Compound ID |
Compound Name |
Compound Formula |
CP0415114
|
methyl 4-[[4-[2-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl]phenyl]carbamoyl]-2-(quinoline-2-carbonylamino)benzoate
Show/Hide
|
C38H36N4O6
|
3
|
1 |
IC50 = 59 nM
|
|
|
2 |
IC50 = 60 nM
|
|
|
3 |
IC50 = 65 nM
|
|
|
CP0563377
|
N-[5-[1-[4-[2-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl]phenyl]triazol-4-yl]-2-propanoylphenyl]-6-nitropyridine-2-carboxamide
Show/Hide
|
C36H35N7O6
|
1
|
1 |
IC50 = 70 nM
|
|
|
CP0500776
|
N-[5-[1-[4-[2-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl]phenyl]triazol-4-yl]-2-propanoylphenyl]quinoline-2-carboxamide
Show/Hide
|
C40H38N6O4
|
1
|
1 |
IC50 = 79 nM
|
|
|
CP0563378
|
N-[5-[1-[4-[2-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl]phenyl]triazol-4-yl]-2-propanoylphenyl]-4-oxochromene-2-carboxamide
Show/Hide
|
C40H37N5O6
|
1
|
1 |
IC50 = 80 nM
|
|
|
CP0552852
|
6-amino-N-[5-[1-[4-[2-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl]phenyl]triazol-4-yl]-2-propanoylphenyl]pyridine-2-carboxamide
Show/Hide
|
C36H37N7O4
|
1
|
1 |
IC50 = 82 nM
|
|
|
CP0531229
|
N-[5-methyl-2-[1-(2-pyrrolidin-1-ylethyl)triazol-4-yl]phenyl]-4-oxochromene-2-carboxamide
Show/Hide
|
C25H25N5O3
|
1
|
1 |
IC50 = 109 nM
|
|
|
CP0533951
|
6-chloro-N-[5-[1-[4-[2-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl]phenyl]triazol-4-yl]-2-propanoylphenyl]pyridine-2-carboxamide
Show/Hide
|
C36H35ClN6O4
|
1
|
1 |
IC50 = 116 nM
|
|
|
CP0563376
|
N-[5-[1-[4-[2-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl]phenyl]triazol-4-yl]-2-propanoylphenyl]-5-methoxypyridine-2-carboxamide
Show/Hide
|
C37H38N6O5
|
1
|
1 |
IC50 = 116 nM
|
|
|
CP0141589
|
3-((3S,6S)-6-Isobutyl-9-methoxy-1,4-dioxo-1,2,3,4,6,7,12,12a-octahydro-pyrazino[1',2':1,6]pyrido[3,4-b]indol-3-yl)-propionic acid tert-butyl ester
Show/Hide
|
C26H35N3O5
|
2
|
1 |
IC50 = 117 nM
|
|
|
2 |
IC50 = 225 nM
|
|
|
CP0373409
|
methyl 4-[[4-[2-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl]phenyl]carbamoyl]-2-(quinoline-3-carbonylamino)benzoate
Show/Hide
|
C38H36N4O6
|
1
|
1 |
IC50 = 119 nM
|
|
|
CP0565434
|
N-[5-[1-[4-[2-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl]phenyl]triazol-4-yl]-2-propanoylphenyl]-1-benzofuran-2-carboxamide
Show/Hide
|
C39H37N5O5
|
1
|
1 |
IC50 = 120 nM
|
|
|
CP0254388
|
5-Methoxy-9-oxo-9,10-dihydro-acridine-4-carboxylic acid {4-[2-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)-ethyl]-phenyl}-amide
Show/Hide
|
C34H33N3O5
|
2
|
1 |
IC50 = 127 nM
|
|
|
2 |
IC50 = 250 nM
|
|
|
CP0437995
|
methyl 4-[[4-[2-[6-methoxy-7-[2-[2-(2-methoxyethoxy)ethoxy]ethoxy]-3,4-dihydro-1H-isoquinolin-2-yl]ethyl]phenyl]carbamoyl]-2-(quinoline-2-carbonylamino)benzoate
Show/Hide
|
C44H48N4O9
|
1
|
1 |
IC50 = 130 nM
|
|
|
CP0486095
|
methyl 4-bromo-2-[(4-oxochromene-2-carbonyl)amino]benzoate
Show/Hide
|
C18H12BrNO5
|
1
|
1 |
IC50 = 140 nM
|
|
|
CP0531228
|
4-oxo-N-[2-propanoyl-5-[1-(2-pyrrolidin-1-ylethyl)triazol-4-yl]phenyl]chromene-2-carboxamide
Show/Hide
|
C27H27N5O4
|
1
|
1 |
IC50 = 158 nM
|
|
|
CP0531227
|
N-[5-[1-[4-[2-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl]phenyl]triazol-4-yl]-2-propanoylphenyl]-6-methylpyridine-2-carboxamide
Show/Hide
|
C37H38N6O4
|
1
|
1 |
IC50 = 166 nM
|
|
|
CP0394488
|
methyl 4-[[4-[2-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl]phenyl]carbamoyl]-2-(quinoline-6-carbonylamino)benzoate
Show/Hide
|
C38H36N4O6
|
2
|
1 |
IC50 = 172 nM
|
|
|
2 |
IC50 = 179 nM
|
|
|
CP0531225
|
N-[5-[1-[4-[2-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl]phenyl]triazol-4-yl]-2-propanoylphenyl]-5,6,7,8-tetrahydroquinoline-2-carboxamide
Show/Hide
|
C40H42N6O4
|
1
|
1 |
IC50 = 180 nM
|
|
|
CP0382010
|
methyl 4-[[4-[2-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl]phenyl]carbamoyl]-2-(quinoxaline-2-carbonylamino)benzoate
Show/Hide
|
C37H35N5O6
|
1
|
1 |
IC50 = 183 nM
|
|
|
CP0373171
|
methyl 4-[[4-[2-[7-methoxy-6-[2-[2-(2-methoxyethoxy)ethoxy]ethoxy]-3,4-dihydro-1H-isoquinolin-2-yl]ethyl]phenyl]carbamoyl]-2-(quinoline-2-carbonylamino)benzoate
Show/Hide
|
C44H48N4O9
|
1
|
1 |
IC50 = 183 nM
|
|
|
CP0486097
|
N-[5-methyl-2-[1-(2-morpholin-4-ylethyl)triazol-4-yl]phenyl]-4-oxochromene-2-carboxamide
Show/Hide
|
C25H25N5O4
|
1
|
1 |
IC50 = 188 nM
|
|
|
CP0417519
|
methyl 4-[4-[[7-methoxy-6-[2-[2-(2-methoxyethoxy)ethoxy]ethoxy]-3,4-dihydro-1H-isoquinolin-2-yl]methyl]phenyl]-2-(quinoline-6-carbonylamino)benzoate
Show/Hide
|
C42H45N3O8
|
1
|
1 |
IC50 = 237 nM
|
|
|
CP0565435
|
N-[5-[1-[4-[2-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl]phenyl]triazol-4-yl]-2-propanoylphenyl]naphthalene-2-carboxamide
Show/Hide
|
C41H39N5O4
|
1
|
1 |
IC50 = 249 nM
|
|
|
CP0531226
|
N-[5-[1-(2-morpholin-4-ylethyl)triazol-4-yl]-2-propanoylphenyl]-4-oxochromene-2-carboxamide
Show/Hide
|
C27H27N5O5
|
1
|
1 |
IC50 = 312 nM
|
|
|
CP0382011
|
N-[5-[[4-[2-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl]phenyl]carbamoyl]-2-methoxyphenyl]quinoline-3-carboxamide
Show/Hide
|
C37H36N4O5
|
1
|
1 |
IC50 = 317 nM
|
|
|
CP0531222
|
N-[5-[1-[4-[2-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl]phenyl]triazol-4-yl]-2-propanoylphenyl]-6-methoxypyridine-2-carboxamide
Show/Hide
|
C37H38N6O5
|
1
|
1 |
IC50 = 322 nM
|
|
|
CP0531223
|
N-[5-[1-[4-[2-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl]phenyl]triazol-4-yl]-2-propanoylphenyl]-6-oxo-1H-pyridine-2-carboxamide
Show/Hide
|
C36H36N6O5
|
1
|
1 |
IC50 = 328 nM
|
|
|
CP0437996
|
methyl 4-[[4-[2-[7-methoxy-6-[2-[2-(2-methoxyethoxy)ethoxy]ethoxy]-3,4-dihydro-1H-isoquinolin-2-yl]ethyl]phenyl]carbamoyl]-2-(quinoline-6-carbonylamino)benzoate
Show/Hide
|
C44H48N4O9
|
1
|
1 |
IC50 = 390 nM
|
|
|
CP0563379
|
N-[2-[1-(2-hydroxyethyl)triazol-4-yl]-5-methylphenyl]-4-oxochromene-2-carboxamide
Show/Hide
|
C21H18N4O4
|
1
|
1 |
IC50 = 447 nM
|
|
|
CP0465345
|
methyl 4-[[4-[2-[6-methoxy-7-[2-[2-(2-methoxyethoxy)ethoxy]ethoxy]-3,4-dihydro-1H-isoquinolin-2-yl]ethyl]phenyl]carbamoyl]-2-(quinoline-6-carbonylamino)benzoate
Show/Hide
|
C44H48N4O9
|
1
|
1 |
IC50 = 508 nM
|
|
|
CP0116921
|
1N-{4-[2-(6,7-dimethoxy-1,2,3,4-tetrahydro-2-isoquinolinyl)ethyl]phenyl}-4,5-dimethoxy-2-(3-quinolylcarboxamido)benzamide
Show/Hide
|
C38H38N4O6
|
3
|
1 |
IC50 = 520 nM
|
|
|
2 |
IC50 = 526 nM
|
|
|
3 |
IC50 = 916 nM
|
|
|
CP0455199
|
methyl 4-[4-[2-[6,7-bis[2-[2-(2-methoxyethoxy)ethoxy]ethoxy]-3,4-dihydro-1H-isoquinolin-2-yl]ethyl]phenyl]-2-(quinoline-2-carbonylamino)benzoate
Show/Hide
|
C49H59N3O11
|
1
|
1 |
IC50 = 544 nM
|
|
|
CP0459693
|
methyl 4-[[4-[2-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl]phenyl]carbamoyl]-2-[(5-methylpyrazine-2-carbonyl)amino]benzoate
Show/Hide
|
C34H35N5O6
|
1
|
1 |
IC50 = 552 nM
|
|
|
CP0417560
|
methyl 4-[4-[[6-methoxy-7-[2-[2-(2-methoxyethoxy)ethoxy]ethoxy]-3,4-dihydro-1H-isoquinolin-2-yl]methyl]phenyl]-2-(quinoline-2-carbonylamino)benzoate
Show/Hide
|
C42H45N3O8
|
1
|
1 |
IC50 = 591 nM
|
|
|
CP0531224
|
methyl 4-[1-[4-[2-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl]phenyl]triazol-4-yl]-2-(quinoline-2-carbonylamino)benzoate
Show/Hide
|
C39H36N6O5
|
1
|
1 |
IC50 = 617 nM
|
|
|
CP0462358
|
methyl 4-[[4-[2-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl]phenyl]carbamoyl]-2-(pyrazine-2-carbonylamino)benzoate
Show/Hide
|
C33H33N5O6
|
1
|
1 |
IC50 = 632 nM
|
|
|
CP0455202
|
methyl 4-[4-(3,4-dihydro-1H-isoquinolin-2-ylmethyl)phenyl]-2-(quinoline-6-carbonylamino)benzoate
Show/Hide
|
C34H29N3O3
|
1
|
1 |
IC50 = 641 nM
|
|
|
CP0046870
|
FTC
Show/Hide
|
C22H25N3O3
|
4
|
1 |
IC50 = 730 nM
|
|
|
2 |
IC50 = 731 nM
|
|
|
3 |
IC50 = 960 nM
|
|
|
4 |
IC50 > 11000 nM
|
|
|
CP0469410
|
methyl 4-[4-[2-[6-methoxy-7-[2-[2-(2-methoxyethoxy)ethoxy]ethoxy]-3,4-dihydro-1H-isoquinolin-2-yl]ethyl]phenyl]-2-(quinoline-2-carbonylamino)benzoate
Show/Hide
|
C43H47N3O8
|
1
|
1 |
IC50 = 760 nM
|
|
|
CP0459998
|
methyl 4-[4-[[6,7-bis[2-[2-(2-methoxyethoxy)ethoxy]ethoxy]-3,4-dihydro-1H-isoquinolin-2-yl]methyl]phenyl]-2-(quinoline-2-carbonylamino)benzoate
Show/Hide
|
C48H57N3O11
|
1
|
1 |
IC50 = 839 nM
|
|
|
CP0502250
|
N-[5-[[4-[2-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl]phenyl]carbamoyl]-2,3-dimethoxyphenyl]quinoline-3-carboxamide
Show/Hide
|
C38H38N4O6
|
1
|
1 |
IC50 = 858 nM
|
|
|
CP0466004
|
N-[5-[(E)-3-[4-[2-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethoxy]phenyl]prop-2-enoyl]-2-methylphenyl]quinoline-2-carboxamide
Show/Hide
|
C39H37N3O5
|
1
|
1 |
IC50 = 880 nM
|
|
|
CP0455201
|
methyl 4-[4-[(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)methyl]phenyl]-2-(quinoline-2-carbonylamino)benzoate
Show/Hide
|
C36H33N3O5
|
1
|
1 |
IC50 = 943 nM
|
|
|
CP0394487
|
N-[3-[[4-[2-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl]phenyl]carbamoyl]-5-methoxyphenyl]quinoline-3-carboxamide
Show/Hide
|
C37H36N4O5
|
1
|
1 |
IC50 = 977 nM
|
|
|
CP0423799
|
methyl 4-[[4-[2-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl]phenyl]carbamoyl]-2-(pyridine-3-carbonylamino)benzoate
Show/Hide
|
C34H34N4O6
|
1
|
1 |
IC50 = 1015 nM
|
|
|
CP0426811
|
methyl 4-[4-[[7-methoxy-6-[2-[2-(2-methoxyethoxy)ethoxy]ethoxy]-3,4-dihydro-1H-isoquinolin-2-yl]methyl]phenyl]-2-(quinoline-2-carbonylamino)benzoate
Show/Hide
|
C42H45N3O8
|
1
|
1 |
IC50 = 1031 nM
|
|
|
CP0410638
|
methyl 4-[4-[2-(3,4-dihydro-1H-isoquinolin-2-yl)ethyl]phenyl]-2-(quinoline-2-carbonylamino)benzoate
Show/Hide
|
C35H31N3O3
|
1
|
1 |
IC50 = 1100 nM
|
|
|
CP0415664
|
N-[3-[2-[6-methoxy-7-[2-[2-(2-methoxyethoxy)ethoxy]ethoxy]-3,4-dihydro-1H-isoquinolin-2-yl]acetyl]phenyl]quinoline-2-carboxamide
Show/Hide
|
C35H39N3O7
|
1
|
1 |
IC50 = 1130 nM
|
|
|
CP0448896
|
methyl 4-[4-(3,4-dihydro-1H-isoquinolin-2-ylmethyl)phenyl]-2-(quinoline-2-carbonylamino)benzoate
Show/Hide
|
C34H29N3O3
|
1
|
1 |
IC50 = 1461 nM
|
|
|
CP0455200
|
methyl 4-[4-[(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)methyl]phenyl]-2-(quinoline-6-carbonylamino)benzoate
Show/Hide
|
C36H33N3O5
|
1
|
1 |
IC50 = 1540 nM
|
|
|
CP0415663
|
N-[5-[(E)-3-[4-[2-[6-methoxy-7-(2-methoxyethoxy)-3,4-dihydro-1H-isoquinolin-2-yl]ethoxy]phenyl]prop-2-enoyl]-2-methylphenyl]quinoline-2-carboxamide
Show/Hide
|
C41H41N3O6
|
1
|
1 |
IC50 = 1550 nM
|
|
|
CP0398616
|
N-[2-(3,4-dimethoxyphenyl)ethyl]-4-oxo-5-phenylmethoxychromene-2-carboxamide
Show/Hide
|
C27H25NO6
|
1
|
1 |
IC50 = 1800 nM
|
|
|
CP0563380
|
methyl 4-bromo-2-(quinoline-2-carbonylamino)benzoate
Show/Hide
|
C18H13BrN2O3
|
1
|
1 |
IC50 = 1918 nM
|
|
|
CP0462357
|
N-[5-[[4-[2-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl]phenyl]carbamoyl]-2-methylphenyl]quinoline-3-carboxamide
Show/Hide
|
C37H36N4O4
|
1
|
1 |
IC50 = 1990 nM
|
|
|
CP0402761
|
N-[3-[(E)-3-[4-[2-[6-methoxy-7-(2-methoxyethoxy)-3,4-dihydro-1H-isoquinolin-2-yl]ethoxy]phenyl]prop-2-enoyl]phenyl]quinoline-2-carboxamide
Show/Hide
|
C40H39N3O6
|
1
|
1 |
IC50 = 2130 nM
|
|
|
CP0432680
|
(E)-1-naphthalen-2-yl-3-(3,4,5-trimethoxyphenyl)prop-2-en-1-one
Show/Hide
|
C22H20O4
|
1
|
1 |
IC50 = 2400 nM
|
|
|
CP0383918
|
N-[5-[(E)-3-[4-[2-[6-methoxy-7-[2-[2-(2-methoxyethoxy)ethoxy]ethoxy]-3,4-dihydro-1H-isoquinolin-2-yl]ethoxy]phenyl]prop-2-enoyl]-2-methylphenyl]quinoline-2-carboxamide
Show/Hide
|
C45H49N3O8
|
1
|
1 |
IC50 = 2720 nM
|
|
|
CP0415665
|
N-[3-[(E)-3-[4-[2-[6-methoxy-7-[2-[2-(2-methoxyethoxy)ethoxy]ethoxy]-3,4-dihydro-1H-isoquinolin-2-yl]ethoxy]phenyl]prop-2-enoyl]phenyl]quinoline-2-carboxamide
Show/Hide
|
C44H47N3O8
|
1
|
1 |
IC50 = 2830 nM
|
|
|
CP0417559
|
methyl 4-[4-[2-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl]phenyl]-2-(quinoline-2-carbonylamino)benzoate
Show/Hide
|
C37H35N3O5
|
1
|
1 |
IC50 = 3214 nM
|
|
|
CP0565380
|
6,7-dimethoxy-2-[2-[4-(4-phenyltriazol-1-yl)phenyl]ethyl]-3,4-dihydro-1H-isoquinoline
Show/Hide
|
C27H28N4O2
|
1
|
1 |
IC50 = 3606 nM
|
|
|
CP0466006
|
N-[3-[(E)-3-[4-[2-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethoxy]phenyl]prop-2-enoyl]phenyl]quinoline-2-carboxamide
Show/Hide
|
C38H35N3O5
|
1
|
1 |
IC50 = 4080 nM
|
|
|
CP0432681
|
(E)-3-(3-bromo-4,5-dimethoxyphenyl)-1-naphthalen-2-ylprop-2-en-1-one
Show/Hide
|
C21H17BrO3
|
1
|
1 |
IC50 = 4900 nM
|
|
|
CP0412836
|
N-[5-[2-[6-methoxy-7-[2-[2-(2-methoxyethoxy)ethoxy]ethoxy]-3,4-dihydro-1H-isoquinolin-2-yl]acetyl]-2-methylphenyl]quinoline-2-carboxamide
Show/Hide
|
C36H41N3O7
|
1
|
1 |
IC50 = 6650 nM
|
|
|
CP0415666
|
N-[3-[2-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)acetyl]phenyl]quinoline-2-carboxamide
Show/Hide
|
C29H27N3O4
|
1
|
1 |
IC50 = 6730 nM
|
|
|
CP0377046
|
1-[3-(3-iodo-4,5-dimethoxyphenyl)-5-naphthalen-2-yl-3,4-dihydropyrazol-2-yl]ethanone
Show/Hide
|
C23H21IN2O3
|
1
|
1 |
IC50 = 7100 nM
|
|
|
CP0442789
|
1-[3-(3-chloro-4,5-dimethoxyphenyl)-5-naphthalen-2-yl-3,4-dihydropyrazol-2-yl]ethanone
Show/Hide
|
C23H21ClN2O3
|
1
|
1 |
IC50 = 7400 nM
|
|
|
CP0377045
|
(E)-3-(3-iodo-4,5-dimethoxyphenyl)-1-naphthalen-2-ylprop-2-en-1-one
Show/Hide
|
C21H17IO3
|
1
|
1 |
IC50 = 7800 nM
|
|
|
CP0442791
|
(E)-3-(3-chloro-4,5-dimethoxyphenyl)-1-naphthalen-2-ylprop-2-en-1-one
Show/Hide
|
C21H17ClO3
|
1
|
1 |
IC50 = 8700 nM
|
|
|
CP0412837
|
N-[5-[2-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)acetyl]-2-methylphenyl]quinoline-2-carboxamide
Show/Hide
|
C30H29N3O4
|
1
|
1 |
IC50 = 8760 nM
|
|
|
CP0458758
|
1-[3-(3-bromo-4,5-dimethoxyphenyl)-5-naphthalen-2-yl-3,4-dihydropyrazol-2-yl]ethanone
Show/Hide
|
C23H21BrN2O3
|
1
|
1 |
IC50 = 8900 nM
|
|
|
CP0395102
|
5-hydroxy-7-methoxy-2-[4-[(4-nitrophenyl)methyl]piperazine-1-carbonyl]chromen-4-one
Show/Hide
|
C22H21N3O7
|
1
|
1 |
IC50 = 12000 nM
|
|
|
CP0388621
|
5,7-dimethoxy-2-[4-(4-nitrophenyl)piperazin-1-yl]chromen-4-one
Show/Hide
|
C21H21N3O6
|
1
|
1 |
IC50 = 12200 nM
|
|
|
CP0415667
|
N-[3-[2-[6-methoxy-7-(2-methoxyethoxy)-3,4-dihydro-1H-isoquinolin-2-yl]acetyl]phenyl]quinoline-2-carboxamide
Show/Hide
|
C31H31N3O5
|
1
|
1 |
IC50 = 14390 nM
|
|
|
CP0398446
|
2-(4-benzylpiperazine-1-carbonyl)-5-phenylmethoxychromen-4-one
Show/Hide
|
C28H26N2O4
|
1
|
1 |
IC50 = 16300 nM
|
|
|
CP0473594
|
N-[5-[2-[6-methoxy-7-(2-methoxyethoxy)-3,4-dihydro-1H-isoquinolin-2-yl]acetyl]-2-methylphenyl]quinoline-2-carboxamide
Show/Hide
|
C32H33N3O5
|
1
|
1 |
IC50 = 23240 nM
|
|
|
CP0462998
|
5-hydroxy-7-methoxy-2-[4-[(2-nitrophenyl)methyl]piperazine-1-carbonyl]chromen-4-one
Show/Hide
|
C22H21N3O7
|
1
|
1 |
IC50 = 34900 nM
|
|
|
CP0433316
|
5,7-dimethoxy-2-[4-[2-(4-nitrophenyl)ethyl]piperazin-1-yl]chromen-4-one
Show/Hide
|
C23H25N3O6
|
1
|
1 |
IC50 = 36900 nM
|
|
|
CP0406172
|
5,7-dimethoxy-2-[4-[(2-nitrophenyl)methyl]piperazin-1-yl]chromen-4-one
Show/Hide
|
C22H23N3O6
|
1
|
1 |
IC50 = 37600 nM
|
|
|
CP0474629
|
5,7-dimethoxy-2-[4-[(3-nitrophenyl)methyl]piperazin-1-yl]chromen-4-one
Show/Hide
|
C22H23N3O6
|
1
|
1 |
IC50 = 38200 nM
|
|
|
CP0898201
|
N-{4-[2-(7-Methoxy-6-{2-[2-(2-methoxy-ethoxy)-ethoxy]-ethoxy}-3,4-dihydro-1H-isoquinolin-2-yl)-ethyl]-phenyl}-2-[(quinoline-2-carbonyl)-amino]-terephthalamic acid trifluoroacetic acid
Show/Hide
|
C45H47F3N4O11
|
1
|
1 |
IC50 > 50000 nM
|
|
|
CP0904106
|
N-{4-[2-(6-Methoxy-7-{2-[2-(2-methoxy-ethoxy)-ethoxy]-ethoxy}-3,4-dihydro-1H-isoquinolin-2-yl)-ethyl]-phenyl}-2-[(quinoline-6-carbonyl)-amino]-terephthalamic acid trifluoroacetic acid
Show/Hide
|
C45H47F3N4O11
|
1
|
1 |
IC50 > 50000 nM
|
|
|
CP0904107
|
N-{4-[2-(7-Methoxy-6-{2-[2-(2-methoxy-ethoxy)-ethoxy]-ethoxy}-3,4-dihydro-1H-isoquinolin-2-yl)-ethyl]-phenyl}-2-[(quinoline-6-carbonyl)-amino]-terephthalamic acid trifluoroacetic acid
Show/Hide
|
C45H47F3N4O11
|
1
|
1 |
IC50 > 50000 nM
|
|
|
CP0390463
|
2-[4-[(3,4-difluorophenyl)methyl]piperazin-1-yl]-5,7-dimethoxychromen-4-one
Show/Hide
|
C22H22F2N2O4
|
1
|
1 |
IC50 = 66600 nM
|
|
|
CP0406265
|
5,7-dimethoxy-2-[4-[(4-nitrophenyl)methyl]piperazin-1-yl]chromen-4-one
Show/Hide
|
C22H23N3O6
|
1
|
1 |
IC50 = 87800 nM
|
|
|
CP0497740
|
4-[[4-(5,7-dimethoxy-4-oxochromen-2-yl)piperazin-1-yl]methyl]benzonitrile
Show/Hide
|
C23H23N3O4
|
1
|
1 |
IC50 = 99700 nM
|
|
|
CP0906528
|
N-{4-[2-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)-ethyl]-phenyl}-2-[(quinoline-6-carbonyl)-amino]-terephthalamic acid trifluoroacetic acid
Show/Hide
|
C39H35F3N4O8
|
1
|
1 |
IC50 > 100000 nM
|
|
|
CP0390465
|
methyl 4-[[4-(5,7-dimethoxy-4-oxochromen-2-yl)piperazin-1-yl]methyl]benzoate
Show/Hide
|
C24H26N2O6
|
1
|
1 |
IC50 > 100000 nM
|
|
|
CP0406171
|
5,7-dimethoxy-2-[4-(2-phenylethyl)piperazin-1-yl]chromen-4-one
Show/Hide
|
C23H26N2O4
|
1
|
1 |
IC50 > 100000 nM
|
|
|
CP0406173
|
5,7-dimethoxy-2-[4-[2-(4-nitrophenyl)ethyl]piperazine-1-carbonyl]chromen-4-one
Show/Hide
|
C24H25N3O7
|
1
|
1 |
IC50 > 100000 nM
|
|
|
CP0434377
|
5,7-dimethoxy-2-[4-[(4-nitrophenyl)methyl]piperazine-1-carbonyl]chromen-4-one
Show/Hide
|
C23H23N3O7
|
1
|
1 |
IC50 > 100000 nM
|
|
|
CP0434379
|
2-[2-(3,4-dimethoxyphenyl)ethylamino]-5,7-dimethoxychromen-4-one
Show/Hide
|
C21H23NO6
|
1
|
1 |
IC50 > 100000 nM
|
|
|
CP0448142
|
5,7-dimethoxy-2-[4-[(4-methoxyphenyl)methyl]piperazin-1-yl]chromen-4-one
Show/Hide
|
C23H26N2O5
|
1
|
1 |
IC50 > 100000 nM
|
|
|
CP0462997
|
5,7-dimethoxy-2-[4-[[4-(trifluoromethylsulfonyl)phenyl]methyl]piperazin-1-yl]chromen-4-one
Show/Hide
|
C23H23F3N2O6S
|
1
|
1 |
IC50 > 100000 nM
|
|
|
CP0483165
|
5,7-dimethoxy-2-[4-[[4-(trifluoromethylsulfanyl)phenyl]methyl]piperazin-1-yl]chromen-4-one
Show/Hide
|
C23H23F3N2O4S
|
1
|
1 |
IC50 > 100000 nM
|
|
|
CP0508791
|
5,7-dimethoxy-2-[4-[[4-(trifluoromethyl)phenyl]methyl]piperazin-1-yl]chromen-4-one
Show/Hide
|
C23H23F3N2O4
|
1
|
1 |
IC50 > 100000 nM
|
|
|
CP0486096
|
N-[5-[1-(2-hydroxyethyl)triazol-4-yl]-2-propanoylphenyl]-4-oxochromene-2-carboxamide
Show/Hide
|
C23H20N4O5
|
1
|
1 |
IC50 > 1102 nM
|
|
|
CP0898202
|
N-{4-[2-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)-ethyl]-phenyl}-2-[(quinoline-2-carbonyl)-amino]-terephthalamic acid trifluoroacetic acid
Show/Hide
|
C39H35F3N4O8
|
1
|
1 |
IC50 > 5000 nM
|
|
|
CP0878929
|
N-{4-[2-(6-Methoxy-7-{2-[2-(2-methoxy-ethoxy)-ethoxy]-ethoxy}-3,4-dihydro-1H-isoquinolin-2-yl)-ethyl]-phenyl}-2-[(quinoline-2-carbonyl)-amino]-terephthalamic acid trifluoroacetic acid
Show/Hide
|
C45H47F3N4O11
|
1
|
1 |
IC50 > 6200 nM
|
|
|