| Compound ID |
Compound Name |
Compound Formula |
|
CP0466200
|
2-methyl-4-[(6-methyl-2-phenylpyrimidin-4-yl)amino]benzonitrile
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|
C19H16N4
|
5
|
| 1 |
Activity = 17.25 nM
|
|
|
| 2 |
Activity = 50 nM
|
|
|
| 3 |
EC50 = 11 nM
|
|
|
| 4 |
IC50 = 93.5 nM
|
|
|
| 5 |
IC50 = 175 nM
|
|
|
|
CP0393143
|
2-(3,4-dimethoxyphenyl)-N-(4-nitrophenyl)quinazolin-4-amine
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|
C22H18N4O4
|
4
|
| 1 |
EC50 = 7.4 nM
|
|
|
| 2 |
EC50 = 12.7 nM
|
|
|
| 3 |
IC50 = 300 nM
|
|
|
| 4 |
IC50 = 320 nM
|
|
|
|
CP0393144
|
N-(4-bromo-3-methoxyphenyl)-2-(3,4-dimethoxyphenyl)quinazolin-4-amine
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|
C23H20BrN3O3
|
3
|
| 1 |
EC50 = 9.7 nM
|
|
|
| 2 |
EC50 = 15.6 nM
|
|
|
| 3 |
IC50 = 47.5 nM
|
|
|
|
CP0387310
|
N-(4-nitrophenyl)-2-pyridin-3-ylquinazolin-4-amine
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|
C19H13N5O2
|
3
|
| 1 |
EC50 = 12.6 nM
|
|
|
| 2 |
EC50 = 21.2 nM
|
|
|
| 3 |
IC50 = 64.1 nM
|
|
|
|
CP0487494
|
2-bromo-4-[(6-methyl-2-phenylpyrimidin-4-yl)amino]benzonitrile
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|
C18H13BrN4
|
3
|
| 1 |
EC50 = 15 nM
|
|
|
| 2 |
IC50 = 59.4 nM
|
|
|
| 3 |
IC50 = 119 nM
|
|
|
|
CP0466208
|
4-[(6-methyl-2-phenylpyrimidin-4-yl)amino]-2-(trifluoromethyl)benzonitrile
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|
C19H13F3N4
|
3
|
| 1 |
EC50 = 15.2 nM
|
|
|
| 2 |
IC50 = 69.3 nM
|
|
|
| 3 |
IC50 = 385 nM
|
|
|
|
CP0425266
|
4-[[2-phenyl-6-(propylamino)pyrimidin-4-yl]amino]benzonitrile
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|
C20H19N5
|
5
|
| 1 |
EC50 = 15.3 nM
|
|
|
| 2 |
GI50 = 334 nM
|
|
|
| 3 |
GI50 = 603 nM
|
|
|
| 4 |
GI50 = 2780 nM
|
|
|
| 5 |
IC50 = 293 nM
|
|
|
|
CP0425267
|
4-[[2-phenyl-6-(pyridin-2-ylmethylamino)pyrimidin-4-yl]amino]benzonitrile
Show/Hide
|
C23H18N6
|
5
|
| 1 |
EC50 = 15.5 nM
|
|
|
| 2 |
GI50 = 334 nM
|
|
|
| 3 |
GI50 = 616 nM
|
|
|
| 4 |
GI50 = 2960 nM
|
|
|
| 5 |
IC50 = 210 nM
|
|
|
|
CP0472565
|
6-methyl-N-(4-nitrophenyl)-2-phenylpyrimidin-4-amine
Show/Hide
|
C17H14N4O2
|
3
|
| 1 |
EC50 = 15.9 nM
|
|
|
| 2 |
IC50 = 52.2 nM
|
|
|
| 3 |
IC50 = 156 nM
|
|
|
|
CP0466206
|
N-(6-methyl-2-phenylpyrimidin-4-yl)quinolin-6-amine
Show/Hide
|
C20H16N4
|
2
|
| 1 |
EC50 = 16.4 nM
|
|
|
| 2 |
IC50 = 151 nM
|
|
|
|
CP0425259
|
4-[[2-phenyl-6-(propan-2-ylamino)pyrimidin-4-yl]amino]benzonitrile
Show/Hide
|
C20H19N5
|
5
|
| 1 |
EC50 = 18 nM
|
|
|
| 2 |
GI50 = 314 nM
|
|
|
| 3 |
GI50 = 717 nM
|
|
|
| 4 |
GI50 = 2930 nM
|
|
|
| 5 |
IC50 = 763 nM
|
|
|
|
CP0440750
|
N-(3-fluorophenyl)-2-(3-methoxyphenyl)-6-nitroquinazolin-4-amine
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|
C21H15FN4O3
|
3
|
| 1 |
EC50 = 19.5 nM
|
|
|
| 2 |
EC50 = 51.1 nM
|
|
|
| 3 |
IC50 = 23.4 nM
|
|
|
|
CP0548061
|
2-fluoro-5-[(6-methyl-2-phenylpyrimidin-4-yl)amino]benzonitrile
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|
C18H13FN4
|
3
|
| 1 |
EC50 = 20.9 nM
|
|
|
| 2 |
IC50 = 86.1 nM
|
|
|
| 3 |
IC50 = 307 nM
|
|
|
|
CP0534852
|
4-[[6-(methylamino)-2-phenylpyrimidin-4-yl]amino]benzonitrile
Show/Hide
|
C18H15N5
|
5
|
| 1 |
EC50 = 21.7 nM
|
|
|
| 2 |
GI50 = 407 nM
|
|
|
| 3 |
GI50 = 917 nM
|
|
|
| 4 |
GI50 = 3620 nM
|
|
|
| 5 |
IC50 = 141 nM
|
|
|
|
CP0427176
|
3-[[6-nitro-2-[3-(trifluoromethyl)phenyl]quinazolin-4-yl]amino]phenol
Show/Hide
|
C21H13F3N4O3
|
2
|
| 1 |
EC50 = 21.8 nM
|
|
|
| 2 |
IC50 = 27.6 nM
|
|
|
|
CP0420361
|
4-[(6-methyl-2-phenylpyrimidin-4-yl)amino]-2-nitrophenol
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|
C17H14N4O3
|
3
|
| 1 |
EC50 = 22 nM
|
|
|
| 2 |
EC50 = 62.3 nM
|
|
|
| 3 |
IC50 = 98.8 nM
|
|
|
|
CP0425271
|
4-[[6-(benzylamino)-2-phenylpyrimidin-4-yl]amino]benzonitrile
Show/Hide
|
C24H19N5
|
5
|
| 1 |
EC50 = 25.5 nM
|
|
|
| 2 |
GI50 = 421 nM
|
|
|
| 3 |
GI50 = 1110 nM
|
|
|
| 4 |
GI50 = 3620 nM
|
|
|
| 5 |
IC50 = 283 nM
|
|
|
|
CP0463432
|
N-(4-methoxyphenyl)-2-phenylpyrido[2,3-d]pyrimidin-4-amine
Show/Hide
|
C20H16N4O
|
3
|
| 1 |
EC50 = 29.4 nM
|
|
|
| 2 |
GI50 = 20.9 nM
|
|
|
| 3 |
IC50 = 238 nM
|
|
|
|
CP0424839
|
4-[[6-(butylamino)-2-phenylpyrimidin-4-yl]amino]benzonitrile
Show/Hide
|
C21H21N5
|
5
|
| 1 |
EC50 = 29.8 nM
|
|
|
| 2 |
GI50 = 731 nM
|
|
|
| 3 |
GI50 = 1680 nM
|
|
|
| 4 |
GI50 = 5810 nM
|
|
|
| 5 |
IC50 = 500 nM
|
|
|
|
CP0478881
|
2-nitro-4-[(6-nitro-2-phenylquinazolin-4-yl)amino]phenol
Show/Hide
|
C20H13N5O5
|
2
|
| 1 |
EC50 = 34 nM
|
|
|
| 2 |
IC50 = 37.4 nM
|
|
|
|
CP0389518
|
N,2-diphenylpyrido[2,3-d]pyrimidin-4-amine
Show/Hide
|
C19H14N4
|
3
|
| 1 |
EC50 = 37.1 nM
|
|
|
| 2 |
GI50 = 8.61 nM
|
|
|
| 3 |
IC50 = 149 nM
|
|
|
|
CP0425269
|
4-[(2,6-diphenylpyrimidin-4-yl)amino]benzonitrile
Show/Hide
|
C23H16N4
|
5
|
| 1 |
EC50 = 40.5 nM
|
|
|
| 2 |
GI50 = 367 nM
|
|
|
| 3 |
GI50 = 1720 nM
|
|
|
| 4 |
GI50 = 4440 nM
|
|
|
| 5 |
IC50 = 4410 nM
|
|
|
|
CP0528180
|
4-[(2-phenylquinazolin-4-yl)amino]benzonitrile
Show/Hide
|
C21H14N4
|
6
|
| 1 |
EC50 = 41 nM
|
|
|
| 2 |
EC50 = 53 nM
|
|
|
| 3 |
GI50 = 4.41 nM
|
|
|
| 4 |
IC50 = 69.9 nM
|
|
|
| 5 |
IC50 = 71.4 nM
|
|
|
| 6 |
IC50 = 84.5 nM
|
|
|
|
CP0444105
|
4-[(6-anilino-2-phenylpyrimidin-4-yl)amino]benzonitrile
Show/Hide
|
C23H17N5
|
5
|
| 1 |
EC50 = 43.5 nM
|
|
|
| 2 |
GI50 = 333 nM
|
|
|
| 3 |
GI50 = 1640 nM
|
|
|
| 4 |
GI50 = 4130 nM
|
|
|
| 5 |
IC50 = 169 nM
|
|
|
|
CP0516921
|
4-[[2-phenyl-6-(pyridin-3-ylmethylamino)pyrimidin-4-yl]amino]benzonitrile
Show/Hide
|
C23H18N6
|
5
|
| 1 |
EC50 = 44.3 nM
|
|
|
| 2 |
GI50 = 415 nM
|
|
|
| 3 |
GI50 = 1730 nM
|
|
|
| 4 |
GI50 = 4660 nM
|
|
|
| 5 |
IC50 = 373 nM
|
|
|
|
CP0444264
|
3-[(6-nitro-2-pyridin-4-ylquinazolin-4-yl)amino]benzonitrile
Show/Hide
|
C20H12N6O2
|
2
|
| 1 |
EC50 = 48.3 nM
|
|
|
| 2 |
IC50 = 63.8 nM
|
|
|
|
CP0389669
|
2-nitro-4-[[6-nitro-2-[3-(trifluoromethyl)phenyl]quinazolin-4-yl]amino]phenol
Show/Hide
|
C21H12F3N5O5
|
2
|
| 1 |
EC50 = 57 nM
|
|
|
| 2 |
IC50 = 33 nM
|
|
|
|
CP0444115
|
4-[[2-phenyl-6-(3-phenylpropylamino)pyrimidin-4-yl]amino]benzonitrile
Show/Hide
|
C26H23N5
|
5
|
| 1 |
EC50 = 67 nM
|
|
|
| 2 |
GI50 = 727 nM
|
|
|
| 3 |
GI50 = 3180 nM
|
|
|
| 4 |
GI50 = 6550 nM
|
|
|
| 5 |
IC50 = 96 nM
|
|
|
|
CP0389584
|
N-(4-methoxyphenyl)-6-nitro-2-pyridin-4-ylquinazolin-4-amine
Show/Hide
|
C20H15N5O3
|
2
|
| 1 |
EC50 = 71.2 nM
|
|
|
| 2 |
IC50 = 75.5 nM
|
|
|
|
CP0444106
|
4-[[2-phenyl-6-(pyridin-4-ylmethylamino)pyrimidin-4-yl]amino]benzonitrile
Show/Hide
|
C23H18N6
|
5
|
| 1 |
EC50 = 72.5 nM
|
|
|
| 2 |
GI50 = 365 nM
|
|
|
| 3 |
GI50 = 2090 nM
|
|
|
| 4 |
GI50 = 4150 nM
|
|
|
| 5 |
IC50 = 435 nM
|
|
|
|
CP0469970
|
3-[(2-pyridin-3-ylquinazolin-4-yl)amino]benzonitrile
Show/Hide
|
C20H13N5
|
2
|
| 1 |
EC50 = 85 nM
|
|
|
| 2 |
IC50 = 108 nM
|
|
|
|
CP0095983
|
(1s,3s)-3-(8-amino-1-(2-phenylquinolin-7-yl)imidazo[1,5-a]pyrazin-3-yl)-1-methylcyclobutanol
Show/Hide
|
C26H23N5O
|
1
|
| 1 |
EC50 = 104 nM
|
|
|
|
CP0327876
|
N-(3,4-dimethoxyphenyl)-2-[4-[(E)-3-(3,4,5-trimethoxyphenyl)prop-2-enoyl]phenoxy]acetamide
Show/Hide
|
C28H29NO8
|
1
|
| 1 |
EC50 = 107 nM
|
|
|
|
CP0430189
|
2-nitro-4-[(2-phenylquinazolin-4-yl)amino]phenol
Show/Hide
|
C20H14N4O3
|
6
|
| 1 |
EC50 = 120 nM
|
|
|
| 2 |
EC50 = 130 nM
|
|
|
| 3 |
GI50 = 68.4 nM
|
|
|
| 4 |
IC50 = 80 nM
|
|
|
| 5 |
IC50 = 81.1 nM
|
|
|
| 6 |
IC50 = 113 nM
|
|
|
|
CP0444112
|
4-[[6-(2-hydroxyanilino)-2-phenylpyrimidin-4-yl]amino]benzonitrile
Show/Hide
|
C23H17N5O
|
5
|
| 1 |
EC50 = 147 nM
|
|
|
| 2 |
GI50 = 441 nM
|
|
|
| 3 |
GI50 = 3070 nM
|
|
|
| 4 |
GI50 = 4620 nM
|
|
|
| 5 |
IC50 = 223 nM
|
|
|
|
CP0425272
|
4-[[6-(4-hydroxyanilino)-2-phenylpyrimidin-4-yl]amino]benzonitrile
Show/Hide
|
C23H17N5O
|
5
|
| 1 |
EC50 = 171 nM
|
|
|
| 2 |
GI50 = 325 nM
|
|
|
| 3 |
GI50 = 2570 nM
|
|
|
| 4 |
GI50 = 3150 nM
|
|
|
| 5 |
IC50 = 387 nM
|
|
|
|
CP0425619
|
4-[[6-(3-hydroxyanilino)-2-phenylpyrimidin-4-yl]amino]benzonitrile
Show/Hide
|
C23H17N5O
|
5
|
| 1 |
EC50 = 181 nM
|
|
|
| 2 |
GI50 = 563 nM
|
|
|
| 3 |
GI50 = 3280 nM
|
|
|
| 4 |
GI50 = 4240 nM
|
|
|
| 5 |
IC50 = 608 nM
|
|
|
|
CP0425270
|
4-[[2-phenyl-6-(4-phenylbutylamino)pyrimidin-4-yl]amino]benzonitrile
Show/Hide
|
C27H25N5
|
5
|
| 1 |
EC50 = 187 nM
|
|
|
| 2 |
GI50 = 494 nM
|
|
|
| 3 |
GI50 = 3750 nM
|
|
|
| 4 |
GI50 = 4840 nM
|
|
|
| 5 |
IC50 = 147 nM
|
|
|
|
CP0016777
|
2-bromo-4-(6,7-dimethoxyquinazolin-4-ylamino)phenol
Show/Hide
|
C16H14BrN3O3
|
1
|
| 1 |
EC50 = 189 nM
|
|
|
|
CP0425268
|
4-[[6-(4-cyanoanilino)-2-phenylpyrimidin-4-yl]amino]benzonitrile
Show/Hide
|
C24H16N6
|
5
|
| 1 |
EC50 = 231 nM
|
|
|
| 2 |
GI50 = 563 nM
|
|
|
| 3 |
GI50 = 4080 nM
|
|
|
| 4 |
GI50 = 5120 nM
|
|
|
| 5 |
IC50 = 133 nM
|
|
|
|
CP0389267
|
4-[(2-phenylpyrido[2,3-d]pyrimidin-4-yl)amino]benzonitrile
Show/Hide
|
C20H13N5
|
2
|
| 1 |
EC50 = 270 nM
|
|
|
| 2 |
IC50 = 1210 nM
|
|
|
|
CP0415982
|
2-[3-(3,4-dimethoxyphenyl)-4-oxochromen-2-yl]oxy-N-naphthalen-1-ylacetamide
Show/Hide
|
C29H23NO6
|
1
|
| 1 |
EC50 = 446 nM
|
|
|
|
CP0256321
|
2-[4-[(E)-3-(2,6-difluorophenyl)prop-2-enoyl]phenoxy]-N-(3,4-dimethoxyphenyl)acetamide
Show/Hide
|
C25H21F2NO5
|
1
|
| 1 |
EC50 = 448 nM
|
|
|
|
CP0415981
|
(E)-1-(4-hydroxy-3-methoxyphenyl)-3-(3,4,5-trimethoxyphenyl)prop-2-en-1-one
Show/Hide
|
C19H20O6
|
1
|
| 1 |
EC50 = 512 nM
|
|
|
|
CP0391069
|
2-[3-(4-methoxyphenyl)-4-oxochromen-2-yl]oxy-N-naphthalen-1-ylacetamide
Show/Hide
|
C28H21NO5
|
1
|
| 1 |
EC50 = 793 nM
|
|
|
|
CP0124997
|
N-(1,3-benzodioxol-5-ylmethyl)-2-[4-[(E)-3-(3,4,5-trimethoxyphenyl)prop-2-enoyl]phenoxy]acetamide
Show/Hide
|
C28H27NO8
|
1
|
| 1 |
EC50 = 989 nM
|
|
|
|
CP0420980
|
N-(1-oxo-3H-2-benzofuran-5-yl)-2-[3-[(E)-3-phenylprop-2-enoyl]phenoxy]acetamide
Show/Hide
|
C25H19NO5
|
1
|
| 1 |
EC50 = 1170 nM
|
|
|
|
CP0391067
|
2-[2-(2-chlorophenyl)-4-oxochromen-3-yl]oxy-N-(1-oxo-3H-2-benzofuran-5-yl)acetamide
Show/Hide
|
C25H16ClNO6
|
1
|
| 1 |
EC50 = 1220 nM
|
|
|
|
CP0391063
|
(E)-1-(4-hydroxyphenyl)-3-(4-propoxyphenyl)prop-2-en-1-one
Show/Hide
|
C18H18O3
|
1
|
| 1 |
EC50 = 1250 nM
|
|
|
|
CP0391014
|
2-[4-(7-methyl-2-pyridin-3-yl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-yl)piperazin-1-yl]-2-phenylacetamide
Show/Hide
|
C28H30N6OS
|
5
|
| 1 |
EC50 = 1310 nM
|
|
|
| 2 |
GI50 = 662 nM
|
|
|
| 3 |
GI50 = 2440 nM
|
|
|
| 4 |
GI50 = 3080 nM
|
|
|
| 5 |
IC50 = 2380 nM
|
|
|
|
CP0201944
|
N-(3,4-dimethoxyphenyl)-2-[4-[(E)-3-(3-methoxyphenyl)prop-2-enoyl]phenoxy]acetamide
Show/Hide
|
C26H25NO6
|
1
|
| 1 |
EC50 = 1390 nM
|
|
|
|
CP0412741
|
4-methoxy-N-[2-[2-(6-methoxypyridin-3-yl)tetrazol-5-yl]phenyl]benzamide
Show/Hide
|
C21H18N6O3
|
5
|
| 1 |
GI50 = 190 nM
|
|
|
| 2 |
GI50 = 202 nM
|
|
|
| 3 |
GI50 = 483 nM
|
|
|
| 4 |
GI50 = 802 nM
|
|
|
| 5 |
IC50 = 61.6 nM
|
|
|
|
CP0517984
|
4-methoxy-N-[2-[5-(4-methoxyphenyl)-1,3,4-oxadiazol-2-yl]phenyl]benzamide
Show/Hide
|
C23H19N3O4
|
5
|
| 1 |
GI50 = 237 nM
|
|
|
| 2 |
GI50 = 396 nM
|
|
|
| 3 |
GI50 = 927 nM
|
|
|
| 4 |
GI50 = 1210 nM
|
|
|
| 5 |
IC50 = 438 nM
|
|
|
|
CP0412739
|
N-[2-(5-phenyl-1,3,4-oxadiazol-2-yl)phenyl]benzamide
Show/Hide
|
C21H15N3O2
|
5
|
| 1 |
GI50 = 272 nM
|
|
|
| 2 |
GI50 = 278 nM
|
|
|
| 3 |
GI50 = 478 nM
|
|
|
| 4 |
GI50 = 1010 nM
|
|
|
| 5 |
IC50 = 112 nM
|
|
|
|
CP0412385
|
N-[2-(4-phenyltriazol-1-yl)phenyl]benzamide
Show/Hide
|
C21H16N4O
|
5
|
| 1 |
GI50 = 299 nM
|
|
|
| 2 |
GI50 = 436 nM
|
|
|
| 3 |
GI50 = 656 nM
|
|
|
| 4 |
GI50 = 982 nM
|
|
|
| 5 |
IC50 = 15300 nM
|
|
|
|
CP0420847
|
3-[[2-(1H-pyrrol-2-yl)quinazolin-4-yl]amino]benzonitrile
Show/Hide
|
C19H13N5
|
2
|
| 1 |
IC50 = 7.98 nM
|
|
|
| 2 |
IC50 = 156 nM
|
|
|
|
CP0409100
|
4-[[2-(3-methoxyphenyl)-6-nitroquinazolin-4-yl]amino]benzonitrile
Show/Hide
|
C22H15N5O3
|
1
|
| 1 |
IC50 = 27.8 nM
|
|
|
|
CP0389588
|
N-(3,4-dimethoxyphenyl)-6-nitro-2-[3-(trifluoromethyl)phenyl]quinazolin-4-amine
Show/Hide
|
C23H17F3N4O4
|
1
|
| 1 |
IC50 = 30.2 nM
|
|
|
|
CP0389587
|
N-(3-methoxyphenyl)-6-nitro-2-phenylquinazolin-4-amine
Show/Hide
|
C21H16N4O3
|
1
|
| 1 |
IC50 = 33.1 nM
|
|
|
|
CP0389672
|
N-(3,4-dimethoxyphenyl)-6-nitro-2-phenylquinazolin-4-amine
Show/Hide
|
C22H18N4O4
|
1
|
| 1 |
IC50 = 37 nM
|
|
|
|
CP0482661
|
N-[3-[[6-nitro-2-[3-(trifluoromethyl)phenyl]quinazolin-4-yl]amino]phenyl]acetamide
Show/Hide
|
C23H16F3N5O3
|
1
|
| 1 |
IC50 = 44.8 nM
|
|
|
|
CP0548216
|
N-(3-fluorophenyl)-6-nitro-2-[3-(trifluoromethyl)phenyl]quinazolin-4-amine
Show/Hide
|
C21H12F4N4O2
|
1
|
| 1 |
IC50 = 44.8 nM
|
|
|
|
CP0466717
|
3-[(2-thiophen-2-ylquinazolin-4-yl)amino]benzonitrile
Show/Hide
|
C19H12N4S
|
2
|
| 1 |
IC50 = 45.3 nM
|
|
|
| 2 |
IC50 = 178 nM
|
|
|
|
CP0435284
|
N-(3-methoxyphenyl)-6-nitro-2-pyridin-3-ylquinazolin-4-amine
Show/Hide
|
C20H15N5O3
|
1
|
| 1 |
IC50 = 47 nM
|
|
|
|
CP0427813
|
3-nitro-N-(2-phenylquinazolin-4-yl)benzamide
Show/Hide
|
C21H14N4O3
|
2
|
| 1 |
IC50 = 47.3 nM
|
|
|
| 2 |
IC50 = 54.5 nM
|
|
|
|
CP0435285
|
4-[(6-nitro-2-phenylquinazolin-4-yl)amino]benzonitrile
Show/Hide
|
C21H13N5O2
|
1
|
| 1 |
IC50 = 48.1 nM
|
|
|
|
CP0389668
|
3-[(6-nitro-2-phenylquinazolin-4-yl)amino]benzonitrile
Show/Hide
|
C21H13N5O2
|
1
|
| 1 |
IC50 = 48.2 nM
|
|
|
|
CP0389585
|
6-nitro-2-phenyl-N-[3-(trifluoromethyl)phenyl]quinazolin-4-amine
Show/Hide
|
C21H13F3N4O2
|
1
|
| 1 |
IC50 = 49.1 nM
|
|
|
|
CP0478880
|
N-(3-fluorophenyl)-6-nitro-2-phenylquinazolin-4-amine
Show/Hide
|
C20H13FN4O2
|
1
|
| 1 |
IC50 = 51.5 nM
|
|
|
|
CP0466626
|
2-(3,4-dimethoxyphenyl)-6-nitro-N-[3-(trifluoromethyl)phenyl]quinazolin-4-amine
Show/Hide
|
C23H17F3N4O4
|
1
|
| 1 |
IC50 = 57.2 nM
|
|
|
|
CP0440751
|
N-(4-methoxyphenyl)-6-nitro-2-pyridin-3-ylquinazolin-4-amine
Show/Hide
|
C20H15N5O3
|
1
|
| 1 |
IC50 = 57.7 nM
|
|
|
|
CP0553309
|
N-(3-chloro-4-nitrophenyl)-6-methyl-2-phenylpyrimidin-4-amine
Show/Hide
|
C17H13ClN4O2
|
2
|
| 1 |
IC50 = 58.9 nM
|
|
|
| 2 |
IC50 = 228 nM
|
|
|
|
CP0538861
|
N-(3-methoxyphenyl)-6-nitro-2-[3-(trifluoromethyl)phenyl]quinazolin-4-amine
Show/Hide
|
C22H15F3N4O3
|
1
|
| 1 |
IC50 = 59 nM
|
|
|
|
CP0409037
|
6-nitro-N-phenyl-2-[3-(trifluoromethyl)phenyl]quinazolin-4-amine
Show/Hide
|
C21H13F3N4O2
|
1
|
| 1 |
IC50 = 59.6 nM
|
|
|
|
CP0541451
|
6-nitro-N-(4-nitrophenyl)-2-[3-(trifluoromethyl)phenyl]quinazolin-4-amine
Show/Hide
|
C21H12F3N5O4
|
1
|
| 1 |
IC50 = 61.4 nM
|
|
|
|
CP0402414
|
N-[2-(2-phenyltetrazol-5-yl)phenyl]benzamide
Show/Hide
|
C20H15N5O
|
2
|
| 1 |
IC50 = 64 nM
|
|
|
| 2 |
IC50 = 66.9 nM
|
|
|
|
CP0398050
|
4-methoxy-N-[2-[2-(4-propylphenyl)tetrazol-5-yl]phenyl]benzamide
Show/Hide
|
C24H23N5O2
|
1
|
| 1 |
IC50 = 64.2 nM
|
|
|
|
CP0389667
|
3-[(6-nitro-2-phenylquinazolin-4-yl)amino]phenol
Show/Hide
|
C20H14N4O3
|
1
|
| 1 |
IC50 = 65.3 nM
|
|
|
|
CP0548215
|
6-nitro-N-(3-nitrophenyl)-2-[3-(trifluoromethyl)phenyl]quinazolin-4-amine
Show/Hide
|
C21H12F3N5O4
|
1
|
| 1 |
IC50 = 66.3 nM
|
|
|
|
CP0443240
|
N-(4-nitrophenyl)-2-phenylquinazolin-4-amine
Show/Hide
|
C20H14N4O2
|
2
|
| 1 |
IC50 = 69.6 nM
|
|
|
| 2 |
IC50 = 970 nM
|
|
|
|
CP0398098
|
4-methoxy-N-[2-[2-[4-(trifluoromethyl)phenyl]tetrazol-5-yl]phenyl]benzamide
Show/Hide
|
C22H16F3N5O2
|
1
|
| 1 |
IC50 = 73 nM
|
|
|
|
CP0380945
|
2-(3,4-dimethoxyphenyl)-N-(3-nitrophenyl)quinazolin-4-amine
Show/Hide
|
C22H18N4O4
|
2
|
| 1 |
IC50 = 76 nM
|
|
|
| 2 |
IC50 = 92 nM
|
|
|
|
CP0427812
|
4-nitro-N-(2-phenylquinazolin-4-yl)benzamide
Show/Hide
|
C21H14N4O3
|
2
|
| 1 |
IC50 = 77.3 nM
|
|
|
| 2 |
IC50 = 93.1 nM
|
|
|
|
CP0529206
|
N-[4-methoxy-2-[2-(4-methoxyphenyl)tetrazol-5-yl]phenyl]-4-(trifluoromethyl)benzamide
Show/Hide
|
C23H18F3N5O3
|
1
|
| 1 |
IC50 = 77.4 nM
|
|
|
|
CP0542831
|
N-[3-[(6-nitro-2-phenylquinazolin-4-yl)amino]phenyl]acetamide
Show/Hide
|
C22H17N5O3
|
1
|
| 1 |
IC50 = 78.7 nM
|
|
|
|
CP0390499
|
N-[2-[2-(3-methoxyphenyl)tetrazol-5-yl]phenyl]-4-nitrobenzamide
Show/Hide
|
C21H16N6O4
|
1
|
| 1 |
IC50 = 78.9 nM
|
|
|
|
CP0398097
|
N-[2-[2-(4-methoxyphenyl)tetrazol-5-yl]phenyl]-4-propylbenzamide
Show/Hide
|
C24H23N5O2
|
1
|
| 1 |
IC50 = 79.4 nM
|
|
|
|
CP0393140
|
N-(4-methylsulfanylphenyl)-2-(3-nitrophenyl)quinazolin-4-amine
Show/Hide
|
C21H16N4O2S
|
1
|
| 1 |
IC50 = 88.6 nM
|
|
|
|
CP0516014
|
N-[2-[5-(4-methoxyphenyl)-1,3,4-oxadiazol-2-yl]phenyl]-4-(trifluoromethyl)benzamide
Show/Hide
|
C23H16F3N3O3
|
1
|
| 1 |
IC50 = 90 nM
|
|
|
|
CP0383541
|
N-(3-methylsulfanylphenyl)-2-(3-nitrophenyl)quinazolin-4-amine
Show/Hide
|
C21H16N4O2S
|
1
|
| 1 |
IC50 = 94.8 nM
|
|
|
|
CP0401070
|
N-[2-(2-phenyltetrazol-5-yl)phenyl]-4-propylbenzamide
Show/Hide
|
C23H21N5O
|
2
|
| 1 |
IC50 = 96.6 nM
|
|
|
| 2 |
IC50 = 212 nM
|
|
|
|
CP0459389
|
N-[2-[2-(4-methylphenyl)tetrazol-5-yl]phenyl]-4-nitrobenzamide
Show/Hide
|
C21H16N6O3
|
1
|
| 1 |
IC50 = 100 nM
|
|
|
|
CP0547260
|
N-(3-methylsulfanylphenyl)-6-nitro-2-[3-(trifluoromethyl)phenyl]quinazolin-4-amine
Show/Hide
|
C22H15F3N4O2S
|
1
|
| 1 |
IC50 = 101 nM
|
|
|
|
CP0412384
|
N-[2-[2-(6-methoxypyridin-3-yl)tetrazol-5-yl]phenyl]benzamide
Show/Hide
|
C20H16N6O2
|
1
|
| 1 |
IC50 = 102 nM
|
|
|
|
CP0387305
|
N-(3-nitrophenyl)-2-pyridin-3-ylquinazolin-4-amine
Show/Hide
|
C19H13N5O2
|
1
|
| 1 |
IC50 = 105 nM
|
|
|
|
CP0445801
|
N-[2-[2-(4-methoxyphenyl)tetrazol-5-yl]phenyl]-4-(trifluoromethyl)benzamide
Show/Hide
|
C22H16F3N5O2
|
1
|
| 1 |
IC50 = 106 nM
|
|
|
|
CP0457689
|
6-nitro-N,2-diphenylquinazolin-4-amine
Show/Hide
|
C20H14N4O2
|
1
|
| 1 |
IC50 = 106 nM
|
|
|
|
CP0393142
|
2-(3-nitrophenyl)-N-phenylquinazolin-4-amine
Show/Hide
|
C20H14N4O2
|
1
|
| 1 |
IC50 = 108 nM
|
|
|
|
CP0415207
|
3-[[2-(3,4-dimethoxyphenyl)quinazolin-4-yl]amino]phenol
Show/Hide
|
C22H19N3O3
|
2
|
| 1 |
IC50 = 110 nM
|
|
|
| 2 |
IC50 = 140 nM
|
|
|
|
CP0459387
|
3,4-dimethoxy-N-[2-[2-(4-methoxyphenyl)tetrazol-5-yl]phenyl]benzamide
Show/Hide
|
C23H21N5O4
|
1
|
| 1 |
IC50 = 117 nM
|
|
|
|
CP0464424
|
N-[2-[2-(4-methylsulfanylphenyl)tetrazol-5-yl]phenyl]-2-nitrobenzamide
Show/Hide
|
C21H16N6O3S
|
2
|
| 1 |
IC50 = 117 nM
|
|
|
| 2 |
IC50 = 221 nM
|
|
|
|
CP0387306
|
N-(3-nitrophenyl)-2-pyridin-4-ylquinazolin-4-amine
Show/Hide
|
C19H13N5O2
|
1
|
| 1 |
IC50 = 117 nM
|
|
|
|
CP0448194
|
N-[2-[2-(4-methoxyphenyl)tetrazol-5-yl]phenyl]-4-nitrobenzamide
Show/Hide
|
C21H16N6O4
|
1
|
| 1 |
IC50 = 118 nM
|
|
|
|
CP0518995
|
4-[(6-nitro-2-phenylquinazolin-4-yl)amino]benzene-1,2-diol
Show/Hide
|
C20H14N4O4
|
1
|
| 1 |
IC50 = 119 nM
|
|
|
|
CP0481652
|
3-[[2-(3-nitrophenyl)quinazolin-4-yl]amino]benzonitrile
Show/Hide
|
C21H13N5O2
|
1
|
| 1 |
IC50 = 120 nM
|
|
|
|
CP0410359
|
3-[(6-methyl-2-phenylpyrimidin-4-yl)amino]benzonitrile
Show/Hide
|
C18H14N4
|
1
|
| 1 |
IC50 = 122 nM
|
|
|
|
CP0401068
|
3-nitro-N-[2-(2-phenyltetrazol-5-yl)phenyl]benzamide
Show/Hide
|
C20H14N6O3
|
2
|
| 1 |
IC50 = 123 nM
|
|
|
| 2 |
IC50 = 127 nM
|
|
|
|
CP0486085
|
N-[3-[[2-(3-nitrophenyl)quinazolin-4-yl]amino]phenyl]acetamide
Show/Hide
|
C22H17N5O3
|
1
|
| 1 |
IC50 = 127 nM
|
|
|
|
CP0141589
|
3-((3S,6S)-6-Isobutyl-9-methoxy-1,4-dioxo-1,2,3,4,6,7,12,12a-octahydro-pyrazino[1',2':1,6]pyrido[3,4-b]indol-3-yl)-propionic acid tert-butyl ester
Show/Hide
|
C26H35N3O5
|
13
|
| 1 |
IC50 = 128 nM
|
|
|
| 2 |
IC50 = 202 nM
|
|
|
| 3 |
IC50 = 215 nM
|
|
|
| 4 |
IC50 = 220 nM
|
|
|
| 5 |
IC50 = 221 nM
|
|
|
| 6 |
IC50 = 227 nM
|
|
|
| 7 |
IC50 = 240 nM
|
|
|
| 8 |
IC50 = 250 nM
|
|
|
| 9 |
IC50 = 260 nM
|
|
|
| 10 |
IC50 = 274 nM
|
|
|
| 11 |
IC50 = 276 nM
|
|
|
| 12 |
IC50 = 330 nM
|
|
|
| 13 |
IC50 = 354 nM
|
|
|
|
CP0528302
|
4-[(6-methyl-2-phenylpyrimidin-4-yl)amino]benzonitrile
Show/Hide
|
C18H14N4
|
2
|
| 1 |
IC50 = 128 nM
|
|
|
| 2 |
IC50 = 189 nM
|
|
|
|
CP0464422
|
N-[2-[2-(4-hydroxyphenyl)tetrazol-5-yl]phenyl]-4-propylbenzamide
Show/Hide
|
C23H21N5O2
|
2
|
| 1 |
IC50 = 129 nM
|
|
|
| 2 |
IC50 = 204 nM
|
|
|
|
CP0542906
|
N-[4-methoxy-2-[2-(4-methoxyphenyl)tetrazol-5-yl]phenyl]-4-nitrobenzamide
Show/Hide
|
C22H18N6O5
|
1
|
| 1 |
IC50 = 129 nM
|
|
|
|
CP0408573
|
(3-Nitro-phenyl)-(2-phenyl-quinazolin-4-yl)-amine
Show/Hide
|
C20H14N4O2
|
1
|
| 1 |
IC50 = 130 nM
|
|
|
|
CP0383766
|
N-[2-[2-(6-methoxypyridin-3-yl)tetrazol-5-yl]phenyl]-4-(trifluoromethyl)benzamide
Show/Hide
|
C21H15F3N6O2
|
1
|
| 1 |
IC50 = 130 nM
|
|
|
|
CP0424640
|
6-methyl-N-(3-nitrophenyl)-2-phenylpyrimidin-4-amine
Show/Hide
|
C17H14N4O2
|
2
|
| 1 |
IC50 = 130 nM
|
|
|
| 2 |
IC50 = 146 nM
|
|
|
|
CP0465045
|
4-methoxy-N-[2-[2-(4-propan-2-ylphenyl)tetrazol-5-yl]phenyl]benzamide
Show/Hide
|
C24H23N5O2
|
2
|
| 1 |
IC50 = 131 nM
|
|
|
| 2 |
IC50 = 136 nM
|
|
|
|
CP0500266
|
4-methoxy-N-[2-[2-(4-methylsulfanylphenyl)tetrazol-5-yl]phenyl]benzamide
Show/Hide
|
C22H19N5O2S
|
2
|
| 1 |
IC50 = 132 nM
|
|
|
| 2 |
IC50 = 251 nM
|
|
|
|
CP0472386
|
3-[(6-methyl-2-pyridin-4-ylpyrimidin-4-yl)amino]benzonitrile
Show/Hide
|
C17H13N5
|
1
|
| 1 |
IC50 = 132 nM
|
|
|
|
CP0410353
|
3-[(2-pyridin-4-ylquinazolin-4-yl)amino]benzonitrile
Show/Hide
|
C20H13N5
|
1
|
| 1 |
IC50 = 134 nM
|
|
|
|
CP0393139
|
3-[[2-(3,4-dimethoxyphenyl)quinazolin-4-yl]amino]benzonitrile
Show/Hide
|
C23H18N4O2
|
3
|
| 1 |
IC50 = 136 nM
|
|
|
| 2 |
IC50 = 190 nM
|
|
|
| 3 |
IC50 = 300 nM
|
|
|
|
CP0410747
|
N-[2-[2-(4-methylphenyl)tetrazol-5-yl]phenyl]-4-(trifluoromethyl)benzamide
Show/Hide
|
C22H16F3N5O
|
1
|
| 1 |
IC50 = 137 nM
|
|
|
|
CP0523463
|
3-[(2-phenylquinazolin-4-yl)amino]benzonitrile
Show/Hide
|
C21H14N4
|
1
|
| 1 |
IC50 = 140 nM
|
|
|
|
CP0389951
|
N-[4-methoxy-3-(trifluoromethyl)phenyl]-2-pyridin-4-ylquinazolin-4-amine
Show/Hide
|
C21H15F3N4O
|
1
|
| 1 |
IC50 = 146 nM
|
|
|
|
CP0421518
|
3-[(2-phenyl-4-quinazolinyl)amino]phenol
Show/Hide
|
C20H15N3O
|
1
|
| 1 |
IC50 = 150 nM
|
|
|
|
CP0464453
|
4-nitro-N-[2-(2-phenyltetrazol-5-yl)phenyl]benzamide
Show/Hide
|
C20H14N6O3
|
2
|
| 1 |
IC50 = 150 nM
|
|
|
| 2 |
IC50 = 321 nM
|
|
|
|
CP0475211
|
N-(3-methoxyphenyl)-2-phenylpyrido[2,3-d]pyrimidin-4-amine
Show/Hide
|
C20H16N4O
|
1
|
| 1 |
IC50 = 150 nM
|
|
|
|
CP0412501
|
2-nitro-4-[[2-(3-nitrophenyl)quinazolin-4-yl]amino]phenol
Show/Hide
|
C20H13N5O5
|
1
|
| 1 |
IC50 = 151 nM
|
|
|
|
CP0388004
|
N-(3,4-dimethoxyphenyl)-2-phenylquinazolin-4-amine
Show/Hide
|
C22H19N3O2
|
2
|
| 1 |
IC50 = 152 nM
|
|
|
| 2 |
IC50 = 190 nM
|
|
|
|
CP0469972
|
N-(3-fluorophenyl)-2-pyridin-3-ylquinazolin-4-amine
Show/Hide
|
C19H13FN4
|
1
|
| 1 |
IC50 = 156 nM
|
|
|
|
CP0513312
|
N-(3,4-difluorophenyl)-2-(3-methoxyphenyl)pyrido[2,3-d]pyrimidin-4-amine
Show/Hide
|
C20H14F2N4O
|
1
|
| 1 |
IC50 = 163 nM
|
|
|
|
CP0475210
|
N-(3-fluorophenyl)-2-phenylpyrido[2,3-d]pyrimidin-4-amine
Show/Hide
|
C19H13FN4
|
1
|
| 1 |
IC50 = 164 nM
|
|
|
|
CP0408063
|
4-[(2-pyridin-3-ylquinazolin-4-yl)amino]benzonitrile
Show/Hide
|
C20H13N5
|
1
|
| 1 |
IC50 = 166 nM
|
|
|
|
CP0393141
|
N-(3-nitrophenyl)-2-(4-nitrophenyl)quinazolin-4-amine
Show/Hide
|
C20H13N5O4
|
1
|
| 1 |
IC50 = 166 nM
|
|
|
|
CP0401067
|
N-[2-[2-(4-methoxyphenyl)tetrazol-5-yl]phenyl]-3-nitrobenzamide
Show/Hide
|
C21H16N6O4
|
2
|
| 1 |
IC50 = 168 nM
|
|
|
| 2 |
IC50 = 247 nM
|
|
|
|
CP0558202
|
N-[2-(2-phenyltetrazol-5-yl)phenyl]quinoline-3-carboxamide
Show/Hide
|
C23H16N6O
|
1
|
| 1 |
IC50 = 176 nM
|
|
|
|
CP0389519
|
2-phenyl-N-[3-(trifluoromethyl)phenyl]pyrido[2,3-d]pyrimidin-4-amine
Show/Hide
|
C20H13F3N4
|
1
|
| 1 |
IC50 = 177 nM
|
|
|
|
CP0441652
|
4-methoxy-N-[2-[2-(2-methoxyphenyl)tetrazol-5-yl]phenyl]benzamide
Show/Hide
|
C22H19N5O3
|
1
|
| 1 |
IC50 = 180 nM
|
|
|
|
CP0481657
|
2-(4-methoxyphenyl)-N-(3-nitrophenyl)quinazolin-4-amine
Show/Hide
|
C21H16N4O3
|
1
|
| 1 |
IC50 = 183 nM
|
|
|
|
CP0410741
|
4-nitro-N-[2-[2-(4-propylphenyl)tetrazol-5-yl]phenyl]benzamide
Show/Hide
|
C23H20N6O3
|
1
|
| 1 |
IC50 = 184 nM
|
|
|
|
CP0472567
|
4-[(6-methyl-2-phenylpyrimidin-4-yl)amino]benzene-1,2-dicarbonitrile
Show/Hide
|
C19H13N5
|
2
|
| 1 |
IC50 = 188 nM
|
|
|
| 2 |
IC50 = 548 nM
|
|
|
|
CP0380381
|
(E)-3-(3,4-dimethoxyphenyl)-1-[4-[[2-(3,4-dimethoxyphenyl)quinazolin-4-yl]amino]phenyl]prop-2-en-1-one
Show/Hide
|
C33H29N3O5
|
1
|
| 1 |
IC50 = 190 nM
|
|
|
|
CP0577964
|
N-[2-(2-phenyltetrazol-5-yl)phenyl]-2,3-dihydro-1,4-benzodioxine-6-carboxamide
Show/Hide
|
C22H17N5O3
|
1
|
| 1 |
IC50 = 190 nM
|
|
|
|
CP0412740
|
4-methoxy-N-[2-[2-(4-methoxyphenyl)tetrazol-5-yl]phenyl]benzamide
Show/Hide
|
C22H19N5O3
|
2
|
| 1 |
IC50 = 199 nM
|
|
|
| 2 |
IC50 = 300 nM
|
|
|
|
CP0385298
|
4-methoxy-N-[2-(2-phenyltetrazol-5-yl)phenyl]benzamide
Show/Hide
|
C21H17N5O2
|
2
|
| 1 |
IC50 = 200 nM
|
|
|
| 2 |
IC50 = 208 nM
|
|
|
|
CP0486869
|
N-[2-[2-(4-ethoxyphenyl)tetrazol-5-yl]phenyl]-3,4-dimethoxybenzamide
Show/Hide
|
C24H23N5O4
|
1
|
| 1 |
IC50 = 201 nM
|
|
|
|
CP0477032
|
N-(3,4-dimethoxyphenyl)-2-thiophen-2-ylquinazolin-4-amine
Show/Hide
|
C20H17N3O2S
|
1
|
| 1 |
IC50 = 202 nM
|
|
|
|
CP0490374
|
N-(4-bromo-3-methoxyphenyl)-2-phenylquinazolin-4-amine
Show/Hide
|
C21H16BrN3O
|
2
|
| 1 |
IC50 = 202 nM
|
|
|
| 2 |
IC50 = 289 nM
|
|
|
|
CP0395884
|
4-[(2-phenylquinazolin-4-yl)amino]phenol
Show/Hide
|
C20H15N3O
|
3
|
| 1 |
IC50 = 204 nM
|
|
|
| 2 |
IC50 = 211 nM
|
|
|
| 3 |
IC50 = 304 nM
|
|
|
|
CP0392202
|
N-(3-methylsulfanylphenyl)-2-phenylpyrido[2,3-d]pyrimidin-4-amine
Show/Hide
|
C20H16N4S
|
1
|
| 1 |
IC50 = 206 nM
|
|
|
|
CP0446423
|
[1-(3,4-dichlorophenyl)-1,3,4,9-tetrahydropyrido[3,4-b]indol-2-yl]-(3-methoxyphenyl)methanone
Show/Hide
|
C25H20Cl2N2O2
|
2
|
| 1 |
IC50 = 206 nM
|
|
|
| 2 |
IC50 = 238 nM
|
|
|
|
CP0401902
|
(E)-1-[3-[[2-(3,4-dimethoxyphenyl)quinazolin-4-yl]amino]phenyl]-3-(4-methoxyphenyl)prop-2-en-1-one
Show/Hide
|
C32H27N3O4
|
1
|
| 1 |
IC50 = 210 nM
|
|
|
|
CP0481653
|
N-(3,4-diethoxyphenyl)-2-(3-nitrophenyl)quinazolin-4-amine
Show/Hide
|
C24H22N4O4
|
1
|
| 1 |
IC50 = 210 nM
|
|
|
|
CP0401071
|
N-[2-[2-(3,4-dimethoxyphenyl)tetrazol-5-yl]phenyl]benzamide
Show/Hide
|
C22H19N5O3
|
2
|
| 1 |
IC50 = 212 nM
|
|
|
| 2 |
IC50 = 230 nM
|
|
|
|
CP0472388
|
2-pyridin-4-yl-N-[3-(trifluoromethyl)phenyl]quinazolin-4-amine
Show/Hide
|
C20H13F3N4
|
1
|
| 1 |
IC50 = 216 nM
|
|
|
|
CP0402502
|
3-N,3-N-dimethyl-1-N-[2-(3-nitrophenyl)quinazolin-4-yl]benzene-1,3-diamine
Show/Hide
|
C22H19N5O2
|
1
|
| 1 |
IC50 = 221 nM
|
|
|
|
CP0401065
|
N-[2-[2-(4-chlorophenyl)tetrazol-5-yl]phenyl]-4-methoxybenzamide
Show/Hide
|
C21H16ClN5O2
|
1
|
| 1 |
IC50 = 223 nM
|
|
|
|
CP0057114
|
MLS001007082
Show/Hide
|
C22H18N4O
|
2
|
| 1 |
IC50 = 224 nM
|
|
|
| 2 |
IC50 = 278 nM
|
|
|
|
CP0393135
|
N-[3-[[2-(3-cyanophenyl)quinazolin-4-yl]amino]phenyl]acetamide
Show/Hide
|
C23H17N5O
|
1
|
| 1 |
IC50 = 225 nM
|
|
|
|
CP0542905
|
N-[2-[2-(4-methoxyphenyl)tetrazol-5-yl]phenyl]quinoline-3-carboxamide
Show/Hide
|
C24H18N6O2
|
1
|
| 1 |
IC50 = 228 nM
|
|
|
|
CP0486084
|
3-N,3-N-diethyl-1-N-[2-(3-nitrophenyl)quinazolin-4-yl]benzene-1,3-diamine
Show/Hide
|
C24H23N5O2
|
1
|
| 1 |
IC50 = 230 nM
|
|
|
|
CP0446488
|
[1-(3,4-dichlorophenyl)-1,3,4,9-tetrahydropyrido[3,4-b]indol-2-yl]-(4-methoxyphenyl)methanone
Show/Hide
|
C25H20Cl2N2O2
|
2
|
| 1 |
IC50 = 233 nM
|
|
|
| 2 |
IC50 = 237 nM
|
|
|
|
CP0486087
|
N,2-bis(3-nitrophenyl)quinazolin-4-amine
Show/Hide
|
C20H13N5O4
|
1
|
| 1 |
IC50 = 236 nM
|
|
|
|
CP0435460
|
2-(3,4-dimethoxyphenyl)-N-[3-(trifluoromethyl)phenyl]quinazolin-4-amine
Show/Hide
|
C23H18F3N3O2
|
2
|
| 1 |
IC50 = 240 nM
|
|
|
| 2 |
IC50 = 300 nM
|
|
|
|
CP0469973
|
2-nitro-4-[(2-pyridin-3-ylquinazolin-4-yl)amino]phenol
Show/Hide
|
C19H13N5O3
|
1
|
| 1 |
IC50 = 245 nM
|
|
|
|
CP0445691
|
2-phenyl-N-[3-(trifluoromethyl)phenyl]quinazolin-4-amine
Show/Hide
|
C21H14F3N3
|
1
|
| 1 |
IC50 = 250 nM
|
|
|
|
CP0472566
|
3-[(6-methyl-2-phenylpyrimidin-4-yl)amino]phenol
Show/Hide
|
C17H15N3O
|
2
|
| 1 |
IC50 = 253 nM
|
|
|
| 2 |
IC50 = 516 nM
|
|
|
|
CP0487637
|
5-[(6-methyl-2-phenylpyrimidin-4-yl)amino]isoindole-1,3-dione
Show/Hide
|
C19H14N4O2
|
2
|
| 1 |
IC50 = 253 nM
|
|
|
| 2 |
IC50 = 416 nM
|
|
|
|
CP0545255
|
N-[2-(2-phenyltetrazol-5-yl)phenyl]-1,3-benzodioxole-5-carboxamide
Show/Hide
|
C21H15N5O3
|
1
|
| 1 |
IC50 = 259 nM
|
|
|
|
CP0407287
|
2-[[2-(3,4-dimethoxyphenyl)quinazolin-4-yl]amino]phenol
Show/Hide
|
C22H19N3O3
|
2
|
| 1 |
IC50 = 260 nM
|
|
|
| 2 |
IC50 = 290 nM
|
|
|
|
CP0410744
|
N-[2-[2-(2-methoxyphenyl)tetrazol-5-yl]phenyl]-4-nitrobenzamide
Show/Hide
|
C21H16N6O4
|
1
|
| 1 |
IC50 = 261 nM
|
|
|
|
CP0393132
|
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-(3-nitrophenyl)quinazolin-4-amine
Show/Hide
|
C22H16N4O4
|
1
|
| 1 |
IC50 = 263 nM
|
|
|
|
CP0477389
|
N-(3-fluorophenyl)-2-(3-methoxyphenyl)pyrido[2,3-d]pyrimidin-4-amine
Show/Hide
|
C20H15FN4O
|
1
|
| 1 |
IC50 = 264 nM
|
|
|
|
CP0464426
|
N-[2-[2-(4-methoxyphenyl)tetrazol-5-yl]phenyl]-2-nitrobenzamide
Show/Hide
|
C21H16N6O4
|
2
|
| 1 |
IC50 = 266 nM
|
|
|
| 2 |
IC50 = 311 nM
|
|
|
|
CP0529202
|
N-[2-[2-(4-methoxyphenyl)tetrazol-5-yl]phenyl]naphthalene-1-carboxamide
Show/Hide
|
C25H19N5O2
|
1
|
| 1 |
IC50 = 267 nM
|
|
|
|
CP0410749
|
3,4-dimethoxy-N-[2-[2-[4-(trifluoromethyl)phenyl]tetrazol-5-yl]phenyl]benzamide
Show/Hide
|
C23H18F3N5O3
|
1
|
| 1 |
IC50 = 269 nM
|
|
|
|
CP0516015
|
N-[2-(2-phenyltetrazol-5-yl)phenyl]thiophene-2-carboxamide
Show/Hide
|
C18H13N5OS
|
1
|
| 1 |
IC50 = 270 nM
|
|
|
|
CP0543103
|
N-(3-methoxyphenyl)-6-methyl-2-pyridin-4-ylpyrimidin-4-amine
Show/Hide
|
C17H16N4O
|
1
|
| 1 |
IC50 = 271 nM
|
|
|
|
CP0507499
|
N-(3-methoxyphenyl)-6-methyl-2-phenylpyrimidin-4-amine
Show/Hide
|
C18H17N3O
|
2
|
| 1 |
IC50 = 271 nM
|
|
|
| 2 |
IC50 = 503 nM
|
|
|
|
CP0546238
|
4-[(2-phenylpyrimidin-4-yl)amino]benzonitrile
Show/Hide
|
C17H12N4
|
1
|
| 1 |
IC50 = 274 nM
|
|
|
|
CP0450330
|
2-nitro-N-[2-(2-phenyltetrazol-5-yl)phenyl]benzamide
Show/Hide
|
C20H14N6O3
|
2
|
| 1 |
IC50 = 280 nM
|
|
|
| 2 |
IC50 = 458 nM
|
|
|
|
CP0466205
|
N-(4-bromo-3-methoxyphenyl)-6-methyl-2-phenylpyrimidin-4-amine
Show/Hide
|
C18H16BrN3O
|
2
|
| 1 |
IC50 = 280 nM
|
|
|
| 2 |
IC50 = 328 nM
|
|
|
|
CP0412502
|
3-N-[2-(3-nitrophenyl)quinazolin-4-yl]benzene-1,3-diamine
Show/Hide
|
C20H15N5O2
|
1
|
| 1 |
IC50 = 284 nM
|
|
|
|
CP0542902
|
N-[2-(2-phenyltetrazol-5-yl)phenyl]cyclohexanecarboxamide
Show/Hide
|
C20H21N5O
|
1
|
| 1 |
IC50 = 287 nM
|
|
|
|
CP0547299
|
N-[2-(2-phenyltetrazol-5-yl)phenyl]pyridine-4-carboxamide
Show/Hide
|
C19H14N6O
|
1
|
| 1 |
IC50 = 287 nM
|
|
|
|
CP0432849
|
N-(3-bromophenyl)-2-(3,4-dimethoxyphenyl)quinazolin-4-amine
Show/Hide
|
C22H18BrN3O2
|
2
|
| 1 |
IC50 = 290 nM
|
|
|
| 2 |
IC50 = 400 nM
|
|
|
|
CP0454937
|
(E)-3-(3,4-dimethoxyphenyl)-1-[4-[(2-phenylquinazolin-4-yl)amino]phenyl]prop-2-en-1-one
Show/Hide
|
C31H25N3O3
|
1
|
| 1 |
IC50 = 290 nM
|
|
|
|
CP0481656
|
N-(3,5-dinitrophenyl)-2-(3-methoxyphenyl)quinazolin-4-amine
Show/Hide
|
C21H15N5O5
|
1
|
| 1 |
IC50 = 291 nM
|
|
|
|
CP0430542
|
3-[4-(3-hydroxy-4-methoxyanilino)quinazolin-2-yl]benzonitrile
Show/Hide
|
C22H16N4O2
|
1
|
| 1 |
IC50 = 297 nM
|
|
|
|
CP0552367
|
tert-butyl 3-[(2-pyridin-4-ylquinazolin-4-yl)amino]benzoate
Show/Hide
|
C24H22N4O2
|
1
|
| 1 |
IC50 = 299 nM
|
|
|
|
CP0424456
|
N-(3-nitrophenyl)-2-thiophen-2-ylquinazolin-4-amine
Show/Hide
|
C18H12N4O2S
|
1
|
| 1 |
IC50 = 300 nM
|
|
|
|
CP0383544
|
4-[[2-(3,4-dimethoxyphenyl)quinazolin-4-yl]amino]-2-nitrophenol
Show/Hide
|
C22H18N4O5
|
1
|
| 1 |
IC50 = 305 nM
|
|
|
|
CP0469080
|
N-[2-[2-(4-ethoxyphenyl)tetrazol-5-yl]phenyl]-2-nitrobenzamide
Show/Hide
|
C22H18N6O4
|
1
|
| 1 |
IC50 = 308 nM
|
|
|
|
CP0454936
|
(E)-1-[3-[[2-(3,4-dimethoxyphenyl)quinazolin-4-yl]amino]phenyl]-3-(3-methoxyphenyl)prop-2-en-1-one
Show/Hide
|
C32H27N3O4
|
1
|
| 1 |
IC50 = 310 nM
|
|
|
|
CP0472564
|
N-(6-methyl-2-phenylpyrimidin-4-yl)quinoxalin-6-amine
Show/Hide
|
C19H15N5
|
1
|
| 1 |
IC50 = 312 nM
|
|
|
|
CP0464421
|
N-[2-[2-(3,4-dimethoxyphenyl)tetrazol-5-yl]phenyl]-4-methoxybenzamide
Show/Hide
|
C23H21N5O4
|
1
|
| 1 |
IC50 = 319 nM
|
|
|
|
CP0395732
|
6,7-dimethoxy-2-N,4-N-bis(3-nitrophenyl)quinazoline-2,4-diamine
Show/Hide
|
C22H18N6O6
|
2
|
| 1 |
IC50 = 320 nM
|
|
|
| 2 |
IC50 = 330 nM
|
|
|
|
CP0443410
|
(E)-1-[3-[(6,7-dimethoxyquinazolin-4-yl)amino]phenyl]-3-(4-methoxyphenyl)prop-2-en-1-one
Show/Hide
|
C26H23N3O4
|
1
|
| 1 |
IC50 = 320 nM
|
|
|
|
CP0473956
|
[1-(3,4-dichlorophenyl)-1,3,4,9-tetrahydropyrido[3,4-b]indol-2-yl]-phenylmethanone
Show/Hide
|
C24H18Cl2N2O
|
2
|
| 1 |
IC50 = 328 nM
|
|
|
| 2 |
IC50 = 365 nM
|
|
|
|
CP0503950
|
N-[2-[2-(3,4-dimethoxyphenyl)tetrazol-5-yl]phenyl]-4-(trifluoromethyl)benzamide
Show/Hide
|
C23H18F3N5O3
|
1
|
| 1 |
IC50 = 330 nM
|
|
|
|
CP0424457
|
N-(4-nitrophenyl)-2-thiophen-2-ylquinazolin-4-amine
Show/Hide
|
C18H12N4O2S
|
1
|
| 1 |
IC50 = 335 nM
|
|
|
|
CP0402504
|
3-[[2-(4-nitrophenyl)quinazolin-4-yl]amino]benzonitrile
Show/Hide
|
C21H13N5O2
|
1
|
| 1 |
IC50 = 336 nM
|
|
|
|
CP0404569
|
N-(3,4-dimethoxyphenyl)-2-phenylpyrido[2,3-d]pyrimidin-4-amine
Show/Hide
|
C21H18N4O2
|
1
|
| 1 |
IC50 = 343 nM
|
|
|
|
CP0541420
|
3-[[2-(3-methoxyphenyl)pyrido[2,3-d]pyrimidin-4-yl]amino]benzonitrile
Show/Hide
|
C21H15N5O
|
1
|
| 1 |
IC50 = 348 nM
|
|
|
|
CP0529203
|
N-[2-[2-(4-methoxyphenyl)tetrazol-5-yl]phenyl]thiophene-2-carboxamide
Show/Hide
|
C19H15N5O2S
|
1
|
| 1 |
IC50 = 351 nM
|
|
|
|
CP0389950
|
N-(3-fluorophenyl)-2-phenylquinazolin-4-amine
Show/Hide
|
C20H14FN3
|
3
|
| 1 |
IC50 = 355 nM
|
|
|
| 2 |
IC50 = 363 nM
|
|
|
| 3 |
IC50 = 405 nM
|
|
|
|
CP0393129
|
3-[[2-(3-methoxyphenyl)quinazolin-4-yl]amino]benzonitrile
Show/Hide
|
C22H16N4O
|
1
|
| 1 |
IC50 = 359 nM
|
|
|
|
CP0403081
|
(E)-1-[4-[[2-(3,4-dimethoxyphenyl)quinazolin-4-yl]amino]phenyl]-3-(3-methoxyphenyl)prop-2-en-1-one
Show/Hide
|
C32H27N3O4
|
1
|
| 1 |
IC50 = 360 nM
|
|
|
|
CP0304737
|
N-[3-[(2-thiophen-2-ylquinazolin-4-yl)amino]phenyl]acetamide
Show/Hide
|
C20H16N4OS
|
1
|
| 1 |
IC50 = 360 nM
|
|
|
|
CP0410357
|
3-(2-Pyridin-3-yl-quinazolin-4-ylamino)-benzoic acid methyl ester
Show/Hide
|
C21H16N4O2
|
1
|
| 1 |
IC50 = 362 nM
|
|
|
|
CP0389586
|
4-N-(3-methoxyphenyl)-2-pyridin-3-ylquinazoline-4,6-diamine
Show/Hide
|
C20H17N5O
|
1
|
| 1 |
IC50 = 369 nM
|
|
|
|
CP0408062
|
N-(3-nitrophenyl)-2-pyridin-2-ylquinazolin-4-amine
Show/Hide
|
C19H13N5O2
|
1
|
| 1 |
IC50 = 376 nM
|
|
|
|
CP0361939
|
[1-(3,4-dichlorophenyl)-6-methoxy-1,3,4,9-tetrahydropyrido[3,4-b]indol-2-yl]-phenylmethanone
Show/Hide
|
C25H20Cl2N2O2
|
1
|
| 1 |
IC50 = 382 nM
|
|
|
|
CP0466213
|
N-(3-bromophenyl)-6-methyl-2-phenylpyrimidin-4-amine
Show/Hide
|
C17H14BrN3
|
2
|
| 1 |
IC50 = 386 nM
|
|
|
| 2 |
IC50 = 892 nM
|
|
|
|
CP0386498
|
(E)-1-[4-[(6,7-dimethoxyquinazolin-4-yl)amino]phenyl]-3-(3-methoxyphenyl)prop-2-en-1-one
Show/Hide
|
C26H23N3O4
|
1
|
| 1 |
IC50 = 390 nM
|
|
|
|
CP0475205
|
3-[(2-phenylpyrido[2,3-d]pyrimidin-4-yl)amino]benzonitrile
Show/Hide
|
C20H13N5
|
1
|
| 1 |
IC50 = 400 nM
|
|
|
|
CP0407967
|
3-[(2-pyridin-4-yl-4-quinazolinyl)amino]benzoic acid methyl ester
Show/Hide
|
C21H16N4O2
|
1
|
| 1 |
IC50 = 405 nM
|
|
|
|
CP0393131
|
N-(3,4-dimethoxyphenyl)-2-(4-methoxyphenyl)quinazolin-4-amine
Show/Hide
|
C23H21N3O3
|
1
|
| 1 |
IC50 = 418 nM
|
|
|
|
CP0388006
|
N,2-bis(3,4-dimethoxyphenyl)quinazolin-4-amine
Show/Hide
|
C24H23N3O4
|
2
|
| 1 |
IC50 = 420 nM
|
|
|
| 2 |
IC50 = 610 nM
|
|
|
|
CP0395159
|
N-(2-phenylquinazolin-4-yl)benzamide
Show/Hide
|
C21H15N3O
|
1
|
| 1 |
IC50 = 424 nM
|
|
|
|
CP0463652
|
N-(4-fluorophenyl)-2-(3-methoxyphenyl)pyrido[2,3-d]pyrimidin-4-amine
Show/Hide
|
C20H15FN4O
|
1
|
| 1 |
IC50 = 425 nM
|
|
|
|
CP0481550
|
2-(3,4-dimethoxyphenyl)-3-methoxybenzo[h]chromen-4-one
Show/Hide
|
C22H18O5
|
2
|
| 1 |
IC50 = 426 nM
|
|
|
| 2 |
IC50 = 468 nM
|
|
|
|
CP0529205
|
N-[2-(2-phenyltetrazol-5-yl)phenyl]naphthalene-1-carboxamide
Show/Hide
|
C24H17N5O
|
1
|
| 1 |
IC50 = 430 nM
|
|
|
|
CP0547345
|
N-[2-(2-phenyltetrazol-5-yl)phenyl]pyridine-3-carboxamide
Show/Hide
|
C19H14N6O
|
1
|
| 1 |
IC50 = 445 nM
|
|
|
|
CP0410745
|
N-[2-[2-(2-methoxyphenyl)tetrazol-5-yl]phenyl]-4-(trifluoromethyl)benzamide
Show/Hide
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C22H16F3N5O2
|
1
|
| 1 |
IC50 = 451 nM
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CP0473013
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N-(3-chlorophenyl)-2-phenylpyrido[2,3-d]pyrimidin-4-amine
Show/Hide
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C19H13ClN4
|
1
|
| 1 |
IC50 = 454 nM
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CP0444348
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2-(4-fluoro-3-methoxyphenyl)benzo[h]chromen-4-one
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C20H13FO3
|
2
|
| 1 |
IC50 = 457 nM
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| 2 |
IC50 = 522 nM
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CP0406749
|
3-(3,4-dimethoxyphenyl)benzo[f]chromen-1-one
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C21H16O4
|
2
|
| 1 |
IC50 = 458 nM
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| 2 |
IC50 = 590 nM
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CP0567720
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(E)-3-(3,4-dimethoxyphenyl)-1-[3-[(2-phenylquinazolin-4-yl)amino]phenyl]prop-2-en-1-one
Show/Hide
|
C31H25N3O3
|
1
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| 1 |
IC50 = 460 nM
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CP0536908
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2-(3,4-dimethoxyphenyl)-N-(3-fluorophenyl)quinazolin-4-amine
Show/Hide
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C22H18FN3O2
|
1
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| 1 |
IC50 = 462 nM
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CP0443797
|
4-[[2-(3,4-dimethoxyphenyl)quinazolin-4-yl]amino]phenol
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C22H19N3O3
|
2
|
| 1 |
IC50 = 470 nM
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| 2 |
IC50 = 680 nM
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CP0484132
|
3-[[2-(3-cyanoanilino)-6,7-dimethoxyquinazolin-4-yl]amino]benzonitrile
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C24H18N6O2
|
2
|
| 1 |
IC50 = 470 nM
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| 2 |
IC50 = 480 nM
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CP0407963
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2-pyridin-4-yl-N-[4-(trifluoromethyl)phenyl]quinazolin-4-amine
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C20H13F3N4
|
1
|
| 1 |
IC50 = 488 nM
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CP0383920
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N-[2-[(E)-3-(3,4-dimethoxyphenyl)prop-2-enoyl]phenyl]thiophene-2-carboxamide
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C22H19NO4S
|
1
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| 1 |
IC50 = 501 nM
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CP0563543
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3-[(2-pyridin-2-ylquinazolin-4-yl)amino]benzonitrile
Show/Hide
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C20H13N5
|
1
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| 1 |
IC50 = 507 nM
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CP0401069
|
3,4-dimethoxy-N-[2-(2-phenyltetrazol-5-yl)phenyl]benzamide
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C22H19N5O3
|
2
|
| 1 |
IC50 = 511 nM
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| 2 |
IC50 = 832 nM
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CP0482674
|
N-(3-ethynylphenyl)-2-phenylquinazolin-4-amine
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C22H15N3
|
2
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| 1 |
IC50 = 513 nM
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| 2 |
IC50 = 672 nM
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CP0575545
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N-(3-nitrophenyl)-2-phenylpyrido[2,3-d]pyrimidin-4-amine
Show/Hide
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C19H13N5O2
|
1
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| 1 |
IC50 = 519 nM
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CP0541418
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2-nitro-4-[(2-phenylpyrido[2,3-d]pyrimidin-4-yl)amino]phenol
Show/Hide
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C19H13N5O3
|
1
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| 1 |
IC50 = 528 nM
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CP0427782
|
(E)-3-(3,4-dimethoxyphenyl)-1-(2-hydroxy-4,6-dimethoxyphenyl)prop-2-en-1-one
Show/Hide
|
C19H20O6
|
1
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| 1 |
IC50 = 530 nM
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CP0412776
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2-(3-methoxyphenyl)-N-[3-(trifluoromethyl)phenyl]pyrido[2,3-d]pyrimidin-4-amine
Show/Hide
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C21H15F3N4O
|
1
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| 1 |
IC50 = 539 nM
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CP0050832
|
2-(3,4-Dimethoxy-phenyl)-5-hydroxy-3,7-dimethoxy-chromen-4-one
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C19H18O7
|
2
|
| 1 |
IC50 = 540 nM
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| 2 |
IC50 = 570 nM
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CP0472563
|
N-[4-methoxy-3-(trifluoromethyl)phenyl]-6-methyl-2-phenylpyrimidin-4-amine
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C19H16F3N3O
|
2
|
| 1 |
IC50 = 544 nM
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| 2 |
IC50 = 598 nM
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CP0410360
|
N-(3,4-dimethoxyphenyl)-2-pyridin-4-ylquinazolin-4-amine
Show/Hide
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C21H18N4O2
|
1
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| 1 |
IC50 = 545 nM
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CP0490377
|
4-[(2-phenylquinazolin-4-yl)amino]benzenesulfonyl fluoride
Show/Hide
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C20H14FN3O2S
|
1
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| 1 |
IC50 = 556 nM
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CP0387308
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N-(3-methoxyphenyl)-2-pyridin-4-ylquinazolin-4-amine
Show/Hide
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C20H16N4O
|
1
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| 1 |
IC50 = 558 nM
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CP0529204
|
N-[2-[2-(4-methoxyphenyl)tetrazol-5-yl]phenyl]cyclohexanecarboxamide
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C21H23N5O2
|
1
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| 1 |
IC50 = 565 nM
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CP0396379
|
N-(3-bromophenyl)-2-phenylquinazolin-4-amine
Show/Hide
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C20H14BrN3
|
1
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| 1 |
IC50 = 570 nM
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CP0416871
|
3-[[2-(3,4-dimethoxyphenyl)quinazolin-4-yl]amino]benzenesulfonyl fluoride
Show/Hide
|
C22H18FN3O4S
|
1
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| 1 |
IC50 = 570 nM
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CP0567376
|
N-(3,4-dimethoxyphenyl)-2-(3-methoxyphenyl)pyrido[2,3-d]pyrimidin-4-amine
Show/Hide
|
C22H20N4O3
|
1
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| 1 |
IC50 = 572 nM
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CP0390839
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(E)-3-(3,4-dimethoxyphenyl)-1-[3-[[2-(3,4-dimethoxyphenyl)quinazolin-4-yl]amino]phenyl]prop-2-en-1-one
Show/Hide
|
C33H29N3O5
|
1
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| 1 |
IC50 = 600 nM
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CP0484131
|
6,7-dimethoxy-2-N,4-N-bis[3-(trifluoromethyl)phenyl]quinazoline-2,4-diamine
Show/Hide
|
C24H18F6N4O2
|
2
|
| 1 |
IC50 = 610 nM
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| 2 |
IC50 = 800 nM
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CP0451507
|
2-(3,4-dimethoxyphenyl)-N-(3,5-dinitrophenyl)quinazolin-4-amine
Show/Hide
|
C22H17N5O6
|
1
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| 1 |
IC50 = 610 nM
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CP0490378
|
N-(4-iodophenyl)-2-phenylquinazolin-4-amine
Show/Hide
|
C20H14IN3
|
1
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| 1 |
IC50 = 612 nM
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CP0470839
|
2-(3-methoxyphenyl)-N-[4-(trifluoromethyl)phenyl]pyrido[2,3-d]pyrimidin-4-amine
Show/Hide
|
C21H15F3N4O
|
1
|
| 1 |
IC50 = 621 nM
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CP0489923
|
N-(3-chlorophenyl)-2-(3-methoxyphenyl)pyrido[2,3-d]pyrimidin-4-amine
Show/Hide
|
C20H15ClN4O
|
1
|
| 1 |
IC50 = 628 nM
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CP0395731
|
2-(3,4-dimethoxyphenyl)-N-(2-nitrophenyl)quinazolin-4-amine
Show/Hide
|
C22H18N4O4
|
2
|
| 1 |
IC50 = 640 nM
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| 2 |
IC50 = 1550 nM
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CP0412505
|
2-(2-methoxyphenyl)-N-(3-nitrophenyl)quinazolin-4-amine
Show/Hide
|
C21H16N4O3
|
1
|
| 1 |
IC50 = 642 nM
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CP0424485
|
4-Anilino quinazoline deriv. 12
Show/Hide
|
C15H13N3O
|
1
|
| 1 |
IC50 = 645 nM
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CP0518996
|
4-N-(4-methoxyphenyl)-2-pyridin-3-ylquinazoline-4,6-diamine
Show/Hide
|
C20H17N5O
|
1
|
| 1 |
IC50 = 646 nM
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CP0565185
|
6-methyl-N,2-diphenylpyrimidin-4-amine
Show/Hide
|
C17H15N3
|
1
|
| 1 |
IC50 = 648 nM
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CP0420849
|
N-(3,4-dimethoxyphenyl)-2-(1H-pyrrol-2-yl)quinazolin-4-amine
Show/Hide
|
C20H18N4O2
|
1
|
| 1 |
IC50 = 652 nM
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CP0407286
|
2-N,4-N-bis(3-bromophenyl)-6,7-dimethoxyquinazoline-2,4-diamine
Show/Hide
|
C22H18Br2N4O2
|
2
|
| 1 |
IC50 = 670 nM
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| 2 |
IC50 = 860 nM
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CP0507006
|
N-[2-[2-(4-methylsulfanylphenyl)tetrazol-5-yl]phenyl]-4-propylbenzamide
Show/Hide
|
C24H23N5OS
|
2
|
| 1 |
IC50 = 679 nM
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| 2 |
IC50 = 783 nM
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CP0401903
|
(E)-3-(3-methoxyphenyl)-1-[4-(quinazolin-4-ylamino)phenyl]prop-2-en-1-one
Show/Hide
|
C24H19N3O2
|
1
|
| 1 |
IC50 = 680 nM
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CP0469625
|
(E)-3-(3-methoxyphenyl)-1-[3-[(2-phenylquinazolin-4-yl)amino]phenyl]prop-2-en-1-one
Show/Hide
|
C30H23N3O2
|
1
|
| 1 |
IC50 = 680 nM
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CP0530755
|
[1-(4-bromophenyl)-1,3,4,9-tetrahydropyrido[3,4-b]indol-2-yl]-phenylmethanone
Show/Hide
|
C24H19BrN2O
|
1
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| 1 |
IC50 = 687 nM
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CP0528175
|
N-(3-fluoro-4-methoxyphenyl)-2-phenylquinazolin-4-amine
Show/Hide
|
C21H16FN3O
|
2
|
| 1 |
IC50 = 689 nM
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| 2 |
IC50 = 872 nM
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CP0446428
|
[1-(3,4-dichlorophenyl)-1,3,4,9-tetrahydropyrido[3,4-b]indol-2-yl]-(3,4-dimethoxyphenyl)methanone
Show/Hide
|
C26H22Cl2N2O3
|
1
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| 1 |
IC50 = 698 nM
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CP0307451
|
N-[2-[[4-[2-(3,4-dihydro-1H-isoquinolin-2-yl)ethyl]phenyl]carbamoyl]phenyl]quinoline-3-carboxamide
Show/Hide
|
C34H30N4O2
|
3
|
| 1 |
IC50 = 704 nM
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| 2 |
IC50 = 721 nM
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| 3 |
IC50 = 741 nM
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CP0441268
|
(E)-3-(3,4-dimethoxyphenyl)-1-(2-hydroxynaphthalen-1-yl)prop-2-en-1-one
Show/Hide
|
C21H18O4
|
1
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| 1 |
IC50 = 720 nM
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CP0397340
|
2-(3,4-dimethoxyphenyl)-3-hydroxybenzo[h]chromen-4-one
Show/Hide
|
C21H16O5
|
2
|
| 1 |
IC50 = 724 nM
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| 2 |
IC50 = 1520 nM
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CP0547259
|
4-N-phenyl-2-[3-(trifluoromethyl)phenyl]quinazoline-4,6-diamine
Show/Hide
|
C21H15F3N4
|
1
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| 1 |
IC50 = 726 nM
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CP0536416
|
N-[2-(2-phenyltetrazol-5-yl)phenyl]pyridine-2-carboxamide
Show/Hide
|
C19H14N6O
|
1
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| 1 |
IC50 = 733 nM
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CP0446426
|
[1-(4-chlorophenyl)-1,3,4,9-tetrahydropyrido[3,4-b]indol-2-yl]-phenylmethanone
Show/Hide
|
C24H19ClN2O
|
2
|
| 1 |
IC50 = 741 nM
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| 2 |
IC50 = 784 nM
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CP0387307
|
(4-methoxyphenyl)-[2-(4-pyridyl)quinazolin-4-yl]amine
Show/Hide
|
C20H16N4O
|
1
|
| 1 |
IC50 = 742 nM
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CP0539340
|
2-(3-methoxyphenyl)-N-(3-nitrophenyl)pyrido[2,3-d]pyrimidin-4-amine
Show/Hide
|
C20H15N5O3
|
1
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| 1 |
IC50 = 747 nM
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CP0552366
|
N-(3,4-dimethoxyphenyl)-2-pyridin-3-ylquinazolin-4-amine
Show/Hide
|
C21H18N4O2
|
1
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| 1 |
IC50 = 753 nM
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CP0477947
|
N-[2-[4-(4-methoxyphenyl)triazol-1-yl]phenyl]-4-(trifluoromethyl)benzamide
Show/Hide
|
C23H17F3N4O2
|
1
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| 1 |
IC50 = 766 nM
|
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CP0466212
|
N-(4-fluoro-3-nitrophenyl)-6-methyl-2-phenylpyrimidin-4-amine
Show/Hide
|
C17H13FN4O2
|
2
|
| 1 |
IC50 = 771 nM
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| 2 |
IC50 = 1010 nM
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CP0466210
|
N-(3-fluorophenyl)-6-methyl-2-phenylpyrimidin-4-amine
Show/Hide
|
C17H14FN3
|
2
|
| 1 |
IC50 = 776 nM
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| 2 |
IC50 = 1110 nM
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CP0482673
|
N-(3-iodophenyl)-2-phenylquinazolin-4-amine
Show/Hide
|
C20H14IN3
|
1
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| 1 |
IC50 = 791 nM
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CP0385297
|
N-[2-[2-(4-ethoxyphenyl)tetrazol-5-yl]phenyl]-4-methoxybenzamide
Show/Hide
|
C23H21N5O3
|
1
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| 1 |
IC50 = 793 nM
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CP0481658
|
2-(3,4-dimethoxyphenyl)-N-[4-methoxy-3-(trifluoromethyl)phenyl]quinazolin-4-amine
Show/Hide
|
C24H20F3N3O3
|
1
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| 1 |
IC50 = 795 nM
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CP0469350
|
3-[[6-amino-2-[3-(trifluoromethyl)phenyl]quinazolin-4-yl]amino]phenol
Show/Hide
|
C21H15F3N4O
|
1
|
| 1 |
IC50 = 799 nM
|
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CP0430535
|
N-(4-bromo-3-methoxyphenyl)-2-(3-nitrophenyl)quinazolin-4-amine
Show/Hide
|
C21H15BrN4O3
|
1
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| 1 |
IC50 = 801 nM
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CP0534954
|
[1-(3,4-difluorophenyl)-1,3,4,9-tetrahydropyrido[3,4-b]indol-2-yl]-(4-methoxyphenyl)methanone
Show/Hide
|
C25H20F2N2O2
|
1
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| 1 |
IC50 = 805 nM
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CP0472569
|
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-6-methyl-2-phenylpyrimidin-4-amine
Show/Hide
|
C19H17N3O2
|
2
|
| 1 |
IC50 = 808 nM
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| 2 |
IC50 = 1630 nM
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CP0388007
|
6,7-dimethoxy-N-(3-nitrophenyl)quinazolin-4-amine
Show/Hide
|
C16H14N4O4
|
2
|
| 1 |
IC50 = 810 nM
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| 2 |
IC50 = 910 nM
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CP0420420
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[3-[(2-pyridin-3-ylquinazolin-4-yl)amino]phenyl]methanol
Show/Hide
|
C20H16N4O
|
1
|
| 1 |
IC50 = 810 nM
|
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CP0383540
|
N,2-bis(3-methoxyphenyl)quinazolin-4-amine
Show/Hide
|
C22H19N3O2
|
1
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| 1 |
IC50 = 811 nM
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CP0550389
|
[1-(3-chlorophenyl)-1,3,4,9-tetrahydropyrido[3,4-b]indol-2-yl]-phenylmethanone
Show/Hide
|
C24H19ClN2O
|
2
|
| 1 |
IC50 = 811 nM
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| 2 |
IC50 = 869 nM
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CP0492412
|
N-(3-chlorophenyl)-6-methyl-2-phenylpyrimidin-4-amine
Show/Hide
|
C17H14ClN3
|
2
|
| 1 |
IC50 = 811 nM
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| 2 |
IC50 = 1000 nM
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CP0037782
|
2-(3,4-dimethoxyphenyl)-3,5,7-trimethoxychromen-4-one
Show/Hide
|
C20H20O7
|
2
|
| 1 |
IC50 = 822 nM
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|
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| 2 |
IC50 = 1880 nM
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CP0490375
|
(4-Chloro-phenyl)-(2-phenyl-quinazolin-4-yl)-amine
Show/Hide
|
C20H14ClN3
|
1
|
| 1 |
IC50 = 830 nM
|
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CP0435283
|
4-N-(3-methoxyphenyl)-2-[3-(trifluoromethyl)phenyl]quinazoline-4,6-diamine
Show/Hide
|
C22H17F3N4O
|
1
|
| 1 |
IC50 = 835 nM
|
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CP0380380
|
(E)-3-(3,4-dimethoxyphenyl)-1-[4-(quinazolin-4-ylamino)phenyl]prop-2-en-1-one
Show/Hide
|
C25H21N3O3
|
1
|
| 1 |
IC50 = 840 nM
|
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CP0482675
|
4-[(2-phenylquinolin-4-yl)amino]benzonitrile
Show/Hide
|
C22H15N3
|
1
|
| 1 |
IC50 = 846 nM
|
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CP0161706
|
(E)-1-(2,4-dihydroxyphenyl)-3-(3,4-dimethoxyphenyl)prop-2-en-1-one
Show/Hide
|
C17H16O5
|
1
|
| 1 |
IC50 = 850 nM
|
|
|
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CP0472568
|
N-(3-fluoro-4-methoxyphenyl)-6-methyl-2-phenylpyrimidin-4-amine
Show/Hide
|
C18H16FN3O
|
2
|
| 1 |
IC50 = 861 nM
|
|
|
| 2 |
IC50 = 1310 nM
|
|
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CP0547394
|
N-(4-methoxyphenyl)-6-methyl-2-pyridin-4-ylpyrimidin-4-amine
Show/Hide
|
C17H16N4O
|
1
|
| 1 |
IC50 = 874 nM
|
|
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CP0513311
|
4-[[2-(3-methoxyphenyl)pyrido[2,3-d]pyrimidin-4-yl]amino]benzonitrile
Show/Hide
|
C21H15N5O
|
1
|
| 1 |
IC50 = 876 nM
|
|
|
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CP0401965
|
(E)-3-(3-methoxyphenyl)-1-[4-[(2-phenylquinazolin-4-yl)amino]phenyl]prop-2-en-1-one
Show/Hide
|
C30H23N3O2
|
1
|
| 1 |
IC50 = 880 nM
|
|
|
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CP0389670
|
N,2-diphenylquinazolin-4-amine
Show/Hide
|
C20H15N3
|
2
|
| 1 |
IC50 = 882 nM
|
|
|
| 2 |
IC50 = 2570 nM
|
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CP0446424
|
[1-(3-chlorophenyl)-1,3,4,9-tetrahydropyrido[3,4-b]indol-2-yl]-(4-methoxyphenyl)methanone
Show/Hide
|
C25H21ClN2O2
|
1
|
| 1 |
IC50 = 883 nM
|
|
|
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CP0388008
|
N-(3-nitrophenyl)quinazolin-4-amine
Show/Hide
|
C14H10N4O2
|
2
|
| 1 |
IC50 = 890 nM
|
|
|
| 2 |
IC50 = 1130 nM
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CP0454935
|
(E)-3-(4-methoxyphenyl)-1-[3-(quinazolin-4-ylamino)phenyl]prop-2-en-1-one
Show/Hide
|
C24H19N3O2
|
1
|
| 1 |
IC50 = 890 nM
|
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CP0518999
|
3-[(6-nitro-2-phenylquinazolin-4-yl)amino]benzoic acid
Show/Hide
|
C21H14N4O4
|
1
|
| 1 |
IC50 = 904 nM
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CP0567254
|
2-(3-methoxyphenyl)-N-(3-methylsulfanylphenyl)pyrido[2,3-d]pyrimidin-4-amine
Show/Hide
|
C21H18N4OS
|
1
|
| 1 |
IC50 = 910 nM
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CP0390685
|
(E)-3-phenyl-1-[4-[(2-phenylquinazolin-4-yl)amino]phenyl]prop-2-en-1-one
Show/Hide
|
C29H21N3O
|
1
|
| 1 |
IC50 = 920 nM
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CP0407965
|
[3-[(2-pyridin-4-ylquinazolin-4-yl)amino]phenyl]methanol
Show/Hide
|
C20H16N4O
|
1
|
| 1 |
IC50 = 921 nM
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CP0130380
|
3-[(6,7-dimethoxyquinazolin-4-yl)amino]benzonitrile
Show/Hide
|
C17H14N4O2
|
2
|
| 1 |
IC50 = 930 nM
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| 2 |
IC50 = 1060 nM
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CP0288954
|
4-Anilino quinazoline deriv. 17
Show/Hide
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C15H10F3N3
|
2
|
| 1 |
IC50 = 940 nM
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| 2 |
IC50 = 1550 nM
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CP0451195
|
4-(2-Phenyl-quinazolin-4-ylamino)-benzoic acid methyl ester
Show/Hide
|
C22H17N3O2
|
1
|
| 1 |
IC50 = 944 nM
|
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CP0490379
|
N-(3-methoxyphenyl)-2-phenylquinolin-4-amine
Show/Hide
|
C22H18N2O
|
1
|
| 1 |
IC50 = 951 nM
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CP0420846
|
N-(3-fluorophenyl)-2-thiophen-2-ylquinazolin-4-amine
Show/Hide
|
C18H12FN3S
|
1
|
| 1 |
IC50 = 953 nM
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CP0567253
|
3-[[2-(3-methoxyphenyl)pyrido[2,3-d]pyrimidin-4-yl]amino]phenol
Show/Hide
|
C20H16N4O2
|
1
|
| 1 |
IC50 = 963 nM
|
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CP0531581
|
(E)-3-(4-methoxyphenyl)-1-[3-[(2-phenylquinazolin-4-yl)amino]phenyl]prop-2-en-1-one
Show/Hide
|
C30H23N3O2
|
1
|
| 1 |
IC50 = 970 nM
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CP0574768
|
2-phenyl-4-[3-(trifluoromethyl)phenoxy]quinazoline
Show/Hide
|
C21H13F3N2O
|
1
|
| 1 |
IC50 = 989 nM
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CP0424484
|
2-nitro-N-(2-phenylquinazolin-4-yl)benzamide
Show/Hide
|
C21H14N4O3
|
1
|
| 1 |
IC50 = 994 nM
|
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CP0500848
|
2-(3,4-Dimethoxy-phenyl)-3-hydroxy-7-methoxy-chromen-4-one
Show/Hide
|
C18H16O6
|
2
|
| 1 |
IC50 = 1010 nM
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| 2 |
IC50 = 1770 nM
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CP0387304
|
N-(3-methoxyphenyl)-2-pyridin-3-ylquinazolin-4-amine
Show/Hide
|
C20H16N4O
|
1
|
| 1 |
IC50 = 1020 nM
|
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CP0441261
|
(E)-1-(2,4-dimethoxyphenyl)-3-(3,4-dimethoxyphenyl)prop-2-en-1-one
Show/Hide
|
C19H20O5
|
1
|
| 1 |
IC50 = 1030 nM
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CP0475286
|
(4-chlorophenyl)-[1-(3,4-dichlorophenyl)-1,3,4,9-tetrahydropyrido[3,4-b]indol-2-yl]methanone
Show/Hide
|
C24H17Cl3N2O
|
1
|
| 1 |
IC50 = 1030 nM
|
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CP0533355
|
N-[4-(3-methoxyanilino)-2-pyridin-3-ylquinazolin-6-yl]pyridine-3-carboxamide
Show/Hide
|
C26H20N6O2
|
1
|
| 1 |
IC50 = 1040 nM
|
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CP0147681
|
(E)-3-(3,4-dimethoxyphenyl)-1-(2-hydroxy-4-methoxyphenyl)prop-2-en-1-one
Show/Hide
|
C18H18O5
|
1
|
| 1 |
IC50 = 1060 nM
|
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CP0376009
|
3-methoxy-2-(4-methoxyphenyl)benzo[h]chromen-4-one
Show/Hide
|
C21H16O4
|
2
|
| 1 |
IC50 = 1060 nM
|
|
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| 2 |
IC50 = 3070 nM
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CP0407966
|
N-(3,4-dimethoxyphenyl)-2-pyridin-2-ylquinazolin-4-amine
Show/Hide
|
C21H18N4O2
|
1
|
| 1 |
IC50 = 1060 nM
|
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CP0476081
|
N-[2-(2-phenyltetrazol-5-yl)phenyl]adamantane-1-carboxamide
Show/Hide
|
C24H25N5O
|
1
|
| 1 |
IC50 = 1060 nM
|
|
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CP0451206
|
N-(4-fluorophenyl)-2-phenylquinazolin-4-amine
Show/Hide
|
C20H14FN3
|
1
|
| 1 |
IC50 = 1060 nM
|
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CP0544530
|
N-(4-tert-butylphenyl)-2-phenylquinazolin-4-amine
Show/Hide
|
C24H23N3
|
1
|
| 1 |
IC50 = 1060 nM
|
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CP0563542
|
3-[(2-pyridin-4-ylquinazolin-4-yl)amino]phenol
Show/Hide
|
C19H14N4O
|
1
|
| 1 |
IC50 = 1070 nM
|
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CP0532849
|
N-(3-tert-butylphenyl)-2-phenylquinazolin-4-amine
Show/Hide
|
C24H23N3
|
1
|
| 1 |
IC50 = 1070 nM
|
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CP0153516
|
4-Anilino quinazoline deriv. 15
Show/Hide
|
C14H10BrN3
|
2
|
| 1 |
IC50 = 1080 nM
|
|
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| 2 |
IC50 = 1480 nM
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CP0544644
|
(E)-1-[4-[[2-(3,4-dimethoxyphenyl)quinazolin-4-yl]amino]phenyl]-3-phenylprop-2-en-1-one
Show/Hide
|
C31H25N3O3
|
1
|
| 1 |
IC50 = 1090 nM
|
|
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CP0475281
|
[1-(3,4-difluorophenyl)-1,3,4,9-tetrahydropyrido[3,4-b]indol-2-yl]-phenylmethanone
Show/Hide
|
C24H18F2N2O
|
2
|
| 1 |
IC50 = 1100 nM
|
|
|
| 2 |
IC50 = 1800 nM
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CP0475283
|
[1-(3,4-difluorophenyl)-1,3,4,9-tetrahydropyrido[3,4-b]indol-2-yl]-(3,4-dimethoxyphenyl)methanone
Show/Hide
|
C26H22F2N2O3
|
1
|
| 1 |
IC50 = 1100 nM
|
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CP0385411
|
(E)-3-(4-chlorophenyl)-1-(2,4-dimethoxyphenyl)prop-2-en-1-one
Show/Hide
|
C17H15ClO3
|
1
|
| 1 |
IC50 = 1130 nM
|
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CP0202859
|
2-(3,4-dimethoxyphenyl)benzo[h]chromen-4-one
Show/Hide
|
C21H16O4
|
2
|
| 1 |
IC50 = 1130 nM
|
|
|
| 2 |
IC50 = 1230 nM
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CP0482660
|
N-[4-(3-methoxyanilino)-2-pyridin-3-ylquinazolin-6-yl]-3-nitrobenzamide
Show/Hide
|
C27H20N6O4
|
1
|
| 1 |
IC50 = 1150 nM
|
|
|
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CP0163255
|
N-(3-methylphenyl)-2-phenylquinazolin-4-amine
Show/Hide
|
C21H17N3
|
1
|
| 1 |
IC50 = 1150 nM
|
|
|
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CP0480465
|
(E)-1-(3',4'-Dimethoxyphenyl)-3-(4''-methoxyphenyl)prop-2-en-1-one
Show/Hide
|
C18H18O4
|
1
|
| 1 |
IC50 = 1160 nM
|
|
|
|
CP0434804
|
2-(3,4-dimethoxyphenyl)-3-methoxychromen-4-one
Show/Hide
|
C18H16O5
|
2
|
| 1 |
IC50 = 1180 nM
|
|
|
| 2 |
IC50 = 1340 nM
|
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|
|
CP0500657
|
FISETIN TETRAMETHYL ETHER
Show/Hide
|
C19H18O6
|
2
|
| 1 |
IC50 = 1180 nM
|
|
|
| 2 |
IC50 = 2140 nM
|
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|
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CP0435467
|
3-(quinazolin-4-ylamino)benzonitrile
Show/Hide
|
C15H10N4
|
2
|
| 1 |
IC50 = 1180 nM
|
|
|
| 2 |
IC50 = 2030 nM
|
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CP0430540
|
N-(4-fluoro-3-nitrophenyl)-2-(3-methoxyphenyl)quinazolin-4-amine
Show/Hide
|
C21H15FN4O3
|
1
|
| 1 |
IC50 = 1190 nM
|
|
|
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CP0451205
|
N-(3-methylsulfanylphenyl)-2-phenylquinazolin-4-amine
Show/Hide
|
C21H17N3S
|
1
|
| 1 |
IC50 = 1190 nM
|
|
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CP0469971
|
3-N,3-N-dimethyl-1-N-(2-pyridin-3-ylquinazolin-4-yl)benzene-1,3-diamine
Show/Hide
|
C21H19N5
|
1
|
| 1 |
IC50 = 1200 nM
|
|
|
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CP0322898
|
3-methoxy-2-phenylchromen-4-one
Show/Hide
|
C16H12O3
|
2
|
| 1 |
IC50 = 1210 nM
|
|
|
| 2 |
IC50 = 1280 nM
|
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|
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CP0414694
|
(E)-3-(3,4-dimethoxyphenyl)-1-[4-[(6,7-dimethoxyquinazolin-4-yl)amino]phenyl]prop-2-en-1-one
Show/Hide
|
C27H25N3O5
|
1
|
| 1 |
IC50 = 1230 nM
|
|
|
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CP0463654
|
3-[(2-phenylpyrido[2,3-d]pyrimidin-4-yl)amino]phenol
Show/Hide
|
C19H14N4O
|
1
|
| 1 |
IC50 = 1230 nM
|
|
|
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CP0568917
|
N-(3-fluorophenyl)-2-pyridin-3-ylpyrido[2,3-d]pyrimidin-4-amine
Show/Hide
|
C18H12FN5
|
1
|
| 1 |
IC50 = 1230 nM
|
|
|
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CP0475293
|
(4-methoxyphenyl)-[1-[4-(trifluoromethyl)phenyl]-1,3,4,9-tetrahydropyrido[3,4-b]indol-2-yl]methanone
Show/Hide
|
C26H21F3N2O2
|
1
|
| 1 |
IC50 = 1230 nM
|
|
|
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CP0509629
|
4-[[2-(3-methoxyphenyl)pyrido[2,3-d]pyrimidin-4-yl]amino]-2-nitrophenol
Show/Hide
|
C20H15N5O4
|
1
|
| 1 |
IC50 = 1260 nM
|
|
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CP0538637
|
(4-chlorophenyl)-[1-(3,4-difluorophenyl)-1,3,4,9-tetrahydropyrido[3,4-b]indol-2-yl]methanone
Show/Hide
|
C24H17ClF2N2O
|
1
|
| 1 |
IC50 = 1260 nM
|
|
|
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CP0424487
|
4-(quinazolin-4-ylamino)benzonitrile
Show/Hide
|
C15H10N4
|
1
|
| 1 |
IC50 = 1270 nM
|
|
|
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CP0074049
|
2-(4-methoxyphenyl)benzo[h]chromen-4-one
Show/Hide
|
C20H14O3
|
2
|
| 1 |
IC50 = 1280 nM
|
|
|
| 2 |
IC50 = 1290 nM
|
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CP0390684
|
(E)-3-(3,4-dimethoxyphenyl)-1-[3-(quinazolin-4-ylamino)phenyl]prop-2-en-1-one
Show/Hide
|
C25H21N3O3
|
1
|
| 1 |
IC50 = 1300 nM
|
|
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CP0568915
|
4-[[2-(3-methoxyphenyl)pyrido[2,3-d]pyrimidin-4-yl]amino]phenol
Show/Hide
|
C20H16N4O2
|
1
|
| 1 |
IC50 = 1300 nM
|
|
|
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CP0038890
|
2-PHENYL-4H-BENZO[H]CHROMEN-4-ONE
Show/Hide
|
C19H12O2
|
2
|
| 1 |
IC50 = 1310 nM
|
|
|
| 2 |
IC50 = 1400 nM
|
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CP0451598
|
(3-methoxyphenyl)-(2-phenylquinazolin-4-yl)amine
Show/Hide
|
C21H17N3O
|
1
|
| 1 |
IC50 = 1320 nM
|
|
|
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CP0446429
|
[1-(3,4-dichlorophenyl)-1,3,4,9-tetrahydropyrido[3,4-b]indol-2-yl]-naphthalen-1-ylmethanone
Show/Hide
|
C28H20Cl2N2O
|
1
|
| 1 |
IC50 = 1320 nM
|
|
|
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CP0424488
|
N-(3-methylsulfanylphenyl)quinazolin-4-amine
Show/Hide
|
C15H13N3S
|
1
|
| 1 |
IC50 = 1350 nM
|
|
|
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CP0565502
|
3-[(2-pyridin-4-ylquinazolin-4-yl)amino]benzenesulfonyl fluoride
Show/Hide
|
C19H13FN4O2S
|
1
|
| 1 |
IC50 = 1380 nM
|
|
|
|
CP0459141
|
N-(2-methyl-1,3-benzothiazol-5-yl)-1-(6-pyrazol-1-ylpyrimidin-4-yl)piperidine-3-carboxamide
Show/Hide
|
C21H21N7OS
|
1
|
| 1 |
IC50 = 1390 nM
|
|
|
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CP0549212
|
[1-(4-methylphenyl)-1,3,4,9-tetrahydropyrido[3,4-b]indol-2-yl]-phenylmethanone
Show/Hide
|
C25H22N2O
|
1
|
| 1 |
IC50 = 1430 nM
|
|
|
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CP0474211
|
(4-methoxyphenyl)-[1-(3-methoxyphenyl)-1,3,4,9-tetrahydropyrido[3,4-b]indol-2-yl]methanone
Show/Hide
|
C26H24N2O3
|
1
|
| 1 |
IC50 = 1450 nM
|
|
|
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CP0553012
|
N-(4-iodo-3-methylphenyl)-2-phenylquinazolin-4-amine
Show/Hide
|
C21H16IN3
|
1
|
| 1 |
IC50 = 1460 nM
|
|
|
|
CP0201213
|
(E)-1-(2-hydroxy-4-methoxyphenyl)-3-(3-methoxyphenyl)prop-2-en-1-one
Show/Hide
|
C17H16O4
|
1
|
| 1 |
IC50 = 1470 nM
|
|
|
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CP0042674
|
N-(4-methylphenyl)-2-phenylquinazolin-4-amine
Show/Hide
|
C21H17N3
|
1
|
| 1 |
IC50 = 1480 nM
|
|
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CP0484130
|
2-N,4-N-bis(3,4-dimethoxyphenyl)-6,7-dimethoxyquinazoline-2,4-diamine
Show/Hide
|
C26H28N4O6
|
2
|
| 1 |
IC50 = 1520 nM
|
|
|
| 2 |
IC50 = 1740 nM
|
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CP0513289
|
2-phenyl-N-[4-(trifluoromethyl)phenyl]quinazolin-4-amine
Show/Hide
|
C21H14F3N3
|
1
|
| 1 |
IC50 = 1530 nM
|
|
|
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CP0567255
|
N-(3-bromophenyl)-2-(3-methoxyphenyl)pyrido[2,3-d]pyrimidin-4-amine
Show/Hide
|
C20H15BrN4O
|
1
|
| 1 |
IC50 = 1530 nM
|
|
|
|
CP0397339
|
3-hydroxy-2-phenylbenzo[h]chromen-4-one
Show/Hide
|
C19H12O3
|
2
|
| 1 |
IC50 = 1590 nM
|
|
|
| 2 |
IC50 = 2890 nM
|
|
|
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CP0566441
|
N-[4-(4-methoxyanilino)-2-pyridin-3-ylquinazolin-6-yl]-3-nitrobenzamide
Show/Hide
|
C27H20N6O4
|
1
|
| 1 |
IC50 = 1620 nM
|
|
|
|
CP0387202
|
N-(3-methoxyphenyl)-2-pyridin-2-ylquinazolin-4-amine
Show/Hide
|
C20H16N4O
|
1
|
| 1 |
IC50 = 1630 nM
|
|
|
|
CP0490376
|
N-[3-[(2-phenylquinolin-4-yl)amino]phenyl]acetamide
Show/Hide
|
C23H19N3O
|
1
|
| 1 |
IC50 = 1630 nM
|
|
|
|
CP0393136
|
N-(3-fluorophenyl)-2-(3-methoxyphenyl)quinazolin-4-amine
Show/Hide
|
C21H16FN3O
|
1
|
| 1 |
IC50 = 1640 nM
|
|
|
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CP0565812
|
N-(3-chloro-4-fluorophenyl)-2-phenylquinazolin-4-amine
Show/Hide
|
C20H13ClFN3
|
1
|
| 1 |
IC50 = 1660 nM
|
|
|
|
CP0434803
|
3-(4-methoxyphenyl)benzo[f]chromen-1-one
Show/Hide
|
C20H14O3
|
2
|
| 1 |
IC50 = 1690 nM
|
|
|
| 2 |
IC50 = 2460 nM
|
|
|
|
CP0469626
|
(E)-3-(3,4-dimethoxyphenyl)-1-[3-[(6,7-dimethoxyquinazolin-4-yl)amino]phenyl]prop-2-en-1-one
Show/Hide
|
C27H25N3O5
|
1
|
| 1 |
IC50 = 1710 nM
|
|
|
|
CP0395784
|
(E)-3-(4-chlorophenyl)-1-(3,4-dimethoxyphenyl)prop-2-en-1-one
Show/Hide
|
C17H15ClO3
|
1
|
| 1 |
IC50 = 1730 nM
|
|
|
|
CP0011998
|
N-(3-bromophenyl)-6,7-dimethoxyquinazolin-4-amine
Show/Hide
|
C16H14BrN3O2
|
2
|
| 1 |
IC50 = 1730 nM
|
|
|
| 2 |
IC50 = 2320 nM
|
|
|
|
CP0534186
|
(4-methoxyphenyl)-(1-phenyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-2-yl)methanone
Show/Hide
|
C25H22N2O2
|
1
|
| 1 |
IC50 = 1750 nM
|
|
|
|
CP0430536
|
N-(4-iodophenyl)-2-(3-nitrophenyl)quinazolin-4-amine
Show/Hide
|
C20H13IN4O2
|
1
|
| 1 |
IC50 = 1770 nM
|
|
|
|
CP0446425
|
[1-(4-bromophenyl)-1,3,4,9-tetrahydropyrido[3,4-b]indol-2-yl]-(4-chlorophenyl)methanone
Show/Hide
|
C24H18BrClN2O
|
1
|
| 1 |
IC50 = 1780 nM
|
|
|
|
CP0475296
|
[1-(4-fluorophenyl)-1,3,4,9-tetrahydropyrido[3,4-b]indol-2-yl]-phenylmethanone
Show/Hide
|
C24H19FN2O
|
1
|
| 1 |
IC50 = 1890 nM
|
|
|
|
CP0528179
|
N-(3-methylsulfanylphenyl)-2-phenylquinolin-4-amine
Show/Hide
|
C22H18N2S
|
1
|
| 1 |
IC50 = 1900 nM
|
|
|
|
CP0342156
|
(E)-1-(2',4'-Dimethoxyphenyl)-3-(4''-methoxyphenyl)prop-2-en-1-one
Show/Hide
|
C18H18O4
|
1
|
| 1 |
IC50 = 1910 nM
|
|
|
|
CP0446422
|
[1-(3-methoxyphenyl)-1,3,4,9-tetrahydropyrido[3,4-b]indol-2-yl]-phenylmethanone
Show/Hide
|
C25H22N2O2
|
1
|
| 1 |
IC50 = 1920 nM
|
|
|
|
CP0418765
|
(E)-1-(2-hydroxynaphthalen-1-yl)-3-(3-methoxyphenyl)prop-2-en-1-one
Show/Hide
|
C20H16O3
|
1
|
| 1 |
IC50 = 1930 nM
|
|
|
|
CP0495661
|
N-(4-methoxyphenyl)-2-phenylquinazolin-4-amine
Show/Hide
|
C21H17N3O
|
1
|
| 1 |
IC50 = 1930 nM
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|
CP0523464
|
(3-Chloro-phenyl)-(2-phenyl-quinazolin-4-yl)-amine; hydrochloride
Show/Hide
|
C20H14ClN3
|
1
|
| 1 |
IC50 = 1930 nM
|
|
|
|
CP0389298
|
(E)-1-(2,4-dihydroxyphenyl)-3-(3-methoxyphenyl)prop-2-en-1-one
Show/Hide
|
C16H14O4
|
1
|
| 1 |
IC50 = 1940 nM
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|
|
CP0441263
|
(E)-3-(3,4-dimethoxyphenyl)-1-(1-hydroxynaphthalen-2-yl)prop-2-en-1-one
Show/Hide
|
C21H18O4
|
1
|
| 1 |
IC50 = 1950 nM
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|
|
CP0033751
|
6,7-dimethoxy-N-[3-(trifluoromethyl)phenyl]quinazolin-4-amine
Show/Hide
|
C17H14F3N3O2
|
2
|
| 1 |
IC50 = 1980 nM
|
|
|
| 2 |
IC50 = 2400 nM
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CP0484129
|
2-(3,4-dimethoxyphenyl)-N-phenylquinazolin-4-amine
Show/Hide
|
C22H19N3O2
|
2
|
| 1 |
IC50 = 1990 nM
|
|
|
| 2 |
IC50 = 4090 nM
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CP0530754
|
3-(2-benzoyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl)benzonitrile
Show/Hide
|
C25H19N3O
|
1
|
| 1 |
IC50 = 2000 nM
|
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|
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CP0424483
|
N-methyl-N-(3-nitrophenyl)-2-phenylquinazolin-4-amine
Show/Hide
|
C21H16N4O2
|
1
|
| 1 |
IC50 = 2025 nM
|
|
|
|
CP0509628
|
4-[(2-phenylpyrido[2,3-d]pyrimidin-4-yl)amino]phenol
Show/Hide
|
C19H14N4O
|
1
|
| 1 |
IC50 = 2040 nM
|
|
|
|
CP0393130
|
3-[[2-(4-methoxyphenyl)quinazolin-4-yl]amino]benzonitrile
Show/Hide
|
C22H16N4O
|
1
|
| 1 |
IC50 = 2120 nM
|
|
|
|
CP0553013
|
N-(3-fluorophenyl)-2-phenylquinolin-4-amine
Show/Hide
|
C21H15FN2
|
1
|
| 1 |
IC50 = 2130 nM
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|
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CP0393138
|
N-(3-methoxyphenyl)-2-(4-methoxyphenyl)quinazolin-4-amine
Show/Hide
|
C22H19N3O2
|
1
|
| 1 |
IC50 = 2140 nM
|
|
|
|
CP0043433
|
1-(2-hydroxy-4-methoxyphenyl)-3-(4-methoxyphenyl)prop-2-en-1-one
Show/Hide
|
C17H16O4
|
1
|
| 1 |
IC50 = 2200 nM
|
|
|
|
CP0475295
|
[1-(4-methoxyphenyl)-1,3,4,9-tetrahydropyrido[3,4-b]indol-2-yl]-phenylmethanone
Show/Hide
|
C25H22N2O2
|
1
|
| 1 |
IC50 = 2210 nM
|
|
|
|
CP0124818
|
N-(2-methoxyphenyl)-2-phenylquinazolin-4-amine
Show/Hide
|
C21H17N3O
|
1
|
| 1 |
IC50 = 2250 nM
|
|
|
|
CP0406748
|
3-methoxy-2-phenylbenzo[h]chromen-4-one
Show/Hide
|
C20H14O3
|
2
|
| 1 |
IC50 = 2310 nM
|
|
|
| 2 |
IC50 = 2710 nM
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|
CP0555177
|
[1-(2-methylpropyl)-1,3,4,9-tetrahydropyrido[3,4-b]indol-2-yl]-phenylmethanone
Show/Hide
|
C22H24N2O
|
1
|
| 1 |
IC50 = 2330 nM
|
|
|
|
CP0529200
|
4-methoxy-N-[2-[4-(4-methoxyphenyl)triazol-1-yl]phenyl]benzamide
Show/Hide
|
C23H20N4O3
|
1
|
| 1 |
IC50 = 2360 nM
|
|
|
|
CP0434124
|
2-(4-fluoro-3-methoxyphenyl)-3-methoxybenzo[h]chromen-4-one
Show/Hide
|
C21H15FO4
|
2
|
| 1 |
IC50 = 2440 nM
|
|
|
| 2 |
IC50 = 4010 nM
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|
|
|
CP0553476
|
N-(4-fluoro-3-nitrophenyl)-2-phenylquinazolin-4-amine
Show/Hide
|
C20H13FN4O2
|
1
|
| 1 |
IC50 = 2460 nM
|
|
|
|
CP0442378
|
6,7-dimethoxy-N-(4-nitrophenyl)quinazolin-4-amine
Show/Hide
|
C16H14N4O4
|
2
|
| 1 |
IC50 = 2460 nM
|
|
|
| 2 |
IC50 = 2920 nM
|
|
|
|
CP0487638
|
2-[4-[(6-methyl-2-phenylpyrimidin-4-yl)amino]phenyl]acetonitrile
Show/Hide
|
C19H16N4
|
2
|
| 1 |
IC50 = 2500 nM
|
|
|
| 2 |
IC50 = 3620 nM
|
|
|
|
CP0548060
|
[3-[(6-methyl-2-phenylpyrimidin-4-yl)amino]phenyl]methanol
Show/Hide
|
C18H17N3O
|
2
|
| 1 |
IC50 = 2520 nM
|
|
|
| 2 |
IC50 = 4220 nM
|
|
|
|
CP0420848
|
N-(4-methoxyphenyl)-2-(1H-pyrrol-2-yl)quinazolin-4-amine
Show/Hide
|
C19H16N4O
|
1
|
| 1 |
IC50 = 2570 nM
|
|
|
|
CP0428495
|
(E)-1-(2-hydroxynaphthalen-1-yl)-3-phenylprop-2-en-1-one
Show/Hide
|
C19H14O2
|
1
|
| 1 |
IC50 = 2580 nM
|
|
|
|
CP0418784
|
(E)-3-(2-chlorophenyl)-1-(2,4-dimethoxyphenyl)prop-2-en-1-one
Show/Hide
|
C17H15ClO3
|
1
|
| 1 |
IC50 = 2630 nM
|
|
|
|
CP0424486
|
4-(quinazolin-4-ylamino)phenol
Show/Hide
|
C14H11N3O
|
1
|
| 1 |
IC50 = 2630 nM
|
|
|
|
CP0508457
|
N-cyclohexyl-2-(3-nitrophenyl)quinazolin-4-amine
Show/Hide
|
C20H20N4O2
|
1
|
| 1 |
IC50 = 2780 nM
|
|
|
|
CP0446487
|
phenyl-(1-phenyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-2-yl)methanone
Show/Hide
|
C24H20N2O
|
1
|
| 1 |
IC50 = 2780 nM
|
|
|
|
CP0389850
|
(E)-3-(2-chlorophenyl)-1-(2-hydroxy-4,6-dimethoxyphenyl)prop-2-en-1-one
Show/Hide
|
C17H15ClO4
|
1
|
| 1 |
IC50 = 2820 nM
|
|
|
|
CP0387978
|
(E)-1-(2-hydroxynaphthalen-1-yl)-3-(4-methoxyphenyl)prop-2-en-1-one
Show/Hide
|
C20H16O3
|
1
|
| 1 |
IC50 = 2890 nM
|
|
|
|
CP0545310
|
2-nitro-4-(quinazolin-4-ylamino)phenol
Show/Hide
|
C14H10N4O3
|
1
|
| 1 |
IC50 = 2900 nM
|
|
|
|
CP0202456
|
FLAVOKAWAIN A
Show/Hide
|
C18H18O5
|
1
|
| 1 |
IC50 = 3000 nM
|
|
|
|
CP0406747
|
2-methoxy-3-(4-methoxyphenyl)benzo[f]chromen-1-one
Show/Hide
|
C21H16O4
|
2
|
| 1 |
IC50 = 3070 nM
|
|
|
| 2 |
IC50 = 8020 nM
|
|
|
|
CP0409714
|
(E)-1-[4-[[2-(3,4-dimethoxyphenyl)quinazolin-4-yl]amino]phenyl]-3-(4-methoxyphenyl)prop-2-en-1-one
Show/Hide
|
C32H27N3O4
|
1
|
| 1 |
IC50 = 3130 nM
|
|
|
|
CP0036082
|
N-(3-chloro-4-fluorophenyl)-7-methoxy-6-(3-morpholin-4-ylpropoxy)quinazolin-4-amine
Show/Hide
|
C22H24ClFN4O3
|
1
|
| 1 |
IC50 = 3190 nM
|
|
|
|
CP0383768
|
N-[2-[2-(4-methoxyphenyl)tetrazol-5-yl]phenyl]acetamide
Show/Hide
|
C16H15N5O2
|
1
|
| 1 |
IC50 = 3230 nM
|
|
|
|
CP0406746
|
MORIN PENTAMETHYL ETHER
Show/Hide
|
C19H18O7
|
2
|
| 1 |
IC50 = 3270 nM
|
|
|
| 2 |
IC50 = 3890 nM
|
|
|
|
CP0418786
|
(E)-1-(2,4-dihydroxyphenyl)-3-(2-chlorophenyl)-2-propen-1-one (6)
Show/Hide
|
C15H11ClO3
|
1
|
| 1 |
IC50 = 3280 nM
|
|
|
|
CP0441258
|
(E)-3-(2-chlorophenyl)-1-(2-hydroxy-4-methoxyphenyl)prop-2-en-1-one
Show/Hide
|
C16H13ClO3
|
1
|
| 1 |
IC50 = 3320 nM
|
|
|
|
CP0422923
|
N-(3,4-dimethoxyphenyl)quinazolin-4-amine
Show/Hide
|
C16H15N3O2
|
2
|
| 1 |
IC50 = 3380 nM
|
|
|
| 2 |
IC50 = 4790 nM
|
|
|
|
CP0409715
|
(E)-3-(4-methoxyphenyl)-1-[4-[(2-phenylquinazolin-4-yl)amino]phenyl]prop-2-en-1-one
Show/Hide
|
C30H23N3O2
|
1
|
| 1 |
IC50 = 3550 nM
|
|
|
|
CP0455724
|
[1-(3,4-dimethoxyphenyl)-1,3,4,9-tetrahydropyrido[3,4-b]indol-2-yl]-phenylmethanone
Show/Hide
|
C26H24N2O3
|
1
|
| 1 |
IC50 = 3620 nM
|
|
|
|
CP0450326
|
N-[2-(2-phenyltetrazol-5-yl)phenyl]-4-(trifluoromethyl)benzamide
Show/Hide
|
C21H14F3N5O
|
2
|
| 1 |
IC50 = 3630 nM
|
|
|
| 2 |
IC50 = 4390 nM
|
|
|
|
CP0523151
|
N-methyl-N-(4-nitrophenyl)-2-phenylquinazolin-4-amine
Show/Hide
|
C21H16N4O2
|
1
|
| 1 |
IC50 = 3669 nM
|
|
|
|
CP0516043
|
N-(2-bromophenyl)-2-phenylquinazolin-4-amine
Show/Hide
|
C20H14BrN3
|
1
|
| 1 |
IC50 = 3750 nM
|
|
|
|
CP0020298
|
(3,4-Dimethoxy-phenyl)-(6,7-dimethoxy-quinazolin-4-yl)-amine
Show/Hide
|
C18H19N3O4
|
2
|
| 1 |
IC50 = 3790 nM
|
|
|
| 2 |
IC50 = 7380 nM
|
|
|
|
CP0197181
|
(E)-1,3-bis(3,4-dimethoxyphenyl)prop-2-en-1-one
Show/Hide
|
C19H20O5
|
1
|
| 1 |
IC50 = 3800 nM
|
|
|
|
CP0435465
|
6,7-dimethoxy-N-(2-nitrophenyl)quinazolin-4-amine
Show/Hide
|
C16H14N4O4
|
2
|
| 1 |
IC50 = 3800 nM
|
|
|
| 2 |
IC50 = 3970 nM
|
|
|
|
CP0528982
|
4-(3-bromophenoxy)-2-phenylquinazoline
Show/Hide
|
C20H13BrN2O
|
1
|
| 1 |
IC50 = 3860 nM
|
|
|
|
CP0528983
|
N-(3-fluorophenyl)-N-methyl-2-phenylquinazolin-4-amine
Show/Hide
|
C21H16FN3
|
1
|
| 1 |
IC50 = 3948 nM
|
|
|
|
CP0534245
|
4-(4-methylpiperazin-1-yl)-6,7,8,9-tetrahydropyrimido[4,5-b]indolizine-10-carbonitrile
Show/Hide
|
C16H20N6
|
1
|
| 1 |
IC50 = 4250 nM
|
|
|
|
CP0547392
|
4-[(2-pyridin-4-ylquinazolin-4-yl)amino]phenol
Show/Hide
|
C19H14N4O
|
1
|
| 1 |
IC50 = 4260 nM
|
|
|
|
CP0434802
|
3-(3,4-dimethoxyphenyl)-2-methoxybenzo[f]chromen-1-one
Show/Hide
|
C22H18O5
|
2
|
| 1 |
IC50 = 4270 nM
|
|
|
| 2 |
IC50 = 5250 nM
|
|
|
|
CP0446427
|
[1-(2-fluorophenyl)-1,3,4,9-tetrahydropyrido[3,4-b]indol-2-yl]-phenylmethanone
Show/Hide
|
C24H19FN2O
|
1
|
| 1 |
IC50 = 4490 nM
|
|
|
|
CP0504951
|
4-(4-benzylpiperazin-1-yl)-5,6-di(cycloheptyl)pyrrolo[3,2-d]pyrimidine-7-carbonitrile
Show/Hide
|
C32H42N6
|
1
|
| 1 |
IC50 = 4680 nM
|
|
|
|
CP0559002
|
4-(3-nitrophenoxy)-2-phenylquinazoline
Show/Hide
|
C20H13N3O3
|
1
|
| 1 |
IC50 = 4780 nM
|
|
|
|
CP0406745
|
3-(3,4-dimethoxyphenyl)-2-hydroxybenzo[f]chromen-1-one
Show/Hide
|
C21H16O5
|
2
|
| 1 |
IC50 = 4840 nM
|
|
|
| 2 |
IC50 = 6120 nM
|
|
|
|
CP0418783
|
Chalcone, 9
Show/Hide
|
C17H16O4
|
1
|
| 1 |
IC50 = 4970 nM
|
|
|
|
CP0434801
|
3-hydroxy-2-(4-methoxyphenyl)benzo[h]chromen-4-one
Show/Hide
|
C20H14O4
|
2
|
| 1 |
IC50 = 4970 nM
|
|
|
| 2 |
IC50 = 6930 nM
|
|
|
|
CP0019844
|
7-methoxy-1-methyl-9H-beta-carboline;hydrochloride
Show/Hide
|
C13H12N2O
|
1
|
| 1 |
IC50 = 5080 nM
|
|
|
|
CP0565811
|
4-[4-(3-bromophenyl)piperazin-1-yl]-2-phenylquinazoline
Show/Hide
|
C24H21BrN4
|
1
|
| 1 |
IC50 = 5120 nM
|
|
|
|
CP0569191
|
N-[3-[(2-phenylpyrido[2,3-d]pyrimidin-4-yl)amino]phenyl]acetamide
Show/Hide
|
C21H17N5O
|
1
|
| 1 |
IC50 = 5270 nM
|
|
|
|
CP0538860
|
[N-[4-(3-methoxyanilino)-2-pyridin-3-ylquinazolin-6-yl]-C-methylcarbonimidoyl] acetate
Show/Hide
|
C24H21N5O3
|
1
|
| 1 |
IC50 = 5310 nM
|
|
|
|
CP0428640
|
(E)-3-(2-chlorophenyl)-1-(2-hydroxynaphthalen-1-yl)prop-2-en-1-one
Show/Hide
|
C19H13ClO2
|
1
|
| 1 |
IC50 = 5580 nM
|
|
|
|
CP0544529
|
tert-butyl 4-[(2-phenylquinazolin-4-yl)amino]benzoate
Show/Hide
|
C25H23N3O2
|
1
|
| 1 |
IC50 = 5650 nM
|
|
|
|
CP0395785
|
(E)-1-(1-hydroxynaphthalen-2-yl)-3-(3-methoxyphenyl)prop-2-en-1-one
Show/Hide
|
C20H16O3
|
1
|
| 1 |
IC50 = 5680 nM
|
|
|
|
CP0523462
|
4-[4-(3-chlorophenyl)piperazin-1-yl]-2-phenylquinazoline
Show/Hide
|
C24H21ClN4
|
1
|
| 1 |
IC50 = 5910 nM
|
|
|
|
CP0420699
|
4-(4-phenylpiperazin-1-yl)-6,7,8,9-tetrahydropyrimido[4,5-b]indolizine-10-carbonitrile
Show/Hide
|
C21H22N6
|
1
|
| 1 |
IC50 = 5910 nM
|
|
|
|
CP0525908
|
N-(2-nitrophenyl)-2-phenylquinazolin-4-amine
Show/Hide
|
C20H14N4O2
|
1
|
| 1 |
IC50 = 5930 nM
|
|
|
|
CP0055377
|
2-(2,4-Dimethoxy-phenyl)-3,5,7-trimethoxy-chromen-4-one
Show/Hide
|
C20H20O7
|
2
|
| 1 |
IC50 = 5940 nM
|
|
|
| 2 |
IC50 = 5980 nM
|
|
|
|
CP0129110
|
3-Phenyl-1H-naphtho[2,1-b]pyran-1-one
Show/Hide
|
C19H12O2
|
2
|
| 1 |
IC50 = 6050 nM
|
|
|
| 2 |
IC50 = 8320 nM
|
|
|
|
CP0509817
|
4-(3-phenylpropylamino)-6,7,8,9-tetrahydropyrimido[4,5-b]indolizine-10-carbonitrile
Show/Hide
|
C20H21N5
|
1
|
| 1 |
IC50 = 6070 nM
|
|
|
|
CP0444049
|
2-hydroxy-3-(4-methoxyphenyl)benzo[f]chromen-1-one
Show/Hide
|
C20H14O4
|
2
|
| 1 |
IC50 = 6120 nM
|
|
|
| 2 |
IC50 = 8930 nM
|
|
|
|
CP0067438
|
substituted chalcone, 5m
Show/Hide
|
C15H11ClO3
|
1
|
| 1 |
IC50 = 6370 nM
|
|
|
|
CP0532850
|
4-[(2-phenylquinazolin-4-yl)amino]benzoic acid
Show/Hide
|
C21H15N3O2
|
1
|
| 1 |
IC50 = 6380 nM
|
|
|
|
CP0575546
|
N-[3-[[2-(3-methoxyphenyl)pyrido[2,3-d]pyrimidin-4-yl]amino]phenyl]acetamide
Show/Hide
|
C22H19N5O2
|
1
|
| 1 |
IC50 = 6400 nM
|
|
|
|
CP0406744
|
3-methoxy-2-(4-methoxyphenyl)chromen-4-one
Show/Hide
|
C17H14O4
|
2
|
| 1 |
IC50 = 6500 nM
|
|
|
| 2 |
IC50 = 7740 nM
|
|
|
|
CP0523465
|
N-(4-bromophenyl)-2-phenylquinazolin-4-amine
Show/Hide
|
C20H14BrN3
|
1
|
| 1 |
IC50 = 6830 nM
|
|
|
|
CP0542890
|
N-[2-(2-phenyltetrazol-5-yl)phenyl]acetamide
Show/Hide
|
C15H13N5O
|
1
|
| 1 |
IC50 = 6910 nM
|
|
|
|
CP0387997
|
(E)-3-(3,4-dichlorophenyl)-1-(2-hydroxynaphthalen-1-yl)prop-2-en-1-one
Show/Hide
|
C19H12Cl2O2
|
1
|
| 1 |
IC50 = 7260 nM
|
|
|
|
CP0545307
|
4-(4-bromophenoxy)-2-phenylquinazoline
Show/Hide
|
C20H13BrN2O
|
1
|
| 1 |
IC50 = 7270 nM
|
|
|
|
CP0545309
|
4-(3-methoxyphenyl)sulfanyl-2-phenylquinazoline
Show/Hide
|
C21H16N2OS
|
1
|
| 1 |
IC50 = 7400 nM
|
|
|
|
CP0402415
|
4-methoxy-N-[2-[2-(4-methoxyphenyl)tetrazol-5-yl]phenyl]benzenesulfonamide
Show/Hide
|
C21H19N5O4S
|
1
|
| 1 |
IC50 = 7670 nM
|
|
|
|
CP0493653
|
4-anilino-6,7,8,9-tetrahydropyrimido[4,5-b]indolizine-10-carbonitrile
Show/Hide
|
C17H15N5
|
1
|
| 1 |
IC50 = 7680 nM
|
|
|
|
CP0441265
|
(E)-3-(2-chlorophenyl)-1-(3,4-dimethoxyphenyl)prop-2-en-1-one
Show/Hide
|
C17H15ClO3
|
1
|
| 1 |
IC50 = 7800 nM
|
|
|
|
CP0490342
|
N-[4-(2-benzoyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl)phenyl]acetamide
Show/Hide
|
C26H23N3O2
|
1
|
| 1 |
IC50 = 7820 nM
|
|
|
|
CP0525911
|
4-[4-(3-nitrophenyl)piperazin-1-yl]-2-phenylquinazoline
Show/Hide
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C24H21N5O2
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1
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| 1 |
IC50 = 7950 nM
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CP0263949
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N-(3-fluorophenyl)quinazolin-4-amine
Show/Hide
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C14H10FN3
|
1
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| 1 |
IC50 = 8120 nM
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CP0504953
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4-(4-Phenethyl-piperazin-1-yl)-6,7,8,9-tetrahydro-pyrimido[4,5-b]indolizine-10-carbonitrile
Show/Hide
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C23H26N6
|
1
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| 1 |
IC50 = 8190 nM
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CP0381604
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4-[4-(3-chloro-4-fluorophenyl)piperazin-1-yl]-2-phenylquinazoline
Show/Hide
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C24H20ClFN4
|
1
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| 1 |
IC50 = 8220 nM
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CP0380589
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4-(4-benzylpiperazin-1-yl)-6,7,8,9-tetrahydropyrimido[4,5-b]indolizine-10-carbonitrile
Show/Hide
|
C22H24N6
|
1
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| 1 |
IC50 = 8240 nM
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CP0383765
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2-phenyl-5-(2-phenylphenyl)tetrazole
Show/Hide
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C19H14N4
|
1
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| 1 |
IC50 = 8340 nM
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CP0451319
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6-[4-[(2-chlorophenyl)methyl]piperazin-1-yl]-11,13-dimethyl-8-thia-3,5,10-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaene
Show/Hide
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C22H22ClN5S
|
1
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| 1 |
IC50 = 8680 nM
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CP0380587
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4-(4-benzhydrylpiperazin-1-yl)-5,6-di(cycloheptyl)pyrrolo[3,2-d]pyrimidine-7-carbonitrile
Show/Hide
|
C38H46N6
|
1
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| 1 |
IC50 = 8710 nM
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CP0436733
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4-[4-(3-methoxyphenyl)piperazin-1-yl]-2-phenylquinazoline
Show/Hide
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C25H24N4O
|
1
|
| 1 |
IC50 = 8900 nM
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CP0443242
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2-phenyl-4-(4-phenylpiperazin-1-yl)quinazoline
Show/Hide
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C24H22N4
|
1
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| 1 |
IC50 = 8920 nM
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CP0144771
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3-hydroxy-5,7-dimethoxy-2-(4-methoxyphenyl)chromen-4-one
Show/Hide
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C18H16O6
|
2
|
| 1 |
IC50 = 8950 nM
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|
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| 2 |
IC50 = 12400 nM
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CP0003356
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(E)-1-(1-hydroxynaphthalen-2-yl)-3-phenylprop-2-en-1-one
Show/Hide
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C19H14O2
|
1
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| 1 |
IC50 = 9230 nM
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CP0443241
|
4-[4-(4-nitrophenyl)piperazin-1-yl]-2-phenylquinazoline
Show/Hide
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C24H21N5O2
|
1
|
| 1 |
IC50 = 9350 nM
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CP0547393
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4-[(2-pyridin-4-ylquinazolin-4-yl)amino]benzoic acid
Show/Hide
|
C20H14N4O2
|
1
|
| 1 |
IC50 = 9640 nM
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CP0418785
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(E)-1-(1-hydroxynaphthalen-2-yl)-3-(4-methoxyphenyl)prop-2-en-1-one
Show/Hide
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C20H16O3
|
1
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| 1 |
IC50 = 9830 nM
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CP0380588
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5,6-di(cycloheptyl)-4-[4-(2-phenylethyl)piperazin-1-yl]pyrrolo[3,2-d]pyrimidine-7-carbonitrile
Show/Hide
|
C33H44N6
|
1
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| 1 |
IC50 = 9940 nM
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CP0385299
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N-[2-[2-(4-methylsulfanylphenyl)tetrazol-5-yl]phenyl]-4-(trifluoromethyl)benzamide
Show/Hide
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C22H16F3N5OS
|
1
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| 1 |
IC50 > 10000 nM
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CP0450329
|
[4-[5-[2-[(4-propylbenzoyl)amino]phenyl]tetrazol-2-yl]phenyl] 4-propylbenzoate
Show/Hide
|
C33H31N5O3
|
1
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| 1 |
IC50 > 10000 nM
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CP0467039
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N-[2-[2-(4-methylsulfanylphenyl)tetrazol-5-yl]phenyl]-4-nitrobenzamide
Show/Hide
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C21H16N6O3S
|
1
|
| 1 |
IC50 > 10000 nM
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|
|
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CP0473221
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N-[2-[2-(4-chlorophenyl)tetrazol-5-yl]phenyl]-4-nitrobenzamide
Show/Hide
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C20H13ClN6O3
|
1
|
| 1 |
IC50 > 10000 nM
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CP0507005
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N-[2-[2-(4-propan-2-ylphenyl)tetrazol-5-yl]phenyl]-4-(trifluoromethyl)benzamide
Show/Hide
|
C24H20F3N5O
|
1
|
| 1 |
IC50 > 10000 nM
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|
|
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CP0510697
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N-[2-[2-(4-phenoxyphenyl)tetrazol-5-yl]phenyl]-4-propylbenzamide
Show/Hide
|
C29H25N5O2
|
1
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| 1 |
IC50 > 10000 nM
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|
|
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CP0519616
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4-methoxy-N-[2-[2-(4-phenoxyphenyl)tetrazol-5-yl]phenyl]benzamide
Show/Hide
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C27H21N5O3
|
1
|
| 1 |
IC50 > 10000 nM
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|
|
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CP0545308
|
2-phenyl-4-phenylsulfanylquinazoline
Show/Hide
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C20H14N2S
|
1
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| 1 |
IC50 = 10000 nM
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CP0455715
|
[1-(3-nitrophenyl)-1,3,4,9-tetrahydropyrido[3,4-b]indol-2-yl]-phenylmethanone
Show/Hide
|
C24H19N3O3
|
1
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| 1 |
IC50 > 10000 nM
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|
|
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CP0488223
|
phenyl-[1-[4-(trifluoromethyl)phenyl]-1,3,4,9-tetrahydropyrido[3,4-b]indol-2-yl]methanone
Show/Hide
|
C25H19F3N2O
|
1
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| 1 |
IC50 > 10000 nM
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CP0530756
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[1-(3,4-dichlorophenyl)-9-ethyl-3,4-dihydro-1H-pyrido[3,4-b]indol-2-yl]-(3-methoxyphenyl)methanone
Show/Hide
|
C27H24Cl2N2O2
|
1
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| 1 |
IC50 > 10000 nM
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CP0531725
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2-benzyl-1-(3,4-dichlorophenyl)-1,3,4,9-tetrahydropyrido[3,4-b]indole
Show/Hide
|
C24H20Cl2N2
|
1
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| 1 |
IC50 > 10000 nM
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|
|
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CP0534953
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2-benzyl-1-phenyl-1,3,4,9-tetrahydropyrido[3,4-b]indole
Show/Hide
|
C24H22N2
|
1
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| 1 |
IC50 > 10000 nM
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|
|
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CP0534955
|
[1-(2-bromophenyl)-1,3,4,9-tetrahydropyrido[3,4-b]indol-2-yl]-phenylmethanone
Show/Hide
|
C24H19BrN2O
|
1
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| 1 |
IC50 > 10000 nM
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|
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CP0550465
|
[1-(2-chlorophenyl)-1,3,4,9-tetrahydropyrido[3,4-b]indol-2-yl]-phenylmethanone
Show/Hide
|
C24H19ClN2O
|
1
|
| 1 |
IC50 > 10000 nM
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|
|
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CP0559003
|
4-[methyl-(2-phenylquinazolin-4-yl)amino]benzonitrile
Show/Hide
|
C22H16N4
|
1
|
| 1 |
IC50 = 10080 nM
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|
|
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CP0030165
|
US8592579, 104
Show/Hide
|
C23H24FN9O
|
1
|
| 1 |
IC50 = 10200 nM
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|
|
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CP0493723
|
2,3-dihydro-1,4-benzodioxin-6-yl-[1-(4-pyrazol-1-ylbenzoyl)piperidin-4-yl]methanone
Show/Hide
|
C24H23N3O4
|
1
|
| 1 |
IC50 = 10400 nM
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CP0474210
|
(9-ethyl-1-phenyl-3,4-dihydro-1H-pyrido[3,4-b]indol-2-yl)-phenylmethanone
Show/Hide
|
C26H24N2O
|
1
|
| 1 |
IC50 = 10400 nM
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|
|
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CP0393133
|
2-(3-nitrophenyl)-N-[3-(trifluoromethyl)phenyl]quinazolin-4-amine
Show/Hide
|
C21H13F3N4O2
|
1
|
| 1 |
IC50 = 10700 nM
|
|
|
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CP0050726
|
4-Anilino quinazoline deriv. 10
Show/Hide
|
C14H11N3
|
1
|
| 1 |
IC50 = 10700 nM
|
|
|
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CP0095207
|
substituted chalcone, 5i
Show/Hide
|
C16H13ClO3
|
1
|
| 1 |
IC50 = 10720 nM
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|
|
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CP0434122
|
2-hydroxy-3-phenylbenzo[f]chromen-1-one
Show/Hide
|
C19H12O3
|
2
|
| 1 |
IC50 = 11000 nM
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|
|
| 2 |
IC50 = 13600 nM
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|
|
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CP0397338
|
2-methoxy-3-phenylbenzo[f]chromen-1-one
Show/Hide
|
C20H14O3
|
2
|
| 1 |
IC50 = 11100 nM
|
|
|
| 2 |
IC50 = 12500 nM
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|
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CP0416672
|
N-[2-[2-(3-methoxyphenyl)tetrazol-5-yl]phenyl]-4-(trifluoromethyl)benzamide
Show/Hide
|
C22H16F3N5O2
|
1
|
| 1 |
IC50 = 11200 nM
|
|
|
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CP0521246
|
2-(1,3-benzodioxol-5-yl)-4-[[4-(2-fluorophenyl)piperazin-1-yl]methyl]-1,3-thiazole
Show/Hide
|
C21H20FN3O2S
|
1
|
| 1 |
IC50 = 11200 nM
|
|
|
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CP0391018
|
11,13-dimethyl-6-[4-(2-naphthalen-1-yloxyethyl)piperazin-1-yl]-4-propyl-3,7,8,10-tetrazatricyclo[7.4.0.02,7]trideca-1,3,5,8,10,12-hexaene
Show/Hide
|
C30H34N6O
|
1
|
| 1 |
IC50 = 11800 nM
|
|
|
|
CP0047641
|
1-(2,4-Dihydroxy-phenyl)-3-(4-methoxy-phenyl)-propenone
Show/Hide
|
C16H14O4
|
1
|
| 1 |
IC50 = 12050 nM
|
|
|
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CP0455914
|
4-(4-benzhydrylpiperazin-1-yl)-6,7,8,9-tetrahydropyrimido[4,5-b]indolizine-10-carbonitrile
Show/Hide
|
C28H28N6
|
1
|
| 1 |
IC50 = 14300 nM
|
|
|
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CP0467720
|
1-[4-(2,3-dihydro-1-benzofuran-5-ylmethyl)piperazin-1-yl]-2-[[5-(4-fluorophenyl)-1,3,4-oxadiazol-2-yl]sulfanyl]ethanone
Show/Hide
|
C23H23FN4O3S
|
1
|
| 1 |
IC50 = 14400 nM
|
|
|
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CP0574767
|
4-phenoxy-2-phenylquinazoline
Show/Hide
|
C20H14N2O
|
1
|
| 1 |
IC50 = 14500 nM
|
|
|
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CP0424482
|
2-phenyl-4-[3-(trifluoromethyl)phenyl]sulfanylquinazoline
Show/Hide
|
C21H13F3N2S
|
1
|
| 1 |
IC50 = 14800 nM
|
|
|
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CP0459137
|
4-[[4-(1-benzyl-3-pyridin-3-ylpyrazole-4-carbonyl)piperazin-1-yl]methyl]benzonitrile
Show/Hide
|
C28H26N6O
|
1
|
| 1 |
IC50 = 15400 nM
|
|
|
|
CP0420065
|
4-(benzylamino)-6,7,8,9-tetrahydropyrimido[4,5-b]indolizine-10-carbonitrile
Show/Hide
|
C18H17N5
|
1
|
| 1 |
IC50 = 15800 nM
|
|
|
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CP0529201
|
2-(4-methoxyphenyl)-5-[2-[5-[4-(trifluoromethyl)phenyl]tetrazol-2-yl]phenyl]tetrazole
Show/Hide
|
C22H15F3N8O
|
1
|
| 1 |
IC50 = 15800 nM
|
|
|
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CP0529577
|
(2-pyridin-3-ylquinolin-4-yl)-[4-(thiophen-2-ylmethyl)piperazin-1-yl]methanone
Show/Hide
|
C24H22N4OS
|
1
|
| 1 |
IC50 = 16000 nM
|
|
|
|
CP0393134
|
N-[4-methoxy-3-(trifluoromethyl)phenyl]-2-(3-nitrophenyl)quinazolin-4-amine
Show/Hide
|
C22H15F3N4O3
|
1
|
| 1 |
IC50 = 16200 nM
|
|
|
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CP0511750
|
3-[(2-pyridin-3-ylpyrido[2,3-d]pyrimidin-4-yl)amino]phenol
Show/Hide
|
C18H13N5O
|
1
|
| 1 |
IC50 = 16900 nM
|
|
|
|
CP0434800
|
2-(4-fluoro-3-methoxyphenyl)-3-hydroxybenzo[h]chromen-4-one
Show/Hide
|
C20H13FO4
|
2
|
| 1 |
IC50 = 17900 nM
|
|
|
| 2 |
IC50 = 22500 nM
|
|
|
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CP0542904
|
N-[3-[2-(4-methoxyphenyl)tetrazol-5-yl]phenyl]-4-(trifluoromethyl)benzamide
Show/Hide
|
C22H16F3N5O2
|
1
|
| 1 |
IC50 = 18500 nM
|
|
|
|
CP0541419
|
N-(4-nitrophenyl)-2-phenylpyrido[2,3-d]pyrimidin-4-amine
Show/Hide
|
C19H13N5O2
|
1
|
| 1 |
IC50 = 19500 nM
|
|
|
|
CP0441259
|
(E)-3-(3,4-dichlorophenyl)-1-(1-hydroxynaphthalen-2-yl)prop-2-en-1-one
Show/Hide
|
C19H12Cl2O2
|
1
|
| 1 |
IC50 = 22390 nM
|
|
|
|
CP0549041
|
N-[3-(quinazolin-4-ylamino)phenyl]acetamide
Show/Hide
|
C16H14N4O
|
1
|
| 1 |
IC50 = 28900 nM
|
|
|
|
CP0031166
|
(E)-1-(2-Hydroxy-4-methoxy-phenyl)-3-phenyl-propenone
Show/Hide
|
C16H14O3
|
1
|
| 1 |
IC50 = 30950 nM
|
|
|
|
CP0557993
|
N-[4-[2-(4-methoxyphenyl)tetrazol-5-yl]phenyl]-4-(trifluoromethyl)benzamide
Show/Hide
|
C22H16F3N5O2
|
1
|
| 1 |
IC50 = 39800 nM
|
|
|
|
CP0472385
|
3-[(2-pyridin-4-ylquinazolin-4-yl)amino]benzoic acid
Show/Hide
|
C20H14N4O2
|
1
|
| 1 |
IC50 = 60000 nM
|
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|
