Brief Information of the Compound and Protein
Compound Name
5-Chloro-3-methyl-benzo[b]thiophene-2-sulfonic acid [3-((S)-1-methyl-pyrrolidin-2-ylmethyl)-1H-indol-5-yl]-amide
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PubChem ID
CID: 11282884
SID: 16369824
Canonical SMILES
Cc1c(S(=O)(=O)Nc2ccc3[nH]cc(C[C@@H]4CCCN4C)c3c2)sc2ccc(Cl)cc12
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Compound Formula C23H24ClN3O2S2
Compound Structure
Protein Name
5-hydroxytryptamine receptor 6
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Monoamine receptor
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Serotonin receptor
Uniprot ID
P50406
Gene Name
HTR6
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000017 HeLa Homo sapiens (Human)  2
1
IC50 = 1.1 nM
   TI
   LI
   LO
   TS
2
Ki = 2 nM
   TI
   LI
   LO
   TS