General Information of the Cell Line
Cell Line ID
CL000111
Cell Line Name
MDA-MB-231
Synonyms
MDA_MB_231
MDA-MB 231
MDA.MB.231
MDA MB 231
MDA MB231
MDA Mb231
MDA-MB231
MDAMB-231
MDAMB231
MDA-231
MDA-231P
MDA231
MDA231-BRE
MB231
MD Anderson-Metastatic Breast-231
Category
Cancer cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_0062
Tissue Information
Pleural effusion
Disease
Breast adenocarcinoma (NCIt: C5214)
Map of Molecular Bioactivity Related to the Cell Line
Map of Molecular Bioactivity Related to the Cell Line

Cell Line
Protein
Compound

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Cell Line
Protein ID: PT03381, 5'-nucleotidase
 Protein Info 
Compound ID Compound Name Compound Formula
CP0143939
 Compound Info 
[[(2R,3S,4R,5R)-5-(6-amino-2-iodopurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl]methylphosphonic acid
   Show/Hide
C11H16IN5O9P2
  1
1
Ki = 3.33 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0357536
 Compound Info 
[[(2R,3S,4R,5R)-5-(5-fluoro-2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl]methylphosphonic acid
   Show/Hide
C10H15FN2O11P2
  1
1
Ki = 4.51 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0135871
 Compound Info 
[[(2R,3S,4R,5R)-5-(6-amino-2-chloropurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl]methylphosphonic acid
   Show/Hide
C11H16ClN5O9P2
  1
1
Ki = 4.57 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0479758
 Compound Info 
[[(2R,3S,4R,5R)-5-(4-benzamido-2-oxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl]methylphosphonic acid
   Show/Hide
C17H21N3O11P2
  1
1
Ki = 5.68 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0535394
 Compound Info 
[[(2R,3S,4R,5R)-3,4-dihydroxy-5-[4-(naphthalen-2-ylmethoxyamino)-2-oxopyrimidin-1-yl]oxolan-2-yl]methoxy-hydroxyphosphoryl]methylphosphonic acid
   Show/Hide
C21H25N3O11P2
  1
1
Ki = 6.29 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0064631
 Compound Info 
[[(2R,3S,4R,5R)-3,4-dihydroxy-5-[(4E)-3-methyl-2-oxo-4-phenylmethoxyiminopyrimidin-1-yl]oxolan-2-yl]methoxy-hydroxyphosphoryl]methylphosphonic acid
   Show/Hide
C18H25N3O11P2
  1
1
Ki = 7.96 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0434811
 Compound Info 
[hydroxy-[[(2R,3S,5R)-3-hydroxy-5-[2-oxo-4-[[4-(trifluoromethyl)phenyl]methoxyamino]pyrimidin-1-yl]oxolan-2-yl]methoxy]phosphoryl]methylphosphonic acid
   Show/Hide
C18H22F3N3O10P2
  1
1
Ki = 10.1 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0488030
 Compound Info 
[[(2R,3S,4R,5R)-5-(6-amino-2-hydrazinylpurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl]methylphosphonic acid
   Show/Hide
C11H19N7O9P2
  1
1
Ki = 15.4 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0434795
 Compound Info 
[[(2R,3S,4R,5R)-5-[5-fluoro-2-oxo-4-(phenylmethoxyamino)pyrimidin-1-yl]-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl]methylphosphonic acid
   Show/Hide
C17H22FN3O11P2
  1
1
Ki = 16.6 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0368770
 Compound Info 
[[(2R,3S,4R,5R)-5-(2-amino-6-chloropurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl]methylphosphonic acid
   Show/Hide
C11H16ClN5O9P2
  1
1
Ki = 32.2 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0426686
 Compound Info 
[[(2R,3S,4R,5R)-5-(2,6-diaminopurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl]methylphosphonic acid
   Show/Hide
C11H18N6O9P2
  1
1
Ki = 35.7 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0064281
 Compound Info 
[[(2R,3S,4R,5R)-5-[6-amino-2-(2-cyclohexylethylsulfanyl)purin-9-yl]-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl]methylphosphonic acid
   Show/Hide
C19H31N5O9P2S
  1
1
Ki = 49.1 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0440395
 Compound Info 
[[(2R,3S,4R,5R)-5-(6-amino-2-prop-2-enylsulfanylpurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl]methylphosphonic acid
   Show/Hide
C14H21N5O9P2S
  1
1
Ki = 65.4 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0136183
 Compound Info 
ADP, alpha beta-me
   Show/Hide
C11H17N5O9P2
  1
1
Ki = 207 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0483092
 Compound Info 
[[(2R,3S,4R,5R)-5-(6-amino-2-piperazin-1-ylpurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl]methylphosphonic acid
   Show/Hide
C15H25N7O9P2
  1
1
Ki = 238 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0240255
 Compound Info 
PHOSPHOMETHYLPHOSPHONIC ACID GUANOSYL ESTER
   Show/Hide
C11H17N5O10P2
  1
1
Ki = 255 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
Protein ID: PT00894, Androgen receptor
 Protein Info 
Protein ID: PT01786, Autotaxin
 Protein Info 
Protein ID: PT07141, B-cell lymphoma 3 protein
 Protein Info 
Protein ID: PT01191, Baculoviral IAP repeat-containing protein 2
 Protein Info 
Protein ID: PT02379, Bifunctional purine biosynthesis protein ATIC
 Protein Info 
Protein ID: PT00818, CaM kinase I delta
 Protein Info 
Protein ID: PT00985, Cell division cycle 7-related protein kinase
 Protein Info 
Protein ID: PT01771, E3 ubiquitin-protein ligase Mdm2
 Protein Info 
Protein ID: PT00922, Epidermal growth factor receptor
 Protein Info 
Protein ID: PT00889, Estrogen receptor beta
 Protein Info 
Protein ID: PT02717, Eukaryotic initiation factor 4A-I
 Protein Info 
Protein ID: PT05453, G-protein coupled receptor 55
 Protein Info 
Protein ID: PT00947, Geranylgeranyl pyrophosphate synthase
 Protein Info 
Protein ID: PT01566, Histone-lysine N-methyltransferase EHMT2
 Protein Info 
Protein ID: PT01557, Indoleamine 2,3-dioxygenase 1
 Protein Info 
Protein ID: PT06082, Integrin alpha-3
 Protein Info 
Protein ID: PT02653, N-lysine methyltransferase SMYD2
 Protein Info 
Protein ID: PT01871, Proteinase-activated receptor 1
 Protein Info 
Protein ID: PT04124, Proteinase-activated receptor 2
 Protein Info 
Protein ID: PT00879, Proto-oncogene tyrosine-protein kinase Src
 Protein Info 
Protein ID: PT06122, Retinoblastoma-associated protein
 Protein Info 
Protein ID: PT01033, Serine/threonine protein kinase PIK3CB
 Protein Info 
Protein ID: PT01065, Serine/threonine-protein kinase mTOR
 Protein Info 
Protein ID: PT01503, Signal transducer and activator of transcription 3
 Protein Info 
Protein ID: PT01466, Telomerase reverse transcriptase
 Protein Info 
Protein ID: PT06229, Transmembrane protein 142A
 Protein Info 
Cell Viability or Cytotoxicity Assay
Compound ID Compound Name Compound Formula
CP0001056
 Compound Info 
N-hydroxy-7-[3-[4-[[(7-hydroxy-21-methyl-14-oxo-3,13,21-triazapentacyclo[11.8.0.02,10.04,9.015,20]henicosa-2(10),4(9),5,7,15(20),16,18-heptaen-17-yl)amino]methyl]phenyl]-1,2,4-oxadiazol-5-yl]heptanamide
   Show/Hide
 C35H37N7O5  1
1
IC50 = 2300 nM
   TI
   LI
   LO
   TS
CP0001881
 Compound Info 
N-(2-aminophenyl)-4-[[4-[4-(pyridin-3-ylmethylcarbamoyl)phenyl]triazol-1-yl]methyl]benzamide
   Show/Hide
 C29H25N7O2  1
1
IC50 = 10000 nM
   TI
   LI
   LO
   TS
CP0002211
 Compound Info 
N-[2-(diethylamino)ethyl]-5-[(Z)-(5-fluoro-2-oxo-1H-indol-3-ylidene)methyl]-2,4-dimethyl-1H-pyrrole-3-carboxamide
   Show/Hide
 C22H27FN4O2  1
1
IC50 = 22.3 nM
   TI
   LI
   LO
   TS
CP0002778
 Compound Info 
4-[(4-methylpiperazin-1-yl)methyl]-N-[4-methyl-3-[(4-pyridin-3-ylpyrimidin-2-yl)amino]phenyl]benzamide
   Show/Hide
 C29H31N7O  1
1
IC50 = 39810.72 nM
   TI
   LI
   LO
   TS
CP0003147
 Compound Info 
ethyl 6-[5-(benzenesulfonamido)pyridin-3-yl]imidazo[1,2-a]pyridine-3-carboxylate
   Show/Hide
 C21H18N4O4S  1
1
IC50 = 760 nM
   TI
   LI
   LO
   TS
CP0003424
 Compound Info 
N-[4-(1,4-diazepan-1-ylsulfonyl)phenyl]-1,3-dimethylpyrazolo[4,3-e][1,2,4]triazin-5-amine
   Show/Hide
 C17H22N8O2S  2
1
IC50 = 150000 nM
   TI
   LI
   LO
   TS
2
IC50 = 155000 nM
   TI
   LI
   LO
   TS
CP0003832
 Compound Info 
N'-hydroxy-N-phenyloctanediamide
   Show/Hide
 C14H20N2O3  7
1
IC50 = 610 nM
   TI
   LI
   LO
   TS
2
IC50 = 1110 nM
   TI
   LI
   LO
   TS
3
IC50 = 1710 nM
   TI
   LI
   LO
   TS
4
IC50 = 1730 nM
   TI
   LI
   LO
   TS
5
IC50 = 1980 nM
   TI
   LI
   LO
   TS
6
IC50 = 2200 nM
   TI
   LI
   LO
   TS
7
IC50 = 7400 nM
   TI
   LI
   LO
   TS
CP0004959
 Compound Info 
S-[(E)-4-[(5R,8S,11S)-5-methyl-6,9,13-trioxo-8-propan-2-yl-10-oxa-3,17-dithia-7,14,19,20-tetrazatricyclo[14.2.1.12,5]icosa-1(18),2(20),16(19)-trien-11-yl]but-3-enyl] octanethioate
   Show/Hide
 C29H42N4O5S3  1
1
IC50 = 4750 nM
   TI
   LI
   LO
   TS
CP0005409
 Compound Info 
1,3-dimethyl-N-(4-morpholin-4-ylsulfonylphenyl)pyrazolo[4,3-e][1,2,4]triazin-5-amine
   Show/Hide
 C16H19N7O3S  1
1
IC50 > 200000 nM
   TI
   LI
   LO
   TS
CP0006391
 Compound Info 
3-[(3-anilino-3-oxopropyl)-octylamino]-N-phenylpropanamide
   Show/Hide
 C26H37N3O2  1
1
IC50 = 5000 nM
   TI
   LI
   LO
   TS
CP0007167
 Compound Info 
4-[(1,3-dimethylpyrazolo[4,3-e][1,2,4]triazin-5-yl)amino]-N-(2-morpholin-4-ylethyl)benzenesulfonamide
   Show/Hide
 C18H24N8O3S  1
1
IC50 = 120000 nM
   TI
   LI
   LO
   TS
CP0007711
 Compound Info 
(E)-3-[4-[[2-(2-methyl-1H-indol-3-yl)ethylamino]methyl]phenyl]-N'-propylprop-2-enehydrazide;2,2,2-trifluoroacetic acid
   Show/Hide
 C26H31F3N4O3  1
1
LC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0010389
 Compound Info 
6-[4-[5,7-dimethoxy-4-(4-methylpiperazin-1-yl)quinazolin-2-yl]-2,6-dimethylphenoxy]-N-hydroxyhexanamide
   Show/Hide
 C29H39N5O5  1
1
IC50 = 1323 nM
   TI
   LI
   LO
   TS
CP0010390
 Compound Info 
6-[4-[4-(1,1-dioxo-1,4-thiazinan-4-yl)-5,7-dimethoxyquinazolin-2-yl]-2,6-dimethylphenoxy]-N-hydroxyhexanamide
   Show/Hide
 C28H36N4O7S  1
1
IC50 = 1335 nM
   TI
   LI
   LO
   TS
CP0012103
 Compound Info 
6-[5-[(2,4-difluorophenyl)sulfonylamino]-6-methoxypyridin-3-yl]-N-(3-morpholin-4-ylpropyl)imidazo[1,2-a]pyridine-3-carboxamide
   Show/Hide
 C27H28F2N6O5S  1
1
IC50 = 300 nM
   TI
   LI
   LO
   TS
CP0015576
 Compound Info 
N-(6-chloro-9H-pyrido[3,4-b]indol-8-yl)pyridine-3-carboxamide
   Show/Hide
 C17H11ClN4O  1
1
IC50 = 900 nM
   TI
   LI
   LO
   TS
CP0019439
 Compound Info 
8-[3-(1-benzofuran-2-yl)-5-chloropyridin-4-yl]-2,8-diazaspiro[4.5]decan-1-one
   Show/Hide
 C21H20ClN3O2  1
1
GI50 = 40710 nM
   TI
   LI
   LO
   TS
CP0036258
 Compound Info 
5-(2,6-difluoroanilino)-N-methylbenzo[c][2,6]naphthyridine-7-carboxamide
   Show/Hide
 C20H14F2N4O  1
1
EC50 = 590 nM
   TI
   LI
   LO
   TS
CP0037780
 Compound Info 
(2S)-2-[(2S,3R)-3-amino-2-hydroxy-4-phenylbutanamido]-4-methylpentanoic acid
   Show/Hide
 C16H24N2O4  2
1
IC50 = 753180 nM
   TI
   LI
   LO
   TS
2
IC50 = 5080000 nM
   TI
   LI
   LO
   TS
CP0040710
 Compound Info 
6-Methoxy-2-(4-methyl-1,4-diazepan-1-yl)-N-(1-methylpiperidin-4-yl)-7-(3-(piperidin-1-yl)propoxy)quinazolin-4-amine
   Show/Hide
 C29H47N7O2  1
1
EC50 = 12000 nM
   TI
   LI
   LO
   TS
CP0042443
 Compound Info 
(S)-1-(5-phenyl-3-(piperidin-3-ylcarbamoyl)thiophen-2-yl)urea
   Show/Hide
 C17H20N4O2S  1
1
GI50 = 596 nM
   TI
   LI
   LO
   TS
CP0044060
 Compound Info 
4-{[(7R)-8-cyclopentyl-7-ethyl-5-methyl-6-oxo-5,6,7,8-tetrahydropteridin-2-yl]amino}-3-methoxy-N-(1-methylpiperidin-4-yl)benzamide
   Show/Hide
 C28H39N7O3  1
1
IC50 = 1 nM
   TI
   LI
   LO
   TS
CP0046554
 Compound Info 
6-[difluoro-[6-(4-fluorophenyl)-[1,2,4]triazolo[4,3-b][1,2,4]triazin-3-yl]methyl]quinoline
   Show/Hide
 C20H11F3N6  1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0046759
 Compound Info 
N-[3-fluoro-4-[2-(1-methylimidazol-4-yl)thieno[3,2-b]pyridin-7-yl]oxyphenyl]-1-phenyl-5-(trifluoromethyl)pyrazole-4-carboxamide
   Show/Hide
 C28H18F4N6O2S  1
1
IC50 = 100 nM
   TI
   LI
   LO
   TS
CP0051683
 Compound Info 
(8S,11S,14S,17S,29S,32S,35S,38S)-10,31-bis[(2S)-3,3-dimethyl-2-[[(2S)-2-(methylamino)propanoyl]amino]butanoyl]-14,35-bis(naphthalen-2-ylmethyl)-12,15,33,36-tetraoxo-2,23-dioxa-5,6,7,10,13,16,26,27,28,31,34,37-dodecazaheptacyclo[38.2.2.219,22.14,7.18,11.125,28.129,32]pentaconta-1(43),4(50),5,19,21,25(46),26,40(44),41,47-decaene-17,38-dicarboxylic acid
   Show/Hide
 C80H96N16O14  1
1
IC50 = 26 nM
   TI
   LI
   LO
   TS
CP0052426
 Compound Info 
(2E)-3-{4-[3-(adamantan-1-yl)-4-hydroxyphenyl]-3-chlorophenyl}prop-2-enoic acid
   Show/Hide
 C25H25ClO3  1
1
IC50 = 950 nM
   TI
   LI
   LO
   TS
CP0055412
 Compound Info 
3-((1H-Indazol-3-yl)ethynyl)aniline
   Show/Hide
 C15H11N3  1
1
GI50 = 8290 nM
   TI
   LI
   LO
   TS
CP0064592
 Compound Info 
[(1S,2S,3R,4S,7R,9S,10S,12R,15S)-4,12-diacetyloxy-15-[(2R,3S)-3-benzamido-2-hydroxy-3-phenylpropanoyl]oxy-1,9-dihydroxy-10,14,17,17-tetramethyl-11-oxo-6-oxatetracyclo[11.3.1.03,10.04,7]heptadec-13-en-2-yl] benzoate
   Show/Hide
 C47H51NO14  1
1
GI50 = 12.5 nM
   TI
   LI
   LO
   TS
CP0068848
 Compound Info 
(5S,8S,10aR)-N-benzhydryl-5-[[(2S)-2-(methylamino)propanoyl]amino]-3-(3-methylbutanoyl)-6-oxo-1,2,4,5,8,9,10,10a-octahydropyrrolo[1,2-a][1,5]diazocine-8-carboxamide
   Show/Hide
 C32H43N5O4  1
1
EC50 = 19 nM
   TI
   LI
   LO
   TS
CP0069223
 Compound Info 
4-[4-chloro-3-(trifluoromethyl)phenyl]-1-[3-(4-fluoro-N-(4-fluorophenyl)anilino)propyl]piperidin-4-ol
   Show/Hide
 C27H26ClF5N2O  1
1
IC50 = 3500 nM
   TI
   LI
   LO
   TS
CP0074041
 Compound Info 
3-(2-chloro-4-hydroxyphenyl)-4-ethyl-7-hydroxychromen-2-one
   Show/Hide
 C17H13ClO4  1
1
IC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0075279
 Compound Info 
5-(2-chloroanilino)-N-ethylbenzo[c][2,6]naphthyridine-7-carboxamide
   Show/Hide
 C21H17ClN4O  1
1
EC50 = 2120 nM
   TI
   LI
   LO
   TS
CP0082560
 Compound Info 
4-[4-chloro-3-(trifluoromethyl)phenyl]-1-(4,4-diphenylbutyl)piperidin-4-ol
   Show/Hide
 C28H29ClF3NO  1
1
IC50 = 9300 nM
   TI
   LI
   LO
   TS
CP0089066
 Compound Info 
(8S,11S,14S,17S,29S,32S,35S,38S)-10,31-bis[(2S)-2-cyclohexyl-2-[[(2S)-2-(methylamino)propanoyl]amino]acetyl]-14,35-bis(naphthalen-2-ylmethyl)-12,15,33,36-tetraoxo-2,23-dioxa-5,6,7,10,13,16,26,27,28,31,34,37-dodecazaheptacyclo[38.2.2.219,22.14,7.18,11.125,28.129,32]pentaconta-1(43),4(50),5,19,21,25(46),26,40(44),41,47-decaene-17,38-dicarboxylic acid
   Show/Hide
 C84H100N16O14  1
1
IC50 = 14 nM
   TI
   LI
   LO
   TS
CP0091315
 Compound Info 
US9422297, AAG145-136
   Show/Hide
 C17H13ClN4  1
1
GI50 = 641 nM
   TI
   LI
   LO
   TS
CP0092308
 Compound Info 
4-[2-amino-5-[4-[(dimethylamino)methyl]thiophen-2-yl]pyridin-3-yl]-2-[(Z,2R)-5,5,5-trifluoropent-3-en-2-yl]oxybenzamide
   Show/Hide
 C24H25F3N4O2S  1
1
GI50 = 4160 nM
   TI
   LI
   LO
   TS
CP0107901
 Compound Info 
6-[4-[4-[[2-[4-[(Z)-1,2-diphenylbut-1-enyl]phenoxy]ethyl-methylamino]methyl]phenyl]triazol-1-yl]-N-hydroxyhexanamide
   Show/Hide
 C40H45N5O3  1
1
IC50 = 10000 nM
   TI
   LI
   LO
   TS
CP0112599
 Compound Info 
US8569511, 2
   Show/Hide
 C23H22F2N6O2  1
1
IC50 = 3540 nM
   TI
   LI
   LO
   TS
CP0114044
 Compound Info 
4-[2-amino-5-[4-[(dimethylamino)methyl]thiophen-2-yl]pyridin-3-yl]-2-[(1R)-1-[2-(trifluoromethyl)phenyl]ethoxy]benzamide
   Show/Hide
 C28H27F3N4O2S  1
1
GI50 = 950 nM
   TI
   LI
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   TS
CP0118102
 Compound Info 
methyl (1R,2R,3S,3aR,8bS)-6-[[(2S,3R,6R)-6-[(1R)-1,2-dihydroxyethyl]-3-methoxy-1,4-dioxan-2-yl]oxy]-1,8b-dihydroxy-8-methoxy-3a-(4-methoxyphenyl)-3-phenyl-2,3-dihydro-1H-cyclopenta[b][1]benzofuran-2-carboxylate
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 C34H38O13  1
1
EC50 = 3 nM
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CP0120515
 Compound Info 
4-({3-[(4-cyclopropanecarbonylpiperazin-1-yl)carbonyl]-4-fluorophenyl}methyl)-1,2-dihydrophthalazin-1-one
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 C24H23FN4O3  3
1
IC50 = 7920 nM
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2
IC50 = 39510 nM
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3
IC50 > 40000 nM
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CP0124520
 Compound Info 
(1S,5S,6R,9S,15E,20R)-5-hydroxy-20-(2-methylsulfanylethyl)-6-propan-2-yl-2-oxa-11,12-dithia-7,19,22-triazabicyclo[7.7.6]docos-15-ene-3,8,18,21-tetrone
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 C22H35N3O6S3  1
1
GI50 = 1.8 nM
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CP0126431
 Compound Info 
US8629141, 21
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 C24H24Cl2FN3O2  2
1
IC50 > 10 nM
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2
IC50 > 3000 nM
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CP0127814
 Compound Info 
N-[4-(hydroxycarbamoyl)phenyl]-4-naphthalen-2-yloxane-4-carboxamide
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 C23H22N2O4  1
1
IC50 = 100 nM
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CP0137418
 Compound Info 
N-[4-[2-(1-ethylimidazol-4-yl)thieno[3,2-b]pyridin-7-yl]oxy-3-fluorophenyl]-3-(4-fluorophenyl)-2-oxoimidazolidine-1-carboxamide
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 C28H22F2N6O3S  1
1
IC50 = 20000 nM
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CP0151685
 Compound Info 
N-(2-aminophenyl)-4-[[4-methyl-3-[(4-pyridin-3-ylpyrimidin-2-yl)amino]anilino]methyl]benzamide
   Show/Hide
 C30H27N7O  1
1
IC50 = 10000 nM
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CP0152361
 Compound Info 
3-chloro-4-[[7-(1H-1,2,4-triazol-5-yl)benzo[c][2,6]naphthyridin-5-yl]amino]phenol
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 C20H13ClN6O  1
1
EC50 = 2380 nM
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CP0154285
 Compound Info 
1-[5,5-bis(4-fluorophenyl)pent-4-enyl]-4-[4-chloro-3-(trifluoromethyl)phenyl]piperidin-4-ol
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 C29H27ClF5NO  2
1
IC50 = 14900 nM
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2
IC50 = 23900 nM
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CP0160473
 Compound Info 
2-(4-(2-(1H-pyrazol-3-ylamino)-1H-benzo[d]imidazol-1-yl)-6-methyl-1,3,5-triazin-2-ylamino)acetonitrile
   Show/Hide
 C16H14N10  1
1
IC50 = 270 nM
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CP0163043
 Compound Info 
4-((1H-Indazol-3-yl)ethynyl)aniline
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 C15H11N3  1
1
GI50 = 8280 nM
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CP0166875
 Compound Info 
(2E)-3-{4-[3-(adamantan-1-yl)-4-fluorophenyl]-3-chlorophenyl}prop-2-enoic acid
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 C25H24ClFO2  1
1
IC50 = 67000 nM
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CP0168317
 Compound Info 
1-(4,4-bis(4-fluorophenyl)butyl)-4-(4-chloro-3-(trifluoromethyl)phenyl)piperidin-4-ol
   Show/Hide
 C28H27ClF5NO  1
1
IC50 = 5100 nM
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CP0176598
 Compound Info 
N-[4-[2-[(2S,3S,5R)-2-[[tert-butyl(dimethyl)silyl]oxymethyl]-5-(5-methyl-2,4-dioxopyrimidin-1-yl)oxolan-3-yl]-1,3-dithian-2-yl]phenyl]-N'-hydroxyoctanediamide
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 C34H52N4O7S2Si  1
1
GI50 = 2511.89 nM
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CP0198449
 Compound Info 
4-[4-chloro-3-(trifluoromethyl)phenyl]-1-[5-(4-fluorophenyl)pentyl]piperidin-4-ol
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 C23H26ClF4NO  1
1
IC50 = 9800 nM
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CP0198450
 Compound Info 
1-[5,5-bis(4-fluorophenyl)pentyl]-4-[4-chloro-3-(trifluoromethyl)phenyl]piperidin-4-ol
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 C29H29ClF5NO  2
1
IC50 = 5300 nM
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2
IC50 = 5700 nM
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CP0202831
 Compound Info 
4-[4-chloro-3-(trifluoromethyl)phenyl]-1-[4-(4-methoxy-N-(4-methoxyphenyl)anilino)butyl]piperidin-4-ol
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 C30H34ClF3N2O3  2
1
IC50 = 5400 nM
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2
IC50 = 7100 nM
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CP0206772
 Compound Info 
(2E)-3-{3-chloro-4-[3-(3,5-dimethyladamantan-1-yl)-4-hydroxyphenyl]phenyl}prop-2-enoic acid
   Show/Hide
 C27H29ClO3  1
1
IC50 > 5000 nM
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CP0224657
 Compound Info 
(3,5-dichlorophenyl)methyl 4-[3-oxo-3-(2-oxo-3H-1,3-benzoxazol-6-yl)propyl]piperazine-1-carboxylate
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 C22H21Cl2N3O5  1
1
IC50 = 4170 nM
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CP0228522
 Compound Info 
4-[[4-[2-fluoro-5-[(4-oxo-3H-phthalazin-1-yl)methyl]benzoyl]piperazin-1-yl]methyl]-N-hydroxybenzamide
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 C28H26FN5O4  1
1
IC50 = 18290 nM
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CP0229896
 Compound Info 
(E)-3-[4-[[4-[2-fluoro-5-[(4-oxo-3H-phthalazin-1-yl)methyl]benzoyl]piperazin-1-yl]methyl]phenyl]-N-hydroxyprop-2-enamide
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 C30H28FN5O4  2
1
IC50 = 940 nM
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2
IC50 = 2680 nM
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CP0229968
 Compound Info 
[1-(2,4-difluoro-5-hydroxybenzoyl)piperidin-4-yl]-(4-phenylsulfanylphenyl)methanone
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 C25H21F2NO3S  1
1
IC50 = 63000 nM
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CP0230298
 Compound Info 
(2S)-1-[(2S)-3,3-dimethyl-2-[[(2S)-2-(methylamino)propanoyl]amino]butanoyl]-N-[(1S,2R)-2-[6-[[(1S,2R)-1-[[(2S)-1-[(2S)-3,3-dimethyl-2-[[(2S)-2-(methylamino)propanoyl]amino]butanoyl]pyrrolidine-2-carbonyl]amino]-2,3-dihydro-1H-inden-2-yl]oxy]hexa-2,4-diynoxy]-2,3-dihydro-1H-inden-1-yl]pyrrolidine-2-carboxamide
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 C54H74N8O8  1
1
GI50 < 2.4 nM
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CP0231485
 Compound Info 
2-[bis(2-methylpropyl)amino]-1-[4-[2-(2,4-dichlorophenyl)-2-(naphthalen-2-ylmethoxy)ethyl]piperazin-1-yl]ethanone
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 C33H43Cl2N3O2  1
1
IC50 = 1660 nM
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CP0231500
 Compound Info 
7-(2-(2-(Dimethylamino)ethoxy)ethoxy)-6-methoxy-2-(4-methyl-1,4-diazepan-1-yl)-N-(1-methylpiperidin-4-yl)quinazolin-4-amine
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 C27H45N7O3  1
1
EC50 > 40000 nM
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CP0236214
 Compound Info 
2-fluoro-N-[2-[4-[(E)-3-(hydroxyamino)-3-oxoprop-1-enyl]phenyl]ethyl]-5-[(4-oxo-3H-phthalazin-1-yl)methyl]benzamide
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 C27H23FN4O4  1
1
IC50 = 220 nM
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CP0241639
 Compound Info 
N-[2-chloro-4-(4-methylpiperazin-1-yl)phenyl]-7-(1H-1,2,4-triazol-5-yl)benzo[c][2,6]naphthyridin-5-amine
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 C25H23ClN8  1
1
EC50 = 2940 nM
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CP0242458
 Compound Info 
N-(1-cyclopropylpiperidin-4-yl)-2-(1,1-dioxo-1,4-thiazinan-4-yl)-6-methoxy-7-(3-pyrrolidin-1-ylpropoxy)quinazolin-4-amine
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 C28H42N6O4S  1
1
EC50 > 50000 nM
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CP0247307
 Compound Info 
(2E)-3-{4-[3-(adamantan-1-yl)-4-acetamidophenyl]-3-chlorophenyl}prop-2-enoic acid
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 C27H28ClNO3  1
1
IC50 > 5000 nM
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CP0247497
 Compound Info 
7-[(6-fluoroquinazolin-4-yl)amino]-N-hydroxyheptanamide
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 C15H19FN4O2  1
1
IC50 = 490 nM
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CP0258426
 Compound Info 
(2S)-1-[(2S)-3,3-dimethyl-2-[[(2S)-2-(methylamino)propanoyl]amino]butanoyl]-N-[(1R,2S)-2-prop-2-ynoxy-1,2,3,4-tetrahydronaphthalen-1-yl]pyrrolidine-2-carboxamide
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 C28H40N4O4  1
1
GI50 = 192 nM
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CP0271917
 Compound Info 
(2R)-N-[(2S,3S)-2-amino-3-hydroxy-3-(4-nitrophenyl)propyl]-2-[[(2S)-3-amino-2-hydroxypropanoyl]amino]-3-phenylpropanamide
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 C21H27N5O6  1
1
IC50 = 4130000 nM
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CP0271918
 Compound Info 
(2S)-2-amino-N-[(2R)-1-[[(2S,3S)-2-amino-3-(4-aminophenyl)-3-hydroxypropyl]amino]-1-oxo-3-phenylpropan-2-yl]-4-methylpentanamide
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 C24H35N5O3  1
1
IC50 = 3650000 nM
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CP0273261
 Compound Info 
2-morpholin-4-yl-1-phenyl-2-sulfanylideneethanone
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 C12H13NO2S  1
1
IC50 > 100000 nM
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CP0283444
 Compound Info 
6-(3-aminophenyl)-3-anilino-2H-isoquinolin-1-one
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 C21H17N3O  1
1
IC50 = 6800 nM
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CP0293714
 Compound Info 
(2S)-N-[(1S)-1-cyclohexyl-2-oxo-2-[[(1R,4S,6S)-2-(2-phenylethyl)-2-azabicyclo[2.2.2]octan-6-yl]amino]ethyl]-2-(methylamino)propanamide
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 C27H42N4O2  1
1
GI50 = 100 nM
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CP0314578
 Compound Info 
4-[4-chloro-3-(trifluoromethyl)phenyl]-1-[4-(4-fluoro-N-(4-fluorophenyl)anilino)butyl]piperidin-4-ol
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 C28H28ClF5N2O  1
1
IC50 = 11300 nM
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CP0327287
 Compound Info 
US9018214, 180
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 C28H37N5O2  1
1
EC50 = 100 nM
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CP0329823
 Compound Info 
2-Acetylfuranonaphthoquinone
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 C14H8O4  1
1
IC50 = 2100 nM
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CP0339039
 Compound Info 
CHEBI:66028
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 C14H10O5  1
1
IC50 = 410 nM
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CP0345034
 Compound Info 
[(2R)-1-(4-tert-butylphenoxy)-3-(2-nitroimidazol-1-yl)propan-2-yl] 4-[(2-hydroxy-5-oxocyclopenta-1,3-dien-1-yl)methylideneamino]benzoate
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 C29H28N4O7  2
1
GI50 = 12000 nM
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2
LC50 = 68000 nM
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CP0350263
 Compound Info 
2-[4-(cyclohexylmethyl)-1,4-diazepan-1-yl]-6-methoxy-N-(1-propan-2-ylpiperidin-4-yl)-7-(3-pyrrolidin-1-ylpropoxy)quinazolin-4-amine
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 C36H59N7O2  1
1
EC50 = 760 nM
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CP0350802
 Compound Info 
(4-benzylphenyl)-[1-(2,4-difluoro-5-hydroxybenzoyl)piperidin-4-yl]methanone
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 C26H23F2NO3  1
1
IC50 = 65000 nM
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CP0354927
 Compound Info 
ethyl 1-[4-[(5-methyl-1H-pyrazol-3-yl)amino]-2-phenylquinazolin-7-yl]piperidine-4-carboxylate
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 C26H28N6O2  1
1
IC50 = 1190 nM
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CP0370065
 Compound Info 
5-(4-chlorophenyl)-2-(4-methoxyphenyl)-[1,3]thiazolo[3,2-b][1,2,4]triazole
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 C17H12ClN3OS  1
1
GI50 = 2060 nM
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CP0373216
 Compound Info 
(2E)-3-{3-chloro-4-[4-hydroxy-3-(1-methylcyclohexyl)phenyl]phenyl}prop-2-enoic acid
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 C22H23ClO3  1
1
IC50 > 5000 nM
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CP0381601
 Compound Info 
(2S)-1-[(2S)-3,3-dimethyl-2-[[(2S)-2-(methylamino)propanoyl]amino]butanoyl]-N-[(1R,2R)-2-[6-[[(1R,2R)-1-[[(2S)-1-[(2S)-3,3-dimethyl-2-[[(2S)-2-(methylamino)propanoyl]amino]butanoyl]pyrrolidine-2-carbonyl]amino]-1,2,3,4-tetrahydronaphthalen-2-yl]oxy]hexa-2,4-diynoxy]-1,2,3,4-tetrahydronaphthalen-1-yl]pyrrolidine-2-carboxamide
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 C56H78N8O8  1
1
GI50 = 61 nM
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CP0383074
 Compound Info 
1,3,10-trichloro-7-(3,5-dichloro-4-hydroxy-2-methoxy-6-methylphenyl)-2,4,6,9-tetrahydroxy-12,12-dimethyltetracen-5-one
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 C28H19Cl5O7  1
1
IC50 > 40000 nM
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CP0383276
 Compound Info 
N-(4-methoxyphenyl)-N,2,6-trimethylfuro[2,3-d]pyrimidin-4-amine
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 C16H17N3O2  1
1
GI50 = 44.3 nM
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CP0384556
 Compound Info 
(2E)-3-{3-chloro-4-[3-(3,3-dimethylbut-1-yn-1-yl)-4-hydroxyphenyl]phenyl}prop-2-enoic acid
   Show/Hide
 C21H19ClO3  1
1
IC50 > 10000 nM
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CP0386603
 Compound Info 
(E)-1-(5-bromo-2-hydroxyphenyl)-3-(2-methoxyphenyl)prop-2-en-1-one
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 C16H13BrO3  1
1
IC50 = 9700 nM
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CP0386673
 Compound Info 
5-[4-[(Z)-1-[4-[2-(dimethylamino)ethoxy]phenyl]-1-(4-hydroxyphenyl)but-1-en-2-yl]phenyl]-N-hydroxypentanamide
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 C31H38N2O4  1
1
IC50 = 1270 nM
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CP0387126
 Compound Info 
4,4-dimethyl-7-(2-methyloctan-2-yl)-1H-chromeno[4,3-c]pyrazole-8,9-dione
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 C21H28N2O3  1
1
IC50 = 8500 nM
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CP0394629
 Compound Info 
4-(3-fluoro-4-hydroxyphenyl)-2-[(E)-N-hydroxy-C-undecylcarbonimidoyl]phenol
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 C24H32FNO3  1
1
IC50 = 45000 nM
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CP0396663
 Compound Info 
2-(1-octyl-5-m-tolyl-1H-indol-3-yl)acetamide
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 C25H32N2O  1
1
IC50 = 21800 nM
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CP0396688
 Compound Info 
[(1R)-1-[[(2S)-2-[(3,4-difluorophenyl)methylcarbamoylamino]-3-phenylpropanoyl]amino]-3-methylbutyl]boronic acid
   Show/Hide
 C22H28BF2N3O4  1
1
IC50 = 28.4 nM
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CP0396691
 Compound Info 
3-(3-fluoro-4-hydroxyphenyl)-7-hydroxychromen-2-one
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 C15H9FO4  1
1
IC50 > 100000 nM
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CP0397385
 Compound Info 
methyl (1R,2R,3S,3aR,8bS)-6-carbamoyl-1,8b-dihydroxy-8-methoxy-3a-(4-methoxyphenyl)-3-phenyl-2,3-dihydro-1H-cyclopenta[b][1]benzofuran-2-carboxylate
   Show/Hide
 C28H27NO8  1
1
EC50 = 80 nM
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CP0397387
 Compound Info 
methyl (1R,2R,3S,3aR,8bS)-6-(dimethylamino)-1,8b-dihydroxy-8-methoxy-3a-(4-methoxyphenyl)-3-phenyl-2,3-dihydro-1H-cyclopenta[b][1]benzofuran-2-carboxylate
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 C29H31NO7  1
1
EC50 > 4000 nM
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CP0397547
 Compound Info 
(2-aminophenyl)-[1-(3-propan-2-ylphenyl)triazol-4-yl]methanone
   Show/Hide
 C18H18N4O  1
1
IC50 = 6900 nM
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CP0402046
 Compound Info 
CHEMBL4449512
   Show/Hide
 C41H42Cl2FN5O5  1
1
IC50 = 39.4 nM
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CP0403368
 Compound Info 
1-benzyl-3-[4-(3-bromoanilino)quinazolin-6-yl]thiourea
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 C22H18BrN5S  1
1
GI50 = 9500 nM
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CP0403677
 Compound Info 
2-(1-octyl-5-o-tolyl-1H-indol-3-yl)acetamide
   Show/Hide
 C25H32N2O  1
1
IC50 = 21200 nM
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CP0407391
 Compound Info 
N-ethyl-N-[(1-octyl-5-pyrimidin-5-ylindol-3-yl)methyl]ethanamine
   Show/Hide
 C25H36N4  1
1
IC50 = 11050 nM
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CP0407392
 Compound Info 
N-ethyl-N-[[5-(3-methylphenyl)-1-octylindol-3-yl]methyl]ethanamine
   Show/Hide
 C28H40N2  1
1
IC50 = 3600 nM
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CP0407852
 Compound Info 
N-[(5,6-dichloro-1H-benzimidazol-2-yl)methyl]-2-morpholin-4-yl-9-pyridin-3-ylpurin-6-amine
   Show/Hide
 C22H19Cl2N9O  1
1
EC50 = 4 nM
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CP0407874
 Compound Info 
1-[4-(3-bromoanilino)quinazolin-6-yl]-3-(3,4-dichlorophenyl)thiourea
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 C21H14BrCl2N5S  1
1
GI50 = 4800 nM
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CP0407945
 Compound Info 
1-[4-(3-bromoanilino)quinazolin-6-yl]-3-methylthiourea
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 C16H14BrN5S  1
1
GI50 > 30000 nM
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CP0408551
 Compound Info 
2-[(2R,5R)-2-[[(2R,5R)-2,5-dimethylmorpholin-4-yl]methyl]-5-methylpiperazin-1-yl]-1-[6-[(4-fluorophenyl)methyl]-3,3-dimethyl-2H-pyrrolo[3,2-b]pyridin-1-yl]ethanone
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 C30H42FN5O2  1
1
IC50 = 26 nM
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CP0409460
 Compound Info 
ethyl 3-methyl-5-[(2-nitrophenyl)sulfonylamino]-1-benzofuran-2-carboxylate
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 C18H16N2O7S  1
1
IC50 = 80400 nM
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CP0410332
 Compound Info 
2-(1H-benzimidazol-2-ylmethyl)-5-(4-chlorophenyl)-1,3,4-oxadiazole
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 C16H11ClN4O  1
1
IC50 = 14500 nM
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CP0410333
 Compound Info 
2-benzhydryl-5-(1H-benzimidazol-2-ylmethyl)-1,3,4-oxadiazole
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 C23H18N4O  1
1
IC50 = 48600 nM
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CP0413318
 Compound Info 
2-morpholin-4-yl-1-(4-nitrophenyl)-2-sulfanylideneethanone
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 C12H12N2O4S  1
1
IC50 > 100000 nM
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CP0413319
 Compound Info 
1-(3-chlorophenyl)-2-morpholin-4-yl-2-sulfanylideneethanone
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 C12H12ClNO2S  1
1
IC50 > 100000 nM
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CP0413707
 Compound Info 
2-(5'-bromo-2'-oxospiro[1,3-dioxolane-2,3'-indole]-1'-yl)-N-hydroxyacetamide
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 C12H11BrN2O5  1
1
IC50 = 57450 nM
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CP0415930
 Compound Info 
2-acetyl-5-hydroxybenzo[f][1]benzofuran-4,9-dione
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 C14H8O5  1
1
IC50 = 170 nM
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CP0416887
 Compound Info 
1,3-dichloro-7-(3-chloro-4-hydroxy-6-methoxy-2-methylphenyl)-2,4,6,9-tetrahydroxy-12,12-dimethyltetracen-5-one
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 C28H21Cl3O7  1
1
IC50 > 40000 nM
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CP0417643
 Compound Info 
4-tert-butyl-N-[4-(hydroxycarbamoyl)phenyl]benzamide
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 C18H20N2O3  1
1
IC50 > 25000 nM
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CP0418687
 Compound Info 
4-(4-chlorophenyl)-2-[(2Z)-2-[1-[1-ethyl-5-[4-[(4-methylpiperazin-1-yl)methyl]-1,3-thiazol-2-yl]indol-3-yl]-2,2,2-trifluoroethylidene]hydrazinyl]-1,3-thiazole-5-carbonitrile
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 C31H28ClF3N8S2  1
1
IC50 = 1560 nM
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CP0422287
 Compound Info 
N-[(Z)-[1-[1-ethyl-5-[4-[(4-methylpiperazin-1-yl)methyl]-1,3-thiazol-2-yl]indol-3-yl]-2,2,2-trifluoroethylidene]amino]-1,3-benzothiazol-2-amine
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 C28H28F3N7S2  1
1
IC50 = 1450 nM
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CP0422288
 Compound Info 
2-[(2Z)-2-[1-[5-[4-[2-(dimethylamino)ethyl]piperazin-1-yl]-6-fluoro-2-methyl-1H-indol-3-yl]-2,2,2-trifluoroethylidene]hydrazinyl]-4-(4-fluorophenyl)-1,3-thiazole-5-carbonitrile
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 C29H29F5N8S  1
1
IC50 = 790 nM
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CP0422907
 Compound Info 
4-(4-chlorophenyl)-2-[(2Z)-2-[1-[1-ethyl-5-[4-[(4-ethylpiperazin-1-yl)methyl]-1,3-thiazol-2-yl]indol-3-yl]-2,2,2-trifluoroethylidene]hydrazinyl]-1,3-thiazole-5-carbonitrile
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 C32H30ClF3N8S2  1
1
IC50 = 3210 nM
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CP0423624
 Compound Info 
methyl (1R,2R,3S,3aR,8bS)-6-acetyl-1,8b-dihydroxy-8-methoxy-3a-(4-methoxyphenyl)-3-phenyl-2,3-dihydro-1H-cyclopenta[b][1]benzofuran-2-carboxylate
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 C29H28O8  1
1
EC50 = 1 nM
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CP0423625
 Compound Info 
methyl (1R,2R,3S,3aR,8bS)-1,8b-dihydroxy-6-[[(2S,6S)-6-(hydroxymethyl)-1,4-dioxan-2-yl]oxy]-8-methoxy-3a-(4-methoxyphenyl)-3-phenyl-2,3-dihydro-1H-cyclopenta[b][1]benzofuran-2-carboxylate
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 C32H34O11  1
1
EC50 = 9 nM
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CP0423628
 Compound Info 
methyl (1R,2R,3S,3aR,8bS)-1,8b-dihydroxy-6-[[(2S,3S,6S)-6-(2-hydroxyethyl)-3-methoxy-1,4-dioxan-2-yl]oxy]-8-methoxy-3a-(4-methoxyphenyl)-3-phenyl-2,3-dihydro-1H-cyclopenta[b][1]benzofuran-2-carboxylate
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 C34H38O12  1
1
EC50 = 70 nM
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CP0423636
 Compound Info 
methyl (1R,2R,3S,3aR,8bS)-1,8b-dihydroxy-6-(methanesulfonamido)-8-methoxy-3a-(4-methoxyphenyl)-3-phenyl-2,3-dihydro-1H-cyclopenta[b][1]benzofuran-2-carboxylate
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 C28H29NO9S  1
1
EC50 > 5000 nM
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CP0423637
 Compound Info 
methyl (1R,2R,3S,3aR,8bS)-1,8b-dihydroxy-8-methoxy-3a-(4-methoxyphenyl)-6-methyl-3-phenyl-2,3-dihydro-1H-cyclopenta[b][1]benzofuran-2-carboxylate
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 C28H28O7  1
1
EC50 > 5000 nM
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CP0423641
 Compound Info 
(1R,2R,3S,3aR,8bS)-1,8b-dihydroxy-6-[[(2S,6S)-6-(hydroxymethyl)-1,4-dioxan-2-yl]oxy]-8-methoxy-3a-(4-methoxyphenyl)-N,N-dimethyl-3-phenyl-2,3-dihydro-1H-cyclopenta[b][1]benzofuran-2-carboxamide
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 C33H37NO10  1
1
EC50 = 5 nM
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CP0423642
 Compound Info 
methyl (1R,2R,3S,3aR,8bS)-3a-(4-cyanophenyl)-1,8b-dihydroxy-6,8-dimethoxy-3-phenyl-2,3-dihydro-1H-cyclopenta[b][1]benzofuran-2-carboxylate
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 C28H25NO7  1
1
EC50 = 3 nM
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CP0423643
 Compound Info 
methyl (1R,2R,3S,3aR,8bS)-1,6,8b-trihydroxy-8-methoxy-3a-(4-methoxyphenyl)-3-phenyl-2,3-dihydro-1H-cyclopenta[b][1]benzofuran-2-carboxylate
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 C27H26O8  1
1
EC50 = 20 nM
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CP0425754
 Compound Info 
2-(5-(3-ethoxyphenyl)-1-octyl-1H-indol-3-yl)-N,N-diethylacetamide
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 C30H42N2O2  1
1
IC50 = 26800 nM
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CP0426073
 Compound Info 
4-nitrooxybutyl (4aS,6aR,6aS,6bR,8aR,10S,12aR,14bS)-2,2,6a,6b,9,9,12a-heptamethyl-10-phenylmethoxy-1,3,4,5,6,6a,7,8,8a,10,11,12,13,14b-tetradecahydropicene-4a-carboxylate
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 C41H61NO6  1
1
IC50 > 10000 nM
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CP0427160
 Compound Info 
2-[[(2R,5R)-1-[2-[6-[(4-fluorophenyl)methyl]-3,3-dimethyl-2H-pyrrolo[3,2-b]pyridin-1-yl]-2-oxoethyl]-5-methylpiperazin-2-yl]methyl]-3H-isoindol-1-one
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 C32H36FN5O2  1
1
IC50 = 8.3 nM
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CP0427571
 Compound Info 
N-ethyl-N-[[1-(3-methylbut-2-enyl)indol-3-yl]methyl]ethanamine
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 C18H26N2  1
1
IC50 = 74000 nM
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CP0435112
 Compound Info 
(2S)-1-[(2S)-3,3-dimethyl-2-[[(2S)-2-(methylamino)propanoyl]amino]butanoyl]-N-[(1S,2R)-2-prop-2-ynoxy-1,2,3,4-tetrahydronaphthalen-1-yl]pyrrolidine-2-carboxamide
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 C28H40N4O4  1
1
GI50 = 16 nM
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CP0437196
 Compound Info 
ethyl 5-[(3,4-dimethoxyphenyl)sulfonylamino]-3-methyl-1-benzofuran-2-carboxylate
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 C20H21NO7S  1
1
IC50 = 35400 nM
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CP0440224
 Compound Info 
N-[3-methoxy-6-[[(E)-2-(2,4,6-trimethoxyphenyl)ethenyl]sulfonylmethyl]pyridin-2-yl]methanesulfonamide
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 C19H24N2O8S2  1
1
GI50 = 641 nM
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CP0442037
 Compound Info 
(2-aminophenyl)-[1-(3-tert-butylphenyl)triazol-4-yl]methanone
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 C19H20N4O  1
1
IC50 = 14900 nM
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CP0443195
 Compound Info 
4-((+/-)-(1H-imidazol-1-yl)-(E)-methylretinoate
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 C24H32N2O2  1
1
IC50 = 7500 nM
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CP0444009
 Compound Info 
2-(5'-bromo-2'-oxospiro[1,3-dioxepane-2,3'-indole]-1'-yl)-N-hydroxyacetamide
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 C14H15BrN2O5  1
1
IC50 = 32850 nM
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CP0445793
 Compound Info 
CHEMBL4436772
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 C48H47Cl2FN6O6  1
1
IC50 > 3000 nM
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CP0447703
 Compound Info 
2-(5-m-tolyl-1H-indol-3-yl)acetamide
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 C17H16N2O  1
1
IC50 > 100000 nM
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CP0447704
 Compound Info 
3-(1-octyl-5-m-tolyl-1H-indol-3-yl)propanamide
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 C26H34N2O  1
1
IC50 = 20700 nM
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CP0447705
 Compound Info 
ethyl 2-[5-(3-methylphenyl)-1-octylindol-3-yl]acetate
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 C27H35NO2  1
1
IC50 > 100000 nM
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CP0449355
 Compound Info 
4'-[5-(4-cyclopropylaminomethyl-phenylamino)-2H-pyrazol-3-yl]-biphenyl-2,4-diol
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 C25H24N4O2  1
1
IC50 = 1 nM
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CP0449859
 Compound Info 
N-ethyl-N-[(4-fluoro-1-octylindol-3-yl)methyl]ethanamine
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 C21H33FN2  1
1
IC50 = 7500 nM
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CP0451689
 Compound Info 
ethyl 5-[(2-bromophenyl)sulfonylamino]-3-methyl-1-benzofuran-2-carboxylate
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 C18H16BrNO5S  1
1
IC50 = 178700 nM
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CP0451721
 Compound Info 
(1S,7R,10S,16E,21R)-7-benzyl-21-propan-2-yl-2-oxa-12,13-dithia-5,8,20,23-tetrazabicyclo[8.7.6]tricos-16-ene-3,6,9,19,22-pentone
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 C26H34N4O6S2  1
1
GI50 = 8.7 nM
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CP0453490
 Compound Info 
methyl (1R,2R,3S,3aR,8bS)-1,8b-dihydroxy-6-[(2S,6S)-6-(hydroxymethyl)oxan-2-yl]oxy-8-methoxy-3a-(4-methoxyphenyl)-3-phenyl-2,3-dihydro-1H-cyclopenta[b][1]benzofuran-2-carboxylate
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 C33H36O10  1
1
EC50 = 200 nM
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CP0453491
 Compound Info 
methyl (1R,2R,3S,3aR,8bS)-1,8b-dihydroxy-6,8-dimethoxy-3a-(4-methylphenyl)-3-phenyl-2,3-dihydro-1H-cyclopenta[b][1]benzofuran-2-carboxylate
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 C28H28O7  1
1
EC50 = 32 nM
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CP0453494
 Compound Info 
(1R,2R,3S,3aR,8bS)-6-cyano-1,8b-dihydroxy-8-methoxy-3a-(4-methoxyphenyl)-N,N-dimethyl-3-phenyl-2,3-dihydro-1H-cyclopenta[b][1]benzofuran-2-carboxamide
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 C29H28N2O6  1
1
EC50 = 2 nM
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CP0453523
 Compound Info 
methyl (1R,2R,3S,3aR,8bS)-6-(dimethylcarbamoyl)-1,8b-dihydroxy-8-methoxy-3a-(4-methoxyphenyl)-3-phenyl-2,3-dihydro-1H-cyclopenta[b][1]benzofuran-2-carboxylate
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 C30H31NO8  1
1
EC50 > 5000 nM
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CP0454552
 Compound Info 
1-[4-(3-bromoanilino)quinazolin-6-yl]-3-(3-chloro-4-fluorophenyl)thiourea
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 C21H14BrClFN5S  1
1
GI50 = 300 nM
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CP0454812
 Compound Info 
ethyl 3-methyl-5-[[4-(trifluoromethyl)phenyl]sulfonylamino]-1-benzofuran-2-carboxylate
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 C19H16F3NO5S  1
1
IC50 = 24300 nM
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CP0454836
 Compound Info 
2-(1H-benzimidazol-2-ylmethyl)-5-benzyl-1,3,4-oxadiazole
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 C17H14N4O  1
1
IC50 = 29800 nM
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CP0454837
 Compound Info 
2-(1H-benzimidazol-2-ylmethyl)-5-(phenoxymethyl)-1,3,4-oxadiazole
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 C17H14N4O2  1
1
IC50 = 35500 nM
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CP0454842
 Compound Info 
ethyl 3-methyl-5-(pyridin-3-ylsulfonylamino)-1-benzofuran-2-carboxylate
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 C17H16N2O5S  1
1
IC50 = 140800 nM
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CP0457636
 Compound Info 
7-hydroxy-3,4-bis(4-hydroxyphenyl)chromen-2-one
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 C21H14O5  1
1
IC50 = 59800 nM
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CP0458420
 Compound Info 
1-benzyl-3-[4-(4-tert-butylanilino)quinazolin-6-yl]thiourea
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 C26H27N5S  1
1
GI50 = 8700 nM
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CP0459930
 Compound Info 
1-(2,4-dichlorophenyl)-3-[3-fluoro-4-[6-(methylamino)pyrimidin-4-yl]oxyphenyl]urea
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 C18H14Cl2FN5O2  1
1
IC50 > 20000 nM
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CP0460196
 Compound Info 
N-[(2S)-1-amino-4-methyl-1-oxopentan-2-yl]-4-[3-[(1R)-1-cyclohexylethyl]-2-(4-methoxyanilino)-8-oxopyrano[3,2-f]benzimidazol-6-yl]benzamide
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 C38H43N5O5  1
1
IC50 = 5000 nM
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CP0461252
 Compound Info 
(2S)-1-[(2S)-3-methyl-2-[[(2S)-2-(methylamino)propanoyl]amino]butanoyl]-N-[(1S,2R)-2-[6-[[(1S,2R)-1-[[(2S)-1-[(2S)-3-methyl-2-[[(2S)-2-(methylamino)propanoyl]amino]butanoyl]pyrrolidine-2-carbonyl]amino]-2,3-dihydro-1H-inden-2-yl]oxy]hexa-2,4-diynoxy]-2,3-dihydro-1H-inden-1-yl]pyrrolidine-2-carboxamide
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 C52H70N8O8  1
1
GI50 = 0.4 nM
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CP0462276
 Compound Info 
(2S)-1-[(2S)-2-cyclohexyl-2-[[(2S)-2-(methylamino)propanoyl]amino]acetyl]-N-[(4R)-1-[6-[(4R)-4-[[(2S)-1-[(2S)-2-cyclohexyl-2-[[(2S)-2-(methylamino)propanoyl]amino]acetyl]pyrrolidine-2-carbonyl]amino]-3,4-dihydro-2H-quinolin-1-yl]hexa-2,4-diynyl]-3,4-dihydro-2H-quinolin-4-yl]pyrrolidine-2-carboxamide
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 C58H80N10O6  1
1
GI50 = 0.1 nM
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CP0462854
 Compound Info 
methyl (1R,2R,3S,3aR,8bS)-1,8b-dihydroxy-6-[[(2S,3R,6S)-6-(hydroxymethyl)-3-methoxy-1,4-dioxan-2-yl]oxy]-8-methoxy-3a-(4-methoxyphenyl)-3-phenyl-2,3-dihydro-1H-cyclopenta[b][1]benzofuran-2-carboxylate
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 C33H36O12  1
1
EC50 = 15 nM
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CP0462855
 Compound Info 
methyl (1R,2R,3S,3aR,8bS)-1,8b-dihydroxy-6-[[(2S,3R,6S)-6-(2-hydroxyethyl)-3-methoxy-1,4-dioxan-2-yl]oxy]-8-methoxy-3a-(4-methoxyphenyl)-3-phenyl-2,3-dihydro-1H-cyclopenta[b][1]benzofuran-2-carboxylate
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 C34H38O12  1
1
EC50 = 1.5 nM
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CP0462863
 Compound Info 
methyl (1R,2R,3S,3aR,8bS)-6-cyano-1,8b-dihydroxy-8-methoxy-3a-(4-methoxyphenyl)-3-phenyl-2,3-dihydro-1H-cyclopenta[b][1]benzofuran-2-carboxylate
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 C28H25NO7  1
1
EC50 = 1.8 nM
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CP0464497
 Compound Info 
2-[(1E,5E,7E,9R,10R,11E)-10-hydroxy-3,7,9,11-tetramethyltrideca-1,5,7,11-tetraenyl]-6-methoxy-3,5-dimethylpyran-4-one
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 C25H36O4  1
1
GI50 = 10500 nM
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CP0465282
 Compound Info 
4-N-(4-methoxyphenyl)-4-N-methyl-9H-pyrimido[4,5-b]indole-2,4-diamine
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 C18H17N5O  1
1
GI50 = 64.6 nM
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CP0465631
 Compound Info 
2-(5'-chloro-2'-oxospiro[1,3-dioxolane-2,3'-indole]-1'-yl)-N-hydroxyacetamide
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 C12H11ClN2O5  1
1
IC50 = 177170 nM
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CP0466665
 Compound Info 
2-(1H-benzimidazol-2-ylmethyl)-5-(4-methoxyphenyl)-1,3,4-oxadiazole
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 C17H14N4O2  1
1
IC50 = 131 nM
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CP0466666
 Compound Info 
2-(1H-benzimidazol-2-ylmethyl)-5-(naphthalen-1-ylmethyl)-1,3,4-oxadiazole
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 C21H16N4O  1
1
IC50 = 13200 nM
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CP0469271
 Compound Info 
2-(5-fluoro-1-(3-methylbut-2-enyl)-1H-indol-3-yl)acetamide
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 C15H17FN2O  1
1
IC50 > 100000 nM
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CP0469291
 Compound Info 
4-((1-(3-methylbut-2-enyl)-5-m-tolyl-1H-indol-3-yl)methyl)morpholine
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 C25H30N2O  1
1
IC50 = 34000 nM
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CP0474304
 Compound Info 
1-benzyl-3-[4-(4-sulfamoylanilino)quinazolin-6-yl]thiourea
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 C22H20N6O2S2  1
1
GI50 > 30000 nM
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CP0474307
 Compound Info 
1-[4-(3-bromoanilino)quinazolin-6-yl]-3-[3-(trifluoromethyl)phenyl]thiourea
   Show/Hide
 C22H15BrF3N5S  1
1
GI50 = 1400 nM
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CP0474429
 Compound Info 
4-((1-octyl-5-m-tolyl-1H-indol-3-yl)methyl)morpholine
   Show/Hide
 C28H38N2O  1
1
IC50 = 24500 nM
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CP0475635
 Compound Info 
1-(5-tert-butyl-1,2-oxazol-3-yl)-3-[2-methyl-4-[6-(methylamino)pyrimidin-4-yl]oxyphenyl]urea
   Show/Hide
 C20H24N6O3  1
1
IC50 = 2100 nM
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CP0475636
 Compound Info 
1-(5-tert-butyl-1,2-oxazol-3-yl)-3-[2-methyl-4-(6-morpholin-4-ylpyrimidin-4-yl)oxyphenyl]urea
   Show/Hide
 C23H28N6O4  1
1
IC50 = 7390 nM
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CP0477432
 Compound Info 
3-chloro-7-(3-chloro-4-hydroxy-6-methoxy-2-methylphenyl)-2,4,6,9-tetrahydroxy-12,12-dimethyltetracen-5-one
   Show/Hide
 C28H22Cl2O7  1
1
IC50 = 18820 nM
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CP0478984
 Compound Info 
6-[2-[4-[2-(dimethylamino)ethoxy]phenyl]-5-hydroxy-4-oxochromen-7-yl]oxy-N-hydroxyhexanamide;hydrochloride
   Show/Hide
 C25H31ClN2O7  1
1
IC50 = 2050 nM
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CP0479885
 Compound Info 
ethyl 3-methyl-5-[(3-methylphenyl)sulfonylamino]-1-benzofuran-2-carboxylate
   Show/Hide
 C19H19NO5S  1
1
IC50 = 29500 nM
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CP0479899
 Compound Info 
2-(1H-benzimidazol-2-ylmethyl)-5-(2-methylphenyl)-1,3,4-oxadiazole
   Show/Hide
 C17H14N4O  1
1
IC50 = 50000 nM
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CP0479900
 Compound Info 
2-[(6-chloro-1H-benzimidazol-2-yl)methyl]-5-(4-chlorophenyl)-1,3,4-oxadiazole
   Show/Hide
 C16H10Cl2N4O  1
1
IC50 = 14700 nM
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CP0479906
 Compound Info 
2-[(6-chloro-1H-benzimidazol-2-yl)methyl]-5-(2,4-dichlorophenyl)-1,3,4-oxadiazole
   Show/Hide
 C16H9Cl3N4O  1
1
IC50 = 29900 nM
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CP0481551
 Compound Info 
(2S)-2-amino-N-[4-[(3,4-dimethoxyphenyl)methylsulfamoyl]phenyl]-4-methylpentanamide
   Show/Hide
 C21H29N3O5S  1
1
IC50 = 5440 nM
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CP0483564
 Compound Info 
ethyl 5-[(2-chlorophenyl)sulfonylamino]-3-methyl-1-benzofuran-2-carboxylate
   Show/Hide
 C18H16ClNO5S  1
1
IC50 > 200000 nM
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CP0483565
 Compound Info 
ethyl 3-methyl-5-[[2-(trifluoromethyl)phenyl]sulfonylamino]-1-benzofuran-2-carboxylate
   Show/Hide
 C19H16F3NO5S  1
1
IC50 = 82400 nM
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CP0483566
 Compound Info 
ethyl 3-methyl-5-(naphthalen-2-ylsulfonylamino)-1-benzofuran-2-carboxylate
   Show/Hide
 C22H19NO5S  1
1
IC50 = 21600 nM
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CP0483581
 Compound Info 
1-(4-fluorophenyl)-2-morpholin-4-yl-2-sulfanylideneethanone
   Show/Hide
 C12H12FNO2S  1
1
IC50 > 100000 nM
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CP0483582
 Compound Info 
1-(4-iodophenyl)-2-morpholin-4-yl-2-sulfanylideneethanone
   Show/Hide
 C12H12INO2S  1
1
IC50 > 100000 nM
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CP0483584
 Compound Info 
1-(2-chlorophenyl)-2-morpholin-4-yl-2-sulfanylideneethanone
   Show/Hide
 C12H12ClNO2S  1
1
IC50 > 100000 nM
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CP0484751
 Compound Info 
(2E)-3-{3-chloro-4-[3-(2,6-dimethylphenyl)-4-hydroxyphenyl]phenyl}prop-2-enoic acid
   Show/Hide
 C23H19ClO3  1
1
IC50 > 10000 nM
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CP0486043
 Compound Info 
2-[[(2R,5R)-1-[2-[3-[(2,4-difluorophenyl)methyl]-7,7-dimethyl-6H-pyrrolo[3,2-c]pyridazin-5-yl]-2-oxoethyl]-5-methylpiperazin-2-yl]methyl]-1-oxo-3H-isoindole-5-carbonitrile
   Show/Hide
 C32H33F2N7O2  1
1
IC50 = 5.2 nM
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CP0486203
 Compound Info 
N-[(2S)-1-amino-1-oxo-3-phenylpropan-2-yl]-4-[3-benzyl-2-(2-methylpropylamino)-8-oxopyrano[3,2-f]benzimidazol-6-yl]benzamide
   Show/Hide
 C37H35N5O4  1
1
IC50 = 5000 nM
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CP0492769
 Compound Info 
4-chloro-N-(2-nitrophenyl)benzamide
   Show/Hide
 C13H9ClN2O3  1
1
IC50 > 100000 nM
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CP0492803
 Compound Info 
N-[3-[2-[4-amino-1-[(2S)-3-hydroxy-2-methylpropyl]pyrazolo[3,4-d]pyrimidin-3-yl]ethynyl]-4-methylphenyl]-3-(trifluoromethyl)benzamide
   Show/Hide
 C26H23F3N6O2  1
1
IC50 = 10 nM
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CP0493559
 Compound Info 
methyl (1R,2R,3S,3aR,8bS)-1,8b-dihydroxy-8-methoxy-3a-(4-methoxyphenyl)-6-(methylamino)-3-phenyl-2,3-dihydro-1H-cyclopenta[b][1]benzofuran-2-carboxylate
   Show/Hide
 C28H29NO7  1
1
EC50 = 120 nM
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CP0500000
 Compound Info 
2-(1-octyl-5-m-tolyl-1H-indol-3-yl)-1-(pyrrolidin-1-yl)ethanone
   Show/Hide
 C29H38N2O  1
1
IC50 = 15600 nM
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CP0500001
 Compound Info 
1-octyl-3-(pyrrolidin-1-ylmethyl)-5-m-tolyl-1H-indole
   Show/Hide
 C28H38N2  1
1
IC50 = 5100 nM
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CP0500023
 Compound Info 
2-(5-(3-methoxyphenyl)-1-octyl-1H-indol-3-yl)acetamide
   Show/Hide
 C25H32N2O2  1
1
IC50 = 22400 nM
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CP0503035
 Compound Info 
(2E)-3-[3-chloro-4-(4-hydroxy-3-{tricyclo[3.3.1.0^{3,7}]nonan-3-yl}phenyl)phenyl]prop-2-enoic acid
   Show/Hide
 C24H23ClO3  1
1
IC50 = 9800 nM
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CP0504740
 Compound Info 
4-(6-methoxy-3,4-dihydro-2H-quinolin-1-yl)-2,6-dimethylfuro[2,3-d]pyrimidine
   Show/Hide
 C18H19N3O2  1
1
GI50 = 11.4 nM
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CP0507077
 Compound Info 
1-benzyl-3-[4-(3-methylanilino)quinazolin-6-yl]thiourea
   Show/Hide
 C23H21N5S  1
1
GI50 = 19500 nM
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CP0507151
 Compound Info 
ethyl 5-[(4-tert-butylphenyl)sulfonylamino]-3-methyl-1-benzofuran-2-carboxylate
   Show/Hide
 C22H25NO5S  1
1
IC50 = 22400 nM
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CP0507200
 Compound Info 
1-(4-methylpiperazin-1-yl)-2-(1-octyl-5-m-tolyl-1H-indol-3-yl)ethanone
   Show/Hide
 C30H41N3O  1
1
IC50 = 19700 nM
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CP0508105
 Compound Info 
2-(1-octyl-1H-indol-3-yl)acetamide
   Show/Hide
 C18H26N2O  1
1
IC50 = 50000 nM
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CP0511796
 Compound Info 
1-[4-(4-benzylpiperazin-1-yl)-6-(1H-indol-3-ylsulfanyl)pyrimidin-2-yl]-3-(2,5-dimethylphenyl)urea
   Show/Hide
 C32H33N7OS  1
1
IC50 = 18960 nM
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CP0514458
 Compound Info 
2-(1-(3-(trifluoromethyl)benzyl)-5-m-tolyl-1H-indol-3-yl)acetamide
   Show/Hide
 C25H21F3N2O  1
1
IC50 = 17200 nM
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CP0517811
 Compound Info 
2-(1H-benzimidazol-2-ylmethyl)-5-(2-chlorophenyl)-1,3,4-oxadiazole
   Show/Hide
 C16H11ClN4O  1
1
IC50 = 21200 nM
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CP0517916
 Compound Info 
1-[4-chloro-3-(trifluoromethyl)phenyl]-3-[2-methyl-4-[6-(methylamino)pyrimidin-4-yl]oxyphenyl]thiourea
   Show/Hide
 C20H17ClF3N5OS  1
1
IC50 = 16730 nM
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CP0517983
 Compound Info 
N-[4-[2-[(2S,3S,5S)-2-[[tert-butyl(dimethyl)silyl]oxymethyl]-5-(5-methyl-2,4-dioxopyrimidin-1-yl)oxolan-3-yl]-1,3-dithian-2-yl]phenyl]-N'-hydroxyoctanediamide
   Show/Hide
 C34H52N4O7S2Si  1
1
GI50 = 3090.3 nM
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CP0519820
 Compound Info 
N-[(5,6-dichloro-1H-benzimidazol-2-yl)methyl]-2-(4-methylpiperazin-1-yl)-9-pyridin-3-ylpurin-6-amine
   Show/Hide
 C23H22Cl2N10  1
1
EC50 < 1 nM
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CP0519872
 Compound Info 
2-(5-fluoro-1-octyl-1H-indol-3-yl)acetamide
   Show/Hide
 C18H25FN2O  1
1
IC50 = 70000 nM
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CP0519874
 Compound Info 
(1-octyl-5-m-tolyl-1H-indol-3-yl)methanamine
   Show/Hide
 C24H32N2  1
1
IC50 = 2900 nM
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CP0519876
 Compound Info 
N-ethyl-N-[[5-(4-methylphenyl)-1-octylindol-3-yl]methyl]ethanamine
   Show/Hide
 C28H40N2  1
1
IC50 = 3400 nM
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CP0521709
 Compound Info 
(7R)-6-[(2S)-2-cyclohexyl-2-[[(2S)-2-(methylamino)propanoyl]amino]acetyl]-N-[(1S,2R)-2-[6-[[(1S,2R)-1-[[(7R)-6-[(2S)-2-cyclohexyl-2-[[(2S)-2-(methylamino)propanoyl]amino]acetyl]-4-thia-6-azaspiro[2.4]heptane-7-carbonyl]amino]-2,3-dihydro-1H-inden-2-yl]oxy]hexa-2,4-diynoxy]-2,3-dihydro-1H-inden-1-yl]-4-thia-6-azaspiro[2.4]heptane-7-carboxamide
   Show/Hide
 C60H78N8O8S2  1
1
GI50 < 0.1 nM
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CP0526259
 Compound Info 
(2-aminophenyl)-[1-(4-propan-2-ylphenyl)triazol-4-yl]methanone
   Show/Hide
 C18H18N4O  1
1
IC50 = 8500 nM
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CP0526919
 Compound Info 
(2E)-3-{3-chloro-4-[4-hydroxy-3-(2-methyl-1,3-dithian-2-yl)phenyl]phenyl}prop-2-enoic acid
   Show/Hide
 C20H19ClO3S2  1
1
IC50 > 20000 nM
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CP0527135
 Compound Info 
2-(1-(2-methylbuta-1,3-dienyl)-5-m-tolyl-1H-indol-3-yl)acetamide
   Show/Hide
 C22H24N2O  1
1
IC50 = 28500 nM
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CP0527139
 Compound Info 
N-[[5-(3-methylphenyl)-1-octylindol-3-yl]methyl]methanesulfonamide
   Show/Hide
 C25H34N2O2S  1
1
IC50 = 17500 nM
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CP0527140
 Compound Info 
N-ethyl-N-[[5-(2-methylphenyl)-1-octylindol-3-yl]methyl]ethanamine
   Show/Hide
 C28H40N2  1
1
IC50 = 5500 nM
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CP0527674
 Compound Info 
1-(4-chloro-2-methylphenyl)-3-[4-(1H-indol-3-ylsulfanyl)-6-morpholin-4-ylpyrimidin-2-yl]urea
   Show/Hide
 C24H23ClN6O2S  1
1
IC50 = 8650 nM
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CP0529676
 Compound Info 
N-ethyl-N-[[5-(3-fluoropyridin-4-yl)-1-octylindol-3-yl]methyl]ethanamine
   Show/Hide
 C26H36FN3  1
1
IC50 = 5140 nM
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CP0529677
 Compound Info 
5-[3-(diethylaminomethyl)-1-octylindol-5-yl]-N,N-dimethylpyridin-2-amine
   Show/Hide
 C28H42N4  1
1
IC50 = 2520 nM
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CP0539480
 Compound Info 
2-(5'-chloro-2'-oxospiro[1,3-dioxane-2,3'-indole]-1'-yl)-N-hydroxyacetamide
   Show/Hide
 C13H13ClN2O5  1
1
IC50 = 259040 nM
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CP0546110
 Compound Info 
1-[4-(cyclopropylamino)-6-(1H-indol-3-ylsulfanyl)pyrimidin-2-yl]-3-phenylurea
   Show/Hide
 C22H20N6OS  1
1
IC50 = 7860 nM
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CP0547399
 Compound Info 
1-benzyl-3-[4-(4-propan-2-ylanilino)quinazolin-6-yl]thiourea
   Show/Hide
 C25H25N5S  1
1
GI50 = 12800 nM
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CP0547446
 Compound Info 
N-[(4,5-difluoro-1H-benzimidazol-2-yl)methyl]-2-morpholin-4-yl-9-thiophen-3-ylpurin-6-amine
   Show/Hide
 C21H18F2N8OS  1
1
EC50 = 43 nM
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CP0547745
 Compound Info 
ethyl 5-[(3-chlorophenyl)sulfonylamino]-3-methyl-1-benzofuran-2-carboxylate
   Show/Hide
 C18H16ClNO5S  1
1
IC50 = 57300 nM
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CP0547746
 Compound Info 
ethyl 5-[(3-bromophenyl)sulfonylamino]-3-methyl-1-benzofuran-2-carboxylate
   Show/Hide
 C18H16BrNO5S  1
1
IC50 = 33700 nM
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CP0547747
 Compound Info 
ethyl 3-methyl-5-[(4-nitrophenyl)sulfonylamino]-1-benzofuran-2-carboxylate
   Show/Hide
 C18H16N2O7S  1
1
IC50 = 33100 nM
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CP0549968
 Compound Info 
5,7-dimethoxy-3-(3-piperidin-1-ylpropoxy)-2-(3,4,5-trimethoxyphenyl)chromen-4-one
   Show/Hide
 C28H35NO8  1
1
IC50 = 2160 nM
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CP0552321
 Compound Info 
1-(4-chloro-2-methylphenyl)-3-[4-(1H-indol-3-ylsulfanyl)-6-pyrrolidin-1-ylpyrimidin-2-yl]urea
   Show/Hide
 C24H23ClN6OS  1
1
IC50 = 9440 nM
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CP0553300
 Compound Info 
2-[(2Z)-2-[1-[1-ethyl-5-[4-[(4-ethylpiperazin-1-yl)methyl]-1,3-thiazol-2-yl]indol-3-yl]-2,2,2-trifluoroethylidene]hydrazinyl]-4-(4-fluorophenyl)-1,3-thiazole-5-carbonitrile
   Show/Hide
 C32H30F4N8S2  1
1
IC50 = 2690 nM
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CP0553579
 Compound Info 
1-[4-[(6-methyl-3,4-dihydro-2H-quinolin-1-yl)sulfonyl]phenyl]pyrrolidin-2-one
   Show/Hide
 C20H22N2O3S  1
1
IC50 = 17 nM
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CP0553580
 Compound Info 
1-[4-[(6-tert-butyl-3,4-dihydro-2H-quinolin-1-yl)sulfonyl]phenyl]pyrrolidin-2-one
   Show/Hide
 C23H28N2O3S  1
1
IC50 = 608 nM
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CP0557086
 Compound Info 
(1S,7S,10S,16E,21R)-7-benzyl-21-propan-2-yl-2-oxa-12,13-dithia-5,8,20,23-tetrazabicyclo[8.7.6]tricos-16-ene-3,6,9,19,22-pentone
   Show/Hide
 C26H34N4O6S2  1
1
GI50 = 1200 nM
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CP0557096
 Compound Info 
2-[5,7-dimethoxy-4-oxo-2-(3,4,5-trimethoxyphenyl)chromen-3-yl]oxy-N-[(E)-(2-fluorophenyl)methylideneamino]acetamide
   Show/Hide
 C29H27FN2O9  1
1
IC50 = 3400 nM
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CP0559081
 Compound Info 
1-[4-(3,4-dihydro-2H-quinolin-1-ylsulfonyl)phenyl]pyrrolidin-2-one
   Show/Hide
 C19H20N2O3S  1
1
IC50 = 15 nM
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CP0561540
 Compound Info 
1-benzyl-3-[4-(3-ethylanilino)quinazolin-6-yl]thiourea
   Show/Hide
 C24H23N5S  1
1
GI50 = 10500 nM
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CP0563880
 Compound Info 
1-[4-(1H-indol-3-ylsulfanyl)-6-(4-pyridin-2-ylpiperazin-1-yl)pyrimidin-2-yl]-3-(4-methoxyphenyl)urea
   Show/Hide
 C29H28N8O2S  1
1
IC50 = 28420 nM
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CP0563909
 Compound Info 
1-(4-chlorophenyl)-3-[4-(1H-indol-3-ylsulfanyl)-6-pyrrolidin-1-ylpyrimidin-2-yl]urea
   Show/Hide
 C23H21ClN6OS  1
1
IC50 = 5850 nM
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CP0564548
 Compound Info 
2-[(2E)-2-[[5-[4-(4-ethylpiperazine-1-carbonyl)piperidin-1-yl]-6-fluoro-2-methyl-1H-indol-3-yl]methylidene]hydrazinyl]-4-(4-fluorophenyl)-1,3-thiazole-5-carbonitrile
   Show/Hide
 C32H34F2N8OS  1
1
IC50 = 1140 nM
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CP0564728
 Compound Info 
1-[3-fluoro-4-[6-(methylamino)pyrimidin-4-yl]oxyphenyl]-3-[3-(trifluoromethyl)phenyl]thiourea
   Show/Hide
 C19H15F4N5OS  1
1
IC50 = 18280 nM
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CP0565042
 Compound Info 
(1S,7S,10S,16E,21R)-7-methyl-21-propan-2-yl-2-oxa-12,13-dithia-5,8,20,23-tetrazabicyclo[8.7.6]tricos-16-ene-3,6,9,19,22-pentone
   Show/Hide
 C20H30N4O6S2  1
1
GI50 = 16000 nM
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CP0565069
 Compound Info 
1-[4-[(6-methoxy-3,4-dihydro-2H-quinolin-1-yl)sulfonyl]phenyl]pyrrolidin-2-one
   Show/Hide
 C20H22N2O4S  1
1
IC50 = 20 nM
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CP0565161
 Compound Info 
ethyl 3-methyl-5-[(2-methylphenyl)sulfonylamino]-1-benzofuran-2-carboxylate
   Show/Hide
 C19H19NO5S  1
1
IC50 = 89200 nM
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CP0565459
 Compound Info 
US9205085, MSX-207
   Show/Hide
 C90H141N33O18S2  1
1
CC50 = 410000 nM
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CP0565779
 Compound Info 
1'-[2-(4-aminophenyl)quinoline-4-carbonyl]-2-tert-butylspiro[6H-pyrano[3,2-c]pyrazole-5,4'-piperidine]-7-one
   Show/Hide
 C30H31N5O3  1
1
IC50 = 4960 nM
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CP0569301
 Compound Info 
4-(4-chlorophenyl)-2-[(2Z)-2-[1-[1-ethyl-5-[4-[[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]methyl]-1,3-thiazol-2-yl]indol-3-yl]-2,2,2-trifluoroethylidene]hydrazinyl]-1,3-thiazole-5-carbonitrile
   Show/Hide
 C31H27ClF3N7OS2  1
1
IC50 = 1210 nM
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CP0571846
 Compound Info 
1-[[2-[3-[(Z)-N-(1,3-benzothiazol-2-ylamino)-C-(trifluoromethyl)carbonimidoyl]-1-ethylindol-5-yl]-1,3-thiazol-4-yl]methyl]piperidin-4-ol
   Show/Hide
 C28H27F3N6OS2  1
1
IC50 = 310 nM
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CP0578961
 Compound Info 
4-(4-chlorophenyl)-2-[(2Z)-2-[1-[1-ethyl-5-[4-[(3-hydroxyazetidin-1-yl)methyl]-1,3-thiazol-2-yl]indol-3-yl]-2,2,2-trifluoroethylidene]hydrazinyl]-1,3-thiazole-5-carbonitrile
   Show/Hide
 C29H23ClF3N7OS2  1
1
IC50 = 3410 nM
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CP0633664
 Compound Info 
2-chloro-N-ethyl-5-(2-methyl-1-oxo-1-(4-(trifluoromethyl)-6H-thiazolo[5,4-e]indazol-2-ylamino)propan-2-ylamino)benzamide
   Show/Hide
 C22H20ClF3N6O2S  1
1
IC50 = 4600 nM
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CP0633740
 Compound Info 
2-chloro-N-methyl-5-(2-methyl-1-oxo-1-(4-(trifluoromethyl)-6H-thiazolo[5,4-e]indazol-2-ylamino)propan-2-ylamino)benzamide
   Show/Hide
 C21H18ClF3N6O2S  1
1
IC50 = 3200 nM
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CP0633742
 Compound Info 
2-(4-chloro-3-(methylsulfonamido)phenylamino)-2-methyl-N-(4-(trifluoromethyl)-6H-thiazolo[5,4-e]indazol-2-yl)propanamide
   Show/Hide
 C20H18ClF3N6O3S2  1
1
IC50 = 4800 nM
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CP0633746
 Compound Info 
2-(4-chloro-3-(2,3-dihydroxypropoxy)phenylamino)-2-methyl-N-(4-(trifluoromethyl)-6H-thiazolo[5,4-e]indazol-2-yl)propanamide
   Show/Hide
 C22H21ClF3N5O4S  1
1
IC50 = 3000 nM
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CP0634074
 Compound Info 
2-(4-chlorophenylamino)-3-hydroxy-N-(6H-thiazolo[5,4-e]indazol-2-yl)propanamide
   Show/Hide
 C17H14ClN5O2S  1
1
IC50 = 1900 nM
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CP0634075
 Compound Info 
2-chloro-5-(2-methyl-1-oxo-1-(4-(trifluoromethyl)-6H-thiazolo[5,4-e]indazol-2-ylamino)propan-2-ylamino)benzamide
   Show/Hide
 C20H16ClF3N6O2S  1
1
IC50 = 1600 nM
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CP0634077
 Compound Info 
1-(3-hydroxyphenylamino)-N-(6H-thiazolo[5,4-e]indazol-2-yl)cyclopropanecarboxamide
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 C18H15N5O2S  1
1
IC50 = 3100 nM
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CP0634484
 Compound Info 
2-(4-fluoro-3-propionamidophenylamino)-2-methyl-N-(4-(trifluoromethyl)-6H-thiazolo[5,4-e]indazol-2-yl)propanamide
   Show/Hide
 C22H20F4N6O2S  1
1
IC50 = 4600 nM
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CP0634528
 Compound Info 
N-(benzyloxy)-2-chloro-5-(2-methyl-1-oxo-1-(4-(trifluoromethyl)-6H-thiazolo[5,4-e]indazol-2-ylamino)propan-2-ylamino)benzamide
   Show/Hide
 C27H22ClF3N6O3S  1
1
IC50 = 2600 nM
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CP0634799
 Compound Info 
2-(3-hydroxyphenylamino)-2-methyl-N-(6H-thiazolo[5,4-e]indazol-2-yl)propanamide
   Show/Hide
 C18H17N5O2S  1
1
IC50 = 2000 nM
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CP0635195
 Compound Info 
2-(3-hydroxyphenylamino)-N-(6H-thiazolo[5,4-e]indazol-2-yl)propanamide
   Show/Hide
 C17H15N5O2S  1
1
IC50 = 1600 nM
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CP0635785
 Compound Info 
2-(4-chlorophenylamino)-N-(6H-thiazolo[5,4-e]indazol-2-yl)propanamide
   Show/Hide
 C17H14ClN5OS  1
1
IC50 = 3800 nM
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CP0636016
 Compound Info 
2-(3-acetamido-4-chlorophenylamino)-2-methyl-N-(6H-thiazolo[5,4-e]indazol-2-yl)propanamide
   Show/Hide
 C20H19ClN6O2S  1
1
IC50 = 4600 nM
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CP0638972
 Compound Info 
(R)-N-(4-(1H-Pyrazol-4-yl)benzyl)-N-cyclopropyl-1-(3-((2-methyl-1-oxo-1-(piperazin-1-yl)propan-2-yl)oxy)phenyl)-piperidine-3-carboxamide Hydrochloride salt
   Show/Hide
 C33H43ClN6O3  1
1
IC50 = 28000 nM
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CP0648741
 Compound Info 
4-Hydroxytamoxifen
   Show/Hide
 C26H29NO2  2
1
IC50 = 2500 nM
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2
IC50 = 3500 nM
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CP0659902
 Compound Info 
7-(5-{4-[(10-Hydroxy-14-methyl-5-oxo-5,7,8,13,13b,14-hexahydro-indolo[2',3':3,4]pyrido[2,1-b]quinazolin-3-ylamino)-methyl]-phenyl}-[1,3,4]oxadiazol-2-yl)-heptanoic acid hydroxyamide
   Show/Hide
 C35H37N7O5  1
1
IC50 = 5700 nM
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CP0659903
 Compound Info 
Pentanedioic acid hydroxyamide (10-hydroxy-14-methyl-5-oxo-5,7,8,13,13b,14-hexahydro-indolo[2',3':3,4]pyrido[2,1-b]quinazolin-3-yl)-amide
   Show/Hide
 C24H25N5O5  1
1
IC50 = 191000 nM
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CP0664321
 Compound Info 
Heptanedioic acid hydroxyamide (10-hydroxy-14-methyl-5-oxo-5,7,8,13,13b,14-hexahydro-indolo[2',3':3,4]pyrido[2,1-b]quinazolin-3-yl)-amide
   Show/Hide
 C26H29N5O5  1
1
IC50 = 58000 nM
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CP0670595
 Compound Info 
Brintonamide D
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 C48H66N6O10  1
1
IC50 = 16700 nM
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CP0689377
 Compound Info 
SPEBRUTINIB
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 C22H22FN5O3  1
1
IC50 > 40000 nM
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CP0689758
 Compound Info 
5-(3-{4-[(10-Hydroxy-14-methyl-5-oxo-5,7,8,13,13b,14-hexahydro-indolo[2',3':3,4]pyrido[2,1-b]quinazolin-3-ylamino)-methyl]-phenyl}-[1,2,4]oxadiazol-5-yl)-pentanoic acid hydroxyamide
   Show/Hide
 C33H33N7O5  1
1
IC50 = 5900 nM
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CP0703209
 Compound Info 
4-Hydroxy-N-[3,5-bis(trifluoromethyl)phenyl]-1,2,5-thiadiazole-3-carboxamide
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 C11H5F6N3O2S  1
1
IC50 = 53000 nM
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CP0756887
 Compound Info 
4-[Cyclopropylidene-(5,5,8,8-tetramethyl-5,6,7,8-tetrahydro-naphthalen-2-yl)-methyl]-benzoic acid
   Show/Hide
 C25H28O2  1
1
IC50 = 1100 nM
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CP0803799
 Compound Info 
(S)-N-((S)-2-(Hydroxyamino)-2-oxo-1-phenylethyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide hydrochloride
   Show/Hide
 C18H20ClN3O3  1
1
IC50 = 590640 nM
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CP0858674
 Compound Info 
N-(4-Methoxyphenyl)-N,2,6-trimethylfuro[2,3-d]pyrimidin-4-amine hydrochloride
   Show/Hide
 C16H18ClN3O2  1
1
IC50 = 147.6 nM
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CP0859380
 Compound Info 
7-(2-(2,6-bis(phenylamino)-9H-purin-9-yl)acetamido)-N-hydroxyheptanamide
   Show/Hide
 C26H30N8O3  1
1
IC50 = 1550 nM
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CP0863011
 Compound Info 
N,N,N-trimethyl-3-(octadec-1-en-2-ylsulfonyl)propan-1-aminium chloride
   Show/Hide
 C24H50ClNO2S  1
1
IC50 = 390 nM
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CP0897293
 Compound Info 
1-(7-Benzyl-2-methyl-5H-pyrrolo[3,2-d]pyrimidin-4-yl)-6-methoxy-1,2,3,4-tetrahydroquinoline hydrochloride
   Show/Hide
 C24H25ClN4O  1
1
GI50 = 641 nM
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CP0899057
 Compound Info 
Brintonamide E
   Show/Hide
 C48H66N6O10  1
1
IC50 = 14900 nM
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CP0906523
 Compound Info 
7-Benzyl-N-(4-methoxyphenyl)-N,2,5-trimethyl-5H-pyrrolo[3,2-d]pyrimidin-4-amine hydrochloride
   Show/Hide
 C23H25ClN4O  1
1
GI50 = 63.7 nM
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CP0944518
 Compound Info 
Octanedioic acid hydroxyamide (10-hydroxy-14-methyl-5-oxo-5,7,8,13,13b,14-hexahydro-indolo[2',3':3,4]pyrido[2,1-b]quinazolin-3-yl)-amide
   Show/Hide
 C27H31N5O5  1
1
IC50 = 54000 nM
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Protein family and CMB statistics Related to the Cell Line
Cell Lines Derived from the same Tissue Source (Pleural effusion)
Cell Line Name Organism Disease
U-937
 Cell Line Info 
Homo sapiens (Human) Adult acute monocytic leukemia
SU-DHL-1
 Cell Line Info 
Homo sapiens (Human) Anaplastic large cell lymphoma, ALK-positive
SR
 Cell Line Info 
Homo sapiens (Human) Anaplastic large cell lymphoma, ALK-positive
MC116
 Cell Line Info 
Homo sapiens (Human) B-cell non-Hodgkin lymphoma
K-562
 Cell Line Info 
Homo sapiens (Human) Blast phase chronic myelogenous leukemia, BCR-ABL1 positive
K562/A02
 Cell Line Info 
Homo sapiens (Human) Blast phase chronic myelogenous leukemia, BCR-ABL1 positive
K562/Adr
 Cell Line Info 
Homo sapiens (Human) Blast phase chronic myelogenous leukemia, BCR-ABL1 positive
K562/R7
 Cell Line Info 
Homo sapiens (Human) Blast phase chronic myelogenous leukemia, BCR-ABL1 positive
K562/DOX
 Cell Line Info 
Homo sapiens (Human) Blast phase chronic myelogenous leukemia, BCR-ABL1 positive
MDA-MB-415
 Cell Line Info 
Homo sapiens (Human) Breast adenocarcinoma
MDA-MB-468
 Cell Line Info 
Homo sapiens (Human) Breast adenocarcinoma
SK-BR-3
 Cell Line Info 
Homo sapiens (Human) Breast adenocarcinoma
AU565
 Cell Line Info 
Homo sapiens (Human) Breast adenocarcinoma
CAL-51
 Cell Line Info 
Homo sapiens (Human) Breast carcinoma
CAL-120
 Cell Line Info 
Homo sapiens (Human) Breast carcinoma
DG-75
 Cell Line Info 
Homo sapiens (Human) Burkitt lymphoma
SUP-T1
 Cell Line Info 
Homo sapiens (Human) Childhood T lymphoblastic lymphoma
Pfeiffer
 Cell Line Info 
Homo sapiens (Human) Diffuse large B-cell lymphoma germinal center B-cell type
WSU-DLCL2
 Cell Line Info 
Homo sapiens (Human) Diffuse large B-cell lymphoma germinal center B-cell type
Karpas-422
 Cell Line Info 
Homo sapiens (Human) Diffuse large B-cell lymphoma germinal center B-cell type
DoHH2
 Cell Line Info 
Homo sapiens (Human) Diffuse large B-cell lymphoma germinal center B-cell type
KATO III
 Cell Line Info 
Homo sapiens (Human) Down syndrome
GIST-T1
 Cell Line Info 
Homo sapiens (Human) Gastrointestinal stromal tumor
GIST-5R
 Cell Line Info 
Homo sapiens (Human) Gastrointestinal stromal tumor
MZ-CRC-1
 Cell Line Info 
Homo sapiens (Human) Hereditary thyroid gland medullary carcinoma
L-428
 Cell Line Info 
Homo sapiens (Human) Hodgkin lymphoma
KM-H2
 Cell Line Info 
Homo sapiens (Human) Hodgkin lymphoma
T-47D
 Cell Line Info 
Homo sapiens (Human) Invasive breast carcinoma of no special type
MCF-7
 Cell Line Info 
Homo sapiens (Human) Invasive breast carcinoma of no special type
MCF-7/2a
 Cell Line Info 
Homo sapiens (Human) Invasive breast carcinoma of no special type
T-47
 Cell Line Info 
Homo sapiens (Human) Invasive breast carcinoma of no special type
MCF-7 MX100
 Cell Line Info 
Homo sapiens (Human) Invasive breast carcinoma of no special type
MCF-7/VP
 Cell Line Info 
Homo sapiens (Human) Invasive breast carcinoma of no special type
MCF-7-2a
 Cell Line Info 
Homo sapiens (Human) Invasive breast carcinoma of no special type
T47D:A18
 Cell Line Info 
Homo sapiens (Human) Invasive breast carcinoma of no special type
MVLN
 Cell Line Info 
Homo sapiens (Human) Invasive breast carcinoma of no special type
MCF/MX
 Cell Line Info 
Homo sapiens (Human) Invasive breast carcinoma of no special type
MCF7/Topo
 Cell Line Info 
Homo sapiens (Human) Invasive breast carcinoma of no special type
MCF-7/NOD2
 Cell Line Info 
Homo sapiens (Human) Invasive breast carcinoma of no special type
MCF-7aro
 Cell Line Info 
Homo sapiens (Human) Invasive breast carcinoma of no special type
MCF7/MRP1-M6
 Cell Line Info 
Homo sapiens (Human) Invasive breast carcinoma of no special type
MCF7/MRP1-10
 Cell Line Info 
Homo sapiens (Human) Invasive breast carcinoma of no special type
MCF7/MRP1-M24
 Cell Line Info 
Homo sapiens (Human) Invasive breast carcinoma of no special type
MCF-7/NOD1
 Cell Line Info 
Homo sapiens (Human) Invasive breast carcinoma of no special type
MCF-7piGST
 Cell Line Info 
Homo sapiens (Human) Invasive breast carcinoma of no special type
MCF7-Y1
 Cell Line Info 
Homo sapiens (Human) Invasive breast carcinoma of no special type
MCF7/ADM
 Cell Line Info 
Homo sapiens (Human) Invasive breast carcinoma of no special type
MCF7:WS8
 Cell Line Info 
Homo sapiens (Human) Invasive breast carcinoma of no special type
MCF-7-FLV1000
 Cell Line Info 
Homo sapiens (Human) Invasive breast carcinoma of no special type
MCF7-neo/Her2
 Cell Line Info 
Homo sapiens (Human) Invasive breast carcinoma of no special type
MCF-7 cl.24
 Cell Line Info 
Homo sapiens (Human) Invasive breast carcinoma of no special type
MCF-7/DX1
 Cell Line Info 
Homo sapiens (Human) Invasive breast carcinoma of no special type
MCF7-LC3
 Cell Line Info 
Homo sapiens (Human) Invasive breast carcinoma of no special type
T47D-KBluc
 Cell Line Info 
Homo sapiens (Human) Invasive breast carcinoma of no special type
Calu-6
 Cell Line Info 
Homo sapiens (Human) Lung adenocarcinoma
Calu-3
 Cell Line Info 
Homo sapiens (Human) Lung adenocarcinoma
HCC78
 Cell Line Info 
Homo sapiens (Human) Lung adenocarcinoma
NCI-H3122
 Cell Line Info 
Homo sapiens (Human) Lung adenocarcinoma
NCI-H3255
 Cell Line Info 
Homo sapiens (Human) Lung adenocarcinoma
NCI-H2122
 Cell Line Info 
Homo sapiens (Human) Lung adenocarcinoma
COR-L105
 Cell Line Info 
Homo sapiens (Human) Lung adenocarcinoma
NCI-H1437
 Cell Line Info 
Homo sapiens (Human) Lung adenocarcinoma
HCC4006
 Cell Line Info 
Homo sapiens (Human) Lung adenocarcinoma
NCI-H1792
 Cell Line Info 
Homo sapiens (Human) Lung adenocarcinoma
DFCI032
 Cell Line Info 
Homo sapiens (Human) Lung adenocarcinoma
NCI-H1355
 Cell Line Info 
Homo sapiens (Human) Lung adenocarcinoma
NCI-H460
 Cell Line Info 
Homo sapiens (Human) Lung large cell carcinoma
U-1810
 Cell Line Info 
Homo sapiens (Human) Lung large cell carcinoma
COR-L23/R
 Cell Line Info 
Homo sapiens (Human) Lung large cell carcinoma
H460/MX20
 Cell Line Info 
Homo sapiens (Human) Lung large cell carcinoma
H460R
 Cell Line Info 
Homo sapiens (Human) Lung large cell carcinoma
H69AR
 Cell Line Info 
Homo sapiens (Human) Lung small cell carcinoma
NCI-H69
 Cell Line Info 
Homo sapiens (Human) Lung small cell carcinoma
GLC-4/ADR
 Cell Line Info 
Homo sapiens (Human) Lung small cell carcinoma
STC 1
 Cell Line Info 
Homo sapiens (Human) Lung small cell carcinoma
RERF-LC-A1
 Cell Line Info 
Homo sapiens (Human) Lung squamous cell carcinoma
Calu-1
 Cell Line Info 
Homo sapiens (Human) Lung squamous cell carcinoma
HCC95
 Cell Line Info 
Homo sapiens (Human) Lung squamous cell carcinoma
RERF-LC-AI Tet-off
 Cell Line Info 
Homo sapiens (Human) Lung squamous cell carcinoma
NCI-H1650
 Cell Line Info 
Homo sapiens (Human) Minimally invasive lung adenocarcinoma
NCI-H1666
 Cell Line Info 
Homo sapiens (Human) Minimally invasive lung adenocarcinoma
NCI-H929
 Cell Line Info 
Homo sapiens (Human) Plasma cell myeloma
KMS-11
 Cell Line Info 
Homo sapiens (Human) Plasma cell myeloma
UTMC-2
 Cell Line Info 
Homo sapiens (Human) Plasma cell myeloma
KMS-12-PE
 Cell Line Info 
Homo sapiens (Human) Plasma cell myeloma
NCI-H226
 Cell Line Info 
Homo sapiens (Human) Pleural epithelioid mesothelioma
Karpas-1106P
 Cell Line Info 
Homo sapiens (Human) Primary mediastinal (thymic) large B-cell lymphoma