| Compound ID |
Compound Name |
Compound Formula |
|
CP0777252
|
2-Iodo-N-(3-(R)-1-pyrrolidin-2-ylmethyl-1H-indol-5-yl)-benzenesulfonamide
Show/Hide
|
C20H22IN3O2S
|
2
|
| 1 |
EC50 = 0.4 nM
|
|
|
| 2 |
Ki = 1 nM
|
|
|
|
CP0916804
|
3,5-Dimethyl-isoxazole-4-sulfonic acid [3-((R)-1-methyl-pyrrolidin-2-ylmethyl)-1H-indol-5-yl]-amide
Show/Hide
|
C19H24N4O3S
|
2
|
| 1 |
EC50 = 0.8 nM
|
|
|
| 2 |
Ki = 1 nM
|
|
|
|
CP0869624
|
3-Chloro-N-(3-(R)-1-pyrrolidin-2-ylmethyl-1H-indol-5-yl)-benzenesulfonamide
Show/Hide
|
C19H20ClN3O2S
|
2
|
| 1 |
EC50 = 1 nM
|
|
|
| 2 |
Ki = 2 nM
|
|
|
|
CP0873359
|
2-Chloro-N-[3-((R)-1-methyl-pyrrolidin-2-ylmethyl)-1H-indol-5-yl]-benzenesulfonamide
Show/Hide
|
C20H22ClN3O2S
|
2
|
| 1 |
EC50 = 1.1 nM
|
|
|
| 2 |
Ki = 1 nM
|
|
|
|
CP0877520
|
4-Fluoro-N-[3-((R)-1-methyl-pyrrolidin-2-ylmethyl)-1H-indol-5-yl]-benzenesulfonamide
Show/Hide
|
C20H22FN3O2S
|
2
|
| 1 |
EC50 = 1.1 nM
|
|
|
| 2 |
Ki = 1 nM
|
|
|
|
CP0853639
|
2-Chloro-N-(3-(R)-1-pyrrolidin-2-ylmethyl-1H-indol-5-yl)-benzenesulfonamide
Show/Hide
|
C19H20ClN3O2S
|
2
|
| 1 |
EC50 = 1.3 nM
|
|
|
| 2 |
Ki = 3 nM
|
|
|
|
CP0874912
|
2-Fluoro-N-[3-((R)-1-methyl-pyrrolidin-2-ylmethyl)-1H-indol-5-yl]-benzenesulfonamide
Show/Hide
|
C20H22FN3O2S
|
2
|
| 1 |
EC50 = 1.3 nM
|
|
|
| 2 |
Ki = 1 nM
|
|
|
|
CP0919321
|
4-Methyl-N-[3-((R)-1-methyl-pyrrolidin-2-ylmethyl)-1H-indol-5-yl]-benzenesulfonamide
Show/Hide
|
C21H25N3O2S
|
2
|
| 1 |
EC50 = 1.3 nM
|
|
|
| 2 |
Ki = 1 nM
|
|
|
|
CP0869661
|
N-(3-(R)-1-Pyrrolidin-2-ylmethyl-1H-indol-5-yl)-benzenesulfonamide
Show/Hide
|
C19H21N3O2S
|
2
|
| 1 |
EC50 = 1.4 nM
|
|
|
| 2 |
Ki = 4 nM
|
|
|
|
CP0860616
|
3-Chloro-N-[3-((R)-1-methyl-pyrrolidin-2-ylmethyl)-1H-indol-5-yl]-benzenesulfonamide
Show/Hide
|
C20H22ClN3O2S
|
2
|
| 1 |
EC50 = 1.6 nM
|
|
|
| 2 |
Ki = 0.4 nM
|
|
|
|
CP0919322
|
4-Methoxy-N-[3-((R)-1-methyl-pyrrolidin-2-ylmethyl)-1H-indol-5-yl]-benzenesulfonamide
Show/Hide
|
C21H25N3O3S
|
2
|
| 1 |
EC50 = 2.2 nM
|
|
|
| 2 |
Ki = 1 nM
|
|
|
|
CP0862924
|
4-Iodo-N-[3-((R)-1-methyl-pyrrolidin-2-ylmethyl)-1H-indol-5-yl]-benzenesulfonamide
Show/Hide
|
C20H22IN3O2S
|
2
|
| 1 |
EC50 = 2.7 nM
|
|
|
| 2 |
Ki = 0.3 nM
|
|
|
|
CP0916803
|
N-[3-((R)-1-Methyl-pyrrolidin-2-ylmethyl)-1H-indol-5-yl]-4-trifluoromethoxy-benzenesulfonamide
Show/Hide
|
C21H22F3N3O3S
|
2
|
| 1 |
EC50 = 2.9 nM
|
|
|
| 2 |
Ki = 1 nM
|
|
|
|
CP0853638
|
N-[3-((R)-1-Methyl-pyrrolidin-2-ylmethyl)-1H-indol-5-yl]-3-trifluoromethyl-benzenesulfonamide
Show/Hide
|
C21H22F3N3O2S
|
2
|
| 1 |
EC50 = 3.2 nM
|
|
|
| 2 |
Ki = 1 nM
|
|
|
|
CP0847609
|
N-(3-(R)-1-Pyrrolidin-2-ylmethyl-1H-indol-5-yl)-4-trifluoromethoxy-benzenesulfonamide
Show/Hide
|
C20H20F3N3O3S
|
2
|
| 1 |
EC50 = 4.2 nM
|
|
|
| 2 |
Ki = 5 nM
|
|
|
|
CP0485541
|
pyrrolidinylindole, (R)-5b
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|
C21H22F3N3O2S
|
2
|
| 1 |
EC50 = 4.5 nM
|
|
|
| 2 |
Ki = 0.4 nM
|
|
|
|
CP0874915
|
4-Chloro-N-(3-(R)-1-pyrrolidin-2-ylmethyl-1H-indol-5-yl)-benzenesulfonamide
Show/Hide
|
C19H20ClN3O2S
|
2
|
| 1 |
EC50 = 4.5 nM
|
|
|
| 2 |
Ki = 3 nM
|
|
|
|
CP0871294
|
2,4-Difluoro-N-(3-(R)-1-pyrrolidin-2-ylmethyl-1H-indol-5-yl)-benzenesulfonamide
Show/Hide
|
C19H19F2N3O2S
|
2
|
| 1 |
EC50 = 5.2 nM
|
|
|
| 2 |
Ki = 8 nM
|
|
|
|
CP0853755
|
N-(3-(R)-1-Pyrrolidin-2-ylmethyl-1H-indol-5-yl)-3-trifluoromethyl-benzenesulfonamide
Show/Hide
|
C20H20F3N3O2S
|
2
|
| 1 |
EC50 = 5.8 nM
|
|
|
| 2 |
Ki = 4 nM
|
|
|
|
CP0144949
|
2-[1-({6-chloroimidazo[2,1-b][1,3]thiazole-5-}sulfonyl)-1H-indol-3-yl]ethan-1-amine
Show/Hide
|
C15H13ClN4O2S2
|
2
|
| 1 |
EC50 = 6.5 nM
|
|
|
| 2 |
Ki = 2 nM
|
|
|
|
CP0380100
|
2-(3-(3-fluorophenylsulfonyl)-1H-pyrrolo[2,3-b]pyridin-1-yl)-N,N-dimethylethanamine
Show/Hide
|
C17H18FN3O2S
|
3
|
| 1 |
EC50 = 7.3 nM
|
|
|
| 2 |
Ki = 4.8 nM
|
|
|
| 3 |
Ki = 4.9 nM
|
|
|
|
CP0405688
|
2-[3-(3-chlorophenyl)sulfonylpyrrolo[2,3-b]pyridin-1-yl]-N,N-dimethylethanamine
Show/Hide
|
C17H18ClN3O2S
|
2
|
| 1 |
EC50 = 15 nM
|
|
|
| 2 |
Ki = 2.3 nM
|
|
|
|
CP0439248
|
2-{3-[(3-Chlorophenyl)sulfonyl]-1H-pyrrolo[2,3-b]pyridin-1-yl}ethylamine
Show/Hide
|
C15H14ClN3O2S
|
2
|
| 1 |
EC50 = 18 nM
|
|
|
| 2 |
Ki = 2 nM
|
|
|
|
CP0431045
|
2-[2-Methyl-3-(phenylsulfonyl)-1H-pyrrolo[2,3-b]pyridin-1-yl]ethylamine
Show/Hide
|
C16H17N3O2S
|
2
|
| 1 |
EC50 = 20 nM
|
|
|
| 2 |
Ki = 4.2 nM
|
|
|
|
CP0439191
|
2-{3-[(3-Fluorophenyl)sulfonyl]-1H-pyrrolo[2,3-b]pyridin-1-yl}ethylamine
Show/Hide
|
C15H14FN3O2S
|
2
|
| 1 |
EC50 = 24 nM
|
|
|
| 2 |
Ki = 4.7 nM
|
|
|
|
CP0914961
|
3-[(6-chloroimidazo[2,1-b][1,3]thiazol-5-yl)sulfonyl]-1-(1-methylpiperidin-3-yl)-1H-pyrrolo[2,3-b]pyridine
Show/Hide
|
C18H20ClN5O2S2
|
2
|
| 1 |
EC50 = 25 nM
|
|
|
| 2 |
Ki = 2 nM
|
|
|
|
CP0431044
|
2-[3-(benzenesulfonyl)pyrrolo[2,3-b]pyridin-1-yl]-N,N-dimethylethanamine
Show/Hide
|
C17H19N3O2S
|
2
|
| 1 |
EC50 = 25 nM
|
|
|
| 2 |
Ki = 23 nM
|
|
|
|
CP0424416
|
2-[3-(Phenylsulfonyl)-1H-pyrrolo[2,3-b]pyridin-1-yl]ethylamine
Show/Hide
|
C15H15N3O2S
|
2
|
| 1 |
EC50 = 27 nM
|
|
|
| 2 |
Ki = 5.5 nM
|
|
|
|
CP0430945
|
2-[3-(3,5-dichlorophenyl)sulfonylpyrrolo[2,3-b]pyridin-1-yl]-N,N-dimethylethanamine
Show/Hide
|
C17H17Cl2N3O2S
|
2
|
| 1 |
EC50 = 28 nM
|
|
|
| 2 |
Ki = 4.3 nM
|
|
|
|
CP0309906
|
3-[(3-chlorophenyl)sulfonyl]-1-piperidin-3-yl-1Hpyrrolo[2,3-b]pyridine
Show/Hide
|
C18H18ClN3O2S
|
2
|
| 1 |
EC50 = 30 nM
|
|
|
| 2 |
Ki = 1.3 nM
|
|
|
|
CP0431016
|
2-[3-(4-fluorophenyl)sulfonylpyrrolo[2,3-b]pyridin-1-yl]-N,N-dimethylethanamine
Show/Hide
|
C17H18FN3O2S
|
2
|
| 1 |
EC50 = 30 nM
|
|
|
| 2 |
Ki = 45 nM
|
|
|
|
CP0502801
|
1-(1-ethylpiperidin-3-yl)-3-(phenylsulfonyl)-1H-indole
Show/Hide
|
C21H24N2O2S
|
2
|
| 1 |
EC50 = 31 nM
|
|
|
| 2 |
Ki = 7.3 nM
|
|
|
|
CP0398876
|
2-[3-(2,6-dichlorophenyl)sulfonylpyrrolo[2,3-b]pyridin-1-yl]-N,N-dimethylethanamine
Show/Hide
|
C17H17Cl2N3O2S
|
2
|
| 1 |
EC50 = 31 nM
|
|
|
| 2 |
Ki = 9 nM
|
|
|
|
CP0398929
|
2-[3-(5-chlorothiophen-2-yl)sulfonylpyrrolo[2,3-b]pyridin-1-yl]-N,N-dimethylethanamine
Show/Hide
|
C15H16ClN3O2S2
|
2
|
| 1 |
EC50 = 32 nM
|
|
|
| 2 |
Ki = 3.3 nM
|
|
|
|
CP0900149
|
3-[(6-chloroimidazo[2,1-b][1,3]thiazol-5-yl)sulfonyl]-1-(1-ethylpiperidin-3-yl)-1H-pyrrolo[2,3-b]pyridine
Show/Hide
|
C19H22ClN5O2S2
|
2
|
| 1 |
EC50 = 34 nM
|
|
|
| 2 |
Ki = 0.7 nM
|
|
|
|
CP0302411
|
3-(3-bromo-benzenesulfonyl)-1-pyrrolidin-3-yl-1Hpyrrolo[2,3-b]pyridine
Show/Hide
|
C17H16BrN3O2S
|
2
|
| 1 |
EC50 = 35 nM
|
|
|
| 2 |
Ki = 1.3 nM
|
|
|
|
CP0431003
|
2-{3-[(3,5-Dichlorophenyl)sulfonyl]-1H-pyrrolo[2,3-b]pyridin-1-yl}ethylamine
Show/Hide
|
C15H13Cl2N3O2S
|
2
|
| 1 |
EC50 = 35 nM
|
|
|
| 2 |
Ki = 2.9 nM
|
|
|
|
CP0497289
|
5-fluoro-3-(3-fluorophenylsulfonyl)-1-(pyrrolidin-3-yl)-1H-indole
Show/Hide
|
C18H16F2N2O2S
|
2
|
| 1 |
EC50 = 38 nM
|
|
|
| 2 |
Ki = 9.6 nM
|
|
|
|
CP0287714
|
3-[(3,5-dichlorophenyl)sulfonyl]-1-(1-methylpiperidin-3-yl)-1H-pyrrolo[2,3-b]pyridine
Show/Hide
|
C19H19Cl2N3O2S
|
2
|
| 1 |
EC50 = 38.7 nM
|
|
|
| 2 |
Ki = 3.9 nM
|
|
|
|
CP0271606
|
3-(phenylsulfonyl)sulfonyl]-1-piperidin-3-yl-1Hpyrrolo[2,3-b]pyridine
Show/Hide
|
C18H19N3O2S
|
2
|
| 1 |
EC50 = 47 nM
|
|
|
| 2 |
Ki = 4.9 nM
|
|
|
|
CP0469533
|
2-[3-(benzenesulfonyl)-2-methylpyrrolo[2,3-b]pyridin-1-yl]-N,N-dimethylethanamine
Show/Hide
|
C18H21N3O2S
|
2
|
| 1 |
EC50 = 47 nM
|
|
|
| 2 |
Ki = 4.7 nM
|
|
|
|
CP0093677
|
3-{[3-(trifluoromethyl)phenyl]sulfonyl}-1-(1-methylpiperidin-3-yl)-1H-pyrrolo[2,3-b]pyridine
Show/Hide
|
C20H20F3N3O2S
|
2
|
| 1 |
EC50 = 49 nM
|
|
|
| 2 |
Ki = 2.1 nM
|
|
|
|
CP0291339
|
3-[(2-chlorophenyl)sulfonyl]-1-piperidin-3-yl-1Hpyrrolo[2,3-b]pyridine
Show/Hide
|
C18H18ClN3O2S
|
2
|
| 1 |
EC50 = 50 nM
|
|
|
| 2 |
Ki = 3.7 nM
|
|
|
|
CP0326103
|
1-(1-ethylpiperidin-3-yl)-3-[(5-chlorothien-2-yl)-sulfonyl]-1H-pyrrolo[2,3-b]pyridine
Show/Hide
|
C18H20ClN3O2S2
|
2
|
| 1 |
EC50 = 50 nM
|
|
|
| 2 |
Ki = 3.2 nM
|
|
|
|
CP0453183
|
1-(2-Fluoro-benzenesulfonyl)-3-(1,2,5,6-tetrahydro-pyridin-3-yl)-1H-indole
Show/Hide
|
C19H17FN2O2S
|
2
|
| 1 |
EC50 = 51 nM
|
|
|
| 2 |
Ki = 9.2 nM
|
|
|
|
CP0419036
|
N,N-dimethyl-2-(3-naphthalen-1-ylsulfonylpyrrolo[2,3-b]pyridin-1-yl)ethanamine
Show/Hide
|
C21H21N3O2S
|
2
|
| 1 |
EC50 = 51 nM
|
|
|
| 2 |
Ki = 1 nM
|
|
|
|
CP0421794
|
2-{1-[(5-bromothiophene-2-)sulfonyl]-1H-indol-3-yl}ethan-1-amine
Show/Hide
|
C14H13BrN2O2S2
|
2
|
| 1 |
EC50 = 54 nM
|
|
|
| 2 |
Ki = 7 nM
|
|
|
|
CP0411169
|
3-(3-fluorophenylsulfonyl)-1-(piperidin-3-yl)-1H-indole
Show/Hide
|
C19H19FN2O2S
|
2
|
| 1 |
EC50 = 56 nM
|
|
|
| 2 |
Ki = 6 nM
|
|
|
|
CP0483699
|
1-(5-Chloro-thiophene-2-sulfonyl)-3-piperidin-3-yl-1H-indole
Show/Hide
|
C17H17ClN2O2S2
|
2
|
| 1 |
EC50 = 58.5 nM
|
|
|
| 2 |
Ki = 3 nM
|
|
|
|
CP0061587
|
1-(1-ethylpiperidin-3-yl)-3-[(3-fluorophenyl)sulfonyl]-1H-pyrrolo[2,3-b]pyridine
Show/Hide
|
C20H22FN3O2S
|
2
|
| 1 |
EC50 = 60 nM
|
|
|
| 2 |
Ki = 4.4 nM
|
|
|
|
CP0504632
|
3-(phenylsulfonyl)-1-(pyrrolidin-3-yl)-1H-indole
Show/Hide
|
C18H18N2O2S
|
2
|
| 1 |
EC50 = 60 nM
|
|
|
| 2 |
Ki = 5 nM
|
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|
|
CP0460408
|
2-[3-(1-Naphthylsulfonyl)-1H-pyrrolo[2,3-b]pyridin-1-yl]ethylamine
Show/Hide
|
C19H17N3O2S
|
2
|
| 1 |
EC50 = 63 nM
|
|
|
| 2 |
Ki = 1.6 nM
|
|
|
|
CP0453185
|
1-(3,4-Difluoro-benzenesulfonyl)-3-piperidin-3-yl-1H-indole
Show/Hide
|
C19H18F2N2O2S
|
2
|
| 1 |
EC50 = 66 nM
|
|
|
| 2 |
Ki = 7 nM
|
|
|
|
CP0910870
|
3-[(6-chloroimidazo[2,1-b][1,3]thiazol-5-yl)sulfonyl]-1-piperidin-3-yl-1H-pyrrolo[2,3-b]pyridine
Show/Hide
|
C17H18ClN5O2S2
|
2
|
| 1 |
EC50 = 66 nM
|
|
|
| 2 |
Ki = 0.7 nM
|
|
|
|
CP0271608
|
3-[(3-fluorophenyl)sulfonyl]-1-piperidin-3-yl-1Hpyrrolo[2,3-b]pyridine
Show/Hide
|
C18H18FN3O2S
|
2
|
| 1 |
EC50 = 67 nM
|
|
|
| 2 |
Ki = 2.4 nM
|
|
|
|
CP0295963
|
1-(1-ethylpiperidin-3-yl)-3-[(3,5-dichlorophenyl)-sulfonyl]-1H-pyrrolo[2,3-b]pyridine
Show/Hide
|
C20H21Cl2N3O2S
|
2
|
| 1 |
EC50 = 67 nM
|
|
|
| 2 |
Ki = 13.5 nM
|
|
|
|
CP0463337
|
3-(3-fluorophenylsulfonyl)-1-(pyrrolidin-3-yl)-1H-indole
Show/Hide
|
C18H17FN2O2S
|
2
|
| 1 |
EC50 = 68 nM
|
|
|
| 2 |
Ki = 4.7 nM
|
|
|
|
CP0287755
|
3-[(5-chlorothien-2-yl)sulfonyl]-1-(1-methylpiperidin-3-yl)-1H-pyrrolo[2,3-b]pyridine
Show/Hide
|
C17H18ClN3O2S2
|
2
|
| 1 |
EC50 = 71 nM
|
|
|
| 2 |
Ki = 1.9 nM
|
|
|
|
CP0295962
|
3-[(3-bromophenyl)sulfonyl]-1-piperidin-3-yl-1Hpyrrolo[2,3-b]pyridine
Show/Hide
|
C18H18BrN3O2S
|
2
|
| 1 |
EC50 = 72 nM
|
|
|
| 2 |
Ki = 3.8 nM
|
|
|
|
CP0449786
|
2-[1-(benzenesulfonyl)-1H-indol-3-yl]ethan-1-amine
Show/Hide
|
C16H16N2O2S
|
3
|
| 1 |
EC50 = 73 nM
|
|
|
| 2 |
Ki = 10 nM
|
|
|
| 3 |
Ki = 10.3 nM
|
|
|
|
CP0402008
|
3-(3-fluorophenylsulfonyl)-5-methoxy-1-(piperidin-3-yl)-1H-indole
Show/Hide
|
C20H21FN2O3S
|
2
|
| 1 |
EC50 = 73 nM
|
|
|
| 2 |
Ki = 10.7 nM
|
|
|
|
CP0899628
|
3-(6-chloro-imidazo[2,1-b]thiazole-5-sulfonyl)-1-pyrrolidin-3-yl-1H-pyrrolo[2,3-b]pyridine
Show/Hide
|
C16H16ClN5O2S2
|
2
|
| 1 |
EC50 = 80 nM
|
|
|
| 2 |
Ki = 1 nM
|
|
|
|
CP0498895
|
3-(phenylsulfonyl)-1-(piperidin-3-yl)-1H-indole
Show/Hide
|
C19H20N2O2S
|
2
|
| 1 |
EC50 = 82 nM
|
|
|
| 2 |
Ki = 13 nM
|
|
|
|
CP0430944
|
2-(3-{[2-(Trifluoromethyl)phenyl]sulfonyl}-1Hpyrrolo[2,3-b]pyridin-1-yl)ethylamine
Show/Hide
|
C16H14F3N3O2S
|
2
|
| 1 |
EC50 = 85 nM
|
|
|
| 2 |
Ki = 2.1 nM
|
|
|
|
CP0446381
|
1-(5-Chloro-3-methyl-pyrazol-1-ylmethanesulfonyl)-3-(1,2,5,6-tetrahydro-pyridin-3-yl)-1H-indole
Show/Hide
|
C18H19ClN4O2S
|
2
|
| 1 |
EC50 = 89.5 nM
|
|
|
| 2 |
Ki = 8 nM
|
|
|
|
CP0421893
|
4-{[3-(2-aminoethyl)-1H-indole-1-]sulfonyl}aniline
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C16H17N3O2S
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2
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| 1 |
EC50 = 91 nM
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| 2 |
Ki = 1 nM
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CP0113794
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3-[(5-chlorothien-2-yl)sulfonyl]-1-piperidin-3-yl-1H-pyrrolo[2,3-b]pyridine
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C16H16ClN3O2S2
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2
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| 1 |
EC50 = 98 nM
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| 2 |
Ki = 1.2 nM
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CP0448063
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1-(5-Bromo-thiophene-2-sulfonyl)-3-((R)-1-methyl-pyrrolidin-2-ylmethyl)-1H-indole
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C18H19BrN2O2S2
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2
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| 1 |
EC50 = 102.8 nM
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| 2 |
Ki = 4 nM
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CP0443001
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2-{1-[(3-chlorobenzene)sulfonyl]-1H-indol-3-yl}ethan-1-amine
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C16H15ClN2O2S
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2
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| 1 |
EC50 = 108.5 nM
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| 2 |
Ki = 6 nM
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CP0430931
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2-(3-{[3-(Trifluoromethyl)phenyl]sulfonyl}-1Hpyrrolo[2,3-b]pyridin-1-yl)ethylamine
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C16H14F3N3O2S
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2
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| 1 |
EC50 = 110 nM
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| 2 |
Ki = 2.1 nM
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CP0443273
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2-[3-(6-chloroimidazo[2,1-b][1,3]thiazol-5-yl)sulfonylpyrrolo[2,3-b]pyridin-1-yl]-N,N-dimethylethanamine
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C16H16ClN5O2S2
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2
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| 1 |
EC50 = 120 nM
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| 2 |
Ki = 0.9 nM
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CP0411090
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3-(3-chlorophenylsulfonyl)-1-(pyrrolidin-3-yl)-1H-indole
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C18H17ClN2O2S
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2
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| 1 |
EC50 = 125 nM
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| 2 |
Ki = 3.2 nM
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CP0443003
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2-{1-[(2-bromobenzene)sulfonyl]-1H-indol-3-yl}ethan-1-amine
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C16H15BrN2O2S
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2
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| 1 |
EC50 = 148 nM
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| 2 |
Ki = 11 nM
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CP0430947
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N,N-dimethyl-2-(3-thiophen-2-ylsulfonylpyrrolo[2,3-b]pyridin-1-yl)ethanamine
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C15H17N3O2S2
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2
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| 1 |
EC50 = 154 nM
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| 2 |
Ki = 15 nM
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CP0439403
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1-Benzenesulfonyl-3-(1,2,5,6-tetrahydro-pyridin-3-yl)-1H-indole
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C19H18N2O2S
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2
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| 1 |
EC50 = 159 nM
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| 2 |
Ki = 4.6 nM
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CP0473651
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2-{3-[(4-Fluorophenyl)sulfonyl]-1H-pyrrolo[2,3-b]pyridin-1-yl}ethylamine
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C15H14FN3O2S
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2
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| 1 |
EC50 = 166 nM
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| 2 |
Ki = 22 nM
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CP0143099
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3-[(3-fluorophenyl)sulfonyl]-1-(1-isopropylpiperidin-3-yl)-1H-pyrrolo[2,3-b]pyridine
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C21H24FN3O2S
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2
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| 1 |
EC50 = 172 nM
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| 2 |
Ki = 3.4 nM
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CP0464519
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2-{1-[(4-chlorobenzene)sulfonyl]-1H-indol-3-yl}ethan-1-amine
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C16H15ClN2O2S
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2
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| 1 |
EC50 = 174 nM
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| 2 |
Ki = 10 nM
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CP0430943
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2-(3-(phenylsulfonyl)-1H-indol-1-yl)ethanamine
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C16H16N2O2S
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2
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| 1 |
EC50 = 178 nM
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| 2 |
Ki = 25 nM
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CP0847576
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N-[3-((S)-1-Methyl-pyrrolidin-2-ylmethyl)-1H-indol-5-yl]-4-trifluoromethoxy-benzenesulfonamide
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C21H22F3N3O3S
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3
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| 1 |
EC50 = 180 nM
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| 2 |
IC50 = 25.8 nM
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| 3 |
Ki = 8 nM
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CP0443285
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2-{1-[(5-chlorothiophene-2-)sulfonyl]-1H-indol-3-yl}ethan-1-amine
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C14H13ClN2O2S2
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2
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| 1 |
EC50 = 181 nM
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| 2 |
Ki = 6 nM
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CP0461937
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2-{1-[(4-methylbenzene)sulfonyl]-1H-indol-3-yl}ethan-1-amine
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C17H18N2O2S
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2
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| 1 |
EC50 = 191 nM
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| 2 |
Ki = 8 nM
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CP0406482
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1-(1-ethylpiperidin-3-yl)-3-(3-fluorophenylsulfonyl)-5-methoxy-1H-indole
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C22H25FN2O3S
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2
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| 1 |
EC50 = 203 nM
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| 2 |
Ki = 16 nM
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CP0302413
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3-(3-fluoro-benzenesulfonyl)-1-(1-methyl-pyrrolidin-3-yl)-1H-pyrrolo[2,3-b]pyridine
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C18H18FN3O2S
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2
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| 1 |
EC50 = 231 nM
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| 2 |
Ki = 1.4 nM
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CP0485466
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1-(3-Fluoro-benzenesulfonyl)-3-(1,2,5,6-tetrahydro-pyridin-3-yl)-1H-indole
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C19H17FN2O2S
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2
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| 1 |
EC50 = 269.5 nM
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| 2 |
Ki = 8.5 nM
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CP0295961
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3-{[3-(trifluoromethyl)phenyl]sulfonyl}-1-piperidin-3-yl-1H-pyrrolo[2,3-b]pyridine
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C19H18F3N3O2S
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2
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| 1 |
EC50 = 273 nM
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| 2 |
Ki = 4.6 nM
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CP0316409
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3-(3-fluoro-benzenesulfonyl)-1-pyrrolidin-3-yl-1Hpyrrolo[2,3-b]pyridine
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C17H16FN3O2S
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2
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| 1 |
EC50 = 278 nM
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| 2 |
Ki = 2.7 nM
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CP0294388
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3-[(3,5-dichlorophenyl)sulfonyl]-1-piperidin-3-yl-1H-pyrrolo[2,3-b]pyridine
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C18H17Cl2N3O2S
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2
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| 1 |
EC50 = 297 nM
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| 2 |
Ki = 6.1 nM
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CP0158829
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3-[(3-fluorophenyl)sulfonyl]-1-(1-methylpiperidin-3-yl)-1H-pyrrolo[2,3-b]pyridine
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C19H20FN3O2S
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2
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| 1 |
EC50 = 306 nM
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| 2 |
Ki = 4.7 nM
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CP0446378
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1-(4-Fluoro-benzenesulfonyl)-3-(1,2,5,6-tetrahydro-pyridin-3-yl)-1H-indole
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C19H17FN2O2S
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2
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| 1 |
EC50 = 344.5 nM
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| 2 |
Ki = 10.5 nM
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CP0439247
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2-[3-(benzenesulfonyl)indol-1-yl]-N,N-dimethylethanamine
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C18H20N2O2S
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2
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| 1 |
EC50 = 366 nM
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| 2 |
Ki = 20 nM
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CP0497291
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3-(3-fluorophenylsulfonyl)-1-(1-methylpyrrolidin-3-yl)-1H-indole
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C19H19FN2O2S
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2
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| 1 |
EC50 = 398 nM
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| 2 |
Ki = 3.5 nM
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CP0297596
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3-{[4-(trifluoromethyl)phenyl]sulfonyl}-1-piperidin-3-yl-1H-pyrrolo[2,3-b]pyridine
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C19H18F3N3O2S
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2
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| 1 |
EC50 = 414 nM
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| 2 |
Ki = 12 nM
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CP0325789
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1-pyrrolidin-3-yl-3-(3-trifluoromethyl-benzenesulfonyl)-1H-pyrrolo[2,3-b]pyridine
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C18H16F3N3O2S
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2
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| 1 |
EC50 = 520 nM
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| 2 |
Ki = 1.3 nM
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CP0411088
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8-(1-(piperidin-3-yl)-1H-indol-3-ylsulfonyl)quinoline
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C22H21N3O2S
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2
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| 1 |
EC50 = 592 nM
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| 2 |
Ki = 5.6 nM
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CP0143094
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3-(4-fluoro-benzenesulfonyl)-1-pyrrolidin-3-yl-1Hpyrrolo[2,3-b]pyridine
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C17H16FN3O2S
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2
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| 1 |
EC50 = 1645 nM
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| 2 |
Ki = 8.5 nM
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CP0275252
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3-(3-chloro-benzenesulfonyl)-1-pyrrolidin-3-yl-1Hpyrrolo[2,3-b]pyridine
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C17H16ClN3O2S
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2
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| 1 |
EC50 = 1680 nM
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| 2 |
Ki = 1.5 nM
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CP0325791
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3-benzenesulfonyl-1-(1-methyl-pyrrolidin-3-yl)-1Hpyrrolo[2,3-b]pyridine
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C18H19N3O2S
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2
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| 1 |
EC50 = 2035 nM
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| 2 |
Ki = 2.5 nM
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CP0377633
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4-[5-Methoxy-3-(1,2,3,6-tetrahydro-pyridin-4-yl)-indole-1-sulfonyl]-phenylamine
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C20H21N3O3S
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2
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| 1 |
IC50 = 0.4 nM
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| 2 |
Ki = 3 nM
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CP0456508
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1-Benzenesulfonyl-3-((R)-1-methyl-pyrrolidin-2-ylmethyl)-1H-indole; oxalic acid
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C20H22N2O2S
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2
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| 1 |
IC50 = 0.6 nM
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| 2 |
Ki = 8 nM
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CP0433586
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1-(2-Chloro-benzenesulfonyl)-3-(1-methyl-1,2,3,6-tetrahydro-pyridin-4-yl)-1H-indole
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C20H19ClN2O2S
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2
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| 1 |
IC50 = 0.7 nM
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| 2 |
Ki = 10 nM
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CP0881020
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2-Bromo-N-[3-((S)-1-methyl-pyrrolidin-2-ylmethyl)-1H-indol-5-yl]-benzenesulfonamide
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C20H22BrN3O2S
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2
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| 1 |
IC50 = 0.8 nM
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| 2 |
Ki = 5 nM
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CP0376998
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4-[3-(1,2,3,6-Tetrahydro-pyridin-4-yl)-indole-1-sulfonyl]-phenylamine
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C19H19N3O2S
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2
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| 1 |
IC50 = 0.8 nM
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| 2 |
Ki = 2 nM
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CP0485096
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1-(3,4-Dimethoxy-benzenesulfonyl)-3-((S)-1-methyl-pyrrolidin-2-ylmethyl)-1H-indole
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C22H26N2O4S
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2
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| 1 |
IC50 = 0.8 nM
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| 2 |
Ki = 8 nM
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CP0399778
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1-(5-Chloro-thiophene-2-sulfonyl)-3-((S)-1-methyl-pyrrolidin-2-ylmethyl)-1H-indole
Show/Hide
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C18H19ClN2O2S2
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2
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| 1 |
IC50 = 1 nM
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| 2 |
Ki = 4 nM
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CP0873366
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5-Chloro-3-methyl-benzo[b]thiophene-2-sulfonic acid [3-((S)-1-methyl-pyrrolidin-2-ylmethyl)-1H-indol-5-yl]-amide
Show/Hide
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C23H24ClN3O2S2
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2
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| 1 |
IC50 = 1.1 nM
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| 2 |
Ki = 2 nM
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CP0476015
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4-(5-Fluoro-3-piperidin-4-yl-indole-1-sulfonyl)-phenylamine
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C19H20FN3O2S
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2
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| 1 |
IC50 = 1.3 nM
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| 2 |
Ki = 2 nM
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CP0443552
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3-(benzenesulfonyl)-7-methyl-2-methylsulfanylpyrido[1,2-a]pyrimidin-4-imine
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C16H15N3O2S2
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1
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| 1 |
IC50 = 1.3 nM
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CP0493862
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1-isobutyl-5-(4-methylpiperazin-1-yl)-3-(naphthalen-1-ylsulfonyl)-1H-indazole
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C26H30N4O2S
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2
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| 1 |
IC50 = 1.4 nM
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| 2 |
Ki = 1.4 nM
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CP0860619
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4-Bromo-N-[3-((S)-1-methyl-pyrrolidin-2-ylmethyl)-1H-indol-5-yl]-benzenesulfonamide
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C20H22BrN3O2S
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2
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| 1 |
IC50 = 1.6 nM
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| 2 |
Ki = 9 nM
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CP0379546
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1-methyl-3-(naphthalen-1-ylsulfonyl)-5-(piperazin-1-yl)-1H-indazole
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C22H22N4O2S
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2
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| 1 |
IC50 = 1.6 nM
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| 2 |
Ki = 1.6 nM
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CP0393292
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4-[7-(1,2,3,6-Tetrahydro-pyridin-4-yl)-[1,3]dioxolo[4,5-f]indole-5-sulfonyl]-phenylamine
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C20H19N3O4S
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2
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| 1 |
IC50 = 1.7 nM
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| 2 |
Ki = 1 nM
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CP0379597
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1-ethyl-5-(4-methylpiperazin-1-yl)-3-(naphthalen-1-ylsulfonyl)-1H-indazole
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C24H26N4O2S
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2
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| 1 |
IC50 = 1.7 nM
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| 2 |
Ki = 1.7 nM
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CP0522157
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1-methyl-5-(4-methylpiperazin-1-yl)-3-(naphthalen-1-ylsulfonyl)-1H-indazole
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C23H24N4O2S
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2
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| 1 |
IC50 = 1.7 nM
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| 2 |
Ki = 1.7 nM
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CP0502707
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1-isopropyl-5-(4-methylpiperazin-1-yl)-3-(naphthalen-1-ylsulfonyl)-1H-indazole
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C25H28N4O2S
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2
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| 1 |
IC50 = 1.8 nM
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| 2 |
Ki = 1.8 nM
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CP0522158
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5-(4-methylpiperazin-1-yl)-3-(naphthalen-1-ylsulfonyl)-1-propyl-1H-indazole
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C25H28N4O2S
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2
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| 1 |
IC50 = 1.8 nM
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| 2 |
Ki = 1.8 nM
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CP0379599
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1-ethyl-3-(naphthalen-1-ylsulfonyl)-5-(piperazin-1-yl)-1H-indazole
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C23H24N4O2S
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2
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| 1 |
IC50 = 1.9 nM
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| 2 |
Ki = 1.9 nM
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CP0479078
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1-benzyl-5-(4-methylpiperazin-1-yl)-3-(naphthalen-1-ylsulfonyl)-1H-indazole
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C29H28N4O2S
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2
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| 1 |
IC50 = 2 nM
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| 2 |
Ki = 2 nM
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CP0471602
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3-(benzenesulfonyl)-2-ethyliminopyrido[1,2-a]pyrimidin-4-amine
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C16H16N4O2S
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1
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| 1 |
IC50 = 2 nM
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CP0502706
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3-(naphthalen-1-ylsulfonyl)-5-(piperazin-1-yl)-1-propyl-1H-indazole
Show/Hide
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C24H26N4O2S
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2
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| 1 |
IC50 = 2.2 nM
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| 2 |
Ki = 2.2 nM
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CP0415729
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3-(benzenesulfonyl)-2-methyliminopyrido[1,2-a]pyrimidin-4-amine
Show/Hide
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C15H14N4O2S
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1
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| 1 |
IC50 = 2.4 nM
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CP0376224
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1-(2-Fluoro-benzenesulfonyl)-3-(1,2,3,6-tetrahydro-pyridin-4-yl)-1H-indole
Show/Hide
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C19H17FN2O2S
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2
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| 1 |
IC50 = 2.7 nM
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| 2 |
Ki = 1 nM
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CP0379601
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1-isopropyl-3-(naphthalen-1-ylsulfonyl)-5-(piperazin-1-yl)-1H-indazole
Show/Hide
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C24H26N4O2S
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2
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| 1 |
IC50 = 2.9 nM
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| 2 |
Ki = 2.9 nM
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CP0523798
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1-ethyl-3-(phenylsulfonyl)-5-(piperazin-1-yl)-1H-indazole
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C19H22N4O2S
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2
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| 1 |
IC50 = 2.9 nM
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| 2 |
Ki = 2.9 nM
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CP0504424
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1-methyl-3-(phenylsulfonyl)-5-(piperazin-1-yl)-1H-indazole
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C18H20N4O2S
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2
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| 1 |
IC50 = 3.2 nM
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| 2 |
Ki = 3.2 nM
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CP0388190
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3-(benzenesulfonyl)-9-methyl-2-methylsulfanylpyrido[1,2-a]pyrimidin-4-imine
Show/Hide
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C16H15N3O2S2
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1
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| 1 |
IC50 = 3.4 nM
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CP0703997
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3-Amino-N-[3-(naphthalen-1-sulfonyl)-1H-indazol-5-yl]-propionamide HCl
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C20H19ClN4O3S
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2
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| 1 |
IC50 = 3.8 nM
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| 2 |
Ki = 1.5 nM
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CP0409802
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1-(2-Fluoro-benzenesulfonyl)-3-(1-methyl-1,2,3,6-tetrahydro-pyridin-4-yl)-1H-indole
Show/Hide
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C20H19FN2O2S
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2
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| 1 |
IC50 = 3.9 nM
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| 2 |
Ki = 10 nM
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CP0043132
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3-Benzenesulfonyl-2-methylsulfanyl-pyrido[1,2-a]pyrimidin-(4E)-ylideneamine
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C15H13N3O2S2
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1
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| 1 |
IC50 = 4 nM
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CP0436439
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5-Methoxy-1-(naphthalene-2-sulfonyl)-3-(1,2,3,6-tetrahydro-pyridin-4-yl)-1H-indole
Show/Hide
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C24H22N2O3S
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2
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| 1 |
IC50 = 4.1 nM
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| 2 |
Ki = 19 nM
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CP0479094
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1-isobutyl-3-(naphthalen-1-ylsulfonyl)-5-(piperazin-1-yl)-1H-indazole
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C25H28N4O2S
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2
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| 1 |
IC50 = 4.6 nM
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| 2 |
Ki = 4.6 nM
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CP0419113
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2-[3-(6-chloroimidazo[2,1-b][1,3]thiazol-5-yl)sulfonylpyrrolo[2,3-b]pyridin-1-yl]-N-methylethanamine
Show/Hide
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C15H14ClN5O2S2
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2
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| 1 |
IC50 = 5.4 nM
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| 2 |
Ki = 0.9 nM
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CP0443276
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2-[3-(3-fluorophenyl)sulfonylpyrrolo[2,3-b]pyridin-1-yl]-N-methylethanamine
Show/Hide
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C16H16FN3O2S
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2
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| 1 |
IC50 = 6.2 nM
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|
| 2 |
Ki = 1 nM
|
|
|
|
CP0436093
|
1-(4-Methoxy-benzenesulfonyl)-3-piperidin-3-yl-1H-indole
Show/Hide
|
C20H22N2O3S
|
2
|
| 1 |
IC50 = 7.3 nM
|
|
|
| 2 |
Ki = 10 nM
|
|
|
|
CP0448064
|
1-(3,4-Dichloro-benzenesulfonyl)-3-((S)-1-methyl-pyrrolidin-2-ylmethyl)-1H-indole
Show/Hide
|
C20H20Cl2N2O2S
|
2
|
| 1 |
IC50 = 7.3 nM
|
|
|
| 2 |
Ki = 12 nM
|
|
|
|
CP0406091
|
1-benzyl-3-(naphthalen-1-ylsulfonyl)-5-(piperazin-1-yl)-1H-indazole
Show/Hide
|
C28H26N4O2S
|
2
|
| 1 |
IC50 = 7.5 nM
|
|
|
| 2 |
Ki = 7.5 nM
|
|
|
|
CP0453187
|
4-(3-(S)-1-Pyrrolidin-2-ylmethyl-indole-1-sulfonyl)-phenylamine
Show/Hide
|
C19H21N3O2S
|
2
|
| 1 |
IC50 = 7.6 nM
|
|
|
| 2 |
Ki = 7 nM
|
|
|
|
CP0073024
|
1-sulfonylindazole, 7a
Show/Hide
|
C23H22N4O3S
|
2
|
| 1 |
IC50 = 8 nM
|
|
|
| 2 |
Ki = 2.3 nM
|
|
|
|
CP0845189
|
3-[(6-chloroimidazo[2,1-b][1,3]thiazol-5-yl)sulfonyl]-1-(1-isopropylpiperidin-3-yl)-1H-pyrrolo[2,3-b]pyridine
Show/Hide
|
C20H24ClN5O2S2
|
2
|
| 1 |
IC50 = 8 nM
|
|
|
| 2 |
Ki = 1.7 nM
|
|
|
|
CP0379542
|
5-(4-Methylpiperazin-1-yl)-3-(1-naphthalenesulfonyl)-1H-indazole
Show/Hide
|
C22H22N4O2S
|
2
|
| 1 |
IC50 = 8 nM
|
|
|
| 2 |
Ki = 1.6 nM
|
|
|
|
CP0436095
|
1-(4-Chloro-benzenesulfonyl)-3-((S)-1-methyl-pyrrolidin-2-ylmethyl)-1H-indole
Show/Hide
|
C20H21ClN2O2S
|
2
|
| 1 |
IC50 = 8.2 nM
|
|
|
| 2 |
Ki = 7 nM
|
|
|
|
CP0671735
|
N-(3-(Naphthalen-1-ylsulfonyl)-1H-indazol-5-yl)piperidine-4-carboxamide HCl
Show/Hide
|
C23H23ClN4O3S
|
2
|
| 1 |
IC50 = 8.2 nM
|
|
|
| 2 |
Ki = 1.1 nM
|
|
|
|
CP0431017
|
2-[3-(3-chlorophenyl)sulfonylpyrrolo[2,3-b]pyridin-1-yl]-N-methylethanamine
Show/Hide
|
C16H16ClN3O2S
|
2
|
| 1 |
IC50 = 8.3 nM
|
|
|
| 2 |
Ki = 0.3 nM
|
|
|
|
CP0393293
|
4-(6-Chloro-3-piperidin-4-yl-indole-1-sulfonyl)-phenylamine
Show/Hide
|
C19H20ClN3O2S
|
2
|
| 1 |
IC50 = 8.5 nM
|
|
|
| 2 |
Ki = 3 nM
|
|
|
|
CP0409239
|
1-(2-Chloro-benzenesulfonyl)-3-(1,2,3,6-tetrahydro-pyridin-4-yl)-1H-indole
Show/Hide
|
C19H17ClN2O2S
|
2
|
| 1 |
IC50 = 8.8 nM
|
|
|
| 2 |
Ki = 0.4 nM
|
|
|
|
CP0379544
|
5-(4-methylpiperazin-1-yl)-3-(phenylsulfonyl)-1H-indazole
Show/Hide
|
C18H20N4O2S
|
2
|
| 1 |
IC50 = 8.8 nM
|
|
|
| 2 |
Ki = 1.9 nM
|
|
|
|
CP0461785
|
3-(benzenesulfonyl)-4-imino-2-methylsulfanylpyrido[1,2-a]pyrimidine-7-carboxamide
Show/Hide
|
C16H14N4O3S2
|
1
|
| 1 |
IC50 = 8.8 nM
|
|
|
|
CP0394049
|
5-Fluoro-1-(naphthalene-1-sulfonyl)-3-(1,2,3,6-tetrahydro-pyridin-4-yl)-1H-indole
Show/Hide
|
C23H19FN2O2S
|
2
|
| 1 |
IC50 = 9 nM
|
|
|
| 2 |
Ki = 4 nM
|
|
|
|
CP0376177
|
1-(3-Chloro-benzenesulfonyl)-3-(1-methyl-1,2,3,6-tetrahydro-pyridin-4-yl)-1H-indole
Show/Hide
|
C20H19ClN2O2S
|
2
|
| 1 |
IC50 = 9.4 nM
|
|
|
| 2 |
Ki = 1 nM
|
|
|
|
CP0869818
|
5-(3-(2-aminoethyl)-1H-indol-1-ylsulfonyl)-3-methyl-2,3-dihydrothiazol-2-amine
Show/Hide
|
C14H18N4O2S2
|
2
|
| 1 |
IC50 = 9.6 nM
|
|
|
| 2 |
Ki = 10 nM
|
|
|
|
CP0436440
|
4-[5-Fluoro-3-(1,2,3,6-tetrahydro-pyridin-4-yl)-indole-1-sulfonyl]-phenylamine
Show/Hide
|
C19H18FN3O2S
|
2
|
| 1 |
IC50 = 9.7 nM
|
|
|
| 2 |
Ki = 1 nM
|
|
|
|
CP0073023
|
1-sulfonylindazole, 7b
Show/Hide
|
C23H22N4O3S
|
2
|
| 1 |
IC50 = 10 nM
|
|
|
| 2 |
Ki = 1.3 nM
|
|
|
|
CP0886304
|
3-(6-chloro-imidazo[2,1-b]thiazole-5-sulfonyl)-1-(1-ethyl-pyrrolidin-3-yl)-1H-pyrrolo[2,3-b]pyridine
Show/Hide
|
C18H20ClN5O2S2
|
2
|
| 1 |
IC50 = 10 nM
|
|
|
| 2 |
Ki = 1.4 nM
|
|
|
|
CP0873365
|
Naphthalene-2-sulfonic acid [3-((S)-1-methyl-pyrrolidin-2-ylmethyl)-1H-indol-5-yl]-amide
Show/Hide
|
C24H25N3O2S
|
2
|
| 1 |
IC50 = 10.4 nM
|
|
|
| 2 |
Ki = 1 nM
|
|
|
|
CP0073022
|
1-sulfonylindazole, 6a
Show/Hide
|
C20H18N4O3S
|
2
|
| 1 |
IC50 = 11 nM
|
|
|
| 2 |
Ki = 7.9 nM
|
|
|
|
CP0405164
|
1-(5-Chloro-3-methyl-benzo[b]thiophene-2-sulfonyl)-3-((S)-1-methyl-pyrrolidin-2-ylmethyl)-1H-indole
Show/Hide
|
C23H23ClN2O2S2
|
2
|
| 1 |
IC50 = 11 nM
|
|
|
| 2 |
Ki = 11 nM
|
|
|
|
CP0373270
|
3-(5-chloro-thiophene-2-sulfonyl)-1-pyrrolidin-3-yl-1H-pyrrolo[2,3-b]pyridine
Show/Hide
|
C16H16ClN3O2S2
|
2
|
| 1 |
IC50 = 11 nM
|
|
|
| 2 |
Ki = 1 nM
|
|
|
|
CP0461790
|
3-(2-chlorophenyl)sulfonyl-2-methylsulfanylpyrido[1,2-a]pyrimidin-4-imine
Show/Hide
|
C15H12ClN3O2S2
|
1
|
| 1 |
IC50 = 11 nM
|
|
|
|
CP0394038
|
4-[6-Chloro-3-(1,2,3,6-tetrahydro-pyridin-4-yl)-indole-1-sulfonyl]-phenylamine
Show/Hide
|
C19H18ClN3O2S
|
2
|
| 1 |
IC50 = 11.2 nM
|
|
|
| 2 |
Ki = 3 nM
|
|
|
|
CP0703995
|
3-(3-Chlorophenylsulfonyl)-N-(piperidin-4-yl)-1H-indazol-5-amine HCl
Show/Hide
|
C18H20Cl2N4O2S
|
2
|
| 1 |
IC50 = 12 nM
|
|
|
| 2 |
Ki = 1 nM
|
|
|
|
CP0388193
|
3-(benzenesulfonyl)-7-bromo-9-methyl-2-methylsulfanylpyrido[1,2-a]pyrimidin-4-imine
Show/Hide
|
C16H14BrN3O2S2
|
1
|
| 1 |
IC50 = 12 nM
|
|
|
|
CP0434472
|
3-(benzenesulfonyl)-2-ethoxypyrido[1,2-a]pyrimidin-4-imine
Show/Hide
|
C16H15N3O3S
|
1
|
| 1 |
IC50 = 12 nM
|
|
|
|
CP0277626
|
(3S)-1-[3-(1-Naphthylsulfonyl)-1H-indazol-5-yl]pyrrolidin-3-amine
Show/Hide
|
C21H20N4O2S
|
1
|
| 1 |
IC50 = 12.5 nM
|
|
|
|
CP0379545
|
3-(Naphthalen-1-ylsulfonyl)-5-(piperazin-1-yl)-1H-indazole
Show/Hide
|
C21H20N4O2S
|
2
|
| 1 |
IC50 = 13 nM
|
|
|
| 2 |
Ki = 1.1 nM
|
|
|
|
CP0916810
|
N1-3-(Napthalene-1-sulfonyl-1H-indazol-5-yl)-ethane-1,2-diamine HCl
Show/Hide
|
C19H19ClN4O2S
|
2
|
| 1 |
IC50 = 13 nM
|
|
|
| 2 |
Ki = 6.7 nM
|
|
|
|
CP0431575
|
1-Benzenesulfonyl-3-(1-methyl-1,2,3,6-tetrahydro-pyridin-4-yl)-1H-indole
Show/Hide
|
C20H20N2O2S
|
2
|
| 1 |
IC50 = 13.8 nM
|
|
|
| 2 |
Ki = 2 nM
|
|
|
|
CP0703996
|
3-(4-Isopropylphenylsulfonyl)-N-(piperidin-4-yl)-1Hindazol-5-amine HCl
Show/Hide
|
C21H27ClN4O2S
|
2
|
| 1 |
IC50 = 14 nM
|
|
|
| 2 |
Ki = 1 nM
|
|
|
|
CP0860617
|
(S)-N-(3-((1-methylpyrrolidin-2-yl)methyl)-1H-indol-5-yl)-3-(trifluoromethyl)benzenesulfonamide
Show/Hide
|
C21H22F3N3O2S
|
2
|
| 1 |
IC50 = 14.1 nM
|
|
|
| 2 |
Ki = 12 nM
|
|
|
|
CP0436433
|
1-(5-Chloro-thiophene-2-sulfonyl)-3-(1,2,3,6-tetrahydro-pyridin-4-yl)-1H-indole
Show/Hide
|
C17H15ClN2O2S2
|
2
|
| 1 |
IC50 = 14.1 nM
|
|
|
| 2 |
Ki = 3 nM
|
|
|
|
CP0193613
|
1-Benzyl-3-(1-methyl-1,2,3,6-tetrahydro-pyridin-4-yl)-1H-indole
Show/Hide
|
C21H22N2
|
2
|
| 1 |
IC50 = 14.8 nM
|
|
|
| 2 |
Ki = 10 nM
|
|
|
|
CP0492307
|
2-[3-(2,5-dichlorophenyl)sulfonylpyrrolo[2,3-b]pyridin-1-yl]-N,N-dimethylethanamine
Show/Hide
|
C17H17Cl2N3O2S
|
2
|
| 1 |
IC50 = 15 nM
|
|
|
| 2 |
Ki = 11.7 nM
|
|
|
|
CP0688856
|
[3-(Naphthalen-1-sulfonyl)-1H-indazol-5-yl]-piperidin-4-yl-amine HCl
Show/Hide
|
C22H23ClN4O2S
|
2
|
| 1 |
IC50 = 15 nM
|
|
|
| 2 |
Ki = 0.7 nM
|
|
|
|
CP0405165
|
4-[3-(1-Methyl-pyrrolidin-3-yl)-indole-1-sulfonyl]-phenylamine
Show/Hide
|
C19H21N3O2S
|
2
|
| 1 |
IC50 = 15.5 nM
|
|
|
| 2 |
Ki = 1 nM
|
|
|
|
CP0038773
|
(3R)-1-[3-(1-Naphthylsulfonyl)-1H-indazol-5-yl]pyrrolidin-3-amine
Show/Hide
|
C21H20N4O2S
|
1
|
| 1 |
IC50 = 15.7 nM
|
|
|
|
CP0742584
|
3-(Naphthalen-2-ylsulfonyl)-N-(piperidin-4-yl)-1H-indazol-5-amine HCl
Show/Hide
|
C22H23ClN4O2S
|
2
|
| 1 |
IC50 = 16 nM
|
|
|
| 2 |
Ki = 0.6 nM
|
|
|
|
CP0277627
|
1-[3-(1-Naphthylsulfonyl)-1H-indazol-5-yl]azetidin-3-amine
Show/Hide
|
C20H18N4O2S
|
1
|
| 1 |
IC50 = 16.5 nM
|
|
|
|
CP0402010
|
3-(3-chlorophenylsulfonyl)-1-(1-methylpyrrolidin-3-yl)-1H-indole
Show/Hide
|
C19H19ClN2O2S
|
2
|
| 1 |
IC50 = 17 nM
|
|
|
| 2 |
Ki = 1.3 nM
|
|
|
|
CP0502282
|
7-(4-methylpiperazin-1-yl)-3-(naphthalen-1-ylsulfonyl)-1H-indazole
Show/Hide
|
C22H22N4O2S
|
2
|
| 1 |
IC50 = 17 nM
|
|
|
| 2 |
Ki = 4.6 nM
|
|
|
|
CP0025667
|
2-[4-(4-Methyl-benzyl)-piperazin-1-yl]-1-(2-methyl-2,3-dihydro-indol-1-yl)-ethanone
Show/Hide
|
C18H19ClN4
|
2
|
| 1 |
IC50 = 17 nM
|
|
|
| 2 |
Ki = 17 nM
|
|
|
|
CP0421798
|
2-{1-[(3,4-dimethoxybenzene)sulfonyl]-1H-indol-3-yl}ethan-1-amine
Show/Hide
|
C18H20N2O4S
|
2
|
| 1 |
IC50 = 17.5 nM
|
|
|
| 2 |
Ki = 7 nM
|
|
|
|
CP0148893
|
(3S)-N,N-Dimethyl-1-[3-(1-naphthylsulfonyl)-1H-indazol-5-yl]pyrrolidin-3-amine
Show/Hide
|
C23H24N4O2S
|
1
|
| 1 |
IC50 = 17.5 nM
|
|
|
|
CP0398840
|
5-fluoro-3-(3-fluorophenylsulfonyl)-1-(piperidin-3-yl)-1H-indole
Show/Hide
|
C19H18F2N2O2S
|
2
|
| 1 |
IC50 = 18 nM
|
|
|
| 2 |
Ki = 4 nM
|
|
|
|
CP0486747
|
3-(3,4-dichlorophenyl)sulfonyl-2-methylsulfanylpyrido[1,2-a]pyrimidin-4-imine
Show/Hide
|
C15H11Cl2N3O2S2
|
1
|
| 1 |
IC50 = 18 nM
|
|
|
|
CP0848237
|
N-(Piperidin-4-yl)-3-(m-tolylsulfonyl)-1H-indazol-5-amine HCl
Show/Hide
|
C19H23ClN4O2S
|
2
|
| 1 |
IC50 = 19 nM
|
|
|
| 2 |
Ki = 0.8 nM
|
|
|
|
CP0862726
|
3-(Naphthalen-1-ylsulfonyl)-5-(piperazin-1-ylmethyl)-1Hindazole HCl
Show/Hide
|
C22H23ClN4O2S
|
2
|
| 1 |
IC50 = 19 nM
|
|
|
| 2 |
Ki = 0.24 nM
|
|
|
|
CP0310110
|
SB-258585
Show/Hide
|
C18H22IN3O3S
|
2
|
| 1 |
IC50 = 19 nM
|
|
|
| 2 |
Ki = 2.512 nM
|
|
|
|
CP0430190
|
1-Benzenesulfonyl-3-piperidin-4-yl-1H-indole
Show/Hide
|
C19H20N2O2S
|
2
|
| 1 |
IC50 = 19.5 nM
|
|
|
| 2 |
Ki = 12 nM
|
|
|
|
CP0371931
|
3-(1-Benzyl-pyrrolidin-3-yl)-1-(2-bromo-benzenesulfonyl)-1H-indole
Show/Hide
|
C25H23BrN2O2S
|
2
|
| 1 |
IC50 = 21 nM
|
|
|
| 2 |
Ki = 14 nM
|
|
|
|
CP0848610
|
3-(Naphthalen-1-ylsulfonyl)-N-(piperidin-4-ylmethyl)-1Hindazol-4-amine HCl
Show/Hide
|
C23H25ClN4O2S
|
2
|
| 1 |
IC50 = 21 nM
|
|
|
| 2 |
Ki = 9.5 nM
|
|
|
|
CP0395622
|
3-(benzenesulfonyl)-2-methoxypyrido[1,2-a]pyrimidin-4-imine
Show/Hide
|
C15H13N3O3S
|
1
|
| 1 |
IC50 = 21 nM
|
|
|
|
CP0847577
|
4-Isopropyl-N-[3-((S)-1-methyl-pyrrolidin-2-ylmethyl)-1H-indol-5-yl]-benzenesulfonamide
Show/Hide
|
C23H29N3O2S
|
2
|
| 1 |
IC50 = 21.1 nM
|
|
|
| 2 |
Ki = 3 nM
|
|
|
|
CP0428335
|
pyrrolidinylindole, (S)-5b
Show/Hide
|
C21H22F3N3O2S
|
2
|
| 1 |
IC50 = 21.6 nM
|
|
|
| 2 |
Ki = 10 nM
|
|
|
|
CP0415724
|
3-(4-fluorophenyl)sulfonyl-2-methylsulfanylpyrido[1,2-a]pyrimidin-4-imine
Show/Hide
|
C15H12FN3O2S2
|
1
|
| 1 |
IC50 = 22 nM
|
|
|
|
CP0451858
|
2-[3-(benzenesulfonyl)-7-methoxyindol-1-yl]-N,N-dimethylethanamine
Show/Hide
|
C19H22N2O3S
|
2
|
| 1 |
IC50 = 23 nM
|
|
|
| 2 |
Ki = 25 nM
|
|
|
|
CP0093674
|
3-(3-bromo-benzenesulfonyl)-1-(1-methyl-pyrrolidin-3-yl)-1H-pyrrolo[2,3-b]pyridine
Show/Hide
|
C18H18BrN3O2S
|
2
|
| 1 |
IC50 = 23 nM
|
|
|
| 2 |
Ki = 0.9 nM
|
|
|
|
CP0855615
|
3-(Dimethylamino)-N-(3-(naphthalen-1-ylsulfonyl)-1Hindazol-7-yl)propanamide HCl
Show/Hide
|
C22H23ClN4O3S
|
2
|
| 1 |
IC50 = 23 nM
|
|
|
| 2 |
Ki = 4.8 nM
|
|
|
|
CP0485095
|
4-[3-((S)-1-Methyl-pyrrolidin-2-ylmethyl)-indole-1-sulfonyl]-phenylamine
Show/Hide
|
C20H23N3O2S
|
2
|
| 1 |
IC50 = 24.5 nM
|
|
|
| 2 |
Ki = 3 nM
|
|
|
|
CP0485446
|
4-[3-(1-Benzyl-pyrrolidin-3-yl)-indole-1-sulfonyl]-phenylamine
Show/Hide
|
C25H25N3O2S
|
2
|
| 1 |
IC50 = 25 nM
|
|
|
| 2 |
Ki = 1 nM
|
|
|
|
CP0504494
|
1-sulfonylindazole, 6d
Show/Hide
|
C21H20N4O3S
|
2
|
| 1 |
IC50 = 26 nM
|
|
|
| 2 |
Ki = 1.2 nM
|
|
|
|
CP0427370
|
1-(1-ethylpiperidin-3-yl)-3-(phenylsulfonyl)-1Hpyrrolo[2,3-b]pyridine
Show/Hide
|
C20H23N3O2S
|
2
|
| 1 |
IC50 = 26 nM
|
|
|
| 2 |
Ki = 3.6 nM
|
|
|
|
CP0876435
|
3-(6-chloro-imidazo[2,1-b]thiazole-5-sulfonyl)-1-(1-methyl-pyrrolidin-3-yl)-1H-pyrrolo[2,3-b]pyridine
Show/Hide
|
C17H18ClN5O2S2
|
2
|
| 1 |
IC50 = 26 nM
|
|
|
| 2 |
Ki = 0.8 nM
|
|
|
|
CP0148007
|
1-{3-[(4-Methyl-1-naphthyl)sulfonyl]-1H-indazol-5-yl}piperidin-4-amine
Show/Hide
|
C23H24N4O2S
|
1
|
| 1 |
IC50 = 26.7 nM
|
|
|
|
CP0848233
|
N-(Piperidin-4-yl)-3-(4-(trifluoromethyl)phenylsulfonyl)-1H-indazol-5-amine HCl
Show/Hide
|
C19H20ClF3N4O2S
|
2
|
| 1 |
IC50 = 27 nM
|
|
|
| 2 |
Ki = 1.5 nM
|
|
|
|
CP0093694
|
3-[(4-chlorophenyl)sulfonyl]-1-(1-methylpiperidin-3-yl)-1H-pyrrolo[2,3-b]pyridine
Show/Hide
|
C19H20ClN3O2S
|
2
|
| 1 |
IC50 = 28 nM
|
|
|
| 2 |
Ki = 11.5 nM
|
|
|
|
CP0309914
|
1-[3-(1-Naphthylsulfonyl)-1H-indazol-5-yl]piperidin-4-amine
Show/Hide
|
C22H22N4O2S
|
1
|
| 1 |
IC50 = 28 nM
|
|
|
|
CP0281465
|
3-Benzenesulfonyl-7-fluoro-2-methylsulfanyl-pyrido[1,2-a]pyrimidin-(4Z)-ylideneamine
Show/Hide
|
C15H12FN3O2S2
|
1
|
| 1 |
IC50 = 28 nM
|
|
|
|
CP0443550
|
3-(benzenesulfonyl)-7-chloro-2-methylsulfanylpyrido[1,2-a]pyrimidin-4-imine
Show/Hide
|
C15H12ClN3O2S2
|
1
|
| 1 |
IC50 = 28 nM
|
|
|
|
CP0899501
|
N1-(3-(Naphthalen-1-ylsulfonyl)-1H-indazol-6-yl)propane-1,2-diamine HCl
Show/Hide
|
C20H21ClN4O2S
|
2
|
| 1 |
IC50 = 30 nM
|
|
|
| 2 |
Ki = 1.4 nM
|
|
|
|
CP0431536
|
5-Fluoro-1-(4-fluoro-benzenesulfonyl)-3-(1,2,3,6-tetrahydro-pyridin-4-yl)-1H-indole
Show/Hide
|
C19H16F2N2O2S
|
2
|
| 1 |
IC50 = 31 nM
|
|
|
| 2 |
Ki = 3 nM
|
|
|
|
CP0430195
|
4-[5-Bromo-3-(1,2,3,6-tetrahydro-pyridin-4-yl)-indole-1-sulfonyl]-phenylamine
Show/Hide
|
C19H18BrN3O2S
|
2
|
| 1 |
IC50 = 33.7 nM
|
|
|
| 2 |
Ki = 7 nM
|
|
|
|
CP0282297
|
1-(3-(3-chlorophenylsulfonyl)-1H-indazol-5-yl)piperidin-4-amine
Show/Hide
|
C18H19ClN4O2S
|
1
|
| 1 |
IC50 = 33.7 nM
|
|
|
|
CP0379541
|
5-(4-Methylpiperazin-1-yl)-3-(m-tolylsulfonyl)-1H-indazole
Show/Hide
|
C19H22N4O2S
|
2
|
| 1 |
IC50 = 38 nM
|
|
|
| 2 |
Ki = 0.9 nM
|
|
|
|
CP0043595
|
(3R)-N,N-Dimethyl-1-[3-(1-naphthylsulfonyl)-1H-indazol-5-yl]pyrrolidin-3-amine
Show/Hide
|
C23H24N4O2S
|
1
|
| 1 |
IC50 = 39.6 nM
|
|
|
|
CP0493858
|
3-(2,6-Dichlorophenylsulfonyl)-5-(4-methylpiperazin-1-yl)-1Hindazole
Show/Hide
|
C18H18Cl2N4O2S
|
2
|
| 1 |
IC50 = 40 nM
|
|
|
| 2 |
Ki = 2.6 nM
|
|
|
|
CP0500603
|
1-(1-(2-(dimethylamino)ethyl)-3-(3-fluorophenylsulfonyl)-1H-pyrrolo[3,2-b]pyridin-5-yl)ethanone
Show/Hide
|
C19H20FN3O3S
|
2
|
| 1 |
IC50 = 41 nM
|
|
|
| 2 |
Ki = 11.3 nM
|
|
|
|
CP0443275
|
3-(benzenesulfonyl)-8-methyl-2-methylsulfanylpyrido[1,2-a]pyrimidin-4-imine
Show/Hide
|
C16H15N3O2S2
|
1
|
| 1 |
IC50 = 41 nM
|
|
|
|
CP0525354
|
CHEMBL3113363
Show/Hide
|
C16H16N4O3S
|
1
|
| 1 |
IC50 = 42 nM
|
|
|
|
CP0376179
|
1-(4-Fluoro-benzenesulfonyl)-3-(1-methyl-1,2,3,6-tetrahydro-pyridin-4-yl)-1H-indole
Show/Hide
|
C20H19FN2O2S
|
2
|
| 1 |
IC50 = 42.7 nM
|
|
|
| 2 |
Ki = 5 nM
|
|
|
|
CP0376208
|
1-Benzenesulfonyl-3-(1,2,3,6-tetrahydro-pyridin-4-yl)-1H-indole
Show/Hide
|
C19H18N2O2S
|
2
|
| 1 |
IC50 = 43 nM
|
|
|
| 2 |
Ki = 2 nM
|
|
|
|
CP0485445
|
1-(4-Iodo-benzenesulfonyl)-3-(1-methyl-pyrrolidin-3-yl)-1H-indole
Show/Hide
|
C19H19IN2O2S
|
2
|
| 1 |
IC50 = 43.6 nM
|
|
|
| 2 |
Ki = 1 nM
|
|
|
|
CP0848466
|
3-(4-Chlorophenylsulfonyl)-N-(piperidin-4-yl)-1H-indazol-5-amine HCl
Show/Hide
|
C18H20Cl2N4O2S
|
2
|
| 1 |
IC50 = 44 nM
|
|
|
| 2 |
Ki = 2.3 nM
|
|
|
|
CP0430085
|
N,N-dimethyl-2-(3-naphthalen-1-ylsulfonylindol-1-yl)ethanamine
Show/Hide
|
C22H22N2O2S
|
2
|
| 1 |
IC50 = 47 nM
|
|
|
| 2 |
Ki = 3.7 nM
|
|
|
|
CP0923319
|
N-(3-(Naphthalen-1-ylsulfonyl)-1H-indazol-7-yl)piperidine-3-carboxamide HCl
Show/Hide
|
C23H23ClN4O3S
|
2
|
| 1 |
IC50 = 48 nM
|
|
|
| 2 |
Ki = 9.8 nM
|
|
|
|
CP0476066
|
1-(4-Iodo-benzenesulfonyl)-3-((S)-1-methyl-pyrrolidin-2-ylmethyl)-1H-indole
Show/Hide
|
C20H21IN2O2S
|
2
|
| 1 |
IC50 = 49.5 nM
|
|
|
| 2 |
Ki = 3 nM
|
|
|
|
CP0277694
|
3-[(2-fluorophenyl)sulfonyl]-1-piperidin-3-yl-1Hpyrrolo[2,3-b]pyridine
Show/Hide
|
C18H18FN3O2S
|
2
|
| 1 |
IC50 = 50 nM
|
|
|
| 2 |
Ki = 2 nM
|
|
|
|
CP0325786
|
3-(2-fluoro-benzenesulfonyl)-1-pyrrolidin-3-yl-1Hpyrrolo[2,3-b]pyridine
Show/Hide
|
C17H16FN3O2S
|
2
|
| 1 |
IC50 = 50 nM
|
|
|
| 2 |
Ki = 2 nM
|
|
|
|
CP0487049
|
3-(4-chloro-2,5-dimethylphenyl)sulfonyl-2-methylsulfanylpyrido[1,2-a]pyrimidin-4-imine
Show/Hide
|
C17H16ClN3O2S2
|
1
|
| 1 |
IC50 = 50 nM
|
|
|
|
CP0214619
|
1-{3-[(4-Isopropylphenyl)sulfonyl]-1H-indazol-5-yl}piperidin-4-amine
Show/Hide
|
C21H26N4O2S
|
1
|
| 1 |
IC50 = 51.7 nM
|
|
|
|
CP0538892
|
3-(benzenesulfonyl)-2-methylsulfanylpyrido[1,2-a]pyrimidin-4-one
Show/Hide
|
C15H12N2O3S2
|
1
|
| 1 |
IC50 = 52 nM
|
|
|
|
CP0371930
|
1-(4-Fluoro-benzenesulfonyl)-3-(1-methyl-pyrrolidin-3-yl)-1H-indole
Show/Hide
|
C19H19FN2O2S
|
2
|
| 1 |
IC50 = 52.5 nM
|
|
|
| 2 |
Ki = 2 nM
|
|
|
|
CP0474546
|
1-sulfonylindazole, 6e
Show/Hide
|
C22H22N4O3S
|
2
|
| 1 |
IC50 = 53 nM
|
|
|
| 2 |
Ki = 1.8 nM
|
|
|
|
CP0039674
|
1-(2-bromophenyl)sulfonyl-3-(1-methylpyrrolidin-3-yl)indole
Show/Hide
|
C19H19BrN2O2S
|
2
|
| 1 |
IC50 = 53.3 nM
|
|
|
| 2 |
Ki = 1 nM
|
|
|
|
CP0493860
|
3-(2-fluorophenylsulfonyl)-5-(4-methylpiperazin-1-yl)-1H-indazole
Show/Hide
|
C18H19FN4O2S
|
2
|
| 1 |
IC50 = 54 nM
|
|
|
| 2 |
Ki = 5.5 nM
|
|
|
|
CP0306929
|
3-Benzenesulfonyl-2-methylsulfanyl-pyrimido[2,1-a]isoquinolin-(4Z)-ylideneamine
Show/Hide
|
C19H15N3O2S2
|
1
|
| 1 |
IC50 = 55 nM
|
|
|
|
CP0291338
|
3-benzenesulfonyl-1-(1-ethyl-pyrrolidin-3-yl)-1Hpyrrolo[2,3-b]pyridine
Show/Hide
|
C19H21N3O2S
|
2
|
| 1 |
IC50 = 56 nM
|
|
|
| 2 |
Ki = 11 nM
|
|
|
|
CP0862082
|
3-(Naphthalen-1-ylsulfonyl)-N-(piperidin-4-yl)-1H-indazol-4-amine HCl
Show/Hide
|
C22H23ClN4O2S
|
2
|
| 1 |
IC50 = 56 nM
|
|
|
| 2 |
Ki = 2.8 nM
|
|
|
|
CP0525353
|
3-(benzenesulfonyl)-7-bromo-2-methylsulfanylpyrido[1,2-a]pyrimidin-4-imine
Show/Hide
|
C15H12BrN3O2S2
|
1
|
| 1 |
IC50 = 56 nM
|
|
|
|
CP0485444
|
3-((S)-1-Methyl-pyrrolidin-2-ylmethyl)-1-(toluene-4-sulfonyl)-1H-indole
Show/Hide
|
C21H24N2O2S
|
2
|
| 1 |
IC50 = 56.3 nM
|
|
|
| 2 |
Ki = 5 nM
|
|
|
|
CP0479077
|
3-(3-Methoxyphenylsulfonyl)-5-(4-methylpiperazin-1-yl)-1Hindazole
Show/Hide
|
C19H22N4O3S
|
2
|
| 1 |
IC50 = 57 nM
|
|
|
| 2 |
Ki = 1.1 nM
|
|
|
|
CP0395621
|
3-(benzenesulfonyl)-2-methylsulfanylpyrimido[1,2-h][1,7]naphthyridin-4-imine
Show/Hide
|
C18H14N4O2S2
|
1
|
| 1 |
IC50 = 57 nM
|
|
|
|
CP0063547
|
2-Methylsulfanyl-3-(naphthalene-2-sulfonyl)-pyrido[1,2-a]pyrimidin-(4Z)-ylideneamine
Show/Hide
|
C19H15N3O2S2
|
1
|
| 1 |
IC50 = 59 nM
|
|
|
|
CP0497290
|
1-(1-methylpyrrolidin-3-yl)-3-(naphthalen-1-ylsulfonyl)-1H-indole
Show/Hide
|
C23H22N2O2S
|
2
|
| 1 |
IC50 = 60 nM
|
|
|
| 2 |
Ki = 6 nM
|
|
|
|
CP0415725
|
3-(benzenesulfonyl)-7-benzyl-9-methyl-2-methylsulfanylpyrido[1,2-a]pyrimidin-4-imine
Show/Hide
|
C23H21N3O2S2
|
1
|
| 1 |
IC50 = 60 nM
|
|
|
|
CP0461788
|
3-(benzenesulfonyl)-7-methyl-2-(5-methylpyridin-2-yl)iminopyrido[1,2-a]pyrimidin-4-amine
Show/Hide
|
C21H19N5O2S
|
1
|
| 1 |
IC50 = 60 nM
|
|
|
|
CP0399779
|
3-(1-Benzyl-pyrrolidin-3-yl)-1-(3,4-dichloro-benzenesulfonyl)-1H-indole
Show/Hide
|
C25H22Cl2N2O2S
|
2
|
| 1 |
IC50 = 61 nM
|
|
|
| 2 |
Ki = 15 nM
|
|
|
|
CP0493861
|
3-(3-Chlorophenylsulfonyl)-5-(4-methylpiperazin-1-yl)-1H-indazole
Show/Hide
|
C18H19ClN4O2S
|
2
|
| 1 |
IC50 = 62 nM
|
|
|
| 2 |
Ki = 1 nM
|
|
|
|
CP0415722
|
3-(4-tert-butylphenyl)sulfonyl-2-methylsulfanylpyrido[1,2-a]pyrimidin-4-imine
Show/Hide
|
C19H21N3O2S2
|
1
|
| 1 |
IC50 = 65 nM
|
|
|
|
CP0291340
|
1-(1-ethylpiperidin-3-yl)-3-[(4-chlorophenyl)sulfonyl]-1H-pyrrolo[2,3-b]pyridine
Show/Hide
|
C20H22ClN3O2S
|
2
|
| 1 |
IC50 = 70 nM
|
|
|
| 2 |
Ki = 33.5 nM
|
|
|
|
CP0062984
|
1-{3-[(5-Chloro-1-naphthyl)sulfonyl]-1H-indazol-5-yl}piperidin-4-amine
Show/Hide
|
C22H21ClN4O2S
|
1
|
| 1 |
IC50 = 70.1 nM
|
|
|
|
CP0502460
|
8-(1-(1-methylpyrrolidin-3-yl)-1H-indol-3-ylsulfonyl)quinoline
Show/Hide
|
C22H21N3O2S
|
2
|
| 1 |
IC50 = 76 nM
|
|
|
| 2 |
Ki = 2.8 nM
|
|
|
|
CP0436094
|
1-(2-Bromo-benzenesulfonyl)-3-((S)-1-methyl-pyrrolidin-2-ylmethyl)-1H-indole
Show/Hide
|
C20H21BrN2O2S
|
2
|
| 1 |
IC50 = 76.5 nM
|
|
|
| 2 |
Ki = 7 nM
|
|
|
|
CP0372405
|
7-(naphthalen-1-ylsulfonyl)-2-(piperazin-1-yl)benzo[d]oxazole
Show/Hide
|
C21H19N3O3S
|
2
|
| 1 |
IC50 = 77 nM
|
|
|
| 2 |
Ki = 7.1 nM
|
|
|
|
CP0411174
|
3-(3-chlorophenylsulfonyl)-6-methoxy-1-(pyrrolidin-3-yl)-1H-indole
Show/Hide
|
C19H19ClN2O3S
|
2
|
| 1 |
IC50 = 80 nM
|
|
|
| 2 |
Ki = 4.6 nM
|
|
|
|
CP0154123
|
3-Benzenesulfonyl-8-ethyl-2-methylsulfanyl-pyrido[1,2-a]pyrimidin-(4Z)-ylideneamine
Show/Hide
|
C17H17N3O2S2
|
1
|
| 1 |
IC50 = 80 nM
|
|
|
|
CP0457934
|
1-Benzenesulfonyl-3-((S)-1-methyl-pyrrolidin-2-ylmethyl)-1H-indole; oxalic acid
Show/Hide
|
C20H22N2O2S
|
2
|
| 1 |
IC50 = 81.4 nM
|
|
|
| 2 |
Ki = 5 nM
|
|
|
|
CP0411092
|
8-(1-(pyrrolidin-3-yl)-1H-indol-3-ylsulfonyl)quinoline
Show/Hide
|
C21H19N3O2S
|
2
|
| 1 |
IC50 = 82 nM
|
|
|
| 2 |
Ki = 1.5 nM
|
|
|
|
CP0443551
|
N-[3-(benzenesulfonyl)-2-methylsulfanylpyrido[1,2-a]pyrimidin-4-ylidene]acetamide
Show/Hide
|
C17H15N3O3S2
|
1
|
| 1 |
IC50 = 83 nM
|
|
|
|
CP0476067
|
1-(4-Chloro-benzenesulfonyl)-3-(1-methyl-pyrrolidin-3-yl)-1H-indole
Show/Hide
|
C19H19ClN2O2S
|
2
|
| 1 |
IC50 = 85.5 nM
|
|
|
| 2 |
Ki = 1 nM
|
|
|
|
CP0862158
|
N1-(3-(Naphthalen-1-ylsulfonyl)-1H-indazol-6-yl)ethane-1,2-diamine HCl
Show/Hide
|
C19H19ClN4O2S
|
2
|
| 1 |
IC50 = 87 nM
|
|
|
| 2 |
Ki = 17 nM
|
|
|
|
CP0916912
|
3-(Naphthalen-1-ylsulfonyl)-N-(piperidin-4-ylmethyl)-1Hindazol-7-amine HCl
Show/Hide
|
C23H25ClN4O2S
|
2
|
| 1 |
IC50 = 87 nM
|
|
|
| 2 |
Ki = 17 nM
|
|
|
|
CP0919293
|
3-(Naphthalen-1-ylsulfonyl)-N-(piperidin-3-yl)-1H-indazol-4-amine HCl
Show/Hide
|
C22H23ClN4O2S
|
2
|
| 1 |
IC50 = 88 nM
|
|
|
| 2 |
Ki = 4.2 nM
|
|
|
|
CP0073585
|
1-[3-(2-Naphthylsulfonyl)-1H-indazol-5-yl]piperidin-4-amine
Show/Hide
|
C22H22N4O2S
|
1
|
| 1 |
IC50 = 88.9 nM
|
|
|
|
CP0916913
|
N-(3-(Naphthalen-1-ylsulfonyl)-1H-indazol-6-yl)-3-(piperidin-1-yl)propanamide HCl
Show/Hide
|
C25H27ClN4O3S
|
2
|
| 1 |
IC50 = 90 nM
|
|
|
| 2 |
Ki = 12 nM
|
|
|
|
CP0357075
|
3-(2-Chloro-benzenesulfonyl)-1-(1-methyl-pyrrolidin-3-yl)-1H-pyrrolo[2,3-b]pyridine
Show/Hide
|
C18H18ClN3O2S
|
2
|
| 1 |
IC50 = 91 nM
|
|
|
| 2 |
Ki = 2.2 nM
|
|
|
|
CP0878446
|
N,N,N'-Trimethyl-N0-{[3-(1-naphthylsulfonyl)-1H-indazol-5-yl]methyl}ethane-1,2-diamine HCl
Show/Hide
|
C23H27ClN4O2S
|
2
|
| 1 |
IC50 = 91 nM
|
|
|
| 2 |
Ki = 14 nM
|
|
|
|
CP0848236
|
N1-(3-(Naphthalene-1-ylsulfonyl)-1H-indazol-7-yl)ethane-1,2-diamine HCl
Show/Hide
|
C19H19ClN4O2S
|
2
|
| 1 |
IC50 = 93 nM
|
|
|
| 2 |
Ki = 17 nM
|
|
|
|
CP0422111
|
5-fluoro-3-(3-fluorophenylsulfonyl)-1-(1-methylpyrrolidin-3-yl)-1H-indole
Show/Hide
|
C19H18F2N2O2S
|
2
|
| 1 |
IC50 = 94 nM
|
|
|
| 2 |
Ki = 5 nM
|
|
|
|
CP0864884
|
3-(3-Fluorophenylsulfonyl)-N-(piperidin-4-yl)-1H-indazol-5-amine HCl
Show/Hide
|
C18H20ClFN4O2S
|
2
|
| 1 |
IC50 = 94 nM
|
|
|
| 2 |
Ki = 6.7 nM
|
|
|
|
CP0089877
|
3-(4-chloro-benzenesulfonyl)-1-(1-methyl-pyrrolidin-3-yl)-1H-pyrrolo[2,3-b]pyridine
Show/Hide
|
C18H18ClN3O2S
|
2
|
| 1 |
IC50 = 95 nM
|
|
|
| 2 |
Ki = 4.2 nM
|
|
|
|
CP0872983
|
3-(Naphthalen-1-ylsulfonyl)-N-(piperidin-5-yl)-1H-indazol-4-amine HCl
Show/Hide
|
C22H23ClN4O2S
|
2
|
| 1 |
IC50 = 95 nM
|
|
|
| 2 |
Ki = 1.7 nM
|
|
|
|
CP0452536
|
4-(naphthalen-1-ylsulfonyl)-2-(piperazin-1-yl)benzo[d]oxazole
Show/Hide
|
C21H19N3O3S
|
2
|
| 1 |
IC50 = 96 nM
|
|
|
| 2 |
Ki = 3.1 nM
|
|
|
|
CP0485094
|
1-(3-Chloro-benzenesulfonyl)-3-((S)-1-methyl-pyrrolidin-2-ylmethyl)-1H-indole
Show/Hide
|
C20H21ClN2O2S
|
2
|
| 1 |
IC50 = 96.2 nM
|
|
|
| 2 |
Ki = 4 nM
|
|
|
|
CP0476068
|
1-(3,4-Dimethoxy-benzenesulfonyl)-3-(1-methyl-pyrrolidin-3-yl)-1H-indole
Show/Hide
|
C21H24N2O4S
|
2
|
| 1 |
IC50 = 96.7 nM
|
|
|
| 2 |
Ki = 5 nM
|
|
|
|
CP0372406
|
4-(3-methoxyphenylsulfonyl)-2-(piperazin-1-yl)benzo[d]oxazole
Show/Hide
|
C18H19N3O4S
|
2
|
| 1 |
IC50 = 100 nM
|
|
|
| 2 |
Ki = 25 nM
|
|
|
|
CP0505378
|
3-(2-Chlorophenylsulfonyl)-5-(4-methylpiperazin-1-yl)-1H-indazole
Show/Hide
|
C18H19ClN4O2S
|
2
|
| 1 |
IC50 = 101 nM
|
|
|
| 2 |
Ki = 4 nM
|
|
|
|
CP0377003
|
3-(1-methylpiperidin-4-yl)-5-(naphthalen-2-ylsulfonyl)-1H-indazole
Show/Hide
|
C23H23N3O2S
|
2
|
| 1 |
IC50 = 102 nM
|
|
|
| 2 |
Ki = 9.6 nM
|
|
|
|
CP0864883
|
N-[2-(Dimethylamino)ethyl]-3-(1-naphthylsulfonyl)-1Hindazole-5-carboxamide HCl
Show/Hide
|
C22H23ClN4O3S
|
2
|
| 1 |
IC50 = 103 nM
|
|
|
| 2 |
Ki = 2.9 nM
|
|
|
|
CP0916814
|
(S)-3-Methyl-N1-[3-(naphthalen-1-sulfonyl)-1H-indazol-5-yl]-butane-1,2-diamine HCl
Show/Hide
|
C22H25ClN4O2S
|
2
|
| 1 |
IC50 = 103 nM
|
|
|
| 2 |
Ki = 4.3 nM
|
|
|
|
CP0434907
|
2-(4-methylpiperazin-1-yl)-4-(naphthalen-1-ylsulfonyl)benzo[d]oxazole
Show/Hide
|
C22H21N3O3S
|
2
|
| 1 |
IC50 = 105 nM
|
|
|
| 2 |
Ki = 9.7 nM
|
|
|
|
CP0402011
|
3-(naphthalen-1-ylsulfonyl)-1-(pyrrolidin-3-yl)-1H-indole
Show/Hide
|
C22H20N2O2S
|
2
|
| 1 |
IC50 = 107 nM
|
|
|
| 2 |
Ki = 23.3 nM
|
|
|
|
CP0411182
|
1-(1-methylpiperidin-3-yl)-3-(naphthalen-1-ylsulfonyl)-1H-indole
Show/Hide
|
C24H24N2O2S
|
2
|
| 1 |
IC50 = 107 nM
|
|
|
| 2 |
Ki = 7.1 nM
|
|
|
|
CP0453188
|
1-(3,4-Dichloro-benzenesulfonyl)-3-(1-methyl-pyrrolidin-3-yl)-1H-indole
Show/Hide
|
C19H18Cl2N2O2S
|
2
|
| 1 |
IC50 = 107.1 nM
|
|
|
| 2 |
Ki = 3 nM
|
|
|
|
CP0502708
|
3-(4-Chlorophenylsulfonyl)-5-(4-methylpiperazin-1-yl)-1H-indazole
Show/Hide
|
C18H19ClN4O2S
|
2
|
| 1 |
IC50 = 108 nM
|
|
|
| 2 |
Ki = 8.1 nM
|
|
|
|
CP0473616
|
5-(4-isopropylphenylsulfonyl)-3-(1-methylpiperidin-4-yl)-1H-indazole
Show/Hide
|
C22H27N3O2S
|
2
|
| 1 |
IC50 = 108 nM
|
|
|
| 2 |
Ki = 14 nM
|
|
|
|
CP0399781
|
5-[3-(1-Benzyl-pyrrolidin-3-yl)-indole-1-sulfonyl]-4-methyl-thiazol-2-ylamine
Show/Hide
|
C23H24N4O2S2
|
2
|
| 1 |
IC50 = 110 nM
|
|
|
| 2 |
Ki = 3 nM
|
|
|
|
CP0436098
|
3-(1-Benzyl-pyrrolidin-3-yl)-1-(5-bromo-thiophene-2-sulfonyl)-1H-indole
Show/Hide
|
C23H21BrN2O2S2
|
2
|
| 1 |
IC50 = 110 nM
|
|
|
| 2 |
Ki = 9 nM
|
|
|
|
CP0448065
|
1-(5-Bromo-thiophene-2-sulfonyl)-3-((S)-1-methyl-pyrrolidin-2-ylmethyl)-1H-indole
Show/Hide
|
C18H19BrN2O2S2
|
2
|
| 1 |
IC50 = 112 nM
|
|
|
| 2 |
Ki = 3 nM
|
|
|
|
CP0399576
|
5-(4-Methylpiperazin-1-yl)-3-tosyl-1H-indazole
Show/Hide
|
C19H22N4O2S
|
2
|
| 1 |
IC50 = 112 nM
|
|
|
| 2 |
Ki = 4.9 nM
|
|
|
|
CP0524275
|
4-(2,5-dichlorophenylsulfonyl)-2-(piperazin-1-yl)benzo[d]oxazole
Show/Hide
|
C17H15Cl2N3O3S
|
2
|
| 1 |
IC50 = 117 nM
|
|
|
| 2 |
Ki = 13 nM
|
|
|
|
CP0858441
|
3-(4-Fluorophenylsulfonyl)-N-(piperidin-4-yl)-1H-indazol-5-amine HCl
Show/Hide
|
C18H20ClFN4O2S
|
2
|
| 1 |
IC50 = 118 nM
|
|
|
| 2 |
Ki = 6.3 nM
|
|
|
|
CP0372404
|
2-(piperazin-1-yl)-4-(3-(trifluoromethyl)phenylsulfonyl)benzo[d]oxazole
Show/Hide
|
C18H16F3N3O3S
|
2
|
| 1 |
IC50 = 120 nM
|
|
|
| 2 |
Ki = 22 nM
|
|
|
|
CP0093676
|
3-(3-chloro-benzenesulfonyl)-1-(1-ethyl-pyrrolidin-3-yl)-1H-pyrrolo[2,3-b]pyridine
Show/Hide
|
C19H20ClN3O2S
|
2
|
| 1 |
IC50 = 120 nM
|
|
|
| 2 |
Ki = 3.3 nM
|
|
|
|
CP0388192
|
3-(benzenesulfonyl)-N-methyl-2-methylsulfanylpyrido[1,2-a]pyrimidin-4-imine
Show/Hide
|
C16H15N3O2S2
|
1
|
| 1 |
IC50 = 120 nM
|
|
|
|
CP0483732
|
3-(1-Benzyl-pyrrolidin-3-yl)-1-(toluene-4-sulfonyl)-1H-indole
Show/Hide
|
C26H26N2O2S
|
2
|
| 1 |
IC50 = 123 nM
|
|
|
| 2 |
Ki = 8 nM
|
|
|
|
CP0858430
|
3-(Phenylsulfonyl)-N-(piperidin-4-yl)-1H-indazol-5-amine HCl
Show/Hide
|
C18H21ClN4O2S
|
2
|
| 1 |
IC50 = 125 nM
|
|
|
| 2 |
Ki = 3.1 nM
|
|
|
|
CP0860487
|
3-(4-Methoxyphenylsulfonyl)-N-(piperidin-4-yl)-1Hindazol-5-amine HCl
Show/Hide
|
C19H23ClN4O3S
|
2
|
| 1 |
IC50 = 126 nM
|
|
|
| 2 |
Ki = 9.8 nM
|
|
|
|
CP0363770
|
3-Benzenesulfonyl-9-bromo-7-methyl-2-methylsulfanyl-pyrido[1,2-a]pyrimidin-(4Z)-ylideneamine
Show/Hide
|
C16H14BrN3O2S2
|
1
|
| 1 |
IC50 = 126 nM
|
|
|
|
CP0037955
|
METHIOTHEPIN
Show/Hide
|
C20H24N2S2
|
1
|
| 1 |
IC50 = 127 nM
|
|
|
|
CP0113787
|
1-(1-ethyl-pyrrolidin-3-yl)-3-(3-fluoro-benzenesulfonyl)-1H-pyrrolo[2,3-b]pyridine
Show/Hide
|
C19H20FN3O2S
|
2
|
| 1 |
IC50 = 132 nM
|
|
|
| 2 |
Ki = 8.3 nM
|
|
|
|
CP0504425
|
3-(3-Fluorophenylsulfonyl)-5-(4-methylpiperazin-1-yl)-1H-indazole
Show/Hide
|
C18H19FN4O2S
|
2
|
| 1 |
IC50 = 132 nM
|
|
|
| 2 |
Ki = 1.7 nM
|
|
|
|
CP0093693
|
3-(4-bromo-benzenesulfonyl)-1-pyrrolidin-3-yl-1Hpyrrolo[2,3-b]pyridine
Show/Hide
|
C17H16BrN3O2S
|
2
|
| 1 |
IC50 = 135 nM
|
|
|
| 2 |
Ki = 4.3 nM
|
|
|
|
CP0862085
|
3-(Diethylamino)-N-(3-(naphthalen-1-ylsulfonyl)-1Hindazol-7-yl)propanamide HCl
Show/Hide
|
C24H27ClN4O3S
|
2
|
| 1 |
IC50 = 137 nM
|
|
|
| 2 |
Ki = 27 nM
|
|
|
|
CP0288554
|
3-(3-chloro-benzenesulfonyl)-1-(1-methyl-pyrrolidin-3-yl)-1H-pyrrolo[2,3-b]pyridine
Show/Hide
|
C18H18ClN3O2S
|
2
|
| 1 |
IC50 = 142 nM
|
|
|
| 2 |
Ki = 1.5 nM
|
|
|
|
CP0870940
|
N-{[3-(1-Naphthylsulfonyl)-1H-indazol-5yl]methyl}ethane-1,2-diamine HCl
Show/Hide
|
C20H21ClN4O2S
|
2
|
| 1 |
IC50 = 156 nM
|
|
|
| 2 |
Ki = 12 nM
|
|
|
|
CP0229727
|
(3R)-1-[1-(1-Methylethyl)-3-(naphthalen-1-ylsulfonyl)-1H-indazol-5-yl]pyrrolidin-3-amine
Show/Hide
|
C24H26N4O2S
|
1
|
| 1 |
IC50 = 157 nM
|
|
|
|
CP0279371
|
6-(2-methoxyphenylsulfonyl)-1,2,3,4,5,6-hexahydroazepino[4,5-b]indole
Show/Hide
|
C19H20N2O3S
|
2
|
| 1 |
IC50 = 162 nM
|
|
|
| 2 |
Ki = 19 nM
|
|
|
|
CP0430194
|
4-[3-(1,2,3,6-Tetrahydro-pyridin-4-yl)-indole-1-sulfonyl]-isothiazolo[4,5-c]pyridine
Show/Hide
|
C19H16N4O2S2
|
2
|
| 1 |
IC50 = 169 nM
|
|
|
| 2 |
Ki = 5 nM
|
|
|
|
CP0435015
|
1-sulfonylindazole, 6g
Show/Hide
|
C25H26N4O3S
|
2
|
| 1 |
IC50 = 170 nM
|
|
|
| 2 |
Ki = 15 nM
|
|
|
|
CP0899169
|
3-(Naphthalen-1-ylsulfonyl)-N-(piperidin-4-ylmethyl)-1Hindazol-5-amine HCl
Show/Hide
|
C23H25ClN4O2S
|
2
|
| 1 |
IC50 = 174 nM
|
|
|
| 2 |
Ki = 3.5 nM
|
|
|
|
CP0277693
|
3-(2-fluoro-benzenesulfonyl)-1-(1-methyl-pyrrolidin-3-yl)-1H-pyrrolo[2,3-b]pyridine
Show/Hide
|
C18H18FN3O2S
|
2
|
| 1 |
IC50 = 186 nM
|
|
|
| 2 |
Ki = 5.6 nM
|
|
|
|
CP0379952
|
7-(4-methylpiperazin-1-yl)-1-(naphthalen-2-ylsulfonyl)-2,3-dihydroquinolin-4(1H)-one
Show/Hide
|
C24H25N3O3S
|
1
|
| 1 |
IC50 = 188 nM
|
|
|
|
CP0398547
|
2-(3-(3-chlorophenylsulfonyl)-1H-pyrrolo[3,2-b]pyridin-1-yl)ethanamine
Show/Hide
|
C15H14ClN3O2S
|
2
|
| 1 |
IC50 = 197 nM
|
|
|
| 2 |
Ki = 35 nM
|
|
|
|
CP0073491
|
(3R)-1-[1-(2-Methylpropyl)-3-(naphthalen-1-ylsulfonyl)-1Hindazol-5-yl]pyrrolidin-3-amine
Show/Hide
|
C25H28N4O2S
|
1
|
| 1 |
IC50 = 203 nM
|
|
|
|
CP0287843
|
3-(4-fluoro-benzenesulfonyl)-1-(1-methyl-pyrrolidin-3-yl)-1H-pyrrolo[2,3-b]pyridine
Show/Hide
|
C18H18FN3O2S
|
2
|
| 1 |
IC50 = 213 nM
|
|
|
| 2 |
Ki = 5 nM
|
|
|
|
CP0434906
|
2-(4-ethylpiperazin-1-yl)-4-(naphthalen-1-ylsulfonyl)benzo[d]oxazole
Show/Hide
|
C23H23N3O3S
|
2
|
| 1 |
IC50 = 248 nM
|
|
|
| 2 |
Ki = 12 nM
|
|
|
|
CP0443190
|
3-(benzenesulfonyl)-2-methylsulfinylpyrido[1,2-a]pyrimidin-4-imine
Show/Hide
|
C15H13N3O3S2
|
1
|
| 1 |
IC50 = 250 nM
|
|
|
|
CP0455014
|
3-(1-methylpiperidin-4-yl)-5-(naphthalen-1-ylsulfonyl)-1H-indazole
Show/Hide
|
C23H23N3O2S
|
2
|
| 1 |
IC50 = 251 nM
|
|
|
| 2 |
Ki = 3.8 nM
|
|
|
|
CP0493125
|
1-sulfonylindazole, 6f
Show/Hide
|
C24H26N4O3S
|
2
|
| 1 |
IC50 = 260 nM
|
|
|
| 2 |
Ki = 2.1 nM
|
|
|
|
CP0414986
|
1-(1-(2-(dimethylamino)ethyl)-3-(naphthalen-1-ylsulfonyl)-1H-pyrrolo[3,2-b]pyridin-5-yl)ethanone
Show/Hide
|
C23H23N3O3S
|
2
|
| 1 |
IC50 = 295 nM
|
|
|
| 2 |
Ki = 1.7 nM
|
|
|
|
CP0087496
|
N-[7-oxo-6-(piperidin-4-ylmethyl)-4,5-dihydro-1H-pyrazolo[3,4-c]pyridin-3-yl]naphthalene-1-sulfonamide
Show/Hide
|
C22H25N5O3S
|
1
|
| 1 |
IC50 = 310 nM
|
|
|
|
CP0364728
|
N-[7-oxo-6-(piperidin-4-ylmethyl)-4,5-dihydro-1H-pyrazolo[3,4-c]pyridin-3-yl]naphthalene-2-sulfonamide
Show/Hide
|
C22H25N5O3S
|
1
|
| 1 |
IC50 = 310 nM
|
|
|
|
CP0148894
|
(3R)-1-[1-Methyl-3-(naphthalen-1-ylsulfonyl)-1H-indazol-5-yl]pyrrolidin-3-amine
Show/Hide
|
C22H22N4O2S
|
1
|
| 1 |
IC50 = 316 nM
|
|
|
|
CP0487047
|
3-(benzenesulfonyl)-9-benzyl-2-methylsulfanylpyrido[1,2-a]pyrimidin-4-imine
Show/Hide
|
C22H19N3O2S2
|
1
|
| 1 |
IC50 = 330 nM
|
|
|
|
CP0399577
|
5-(4-Methylpiperazin-1-yl)-3-(thiophen-2-ylsulfonyl)-1H-indazole
Show/Hide
|
C16H18N4O2S2
|
2
|
| 1 |
IC50 = 331 nM
|
|
|
| 2 |
Ki = 7.8 nM
|
|
|
|
CP0143098
|
3-[(4-chlorophenyl)sulfonyl]-1-(1-isopropylpiperidin-3-yl)-1H-pyrrolo[2,3-b]pyridine
Show/Hide
|
C21H24ClN3O2S
|
2
|
| 1 |
IC50 = 338 nM
|
|
|
| 2 |
Ki = 11.1 nM
|
|
|
|
CP0325788
|
3-(4-chloro-benzenesulfonyl)-1-pyrrolidin-3-yl-1Hpyrrolo[2,3-b]pyridine
Show/Hide
|
C17H16ClN3O2S
|
2
|
| 1 |
IC50 = 340 nM
|
|
|
| 2 |
Ki = 5.5 nM
|
|
|
|
CP0469508
|
N-methyl-2-(3-naphthalen-1-ylsulfonylindol-1-yl)ethanamine
Show/Hide
|
C21H20N2O2S
|
2
|
| 1 |
IC50 = 359 nM
|
|
|
| 2 |
Ki = 5.7 nM
|
|
|
|
CP0043596
|
(3R)-1-[2-(1-Methylethyl)-3-(naphthalen-1-ylsulfonyl)-2Hindazol-5-yl]pyrrolidin-3-amine
Show/Hide
|
C24H26N4O2S
|
1
|
| 1 |
IC50 = 380 nM
|
|
|
|
CP0405509
|
1-(3-(4-bromophenylsulfonyl)-1-(2-(dimethylamino)ethyl)-1H-pyrrolo[3,2-b]pyridin-5-yl)ethanone
Show/Hide
|
C19H20BrN3O3S
|
2
|
| 1 |
IC50 = 385 nM
|
|
|
| 2 |
Ki = 3.9 nM
|
|
|
|
CP0415730
|
2-methylsulfanyl-3-[4-(trifluoromethoxy)phenyl]sulfonylpyrido[1,2-a]pyrimidin-4-imine
Show/Hide
|
C16H12F3N3O3S2
|
1
|
| 1 |
IC50 = 420 nM
|
|
|
|
CP0208161
|
(3R)-1-[2-(2-Methylpropyl)-3-(naphthalen-1-ylsulfonyl)-2Hindazol-5-yl]pyrrolidin-3-amine
Show/Hide
|
C25H28N4O2S
|
1
|
| 1 |
IC50 = 433 nM
|
|
|
|
CP0330836
|
(3R)-1-[2-Methyl-3-(naphthalen-1-ylsulfonyl)-2H-indazol-5-yl]pyrrolidin-3-amine
Show/Hide
|
C22H22N4O2S
|
1
|
| 1 |
IC50 = 444 nM
|
|
|
|
CP0864882
|
3-Amino-N-(3-(naphthalen-1-ylsulfonyl)-1H-indazol-6-yl)propanamide HCl
Show/Hide
|
C20H19ClN4O3S
|
2
|
| 1 |
IC50 = 456 nM
|
|
|
| 2 |
Ki = 24 nM
|
|
|
|
CP0511778
|
3-(4-Fluorophenylsulfonyl)-5-(4-methylpiperazin-1-yl)-1H-indazole
Show/Hide
|
C18H19FN4O2S
|
2
|
| 1 |
IC50 = 467 nM
|
|
|
| 2 |
Ki = 5.2 nM
|
|
|
|
CP0388191
|
methyl 3-(benzenesulfonyl)-4-imino-2-methylsulfanylpyrido[1,2-a]pyrimidine-7-carboxylate
Show/Hide
|
C17H15N3O4S2
|
1
|
| 1 |
IC50 = 470 nM
|
|
|
|
CP0104220
|
3-[(3-bromophenyl)sulfonyl]-1-(1-isopropylpiperidin-3-yl)-1H-pyrrolo[2,3-b]pyridine
Show/Hide
|
C21H24BrN3O2S
|
2
|
| 1 |
IC50 = 492 nM
|
|
|
| 2 |
Ki = 9.4 nM
|
|
|
|
CP0403554
|
3-(4-Methoxyphenylsulfonyl)-5-(4-methylpiperazin-1-yl)-1Hindazole
Show/Hide
|
C19H22N4O3S
|
2
|
| 1 |
IC50 = 544 nM
|
|
|
| 2 |
Ki = 12 nM
|
|
|
|
CP0087495
|
3-fluoro-N-[6-(4-methoxyphenyl)-7-oxo-4,5-dihydro-1H-pyrazolo[3,4-c]pyridin-3-yl]benzenesulfonamide
Show/Hide
|
C19H17FN4O4S
|
1
|
| 1 |
IC50 = 580 nM
|
|
|
|
CP0176560
|
5,7-dichloro-3-(4-hydroxyphenyl)-3-methylquinoline-2,4(1H,3H)-dione
Show/Hide
|
C16H11Cl2NO3
|
1
|
| 1 |
IC50 = 615 nM
|
|
|
|
CP0269589
|
8-(1-pyrrolidin-3-yl-1H-pyrrolo[2,3-b]pyridine-3-sulfonyl)-quinoline
Show/Hide
|
C20H18N4O2S
|
2
|
| 1 |
IC50 = 643 nM
|
|
|
| 2 |
Ki = 5.7 nM
|
|
|
|
CP0271607
|
3-[(4-chlorophenyl)sulfonyl]-1-piperidin-3-yl-1Hpyrrolo[2,3-b]pyridine
Show/Hide
|
C18H18ClN3O2S
|
2
|
| 1 |
IC50 = 682 nM
|
|
|
| 2 |
Ki = 7.6 nM
|
|
|
|
CP0434471
|
3-(benzenesulfonyl)-2-methylsulfanyl-8-propylpyrido[1,2-a]pyrimidin-4-imine
Show/Hide
|
C18H19N3O2S2
|
1
|
| 1 |
IC50 = 700 nM
|
|
|
|
CP0380698
|
5-(3-chlorophenylsulfonyl)-3-(1-methylpiperidin-4-yl)-1H-indazole
Show/Hide
|
C19H20ClN3O2S
|
2
|
| 1 |
IC50 = 754 nM
|
|
|
| 2 |
Ki = 19 nM
|
|
|
|
CP0373060
|
N-[3-[4-(3,4-dichlorophenyl)piperazin-1-yl]propyl]naphthalene-2-sulfonamide
Show/Hide
|
C23H25Cl2N3O2S
|
1
|
| 1 |
IC50 = 768 nM
|
|
|
|
CP0087497
|
N-(7-oxo-6-piperidin-4-yl-4,5-dihydro-1H-pyrazolo[3,4-c]pyridin-3-yl)naphthalene-1-sulfonamide
Show/Hide
|
C21H23N5O3S
|
1
|
| 1 |
IC50 = 770 nM
|
|
|
|
CP0484146
|
N,N-dimethyl-2-[3-[2-(trifluoromethoxy)phenyl]sulfonylindol-1-yl]ethanamine
Show/Hide
|
C19H19F3N2O3S
|
2
|
| 1 |
IC50 = 792 nM
|
|
|
| 2 |
Ki = 16 nM
|
|
|
|
CP0405511
|
2-(3-(3-fluorophenylsulfonyl)-1H-pyrrolo[3,2-b]pyridin-1-yl)ethanamine
Show/Hide
|
C15H14FN3O2S
|
2
|
| 1 |
IC50 = 823 nM
|
|
|
| 2 |
Ki = 76 nM
|
|
|
|
CP0409004
|
N-[[5-(2-methylpropyl)-1-phenylpyrazol-3-yl]methyl]quinoline-8-sulfonamide
Show/Hide
|
C23H24N4O2S
|
1
|
| 1 |
IC50 = 1420 nM
|
|
|
|
CP0538002
|
3-chloro-2-methyl-N-[6-(4-methylphenyl)-7-oxo-4,5-dihydro-1H-pyrazolo[3,4-c]pyridin-3-yl]benzenesulfonamide
Show/Hide
|
C20H19ClN4O3S
|
1
|
| 1 |
IC50 = 1660 nM
|
|
|
|
CP0419804
|
N-[[1-(4-fluorophenyl)-5-(2-methylpropyl)pyrazol-3-yl]methyl]quinoline-8-sulfonamide
Show/Hide
|
C23H23FN4O2S
|
1
|
| 1 |
IC50 = 1780 nM
|
|
|
|
CP0419082
|
N-[3-[4-[3-(trifluoromethyl)phenyl]piperazin-1-yl]propyl]naphthalene-2-sulfonamide
Show/Hide
|
C24H26F3N3O2S
|
1
|
| 1 |
IC50 = 1956 nM
|
|
|
|
CP0132624
|
N-[[5-(2-methylpropyl)-1-phenylpyrazol-3-yl]methyl]naphthalene-1-sulfonamide
Show/Hide
|
C24H25N3O2S
|
1
|
| 1 |
IC50 = 2430 nM
|
|
|
|
CP0259093
|
N-[3-[4-(2-methoxyphenyl)piperazin-1-yl]propyl]naphthalene-2-sulfonamide
Show/Hide
|
C24H29N3O3S
|
1
|
| 1 |
IC50 = 2634 nM
|
|
|
|
CP0419080
|
4-Methoxy-N-{3-[4-(m-trifluoromethylphenyl)-piperazin-1-yl]-propyl}-benzenesulfonamide
Show/Hide
|
C21H26F3N3O3S
|
1
|
| 1 |
IC50 = 2839 nM
|
|
|
|
CP0397391
|
N-[6-(4-methylphenyl)-7-oxo-4,5-dihydro-1H-pyrazolo[3,4-c]pyridin-3-yl]-3-(trifluoromethyl)benzenesulfonamide
Show/Hide
|
C20H17F3N4O3S
|
1
|
| 1 |
IC50 = 3280 nM
|
|
|
|
CP0238043
|
N-[[5-(2-methylpropyl)-1-phenylpyrazol-3-yl]methyl]naphthalene-2-sulfonamide
Show/Hide
|
C24H25N3O2S
|
1
|
| 1 |
IC50 = 3300 nM
|
|
|
|
CP0247429
|
3-chloro-2-methyl-N-[[5-(2-methylpropyl)-1-phenylpyrazol-3-yl]methyl]benzenesulfonamide
Show/Hide
|
C21H24ClN3O2S
|
1
|
| 1 |
IC50 = 4010 nM
|
|
|
|
CP0540585
|
4-fluoro-N-[6-(4-methylphenyl)-7-oxo-4,5-dihydro-1H-pyrazolo[3,4-c]pyridin-3-yl]benzenesulfonamide
Show/Hide
|
C19H17FN4O3S
|
1
|
| 1 |
IC50 = 5220 nM
|
|
|
|
CP0464391
|
2,6-dichloro-N-[[5-(2-methylpropyl)-1-phenylpyrazol-3-yl]methyl]benzenesulfonamide
Show/Hide
|
C20H21Cl2N3O2S
|
1
|
| 1 |
IC50 = 5650 nM
|
|
|
|
CP0397433
|
3-methoxy-N-[6-(4-methylphenyl)-7-oxo-4,5-dihydro-1H-pyrazolo[3,4-c]pyridin-3-yl]benzenesulfonamide
Show/Hide
|
C20H20N4O4S
|
1
|
| 1 |
IC50 = 6770 nM
|
|
|
|
CP0459682
|
4-Methoxy-N-{3-[4-(m-trifluoromethylphenyl)-piperazin-1-yl]-1-methyl-propyl}-benzenesulfonamide
Show/Hide
|
C22H28F3N3O3S
|
1
|
| 1 |
IC50 = 6925 nM
|
|
|
|
CP0446773
|
3-methoxy-N-[6-(4-methoxyphenyl)-7-oxo-4,5-dihydro-1H-pyrazolo[3,4-c]pyridin-3-yl]benzenesulfonamide
Show/Hide
|
C20H20N4O5S
|
1
|
| 1 |
IC50 = 7080 nM
|
|
|
|
CP0419803
|
4-tert-butyl-N-[[5-(2-methylpropyl)-1-phenylpyrazol-3-yl]methyl]benzenesulfonamide
Show/Hide
|
C24H31N3O2S
|
1
|
| 1 |
IC50 = 8780 nM
|
|
|
|
CP0233824
|
4-Methoxy-N-{3-[4-(2-methoxy-phenyl)-piperazin-1-yl]-propyl}-benzenesulfonamide
Show/Hide
|
C21H29N3O4S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0501817
|
4-Methoxy-N-{3-[4-(p-fluorophenyl)-piperazin-1-yl]-propyl}-benzenesulfonamide
Show/Hide
|
C20H26FN3O3S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0476259
|
3-chloro-N-[[5-(2-methylpropyl)-1-phenylpyrazol-3-yl]methyl]benzenesulfonamide
Show/Hide
|
C20H22ClN3O2S
|
1
|
| 1 |
IC50 = 10900 nM
|
|
|
|
CP0506507
|
10-(benzenesulfonyl)-N-methyl-1,8,12-triazatricyclo[7.3.0.02,6]dodeca-2(6),7,9,11-tetraen-11-amine
Show/Hide
|
C16H16N4O2S
|
1
|
| 1 |
Ki = 0.088 nM
|
|
|
|
CP0438807
|
3-(benzenesulfonyl)-N-methyl-6,7,8,9-tetrahydropyrazolo[1,5-a]quinazolin-2-amine
Show/Hide
|
C17H18N4O2S
|
1
|
| 1 |
Ki = 0.112 nM
|
|
|
|
CP0370584
|
4-(2-bromo-6-piperazin-1-ylpyridin-4-yl)sulfonylaniline
Show/Hide
|
C15H17BrN4O2S
|
1
|
| 1 |
Ki = 0.1148 nM
|
|
|
|
CP0374246
|
10-(benzenesulfonyl)-N,7-dimethyl-1,8,12-triazatricyclo[7.3.0.02,6]dodeca-2(6),7,9,11-tetraen-11-amine
Show/Hide
|
C17H18N4O2S
|
1
|
| 1 |
Ki = 0.202 nM
|
|
|
|
CP0515952
|
1-(3-chlorophenyl)sulfonyl-4-piperazin-1-ylindole
Show/Hide
|
C18H18ClN3O2S
|
1
|
| 1 |
Ki = 0.2512 nM
|
|
|
|
CP0446623
|
3-(benzenesulfonyl)-N,9-dimethyl-5,6,7,8-tetrahydropyrazolo[5,1-b]quinazolin-2-amine
Show/Hide
|
C18H20N4O2S
|
1
|
| 1 |
Ki = 0.256 nM
|
|
|
|
CP0144979
|
1-(phenylsulfonyl)-4-(piperazin-1-yl)-1H-indole
Show/Hide
|
C18H19N3O2S
|
1
|
| 1 |
Ki = 0.3162 nM
|
|
|
|
CP0485606
|
3-(3-chlorophenyl)sulfonyl-7-piperazin-1-yl-1H-indole
Show/Hide
|
C18H18ClN3O2S
|
1
|
| 1 |
Ki = 0.3162 nM
|
|
|
|
CP0541698
|
3-chloro-1-(3-chlorophenyl)sulfonyl-4-piperazin-1-ylindole
Show/Hide
|
C18H17Cl2N3O2S
|
1
|
| 1 |
Ki = 0.3162 nM
|
|
|
|
CP0541703
|
7-chloro-1-(3-chlorophenyl)sulfonyl-4-piperazin-1-ylindole
Show/Hide
|
C18H17Cl2N3O2S
|
1
|
| 1 |
Ki = 0.3162 nM
|
|
|
|
CP0175237
|
5-(benzenesulfonyl)-N,11-dimethyl-2,3,7,11-tetrazatricyclo[7.4.0.02,6]trideca-1(9),3,5,7-tetraen-4-amine
Show/Hide
|
C17H19N5O2S
|
1
|
| 1 |
Ki = 0.39 nM
|
|
|
|
CP0485577
|
1-(3-chlorophenyl)sulfonyl-2-methyl-4-piperazin-1-ylindole
Show/Hide
|
C19H20ClN3O2S
|
1
|
| 1 |
Ki = 0.3981 nM
|
|
|
|
CP0541577
|
1-(2-chlorophenyl)sulfonyl-4-piperazin-1-ylindole
Show/Hide
|
C18H18ClN3O2S
|
1
|
| 1 |
Ki = 0.3981 nM
|
|
|
|
CP0485300
|
5-methyl-2-(methylthio)-3-(phenylsulfonyl)-6,7,8,9-tetrahydropyrazolo[1,5-a]quinazoline
Show/Hide
|
C18H19N3O2S2
|
1
|
| 1 |
Ki = 0.44 nM
|
|
|
|
CP0485301
|
2-(methylthio)-3-(phenylsulfonyl)-7,8-dihydro-6H-cyclopenta[e]pyrazolo[1,5-a]pyrimidine
Show/Hide
|
C16H15N3O2S2
|
1
|
| 1 |
Ki = 0.458 nM
|
|
|
|
CP0508300
|
3-(benzenesulfonyl)-N,5-dimethyl-6,7,8,9-tetrahydropyrazolo[1,5-a]quinazolin-2-amine
Show/Hide
|
C18H20N4O2S
|
1
|
| 1 |
Ki = 0.49 nM
|
|
|
|
CP0430801
|
3-(benzenesulfonyl)-N-methyl-5,6,7,8-tetrahydropyrazolo[5,1-b]quinazolin-2-amine
Show/Hide
|
C17H18N4O2S
|
1
|
| 1 |
Ki = 0.499 nM
|
|
|
|
CP0398424
|
1-sulfonylindazole, 6c
Show/Hide
|
C20H18N4O3S
|
1
|
| 1 |
Ki = 0.5 nM
|
|
|
|
CP0339112
|
4-phenyl-N-(4-piperazin-1-ylquinolin-6-yl)benzenesulfonamide
Show/Hide
|
C25H24N4O2S
|
1
|
| 1 |
Ki = 0.5012 nM
|
|
|
|
CP0452979
|
1-[3-(benzenesulfonyl)-1-benzothiophen-7-yl]piperazine
Show/Hide
|
C18H18N2O2S2
|
1
|
| 1 |
Ki = 0.5012 nM
|
|
|
|
CP0527897
|
5-chloro-4-piperazin-1-yl-1-pyridin-2-ylsulfonylindole
Show/Hide
|
C17H17ClN4O2S
|
1
|
| 1 |
Ki = 0.5012 nM
|
|
|
|
CP0406285
|
2-(methylthio)-3-(phenylsulfonyl)-6,7,8,9-tetrahydropyrazolo[1,5-a]quinazoline
Show/Hide
|
C17H17N3O2S2
|
1
|
| 1 |
Ki = 0.549 nM
|
|
|
|
CP0150364
|
2,8-Dimethyl-5-((Z)-styryl)-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
Show/Hide
|
C21H22N2
|
1
|
| 1 |
Ki = 0.6166 nM
|
|
|
|
CP0113176
|
5-Chloro-3-methyl-benzo[b]thiophene-2-sulfonic acid [4-methoxy-3-(4-methyl-piperazin-1-yl)-phenyl]-amide
Show/Hide
|
C21H24ClN3O3S2
|
1
|
| 1 |
Ki = 0.631 nM
|
|
|
|
CP0081712
|
4-tert-butyl-N-(4-piperazin-1-ylquinolin-6-yl)benzenesulfonamide
Show/Hide
|
C23H28N4O2S
|
1
|
| 1 |
Ki = 0.631 nM
|
|
|
|
CP0483556
|
1-(3-chlorophenyl)sulfonyl-3-methyl-4-piperazin-1-ylindole
Show/Hide
|
C19H20ClN3O2S
|
1
|
| 1 |
Ki = 0.631 nM
|
|
|
|
CP0041243
|
5-chloro-N-[4-methoxy-3-(piperazin-1-yl)phenyl]-3-methyl-1-benzothiophene-2-sulfonamide hydrochloride
Show/Hide
|
C20H22ClN3O3S2
|
3
|
| 1 |
Ki = 0.631 nM
|
|
|
| 2 |
Ki = 1.259 nM
|
|
|
| 3 |
Ki = 1.3 nM
|
|
|
|
CP0226262
|
4-(benzenesulfonyl)-N,8,11-trimethyl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1,3,5,8-tetraen-5-amine
Show/Hide
|
C18H21N5O2S
|
1
|
| 1 |
Ki = 0.66 nM
|
|
|
|
CP0294753
|
9-methyl-2-(methylthio)-3-(phenylsulfonyl)-5,6,7,8-tetrahydropyrazolo[5,1-b]quinazoline
Show/Hide
|
C18H19N3O2S2
|
1
|
| 1 |
Ki = 0.68 nM
|
|
|
|
CP0329025
|
5-(benzenesulfonyl)-N,8,11-trimethyl-2,3,7,11-tetrazatricyclo[7.4.0.02,6]trideca-1(9),3,5,7-tetraen-4-amine
Show/Hide
|
C18H21N5O2S
|
1
|
| 1 |
Ki = 0.68 nM
|
|
|
|
CP0199114
|
SB-399885
Show/Hide
|
C18H21Cl2N3O4S
|
1
|
| 1 |
Ki = 0.7244 nM
|
|
|
|
CP0894752
|
3-Iodo-N-[4-methoxy-3-(4-methyl-piperazin-1-yl)-phenyl]-benzenesulfonamide
Show/Hide
|
C18H22IN3O3S
|
1
|
| 1 |
Ki = 0.7943 nM
|
|
|
|
CP0911387
|
5-Chloro-naphthalene-2-sulfonic acid [4-methoxy-3-(4-methyl-piperazin-1-yl)-phenyl]-amide
Show/Hide
|
C22H24ClN3O3S
|
1
|
| 1 |
Ki = 0.7943 nM
|
|
|
|
CP0165719
|
N-[3-[(8aR)-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]-4-methoxyphenyl]-5-chloro-3-methyl-1-benzothiophene-2-sulfonamide
Show/Hide
|
C23H26ClN3O3S2
|
1
|
| 1 |
Ki = 0.7943 nM
|
|
|
|
CP0183577
|
5-Chloro-3-methyl-benzo[b]thiophene-2-sulfonic acid ((S)-3-hexahydro-pyrrolo[1,2-a]pyrazin-2-yl-4-methoxy-phenyl)-amide
Show/Hide
|
C23H26ClN3O3S2
|
1
|
| 1 |
Ki = 0.7943 nM
|
|
|
|
CP0016259
|
4-(benzenesulfonyl)-N,11-dimethyl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1,3,5,8-tetraen-5-amine
Show/Hide
|
C17H19N5O2S
|
1
|
| 1 |
Ki = 0.82 nM
|
|
|
|
CP0860241
|
5-Iodo-N-[4-methoxy-3-(4-methyl-piperazin-1-yl)-phenyl]-2-methyl-benzenesulfonamide
Show/Hide
|
C19H24IN3O3S
|
1
|
| 1 |
Ki = 1 nM
|
|
|
|
CP0111551
|
5-chloro-N-(4-piperazin-1-ylquinolin-6-yl)naphthalene-2-sulfonamide
Show/Hide
|
C23H21ClN4O2S
|
1
|
| 1 |
Ki = 1 nM
|
|
|
|
CP0208303
|
5-chloro-2-methyl-N-(4-piperazin-1-ylquinolin-6-yl)-1-benzothiophene-3-sulfonamide
Show/Hide
|
C22H21ClN4O2S2
|
1
|
| 1 |
Ki = 1 nM
|
|
|
|
CP0306083
|
5-chloro-3-methyl-N-[4-(4-methylpiperazin-1-yl)quinolin-6-yl]-1-benzothiophene-2-sulfonamide
Show/Hide
|
C23H23ClN4O2S2
|
1
|
| 1 |
Ki = 1 nM
|
|
|
|
CP0370117
|
4-(2-Bromo-6-pyrrolidin-1-yl-pyridine-4-sulfonyl)-phenylamine
Show/Hide
|
C15H16BrN3O2S
|
1
|
| 1 |
Ki = 1 nM
|
|
|
|
CP0860575
|
N-[3-((R)-1-Methyl-pyrrolidin-2-ylmethyl)-1H-indol-5-yl]-benzenesulfonamide
Show/Hide
|
C20H23N3O2S
|
1
|
| 1 |
Ki = 1 nM
|
|
|
|
CP0889329
|
4-Iodo-N-(3-(R)-1-pyrrolidin-2-ylmethyl-1H-indol-5-yl)-benzenesulfonamide
Show/Hide
|
C19H20IN3O2S
|
1
|
| 1 |
Ki = 1 nM
|
|
|
|
CP0911038
|
4-Isopropyl-N-[3-((R)-1-methyl-pyrrolidin-2-ylmethyl)-1H-indol-5-yl]-benzenesulfonamide
Show/Hide
|
C23H29N3O2S
|
1
|
| 1 |
Ki = 1 nM
|
|
|
|
CP0914848
|
3,4-Dichloro-N-[3-((R)-1-methyl-pyrrolidin-2-ylmethyl)-1H-indol-5-yl]-benzenesulfonamide
Show/Hide
|
C20H21Cl2N3O2S
|
1
|
| 1 |
Ki = 1 nM
|
|
|
|
CP0936954
|
Naphthalene-2-sulfonic acid [3-((R)-1-methyl-pyrrolidin-2-ylmethyl)-1H-indol-5-yl]-amide
Show/Hide
|
C24H25N3O2S
|
1
|
| 1 |
Ki = 1 nM
|
|
|
|
CP0957083
|
4-Isopropyl-N-(3-(R)-1-pyrrolidin-2-ylmethyl-1H-indol-5-yl)-benzenesulfonamide
Show/Hide
|
C22H27N3O2S
|
1
|
| 1 |
Ki = 1 nM
|
|
|
|
CP0441845
|
5-chloro-1-(2-chlorophenyl)sulfonyl-4-piperazin-1-ylindole
Show/Hide
|
C18H17Cl2N3O2S
|
1
|
| 1 |
Ki = 1 nM
|
|
|
|
CP0541578
|
4-piperazin-1-yl-1-pyridin-2-ylsulfonylindole
Show/Hide
|
C17H18N4O2S
|
1
|
| 1 |
Ki = 1 nM
|
|
|
|
CP0888590
|
2-(1-(5-(4-methoxyphenylsulfonamido)-1H-indol-3-yl)ethylidene)hydrazinecarboximidamide
Show/Hide
|
C18H20N6O3S
|
1
|
| 1 |
Ki = 1 nM
|
|
|
|
CP0911118
|
2-(1-(5-(phenylsulfonamido)-1H-indol-3-yl)ethylidene)hydrazinecarboximidamide
Show/Hide
|
C17H18N6O2S
|
1
|
| 1 |
Ki = 1 nM
|
|
|
|
CP0449695
|
3-(benzenesulfonyl)-N,N-dimethyl-6,7,8,9-tetrahydrobenzo[e]indol-8-amine
Show/Hide
|
C20H22N2O2S
|
1
|
| 1 |
Ki = 1 nM
|
|
|
|
CP0674190
|
5-Chloro-3-methyl-benzo[b]thiophene-2-sulfonic acid (4-methoxy-3-piperazin-1-yl-phenyl)-amide hydrochloride
Show/Hide
|
C20H23Cl2N3O3S2
|
1
|
| 1 |
Ki = 1.259 nM
|
|
|
|
CP0894716
|
5-Chloro-2-methyl-benzo[b]thiophene-3-sulfonic acid [4-methoxy-3-(4-methyl-piperazin-1-yl)-phenyl]-amide
Show/Hide
|
C21H24ClN3O3S2
|
1
|
| 1 |
Ki = 1.259 nM
|
|
|
|
CP0082421
|
5-chloro-3-methyl-N-(2-methyl-4-piperazin-1-ylquinolin-6-yl)-1-benzothiophene-2-sulfonamide
Show/Hide
|
C23H23ClN4O2S2
|
1
|
| 1 |
Ki = 1.259 nM
|
|
|
|
CP0170807
|
5-chloro-3-ethyl-N-(4-piperazin-1-ylquinolin-6-yl)-1-benzothiophene-2-sulfonamide
Show/Hide
|
C23H23ClN4O2S2
|
1
|
| 1 |
Ki = 1.259 nM
|
|
|
|
CP0343547
|
5-chloro-3-methyl-N-[4-[(3S)-3-methylpiperazin-1-yl]quinolin-6-yl]-1-benzothiophene-2-sulfonamide
Show/Hide
|
C23H23ClN4O2S2
|
1
|
| 1 |
Ki = 1.259 nM
|
|
|
|
CP0436209
|
1-[3-(benzenesulfonyl)-1-benzofuran-7-yl]piperazine
Show/Hide
|
C18H18N2O3S
|
1
|
| 1 |
Ki = 1.259 nM
|
|
|
|
CP0138731
|
1-(3-chlorophenylsulfonyl)-7-methyl-1,5,6,7,8,9-hexahydroazepino[4,5-f]indole
Show/Hide
|
C19H19ClN2O2S
|
1
|
| 1 |
Ki = 1.259 nM
|
|
|
|
CP0286684
|
(2-{2-[3-(3-Methoxy-benzyl)-[1,2,4]oxadiazol-5-yl]-1H-indol-3-yl}-ethyl)-dimethyl-amine
Show/Hide
|
C22H24N4O2
|
1
|
| 1 |
Ki = 1.3 nM
|
|
|
|
CP0330654
|
2-[1-(benzenesulfonyl)indol-4-yl]-N,N-dimethylethanamine
Show/Hide
|
C18H20N2O2S
|
1
|
| 1 |
Ki = 1.5 nM
|
|
|
|
CP0515649
|
(1-Benzenesulfonyl-5-methoxy-1H-indol-3-ylmethyl)-dimethyl-amine
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C18H20N2O3S
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1
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| 1 |
Ki = 1.5 nM
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CP0393159
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1-(benzenesulfonyl)-5-chloro-4-piperazin-1-ylindole
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C18H18ClN3O2S
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1
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| 1 |
Ki = 1.585 nM
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CP0158281
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1-(phenylsulfonyl)-1,5,6,7,8,9-hexahydroazepino[4,5-f]indole
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C18H18N2O2S
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1
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| 1 |
Ki = 1.585 nM
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CP0279822
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1-(3-chlorophenylsulfonyl)-1,5,6,7,8,9-hexahydroazepino[4,5-f]indole
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C18H17ClN2O2S
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1
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| 1 |
Ki = 1.585 nM
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CP0931217
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3,5-Dichloro-N-[4-methoxy-3-(4-methyl-piperazin-1-yl)-phenyl]-benzenesulfonamide
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C18H21Cl2N3O3S
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1
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| 1 |
Ki = 1.995 nM
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CP0173778
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5-chloro-3-methyl-N-(4-piperazin-1-ylquinolin-6-yl)-1-benzothiophene-2-sulfonamide
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C22H21ClN4O2S2
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1
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| 1 |
Ki = 1.995 nM
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CP0467170
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1-(4-chlorophenyl)sulfonyl-4-piperazin-1-ylindole
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C18H18ClN3O2S
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1
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| 1 |
Ki = 1.995 nM
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CP0158282
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1-methyl-3-(phenylsulfonyl)-1,5,6,7,8,9-hexahydroazepino[4,5-f]indole
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C19H20N2O2S
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1
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| 1 |
Ki = 1.995 nM
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CP0254730
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1-(3-methoxyphenylsulfonyl)-1,5,6,7,8,9-hexahydroazepino[4,5-f]indole
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C19H20N2O3S
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1
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| 1 |
Ki = 1.995 nM
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CP0237538
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2,8-Dimethyl-5-phenethyl-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
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C21H24N2
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1
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| 1 |
Ki = 1.995 nM
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CP0419508
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1-(3-Chloro-benzenesulfonyl)-3-piperidin-3-yl-1H-indole
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C19H19ClN2O2S
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1
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| 1 |
Ki = 2 nM
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CP0415376
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4-(4-aminophenyl)sulfonyl-6-bromo-N-methylpyridin-2-amine
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C12H12BrN3O2S
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1
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| 1 |
Ki = 2.291 nM
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CP0045069
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2-[1-(benzenesulfonyl)-5-methoxyindol-3-yl]-N,N-dimethylethanamine
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C19H22N2O3S
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1
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| 1 |
Ki = 2.3 nM
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CP0353494
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2,8-Dimethyl-5-(2-p-tolylethyl)-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
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C22H26N2
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1
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| 1 |
Ki = 2.399 nM
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CP0379189
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2-(1-Benzenesulfonyl-1H-indol-4-yl)-ethylamine
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C16H16N2O2S
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1
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| 1 |
Ki = 2.4 nM
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CP0436431
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1-Benzenesulfonyl-5-fluoro-3-(1,2,3,6-tetrahydro-pyridin-4-yl)-1H-indole
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C19H17FN2O2S
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1
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| 1 |
Ki = 2.4 nM
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CP0481923
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5-chloro-1-(3-chlorophenyl)sulfonyl-4-piperazin-1-ylindole
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C18H17Cl2N3O2S
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1
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| 1 |
Ki = 2.512 nM
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CP0486685
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3-(3-chlorophenyl)sulfonyl-1-methyl-7-piperazin-1-ylindole
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C19H20ClN3O2S
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1
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| 1 |
Ki = 2.512 nM
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CP0170546
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3-chloro-1-(phenylsulfonyl)-1,5,6,7,8,9-hexahydroazepino[4,5-f]indole
Show/Hide
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C18H17ClN2O2S
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1
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| 1 |
Ki = 2.512 nM
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CP0255950
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2-[1-(benzenesulfonyl)indol-3-yl]-N,N-dimethylethanamine
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C18H20N2O2S
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1
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| 1 |
Ki = 2.9 nM
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CP0418991
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[1-(benzenesulfonyl)-4-[2-(dimethylamino)ethyl]indol-2-yl]-phenylmethanone
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C25H24N2O3S
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1
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| 1 |
Ki = 3 nM
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CP0847593
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4-Bromo-N-(3-(R)-1-pyrrolidin-2-ylmethyl-1H-indol-5-yl)-benzenesulfonamide
Show/Hide
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C19H20BrN3O2S
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1
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| 1 |
Ki = 3 nM
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CP0871296
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3,4-Dichloro-N-(3-(R)-1-pyrrolidin-2-ylmethyl-1H-indol-5-yl)-benzenesulfonamide
Show/Hide
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C19H19Cl2N3O2S
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1
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| 1 |
Ki = 3 nM
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CP0880589
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2,5-Dibromo-3,6-difluoro-N-[4-methoxy-3-(4-methyl-piperazin-1-yl)-phenyl]-benzenesulfonamide
Show/Hide
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C18H19Br2F2N3O3S
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1
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| 1 |
Ki = 3.162 nM
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CP0393156
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1-[(5-chloro-3-methyl-1-benzothiophen-2-yl)sulfonyl]-4-piperazin-1-ylindole
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C21H20ClN3O2S2
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1
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| 1 |
Ki = 3.162 nM
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CP0877372
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(S)-N-(1-(naphthalen-1-ylsulfonyl)-1H-indazol-6-yl)piperidine-3-carboxamide
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C23H22N4O3S
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1
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| 1 |
Ki = 3.2 nM
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CP0848234
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3-Amino-N-(3-(naphthalen-1-ylsulfonyl)-1H-indazol-7-yl)propanamide HCl
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C20H19ClN4O3S
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1
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| 1 |
Ki = 3.4 nM
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CP0218959
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1-(4-Isopropylbenzenesulfonyl)-3-(4-methylpiperazin-1-yl)-1H-indole
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C22H27N3O2S
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1
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| 1 |
Ki = 3.4 nM
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CP0279824
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3-chloro-1-(3-chlorophenylsulfonyl)-1,5,6,7,8,9-hexahydroazepino[4,5-f]indole
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C18H16Cl2N2O2S
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1
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| 1 |
Ki = 3.981 nM
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CP0852739
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(R)-N-(1-(naphthalen-1-ylsulfonyl)-1H-indazol-6-yl)piperidine-3-carboxamide
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C23H22N4O3S
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1
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| 1 |
Ki = 4 nM
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CP0847910
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2-Fluoro-N-(3-(R)-1-pyrrolidin-2-ylmethyl-1H-indol-5-yl)-benzenesulfonamide
Show/Hide
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C19H20FN3O2S
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1
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| 1 |
Ki = 4 nM
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CP0911231
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4-Methyl-N-(3-(R)-1-pyrrolidin-2-ylmethyl-1H-indol-5-yl)-benzenesulfonamide
Show/Hide
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C20H23N3O2S
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1
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| 1 |
Ki = 4 nM
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CP0936994
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4-Fluoro-N-(3-(R)-1-pyrrolidin-2-ylmethyl-1H-indol-5-yl)-benzenesulfonamide
Show/Hide
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C19H20FN3O2S
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1
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| 1 |
Ki = 4 nM
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CP0451840
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2-[1-(benzenesulfonyl)indol-3-yl]-N-methylethanamine
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C17H18N2O2S
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1
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| 1 |
Ki = 5 nM
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CP0046703
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1-(2-{4-[5-chloro-1-(4-fluorophenyl)-1H-indol-3-yl]piperidin-1-yl}ethyl)imidazolidin-2-one
Show/Hide
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C24H26ClFN4O
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1
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| 1 |
Ki = 5 nM
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CP0185590
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4-Bromo-N-[4-methoxy-3-(4-methyl-piperazin-1-yl)-phenyl]-benzenesulfonamide
Show/Hide
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C18H22BrN3O3S
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1
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| 1 |
Ki = 5.012 nM
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CP0216543
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N-[3-(1,3,4,6,7,8,9,9a-octahydropyrido[1,2-a]pyrazin-2-yl)-4-methoxyphenyl]-5-chloro-3-methyl-1-benzothiophene-2-sulfonamide
Show/Hide
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C24H28ClN3O3S2
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1
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| 1 |
Ki = 5.012 nM
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CP0393158
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1-(3-chlorophenyl)sulfonyl-4-piperazin-1-ylindole-5-carbonitrile
Show/Hide
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C19H17ClN4O2S
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1
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| 1 |
Ki = 5.012 nM
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CP0045063
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2-methyl-4-(4-methylpiperazin-1-yl)-10H-thieno[2,3-b][1,5]benzodiazepine
Show/Hide
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C17H20N4S
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1
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| 1 |
Ki = 6 nM
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CP0393160
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5-chloro-1-(4-chlorophenyl)sulfonyl-4-piperazin-1-ylindole
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C18H17Cl2N3O2S
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1
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| 1 |
Ki = 6.31 nM
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CP0045725
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(4R,7R)-N,N-diethyl-6-methyl-6,11-diazatetracyclo[7.6.1.0^{2,7}.0^{12,16}]hexadeca-1(16),2,9,12,14-pentaene-4-carboxamide
Show/Hide
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C20H25N3O
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1
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| 1 |
Ki = 6.31 nM
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CP0919323
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3,4-Dichloro-N-[3-((S)-1-methyl-pyrrolidin-2-ylmethyl)-1H-indol-5-yl]-benzenesulfonamide
Show/Hide
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C20H21Cl2N3O2S
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1
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| 1 |
Ki = 7 nM
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CP0186950
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(4S,5S)-4-Dimethylamino-1-(toluene-4-sulfonyl)-1,3,4,5-tetrahydro-benzo[cd]indol-5-ol
Show/Hide
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C20H22N2O3S
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1
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| 1 |
Ki = 7.2 nM
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CP0293425
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5-(benzenesulfonyl)-11-methyl-4-methylsulfanyl-2,3,7,11-tetrazatricyclo[7.4.0.02,6]trideca-1(9),3,5,7-tetraene
Show/Hide
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C17H18N4O2S2
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1
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| 1 |
Ki = 7.7 nM
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CP0402960
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5-Bromo-1-(3-chlorobenzenesulfonyl)-3-(4-methylpiperazin-1-yl)-1H-indole
Show/Hide
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C19H19BrClN3O2S
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1
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| 1 |
Ki = 7.8 nM
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CP0492179
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2-[1-(3-chlorophenyl)sulfonyl-5-methoxyindol-3-yl]-N,N-dimethylethanamine
Show/Hide
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C19H21ClN2O3S
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1
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| 1 |
Ki = 7.9 nM
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CP0087260
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3-[1-(benzenesulfonyl)indol-4-yl]-N,N-dimethylpropan-1-amine
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C19H22N2O2S
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1
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| 1 |
Ki = 7.9 nM
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CP0393155
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3-(benzenesulfonyl)-7-piperazin-1-yl-1H-pyrrolo[3,2-b]pyridine
Show/Hide
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C17H18N4O2S
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1
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| 1 |
Ki = 7.943 nM
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CP0436008
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5-chloro-1-naphthalen-1-ylsulfonyl-4-piperazin-1-ylindole
Show/Hide
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C22H20ClN3O2S
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1
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| 1 |
Ki = 7.943 nM
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CP0316955
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1-(thiophen-3-ylsulfonyl)-1,5,6,7,8,9-hexahydroazepino[4,5-f]indole
Show/Hide
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C16H16N2O2S2
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1
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| 1 |
Ki = 7.943 nM
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CP0327703
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1-(2-chlorophenylsulfonyl)-1,5,6,7,8,9-hexahydroazepino[4,5-f]indole
Show/Hide
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C18H17ClN2O2S
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1
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| 1 |
Ki = 7.943 nM
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CP0805875
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1-(4-chlorophenylsulfonyl)-1,5,6,7,8,9-hexahydroazepino[4,5-f]indole
Show/Hide
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C18H17ClN2O2S
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1
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| 1 |
Ki = 7.943 nM
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CP0373093
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2-Methylsulfanyl-3-phenylsulfonyl-5,6,7,8-tetrahydro-pyrazolo[5,1-b]quinazoline
Show/Hide
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C17H17N3O2S2
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1
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| 1 |
Ki = 7.97 nM
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CP0890154
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2-(1-(1-(6-chloroimidazo[2,1-b]thiazol-5-ylsulfonyl)-1H-indol-3-yl)ethylidene)hydrazinecarboximidamide
Show/Hide
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C16H14ClN7O2S2
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1
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| 1 |
Ki <= 8 nM
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CP0948723
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2-(1-(1-(4-aminophenylsulfonyl)-1H-indol-3-yl)ethylidene)hydrazinecarboximidamide
Show/Hide
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C17H18N6O2S
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1
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| 1 |
Ki <= 8 nM
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CP0541011
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2-(5-methoxy-1-thiophen-2-ylsulfonylindol-3-yl)-N,N-dimethylethanamine
Show/Hide
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C17H20N2O3S2
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1
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| 1 |
Ki = 8.3 nM
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CP0477210
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3-(4-ethylpiperazin-1-yl)-1-(4-isopropylphenylsulfonyl)-1H-indole
Show/Hide
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C23H29N3O2S
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1
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| 1 |
Ki = 8.6 nM
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CP0871295
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2-Chloro-4-fluoro-N-(3-(R)-1-pyrrolidin-2-ylmethyl-1H-indol-5-yl)-benzenesulfonamide
Show/Hide
|
C19H19ClFN3O2S
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1
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| 1 |
Ki = 9 nM
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CP0231487
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5-Bromo-1-(4-fluorobenzenesulfonyl)-3-(4-methylpiperazin-1-yl)-1H-indole
Show/Hide
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C19H19BrFN3O2S
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1
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| 1 |
Ki = 9.2 nM
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CP0152148
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2-(5-methoxy-1-naphthalen-2-ylsulfonylindol-3-yl)-N,N-dimethylethanamine
Show/Hide
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C23H24N2O3S
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1
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| 1 |
Ki = 9.8 nM
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CP0453186
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3-Piperidin-3-yl-1-(thiophene-2-sulfonyl)-1H-indole
Show/Hide
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C17H18N2O2S2
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1
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| 1 |
Ki = 9.8 nM
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CP0911382
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N-[4-Methoxy-3-(4-methyl-piperazin-1-yl)-phenyl]-benzenesulfonamide
Show/Hide
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C18H23N3O3S
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1
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| 1 |
Ki = 10 nM
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CP0419509
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3-Piperidin-3-yl-1-(4-trifluoromethyl-benzenesulfonyl)-1H-indole
Show/Hide
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C20H19F3N2O2S
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1
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| 1 |
Ki = 10 nM
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CP0073333
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3-benzenesulfonyl-8-piperazin-1-ylquinoline
Show/Hide
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C19H19N3O2S
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1
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| 1 |
Ki < 10 nM
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CP0549838
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5-Bromo-1-(2-bromobenzenesulfonyl)-3-(4-methylpiperazin-1-yl)-1H-indole
Show/Hide
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C19H19Br2N3O2S
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1
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| 1 |
Ki = 10.2 nM
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CP0454961
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(2-{3-[(3-fluorobenzene)sulfonyl]-1H-indol-1-yl}ethyl)dimethylamine
Show/Hide
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C18H19FN2O2S
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2
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| 1 |
Ki = 10.3 nM
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| 2 |
Ki = 13 nM
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CP0506044
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5-Bromo-1-(4-fluorobenzenesulfonyl)-3-(4-ethylpiperazin-1-yl)-1H-indole
Show/Hide
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C20H21BrFN3O2S
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1
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| 1 |
Ki = 10.6 nM
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CP0379693
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5-Chloro-1-(4-fluorobenzenesulfonyl)-3-(4-ethylpiperazin-1-yl)-1H-indole
Show/Hide
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C20H21ClFN3O2S
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1
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| 1 |
Ki = 10.7 nM
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CP0487279
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1-(3-chlorophenylsulfonyl)-3-(4-methylpiperazin-1-yl)-1H-indole
Show/Hide
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C19H20ClN3O2S
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1
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| 1 |
Ki = 10.8 nM
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CP0441765
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2-[1-(2-chlorophenyl)sulfonyl-5-methoxyindol-3-yl]-N,N-dimethylethanamine
Show/Hide
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C19H21ClN2O3S
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1
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| 1 |
Ki = 11 nM
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CP0862925
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3-Chloro-N-[3-((S)-1-methyl-pyrrolidin-2-ylmethyl)-1H-indol-5-yl]-benzenesulfonamide
Show/Hide
|
C20H22ClN3O2S
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1
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| 1 |
Ki = 11 nM
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CP0528634
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3-(3-fluorophenylsulfonyl)-6-(piperazin-1-yl)-1H-indazole
Show/Hide
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C17H17FN4O2S
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1
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| 1 |
Ki = 11 nM
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CP0059145
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1-(4-Fluorobenzenesulfonyl)-3-(4-methylpiperazin-1-yl)-1H-indole
Show/Hide
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C19H20FN3O2S
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1
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| 1 |
Ki = 11.8 nM
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CP0508561
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2-[1-(benzenesulfonyl)-5-methoxy-2-methylindol-3-yl]-N,N-dimethylethanamine
Show/Hide
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C20H24N2O3S
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1
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| 1 |
Ki = 12 nM
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CP0456180
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3-ethyl-6-(phenylsulfonyl)-1,2,3,4,5,6-hexahydroazepino[4,5-b]indole
Show/Hide
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C20H22N2O2S
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1
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| 1 |
Ki = 12 nM
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CP0489374
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6-(3-methoxyphenylsulfonyl)-1,2,3,4,5,6-hexahydroazepino[4,5-b]indole
Show/Hide
|
C19H20N2O3S
|
1
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| 1 |
Ki = 12 nM
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CP0080436
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4-Amino-N-(2,6-bis-methylamino-pyridin-4-yl)-benzenesulfonamide
Show/Hide
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C13H17N5O2S
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2
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| 1 |
Ki = 12 nM
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| 2 |
Ki = 12.59 nM
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CP0434905
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2-(4-isopropylpiperazin-1-yl)-4-(naphthalen-1-ylsulfonyl)benzo[d]oxazole
Show/Hide
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C24H25N3O3S
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1
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| 1 |
Ki = 13 nM
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CP0456530
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1-(2-Chloro-benzenesulfonyl)-3-(1,2,5,6-tetrahydro-pyridin-3-yl)-1H-indole
Show/Hide
|
C19H17ClN2O2S
|
1
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| 1 |
Ki = 13 nM
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CP0515645
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1-(2,4-Difluoro-benzenesulfonyl)-3-(1,2,5,6-tetrahydro-pyridin-3-yl)-1H-indole
Show/Hide
|
C19H16F2N2O2S
|
1
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| 1 |
Ki = 13 nM
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CP0421793
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2-{1-[(4-iodobenzene)sulfonyl]-1H-indol-3-yl}ethan-1-amine
Show/Hide
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C16H15IN2O2S
|
1
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| 1 |
Ki = 14 nM
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CP0540194
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1-(4-Chloro-benzenesulfonyl)-5-fluoro-3-(1,2,3,6-tetrahydro-pyridin-4-yl)-1H-indole
Show/Hide
|
C19H16ClFN2O2S
|
1
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| 1 |
Ki = 14 nM
|
|
|
|
CP0419505
|
1-(3-Chloro-benzenesulfonyl)-3-(1,2,5,6-tetrahydro-pyridin-3-yl)-1H-indole
Show/Hide
|
C19H17ClN2O2S
|
1
|
| 1 |
Ki = 14 nM
|
|
|
|
CP0402014
|
5-chloro-3-(3-fluorophenylsulfonyl)-1-(pyrrolidin-3-yl)-1H-indole
Show/Hide
|
C18H16ClFN2O2S
|
1
|
| 1 |
Ki = 15 nM
|
|
|
|
CP0379691
|
1-(2-bromophenylsulfonyl)-3-(4-methylpiperazin-1-yl)-1H-indole
Show/Hide
|
C19H20BrN3O2S
|
1
|
| 1 |
Ki = 15.2 nM
|
|
|
|
CP0509829
|
2-[3-(benzenesulfonyl)indol-1-yl]-N-methylethanamine
Show/Hide
|
C17H18N2O2S
|
1
|
| 1 |
Ki = 15.5 nM
|
|
|
|
CP0379692
|
3-(4-methylpiperazin-1-yl)-1-(phenylsulfonyl)-1H-indole
Show/Hide
|
C19H21N3O2S
|
1
|
| 1 |
Ki = 15.9 nM
|
|
|
|
CP0457904
|
2-{1-[(2-iodobenzene)sulfonyl]-1H-indol-3-yl}ethan-1-amine
Show/Hide
|
C16H15IN2O2S
|
1
|
| 1 |
Ki = 16 nM
|
|
|
|
CP0916805
|
N-[3-((S)-1-Methyl-pyrrolidin-2-ylmethyl)-1H-indol-5-yl]-benzenesulfonamide
Show/Hide
|
C20H23N3O2S
|
1
|
| 1 |
Ki = 16 nM
|
|
|
|
CP0419507
|
1-(4-Methoxy-benzenesulfonyl)-3-(1,2,5,6-tetrahydro-pyridin-3-yl)-1H-indole
Show/Hide
|
C20H20N2O3S
|
1
|
| 1 |
Ki = 16 nM
|
|
|
|
CP0126862
|
1-(8-chloro-10,11-dihydrodibenzo[b,f]thiepin-10-yl)-4-methylpiperazine
Show/Hide
|
C24H23FN4
|
1
|
| 1 |
Ki = 16 nM
|
|
|
|
CP0393102
|
2-[1-(4-chlorophenyl)sulfonyl-5-methoxyindol-3-yl]-N,N-dimethylethanamine
Show/Hide
|
C19H21ClN2O3S
|
1
|
| 1 |
Ki = 17 nM
|
|
|
|
CP0467142
|
2-[3-(benzenesulfonyl)-2-methylindol-1-yl]-N,N-dimethylethanamine
Show/Hide
|
C19H22N2O2S
|
1
|
| 1 |
Ki = 18 nM
|
|
|
|
CP0417831
|
1-(naphthalene-1-sulfonyl)-N-(piperidin-4-ylmethyl)-1H-indazol-6-amine
Show/Hide
|
C23H24N4O2S
|
1
|
| 1 |
Ki = 18 nM
|
|
|
|
CP0431537
|
1-(4-Methoxy-benzenesulfonyl)-3-(1,2,3,6-tetrahydro-pyridin-4-yl)-1H-indole
Show/Hide
|
C20H20N2O3S
|
1
|
| 1 |
Ki = 18 nM
|
|
|
|
CP0402013
|
6-fluoro-3-(3-fluorophenylsulfonyl)-1-(pyrrolidin-3-yl)-1H-indole
Show/Hide
|
C18H16F2N2O2S
|
1
|
| 1 |
Ki = 18 nM
|
|
|
|
CP0411093
|
4-fluoro-3-(3-fluorophenylsulfonyl)-1-(pyrrolidin-3-yl)-1H-indole
Show/Hide
|
C18H16F2N2O2S
|
1
|
| 1 |
Ki = 18 nM
|
|
|
|
CP0434888
|
6-(4-chlorophenylsulfonyl)-1,2,3,4,5,6-hexahydroazepino[4,5-b]indole
Show/Hide
|
C18H17ClN2O2S
|
1
|
| 1 |
Ki = 18 nM
|
|
|
|
CP0292029
|
1-Benzenesulfonyl-3-(2-dimethylamino-ethyl)-1H-indol-5-ol
Show/Hide
|
C18H20N2O3S
|
1
|
| 1 |
Ki = 19 nM
|
|
|
|
CP0399195
|
6-(3-methoxyphenylsulfonyl)-3-methyl-1,2,3,4,5,6-hexahydroazepino[4,5-b]indole
Show/Hide
|
C20H22N2O3S
|
1
|
| 1 |
Ki = 19 nM
|
|
|
|
CP0461400
|
6-(2-chlorophenylsulfonyl)-1,2,3,4,5,6-hexahydroazepino[4,5-b]indole
Show/Hide
|
C18H17ClN2O2S
|
1
|
| 1 |
Ki = 19 nM
|
|
|
|
CP0539489
|
1-(4-Methoxy-benzenesulfonyl)-3-((S)-1-methyl-pyrrolidin-2-ylmethyl)-1H-indole
Show/Hide
|
C21H24N2O3S
|
1
|
| 1 |
Ki = 19.3 nM
|
|
|
|
CP0318039
|
3-(2-Dimethylamino-ethyl)-1H-indole-2-carboxylic acid ethyl ester
Show/Hide
|
C15H20N2O2
|
1
|
| 1 |
Ki = 20 nM
|
|
|
|
CP0430191
|
1-Benzenesulfonyl-5-fluoro-3-piperidin-4-yl-1H-indole
Show/Hide
|
C19H19FN2O2S
|
1
|
| 1 |
Ki = 20 nM
|
|
|
|
CP0525860
|
3-(1,2,3,6-Tetrahydro-pyridin-4-yl)-1-(4-trifluoromethyl-benzenesulfonyl)-1H-indole
Show/Hide
|
C20H17F3N2O2S
|
1
|
| 1 |
Ki = 20 nM
|
|
|
|
CP0483698
|
1-(2,3-Dichloro-benzenesulfonyl)-3-(1,2,5,6-tetrahydro-pyridin-3-yl)-1H-indole
Show/Hide
|
C19H16Cl2N2O2S
|
1
|
| 1 |
Ki = 20 nM
|
|
|
|
CP0510283
|
1-(5-Bromo-thiophene-2-sulfonyl)-3-(S)-1-pyrrolidin-2-ylmethyl-1H-indole
Show/Hide
|
C17H17BrN2O2S2
|
1
|
| 1 |
Ki = 20 nM
|
|
|
|
CP0514875
|
5-Chloro-1-(2-bromobenzenesulfonyl)-3-(4-ethylpiperazin-1-yl)-1H-indole
Show/Hide
|
C20H21BrClN3O2S
|
1
|
| 1 |
Ki = 20.3 nM
|
|
|
|
CP0497532
|
2-{1-[(4-fluorobenzene)sulfonyl]-1H-indol-3-yl}ethan-1-amine
Show/Hide
|
C16H15FN2O2S
|
1
|
| 1 |
Ki = 21 nM
|
|
|
|
CP0402009
|
3-(naphthalen-1-ylsulfonyl)-1-(piperidin-3-yl)-1H-indole
Show/Hide
|
C23H22N2O2S
|
1
|
| 1 |
Ki = 21 nM
|
|
|
|
CP0483471
|
3-(1,2,5,6-Tetrahydro-pyridin-3-yl)-1-(2-trifluoromethyl-benzenesulfonyl)-1H-indole
Show/Hide
|
C20H17F3N2O2S
|
1
|
| 1 |
Ki = 21.7 nM
|
|
|
|
CP0434904
|
4-(4-isopropylphenylsulfonyl)-2-(piperazin-1-yl)benzo[d]oxazole
Show/Hide
|
C20H23N3O3S
|
1
|
| 1 |
Ki = 22 nM
|
|
|
|
CP0926578
|
2-Chloro-N-[3-((S)-1-methyl-pyrrolidin-2-ylmethyl)-1H-indol-5-yl]-benzenesulfonamide
Show/Hide
|
C20H22ClN3O2S
|
1
|
| 1 |
Ki = 22 nM
|
|
|
|
CP0446384
|
1-(3-Chloro-benzenesulfonyl)-3-(S)-1-pyrrolidin-2-ylmethyl-1H-indole
Show/Hide
|
C19H19ClN2O2S
|
1
|
| 1 |
Ki = 22 nM
|
|
|
|
CP0483472
|
1-(4-Chloro-benzenesulfonyl)-3-(1,2,5,6-tetrahydro-pyridin-3-yl)-1H-indole
Show/Hide
|
C19H17ClN2O2S
|
1
|
| 1 |
Ki = 22 nM
|
|
|
|
CP0523797
|
3-(naphthalen-1-ylsulfonyl)-6-(piperazin-1-yl)-1H-indazole
Show/Hide
|
C21H20N4O2S
|
1
|
| 1 |
Ki = 22 nM
|
|
|
|
CP0485469
|
1-(5-Chloro-thiophene-2-sulfonyl)-3-(1,2,5,6-tetrahydro-pyridin-3-yl)-1H-indole
Show/Hide
|
C17H15ClN2O2S2
|
1
|
| 1 |
Ki = 22.7 nM
|
|
|
|
CP0467118
|
2-[3-(benzenesulfonyl)-6-methoxyindol-1-yl]-N,N-dimethylethanamine
Show/Hide
|
C19H22N2O3S
|
1
|
| 1 |
Ki = 23 nM
|
|
|
|
CP0483458
|
1-(3,4-Dimethoxy-benzenesulfonyl)-3-(S)-1-pyrrolidin-2-ylmethyl-1H-indole
Show/Hide
|
C21H24N2O4S
|
1
|
| 1 |
Ki = 23 nM
|
|
|
|
CP0485504
|
6-(4-fluorophenylsulfonyl)-1,2,3,4,5,6-hexahydroazepino[4,5-b]indole
Show/Hide
|
C18H17FN2O2S
|
1
|
| 1 |
Ki = 23 nM
|
|
|
|
CP0486182
|
7-(2-Methoxy-phenylsulfanyl)-1,2,3,4,10,10a-hexahydro-pyrazino[1,2-a]indole
Show/Hide
|
C18H20N2OS
|
1
|
| 1 |
Ki = 23 nM
|
|
|
|
CP0477211
|
5-Bromo-1-(4-isopropylbenzenesulfonyl)-3-(4-methylpiperazin-1-yl)-1H-indole
Show/Hide
|
C22H26BrN3O2S
|
1
|
| 1 |
Ki = 23.2 nM
|
|
|
|
CP0496085
|
5-chloro-2-methoxy-N-[3-[[(2S)-1-methylpyrrolidin-2-yl]methyl]-1H-indol-5-yl]benzenesulfonamide
Show/Hide
|
C21H24ClN3O3S
|
1
|
| 1 |
Ki = 24 nM
|
|
|
|
CP0373085
|
6-(5-chloronaphthalen-2-ylsulfonyl)-1,2,3,4,5,6-hexahydroazepino[4,5-b]indole
Show/Hide
|
C22H19ClN2O2S
|
1
|
| 1 |
Ki = 24 nM
|
|
|
|
CP0862086
|
N-(3-(Naphthalen-1-ylsulfonyl)-1H-indazol-7-yl)-3-(piperidin-1-yl)propanamide HCl
Show/Hide
|
C25H27ClN4O3S
|
1
|
| 1 |
Ki = 24 nM
|
|
|
|
CP0102529
|
[3-[2-(dimethylamino)ethyl]-5-methoxyindol-1-yl]-phenylmethanone
Show/Hide
|
C20H22N2O2
|
1
|
| 1 |
Ki = 25 nM
|
|
|
|
CP0483729
|
1-(5-Chloro-thiophene-2-sulfonyl)-3-(S)-1-pyrrolidin-2-ylmethyl-1H-indole
Show/Hide
|
C17H17ClN2O2S2
|
1
|
| 1 |
Ki = 25 nM
|
|
|
|
CP0393161
|
5-chloro-1-naphthalen-2-ylsulfonyl-4-piperazin-1-ylindole
Show/Hide
|
C22H20ClN3O2S
|
1
|
| 1 |
Ki = 25.12 nM
|
|
|
|
CP0485607
|
3-(benzenesulfonyl)-7-piperazin-1-yl-1H-pyrrolo[2,3-c]pyridine
Show/Hide
|
C17H18N4O2S
|
1
|
| 1 |
Ki = 25.12 nM
|
|
|
|
CP0514877
|
6-Chloro-1-(2-naphthylsulfonyl)-3-(4-ethylpiperazin-1-yl)-1H-indole
Show/Hide
|
C24H24ClN3O2S
|
1
|
| 1 |
Ki = 25.5 nM
|
|
|
|
CP0397846
|
2-[5-methoxy-1-(4-methoxyphenyl)sulfonylindol-3-yl]-N,N-dimethylethanamine
Show/Hide
|
C20H24N2O4S
|
1
|
| 1 |
Ki = 26 nM
|
|
|
|
CP0446379
|
1-(3,4-Difluoro-benzenesulfonyl)-3-(1,2,5,6-tetrahydro-pyridin-3-yl)-1H-indole
Show/Hide
|
C19H16F2N2O2S
|
1
|
| 1 |
Ki = 26 nM
|
|
|
|
CP0449364
|
2-(3-Benzenesulfonyl-5-fluoro-indol-1-yl)-ethylamine
Show/Hide
|
C16H15FN2O2S
|
1
|
| 1 |
Ki = 27 nM
|
|
|
|
CP0500522
|
1-(Naphthalene-2-sulfonyl)-3-(1,2,3,6-tetrahydro-pyridin-4-yl)-1H-indole
Show/Hide
|
C23H20N2O2S
|
1
|
| 1 |
Ki = 27 nM
|
|
|
|
CP0504423
|
6-(piperazin-1-yl)-3-tosyl-1H-indazole
Show/Hide
|
C18H20N4O2S
|
1
|
| 1 |
Ki = 27 nM
|
|
|
|
CP0510282
|
1-Benzenesulfonyl-3-(S)-1-pyrrolidin-2-ylmethyl-1H-indole; oxalic acid
Show/Hide
|
C19H20N2O2S
|
1
|
| 1 |
Ki = 27.7 nM
|
|
|
|
CP0878445
|
N-(3-(Naphthalen-1-ylsulfonyl)-1H-indazol-7-yl)piperidine-4-carboxamide HCl
Show/Hide
|
C23H23ClN4O3S
|
1
|
| 1 |
Ki = 28 nM
|
|
|
|
CP0430188
|
4-[5-Nitro-3-(1,2,3,6-tetrahydro-pyridin-4-yl)-indole-1-sulfonyl]-phenylamine
Show/Hide
|
C19H18N4O4S
|
1
|
| 1 |
Ki = 29 nM
|
|
|
|
CP0440513
|
6-tosyl-1,2,3,4,5,6-hexahydroazepino[4,5-b]indole
Show/Hide
|
C19H20N2O2S
|
1
|
| 1 |
Ki = 29 nM
|
|
|
|
CP0421891
|
2-{1-[(3,4-dichlorobenzene)sulfonyl]-1H-indol-3-yl}ethan-1-amine
Show/Hide
|
C16H14Cl2N2O2S
|
1
|
| 1 |
Ki = 30 nM
|
|
|
|
CP0848609
|
3-(Naphthalen-1-ylsulfonyl)-N-(piperidin-4-yl)-1H-indazol-7-amine HCl
Show/Hide
|
C22H23ClN4O2S
|
1
|
| 1 |
Ki = 30 nM
|
|
|
|
CP0538821
|
5-Bromo-1-(4-isopropylbenzenesulfonyl)-3-(4-ethylpiperazin-1-yl)-1H-indole
Show/Hide
|
C23H28BrN3O2S
|
1
|
| 1 |
Ki = 30.1 nM
|
|
|
|
CP0511747
|
6-Chloro-1-(2-bromobenzenesulfonyl)-3-(4-methylpiperazin-1-yl)-1H-indole
Show/Hide
|
C19H19BrClN3O2S
|
1
|
| 1 |
Ki = 30.2 nM
|
|
|
|
CP0477212
|
5-Chloro-1-(4-isopropylbenzenesulfonyl)-3-(4-ethylpiperazin-1-yl)-1H-indole
Show/Hide
|
C23H28ClN3O2S
|
1
|
| 1 |
Ki = 30.5 nM
|
|
|
|
CP0447857
|
4-(3-chlorophenylsulfonyl)-2-(piperazin-1-yl)benzo[d]oxazole
Show/Hide
|
C17H16ClN3O3S
|
1
|
| 1 |
Ki = 31 nM
|
|
|
|
CP0442996
|
2-{1-[(4,5-dichlorothiophene-2-)sulfonyl]-1H-indol-3-yl}ethan-1-amine
Show/Hide
|
C14H12Cl2N2O2S2
|
1
|
| 1 |
Ki = 31 nM
|
|
|
|
CP0394050
|
4-[6-Nitro-3-(1,2,3,6-tetrahydro-pyridin-4-yl)-indole-1-sulfonyl]-phenylamine
Show/Hide
|
C19H18N4O4S
|
1
|
| 1 |
Ki = 31 nM
|
|
|
|
CP0848235
|
N-(3-(Naphthalen-1-ylsulfonyl)-1H-indazol-6-yl)piperidine-4-carboxamide HCl
Show/Hide
|
C23H23ClN4O3S
|
1
|
| 1 |
Ki = 31 nM
|
|
|
|
CP0544026
|
1-Benzenesulfonyl-3-(2-dimethylamino-ethyl)-1H-indole-5-carbonitrile
Show/Hide
|
C19H19N3O2S
|
1
|
| 1 |
Ki = 33 nM
|
|
|
|
CP0447858
|
2-(piperazin-1-yl)-4-(4-(trifluoromethyl)phenylsulfonyl)benzo[d]oxazole
Show/Hide
|
C18H16F3N3O3S
|
1
|
| 1 |
Ki = 33 nM
|
|
|
|
CP0515647
|
3-(S)-1-Pyrrolidin-2-ylmethyl-1-(toluene-4-sulfonyl)-1H-indole
Show/Hide
|
C20H22N2O2S
|
1
|
| 1 |
Ki = 33 nM
|
|
|
|
CP0399196
|
6-(4-methoxyphenylsulfonyl)-1,2,3,4,5,6-hexahydroazepino[4,5-b]indole
Show/Hide
|
C19H20N2O3S
|
1
|
| 1 |
Ki = 33 nM
|
|
|
|
CP0434890
|
6-(3-fluorophenylsulfonyl)-1,2,3,4,5,6-hexahydroazepino[4,5-b]indole
Show/Hide
|
C18H17FN2O2S
|
1
|
| 1 |
Ki = 33 nM
|
|
|
|
CP0017601
|
2,8-dimethyl-5-[2-(6-methylpyridin-3-yl)ethyl]-3,4-dihydro-1H-pyrido[4,3-b]indole
Show/Hide
|
C21H25N3
|
1
|
| 1 |
Ki = 33.88 nM
|
|
|
|
CP0845006
|
4-Methoxy-N-[3-((S)-1-methyl-pyrrolidin-2-ylmethyl)-1H-indol-5-yl]-benzenesulfonamide
Show/Hide
|
C21H25N3O3S
|
1
|
| 1 |
Ki = 34 nM
|
|
|
|
CP0419510
|
1-(4-Iodo-benzenesulfonyl)-3-(S)-1-pyrrolidin-2-ylmethyl-1H-indole
Show/Hide
|
C19H19IN2O2S
|
1
|
| 1 |
Ki = 34 nM
|
|
|
|
CP0940320
|
2-Chloro-4-fluoro-N-[3-((S)-1-methyl-pyrrolidin-2-ylmethyl)-1H-indol-5-yl]-benzenesulfonamide
Show/Hide
|
C20H21ClFN3O2S
|
1
|
| 1 |
Ki = 35 nM
|
|
|
|
CP0476944
|
5-(4-fluorophenyl)sulfonyl-11-methyl-4-methylsulfanyl-2,3,7,11-tetrazatricyclo[7.4.0.02,6]trideca-1(9),3,5,7-tetraene
Show/Hide
|
C17H17FN4O2S2
|
1
|
| 1 |
Ki = 35.7 nM
|
|
|
|
CP0498918
|
4-(naphthalen-1-ylsulfonyl)-2-(4-propylpiperazin-1-yl)benzo[d]oxazole
Show/Hide
|
C24H25N3O3S
|
1
|
| 1 |
Ki = 36 nM
|
|
|
|
CP0889334
|
3-Chloro-N-(3-(S)-1-pyrrolidin-2-ylmethyl-1H-indol-5-yl)-benzenesulfonamide
Show/Hide
|
C19H20ClN3O2S
|
1
|
| 1 |
Ki = 36 nM
|
|
|
|
CP0950483
|
1-(phenylsulfonyl)-2,3,4,6,7,8,9,10-octahydro-1H-azepino[4,5-g]quinoline
Show/Hide
|
C19H22N2O2S
|
1
|
| 1 |
Ki = 39.81 nM
|
|
|
|
CP0541790
|
2-(1-Benzenesulfonyl-5-methoxy-1H-indol-3-yl)-ethylamine
Show/Hide
|
C17H18N2O3S
|
1
|
| 1 |
Ki = 40 nM
|
|
|
|
CP0515648
|
1-(4-Methoxy-benzenesulfonyl)-3-(S)-1-pyrrolidin-2-ylmethyl-1H-indole
Show/Hide
|
C20H22N2O3S
|
1
|
| 1 |
Ki = 40 nM
|
|
|
|
CP0372403
|
4-(phenylsulfonyl)-2-(piperazin-1-yl)benzo[d]oxazole
Show/Hide
|
C17H17N3O3S
|
1
|
| 1 |
Ki = 41 nM
|
|
|
|
CP0384531
|
6-(3-chlorophenylsulfonyl)-1,2,3,4,5,6-hexahydroazepino[4,5-b]indole
Show/Hide
|
C18H17ClN2O2S
|
1
|
| 1 |
Ki = 41 nM
|
|
|
|
CP0371932
|
9-(3-Chloro-benzenesulfonyl)-2,3,4,9-tetrahydro-1H-beta-carboline
Show/Hide
|
C17H15ClN2O2S
|
1
|
| 1 |
Ki = 41.7 nM
|
|
|
|
CP0509838
|
2-[3-(benzenesulfonyl)-6-chloroindol-1-yl]-N,N-dimethylethanamine
Show/Hide
|
C18H19ClN2O2S
|
1
|
| 1 |
Ki = 42 nM
|
|
|
|
CP0500604
|
2-(3-(6-chloroimidazo[2,1-b]thiazol-5-ylsulfonyl)-1H-pyrrolo[3,2-b]pyridin-1-yl)ethanamine
Show/Hide
|
C14H12ClN5O2S2
|
1
|
| 1 |
Ki = 42 nM
|
|
|
|
CP0536751
|
N-(4-aminophenyl)-2-bromo-6-(methylamino)pyridine-4-sulfonamide
Show/Hide
|
C12H13BrN4O2S
|
1
|
| 1 |
Ki = 42.66 nM
|
|
|
|
CP0485442
|
1-(2-Bromo-benzenesulfonyl)-3-(S)-1-pyrrolidin-2-ylmethyl-1H-indole
Show/Hide
|
C19H19BrN2O2S
|
1
|
| 1 |
Ki = 43 nM
|
|
|
|
CP0529898
|
1-Benzenesulfonyl-5-methoxy-3-(2-pyrrolidin-1-yl-ethyl)-1H-indole
Show/Hide
|
C21H24N2O3S
|
1
|
| 1 |
Ki = 44 nM
|
|
|
|
CP0421112
|
2-[3-(benzenesulfonyl)-5-fluoroindol-1-yl]-N,N-dimethylethanamine
Show/Hide
|
C18H19FN2O2S
|
1
|
| 1 |
Ki = 44 nM
|
|
|
|
CP0399777
|
1-(5-Chloro-3-methyl-benzo[b]thiophene-2-sulfonyl)-3-piperidin-3-yl-1H-indole
Show/Hide
|
C22H21ClN2O2S2
|
1
|
| 1 |
Ki = 44 nM
|
|
|
|
CP0906623
|
3-(Dimethylamino)-N-(3-(naphthalen-1-ylsulfonyl)-1Hindazol-6-yl)propanamide HCl
Show/Hide
|
C22H23ClN4O3S
|
1
|
| 1 |
Ki = 44 nM
|
|
|
|
CP0941017
|
3-(Naphthalen-1-ylsulfonyl)-N-(piperidin-4-ylmethyl)-1Hindazol-6-amine HCl
Show/Hide
|
C23H25ClN4O2S
|
1
|
| 1 |
Ki = 44 nM
|
|
|
|
CP0419506
|
3-(1,2,5,6-Tetrahydro-pyridin-3-yl)-1-(3-trifluoromethyl-benzenesulfonyl)-1H-indole
Show/Hide
|
C20H17F3N2O2S
|
1
|
| 1 |
Ki = 44.7 nM
|
|
|
|
CP0538241
|
2-[5-methoxy-1-(4-methylphenyl)sulfonylindol-3-yl]-N,N-dimethylethanamine
Show/Hide
|
C20H24N2O3S
|
1
|
| 1 |
Ki = 45 nM
|
|
|
|
CP0439249
|
3-[(3-Chlorophenyl)sulfonyl]-1-(2-pyrrolidin-1-ylethyl)-1H-pyrrolo[2,3-b]pyridine
Show/Hide
|
C19H20ClN3O2S
|
1
|
| 1 |
Ki = 45 nM
|
|
|
|
CP0522567
|
2-[3-(benzenesulfonyl)-6-fluoroindol-1-yl]-N,N-dimethylethanamine
Show/Hide
|
C18H19FN2O2S
|
1
|
| 1 |
Ki = 46 nM
|
|
|
|
CP0441457
|
6-(4-(trifluoromethyl)phenylsulfonyl)-1,2,3,4,5,6-hexahydroazepino[4,5-b]indole
Show/Hide
|
C19H17F3N2O2S
|
1
|
| 1 |
Ki = 46 nM
|
|
|
|
CP0421534
|
2-(3-(m-tolylsulfonyl)-1H-pyrrolo[3,2-b]pyridin-1-yl)ethanamine
Show/Hide
|
C16H17N3O2S
|
1
|
| 1 |
Ki = 46 nM
|
|
|
|
CP0487352
|
3-(1-methylpiperidin-4-yl)-5-(4-(trifluoromethyl)phenylsulfonyl)-1H-indazole
Show/Hide
|
C20H20F3N3O2S
|
1
|
| 1 |
Ki = 46 nM
|
|
|
|
CP0442997
|
2-{1-[(4-methoxybenzene)sulfonyl]-1H-indol-3-yl}ethan-1-amine
Show/Hide
|
C17H18N2O3S
|
1
|
| 1 |
Ki = 47 nM
|
|
|
|
CP0510281
|
1-(3,4-Dichloro-benzenesulfonyl)-3-(1,2,5,6-tetrahydro-pyridin-3-yl)-1H-indole
Show/Hide
|
C19H16Cl2N2O2S
|
1
|
| 1 |
Ki = 48 nM
|
|
|
|
CP0522155
|
3-(naphthalen-1-ylsulfonyl)-4-(piperazin-1-yl)-1H-indazole
Show/Hide
|
C21H20N4O2S
|
1
|
| 1 |
Ki = 48 nM
|
|
|
|
CP0521659
|
3-(1-methylpiperidin-4-yl)-5-(4-(trifluoromethoxy)phenylsulfonyl)-1H-indazole
Show/Hide
|
C20H20F3N3O3S
|
1
|
| 1 |
Ki = 48 nM
|
|
|
|
CP0483700
|
1-(4-Chloro-benzenesulfonyl)-3-(S)-1-pyrrolidin-2-ylmethyl-1H-indole
Show/Hide
|
C19H19ClN2O2S
|
1
|
| 1 |
Ki = 49 nM
|
|
|
|
CP0485093
|
1-(3,4-Dichloro-benzenesulfonyl)-3-(S)-1-pyrrolidin-2-ylmethyl-1H-indole
Show/Hide
|
C19H18Cl2N2O2S
|
1
|
| 1 |
Ki = 49 nM
|
|
|
|
CP0489541
|
1-(1-benzylpiperidin-4-yl)-3-(phenylsulfonyl)-1H-indole
Show/Hide
|
C26H26N2O2S
|
1
|
| 1 |
Ki = 49 nM
|
|
|
|
CP0398423
|
1-sulfonylindazole, 6b
Show/Hide
|
C20H18N4O3S
|
1
|
| 1 |
Ki = 50 nM
|
|
|
|
CP0502539
|
4-[5-Benzyloxy-3-(1,2,3,6-tetrahydro-pyridin-4-yl)-indole-1-sulfonyl]-phenylamine
Show/Hide
|
C26H25N3O3S
|
1
|
| 1 |
Ki = 50 nM
|
|
|
|
CP0522399
|
3-ethyl-6-(3-methoxyphenylsulfonyl)-1,2,3,4,5,6-hexahydroazepino[4,5-b]indole
Show/Hide
|
C21H24N2O3S
|
1
|
| 1 |
Ki = 50 nM
|
|
|
|
CP0389550
|
3-(1-methylpiperidin-4-yl)-5-(m-tolylsulfonyl)-1H-indazole
Show/Hide
|
C20H23N3O2S
|
1
|
| 1 |
Ki = 50 nM
|
|
|
|
CP0459250
|
7-m-Tolylsulfanyl-1,2,3,4,10,10a-hexahydro-pyrazino[1,2-a]indole
Show/Hide
|
C18H20N2S
|
1
|
| 1 |
Ki = 50 nM
|
|
|
|
CP0118951
|
4-Amino-N-(2,6-bis-dimethylamino-pyrimidin-4-yl)-benzenesulfonamide
Show/Hide
|
C12H16N6O2S
|
2
|
| 1 |
Ki = 50.12 nM
|
|
|
| 2 |
Ki = 55 nM
|
|
|
|
CP0170130
|
(6aR,9R)-N-[(2R,5S,8S,8aS)-8-benzyl-8a-hydroxy-2-methyl-5-(2-methylpropyl)-3,6-dioxo-7,8-dihydro-5H-[1,3]oxazolo[3,2-a]pyrazin-2-yl]-7-methyl-6,6a,8,9-tetrahydro-4H-indolo[4,3-fg]quinoline-9-carboxamide
Show/Hide
|
C34H39N5O5
|
1
|
| 1 |
Ki = 50.12 nM
|
|
|
|
CP0491336
|
5-(naphthalen-1-ylsulfonyl)-2-(piperazin-1-yl)benzo[d]oxazole
Show/Hide
|
C21H19N3O3S
|
1
|
| 1 |
Ki = 52 nM
|
|
|
|
CP0848232
|
3-(Naphthalen-1-ylsulfonyl)-N-(piperidin-4-yl)-1H-indazol-6-amine HCl
Show/Hide
|
C22H23ClN4O2S
|
1
|
| 1 |
Ki = 53 nM
|
|
|
|
CP0310112
|
4-(2,6-dibromopyridin-4-yl)sulfonylaniline
Show/Hide
|
C11H8Br2N2O2S
|
1
|
| 1 |
Ki = 53.7 nM
|
|
|
|
CP0409092
|
[3-[2-(dimethylamino)ethyl]-5-hydroxyindol-1-yl]-phenylmethanone
Show/Hide
|
C19H20N2O2
|
1
|
| 1 |
Ki = 54 nM
|
|
|
|
CP0459139
|
4-(3-fluorophenylsulfonyl)-2-(piperazin-1-yl)benzo[d]oxazole
Show/Hide
|
C17H16FN3O3S
|
1
|
| 1 |
Ki = 54 nM
|
|
|
|
CP0409238
|
4-(1-Benzenesulfonyl-1H-indol-3-yl)-3,6-dihydro-2H-pyridine-1-carboxylic acid tert-butyl ester
Show/Hide
|
C24H26N2O4S
|
1
|
| 1 |
Ki = 54 nM
|
|
|
|
CP0874735
|
4-Amino-N-(2,6-bis-methylamino-pyrimidin-4-yl)-benzenesulfonamide dihydrobromide
Show/Hide
|
C12H18Br2N6O2S
|
1
|
| 1 |
Ki = 54.95 nM
|
|
|
|
CP0380693
|
3-(1-methylpiperidin-4-yl)-5-(phenylsulfonyl)-1H-indazole
Show/Hide
|
C19H21N3O2S
|
1
|
| 1 |
Ki = 55 nM
|
|
|
|
CP0514876
|
6-Chloro-1-(4-isopropylbenzenesulfonyl)-3-(4-methylpiperazin-1-yl)-1H-indole
Show/Hide
|
C22H26ClN3O2S
|
1
|
| 1 |
Ki = 55.3 nM
|
|
|
|
CP0480038
|
1-(1-(2-(dimethylamino)ethyl)-3-(phenylsulfonyl)-1H-pyrrolo[3,2-b]pyridin-5-yl)ethanone
Show/Hide
|
C19H21N3O3S
|
1
|
| 1 |
Ki = 56 nM
|
|
|
|
CP0494988
|
N,N-dimethyl-2-[3-(4-methylphenyl)sulfonylindol-1-yl]ethanamine
Show/Hide
|
C19H22N2O2S
|
1
|
| 1 |
Ki = 57 nM
|
|
|
|
CP0847591
|
4-Bromo-N-(3-(S)-1-pyrrolidin-2-ylmethyl-1H-indol-5-yl)-benzenesulfonamide
Show/Hide
|
C19H20BrN3O2S
|
1
|
| 1 |
Ki = 57 nM
|
|
|
|
CP0862083
|
3-(Naphthalen-1-ylsulfonyl)-N-(piperidin-6-yl)-1H-indazol-6-amine HCl
Show/Hide
|
C22H23ClN4O2S
|
1
|
| 1 |
Ki = 57 nM
|
|
|
|
CP0515646
|
1-(2,4-Dimethyl-oxazole-5-sulfonyl)-3-(1,2,5,6-tetrahydro-pyridin-3-yl)-1H-indole
Show/Hide
|
C18H19N3O3S
|
1
|
| 1 |
Ki = 58 nM
|
|
|
|
CP0488669
|
6-(benzenesulfonyl)-2,3,4,9-tetrahydro-1H-carbazol-3-amine
Show/Hide
|
C18H18N2O2S
|
1
|
| 1 |
Ki = 58 nM
|
|
|
|
CP0513900
|
5-(benzenesulfonyl)-4,11-dimethyl-2,3,7,11-tetrazatricyclo[7.4.0.02,6]trideca-1(9),3,5,7-tetraene
Show/Hide
|
C17H18N4O2S
|
1
|
| 1 |
Ki = 60.4 nM
|
|
|
|
CP0056386
|
5-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-6-chloroindolin-2-one
Show/Hide
|
C21H21ClN4OS
|
1
|
| 1 |
Ki = 61 nM
|
|
|
|
CP0529873
|
2-[1-(benzenesulfonyl)-5-methoxy-2,3-dihydroindol-3-yl]-N,N-dimethylethanamine
Show/Hide
|
C19H24N2O3S
|
1
|
| 1 |
Ki = 63 nM
|
|
|
|
CP0942002
|
3-Cyano-N-[4-methoxy-3-(4-methyl-piperazin-1-yl)-phenyl]-benzenesulfonamide
Show/Hide
|
C19H22N4O3S
|
1
|
| 1 |
Ki = 63.1 nM
|
|
|
|
CP0379694
|
6-Chloro-1-(2,5-dimethoxybenzenesulfonyl)-3-(4-ethylpiperazin-1-yl)-1H-indole
Show/Hide
|
C22H26ClN3O4S
|
1
|
| 1 |
Ki = 63.5 nM
|
|
|
|
CP0515687
|
4-(4-fluorophenylsulfonyl)-2-(piperazin-1-yl)benzo[d]oxazole
Show/Hide
|
C17H16FN3O3S
|
1
|
| 1 |
Ki = 64 nM
|
|
|
|
CP0941018
|
3-(Diethylamino)-N-(3-(naphthalen-1-ylsulfonyl)-1Hindazol-6-yl)propanamide HCl
Show/Hide
|
C24H27ClN4O3S
|
1
|
| 1 |
Ki = 65 nM
|
|
|
|
CP0862084
|
3-(Naphthalen-1-ylsulfonyl)-N-(piperidin-7-yl)-1H-indazol-7-amine HCl
Show/Hide
|
C22H23ClN4O2S
|
1
|
| 1 |
Ki = 66 nM
|
|
|
|
CP0479483
|
5-(4-fluorophenylsulfonyl)-3-(1-methylpiperidin-4-yl)-1H-indazole
Show/Hide
|
C19H20FN3O2S
|
1
|
| 1 |
Ki = 66 nM
|
|
|
|
CP0411171
|
3-(3-fluorophenylsulfonyl)-5-methoxy-1-(1-methylpiperidin-3-yl)-1H-indole
Show/Hide
|
C21H23FN2O3S
|
1
|
| 1 |
Ki = 68 nM
|
|
|
|
CP0375394
|
6-(m-tolylsulfonyl)-1,2,3,4,5,6-hexahydroazepino[4,5-b]indole
Show/Hide
|
C19H20N2O2S
|
1
|
| 1 |
Ki = 68 nM
|
|
|
|
CP0506389
|
2-(4-cyclobutylpiperazin-1-yl)-4-(naphthalen-1-ylsulfonyl)benzo[d]oxazole
Show/Hide
|
C25H25N3O3S
|
1
|
| 1 |
Ki = 72 nM
|
|
|
|
CP0411089
|
6-chloro-3-(3-fluorophenylsulfonyl)-1-(pyrrolidin-3-yl)-1H-indole
Show/Hide
|
C18H16ClFN2O2S
|
1
|
| 1 |
Ki = 72 nM
|
|
|
|
CP0448880
|
1-(Butane-1-sulfonyl)-3-(1,2,3,6-tetrahydro-pyridin-4-yl)-1H-indole
Show/Hide
|
C17H22N2O2S
|
1
|
| 1 |
Ki = 77 nM
|
|
|
|
CP0478229
|
7-(4-Methoxy-phenylsulfanyl)-1,2,3,4,10,10a-hexahydro-pyrazino[1,2-a]indole
Show/Hide
|
C18H20N2OS
|
1
|
| 1 |
Ki = 78 nM
|
|
|
|
CP0504995
|
2-(4-cyclopentylpiperazin-1-yl)-4-(naphthalen-1-ylsulfonyl)benzo[d]oxazole
Show/Hide
|
C26H27N3O3S
|
1
|
| 1 |
Ki = 79 nM
|
|
|
|
CP0277471
|
N-[4-methoxy-3-(4-methylpiperazin-1-yl)phenyl]-3-nitrobenzenesulfonamide
Show/Hide
|
C18H22N4O5S
|
1
|
| 1 |
Ki = 79.43 nM
|
|
|
|
CP0486181
|
7-o-Tolylsulfanyl-1,2,3,4,10,10a-hexahydro-pyrazino[1,2-a]indole
Show/Hide
|
C18H20N2S
|
1
|
| 1 |
Ki = 81 nM
|
|
|
|
CP0473062
|
6-Chloro-1-(4-methoxybenzenesulfonyl)-3-(4-ethylpiperazin-1-yl)-1H-indole
Show/Hide
|
C21H24ClN3O3S
|
1
|
| 1 |
Ki = 82.3 nM
|
|
|
|
CP0384529
|
3-isopropyl-6-(3-methoxyphenylsulfonyl)-1,2,3,4,5,6-hexahydroazepino[4,5-b]indole
Show/Hide
|
C22H26N2O3S
|
1
|
| 1 |
Ki = 85 nM
|
|
|
|
CP0452535
|
2-(4-butylpiperazin-1-yl)-4-(naphthalen-1-ylsulfonyl)benzo[d]oxazole
Show/Hide
|
C25H27N3O3S
|
1
|
| 1 |
Ki = 88 nM
|
|
|
|
CP0439175
|
3-[(3-Fluorophenyl)sulfonyl]-1-(2-pyrrolidin-1-ylethyl)-1H-pyrrolo[2,3-b]pyridine
Show/Hide
|
C19H20FN3O2S
|
1
|
| 1 |
Ki = 88 nM
|
|
|
|
CP0543149
|
3-(4-methoxyphenylsulfonyl)-4-(piperazin-1-yl)-1H-indazole
Show/Hide
|
C18H20N4O3S
|
1
|
| 1 |
Ki = 88 nM
|
|
|
|
CP0036840
|
2-(5-methoxy-2-methyl-1H-indol-3-yl)-N,N-dimethylethanamine
Show/Hide
|
C14H20N2O
|
1
|
| 1 |
Ki = 89 nM
|
|
|
|
CP0373083
|
6-(3-(trifluoromethyl)phenylsulfonyl)-1,2,3,4,5,6-hexahydroazepino[4,5-b]indole
Show/Hide
|
C19H17F3N2O2S
|
1
|
| 1 |
Ki = 89 nM
|
|
|
|
CP0402012
|
3-(phenylsulfonyl)-1-(piperidin-4-yl)-1H-indole
Show/Hide
|
C19H20N2O2S
|
1
|
| 1 |
Ki = 91 nM
|
|
|
|
CP0436090
|
5-(3-fluorophenylsulfonyl)-3-(1-methylpiperidin-4-yl)-1H-indazole
Show/Hide
|
C19H20FN3O2S
|
1
|
| 1 |
Ki = 93 nM
|
|
|
|
CP0515368
|
2-[3-(benzenesulfonyl)-4-fluoroindol-1-yl]-N,N-dimethylethanamine
Show/Hide
|
C18H19FN2O2S
|
1
|
| 1 |
Ki = 98 nM
|
|
|
|
CP0281101
|
3-(1-methyl-3,6-dihydro-2H-pyridin-4-yl)-1H-indole
Show/Hide
|
C14H16N2
|
1
|
| 1 |
Ki = 98 nM
|
|
|
|
CP0500169
|
[3-(1-methyl-3,6-dihydro-2H-pyridin-4-yl)indol-1-yl]-phenylmethanone
Show/Hide
|
C21H20N2O
|
1
|
| 1 |
Ki = 99 nM
|
|
|
|
CP0279823
|
1-(pyridin-2-ylsulfonyl)-1,5,6,7,8,9-hexahydroazepino[4,5-f]indole
Show/Hide
|
C17H17N3O2S
|
1
|
| 1 |
Ki = 100 nM
|
|
|
|
CP0899515
|
3-(Naphthalen-1-ylsulfonyl)-N-(2-piperidin-1-ylethyl)-1Hindazole-5-carboxamide HCl
Show/Hide
|
C25H27ClN4O3S
|
1
|
| 1 |
Ki = 107 nM
|
|
|
|
CP0502325
|
3-(4-chlorophenylsulfonyl)-6-(piperazin-1-yl)-1H-indazole
Show/Hide
|
C17H17ClN4O2S
|
1
|
| 1 |
Ki = 110 nM
|
|
|
|
CP0502901
|
7-p-Tolylsulfanyl-1,2,3,4,10,10a-hexahydro-pyrazino[1,2-a]indole
Show/Hide
|
C18H20N2S
|
1
|
| 1 |
Ki = 110 nM
|
|
|
|
CP0512515
|
7-(3-Methoxy-phenylsulfanyl)-1,2,3,4,10,10a-hexahydro-pyrazino[1,2-a]indole
Show/Hide
|
C18H20N2OS
|
1
|
| 1 |
Ki = 110 nM
|
|
|
|
CP0502802
|
1-(1-benzylpyrrolidin-3-yl)-3-(phenylsulfonyl)-1H-indole
Show/Hide
|
C25H24N2O2S
|
1
|
| 1 |
Ki = 113 nM
|
|
|
|
CP0401315
|
4-(1,2,3,4-Tetrahydro-beta-carboline-9-sulfonyl)-phenylamine
Show/Hide
|
C17H17N3O2S
|
1
|
| 1 |
Ki = 116 nM
|
|
|
|
CP0431597
|
3-(1-Methyl-1,2,3,6-tetrahydro-pyridin-4-yl)-indole-1-carboxylic acid phenylamide
Show/Hide
|
C21H21N3O
|
1
|
| 1 |
Ki = 118 nM
|
|
|
|
CP0497288
|
1-(1-benzylpiperidin-3-yl)-3-(phenylsulfonyl)-1H-indole
Show/Hide
|
C26H26N2O2S
|
1
|
| 1 |
Ki = 122 nM
|
|
|
|
CP0522012
|
5-(4-methoxyphenylsulfonyl)-3-(1-methylpiperidin-4-yl)-1H-indazole
Show/Hide
|
C20H23N3O3S
|
1
|
| 1 |
Ki = 123 nM
|
|
|
|
CP0480571
|
6-(3-methoxyphenylsulfonyl)-3-propyl-1,2,3,4,5,6-hexahydroazepino[4,5-b]indole
Show/Hide
|
C22H26N2O3S
|
1
|
| 1 |
Ki = 124 nM
|
|
|
|
CP0522156
|
3-(4-methoxyphenylsulfonyl)-6-(piperazin-1-yl)-1H-indazole
Show/Hide
|
C18H20N4O3S
|
1
|
| 1 |
Ki = 124 nM
|
|
|
|
CP0399575
|
3-(4-chlorophenylsulfonyl)-4-(piperazin-1-yl)-1H-indazole
Show/Hide
|
C17H17ClN4O2S
|
1
|
| 1 |
Ki = 125 nM
|
|
|
|
CP0001238
|
14C-5-hydroxy tryptamine creatinine disulfate
Show/Hide
|
C10H12N2O
|
1
|
| 1 |
Ki = 125.89 nM
|
|
|
|
CP0312260
|
2-Dipropylamino-1,2,3,4-tetrahydro-naphthalene-1,8-diol
Show/Hide
|
C16H26N2O
|
1
|
| 1 |
Ki = 125.89 nM
|
|
|
|
CP0515688
|
4-(naphthalen-1-ylsulfonyl)-2-(4-phenethylpiperazin-1-yl)benzo[d]oxazole
Show/Hide
|
C30H29N3O3S
|
1
|
| 1 |
Ki = 127 nM
|
|
|
|
CP0529821
|
(4S,5S)-5-methoxy-N,N-dimethyl-1-(4-methylphenyl)sulfonyl-4,5-dihydro-3H-benzo[cd]indol-4-amine
Show/Hide
|
C21H24N2O3S
|
1
|
| 1 |
Ki = 130 nM
|
|
|
|
CP0949354
|
2,4-Difluoro-N-(3-(S)-1-pyrrolidin-2-ylmethyl-1H-indol-5-yl)-benzenesulfonamide
Show/Hide
|
C19H19F2N3O2S
|
1
|
| 1 |
Ki = 131 nM
|
|
|
|
CP0520000
|
4-(piperazin-1-yl)-3-tosyl-1H-indazole
Show/Hide
|
C18H20N4O2S
|
1
|
| 1 |
Ki = 134 nM
|
|
|
|
CP0523796
|
3-(3-fluorophenylsulfonyl)-4-(piperazin-1-yl)-1H-indazole
Show/Hide
|
C17H17FN4O2S
|
1
|
| 1 |
Ki = 134 nM
|
|
|
|
CP0399194
|
3-benzyl-6-(3-methoxyphenylsulfonyl)-1,2,3,4,5,6-hexahydroazepino[4,5-b]indole
Show/Hide
|
C26H26N2O3S
|
1
|
| 1 |
Ki = 139 nM
|
|
|
|
CP0496760
|
2-(3-Benzenesulfonyl-6-chloro-indol-1-yl)-ethylamine
Show/Hide
|
C16H15ClN2O2S
|
1
|
| 1 |
Ki = 141 nM
|
|
|
|
CP0502908
|
7-(2-Fluoro-phenylsulfanyl)-1,2,3,4,10,10a-hexahydro-pyrazino[1,2-a]indole
Show/Hide
|
C17H17FN2S
|
1
|
| 1 |
Ki = 150 nM
|
|
|
|
CP0465079
|
7-(4-Fluoro-phenylsulfanyl)-1,2,3,4,10,10a-hexahydro-pyrazino[1,2-a]indole
Show/Hide
|
C17H17FN2S
|
1
|
| 1 |
Ki = 160 nM
|
|
|
|
CP0472250
|
2-(4-isobutylpiperazin-1-yl)-4-(naphthalen-1-ylsulfonyl)benzo[d]oxazole
Show/Hide
|
C25H27N3O3S
|
1
|
| 1 |
Ki = 176 nM
|
|
|
|
CP0375451
|
6-(phenylsulfonyl)-1,2,3,4,5,6-hexahydroazepino[4,5-b]indole
Show/Hide
|
C18H18N2O2S
|
1
|
| 1 |
Ki = 193 nM
|
|
|
|
CP0549459
|
6-(naphthalen-1-ylsulfonyl)-2-(piperazin-1-yl)benzo[d]oxazole
Show/Hide
|
C21H19N3O3S
|
1
|
| 1 |
Ki = 196 nM
|
|
|
|
CP0388399
|
2-(3-(3-fluorophenylsulfonyl)-1H-pyrrolo[3,2-b]pyridin-1-yl)-N,N-dimethylethanamine
Show/Hide
|
C17H18FN3O2S
|
1
|
| 1 |
Ki = 200 nM
|
|
|
|
CP0497839
|
6-(piperazin-1-yl)-3-(4-(trifluoromethyl)phenylsulfonyl)-1H-indazole
Show/Hide
|
C18H17F3N4O2S
|
1
|
| 1 |
Ki = 207 nM
|
|
|
|
CP0471925
|
2-(5-chloro-3-(phenylsulfonyl)-1H-pyrrolo[3,2-b]pyridin-1-yl)-N,N-dimethylethanamine
Show/Hide
|
C17H18ClN3O2S
|
1
|
| 1 |
Ki = 214 nM
|
|
|
|
CP0039958
|
(risperidone)3-{2-[4-(6-Fluoro-benzo[d]isoxazol-3-yl)-piperidin-1-yl]-ethyl}-2-methyl-6,7,8,9-tetrahydro-pyrido[1,2-a]pyrimidin-4-one
Show/Hide
|
C23H27FN4O2
|
1
|
| 1 |
Ki = 224 nM
|
|
|
|
CP0542115
|
1-Benzenesulfonyl-3-(1-benzyl-1,2,3,6-tetrahydro-pyridin-4-yl)-1H-indole
Show/Hide
|
C26H24N2O2S
|
1
|
| 1 |
Ki = 246 nM
|
|
|
|
CP0453190
|
9-Benzenesulfonyl-2,3,4,9-tetrahydro-1H-beta-carboline
Show/Hide
|
C17H16N2O2S
|
1
|
| 1 |
Ki = 252.7 nM
|
|
|
|
CP0500723
|
3-cyclohexyl-6-(3-methoxyphenylsulfonyl)-1,2,3,4,5,6-hexahydroazepino[4,5-b]indole
Show/Hide
|
C25H30N2O3S
|
1
|
| 1 |
Ki = 253 nM
|
|
|
|
CP0514846
|
[4-[2-(dimethylamino)ethyl]-1H-indol-2-yl]-phenylmethanone
Show/Hide
|
C19H20N2O
|
1
|
| 1 |
Ki = 260 nM
|
|
|
|
CP0399783
|
9-(Toluene-4-sulfonyl)-2,3,4,9-tetrahydro-1H-beta-carboline
Show/Hide
|
C18H18N2O2S
|
1
|
| 1 |
Ki = 271.3 nM
|
|
|
|
CP0476065
|
1-(5-Chloro-3-methyl-benzo[b]thiophene-2-sulfonyl)-3-(R)-1-pyrrolidin-2-ylmethyl-1H-indole
Show/Hide
|
C22H21ClN2O2S2
|
1
|
| 1 |
Ki = 283.7 nM
|
|
|
|
CP0502909
|
7-(3-Trifluoromethyl-phenylsulfanyl)-1,2,3,4,10,10a-hexahydro-pyrazino[1,2-a]indole
Show/Hide
|
C18H17F3N2S
|
1
|
| 1 |
Ki = 300 nM
|
|
|
|
CP0392698
|
2-[1-(benzenesulfonyl)-5-phenylmethoxyindol-3-yl]-N,N-dimethylethanamine
Show/Hide
|
C25H26N2O3S
|
1
|
| 1 |
Ki = 320 nM
|
|
|
|
CP0493602
|
3-cyclopentyl-6-(3-methoxyphenylsulfonyl)-1,2,3,4,5,6-hexahydroazepino[4,5-b]indole
Show/Hide
|
C24H28N2O3S
|
1
|
| 1 |
Ki = 324 nM
|
|
|
|
CP0374984
|
7-(2-Trifluoromethyl-phenylsulfanyl)-1,2,3,4,10,10a-hexahydro-pyrazino[1,2-a]indole
Show/Hide
|
C18H17F3N2S
|
1
|
| 1 |
Ki = 330 nM
|
|
|
|
CP0437406
|
1-Benzenesulfonyl-5-methoxy-3-(2-piperidin-1-yl-ethyl)-1H-indole
Show/Hide
|
C22H26N2O3S
|
1
|
| 1 |
Ki = 350 nM
|
|
|
|
CP0414985
|
2-[3-(benzenesulfonyl)pyrrolo[3,2-b]pyridin-1-yl]-N,N-dimethylethanamine
Show/Hide
|
C17H19N3O2S
|
1
|
| 1 |
Ki = 368 nM
|
|
|
|
CP0535322
|
3-(2-Dimethylamino-ethyl)-5-hydroxy-indole-1-carboxylic acid tert-butyl ester
Show/Hide
|
C17H24N2O3
|
1
|
| 1 |
Ki = 370 nM
|
|
|
|
CP0321822
|
4-(benzenesulfonyl)-11-methyl-5-methylsulfanyl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1,3,5,8-tetraene
Show/Hide
|
C17H18N4O2S2
|
1
|
| 1 |
Ki = 372 nM
|
|
|
|
CP0417789
|
3-(phenylsulfonyl)-1H-indole, 18i
Show/Hide
|
C21H24N2O2S
|
1
|
| 1 |
Ki = 434 nM
|
|
|
|
CP0388359
|
N-[3-[(5-chloro-6-oxo-4-piperazin-1-ylpyridazin-1-yl)methyl]phenyl]-4-phenylbenzamide
Show/Hide
|
C28H26ClN5O2
|
1
|
| 1 |
Ki = 489.78 nM
|
|
|
|
CP0464599
|
1-Benzenesulfonyl-5-methoxy-3-[2-(4-methyl-piperazin-1-yl)-ethyl]-1H-indole
Show/Hide
|
C22H27N3O3S
|
1
|
| 1 |
Ki = 490 nM
|
|
|
|
CP0399193
|
6-(3-methoxyphenylsulfonyl)-3-phenethyl-1,2,3,4,5,6-hexahydroazepino[4,5-b]indole
Show/Hide
|
C27H28N2O3S
|
1
|
| 1 |
Ki = 504 nM
|
|
|
|
CP0042927
|
7-{4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butoxy}-3,4-dihydroquinolin-2(1H)-one
Show/Hide
|
C23H27Cl2N3O2
|
1
|
| 1 |
Ki = 574 nM
|
|
|
|
CP0562565
|
N,N-dimethyl-2-(1-methylsulfonylindol-3-yl)ethanamine
Show/Hide
|
C13H18N2O2S
|
1
|
| 1 |
Ki = 620 nM
|
|
|
|
CP0505191
|
7-(4-Trifluoromethyl-phenylsulfanyl)-1,2,3,4,10,10a-hexahydro-pyrazino[1,2-a]indole
Show/Hide
|
C18H17F3N2S
|
1
|
| 1 |
Ki = 760 nM
|
|
|
|
CP0850005
|
1-Methyl-1H-imidazole-4-sulfonic acid [4-methoxy-3-(4-methyl-piperazin-1-yl)-phenyl]-amide
Show/Hide
|
C16H23N5O3S
|
1
|
| 1 |
Ki = 794.33 nM
|
|
|
|
CP0399906
|
N-[5-[(5-chloro-6-oxo-4-piperazin-1-ylpyridazin-1-yl)methyl]-2-methylphenyl]-4-phenylbenzamide
Show/Hide
|
C29H28ClN5O2
|
1
|
| 1 |
Ki = 831.76 nM
|
|
|
|
CP0099712
|
3-(2-aminoethyl)-1H-indole-5-carboxamide
Show/Hide
|
C11H13N3O
|
1
|
| 1 |
Ki = 1000 nM
|
|
|
|
CP0466992
|
2-(3-benzylsulfonylindol-1-yl)-N,N-dimethylethanamine
Show/Hide
|
C19H22N2O2S
|
1
|
| 1 |
Ki = 1011 nM
|
|
|
|
CP0497701
|
1-Benzenesulfonyl-5-methoxy-3-(2-morpholin-4-yl-ethyl)-1H-indole
Show/Hide
|
C21H24N2O4S
|
1
|
| 1 |
Ki = 1700 nM
|
|
|
|
CP0388360
|
N-[3-[(5-chloro-6-oxo-4-piperazin-1-ylpyridazin-1-yl)methyl]-2-methylphenyl]-4-phenylbenzamide
Show/Hide
|
C29H28ClN5O2
|
1
|
| 1 |
Ki = 3388.44 nM
|
|
|
|
CP0861232
|
3-Cyclopentyl-N-(2-dimethylamino-ethyl)-N-[4'-(phenethylamino-methyl)-biphenyl-4-ylmethyl]-propionamide with di TFA
Show/Hide
|
C38H47F6N3O5
|
1
|
| 1 |
Ki = 3981.07 nM
|
|
|
|
CP0332842
|
6-[[1-[2-(7-chloro-2-methylquinolin-5-yl)oxyethyl]piperidin-4-yl]methyl]-7-fluoro-4H-1,4-benzoxazin-3-one
Show/Hide
|
C26H27ClFN3O3
|
1
|
| 1 |
Ki = 7943.28 nM
|
|
|
|
CP0413897
|
4-(benzenesulfonyl)-5,11-dimethyl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1,3,5,8-tetraene
Show/Hide
|
C17H18N4O2S
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0296883
|
7-fluoro-6-[[1-[2-(7-fluoro-2-methylquinolin-5-yl)oxyethyl]piperidin-4-yl]methyl]-4H-1,4-benzoxazin-3-one
Show/Hide
|
C26H27F2N3O3
|
1
|
| 1 |
Ki < 1000 nM
|
|
|
|
CP0847634
|
(E)-N-[4'-(Phenethylamino-methyl)-biphenyl-4-ylmethyl]-3-phenyl-N-pyridin-3-ylmethyl-acrylamide TFA
Show/Hide
|
C39H36F3N3O3
|
1
|
| 1 |
Ki < 1995.26 nM
|
|
|
|
CP0371948
|
8-fluoro-6-[[1-[2-(7-fluoro-2-methylquinolin-5-yl)oxyethyl]piperidin-4-yl]methyl]-4H-1,4-benzoxazin-3-one
Show/Hide
|
C26H27F2N3O3
|
1
|
| 1 |
Ki < 6309.57 nM
|
|
|
|
CP0853819
|
(E)-N-(2-Dimethylamino-ethyl)-N-[4'-(phenethylamino-methyl)-biphenyl-4-ylmethyl]-3-phenyl-acrylamide TFA
Show/Hide
|
C37H40F3N3O3
|
1
|
| 1 |
Ki < 7943.28 nM
|
|
|
|
CP0035199
|
5-fluoro-6-[[1-[2-(7-fluoro-2-methylquinolin-5-yl)oxyethyl]piperidin-4-yl]methyl]-4H-1,4-benzoxazin-3-one
Show/Hide
|
C26H27F2N3O3
|
1
|
| 1 |
Ki < 10000 nM
|
|
|
|
CP0152118
|
6-[[1-[2-(2-methylquinolin-5-yl)oxyethyl]piperidin-4-yl]methyl]-4H-1,4-benzoxazin-3-one
Show/Hide
|
C26H29N3O3
|
1
|
| 1 |
Ki < 10000 nM
|
|
|
|
CP0295528
|
6-[[1-[2-(7-chloro-2-methylquinolin-5-yl)oxyethyl]piperidin-4-yl]methyl]-5-fluoro-4H-1,4-benzoxazin-3-one
Show/Hide
|
C26H27ClFN3O3
|
1
|
| 1 |
Ki < 10000 nM
|
|
|
|
CP0332841
|
6-[[1-[2-(7-chloro-2-methylquinolin-5-yl)oxyethyl]piperidin-4-yl]methyl]-8-fluoro-4H-1,4-benzoxazin-3-one
Show/Hide
|
C26H27ClFN3O3
|
1
|
| 1 |
Ki < 10000 nM
|
|
|
|
CP0156235
|
3,N-Dimethyl-N-[(R)-1-methyl-3-(4-methyl-piperidin-1-yl)-propyl]-benzenesulfonamide
Show/Hide
|
C18H30N2O2S
|
1
|
| 1 |
Ki < 15848.93 nM
|
|
|
