General Information of the Compound
Compound ID
CP0116953
Compound Name
1,1'-sulfonylbis(4-aminobenzene)
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Synonyms
(4-sulfanilylphenyl)amine
1,1'-Sulfonylbis(4-aminobenzene)
1,1'-Sulfonylbis[4-aminobenzene]
1,1'-Sulphonylbis(4-aminobenzene)
4,4' Diaminophenyl Sulfone
4,4'-Dapsone
4,4'-Diaminodiphenyl sulfone
4,4'-Diaminodiphenyl suphone
4,4'-Diaminodiphenylsulfone
4,4'-Sulfonylbisaniline
4,4'-Sulfonylbisbenzamine
4,4'-Sulfonylbisbenzenamine
4,4'-Sulfonyldianiline;4,4'-Sulfonyldianiline (Dapsone)
4,4'-Sulphonylbisbenzamine
4,4'-Sulphonylbisbenzenamine
4,4'-Sulphonyldianiline
4,4'-diaminophenyl sulfone
4,4-Diaminodifenylsulfon
4,4-Diaminodifenylsulfon [Czech]
4,4-Sulfonyldianiline
4-(4-aminophenyl)sulfonylaniline
4-Aminop henyl sulfone
4-Aminophenyl sulfone
4-Aminophenylsulfone
4-[(4-aminobenzene)sulfonyl]aniline
4-[(4-aminophenyl)sulfonyl]aniline
ALBB-005917
AZT + Dapsone cominbation
Aczone
Aczone (TN)
Araldite HT
Araldite HT 976
Atrisone
Avlosulfon
Avlosulfone
Avlosulphone
Avsulfor
Bis(4-aminophenyl) sulfone
Bis(4-aminophenyl)sulfone
Bis(4-aminophenyl)sulphone
Bis(p-aminophenyl) sulfone
Bis(p-aminophenyl)sulphone
Croysulfone
Croysulphone
D SS
DADPS
DDS
DDS (pharmaceutical)
DDS, diaphenylsulfone
DDS, pharmaceutical
DSS (VAN)
Dapsoderm-X
Dapson
Dapson-Fatol
Dapsona
Dapsona [INN-Spanish]
Dapsone
Dapsone (USP)
Dapsone [USAN:BAN]
Dapsonum
Dapsonum [INN-Latin];Diamino-diphenyl sulphone
Di(4-aminophenyl) sulfone
Di(4-aminophenyl)sulfone
Di(4-aminophenyl)sulphone
Di(p-aminophenyl) sulfone
Di(p-aminophenyl)sulphone
Diamino-4,4'-diphenyl sulfone
Diamino-4,4'-diphenyl sulphone
Diaminodifenilsulfona
Diaminodifenilsulfona [Spanish]
Diaminodiphenyl sulfone;Fatol Brand of Dapsone
Diaminodiphenylsulfone
Diaphenylsulfon
Diaphenylsulfone
Diaphenylsulfone (JAN)
Diaphenylsulphon
Diaphenylsulphone
Diphenasone
Diphone
Disulone
Dubronax
Dubronaz
Dumitone
Eporal
F 1358
HT 976
HY 976
Hardener HT 976
IN-201
Metabolite C
Mex-America Brand of Dapsone
N, N'-Diphenyl sulfondiamide
N,N'-Diphenyl sulfondiamide
Novophone
Orsade Brand of Dapsone
P, p'-Sulfonyldianiline
P,p'-Diaminodiphenyl sulfone
P,p'-sulfonyldianiline
P,p-Diaminodiphenyl sulphone
P,p-Sulfonylbisbenzamine
P,p-Sulfonylbisbenzenamine
P,p-Sulphonylbisbenzamine
P,p-Sulphonylbisbenzenamine
P,p-Sulphonyldianiline
P-Aminophenyl sulfone
Protogen
Sulfadione
Sulfanona-mae
Sulfon-mere
Sulfona
Sulfona-MAE
Sulfone ucb
Sulfone, 4,4'-Diaminophenyl
Sulfonyldianiline
Sulphadione
Sulphon-mere
Sulphonyldianiline
Sumicure S
Tarimyl
Udolac
W R 448
WR 448
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Structure
Formula
C12H12N2O2S
Molecular Weight
248.307
Canonical SMILES
Nc1ccc(cc1)S(=O)(=O)c1ccc(N)cc1
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InChI
InChI=1S/C12H12N2O2S/c13-9-1-5-11(6-2-9)17(15,16)12-7-3-10(14)4-8-12/h1-8H,13-14H2
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InChIKey
MQJKPEGWNLWLTK-UHFFFAOYSA-N
CAS
80-08-0
Physicochemical Property
logP
1.6838
Rotatable Bonds
2
Heavy Atom Count
17
Polar Areas
86.18
Hydrogen Bond Donor Count
2
Hydrogen Bond Acceptor Count
4
Complexity
17

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 2955
SID: 15196656
ChEMBL ID
CHEMBL1043
DrugBank ID
DB00250
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT01354, 5-hydroxytryptamine receptor 6
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
Ki = 183 nM
   TI
   LI
   LO
   TS
Clinical Information about the Compound
Drug 1 ( Dapsone )
Drug Name Dapsone
Indication
Pneumocystis pneumonia
Approved