General Information of the Compound
Compound ID
CP0848183
Compound Name
1-methyl-4-[1-(oxane-4-sulfonyl)-4-[4-(trifluoromethyl)phenyl]-1H-pyrrolo[2,3-b]pyridin-6-yl]piperazine
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Structure
Formula
C24H27F3N4O3S
Molecular Weight
508.566
Canonical SMILES
CN1CCN(c2cc(-c3ccc(C(F)(F)F)cc3)c3ccn(S(=O)(=O)C4CCOCC4)c3n2)CC1
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InChI
InChI=1S/C24H27F3N4O3S/c1-29-10-12-30(13-11-29)22-16-21(17-2-4-18(5-3-17)24(25,26)27)20-6-9-31(23(20)28-22)35(32,33)19-7-14-34-15-8-19/h2-6,9,16,19H,7-8,10-15H2,1H3
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InChIKey
YDIDXPKIMIHSET-UHFFFAOYSA-N
Physicochemical Property
logP
3.8308
Rotatable Bonds
4
Heavy Atom Count
35
Polar Areas
67.67
Hydrogen Bond Donor Count
0
Hydrogen Bond Acceptor Count
7
Complexity
35

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 127047537
ChEMBL ID
CHEMBL3799448
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT01354, 5-hydroxytryptamine receptor 6
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
Ki = 7 nM
   TI
   LI
   LO
   TS
Protein ID: PT01005, D(2) dopamine receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
Ki > 2000 nM
   TI
   LI
   LO
   TS