General Information of the Compound
Compound ID
CP0380381
Compound Name
(E)-3-(3,4-dimethoxyphenyl)-1-[4-[[2-(3,4-dimethoxyphenyl)quinazolin-4-yl]amino]phenyl]prop-2-en-1-one
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Structure
Formula
C33H29N3O5
Molecular Weight
547.611
Canonical SMILES
COc1ccc(\C=C\C(=O)c2ccc(Nc3nc(nc4ccccc34)-c3ccc(OC)c(OC)c3)cc2)cc1OC
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InChI
InChI=1S/C33H29N3O5/c1-38-28-17-10-21(19-30(28)40-3)9-16-27(37)22-11-14-24(15-12-22)34-33-25-7-5-6-8-26(25)35-32(36-33)23-13-18-29(39-2)31(20-23)41-4/h5-20H,1-4H3,(H,34,35,36)/b16-9+
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InChIKey
UELXDXUOBOULEV-CXUHLZMHSA-N
Physicochemical Property
logP
6.9709
Rotatable Bonds
10
Heavy Atom Count
41
Polar Areas
91.8
Hydrogen Bond Donor Count
1
Hydrogen Bond Acceptor Count
8
Complexity
41

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 127045064
ChEMBL ID
CHEMBL3809529
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT01546, ATP-dependent translocase ABCB1
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000135 A2780ADR Homo sapiens (Human)  1
1
IC50 = 14900 nM
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   LI
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Protein ID: PT02718, Broad substrate specificity ATP-binding cassette transporter ABCG2
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000036 MDCK-II Canis lupus familiaris (Dog)  1
1
IC50 = 190 nM
   TI
   LI
   LO
   TS