Brief Information of the Compound and Protein
Compound Name
2-{1-[(5-chlorothiophene-2-)sulfonyl]-1H-indol-3-yl}ethan-1-amine
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PubChem ID
CID: 23655468
SID: 46527774
Canonical SMILES
NCCc1cn(c2ccccc12)S(=O)(=O)c1ccc(Cl)s1
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Compound Formula C14H13ClN2O2S2
Compound Structure
Protein Name
5-hydroxytryptamine receptor 6
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Monoamine receptor
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Serotonin receptor
Uniprot ID
P50406
Gene Name
HTR6
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000017 HeLa Homo sapiens (Human)  2
1
EC50 = 181 nM
   TI
   LI
   LO
   TS
2
Ki = 6 nM
   TI
   LI
   LO
   TS