Brief Information of the Compound and Protein
Compound Name
3-chloro-2-methyl-N-[6-(4-methylphenyl)-7-oxo-4,5-dihydro-1H-pyrazolo[3,4-c]pyridin-3-yl]benzenesulfonamide
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PubChem ID
CID: 71813838
Canonical SMILES
Cc1ccc(cc1)N1CCc2c(NS(=O)(=O)c3cccc(Cl)c3C)n[nH]c2C1=O
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Compound Formula C20H19ClN4O3S
Compound Structure
Protein Name
5-hydroxytryptamine receptor 6
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Monoamine receptor
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Serotonin receptor
Uniprot ID
P50406
Gene Name
HTR6
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000017 HeLa Homo sapiens (Human)  1
1
IC50 = 1660 nM
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