| Compound ID |
Compound Name |
Compound Formula |
|
CP0537644
|
2-(4-chlorophenyl)-8-hexyl-7-methylimidazo[1,2-a]pyrimidin-5-one
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|
C19H22ClN3O
|
1
|
| 1 |
IC50 = 30 nM
|
|
|
|
CP0018950
|
2-(4-{[(3-Trifluoromethylphenyl)amino]carbonothioyl}-1-piperazinyl)-8-ethyl-5-oxo-5,8-dihydropyrido[2,3-d]pyrimidine-6-carboxylic Acid
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|
C22H21F3N6O3S
|
2
|
| 1 |
IC50 = 900 nM
|
|
|
| 2 |
Ki = 700 nM
|
|
|
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CP0491615
|
2-(4-{[(2,5-Dichlorophenyl)amino]carbonothioyl}-1-piperazinyl)-8-ethyl-5-oxo-5,8-dihydropyrido[2,3-d]pyrimidine-6-carboxylic Acid
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|
C21H20Cl2N6O3S
|
3
|
| 1 |
IC50 = 1300 nM
|
|
|
| 2 |
Ki = 3400 nM
|
|
|
| 3 |
Ki = 22000 nM
|
|
|
|
CP0455141
|
2-(4-{[(4-Trifluoromethylphenyl)amino]carbonothioyl}-1-piperazinyl)-8-ethyl-5-oxo-5,8-dihydropyrido[2,3-d]pyrimidine-6-carboxylic Acid
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|
C22H21F3N6O3S
|
2
|
| 1 |
IC50 = 1500 nM
|
|
|
| 2 |
Ki = 13200 nM
|
|
|
|
CP0227783
|
2-(4-((3,5-dichlorophenyl)carbamothioyl)piperazin-1-yl)-8-ethyl-5-oxo-5,8-dihydropyrido[2,3-d]pyrimidine-6-carboxylic acid
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|
C21H20Cl2N6O3S
|
2
|
| 1 |
IC50 = 1600 nM
|
|
|
| 2 |
Ki = 1900 nM
|
|
|
|
CP0439134
|
2-(4-{[(3-Iodophenyl)amino]carbonothioyl}-1-piperazinyl)-8-ethyl-5-oxo-5,8-dihydropyrido[2,3-d]pyrimidine-6-carboxylic Acid
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|
C21H21IN6O3S
|
3
|
| 1 |
IC50 = 1600 nM
|
|
|
| 2 |
Ki = 7400 nM
|
|
|
| 3 |
Ki = 11000 nM
|
|
|
|
CP0029804
|
2-(4-{[(3-Chlorophenyl)amino]carbonothioyl}-1-piperazinyl)-8-ethyl-5-oxo-5,8-dihydropyrido[2,3-d]pyrimidine-6-carboxylic Acid
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|
C21H21ClN6O3S
|
3
|
| 1 |
IC50 = 2500 nM
|
|
|
| 2 |
Ki = 2600 nM
|
|
|
| 3 |
Ki = 47300 nM
|
|
|
|
CP0497056
|
2-(4-{[(3,5-Bis(trifluoromethyl)phenyl)amino]carbonothioyl}-1-piperazinyl)-8-ethyl-5-oxo-5,8-dihydropyrido[2,3-d]pyrimidine-6-carboxylic Acid
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|
C23H20F6N6O3S
|
2
|
| 1 |
IC50 = 4400 nM
|
|
|
| 2 |
Ki = 4000 nM
|
|
|
|
CP0439131
|
2-(4-{[(4-Iodophenyl)amino]carbonothioyl}-1-piperazinyl)-8-ethyl-5-oxo-5,8-dihydropyrido[2,3-d]pyrimidine-6-carboxylic Acid
Show/Hide
|
C21H21IN6O3S
|
3
|
| 1 |
IC50 = 5600 nM
|
|
|
| 2 |
Ki = 13200 nM
|
|
|
| 3 |
Ki = 34100 nM
|
|
|
|
CP0501469
|
2-(4-{[(3,5-Dimethylphenyl)amino]carbonothioyl}-1-piperazinyl)-8-ethyl-5-oxo-5,8-dihydropyrido[2,3-d]pyrimidine-6-carboxylic Acid
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|
C23H26N6O3S
|
2
|
| 1 |
IC50 = 9000 nM
|
|
|
| 2 |
Ki = 4200 nM
|
|
|
|
CP0431026
|
2-(4-{[(4-Chlorophenyl)amino]carbonothioyl}-1-piperazinyl)-8-ethyl-5-oxo-5,8-dihydropyrido[2,3-d]pyrimidine-6-carboxylic Acid
Show/Hide
|
C21H21ClN6O3S
|
2
|
| 1 |
IC50 = 10700 nM
|
|
|
| 2 |
Ki = 5700 nM
|
|
|
|
CP0430933
|
2-(4-{[(3-Benzothiadiazolphenyl)amino]carbonothioyl}-1-piperazinyl)-8-ethyl-5-oxo-5,8-dihydropyrido[2,3-d]pyrimidine-6-carboxylic Acid
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|
C21H20N8O3S2
|
2
|
| 1 |
IC50 = 12100 nM
|
|
|
| 2 |
Ki = 7100 nM
|
|
|
|
CP0491621
|
2-(4-{[(3-Methylphenyl)amino]carbonothioyl}-1-piperazinyl)-8-ethyl-5-oxo-5,8-dihydropyrido[2,3-d]pyrimidine-6-carboxylic Acid
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|
C22H24N6O3S
|
2
|
| 1 |
IC50 = 13500 nM
|
|
|
| 2 |
Ki = 4500 nM
|
|
|
|
CP0439135
|
2-(4-{[(4-Methylphenyl)amino]carbonothioyl}-1-piperazinyl)-8-ethyl-5-oxo-5,8-dihydropyrido[2,3-d]pyrimidine-6-carboxylic Acid
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|
C22H24N6O3S
|
1
|
| 1 |
IC50 = 16100 nM
|
|
|
|
CP0502984
|
2-(4-{[(3-Fluorophenyl)amino]carbonothioyl}-1-piperazinyl)-8-ethyl-5-oxo-5,8-dihydropyrido[2,3-d]pyrimidine-6-carboxylic Acid
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|
C21H21FN6O3S
|
1
|
| 1 |
IC50 = 16100 nM
|
|
|
|
CP0252311
|
2-(4-{[(4-Fluorophenyl)amino]carbonothioyl}-1-piperazinyl)-8-ethyl-5-oxo-5,8-dihydropyrido[2,3-d]pyrimidine-6-carboxylic Acid
Show/Hide
|
C21H21FN6O3S
|
1
|
| 1 |
IC50 = 17700 nM
|
|
|
|
CP0431027
|
2-(4-{[(3-Methoxyphenyl)amino]carbonothioyl}-1-piperazinyl)-8-ethyl-5-oxo-5,8-dihydropyrido[2,3-d]pyrimidine-6-carboxylic Acid
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|
C22H24N6O4S
|
1
|
| 1 |
IC50 = 17700 nM
|
|
|
|
CP0125579
|
(R)-Octadec-9-enoic acid 2-hydroxy-3-phosphonooxy-propyl ester
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|
C21H41O7P
|
1
|
| 1 |
Ki = 100 nM
|
|
|
|
CP0497058
|
4-amino-4-(hydroxymethyl)-6-(4-octylphenyl)hexylphosphonic acid
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|
C21H38NO4P
|
1
|
| 1 |
Ki = 200 nM
|
|
|
