5-(4-methylpiperazin-1-yl)-2-nitrophenyl)-4-phenylphthalazin-1(2H)-one
Show/Hide
|
C25H23N5O3
|
1
|
| 1 |
Ki = 1221 nM
|
|
|
|
CP0576382
|
1-[1-[(3-chlorophenyl)methyl]pyrrolo[3,2-c]quinolin-4-yl]piperidin-3-ol
Show/Hide
|
C23H22ClN3O
|
1
|
| 1 |
Ki = 1227 nM
|
|
|
|
CP0466616
|
3-[2-(3-chlorophenyl)ethyl]-7-piperazin-1-ylimidazo[4,5-b]pyridine
Show/Hide
|
C18H20ClN5
|
1
|
| 1 |
Ki = 1251 nM
|
|
|
|
CP0487358
|
3-[4-[2-[(2R)-1-quinolin-4-ylsulfonylpiperidin-2-yl]ethyl]piperazin-1-yl]-1,2-benzothiazole
Show/Hide
|
C27H31N5O2S2
|
1
|
| 1 |
Ki = 1259 nM
|
|
|
|
CP0416052
|
4-[(2R)-2-[2-[4-(2,3-dihydro-1,4-benzodioxin-5-yl)piperazin-1-yl]ethyl]pyrrolidin-1-yl]sulfonylisoquinoline
Show/Hide
|
C27H32N4O4S
|
1
|
| 1 |
Ki = 1263 nM
|
|
|
|
CP0528079
|
5-(4-methylpiperazin-1-yl)-2-nitro-N-(pyridin-3-ylmethyl)benzenamine
Show/Hide
|
C17H21N5O2
|
1
|
| 1 |
Ki = 1267 nM
|
|
|
|
CP0469370
|
1,1-dioxo-2-[6-[4-[2-(trifluoromethyl)phenyl]piperazin-1-yl]hexyl]-1,2-benzothiazol-3-one
Show/Hide
|
C24H28F3N3O3S
|
1
|
| 1 |
Ki = 1272 nM
|
|
|
|
CP0424758
|
2-(benzyloxy)-5-(4-methylpiperazin-1-yl)-N-phenethylbenzenamine
Show/Hide
|
C26H31N3O
|
1
|
| 1 |
Ki = 1284 nM
|
|
|
|
CP0568969
|
3-[2-(3-fluorophenyl)ethyl]-7-piperazin-1-ylimidazo[4,5-b]pyridine
Show/Hide
|
C18H20FN5
|
1
|
| 1 |
Ki = 1298 nM
|
|
|
|
CP0423148
|
4-(4-chlorophenyl)-2-[4-[3-(1H-indol-3-yl)piperidin-1-yl]butyl]-5,6,7,8-tetrahydropyrido[1,2-c]pyrimidine-1,3-dione
Show/Hide
|
C31H35ClN4O2
|
1
|
| 1 |
Ki = 1320 nM
|
|
|
|
CP0418452
|
N-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butyl]quinoline-3-sulfonamide
Show/Hide
|
C23H26Cl2N4O2S
|
1
|
| 1 |
Ki = 1331 nM
|
|
|
|
CP0426091
|
N-[1-[2-(2-phenylphenoxy)ethyl]pyrrolidin-3-yl]quinoline-2-carboxamide
Show/Hide
|
C28H27N3O2
|
1
|
| 1 |
Ki = 1335 nM
|
|
|
|
CP0376750
|
N-[[4-(2-hydroxyethoxy)phenyl]methyl]-6-[4-[2-(4-methoxyphenyl)phenyl]piperazin-1-yl]hexanamide
Show/Hide
|
C32H41N3O4
|
1
|
| 1 |
Ki = 1336 nM
|
|
|
|
CP0568394
|
1-[1-[(3-methoxyphenyl)methyl]pyrrolo[3,2-c]quinolin-4-yl]piperidin-4-ol
Show/Hide
|
C24H25N3O2
|
1
|
| 1 |
Ki = 1338 nM
|
|
|
|
CP0440391
|
5-bromo-3-(3-ethylimidazol-4-yl)-1H-indole
Show/Hide
|
C13H12BrN3
|
1
|
| 1 |
Ki = 1349 nM
|
|
|
|
CP0543362
|
1,1-dioxo-2-[5-[4-[3-(trifluoromethyl)phenyl]piperazin-1-yl]pentyl]-1,2-benzothiazol-3-one
Show/Hide
|
C23H26F3N3O3S
|
1
|
| 1 |
Ki = 1354 nM
|
|
|
|
CP0577335
|
7-[1-[(3-chlorophenyl)methyl]pyrrolo[3,2-c]quinolin-4-yl]-2-oxa-7-azaspiro[3.4]octane
Show/Hide
|
C24H22ClN3O
|
1
|
| 1 |
Ki = 1362 nM
|
|
|
|
CP0528082
|
2-(furan-2-ylmethylamino)-4-(4-methylpiperazin-1-yl)benzonitrile
Show/Hide
|
C17H20N4O
|
1
|
| 1 |
Ki = 1365 nM
|
|
|
|
CP0499149
|
5,7-Dimethyl-3-(phenylsulfonyl)-2-piperazin-1-ylpyrazolo[1,5-a]pyrimidine
Show/Hide
|
C18H21N5O2S
|
1
|
| 1 |
Ki = 1380 nM
|
|
|
|
CP0530508
|
3-(3-ethylimidazol-4-yl)-5-(trifluoromethyl)-1H-indole
Show/Hide
|
C14H12F3N3
|
1
|
| 1 |
Ki = 1380 nM
|
|
|
|
CP0387337
|
N-[1-(4-chlorophenyl)ethyl]-3-(furan-2-yl)-4-phenylbutan-1-amine
Show/Hide
|
C22H24ClNO
|
1
|
| 1 |
Ki = 1400 nM
|
|
|
|
CP0202831
|
4-[4-chloro-3-(trifluoromethyl)phenyl]-1-[4-(4-methoxy-N-(4-methoxyphenyl)anilino)butyl]piperidin-4-ol
Show/Hide
|
C30H34ClF3N2O3
|
1
|
| 1 |
Ki = 1400 nM
|
|
|
|
CP0848620
|
(E)-5-((7-bromo-1H-indol-3-yl)methylene)-2-iminoimidazolidin-4-one
Show/Hide
|
C12H9BrN4O
|
1
|
| 1 |
Ki = 1405 nM
|
|
|
|
CP0237317
|
CHEMBL2058415
Show/Hide
|
C14H13BrN4O
|
1
|
| 1 |
Ki = 1409 nM
|
|
|
|
CP0495705
|
2-[6-[4-(2-nitrophenyl)piperazin-1-yl]hexyl]benzo[de]isoquinoline-1,3-dione
Show/Hide
|
C28H30N4O4
|
1
|
| 1 |
Ki = 1410 nM
|
|
|
|
CP0282006
|
6-[4-[4-(4-chlorophenyl)piperazin-1-yl]butyl]-2,4,7-trimethylpurino[7,8-a]imidazole-1,3-dione
Show/Hide
|
C24H30ClN7O2
|
1
|
| 1 |
Ki = 1456 nM
|
|
|
|
CP0417573
|
5-[4-[2-[4-(4-fluorophenyl)piperazin-1-yl]ethyl]piperidin-1-yl]sulfonylquinoline
Show/Hide
|
C26H31FN4O2S
|
1
|
| 1 |
Ki = 1459 nM
|
|
|
|
CP0384570
|
1-[6-(4-pyridin-2-ylpiperazin-1-yl)hexyl]benzo[cd]indol-2-one
Show/Hide
|
C26H30N4O
|
1
|
| 1 |
Ki = 1461 nM
|
|
|
|
CP0421346
|
[4-[5-[[2-(1H-indol-3-yl)ethylamino]methyl]furan-2-yl]phenyl] acetate
Show/Hide
|
C23H22N2O3
|
1
|
| 1 |
Ki = 1463 nM
|
|
|
|
CP0396073
|
4-[(2S)-2-[2-[4-(2,3-dihydro-1,4-benzodioxin-5-yl)piperazin-1-yl]ethyl]pyrrolidin-1-yl]sulfonylisoquinoline
Show/Hide
|
C27H32N4O4S
|
1
|
| 1 |
Ki = 1483 nM
|
|
|
|
CP0471366
|
1-N-(2-aminoethyl)-3-N-benzyl-4-nitrobenzene-1,3-diamine
Show/Hide
|
C15H18N4O2
|
1
|
| 1 |
Ki = 1490 nM
|
|
|
|
CP0510210
|
N-[3-[4-(1,2-benzoxazol-3-yl)piperazin-1-yl]propyl]-3-methylbenzenesulfonamide
Show/Hide
|
C21H26N4O3S
|
1
|
| 1 |
Ki = 1500 nM
|
|
|
|
CP0525861
|
N-[1-(cyclopropylmethoxy)-2-methoxy-6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-10-yl]acetamide
Show/Hide
|
C24H28N2O3
|
1
|
| 1 |
Ki = 1500 nM
|
|
|
|
CP0530888
|
N-[[4-[(dimethylamino)methyl]phenyl]methyl]-6-[4-(2-phenylphenyl)piperazin-1-yl]hexanamide
Show/Hide
|
C32H42N4O
|
1
|
| 1 |
Ki = 1506 nM
|
|
|
|
CP0335494
|
2-nitro-5-(piperazin-1-yl)-N-(pyridin-3-ylmethyl)benzenamine
Show/Hide
|
C16H19N5O2
|
1
|
| 1 |
Ki = 1512 nM
|
|
|
|
CP0395154
|
N-[4-(3,4-dihydro-1H-isoquinolin-2-yl)butyl]quinoline-6-sulfonamide
Show/Hide
|
C22H25N3O2S
|
1
|
| 1 |
Ki = 1518 nM
|
|
|
|
CP0576365
|
1-(3-chlorophenyl)-4-[6-(sulfamoylamino)hexyl]piperazine
Show/Hide
|
C16H27ClN4O2S
|
1
|
| 1 |
Ki = 1531 nM
|
|
|
|
CP0934499
|
N-{4-[4-(4-Chlorophenyl)-piperazin-1-yl]-butyl}-6-quinolinesulfonamide hydrochloride
Show/Hide
|
C23H28Cl2N4O2S
|
1
|
| 1 |
Ki = 1535 nM
|
|
|
|
CP0379116
|
3-(benzenesulfonyl)-6-chloro-N-(4-methylphenyl)quinolin-4-amine
Show/Hide
|
C22H17ClN2O2S
|
1
|
| 1 |
Ki = 1574 nM
|
|
|
|
CP0133391
|
N,N,6-trimethyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-10-amine
Show/Hide
|
C19H22N2
|
1
|
| 1 |
Ki = 1588 nM
|
|
|
|
CP0441366
|
6-[5-[4-(4-chlorophenyl)piperazin-1-yl]pentyl]-2,4-dimethylpurino[7,8-a]imidazole-1,3-dione
Show/Hide
|
C24H30ClN7O2
|
1
|
| 1 |
Ki = 1591 nM
|
|
|
|
CP0156548
|
(PHENYLSULFONYL)BENZENE
Show/Hide
|
C12H10O2S
|
1
|
| 1 |
Ki = 1598 nM
|
|
|
|
CP0548414
|
N-[3-[4-(1,2-benzoxazol-3-yl)piperazin-1-yl]propyl]naphthalene-2-sulfonamide
Show/Hide
|
C24H26N4O3S
|
1
|
| 1 |
Ki = 1600 nM
|
|
|
|
CP0432718
|
2-[6-[4-(2-fluorophenyl)piperazin-1-yl]hexyl]-1,1-dioxo-1,2-benzothiazol-3-one
Show/Hide
|
C23H28FN3O3S
|
1
|
| 1 |
Ki = 1619 nM
|
|
|
|
CP0376744
|
N-[(4-cyanophenyl)methyl]-3-[2-[4-[3-(4-fluorophenyl)pyridin-2-yl]piperazin-1-yl]ethoxy]propanamide
Show/Hide
|
C28H30FN5O2
|
1
|
| 1 |
Ki = 1621 nM
|
|
|
|
CP0528510
|
5-chloro-3-(3-ethylimidazol-4-yl)-4-fluoro-1H-indole
Show/Hide
|
C13H11ClFN3
|
1
|
| 1 |
Ki = 1622 nM
|
|
|
|
CP0445705
|
6-[4-[2-(4-methoxyphenyl)phenyl]piperazin-1-yl]-N-[[4-(3-morpholin-4-ylpropoxy)phenyl]methyl]hexanamide
Show/Hide
|
C37H50N4O4
|
1
|
| 1 |
Ki = 1623 nM
|
|
|
|
CP0376747
|
N-[(4-cyanophenyl)methyl]-3-[2-[4-(3-phenylpyridin-2-yl)piperazin-1-yl]ethoxy]propanamide
Show/Hide
|
C28H31N5O2
|
1
|
| 1 |
Ki = 1633 nM
|
|
|
|
CP0525902
|
(1S,2R,6S,7R)-4-[6-[4-(2-chlorophenyl)piperazin-1-yl]hexyl]-4-azatricyclo[5.2.1.02,6]decane-3,5-dione
Show/Hide
|
C25H34ClN3O2
|
1
|
| 1 |
Ki = 1641 nM
|
|
|
|
CP0384283
|
4-(4-fluorophenyl)-2-[4-[3-(1H-indol-3-yl)piperidin-1-yl]butyl]-5,6,7,8-tetrahydropyrido[1,2-c]pyrimidine-1,3-dione
Show/Hide
|
C31H35FN4O2
|
1
|
| 1 |
Ki = 1651 nM
|
|
|
|
CP0413064
|
3-(3-ethylimidazol-4-yl)-5-iodo-1H-indole
Show/Hide
|
C13H12IN3
|
2
|
| 1 |
Ki = 1660 nM
|
|
|
| 2 |
Ki = 1673 nM
|
|
|
|
CP0314578
|
4-[4-chloro-3-(trifluoromethyl)phenyl]-1-[4-(4-fluoro-N-(4-fluorophenyl)anilino)butyl]piperidin-4-ol
Show/Hide
|
C28H28ClF5N2O
|
1
|
| 1 |
Ki = 1670 nM
|
|
|
|
CP0198450
|
1-[5,5-bis(4-fluorophenyl)pentyl]-4-[4-chloro-3-(trifluoromethyl)phenyl]piperidin-4-ol
Show/Hide
|
C29H29ClF5NO
|
1
|
| 1 |
Ki = 1671 nM
|
|
|
|
CP0069223
|
4-[4-chloro-3-(trifluoromethyl)phenyl]-1-[3-(4-fluoro-N-(4-fluorophenyl)anilino)propyl]piperidin-4-ol
Show/Hide
|
C27H26ClF5N2O
|
1
|
| 1 |
Ki = 1680 nM
|
|
|
|
CP0416669
|
1-[6-[4-(2-chlorophenyl)piperazin-1-yl]hexyl]benzo[cd]indol-2-one;hydrochloride
Show/Hide
|
C27H31Cl2N3O
|
1
|
| 1 |
Ki = 1681 nM
|
|
|
|
CP0456106
|
1'-[2-[4-(4-chlorophenoxy)piperidin-1-yl]ethyl]spiro[1H-indole-3,3'-pyrrolidine]-2-one
Show/Hide
|
C24H28ClN3O2
|
1
|
| 1 |
Ki = 1693 nM
|
|
|
|
CP0545009
|
3-[6-[4-(3-chlorophenyl)piperazin-1-yl]hexyl]-2lambda6-thia-1,3-diazatricyclo[6.3.1.04,12]dodeca-4,6,8(12)-triene 2,2-dioxide
Show/Hide
|
C25H33ClN4O2S
|
1
|
| 1 |
Ki = 1694 nM
|
|
|
|
CP0082560
|
4-[4-chloro-3-(trifluoromethyl)phenyl]-1-(4,4-diphenylbutyl)piperidin-4-ol
Show/Hide
|
C28H29ClF3NO
|
1
|
| 1 |
Ki = 1695 nM
|
|
|
|
CP0562346
|
4-[5-[[2-(5-methoxy-1-benzofuran-3-yl)ethylamino]methyl]furan-2-yl]phenol
Show/Hide
|
C22H21NO4
|
1
|
| 1 |
Ki = 1696 nM
|
|
|
|
CP0417069
|
1-[6-[4-(3-methoxyphenyl)piperazin-1-yl]hexyl]benzo[cd]indol-2-one
Show/Hide
|
C28H33N3O2
|
1
|
| 1 |
Ki = 1699 nM
|
|
|
|
CP0476102
|
6-[4-[2-(4-methoxyphenyl)phenyl]piperazin-1-yl]-N-[[4-(2-morpholin-4-ylethoxy)phenyl]methyl]hexanamide
Show/Hide
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C36H48N4O4
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1
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| 1 |
Ki = 1706 nM
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CP0542758
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2-N-[2-(1H-indol-3-yl)ethyl]-4-N-[4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]-1,3,5-triazine-2,4,6-triamine
Show/Hide
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C28H37N9O
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1
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| 1 |
Ki = 1706 nM
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CP0530347
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2-[4-[3-(1H-indol-3-yl)piperidin-1-yl]butyl]-4-(4-methoxyphenyl)pyrido[1,2-c]pyrimidine-1,3-dione
Show/Hide
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C32H34N4O3
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1
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| 1 |
Ki = 1709 nM
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CP0580239
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1-[1-[(3-chlorophenyl)methyl]pyrrolo[3,2-c]quinolin-4-yl]piperidin-4-ol
Show/Hide
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C23H22ClN3O
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1
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| 1 |
Ki = 1713 nM
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CP0124959
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METHYLAPLYSINOPSIN
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C15H16N4O
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1
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| 1 |
Ki = 1716 nM
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CP0462115
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1,1-dioxo-2-[6-(4-quinolin-8-ylpiperazin-1-yl)hexyl]-1,2-benzothiazol-3-one
Show/Hide
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C26H30N4O3S
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1
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| 1 |
Ki = 1716 nM
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CP0377049
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N-[[4-(2-morpholin-4-ylethoxy)phenyl]methyl]-6-[4-(2-phenylphenyl)piperazin-1-yl]hexanamide
Show/Hide
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C35H46N4O3
|
1
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| 1 |
Ki = 1724 nM
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CP0944094
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N-{4-[4-(4-Chlorophenyl)-piperazin-1-yl]-butyl}-7-quinolinesulfonamide hydrochloride
Show/Hide
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C23H28Cl2N4O2S
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1
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| 1 |
Ki = 1725 nM
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CP0384691
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1-[6-[4-(2-fluorophenyl)piperazin-1-yl]hexyl]benzo[cd]indol-2-one;hydrochloride
Show/Hide
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C27H31ClFN3O
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1
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| 1 |
Ki = 1726 nM
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CP0577334
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1-[(3-chlorophenyl)methyl]-N-[(3S)-oxolan-3-yl]pyrrolo[3,2-c]quinolin-4-amine
Show/Hide
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C22H20ClN3O
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1
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| 1 |
Ki = 1742 nM
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CP0508202
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N-[1-[2-(2-propan-2-ylphenoxy)ethyl]pyrrolidin-3-yl]quinoline-2-carboxamide
Show/Hide
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C25H29N3O2
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1
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| 1 |
Ki = 1761 nM
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CP0510465
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3-[(4-fluorophenyl)methyl]-1-[5-[4-(4-fluorophenyl)piperazin-1-yl]pentyl]-5,5-dimethylimidazolidine-2,4-dione;hydrochloride
Show/Hide
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C27H34F2N4O2
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1
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| 1 |
Ki = 1762 nM
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CP0533329
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5-Methyl-3-(phenylsulfonyl)-2-piperazin-1-yl-6,7,8,9-tetrahydropyrazolo[1,5-a]quinazoline
Show/Hide
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C21H25N5O2S
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1
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| 1 |
Ki = 1764 nM
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CP0453915
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N-[1-[2-(3-fluorophenoxy)ethyl]pyrrolidin-3-yl]thiophene-2-sulfonamide
Show/Hide
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C16H19FN2O3S2
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1
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| 1 |
Ki = 1779 nM
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CP0544198
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6-[4-(2,3-dichlorophenyl)piperazin-1-yl]-2-N-[2-(1H-indol-3-yl)ethyl]-1,3,5-triazine-2,4-diamine
Show/Hide
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C23H24Cl2N8
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1
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| 1 |
Ki = 1781 nM
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CP0381349
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2,3-difluoro-N-[1-[2-(2-phenylphenoxy)ethyl]pyrrolidin-3-yl]benzamide
Show/Hide
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C25H24F2N2O2
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1
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| 1 |
Ki = 1799 nM
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CP0552435
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3-(4-fluorophenyl)-3-(furan-2-yl)-N-[1-(4-methylphenyl)ethyl]propan-1-amine
Show/Hide
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C22H24FNO
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1
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| 1 |
Ki = 1800 nM
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CP0390940
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4-[4-[2-[(2R)-1-isoquinolin-4-ylsulfonylpyrrolidin-2-yl]ethyl]piperazin-1-yl]-3H-1,3-benzoxazol-2-one
Show/Hide
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C26H29N5O4S
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1
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| 1 |
Ki = 1810 nM
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CP0571734
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4-(4-methylpiperazin-1-yl)-6-(pyridin-4-ylmethyl)-1,3,5-triazin-2-amine
Show/Hide
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C14H19N7
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1
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| 1 |
Ki = 1828 nM
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CP0558696
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1,1-dioxo-2-[5-(4-phenylpiperazin-1-yl)pentyl]-1,2-benzothiazol-3-one
Show/Hide
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C22H27N3O3S
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1
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| 1 |
Ki = 1836 nM
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CP0390184
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1-(5-naphthalen-1-yloxypentyl)azepane
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C21H29NO
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1
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| 1 |
Ki = 1837 nM
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CP0416667
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1-[6-[4-(3,4-dichlorophenyl)piperazin-1-yl]hexyl]benzo[cd]indol-2-one;hydrochloride
Show/Hide
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C27H30Cl3N3O
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1
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| 1 |
Ki = 1860 nM
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CP0448725
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4-[4-[2-[4-(4-fluorophenyl)piperazin-1-yl]ethyl]piperidin-1-yl]sulfonylisoquinoline
Show/Hide
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C26H31FN4O2S
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1
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| 1 |
Ki = 1863 nM
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CP0371743
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methyl 2-(benzylamino)-5-(4-methylpiperazin-1-yl)benzoate
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C20H25N3O2
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1
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| 1 |
Ki = 1888 nM
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CP0412481
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3-benzyl-2-phenyl-5-(pyridin-2-ylamino)-5-(trifluoromethyl)imidazol-4-one
Show/Hide
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C22H17F3N4O
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1
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| 1 |
Ki = 1900 nM
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CP0543164
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7-[4-[4-(3,4-dichlorophenyl)piperazin-1-yl]butyl]-1,3-dimethylpurine-2,6-dione;hydrochloride
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C21H26Cl2N6O2
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1
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| 1 |
Ki = 1902 nM
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CP0417089
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1-[6-[4-(2-ethoxyphenyl)piperazin-1-yl]hexyl]benzo[cd]indol-2-one
Show/Hide
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C29H35N3O2
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1
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| 1 |
Ki = 1916 nM
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CP0390723
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N-ethyl-N-[3-[4-(2-methoxyphenyl)piperazin-1-yl]propyl]quinoline-6-sulfonamide
Show/Hide
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C25H32N4O3S
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1
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| 1 |
Ki = 1920 nM
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CP0489716
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3-benzyl-1-[5-[4-(4-fluorophenyl)piperazin-1-yl]pentyl]-5,5-dimethylimidazolidine-2,4-dione;hydrochloride
Show/Hide
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C27H35FN4O2
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1
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| 1 |
Ki = 1945 nM
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CP0387489
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N-[4-(3,4,4a,5,6,7,8,8a-octahydro-1H-isoquinolin-2-yl)butyl]-N-ethylquinoline-8-sulfonamide
Show/Hide
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C24H35N3O2S
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1
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| 1 |
Ki = 1950 nM
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CP0680890
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{2-[4-(2-Chloro-1,2-diphenyl-vinyl)-phenoxy]-ethyl}-diethyl-amine
Show/Hide
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C26H28ClNO
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1
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| 1 |
Ki = 1956 nM
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CP0541083
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2-[6-(4-pyridin-2-ylpiperazin-1-yl)hexyl]benzo[de]isoquinoline-1,3-dione
Show/Hide
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C27H30N4O2
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1
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| 1 |
Ki = 1966 nM
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CP0513026
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7-[4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]-1,3-dimethylpurine-2,6-dione;hydrochloride
Show/Hide
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C22H30N6O3
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1
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| 1 |
Ki = 1970 nM
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CP0540390
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2-[5-[4-(2-methoxyphenyl)piperazin-1-yl]pentyl]-1,1-dioxo-1,2-benzothiazol-3-one
Show/Hide
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C23H29N3O4S
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1
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| 1 |
Ki = 1991 nM
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CP0456103
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1'-[2-[4-(3-chlorophenyl)piperazin-1-yl]ethyl]spiro[1H-indole-3,3'-pyrrolidine]-2-one
Show/Hide
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C23H27ClN4O
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1
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| 1 |
Ki = 2005 nM
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CP0508642
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2-(benzenesulfonyl)-N,N-dimethylaniline
Show/Hide
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C14H15NO2S
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1
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| 1 |
Ki = 2039 nM
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CP0417078
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1-[6-[4-[4-(trifluoromethyl)phenyl]piperazin-1-yl]hexyl]benzo[cd]indol-2-one;hydrochloride
Show/Hide
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C28H31ClF3N3O
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1
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| 1 |
Ki = 2045 nM
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CP0487624
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4-[(2S)-2-[2-[4-(1H-indol-4-yl)piperazin-1-yl]ethyl]pyrrolidin-1-yl]sulfonylisoquinoline
Show/Hide
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C27H31N5O2S
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1
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| 1 |
Ki = 2057 nM
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CP0484861
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4-fluoro-N-[[1-[2-(3-fluorophenoxy)ethyl]piperidin-4-yl]methyl]benzenesulfonamide
Show/Hide
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C20H24F2N2O3S
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1
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| 1 |
Ki = 2124 nM
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CP0545011
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2-[[4-[[4-(4-chlorophenyl)piperazin-1-yl]methyl]phenyl]methyl]-[1,2,4]triazolo[4,3-a]pyridin-3-one
Show/Hide
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C24H24ClN5O
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1
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| 1 |
Ki = 2144 nM
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CP0461751
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N-[3-[4-(2-methoxyphenyl)piperazin-1-yl]propyl]quinoline-8-sulfonamide
Show/Hide
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C23H28N4O3S
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1
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| 1 |
Ki = 2159 nM
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CP0530449
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(2-{[5,7-Dimethyl-3-(phenylsulfonyl)pyrazolo[1,5-a]pyrimidin-2-yl]oxy}ethyl)dimethylamine
Show/Hide
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C18H22N4O3S
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1
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| 1 |
Ki = 2200 nM
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CP0497340
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N-[3-[4-(1,2-benzoxazol-3-yl)piperazin-1-yl]propyl]-4-(trifluoromethoxy)benzenesulfonamide
Show/Hide
|
C21H23F3N4O4S
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1
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| 1 |
Ki = 2200 nM
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CP0315737
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2-[4-(1H-imidazol-5-ylmethyl)-5-phenyl-4,5-dihydro-1,3-thiazol-2-yl]phenol
Show/Hide
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C19H17N3OS
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1
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| 1 |
Ki = 2200 nM
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CP0525901
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(1R,2S,6R,7S)-4-[6-[4-[3-(trifluoromethyl)phenyl]piperazin-1-yl]hexyl]-4-azatricyclo[5.2.1.02,6]decane-3,5-dione
Show/Hide
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C26H34F3N3O2
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1
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| 1 |
Ki = 2205 nM
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CP0880895
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N-{5-[4-(4-Chlorophenyl)-piperazin-1-yl]-pentyl}-3-quinolinesulfonamide hydrochloride
Show/Hide
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C24H30Cl2N4O2S
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1
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| 1 |
Ki = 2209 nM
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CP0384692
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1-[6-[4-[3-(trifluoromethyl)phenyl]piperazin-1-yl]hexyl]benzo[cd]indol-2-one;hydrochloride
Show/Hide
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C28H31ClF3N3O
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1
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| 1 |
Ki = 2214 nM
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CP0525594
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3-[2-[4-(2-phenylpyridin-3-yl)piperazin-1-yl]ethoxy]-N-[[4-(trifluoromethyl)phenyl]methyl]propanamide
Show/Hide
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C28H31F3N4O2
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1
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| 1 |
Ki = 2215 nM
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CP0550470
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6-[1-[(3-chlorophenyl)methyl]pyrrolo[3,2-c]quinolin-4-yl]-2-oxa-6-azaspiro[3.3]heptane
Show/Hide
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C23H20ClN3O
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1
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| 1 |
Ki = 2243 nM
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CP0497341
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N-[3-[4-(1,2-benzoxazol-3-yl)piperazin-1-yl]propyl]-6-chloronaphthalene-2-sulfonamide
Show/Hide
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C24H25ClN4O3S
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1
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| 1 |
Ki = 2300 nM
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CP0146890
|
CHEMBL2058418
Show/Hide
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C14H13BrN4O
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1
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| 1 |
Ki = 2306 nM
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CP0391293
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5-[(2S)-2-[2-[4-(1H-indol-4-yl)piperazin-1-yl]ethyl]pyrrolidin-1-yl]sulfonylquinoline
Show/Hide
|
C27H31N5O2S
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1
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| 1 |
Ki = 2310 nM
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CP0432567
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1,1-dioxo-2-[6-(4-pyridin-2-ylpiperazin-1-yl)hexyl]-1,2-benzothiazol-3-one
Show/Hide
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C22H28N4O3S
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1
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| 1 |
Ki = 2352 nM
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CP0853815
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3-(S)-1-Pyrrolidin-2-ylmethyl-1H-indole hydrochloride
Show/Hide
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C13H17ClN2
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1
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| 1 |
Ki = 2400 nM
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CP0534907
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3-(furan-2-yl)-3-(2-methoxyphenyl)-N-[(4-methoxyphenyl)methyl]propan-1-amine
Show/Hide
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C22H25NO3
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1
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| 1 |
Ki = 2400 nM
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CP0460397
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4-[4-[2-(4-phenylpiperazin-1-yl)ethyl]piperidin-1-yl]sulfonylisoquinoline
Show/Hide
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C26H32N4O2S
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1
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| 1 |
Ki = 2412 nM
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CP0421837
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3-(3-ethylimidazol-4-yl)-7-fluoro-5-iodo-1H-indole
Show/Hide
|
C13H11FIN3
|
1
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| 1 |
Ki = 2455 nM
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CP0387335
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N-[1-(4-chlorophenyl)ethyl]-3-(furan-2-yl)-3-(4-methylphenyl)propan-1-amine
Show/Hide
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C22H24ClNO
|
1
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| 1 |
Ki = 2500 nM
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CP0382641
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3-benzyl-1-[5-[4-(2-fluorophenyl)piperazin-1-yl]pentyl]-5,5-dimethylimidazolidine-2,4-dione;hydrochloride
Show/Hide
|
C27H36ClFN4O2
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1
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| 1 |
Ki = 2506 nM
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CP0382644
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3-[2-[4-(2-phenylphenyl)piperazin-1-yl]ethoxy]-N-(pyridin-4-ylmethyl)propanamide
Show/Hide
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C27H32N4O2
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1
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| 1 |
Ki = 2518 nM
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CP0498238
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4-(1H-Indol-3-ylmethyl)-phenylamine
Show/Hide
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C15H14N2
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1
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| 1 |
Ki = 2530 nM
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CP0396619
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5-[(2S)-2-[2-[4-(2,3-dihydro-1,4-benzodioxin-5-yl)piperazin-1-yl]ethyl]pyrrolidin-1-yl]sulfonylquinoline
Show/Hide
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C27H32N4O4S
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1
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| 1 |
Ki = 2533 nM
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CP0331699
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1-(5-naphthalen-1-yloxypentyl)piperidine
Show/Hide
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C20H27NO
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1
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| 1 |
Ki = 2539 nM
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CP0569187
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4-(3-chlorophenyl)-N-[6-(3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2-yl)hexyl]piperazine-1-carboxamide
Show/Hide
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C23H29ClN6O2
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1
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| 1 |
Ki = 2550 nM
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CP0466167
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N-[3-(benzenesulfonyl)-5,7-dimethylpyrazolo[1,5-a]pyrimidin-2-yl]-N',N'-dimethylethane-1,2-diamine
Show/Hide
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C18H23N5O2S
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1
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| 1 |
Ki = 2600 nM
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CP0487823
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2-{2-phenyl-1H-pyrrolo[3,2-c]pyridin-3-yl}ethan-1-amine, 20
Show/Hide
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C15H15N3
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1
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| 1 |
Ki = 2600 nM
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CP0444342
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2-[(4S,5S)-4-(1H-imidazol-5-ylmethyl)-5-methyl-4,5-dihydro-1,3-thiazol-2-yl]phenol
Show/Hide
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C14H15N3OS
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1
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| 1 |
Ki = 2600 nM
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CP0543385
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1,1-dioxo-2-[5-(4-pyridin-2-ylpiperazin-1-yl)pentyl]-1,2-benzothiazol-3-one
Show/Hide
|
C21H26N4O3S
|
1
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| 1 |
Ki = 2626 nM
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CP0376746
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3-[2-[4-[2-(4-fluorophenyl)pyridin-3-yl]piperazin-1-yl]ethoxy]-N-[[4-(trifluoromethyl)phenyl]methyl]propanamide
Show/Hide
|
C28H30F4N4O2
|
1
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| 1 |
Ki = 2634 nM
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CP0480533
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N-[4-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)butyl]quinoline-7-sulfonamide
Show/Hide
|
C20H23N3O2S2
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1
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| 1 |
Ki = 2652 nM
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CP0540392
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2-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butyl]-1,1-dioxo-1,2-benzothiazol-3-one
Show/Hide
|
C21H23Cl2N3O3S
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1
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| 1 |
Ki = 2662 nM
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CP0069240
|
4-(piperazin-1-yl)-1H-indole
Show/Hide
|
C12H15N3
|
1
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| 1 |
Ki = 2700 nM
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CP0548225
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2-(cyclohexen-1-yl)-N-[(3-methoxy-4-phenylmethoxyphenyl)methyl]ethanamine
Show/Hide
|
C23H29NO2
|
1
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| 1 |
Ki = 2700 nM
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CP0209146
|
4-(4-chlorophenyl)-6-(4-methylpiperazin-1-yl)-1,3,5-triazin-2-amine
Show/Hide
|
C14H17ClN6
|
1
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| 1 |
Ki = 2707 nM
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CP0860970
|
N-{3-[4-(4-Chlorophenyl)-piperazin-1-yl]-propyl}-4-isoquinolinesulfonamide hydrochloride
Show/Hide
|
C22H26Cl2N4O2S
|
1
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| 1 |
Ki = 2757 nM
|
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CP0481686
|
N-[[1-[2-(3-fluorophenoxy)ethyl]piperidin-4-yl]methyl]thiophene-2-sulfonamide
Show/Hide
|
C18H23FN2O3S2
|
1
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| 1 |
Ki = 2759 nM
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CP0542759
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4-N-[2-(1H-indol-3-yl)ethyl]-2-N-[2-(2-methoxyanilino)ethyl]-1,3,5-triazine-2,4,6-triamine
Show/Hide
|
C22H26N8O
|
1
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| 1 |
Ki = 2798 nM
|
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CP0376741
|
N-[(4-cyanophenyl)methyl]-3-[2-[4-[2-(4-fluorophenyl)pyridin-3-yl]piperazin-1-yl]ethoxy]propanamide
Show/Hide
|
C28H30FN5O2
|
1
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| 1 |
Ki = 2815 nM
|
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CP0528129
|
N-(3-aminophenyl)benzenesulfonamide
Show/Hide
|
C12H12N2O2S
|
1
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| 1 |
Ki = 2840 nM
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CP0569767
|
2-[6-[4-(2,3-dihydro-1,4-benzodioxin-5-yl)piperazin-1-yl]hexyl]-[1,2,4]triazolo[4,3-a]pyridin-3-one
Show/Hide
|
C24H31N5O3
|
1
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| 1 |
Ki = 2841 nM
|
|
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CP0456107
|
1'-[2-[4-(2-chlorophenyl)piperazin-1-yl]ethyl]spiro[1H-indole-3,3'-pyrrolidine]-2-one
Show/Hide
|
C23H27ClN4O
|
1
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| 1 |
Ki = 2843 nM
|
|
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CP0489717
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1-[5-[4-(4-chlorophenyl)piperazin-1-yl]pentyl]-3-[(2,4-dichlorophenyl)methyl]-5,5-dimethylimidazolidine-2,4-dione;hydrochloride
Show/Hide
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C27H33Cl3N4O2
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1
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| 1 |
Ki = 2879 nM
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CP0344919
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3-(3-ethylimidazol-4-yl)-4-fluoro-5-iodo-1H-indole
Show/Hide
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C13H11FIN3
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1
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| 1 |
Ki = 2884 nM
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CP0499307
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(2-{2-ethyl-1H-pyrrolo[3,2-c]pyridin-3-yl}ethyl)dimethylamine, 24
Show/Hide
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C13H19N3
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1
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| 1 |
Ki = 2900 nM
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CP0542764
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2-N-[2-(1H-indol-3-yl)ethyl]-6-[4-(2-methoxyphenyl)piperazin-1-yl]-1,3,5-triazine-2,4-diamine
Show/Hide
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C24H28N8O
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1
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| 1 |
Ki = 2907 nM
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CP0382801
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3-benzyl-1-[5-[4-(3-methoxyphenyl)piperazin-1-yl]pentyl]-5,5-dimethylimidazolidine-2,4-dione;hydrochloride
Show/Hide
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C28H38N4O3
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1
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| 1 |
Ki = 2926 nM
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CP0400395
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3-(4-chlorophenyl)sulfonyl-1-(2-methoxyethyl)-4,5-dimethylpyrrol-2-amine
Show/Hide
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C15H19ClN2O3S
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1
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| 1 |
Ki = 2945 nM
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CP0421834
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5-bromo-3-(3-ethylimidazol-4-yl)-4-fluoro-1H-indole
Show/Hide
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C13H11BrFN3
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1
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| 1 |
Ki = 2951 nM
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CP0473972
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5,7-Dimethyl-2-(methylsulfinyl)-3-(phenylsulfonyl)pyrazolo[1,5-a]pyrimidine
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C15H15N3O3S2
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1
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| 1 |
Ki = 2960 nM
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CP0396620
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4-[4-[2-[(2S)-1-isoquinolin-4-ylsulfonylpyrrolidin-2-yl]ethyl]piperazin-1-yl]-3H-1,3-benzoxazol-2-one
Show/Hide
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C26H29N5O4S
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1
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| 1 |
Ki = 2990 nM
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CP0553532
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3-(3-ethylimidazol-4-yl)-1H-indole
Show/Hide
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C13H13N3
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1
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| 1 |
Ki = 3020 nM
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CP0577942
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1-[(3-methoxyphenyl)methyl]-N-(oxan-4-yl)pyrrolo[3,2-c]quinolin-4-amine
Show/Hide
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C24H25N3O2
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1
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| 1 |
Ki = 3024 nM
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CP0473054
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(1S,2R,6S,7R)-4-[6-[4-(4-chlorophenyl)piperazin-1-yl]hexyl]-4-azatricyclo[5.2.1.02,6]decane-3,5-dione
Show/Hide
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C25H34ClN3O2
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1
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| 1 |
Ki = 3028 nM
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CP0411591
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3-methyl-5,5-diphenyl-1-[5-(4-phenylpiperazin-1-yl)pentyl]imidazolidine-2,4-dione;hydrochloride
Show/Hide
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C31H36N4O2
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1
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| 1 |
Ki = 3071 nM
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CP0908603
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1-(1H-indol-3-yl)-2-(phenylsulfonyl)-1,2-dihydroisoquinoline
Show/Hide
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C23H18N2O2S
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1
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| 1 |
Ki = 3104 nM
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CP0051242
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(R)-1-(2-(1-(3-bromo-benzenesulfonyl)-pyrrolidin-2-yl)-ethyl)-4-methyl piperidine
Show/Hide
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C18H27BrN2O2S
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1
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| 1 |
Ki = 3162.28 nM
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CP0416670
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1-[6-[4-(4-bromophenyl)piperazin-1-yl]hexyl]benzo[cd]indol-2-one;hydrochloride
Show/Hide
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C27H31BrClN3O
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1
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| 1 |
Ki = 3187 nM
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CP0400393
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N-[(E)-(6-chloro-2,3,4,9-tetrahydrocarbazol-1-ylidene)amino]-4-methylbenzenesulfonamide
Show/Hide
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C19H18ClN3O2S
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1
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| 1 |
Ki = 3213 nM
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CP0575068
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2-N-[2-(1H-indol-3-yl)ethyl]-6-(4-phenylpiperazin-1-yl)-1,3,5-triazine-2,4-diamine
Show/Hide
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C23H26N8
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1
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| 1 |
Ki = 3220 nM
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CP0417068
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3-[6-[4-(2-methoxyphenyl)piperazin-1-yl]hexyl]-1,3-diazatricyclo[6.3.1.04,12]dodeca-4,6,8(12)-trien-2-one
Show/Hide
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C27H36N4O2
|
1
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| 1 |
Ki = 3270 nM
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CP0548183
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N-[(3,4-dimethoxyphenyl)methyl]-2-[2-ethyl-2-methyl-4-(4-methylphenyl)oxan-4-yl]ethanamine
Show/Hide
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C26H37NO3
|
1
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| 1 |
Ki = 3400 nM
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CP0445867
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N-[(4-cyanophenyl)methyl]-3-[2-[4-(2-phenylpyridin-3-yl)piperazin-1-yl]ethoxy]propanamide
Show/Hide
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C28H31N5O2
|
1
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| 1 |
Ki = 3441 nM
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CP0528509
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3-(3-ethylimidazol-4-yl)-4-fluoro-5-methoxy-1H-indole
Show/Hide
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C14H14FN3O
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1
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| 1 |
Ki = 3467 nM
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CP0541126
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3-(3-ethylimidazol-4-yl)-5-(trifluoromethoxy)-1H-indole
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C14H12F3N3O
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1
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| 1 |
Ki = 3467 nM
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CP0258551
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1-[4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]-3-methyl-5,5-diphenylimidazolidine-2,4-dione
Show/Hide
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C31H36N4O3
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1
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| 1 |
Ki = 3567 nM
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CP0431611
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4-[(2-chlorophenyl)sulfonylmethyl]-6-(4-methylpiperazin-1-yl)-1,3,5-triazin-2-amine
Show/Hide
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C15H19ClN6O2S
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1
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| 1 |
Ki = 3574 nM
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CP0384571
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1-[6-[4-(4-methoxyphenyl)piperazin-1-yl]hexyl]benzo[cd]indol-2-one
Show/Hide
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C28H33N3O2
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1
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| 1 |
Ki = 3666 nM
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CP0412479
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(3-Benzo[1,3]dioxol-5-yl-3-phenyl-propyl)-(4-methoxy-benzyl)-amine
Show/Hide
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C24H25NO3
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1
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| 1 |
Ki = 3700 nM
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CP0699214
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(5Z)-5-((4-bromo-1H-indol-3-yl)methylene)-2-(methylimino)imidazolidin-4-one
Show/Hide
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C13H11BrN4O
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1
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| 1 |
Ki = 3733 nM
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CP0854352
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N-{4-[4-(3-Chlorophenyl)-piperazin-1-yl]-butyl}-8-quinolinesulfonamide hydrochloride
Show/Hide
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C23H28Cl2N4O2S
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1
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| 1 |
Ki = 3765 nM
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CP0433626
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2-ethoxy-N-[1-[2-(3-fluorophenoxy)ethyl]piperidin-4-yl]benzamide
Show/Hide
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C22H27FN2O3
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1
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| 1 |
Ki = 3785 nM
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CP0448724
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4-[4-[2-[4-(3-fluorophenyl)piperazin-1-yl]ethyl]piperidin-1-yl]sulfonylisoquinoline
Show/Hide
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C26H31FN4O2S
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1
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| 1 |
Ki = 3802 nM
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CP0528511
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4-fluoro-5-methoxy-3-(3-methylimidazol-4-yl)-1H-indole
Show/Hide
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C13H12FN3O
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1
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| 1 |
Ki = 3802 nM
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CP0034610
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1-[(3-chlorophenyl)methyl]-4-(4,4-difluoropiperidin-1-yl)pyrrolo[3,2-c]quinoline
Show/Hide
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C23H20ClF2N3
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1
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| 1 |
Ki = 3827 nM
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CP0472438
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4-[4-[2-[(2S)-1-quinolin-5-ylsulfonylpyrrolidin-2-yl]ethyl]piperazin-1-yl]-3H-1,3-benzoxazol-2-one
Show/Hide
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C26H29N5O4S
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1
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| 1 |
Ki = 3912 nM
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CP0505675
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4-(2-benzenesulfonylphenyl)piperazine
Show/Hide
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C16H18N2O2S
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1
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| 1 |
Ki = 4000 nM
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CP0067163
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2-[4-[(Z)-4-chloranyl-1,2-diphenyl-but-1-enyl]phenoxy]-N,N-dimethyl-ethanamine;2-oxidanylpropane-1,2,3-tricarboxylic acid
Show/Hide
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C26H28ClNO
|
1
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| 1 |
Ki = 4125 nM
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CP0401239
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1-[3-[4-(2-ethoxyphenyl)piperazin-1-yl]propyl]-3-methyl-5,5-diphenylimidazolidine-2,4-dione
Show/Hide
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C31H36N4O3
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1
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| 1 |
Ki = 4139 nM
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CP0568316
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2-[6-(4-quinolin-8-ylpiperazin-1-yl)hexyl]-[1,2,4]triazolo[4,3-a]pyridin-3-one
Show/Hide
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C25H30N6O
|
1
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| 1 |
Ki = 4144 nM
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CP0440390
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5-chloro-3-(3-ethylimidazol-4-yl)-1H-indole
Show/Hide
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C13H12ClN3
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1
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| 1 |
Ki = 4169 nM
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CP0498609
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4-(Indan-1-ylsulfanyl)-phenylamine
Show/Hide
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C15H15NS
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1
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| 1 |
Ki = 4200 nM
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CP0480126
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3-benzyl-5,5-dimethyl-1-[5-(4-phenylpiperazin-1-yl)pentyl]imidazolidine-2,4-dione;hydrochloride
Show/Hide
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C27H36N4O2
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1
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| 1 |
Ki = 4368 nM
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CP0498236
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4-(1H-Inden-1-ylmethyl)-phenylamine
Show/Hide
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C16H15N
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1
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| 1 |
Ki = 4470 nM
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CP0428021
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N-benzhydryl-5-(4-methylpiperazin-1-yl)-2-nitroaniline
Show/Hide
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C24H26N4O2
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1
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| 1 |
Ki = 4489 nM
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CP0872933
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[2-(6,6-dioxo-10b,10c-dihydro-6H-6lambda6-thia-5a-aza-acephenanthrylen-4-yl)-ethyl]-dimethyl-amine
Show/Hide
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C18H18N2O2S
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1
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| 1 |
Ki = 4500 nM
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CP0456105
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1'-[2-[4-(4-chlorophenyl)piperidin-1-yl]ethyl]spiro[1H-indole-3,3'-pyrrolidine]-2-one
Show/Hide
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C24H28ClN3O
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1
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| 1 |
Ki = 4577 nM
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CP0545013
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2-[[4-[[4-(3-chlorophenyl)piperazin-1-yl]methyl]cyclohexyl]methyl]-[1,2,4]triazolo[4,3-a]pyridin-3-one
Show/Hide
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C24H30ClN5O
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1
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| 1 |
Ki = 4581 nM
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CP0427385
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N-[5-(3,4,4a,5,6,7,8,8a-octahydro-1H-isoquinolin-2-yl)pentyl]-N-ethylquinoline-8-sulfonamide
Show/Hide
|
C25H37N3O2S
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1
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| 1 |
Ki = 4587 nM
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CP0542995
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2-N-(2-anilinoethyl)-4-N-[2-(1H-indol-3-yl)ethyl]-1,3,5-triazine-2,4,6-triamine
Show/Hide
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C21H24N8
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1
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| 1 |
Ki = 4736 nM
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CP0456102
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1'-[2-[4-(4-chlorophenyl)piperazin-1-yl]ethyl]spiro[1H-indole-3,3'-pyrrolidine]-2-one
Show/Hide
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C23H27ClN4O
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1
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| 1 |
Ki = 4737 nM
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CP0485157
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1'-[2-[4-(4-fluorophenyl)piperazin-1-yl]ethyl]spiro[1H-indole-3,3'-pyrrolidine]-2-one
Show/Hide
|
C23H27FN4O
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1
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| 1 |
Ki = 4744 nM
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CP0461296
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N-[4-[4-(1,2-benzoxazol-3-yl)piperazin-1-yl]butyl]-4-(trifluoromethoxy)benzenesulfonamide
Show/Hide
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C22H25F3N4O4S
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1
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| 1 |
Ki = 4800 nM
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CP0473055
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(1R,2S,6R,7S)-4-[6-[4-(2-methoxyphenyl)piperazin-1-yl]hexyl]-4-azatricyclo[5.2.1.02,6]decane-3,5-dione
Show/Hide
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C26H37N3O3
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1
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| 1 |
Ki = 4874 nM
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CP0421838
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3-(3-ethylimidazol-4-yl)-5-fluoro-1H-indole
Show/Hide
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C13H12FN3
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1
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| 1 |
Ki = 4898 nM
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CP0388312
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2-{2-ethyl-1H-pyrrolo[3,2-c]pyridin-3-yl}ethan-1-amine, 23
Show/Hide
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C11H15N3
|
1
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| 1 |
Ki = 4900 nM
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CP0568128
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6-[4-(3-chlorophenyl)piperazin-1-yl]hexylurea
Show/Hide
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C17H27ClN4O
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1
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| 1 |
Ki = 4929 nM
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CP0860969
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N-(3-(4-(3-chlorophenyl)piperazin-1-yl)propyl)quinoline-3-sulfonamide hydrochloride
Show/Hide
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C22H26Cl2N4O2S
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1
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| 1 |
Ki = 5043 nM
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CP0387338
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N-[[5-bromo-2-[(4-methylphenyl)methoxy]phenyl]methyl]-1-phenylethanamine
Show/Hide
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C23H24BrNO
|
1
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| 1 |
Ki = 5100 nM
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CP0418216
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7-[4-[4-(3-chlorophenyl)piperazin-1-yl]butyl]-1,3-dimethylpurine-2,6-dione;hydrochloride
Show/Hide
|
C21H27ClN6O2
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1
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| 1 |
Ki = 5150 nM
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CP0497344
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N-[4-[4-(1,2-benzoxazol-3-yl)piperazin-1-yl]butyl]thiophene-2-sulfonamide
Show/Hide
|
C19H24N4O3S2
|
1
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| 1 |
Ki = 5200 nM
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CP0417064
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1-[6-(4-pyrimidin-2-ylpiperazin-1-yl)hexyl]benzo[cd]indol-2-one
Show/Hide
|
C25H29N5O
|
1
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| 1 |
Ki = 5253 nM
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CP0412402
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1'-[2-[4-(4-fluorophenyl)piperidin-1-yl]ethyl]spiro[1H-indole-3,3'-pyrrolidine]-2-one
Show/Hide
|
C24H28FN3O
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1
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| 1 |
Ki = 5285 nM
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CP0383204
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1'-[3-[4-(4-chlorophenyl)piperazin-1-yl]propyl]spiro[1H-indole-3,3'-pyrrolidine]-2-one
Show/Hide
|
C24H29ClN4O
|
1
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| 1 |
Ki = 5559 nM
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CP0387336
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N-benzyl-2-[2-ethyl-2-methyl-4-(4-methylphenyl)oxan-4-yl]ethanamine
Show/Hide
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C24H33NO
|
1
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| 1 |
Ki = 5600 nM
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CP0379117
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1-[3-(benzenesulfonyl)-6-chloroquinolin-4-yl]piperidine-4-carboxamide
Show/Hide
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C21H20ClN3O3S
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1
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| 1 |
Ki = 5676 nM
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CP0417063
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2-[6-[4-(4-methoxyphenyl)piperazin-1-yl]hexyl]benzo[de]isoquinoline-1,3-dione
Show/Hide
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C29H33N3O3
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1
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| 1 |
Ki = 5765 nM
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CP0438306
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4-methyl-4-(5-methylfuran-2-yl)-N-[[4-(trifluoromethyl)phenyl]methyl]pentan-2-amine
Show/Hide
|
C19H24F3NO
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1
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| 1 |
Ki = 5800 nM
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CP0384209
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4-chloro-N-(2-isoquinolin-1-ylphenyl)benzenesulfonamide
Show/Hide
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C21H15ClN2O2S
|
1
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| 1 |
Ki = 5805 nM
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CP0523197
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2-(4-fluorophenyl)sulfonyl-1-(1H-indol-3-yl)-3H-isoquinoline
Show/Hide
|
C23H17FN2O2S
|
1
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| 1 |
Ki = 5826 nM
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CP0541121
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3-(3-ethylimidazol-4-yl)-6-fluoro-1H-indole
Show/Hide
|
C13H12FN3
|
1
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| 1 |
Ki = 5888 nM
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CP0909449
|
2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-9H-xanthen-9-one hydrochloride
Show/Hide
|
C25H25ClN2O3
|
1
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| 1 |
Ki = 5939 nM
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CP0533096
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4-((5,6,7,8-tetrahydrocarbazol-9-yl)methyl)benzenamine
Show/Hide
|
C19H20N2
|
1
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| 1 |
Ki = 6000 nM
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CP0900183
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methyl 3-(1-ethyl-1H-imidazol-5-yl)-1H-indole-5-carboxylate
Show/Hide
|
C15H15N3O2
|
1
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| 1 |
Ki = 6062 nM
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CP0406518
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4-Indan-1-ylmethyl-phenylamine
Show/Hide
|
C16H17N
|
1
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| 1 |
Ki = 6100 nM
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CP0456104
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1'-[2-[4-(4-fluorophenyl)-3,6-dihydro-2H-pyridin-1-yl]ethyl]spiro[1H-indole-3,3'-pyrrolidine]-2-one
Show/Hide
|
C24H26FN3O
|
1
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| 1 |
Ki = 6267 nM
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CP0096286
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(R)-3-(2-(2-(4-methylpiperidin-1-yl)ethyl)pyrrolidin-1-ylsulfonyl)phenol
Show/Hide
|
C18H28N2O3S
|
1
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| 1 |
Ki = 6309.57 nM
|
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CP0418579
|
2-(benzenesulfonyl)-4,6-diphenylthieno[2,3-b]pyridin-3-amine
Show/Hide
|
C25H18N2O2S2
|
1
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| 1 |
Ki = 6401 nM
|
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CP0562326
|
3-(3-ethylimidazol-4-yl)-4-fluoro-1H-indole
Show/Hide
|
C13H12FN3
|
1
|
| 1 |
Ki = 6457 nM
|
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CP0504617
|
4-[(4-chlorophenyl)methylsulfanyl]-6-fluoro-3-(4-methylphenyl)sulfonylquinoline
Show/Hide
|
C23H17ClFNO2S2
|
1
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| 1 |
Ki = 6505 nM
|
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CP0880894
|
N-{3-[4-(4-Chlorophenyl)-piperazin-1-yl]-propyl}-3-quinolinesulfonamide hydrochloride
Show/Hide
|
C22H26Cl2N4O2S
|
1
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| 1 |
Ki = 6548 nM
|
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CP0485159
|
1'-[2-(4-phenylpiperazin-1-yl)ethyl]spiro[1H-indole-3,3'-pyrrolidine]-2-one
Show/Hide
|
C23H28N4O
|
1
|
| 1 |
Ki = 6556 nM
|
|
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CP0542761
|
2-N-[5-[4-(2-methoxyphenyl)piperazin-1-yl]pentyl]-1,3,5-triazine-2,4,6-triamine
Show/Hide
|
C19H30N8O
|
1
|
| 1 |
Ki = 6652 nM
|
|
|
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CP0470500
|
5-[4-[2-(4-phenylpiperazin-1-yl)ethyl]piperidin-1-yl]sulfonylquinoline
Show/Hide
|
C26H32N4O2S
|
1
|
| 1 |
Ki = 6712 nM
|
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CP0369306
|
4-[4-imidazo[1,2-a]pyridin-5-yl-3-(trifluoromethyl)phenoxy]furo[3,2-c]pyridine
Show/Hide
|
C21H12F3N3O2
|
1
|
| 1 |
Ki = 6900 nM
|
|
|
|
CP0757055
|
3-(1-methyl-1H-imidazol-5-yl)-1H-indole-5-carboxamide
Show/Hide
|
C13H12N4O
|
1
|
| 1 |
Ki = 6910 nM
|
|
|
|
CP0528508
|
3-(3-ethylimidazol-4-yl)-5-methoxy-1H-indole
Show/Hide
|
C14H15N3O
|
1
|
| 1 |
Ki = 6918 nM
|
|
|
|
CP0421833
|
5-ethoxy-3-(3-ethylimidazol-4-yl)-1H-indole
Show/Hide
|
C15H17N3O
|
1
|
| 1 |
Ki = 7079 nM
|
|
|
|
CP0548406
|
1,1-dioxo-2-[5-(4-pyrimidin-2-ylpiperazin-1-yl)pentyl]-1,2-benzothiazol-3-one
Show/Hide
|
C20H25N5O3S
|
1
|
| 1 |
Ki = 7097 nM
|
|
|
|
CP0244206
|
7-[4-imidazo[1,2-a]pyridin-5-yl-3-(trifluoromethyl)phenoxy]thieno[2,3-c]pyridine
Show/Hide
|
C21H12F3N3OS
|
1
|
| 1 |
Ki = 7200 nM
|
|
|
|
CP0859942
|
3-(1-ethyl-1H-imidazol-5-yl)-1H-indole-5-sulfonamide
Show/Hide
|
C13H14N4O2S
|
1
|
| 1 |
Ki = 7271 nM
|
|
|
|
CP0114041
|
CHEMBL2058429
Show/Hide
|
C15H15BrN4O
|
1
|
| 1 |
Ki = 7300 nM
|
|
|
|
CP0510463
|
3-benzyl-1-[5-[4-(2,4-difluorophenyl)piperazin-1-yl]pentyl]-5,5-dimethylimidazolidine-2,4-dione;hydrochloride
Show/Hide
|
C27H34F2N4O2
|
1
|
| 1 |
Ki = 7469 nM
|
|
|
|
CP0545394
|
4-(3-chlorophenyl)piperazine-1-carboxamide
Show/Hide
|
C11H14ClN3O
|
1
|
| 1 |
Ki = 7489 nM
|
|
|
|
CP0114039
|
CHEMBL2058426
Show/Hide
|
C15H15BrN4O
|
1
|
| 1 |
Ki = 7523 nM
|
|
|
|
CP0568014
|
2-N-[6-[4-(2-methoxyphenyl)piperazin-1-yl]hexyl]-1,3,5-triazine-2,4,6-triamine
Show/Hide
|
C20H32N8O
|
1
|
| 1 |
Ki = 7704 nM
|
|
|
|
CP0456108
|
1'-[2-[4-(4-chlorobenzoyl)piperazin-1-yl]ethyl]spiro[1H-indole-3,3'-pyrrolidine]-2-one
Show/Hide
|
C24H27ClN4O2
|
1
|
| 1 |
Ki = 7746 nM
|
|
|
|
CP0098968
|
3-(3-ethylimidazol-4-yl)-1H-indole-5-carboxamide
Show/Hide
|
C14H14N4O
|
2
|
| 1 |
Ki = 7762 nM
|
|
|
| 2 |
Ki > 10000 nM
|
|
|
|
CP0056178
|
4-fluoranyl-N-(4-oxidanyl-3-quinolin-8-ylsulfanyl-naphthalen-1-yl)benzenesulfonamide
Show/Hide
|
C25H17FN2O3S2
|
1
|
| 1 |
Ki = 7886 nM
|
|
|
|
CP0415883
|
4-[4-[1-[4-[1-[6-[(2-methylpropan-2-yl)oxycarbonylamino]hexyl]triazol-4-yl]butyl]piperidin-4-yl]phenyl]-7-[4-(trifluoromethyl)phenyl]naphthalene-2-carboxylic acid
Show/Hide
|
C46H54F3N5O4
|
1
|
| 1 |
Ki = 7900 nM
|
|
|
|
CP0064188
|
4-[4-(6-methylimidazo[1,2-a]pyrazin-5-yl)-3-(trifluoromethyl)phenoxy]furo[3,2-c]pyridine
Show/Hide
|
C21H13F3N4O2
|
1
|
| 1 |
Ki = 7900 nM
|
|
|
|
CP0064183
|
4-[3-methyl-4-(6-methylimidazo[1,2-a]pyrazin-5-yl)phenoxy]furo[3,2-c]pyridine
Show/Hide
|
C21H16N4O2
|
1
|
| 1 |
Ki = 8100 nM
|
|
|
|
CP0513126
|
1-[5-[4-(2,4-difluorophenyl)piperazin-1-yl]pentyl]-3-[(4-fluorophenyl)methyl]-5,5-dimethylimidazolidine-2,4-dione;hydrochloride
Show/Hide
|
C27H33F3N4O2
|
1
|
| 1 |
Ki = 8104 nM
|
|
|
|
CP0504962
|
4-((1H-indol-1-yl)methyl)benzenamine
Show/Hide
|
C15H14N2
|
1
|
| 1 |
Ki = 8200 nM
|
|
|
|
CP0417574
|
5-[4-[2-[4-(3-fluorophenyl)piperazin-1-yl]ethyl]piperidin-1-yl]sulfonylquinoline
Show/Hide
|
C26H31FN4O2S
|
1
|
| 1 |
Ki = 8279 nM
|
|
|
|
CP0510464
|
3-benzyl-1-[5-[4-(2-methoxyphenyl)piperazin-1-yl]pentyl]-5,5-dimethylimidazolidine-2,4-dione;hydrochloride
Show/Hide
|
C28H39ClN4O3
|
1
|
| 1 |
Ki = 8611 nM
|
|
|
|
CP0886023
|
1-((S)-1-Methyl-pyrrolidin-2-ylmethyl)-1H-indole hydrochloride
Show/Hide
|
C14H19ClN2
|
1
|
| 1 |
Ki = 8750 nM
|
|
|
|
CP0253203
|
(E)-5-((1H-Indol-3yl)methylene)-2-imino-1,3-dimethylimidazolidin-4-one
Show/Hide
|
C14H14N4O
|
1
|
| 1 |
Ki = 8768 nM
|
|
|
|
CP0846085
|
6-methoxy-2-{[4-(benzyl)piperazin-1-yl]methyl}-9H-xanthen-9-one dihydrochloride
Show/Hide
|
C26H28Cl2N2O3
|
1
|
| 1 |
Ki = 8836 nM
|
|
|
|
CP0481901
|
7-[5-[4-(2-methoxyphenyl)piperazin-1-yl]pentyl]-1,3-dimethylpurine-2,6-dione;hydrochloride
Show/Hide
|
C23H32N6O3
|
1
|
| 1 |
Ki = 8987 nM
|
|
|
|
CP0438307
|
(1R)-3-[3-(3,4-difluorophenyl)-6,7-dihydro-4H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-1-phenylpropan-1-ol
Show/Hide
|
C21H20F2N2O2
|
1
|
| 1 |
Ki = 9000 nM
|
|
|
|
CP0527834
|
7-[5-(3,4-dihydro-1H-isoquinolin-2-yl)pentyl]-1,3-dimethylpurine-2,6-dione;hydrochloride
Show/Hide
|
C21H27N5O2
|
1
|
| 1 |
Ki = 9141 nM
|
|
|
|
CP0542994
|
2-N-[5-(4-phenylpiperazin-1-yl)pentyl]-1,3,5-triazine-2,4,6-triamine
Show/Hide
|
C18H28N8
|
1
|
| 1 |
Ki = 9302 nM
|
|
|
|
CP0876492
|
3-Methoxy-5-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-9H-xanthen-9-one hydrochloride
Show/Hide
|
C26H27ClN2O4
|
1
|
| 1 |
Ki = 9363 nM
|
|
|
|
CP0095011
|
3,5-dimethyl-5-phenyl-1-[5-(4-phenylpiperazin-1-yl)pentyl]imidazolidine-2,4-dione;hydrochloride
Show/Hide
|
C26H34N4O2
|
1
|
| 1 |
Ki = 9600 nM
|
|
|
|
CP0504618
|
N-(10a-morpholin-4-yl-7,8,9,10-tetrahydro-6bH-naphtho[1,2-b][1]benzofuran-5-yl)benzenesulfonamide
Show/Hide
|
C26H28N2O4S
|
1
|
| 1 |
Ki = 9669 nM
|
|
|
|
CP0372923
|
2-[3-[(2S,5S)-5-[(6-bromo-1H-indol-3-yl)methyl]-3,6-dioxopiperazin-2-yl]propyl]guanidine
Show/Hide
|
C17H21BrN6O2
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0845072
|
(cyclo[(6-bromo-8-entryptophan)arginine])
Show/Hide
|
C17H19BrN6O2
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0635067
|
2-amino-6-chloro-3,4-dihydroquinazoline hydrochloride
Show/Hide
|
C8H9Cl2N3
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0395878
|
N-[3-[4-(1,2-benzoxazol-3-yl)piperazin-1-yl]propyl]-5-fluoro-3-methyl-1-benzothiophene-2-sulfonamide
Show/Hide
|
C23H25FN4O3S2
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0395880
|
N-[4-[4-(1,2-benzoxazol-3-yl)piperazin-1-yl]butyl]-1,3-benzothiazole-4-sulfonamide
Show/Hide
|
C22H25N5O3S2
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0447126
|
N-[3-[4-(1,2-benzoxazol-3-yl)piperazin-1-yl]propyl]-1,3-benzothiazole-4-sulfonamide
Show/Hide
|
C21H23N5O3S2
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0447212
|
N-[3-[4-(1,2-benzoxazol-3-yl)piperazin-1-yl]propyl]thiophene-2-sulfonamide
Show/Hide
|
C18H22N4O3S2
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0054519
|
(1R,12R,13S,17R,21S)-12-ethyl-18-propyl-7-(trifluoromethyl)-10,18-diazapentacyclo[11.7.1.02,11.04,9.017,21]henicosa-2(11),3,5,7,9-pentaene
Show/Hide
|
C25H31F3N2
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0085414
|
(3aS,6R,6aS,9aR,9bR)-6-benzyl-1-methyl-3,3a,4,6,6a,7,8,9,9a,9b-decahydro-2H-benzo[de]quinolin-5-one
Show/Hide
|
C20H27NO
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0110111
|
[(4S,5S)-5-methyl-2-thiophen-3-yl-4,5-dihydro-1,3-thiazol-4-yl]methanol
Show/Hide
|
C9H11NOS2
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0176519
|
(4R,5S)-4-(1H-imidazol-5-ylmethyl)-5-methyl-2-phenyl-4,5-dihydro-1,3-thiazole
Show/Hide
|
C14H15N3S
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0315736
|
2-[4-(1H-imidazol-5-ylmethyl)-4,5-dihydro-1,3-thiazol-2-yl]phenol
Show/Hide
|
C13H13N3OS
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0315738
|
[(4S,5S)-5-methyl-2-phenyl-4,5-dihydro-1,3-thiazol-4-yl]methanol
Show/Hide
|
C11H13NOS
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0315739
|
[(4S,5S)-2-(1H-indol-3-yl)-5-methyl-4,5-dihydro-1,3-thiazol-4-yl]methanol
Show/Hide
|
C13H14N2OS
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0315740
|
[(4S,5S)-5-methyl-2-thiophen-2-yl-4,5-dihydro-1,3-thiazol-4-yl]methanol
Show/Hide
|
C9H11NOS2
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0369530
|
methyl (2S)-2-[[(4S,5R)-2-(2-hydroxyphenyl)-5-methyl-4,5-dihydro-1,3-thiazole-4-carbonyl]amino]-3-(1H-imidazol-5-yl)propanoate
Show/Hide
|
C18H20N4O4S
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0396119
|
2-[(3aR,6aS)-4,5,6,6a-tetrahydro-3aH-cyclopenta[d][1,3]thiazol-2-yl]phenol
Show/Hide
|
C12H13NOS
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0396120
|
[(4S,5S)-5-methyl-2-(4-octoxyphenyl)-4,5-dihydro-1,3-thiazol-4-yl]methanol
Show/Hide
|
C19H29NO2S
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0396121
|
[(4S,5S)-2-(4-butoxyphenyl)-5-methyl-4,5-dihydro-1,3-thiazol-4-yl]methanol
Show/Hide
|
C15H21NO2S
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0396122
|
[(4S,5S)-2-(4-hexoxyphenyl)-5-methyl-4,5-dihydro-1,3-thiazol-4-yl]methanol
Show/Hide
|
C17H25NO2S
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0396185
|
[(4S,5S)-5-methyl-2-[2-(methylamino)phenyl]-4,5-dihydro-1,3-thiazol-4-yl]methanol
Show/Hide
|
C12H16N2OS
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0408362
|
(4S,5S)-4-(1H-imidazol-5-ylmethyl)-5-methyl-2-phenyl-4,5-dihydro-1,3-thiazole
Show/Hide
|
C14H15N3S
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0444340
|
3-[(4S,5S)-4-(hydroxymethyl)-5-methyl-4,5-dihydro-1,3-thiazol-2-yl]naphthalen-2-ol
Show/Hide
|
C15H15NO2S
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0475794
|
[(4S,5S)-2-(furan-2-yl)-5-methyl-4,5-dihydro-1,3-thiazol-4-yl]methanol
Show/Hide
|
C9H11NO2S
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0391908
|
3-(4-fluorophenyl)-5,6,7,8-tetrahydro-4H-[1,2]oxazolo[4,5-d]azepine
Show/Hide
|
C13H13FN2O
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0421663
|
5-chloro-3-(3-ethylimidazol-4-yl)-6-fluoro-1H-indole
Show/Hide
|
C13H11ClFN3
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0421836
|
3-(3-ethylimidazol-4-yl)-4-fluoro-1H-indole-5-carboxamide
Show/Hide
|
C14H13FN4O
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0440388
|
3-(3-ethylimidazol-4-yl)-5-methyl-1H-indole
Show/Hide
|
C14H15N3
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0537948
|
4-fluoro-3-(3-methylimidazol-4-yl)-1H-indole-5-carboxamide
Show/Hide
|
C13H11FN4O
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0127400
|
(-)-Pramipexole
Show/Hide
|
C10H17N3S
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0514794
|
2-[[4-[[4-(2-methoxyphenyl)piperazin-1-yl]methyl]phenyl]methyl]-1,1-dioxo-1,2-benzothiazol-3-one
Show/Hide
|
C26H27N3O4S
|
1
|
| 1 |
Ki = 10090 nM
|
|
|
|
CP0398059
|
1,3-dimethyl-7-[5-(4-phenylpiperazin-1-yl)pentyl]purine-2,6-dione;hydrochloride
Show/Hide
|
C22H30N6O2
|
1
|
| 1 |
Ki = 10350 nM
|
|
|
|
CP0893594
|
3-{4-[4-(4-Chlorophenyl)-piperazin-1-ylmethyl]-piperidine-1-sulfonyl}-quinoline hydrochloride
Show/Hide
|
C25H30Cl2N4O2S
|
1
|
| 1 |
Ki = 10570 nM
|
|
|
|
CP0382069
|
5-(4-fluorophenyl)-3-[2-hydroxy-3-[4-(2-methoxyphenyl)piperazin-1-yl]propyl]-5-methylimidazolidine-2,4-dione;hydrochloride
Show/Hide
|
C24H29FN4O4
|
1
|
| 1 |
Ki = 10790 nM
|
|
|
|
CP0569637
|
2-N-[4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]-1,3,5-triazine-2,4,6-triamine
Show/Hide
|
C18H28N8O
|
1
|
| 1 |
Ki = 10870 nM
|
|
|
|
CP0481865
|
N-(5-chloro-2-methylphenyl)-2-(2,4-difluorophenyl)-N-methyl-1-oxoisoquinoline-4-carboxamide
Show/Hide
|
C24H17ClF2N2O2
|
1
|
| 1 |
Ki = 11360 nM
|
|
|
|
CP0483411
|
7-[4-(3,4-dihydro-1H-isoquinolin-2-yl)butyl]-1,3-dimethylpurine-2,6-dione;hydrochloride
Show/Hide
|
C20H25N5O2
|
1
|
| 1 |
Ki = 11670 nM
|
|
|
|
CP0528323
|
4-(3H-Inden-1-ylmethyl)-phenylamine
Show/Hide
|
C16H15N
|
1
|
| 1 |
Ki = 11800 nM
|
|
|
|
CP0379113
|
5-bromo-N-[1-(naphthalen-1-ylmethyl)pyrazol-3-yl]thiophene-2-sulfonamide
Show/Hide
|
C18H14BrN3O2S2
|
1
|
| 1 |
Ki = 11980 nM
|
|
|
|
CP0558478
|
7-[3-[4-(2-methoxyphenyl)piperazin-1-yl]propyl]-1,3-dimethylpurine-2,6-dione;hydrochloride
Show/Hide
|
C21H28N6O3
|
1
|
| 1 |
Ki = 12100 nM
|
|
|
|
CP0543165
|
7-[3-(3,4-dihydro-1H-isoquinolin-2-yl)propyl]-1,3-dimethylpurine-2,6-dione;hydrochloride
Show/Hide
|
C19H23N5O2
|
1
|
| 1 |
Ki = 12250 nM
|
|
|
|
CP0400006
|
4-benzyl-12-bromo-1,4-diazatetracyclo[7.6.1.05,16.010,15]hexadeca-9(16),10(15),11,13-tetraene
Show/Hide
|
C21H21BrN2
|
1
|
| 1 |
Ki = 12730 nM
|
|
|
|
CP0379115
|
10-[(4-chloro-2-fluorophenyl)methyl]phenothiazine 5,5-dioxide
Show/Hide
|
C19H13ClFNO2S
|
1
|
| 1 |
Ki = 13330 nM
|
|
|
|
CP0876491
|
6-Methoxy-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-9H-xanthen-9-one hydrochloride
Show/Hide
|
C26H27ClN2O4
|
1
|
| 1 |
Ki = 13600 nM
|
|
|
|
CP0542757
|
2-N-[6-(4-phenylpiperazin-1-yl)hexyl]-1,3,5-triazine-2,4,6-triamine
Show/Hide
|
C19H30N8
|
1
|
| 1 |
Ki = 13650 nM
|
|
|
|
CP0398057
|
1,3-dimethyl-7-[4-(4-phenylpiperazin-1-yl)butyl]purine-2,6-dione;hydrochloride
Show/Hide
|
C21H28N6O2
|
1
|
| 1 |
Ki = 14210 nM
|
|
|
|
CP0876490
|
3-Chloro-5-{[4-(2-hydroxyethyl)piperazin-1-yl]methyl}-9H-xanthen-9-one dihydrochloride
Show/Hide
|
C20H24Cl4N2O3
|
1
|
| 1 |
Ki = 14420 nM
|
|
|
|
CP0456382
|
N-[4-(3,4,4a,5,6,7,8,8a-octahydro-1H-isoquinolin-2-yl)butyl]-N-ethylquinoline-3-sulfonamide
Show/Hide
|
C24H35N3O2S
|
1
|
| 1 |
Ki = 14460 nM
|
|
|
|
CP0382640
|
1-[5-[4-(2-methoxyphenyl)piperazin-1-yl]pentyl]-3,5-dimethyl-5-phenylimidazolidine-2,4-dione;hydrochloride
Show/Hide
|
C27H36N4O3
|
1
|
| 1 |
Ki = 14650 nM
|
|
|
|
CP0147070
|
N-(4-hydroxy-3-quinolin-8-ylsulfanylnaphthalen-1-yl)benzenesulfonamide
Show/Hide
|
C25H18N2O3S2
|
1
|
| 1 |
Ki = 15610 nM
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CP0418580
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N-(3-chlorophenyl)-2-(3-methoxyphenyl)-N-methyl-1-oxoisoquinoline-4-carboxamide
Show/Hide
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C24H19ClN2O3
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1
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| 1 |
Ki = 16550 nM
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CP0834204
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4-(4-{2-[4-(4-Chlorophenyl)-piperazin-1-yl]-ethyl}-piperidine-1-sulfonyl)-isoquinoline hydrochloride
Show/Hide
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C26H32Cl2N4O2S
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1
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| 1 |
Ki = 16650 nM
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CP0059583
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1,1-Dioxo-2-[4-(4-pyrimidin-2-yl-piperazin-1-yl)-butyl]-1,2-dihydro-1lambda*6*-benzo[d]isothiazol-3-one
Show/Hide
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C19H23N5O3S
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1
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| 1 |
Ki = 16800 nM
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CP0860958
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7-{4-[4-(4-Chlorophenyl)-piperazin-1-ylmethyl]-piperidine-1-sulfonyl}-quinoline hydrochloride
Show/Hide
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C25H30Cl2N4O2S
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1
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| 1 |
Ki = 17150 nM
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CP0542765
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2-N-[4-(4-phenylpiperazin-1-yl)butyl]-1,3,5-triazine-2,4,6-triamine
Show/Hide
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C17H26N8
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1
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| 1 |
Ki = 17350 nM
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CP0856666
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6-Methoxy-2-[(4-methylpiperazin-1-yl)methyl]-9H-xanthen-9-one dihydrochloride
Show/Hide
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C20H24Cl2N2O3
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1
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| 1 |
Ki = 19100 nM
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CP0850785
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3-Chloro-5-[(4-methylpiperazin-1-yl)methyl]-9H-xanthen-9-one dihydrochloride
Show/Hide
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C19H22Cl4N2O2
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1
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| 1 |
Ki = 19460 nM
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CP0413125
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5-(6-oxo-1H-pyridazin-3-yl)-N-(5,6,7,8-tetrahydronaphthalen-1-yl)thiophene-2-sulfonamide
Show/Hide
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C18H17N3O3S2
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1
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| 1 |
Ki = 19810 nM
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CP0418218
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1,3-dimethyl-7-[3-(4-phenylpiperazin-1-yl)propyl]purine-2,6-dione;hydrochloride
Show/Hide
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C20H26N6O2
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1
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| 1 |
Ki = 20080 nM
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CP0418217
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7-[3-[4-(3-chlorophenyl)piperazin-1-yl]propyl]-1,3-dimethylpurine-2,6-dione;hydrochloride
Show/Hide
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C20H25ClN6O2
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1
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| 1 |
Ki = 20290 nM
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CP0382070
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1-[2-hydroxy-3-(4-phenylpiperazin-1-yl)propyl]-3-methyl-5,5-diphenylimidazolidine-2,4-dione
Show/Hide
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C29H32N4O3
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1
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| 1 |
Ki = 20410 nM
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CP0676509
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3-(4-{2-[4-(4-Chlorophenyl)-piperazin-1-yl]-ethyl}-piperidine-1-sulfonyl)-quinoline hydrochloride
Show/Hide
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C26H32Cl2N4O2S
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1
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| 1 |
Ki = 24840 nM
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CP0095010
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1-[5-[4-(2-fluorophenyl)piperazin-1-yl]pentyl]-3,5-dimethyl-5-phenylimidazolidine-2,4-dione;hydrochloride
Show/Hide
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C26H33FN4O2
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1
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| 1 |
Ki = 25520 nM
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CP0457198
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1-[3-[4-(2-methoxyphenyl)piperazin-1-yl]propyl]-3-methyl-5,5-diphenylimidazolidine-2,4-dione
Show/Hide
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C30H34N4O3
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1
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| 1 |
Ki = 29070 nM
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CP0568392
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1-[(3-chlorophenyl)methyl]-N-(oxan-4-yl)pyrrolo[3,2-c]quinolin-4-amine
Show/Hide
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C23H22ClN3O
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1
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| 1 |
Ki = 33060 nM
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CP0545512
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2-[[1-[(3-chlorophenyl)methyl]pyrrolo[3,2-c]quinolin-4-yl]-methylamino]ethanol
Show/Hide
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C21H20ClN3O
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1
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| 1 |
Ki = 40300 nM
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CP0085824
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2-[(4S,5R)-4-(hydroxymethyl)-5-methyl-4,5-dihydro-1,3-thiazol-2-yl]phenol
Show/Hide
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C11H13NO2S
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1
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| 1 |
Ki > 10 nM
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CP0110059
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2-[(4S,5S)-4-(hydroxymethyl)-5-methyl-4,5-dihydro-1,3-thiazol-2-yl]phenol
Show/Hide
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C11H13NO2S
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1
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| 1 |
Ki > 10 nM
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CP0475795
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2-[(4R,5R)-4-(hydroxymethyl)-5-methyl-4,5-dihydro-1,3-thiazol-2-yl]phenol
Show/Hide
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C11H13NO2S
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1
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| 1 |
Ki > 10 nM
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CP0372867
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7-chloro-3-methyl-3-phenylquinoline-2,4(1H,3H)-dione
Show/Hide
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C16H12ClNO2
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1
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| 1 |
Ki > 1000 nM
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CP0444330
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3-(4-(benzyloxy)-3-bromophenyl)-5,7-dichloro-3-methylquinoline-2,4(1H,3H)-dione
Show/Hide
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C23H16BrCl2NO3
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1
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| 1 |
Ki > 1000 nM
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CP0444331
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5,7-dichloro-3-(4-methoxy-3-nitrophenyl)-3-methylquinoline-2,4(1H,3H)-dione
Show/Hide
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C17H12Cl2N2O5
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1
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| 1 |
Ki > 1000 nM
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CP0444375
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6,7-dichloro-3-methyl-3-phenylquinoline-2,4(1H,3H)-dione
Show/Hide
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C16H11Cl2NO2
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1
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| 1 |
Ki > 1000 nM
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CP0454145
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3-methyl-3-phenylquinoline-2,4(1H,3H)-dione
Show/Hide
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C16H13NO2
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1
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| 1 |
Ki > 1000 nM
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CP0471141
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6,8-dibromo-3-methyl-3-phenylquinoline-2,4(1H,3H)-dione
Show/Hide
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C16H11Br2NO2
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1
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| 1 |
Ki > 1000 nM
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CP0471142
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5,7-dichloro-3-(4-hydroxy-3-nitrophenyl)-3-methylquinoline-2,4(1H,3H)-dione
Show/Hide
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C16H10Cl2N2O5
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1
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| 1 |
Ki > 1000 nM
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CP0552893
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5,7-dichloro-3-methyl-3-(4-nitrophenyl)quinoline-2,4(1H,3H)-dione
Show/Hide
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C16H10Cl2N2O4
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1
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| 1 |
Ki > 1000 nM
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CP0370109
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6-Chloro-imidazo[2,1-b]thiazole-5-sulfonic acid [1-(3-piperidin-1-yl-propyl)-1H-indol-5-yl]-amide
Show/Hide
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C21H24ClN5O2S2
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1
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| 1 |
Ki > 1000 nM
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CP0375945
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1-[1-(5-Bromo-2-methoxy-benzenesulfonyl)-piperidin-4-yl]-8-methyl-1,4-dihydro-benzo[d][1,3]oxazin-2-one
Show/Hide
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C21H23BrN2O5S
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1
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| 1 |
Ki > 1000 nM
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CP0376104
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N,N-diethyl-2-[5-(naphthalen-1-ylsulfonylamino)-1H-indol-3-yl]-2-oxoacetamide
Show/Hide
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C24H23N3O4S
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1
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| 1 |
Ki > 1000 nM
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CP0392407
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N,N-diethyl-2-oxo-2-[5-(quinolin-8-ylsulfonylamino)-1H-indol-3-yl]acetamide
Show/Hide
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C23H22N4O4S
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1
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| 1 |
Ki > 1000 nM
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CP0431325
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Biphenyl-4-sulfonic acid [1-(2-diethylamino-ethyl)-1H-indol-5-yl]-amide
Show/Hide
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C26H29N3O2S
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1
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| 1 |
Ki > 1000 nM
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CP0445698
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5-Chloro-3-methyl-benzo[b]thiophene-2-sulfonic acid [1-(2-dimethylamino-ethyl)-2-methyl-1H-indol-6-yl]-amide
Show/Hide
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C22H24ClN3O2S2
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1
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| 1 |
Ki > 1000 nM
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CP0445714
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2-[5-(5-Chloro-3-methyl-benzo[b]thiophene-2-sulfonylamino)-1H-indol-3-yl]-N,N-dimethyl-2-oxo-acetamide
Show/Hide
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C21H18ClN3O4S2
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1
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| 1 |
Ki > 1000 nM
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CP0502558
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N-[1-[2-(dimethylamino)ethyl]indol-5-yl]-1-phenylmethanesulfonamide
Show/Hide
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C19H23N3O2S
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1
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| 1 |
Ki > 1000 nM
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CP0430917
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[6-(4-methylpiperazin-1-yl)-1H-benzimidazol-2-yl]-naphthalen-1-ylmethanone
Show/Hide
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C23H22N4O
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1
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| 1 |
Ki > 1000 nM
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CP0439115
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[4-(4-methylpiperazin-1-yl)-1H-benzimidazol-2-yl]-phenylmethanone
Show/Hide
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C19H20N4O
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1
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| 1 |
Ki > 1000 nM
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CP0439116
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phenyl-(4-piperazin-1-yl-1H-benzimidazol-2-yl)methanone
Show/Hide
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C18H18N4O
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1
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| 1 |
Ki > 1000 nM
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CP0439118
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2-(2-Naphthylmethyl)-5-piperazin-1-yl-1H-benzimidazole
Show/Hide
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C22H22N4
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1
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| 1 |
Ki > 1000 nM
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CP0439119
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2-(1-Naphthylmethyl)-5-piperazin-1-yl-1H-benzimidazole
Show/Hide
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C22H22N4
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1
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| 1 |
Ki > 1000 nM
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CP0453092
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4-(4-Methyl-piperazin-1-yl)-1H-benzoimidazole
Show/Hide
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C12H16N4
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1
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| 1 |
Ki > 1000 nM
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CP0484606
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[6-(4-methylpiperazin-1-yl)-1H-benzimidazol-2-yl]-naphthalen-2-ylmethanone
Show/Hide
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C23H22N4O
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1
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| 1 |
Ki > 1000 nM
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CP0484612
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[6-(4-methylpiperazin-1-yl)-1H-benzimidazol-2-yl]-phenylmethanone
Show/Hide
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C19H20N4O
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1
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| 1 |
Ki > 1000 nM
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CP0484613
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2-Benzyl-5-(4-methylpiperazin-1-yl)-1H-benzimidazole
Show/Hide
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C19H22N4
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1
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| 1 |
Ki > 1000 nM
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CP0484878
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2-Naphthyl-(5-piperazin-1-yl-1H-benzimidazol-2-yl)methanone
Show/Hide
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C22H20N4O
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1
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| 1 |
Ki > 1000 nM
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CP0496953
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[4-(4-methylpiperazin-1-yl)-1H-benzimidazol-2-yl]-naphthalen-2-ylmethanone
Show/Hide
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C23H22N4O
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1
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| 1 |
Ki > 1000 nM
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CP0496956
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5-(4-Methylpiperazin-1-yl)-2-(2-naphthylmethyl)-1H-benzimidazole
Show/Hide
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C23H24N4
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1
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| 1 |
Ki > 1000 nM
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CP0498419
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2-Benzyl-5-piperazin-1-yl-1H-benzimidazole
Show/Hide
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C18H20N4
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1
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| 1 |
Ki > 1000 nM
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CP0510401
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5-(4-Methylpiperazin-1-yl)-2-(1-naphthylmethyl)-1H-benzimidazole
Show/Hide
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C23H24N4
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1
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| 1 |
Ki > 1000 nM
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CP0452472
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1-benzyl-5-(4-ethylpiperazin-1-yl-methyl)-1H-indole
Show/Hide
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C22H27N3
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1
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| 1 |
Ki > 1000 nM
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CP0505289
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1-Benzoyl-5-(4-methylpiperazin-1-yl-methyl)-1H-indole
Show/Hide
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C21H23N3O
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1
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| 1 |
Ki > 1000 nM
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CP0118231
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9-[5-[4-(2-hydroxyphenyl)piperazin-1-yl]pentyl]-1,3-dimethylpurino[7,8-a]pyrimidine-2,4,8-trione
Show/Hide
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C25H31N7O4
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1
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| 1 |
Ki > 1000 nM
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CP0475565
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N,N-dimethyl-4-[6-(4-methylpiperazin-1-yl)-1-(2-methylpropylsulfonyl)pyrrolo[2,3-b]pyridin-4-yl]benzamide
Show/Hide
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C25H33N5O3S
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1
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| 1 |
Ki > 2000 nM
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