Brief Information of the Compound and Protein
Compound Name
 Compound Info 
5,7-Dimethyl-2-(ethylthio)-3-phenylsulfonyl-pyrazolo[1,5-a]pyrimidine
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 PubChem ID
CID: 44155875
SID: 85155758
Canonical SMILES
CCSc1nn2c(C)cc(C)nc2c1S(=O)(=O)c1ccccc1
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Compound Formula C16H17N3O2S2
Compound Structure
Protein Name
 Protein Info 
5-hydroxytryptamine receptor 6
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
>
Small molecule receptor (family A GPCR)
>
Monoamine receptor
>
Serotonin receptor
Uniprot ID
P50406
Gene Name
HTR6
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293
 Cell Line Info 
Homo sapiens (Human)  1
1
Ki = 1.91 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 IC50 = 50 nM