3-amino-N-[(2R)-3,3,3-trifluoro-2-hydroxypropyl]-5-[2-(trifluoromethoxy)phenyl]sulfonylpyridine-2-carboxamide

[3-amino-5-(4-fluorophenyl)sulfonylpyridin-2-yl]-[3-hydroxy-3-(trifluoromethyl)azetidin-1-yl]methanone

3-amino-N-[(1-hydroxycyclopropyl)methyl]-5-[4-(trifluoromethoxy)phenyl]sulfonylpyridine-2-carboxamide

3-amino-N-[(2R)-3,3,3-trifluoro-2-hydroxypropyl]-5-[4-(trifluoromethoxy)phenyl]sulfonylpyridine-2-carboxamide

3-amino-N-(3,3,3-trifluoro-2-hydroxypropyl)-5-[4-(trifluoromethoxy)piperidin-1-yl]sulfonylpyridine-2-carboxamide

3-amino-5-(4-fluorophenyl)sulfonyl-N-[(2R)-3,3,3-trifluoro-2-hydroxypropyl]pyridine-2-carboxamide

3-amino-N-[(2S)-2-hydroxypropyl]-5-[4-(trifluoromethoxy)phenyl]sulfonylpyridine-2-carboxamide

N-(3-carbamoyl-5-piperidin-1-ylsulfonylthiophen-2-yl)-1H-pyrazole-5-carboxamide

1-(1,3-benzodioxol-5-yl)-N-[4-phenyl-5-(4-propoxybenzoyl)-1,3-thiazol-2-yl]cyclopropane-1-carboxamide

N-[5-[benzyl(methyl)sulfamoyl]-3-carbamoylthiophen-2-yl]-1H-pyrazole-5-carboxamide

2-[(2-hydroxy-2-methylpropanoyl)amino]-5-(4-methoxyphenyl)sulfonylthiophene-3-carboxamide

5-(4-fluorophenyl)sulfonyl-2-[(2-hydroxy-2-methylpropanoyl)amino]thiophene-3-carboxamide

N-[3-carbamoyl-5-(4-fluorophenyl)sulfonylthiophen-2-yl]-1H-pyrazole-5-carboxamide

3-amino-N-(2-hydroxy-2-methylpropyl)-5-[4-(trifluoromethoxy)phenyl]sulfonylpyridine-2-carboxamide

1-(1,3-benzodioxol-5-yl)-N-[4-phenyl-5-(4-phenylbenzoyl)-1,3-thiazol-2-yl]cyclopropane-1-carboxamide

5-(4-fluorophenyl)sulfonyl-2-[(1-hydroxycyclopropanecarbonyl)amino]thiophene-3-carboxamide

1-(1,3-benzodioxol-5-yl)-N-[5-(3-methoxybenzoyl)-4-phenyl-1,3-thiazol-2-yl]cyclopropane-1-carboxamide

1-(1,3-benzodioxol-5-yl)-N-[5-(4-methylsulfanylbenzoyl)-4-phenyl-1,3-thiazol-2-yl]cyclopropane-1-carboxamide

N-[5-(1,3-benzodioxole-5-carbonyl)-4-phenyl-1,3-thiazol-2-yl]-1-(1,3-benzodioxol-5-yl)cyclopropane-1-carboxamide

1-(1,3-benzodioxol-5-yl)-N-[5-(2,5-dimethoxybenzoyl)-4-phenyl-1,3-thiazol-2-yl]cyclopropane-1-carboxamide

1-(2,2-difluorobenzo[d][1,3]dioxol-5-yl)-N-((2R,4R)-2-(3,4-dimethoxyphenyl)-7-methoxychroman-4-yl)cyclopropanecarboxamide

1-(1,3-benzodioxol-5-yl)-N-[5-(3-fluorobenzoyl)-4-phenyl-1,3-thiazol-2-yl]cyclopropane-1-carboxamide

1-(1,3-benzodioxol-5-yl)-N-[5-(2-methoxybenzoyl)-4-phenyl-1,3-thiazol-2-yl]cyclopropane-1-carboxamide

1-(1,3-benzodioxol-5-yl)-N-[4-phenyl-5-(3-propoxybenzoyl)-1,3-thiazol-2-yl]cyclopropane-1-carboxamide

1-(1,3-benzodioxol-5-yl)-N-[5-(3-bromobenzoyl)-4-phenyl-1,3-thiazol-2-yl]cyclopropane-1-carboxamide

N,N-dimethyl-2-[4-[2-pyridin-2-yl-6-(thiophen-3-ylmethyl)-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl]piperazin-1-yl]ethanamine

N-(3-imidazol-1-ylpropyl)-6-[(4-methoxyphenyl)methyl]-2-pyridin-2-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-amine

6-[(4-fluorophenyl)methyl]-2-pyridin-2-yl-N-(3-pyrrolidin-1-ylpropyl)-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-amine

N-[3-[[6-[(4-fluorophenyl)methyl]-2-pyridin-2-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl]amino]propyl]acetamide

1-(2,2-Difluoro-1,3-benzodioxol-5-yl)-N-[2-(3,4-dimethoxyphenyl)-7-methoxy-3,4-dihydro-2H-chromen-4-yl]cyclopropanecarboxamide

1-(1,3-benzodioxol-5-yl)-N-[5-[4-(diethylamino)benzoyl]-4-phenyl-1,3-thiazol-2-yl]cyclopropane-1-carboxamide

3-[(2R,4R)-4-({[1-(2,2-Difluoro-1,3-benzodioxol-5-yl)cyclopropyl]-carbonyl}amino)-7-methoxy-3,4-dihydro-2H-chromen-2-yl]benzoic acid

1-(1,3-benzodioxol-5-yl)-N-[4-phenyl-5-(3-phenylbenzoyl)-1,3-thiazol-2-yl]cyclopropane-1-carboxamide

3-[(2R,4S,6S)-4-[[1-(2,2-difluoro-1,3-benzodioxol-5-yl)cyclopropanecarbonyl]amino]-6-phenyloxan-2-yl]benzoic acid

1-(1,3-benzodioxol-5-yl)-N-[5-(4-hydroxy-3-prop-2-enylbenzoyl)-4-phenyl-1,3-thiazol-2-yl]cyclopropane-1-carboxamide

4-[(2R,4S,6S)-4-[[1-(2,2-difluoro-1,3-benzodioxol-5-yl)cyclopropanecarbonyl]amino]-6-phenyloxan-2-yl]benzoic acid

N,N-dimethyl-2-[4-[6-[(4-propan-2-ylphenyl)methyl]-2-pyridin-2-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl]piperazin-1-yl]ethanamine

N-ethyl-N-[1-[6-[(4-methoxyphenyl)methyl]-2-pyridin-2-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl]pyrrolidin-3-yl]acetamide

2-(2-chlorobenzamido)-4,5,6,7-tetrahydrobenzo[b]thiophene-3-carboxamide

2-(2,2-dimethylpropanoylamino)-5-(4-fluorophenyl)sulfonylthiophene-3-carboxamide

1-(1,3-benzodioxol-5-yl)-N-[4-phenyl-5-[4-(trifluoromethoxy)benzoyl]-1,3-thiazol-2-yl]cyclopropane-1-carboxamide

1-(1,3-benzodioxol-5-yl)-N-[4-phenyl-5-(4-pyrrolidin-1-ylbenzoyl)-1,3-thiazol-2-yl]cyclopropane-1-carboxamide

2-[4-[6-[(4-methoxyphenyl)methyl]-2-pyridin-2-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl]piperazin-1-yl]ethanol

1-(1,3-benzodioxol-5-yl)-N-[5-(2,4-dimethoxybenzoyl)-4-phenyl-1,3-thiazol-2-yl]cyclopropane-1-carboxamide

1-(1,3-benzodioxol-5-yl)-N-[5-(3-chloro-4-methoxybenzoyl)-4-phenyl-1,3-thiazol-2-yl]cyclopropane-1-carboxamide

ethyl 4-[2-[[1-(1,3-benzodioxol-5-yl)cyclopropanecarbonyl]amino]-4-phenyl-1,3-thiazole-5-carbonyl]benzoate

1-(1,3-benzodioxol-5-yl)-N-[5-(4-pentylbenzoyl)-4-phenyl-1,3-thiazol-2-yl]cyclopropane-1-carboxamide

1-(2,2-Difluoro-1,3-benzodioxol-5-yl)-N-(7-methoxy-2-phenyl-3,4-dihydro-2H-chromen-4-yl)cyclopropanecarboxamide

1-(1,3-benzodioxol-5-yl)-N-[5-(4-methoxybenzoyl)-4-phenyl-1,3-thiazol-2-yl]cyclopropane-1-carboxamide

1-(1,3-benzodioxol-5-yl)-N-[5-(4-bromobenzoyl)-4-phenyl-1,3-thiazol-2-yl]cyclopropane-1-carboxamide

MLS000561583

N-[1-[6-[(4-chlorophenyl)methyl]-2-pyridin-2-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl]piperidin-4-yl]acetamide

N,5-dibenzyl-3-[2-(2,2-dimethylpropanoylamino)-4-methyl-1,3-thiazol-5-yl]pyrazole-1-carboxamide

1-(1,3-benzodioxol-5-yl)-N-[4-phenyl-5-(pyridine-3-carbonyl)-1,3-thiazol-2-yl]cyclopropane-1-carboxamide

3-[(2R,4S)-4-[[1-(2,2-difluoro-1,3-benzodioxol-5-yl)cyclopropanecarbonyl]amino]oxan-2-yl]benzoic acid

2-[4-[6-(cyclohexylmethyl)-2-pyridin-2-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl]piperazin-1-yl]-N,N-dimethylethanamine

3-[2-(2,2-dimethylpropanoylamino)-4-methyl-1,3-thiazol-5-yl]-N-(4-methoxyphenyl)-5-prop-2-enylpyrazole-1-carboxamide

N-[2-(4-chlorophenyl)-3,4-dihydro-2H-chromen-4-yl]-1-(2,2-difluoro-1,3-benzodioxol-5-yl)cyclopropanecarboxamide

1-(2,2-Difluoro-1,3-benzodioxol-5-yl)-N-[(2S,4S)-2-(3,4-dimethoxyphenyl)-7-methoxy-3,4-dihydro-2H-chromen-4-yl]cyclopropanecarboxamide

5-[(5-chloro-2-methoxyphenyl)methyl]-3-[2-(2,2-dimethylpropanoylamino)-4-methyl-1,3-thiazol-5-yl]-N-(4-methoxyphenyl)pyrazole-1-carboxamide

N-[5-[5-[(5-chloro-2-methoxyphenyl)methyl]-1-(morpholine-4-carbonyl)pyrazol-3-yl]-4-methyl-1,3-thiazol-2-yl]-2,2-dimethylpropanamide

(2S,3S,4S,5S)-1-(cyclohexanecarbonyl)-3-(2-methoxypropan-2-yl)-4-[(2-methoxy-5-propan-2-ylpyridin-3-yl)methylamino]-5-phenylpyrrolidine-2-carboxylic acid

1-(1,3-benzodioxol-5-yl)-N-[4-phenyl-5-(4-thiophen-2-ylbenzoyl)-1,3-thiazol-2-yl]cyclopropane-1-carboxamide

N-[5-[2-(5-chloro-2-methoxyanilino)-1,3-thiazol-4-yl]-4-methyl-1,3-thiazol-2-yl]benzamide

ethyl 3-[(2R,4S,6S)-4-[[1-(2,2-difluoro-1,3-benzodioxol-5-yl)cyclopropanecarbonyl]amino]-6-phenyloxan-2-yl]-5-methylbenzoate

2-[[1-(1,3-benzodioxol-5-yl)cyclopropanecarbonyl]amino]-N,4-diphenyl-1,3-thiazole-5-carboxamide

1-(6-benzyl-2-pyridin-2-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl)piperidine-4-carboxamide

2-[4-(6-benzyl-2-pyridin-2-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl)piperazin-1-yl]-N,N-dimethylethanamine

N-[2-[(3-cyano-5,7-dimethylquinolin-2-yl)amino]ethyl]-3,4-dimethoxybenzamide

1-(2,2-difluoro-1,3-benzodioxol-5-yl)-N-{(2R)-2-[3-(hydroxymethyl)phenyl]-3,4-dihydro-2H-chromen-4-yl}cyclopropanecarboxamide

1-(1,3-benzodioxol-5-yl)-N-[5-(5-chloro-2-hydroxybenzoyl)-4-phenyl-1,3-thiazol-2-yl]cyclopropane-1-carboxamide

N-[2-[[1-(1,3-benzodioxol-5-yl)cyclopropanecarbonyl]amino]-4-(4-methoxyphenyl)-1,3-thiazol-5-yl]benzamide

(2S,3R,4S,5R)-1-benzoyl-3-tert-butyl-4-(2,5-dichlorobenzoyl)-5-phenylpyrrolidine-2-carboxylic acid

(2S,3R,4S,5R)-3-tert-butyl-1-(cyclohexanecarbonyl)-4-(2,5-dichlorobenzoyl)-5-phenylpyrrolidine-2-carboxylic acid

1-benzoyl-3-tert-butyl-4-(2,5-dichlorobenzoyl)-5-phenylpyrrolidine-2-carboxylic acid

4-cyclohexyloxy-2-[1-[4-(4-methoxyphenyl)sulfonylpiperazin-1-yl]ethyl]quinazoline

N-[2-[(3-cyano-5,7-dimethylquinolin-2-yl)amino]ethyl]-3-methoxybenzamide

2-[4-[6-[(4-methoxyphenyl)methyl]-2-pyridin-2-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl]piperazin-1-yl]acetamide

N-[(4R)-8-chloro-7-fluoro-2,2-dimethyl-3,4-dihydro-2H-chromen-4-yl]-1-(2,2-difluoro-1,3-benzodioxol-5-yl)cyclopropanecarboxamide

1-(2,2-difluoro-1,3-benzodioxol-5-yl)-N-[2-(4-fluorophenyl)-3,4-dihydro-2H-chromen-4-yl]cyclopropanecarboxamide

1-(2,2-difluoro-1,3-benzodioxol-5-yl)-N-(2-phenyl-3,4-dihydro-2H-chromen-4-yl)cyclopropanecarboxamide

1-(1,3-benzodioxol-5-yl)-N-[5-(4-methylbenzoyl)-1,3-thiazol-2-yl]cyclopropane-1-carboxamide

Lumacaftor

N-[2-[(3-cyano-5,7-dimethylquinolin-2-yl)amino]ethyl]pyridine-3-carboxamide

N-[2-[(3-cyano-5,7-dimethylquinolin-2-yl)amino]ethyl]-5-methoxypyridine-2-carboxamide

1-(2,2-Difluoro-1,3-benzodioxol-5-yl)-N-[(4R)-7-fluoro-2,2-dimethyl-3,4-dihydro-2H-chromen-4-yl]cyclopropanecarboxamide

N-(5-acetyl-4-phenyl-1,3-thiazol-2-yl)-1-(1,3-benzodioxol-5-yl)cyclopropane-1-carboxamide

1-(6-benzyl-2-pyridin-2-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl)piperidin-3-ol

2-[4-(6-benzyl-2-pyridin-2-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl)piperazin-1-yl]acetamide

4-[(2R,4S)-4-[[1-(2,2-difluoro-1,3-benzodioxol-5-yl)cyclopropanecarbonyl]amino]oxan-2-yl]benzoic acid

N-[2-[(3-cyano-5,7-dimethylquinolin-2-yl)amino]ethyl]-4-methoxybenzamide

N-[3-[(3-cyano-5,7-dimethylquinolin-2-yl)amino]propyl]pyridine-3-carboxamide

3-[2-(2,2-dimethylpropanoylamino)-4-methyl-1,3-thiazol-5-yl]-N-phenyl-5-prop-2-enylpyrazole-1-carboxamide

5-[(5-chloro-2-methoxyphenyl)methyl]-3-[2-(2,2-dimethylpropanoylamino)-4-methyl-1,3-thiazol-5-yl]-N-(2-hydroxyethyl)pyrazole-1-carboxamide

6-benzyl-N-[3-(4-methylpiperazin-1-yl)propyl]-2-pyridin-2-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-amine

1-(4-bromophenyl)-5-[2-(2,2-dimethylpropanoylamino)-4-methyl-1,3-thiazol-5-yl]-N-(4-methoxyphenyl)pyrazole-3-carboxamide

1-[6-[(4-methoxyphenyl)methyl]-2-pyridin-2-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl]piperidine-4-carboxamide

N-[2-[(3-cyano-5,7-dimethylquinolin-2-yl)amino]ethyl]-2,6-dimethoxybenzamide

N-[2-(3-chlorophenyl)-3,4-dihydro-2H-chromen-4-yl]-1-(2,2-difluoro-1,3-benzodioxol-5-yl)cyclopropanecarboxamide

N-[2-[(3-cyano-5,7-dimethylquinolin-2-yl)amino]ethyl]-2,4-dimethoxybenzamide

N-[3-[(3-cyano-5,7-dimethylquinolin-2-yl)amino]propyl]-4-methoxybenzamide

1-(2,2-difluoro-1,3-benzodioxol-5-yl)-N-[(4R)-7-fluoro-2,2-bis(fluoromethyl)-3,4-dihydro-2H-chromen-4-yl]cyclopropanecarboxamide

N-[3-[(3-cyano-5,7-dimethylquinolin-2-yl)amino]propyl]-3-methoxybenzamide

4-(3-chlorophenyl)-N-(3-methylsulfanylphenyl)-1,3-thiazol-2-amine

4-(4-methyl-2-phenyl-1,3-thiazol-5-yl)-N-(3-methylsulfanylphenyl)-1,3-thiazol-2-amine

6-[2-(3-methylsulfanylanilino)-1,3-thiazol-4-yl]-3H-1,3-benzoxazol-2-one

N-[2-[(3-cyano-5,7-dimethylquinolin-2-yl)amino]ethyl]pyrazine-2-carboxamide

N-[2-[(3-cyano-5,7-dimethylquinolin-2-yl)amino]ethyl]pyridine-4-carboxamide

4-[2-[[1-(1,3-benzodioxol-5-yl)cyclopropanecarbonyl]amino]-4-phenyl-1,3-thiazole-5-carbonyl]benzoic acid

N-(3-methylsulfanylphenyl)-4-thiophen-2-yl-1,3-thiazol-2-amine

1-(1,3-benzodioxol-5-yl)-N-[5-(morpholine-4-carbonyl)-4-phenyl-1,3-thiazol-2-yl]cyclopropane-1-carboxamide

ethyl 5-benzyl-3-[2-(2,2-dimethylpropanoylamino)-4-methyl-1,3-thiazol-5-yl]pyrazole-1-carboxylate

1-(1,3-benzodioxol-5-yl)-N-[5-(4-methoxybenzoyl)-1,3-thiazol-2-yl]cyclopropane-1-carboxamide

N-(3-methylsulfanylphenyl)-4-(1,3-thiazol-2-yl)-1,3-thiazol-2-amine

MLS001204421

N-[2-(2-chlorophenyl)-3,4-dihydro-2H-chromen-4-yl]-1-(2,2-difluoro-1,3-benzodioxol-5-yl)cyclopropanecarboxamide

N-[3-[(3-cyano-5,7-dimethylquinolin-2-yl)amino]propyl]pyridine-4-carboxamide

5-[2-[[1-(1,3-benzodioxol-5-yl)cyclopropanecarbonyl]amino]-4-phenyl-1,3-thiazole-5-carbonyl]-2-hydroxybenzamide

4-(3,4-dichlorophenyl)-N-(3-methylsulfanylphenyl)-1,3-thiazol-2-amine

4-(4-chlorothiophen-2-yl)-N-(3-methylsulfanylphenyl)-1,3-thiazol-2-amine

1-(2,2-Difluoro-1,3-benzodioxol-5-yl)-N-[(4S)-6-fluoro-2,2-dimethyl-3,4-dihydro-2H-chromen-4-yl]cyclopropanecarboxamide

3-[(2S,4R,6R)-4-[[1-(2,2-difluoro-1,3-benzodioxol-5-yl)cyclopropanecarbonyl]amino]-6-phenyloxan-2-yl]benzoic acid

4-(4-fluorophenyl)-N-(3-methylsulfanylphenyl)-1,3-thiazol-2-amine

4-(3-chlorophenyl)-N-[3-(trifluoromethylsulfanyl)phenyl]-1,3-thiazol-2-amine

4-[2-(3-methylsulfanylanilino)-1,3-thiazol-4-yl]benzonitrile

ethyl 5-[2-(3-methylsulfanylanilino)-1,3-thiazol-4-yl]-1,2-oxazole-3-carboxylate

4-(1,3-benzodioxol-5-yl)-N-(3-methylsulfanylphenyl)-1,3-thiazol-2-amine

2-[4-(6-benzyl-2-pyridin-4-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl)piperazin-1-yl]-N,N-dimethylethanamine

N-[1-[6-[(4-chlorophenyl)methyl]-2-pyridin-2-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl]pyrrolidin-3-yl]-N-ethylacetamide

2-[4-(6-benzyl-2-pyridin-3-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl)piperazin-1-yl]acetamide

6-benzyl-N-[3-(4-methylpiperazin-1-yl)propyl]-2-pyridin-3-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-amine

[4-[4-[2-(dimethylamino)ethyl]piperazin-1-yl]-2-pyridin-2-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl]-phenylmethanone

6-benzyl-N-[3-(4-methylpiperazin-1-yl)propyl]-2-pyridin-4-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-amine

2-[4-[6-(benzenesulfonyl)-2-pyridin-2-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl]piperazin-1-yl]-N,N-dimethylethanamine

2-[4-[6-[(4-fluorophenyl)methyl]-2-pyridin-2-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl]piperazin-1-yl]-N,N-dimethylethanamine

N-[2-[(3-cyano-5,7-dimethylquinolin-2-yl)amino]ethyl]pyridine-2-carboxamide

1-(6-benzyl-2-pyridin-3-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl)piperidine-4-carboxamide

2-[4-(3-methoxybenzoyl)piperazin-1-yl]-5,7-dimethylquinoline-3-carbonitrile

2-[4-(4-methoxybenzoyl)piperazin-1-yl]-5,7-dimethylquinoline-3-carbonitrile

2-[4-(6-benzyl-2-pyridin-3-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl)piperazin-1-yl]-N,N-dimethylethanamine

2-[4-(2-methoxybenzoyl)piperazin-1-yl]-5,7-dimethylquinoline-3-carbonitrile

2-[4-[6-[(4-methoxyphenyl)methyl]-2-pyridin-2-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl]piperazin-1-yl]-N,N-dimethylethanamine

5,7-dimethyl-2-[4-(pyridine-2-carbonyl)piperazin-1-yl]quinoline-3-carbonitrile

N-[3-[(3-cyano-5,7-dimethylquinolin-2-yl)amino]propyl]pyridine-2-carboxamide

N-[3-[(3-cyano-5,7-dimethylquinolin-2-yl)amino]propyl]-2-methoxybenzamide

N-[2-[(3-cyano-5,7-dimethylquinolin-2-yl)amino]ethyl]benzamide

5,7-dimethyl-2-[4-(pyridine-4-carbonyl)piperazin-1-yl]quinoline-3-carbonitrile

5,7-dimethyl-2-[4-(pyridine-3-carbonyl)piperazin-1-yl]quinoline-3-carbonitrile

(2S,3S,4S,5S)-3-tert-butyl-1-(cyclohexanecarbonyl)-4-[[5-(2,3-difluorophenyl)-2-methoxyphenyl]methylamino]-5-phenylpyrrolidine-2-carboxylic acid

(2S,3S,4S,5S)-3-tert-butyl-4-[[2-methoxy-5-(1-methylcyclobutyl)phenyl]methylamino]-5-(2-methylphenyl)-1-[(2S)-oxane-2-carbonyl]pyrrolidine-2-carboxylic acid

(2S,3S,4S,5S)-3-tert-butyl-1-(cyclohexanecarbonyl)-4-[(3-methoxy-5,5,8,8-tetramethyl-6,7-dihydronaphthalen-2-yl)methylamino]-5-phenylpyrrolidine-2-carboxylic acid

(2S,3S,4S,5S)-3-tert-butyl-4-[(2,2-dimethyl-3H-1-benzofuran-7-yl)methylamino]-1-[(2S)-oxane-2-carbonyl]-5-(2-propan-2-ylphenyl)pyrrolidine-2-carboxylic acid

(2S,3S,4S,5S)-3-tert-butyl-1-(cyclohexanecarbonyl)-4-[(2-methoxy-5-trimethylsilylphenyl)methylamino]-5-phenylpyrrolidine-2-carboxylic acid

(2S,3S,4S,5S)-3-tert-butyl-4-[(5-tert-butyl-2-methoxyphenyl)methylamino]-1-(cyclohexanecarbonyl)-5-[2-(dimethylamino)pyridin-3-yl]pyrrolidine-2-carboxylic acid

(2S,3S,4S,5S)-3-tert-butyl-4-[(5-tert-butyl-2-methoxyphenyl)methylamino]-1-[(2S)-2,3-dihydro-1-benzofuran-2-carbonyl]-5-phenylpyrrolidine-2-carboxylic acid

(2S,3S,4S,5S)-3-tert-butyl-4-[(5-cyclobutyl-2-methoxypyridin-3-yl)methylamino]-1-(cyclohexanecarbonyl)-5-(2-methylphenyl)pyrrolidine-2-carboxylic acid

[3-amino-5-[4-(trifluoromethyl)phenyl]sulfonylpyridin-2-yl]-[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]methanone

3-amino-5-(4-fluorophenyl)sulfonyl-N-methyl-N-[(2R)-3,3,3-trifluoro-2-hydroxypropyl]pyridine-2-carboxamide