Brief Information of the Compound and Protein
Compound Name
 Compound Info 
3-(4-fluorophenyl)sulfonyl-5,7-dimethyl-2-methylsulfanylpyrazolo[1,5-a]pyrimidine
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 PubChem ID
CID: 44155876
SID: 85155759
Canonical SMILES
CSc1nn2c(C)cc(C)nc2c1S(=O)(=O)c1ccc(F)cc1
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Compound Formula C15H14FN3O2S2
Compound Structure
Protein Name
 Protein Info 
5-hydroxytryptamine receptor 6
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
>
Small molecule receptor (family A GPCR)
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Monoamine receptor
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Serotonin receptor
Uniprot ID
P50406
Gene Name
HTR6
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293
 Cell Line Info 
Homo sapiens (Human)  1
1
Ki = 6.761 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 IC50 < 10 nM
2 IC50 = 112 nM