Compound ID |
Compound Name |
Compound Formula |
CP0941656
|
SID131413872
Show/Hide
|
C30H32N4O7S
|
1
|
1 |
AC50 = 264 nM
|
|
|
CP0654294
|
SID87677872
Show/Hide
|
C14H21ClN4S
|
1
|
1 |
AC50 = 267 nM
|
|
|
CP0821924
|
SID26661232
Show/Hide
|
C28H23N3O5
|
1
|
1 |
AC50 = 286 nM
|
|
|
CP0667245
|
4-amino-7-((2R,3R,4S,5R)-3,4-dihydroxy-5-(hydroxymethyl)tetrahydrofuran-2-yl)-7H-pyrrolo[2,3-d]pyrimidine-5-carbothioamide
Show/Hide
|
C12H15N5O4S
|
1
|
1 |
AC50 = 294 nM
|
|
|
CP0313028
|
3-(2-methoxyphenyl)-6-p-phenetyl-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine
Show/Hide
|
C19H18N4O2S
|
1
|
1 |
AC50 = 317 nM
|
|
|
CP0133489
|
2-(3-chloro-N-(2-chloro-1-oxoethyl)-4-methoxyanilino)-N-(2-phenylethyl)-2-thiophen-2-ylacetamide
Show/Hide
|
C23H22Cl2N2O3S
|
1
|
1 |
AC50 = 323 nM
|
|
|
CP0418031
|
2,3,4-trihydroxy-3,4,4a,5-tetrahydro-2H-[1,3]dioxolo[4,5-j]phenanthridin-6-one
Show/Hide
|
C14H13NO6
|
1
|
1 |
AC50 = 325 nM
|
|
|
CP0865239
|
SID92763929
Show/Hide
|
C49H76O19
|
1
|
1 |
AC50 = 345 nM
|
|
|
CP0847686
|
SID51090288
Show/Hide
|
C20H23NO5
|
1
|
1 |
AC50 = 370 nM
|
|
|
CP0429330
|
MLS001065900
Show/Hide
|
C19H20N2O2S
|
1
|
1 |
AC50 = 379 nM
|
|
|
CP0054979
|
DIGOXIN
Show/Hide
|
C41H64O14
|
1
|
1 |
AC50 = 414 nM
|
|
|
CP0921060
|
SID92763413
Show/Hide
|
C25H34O10
|
1
|
1 |
AC50 = 426 nM
|
|
|
CP0887200
|
SID99356072
Show/Hide
|
C17H13ClN2O3S
|
1
|
1 |
AC50 = 449 nM
|
|
|
CP0908025
|
SID134215382
Show/Hide
|
C28H27FO8
|
1
|
1 |
AC50 = 465 nM
|
|
|
CP0411497
|
2-(9-hydroxy-1-methyl-5,10-dioxo-3,4-dihydro-1H-benzo[g][2]benzopyran-3-yl)acetic acid
Show/Hide
|
C16H14O6
|
1
|
1 |
AC50 = 469 nM
|
|
|
CP0886278
|
SID85812889
Show/Hide
|
C27H36N6O4S
|
1
|
1 |
AC50 = 480 nM
|
|
|
CP0447170
|
2-(N-(2-chloro-1-oxoethyl)-4-methylanilino)-N-cyclohexyl-2-(4-methoxyphenyl)acetamide
Show/Hide
|
C24H29ClN2O3
|
1
|
1 |
AC50 = 533 nM
|
|
|
CP0858621
|
SID121284991
Show/Hide
|
C24H29N7OS
|
1
|
1 |
AC50 = 538 nM
|
|
|
CP0871543
|
SID92763388
Show/Hide
|
C14H20Cl2N2O6
|
1
|
1 |
AC50 = 546 nM
|
|
|
CP0885641
|
SID56463219
Show/Hide
|
C22H30ClN7O5
|
1
|
1 |
AC50 = 546 nM
|
|
|
CP0884688
|
6-Amino-8-(3,4,5-trimethoxyphenyl)-8H-[1,3]dioxolo[4,5-g]chromene-7-carbonitrile
Show/Hide
|
C20H18N2O6
|
1
|
1 |
AC50 = 553 nM
|
|
|
CP0752656
|
SID24835936
Show/Hide
|
C16H13ClN2OS
|
1
|
1 |
AC50 = 572 nM
|
|
|
CP0862634
|
SID56322476
Show/Hide
|
C19H20N2O5S
|
1
|
1 |
AC50 = 619 nM
|
|
|
CP0652574
|
SID24815158
Show/Hide
|
C15H14N2O4
|
1
|
1 |
AC50 = 635 nM
|
|
|
CP0759343
|
SID49680425
Show/Hide
|
C20H18ClN3O3
|
1
|
1 |
AC50 = 650 nM
|
|
|
CP0905919
|
SID121283285
Show/Hide
|
C29H35NO5
|
1
|
1 |
AC50 = 673 nM
|
|
|
CP0342820
|
2-Chloro-N-[2,2,2-trifluoro-1-(6-nitro-benzothiazol-2-ylamino)-1-trifluoromethyl-ethyl]-benzamide
Show/Hide
|
C17H9ClF6N4O3S
|
1
|
1 |
AC50 = 676 nM
|
|
|
CP0884737
|
4-heptyl-2,3,5,6,7,8-hexahydro-1H-cyclopenta[b]quinolin-9-imine;hydrobromide
Show/Hide
|
C19H31BrN2
|
1
|
1 |
AC50 = 677 nM
|
|
|
CP0692800
|
SID50106605
Show/Hide
|
C22H30Cl2N4O6
|
1
|
1 |
AC50 = 690 nM
|
|
|
CP0386922
|
4-[(2,6-dibromo-4-methyl-phenoxy)methyl]-N'-[(Z)-pyrrol-2-ylidenemethyl]benzohydrazide
Show/Hide
|
C20H17Br2N3O2
|
1
|
1 |
AC50 = 693 nM
|
|
|
CP0386935
|
MLS001234557
Show/Hide
|
C21H25N3O5S
|
1
|
1 |
AC50 = 709 nM
|
|
|
CP0895291
|
SID49824126
Show/Hide
|
C24H22N2O5
|
1
|
1 |
AC50 = 728 nM
|
|
|
CP0912666
|
SID164339393
Show/Hide
|
C25H23N3O2S
|
1
|
1 |
AC50 = 733 nM
|
|
|
CP0426501
|
4-(2-cyclopropyl-1,3-oxazol-5-yl)-N-(2-methoxy-5-methyl-phenyl)benzenesulfonamide
Show/Hide
|
C20H20N2O4S
|
1
|
1 |
AC50 = 734 nM
|
|
|
CP0307430
|
Helenalin acetate
Show/Hide
|
C17H20O5
|
1
|
1 |
AC50 = 742 nM
|
|
|
CP0850666
|
SID85146197
Show/Hide
|
C15H10N6O2S2
|
1
|
1 |
AC50 = 747 nM
|
|
|
CP0907963
|
SID92764525
Show/Hide
|
C17H19N5O5
|
1
|
1 |
AC50 = 759 nM
|
|
|
CP0885259
|
SID17507542
Show/Hide
|
C22H20N2O2
|
1
|
1 |
AC50 = 770 nM
|
|
|
CP0480682
|
4H-Imidazo[4,5-d]-v-triazin-4-one, 3,7-dihydro-7-.beta.-D-ribofuranosyl-
Show/Hide
|
C9H11N5O5
|
1
|
1 |
AC50 = 785 nM
|
|
|
CP0900643
|
SID85811243
Show/Hide
|
C32H37F3N4O6S
|
1
|
1 |
AC50 = 799 nM
|
|
|
CP0432063
|
Lanatoside-C
Show/Hide
|
C49H76O20
|
1
|
1 |
AC50 = 801 nM
|
|
|
CP0897508
|
SID92764012
Show/Hide
|
C29H44O10
|
1
|
1 |
AC50 = 809 nM
|
|
|
CP0673299
|
SID49724927
Show/Hide
|
C17H10F3N3O3
|
1
|
1 |
AC50 = 811 nM
|
|
|
CP0865662
|
SID92763380
Show/Hide
|
C29H33NO11
|
1
|
1 |
AC50 = 833 nM
|
|
|
CP0411574
|
IRINOTECAN HCl )trihydrate)
Show/Hide
|
C33H41ClN4O7
|
1
|
1 |
AC50 = 844 nM
|
|
|
CP0250486
|
(2Z,4Z)-8-methyl-2,4-bis(2-pyridinylmethylidene)-8-azabicyclo[3.2.1]octan-3-one
Show/Hide
|
C20H19N3O
|
1
|
1 |
AC50 = 852 nM
|
|
|
CP0314157
|
5-nitro-2-(2-pyrrolidin-1-ylethyl)benzo[de]isoquinoline-1,3-dione
Show/Hide
|
C18H17N3O4
|
1
|
1 |
AC50 = 870 nM
|
|
|
CP0838009
|
SID851517
Show/Hide
|
C23H27N3O5S2
|
1
|
1 |
AC50 = 871 nM
|
|
|
CP0881646
|
SID57260400
Show/Hide
|
C22H26N6O3
|
1
|
1 |
AC50 = 879 nM
|
|
|
CP0912662
|
SID131448213
Show/Hide
|
C24H27FN2O2
|
1
|
1 |
AC50 = 895 nM
|
|
|
CP0701025
|
SID24801420
Show/Hide
|
C24H30BrN3OS
|
1
|
1 |
AC50 = 906 nM
|
|
|
CP0376097
|
MLS001123206
Show/Hide
|
C23H23ClN2O4S
|
1
|
1 |
AC50 = 921 nM
|
|
|
CP0897595
|
SID17432774
Show/Hide
|
C20H22N2O3
|
1
|
1 |
AC50 = 929 nM
|
|
|
CP0886257
|
SID14733294
Show/Hide
|
C24H27N3O5S
|
1
|
1 |
AC50 = 931 nM
|
|
|
CP0912548
|
SID99360537
Show/Hide
|
C20H19ClN2O5
|
1
|
1 |
AC50 = 966 nM
|
|
|
CP0039843
|
2-methyl-4,5-dioxo-3H-benzo[e]indole-1-carboxylic acid ethyl ester
Show/Hide
|
C16H13NO4
|
1
|
1 |
AC50 = 1050 nM
|
|
|
CP0158825
|
1-amino-8-methoxy-benzo[f]quinazoline-7,10-quinone
Show/Hide
|
C13H9N3O3
|
1
|
1 |
AC50 = 1060 nM
|
|
|
CP0902497
|
SID87334312
Show/Hide
|
C24H19FO5
|
1
|
1 |
AC50 = 1080 nM
|
|
|
CP0874166
|
SID103074497
Show/Hide
|
C24H29N3O2
|
1
|
1 |
AC50 = 1090 nM
|
|
|
CP0178113
|
9-Glycineamido-20(S)-camptothecin.HCl
Show/Hide
|
C22H21ClN4O5
|
1
|
1 |
AC50 = 1110 nM
|
|
|
CP0856715
|
SID92763873
Show/Hide
|
C27H21Cl2N3O7
|
1
|
1 |
AC50 = 1110 nM
|
|
|
CP0851436
|
SID92763407
Show/Hide
|
C23H33NO6
|
1
|
1 |
AC50 = 1120 nM
|
|
|
CP0090336
|
3-[(4-methoxyphenoxy)methyl]-N-(4-nitro-1-pyrazolyl)benzamide
Show/Hide
|
C18H16N4O5
|
1
|
1 |
AC50 = 1130 nM
|
|
|
CP0480193
|
2-amino-9-[(2R,3R,4S,5R)-3,4-dihydroxy-5-(hydroxymethyl)-2-oxolanyl]-3H-purine-6-thione
Show/Hide
|
C10H13N5O4S
|
1
|
1 |
AC50 = 1160 nM
|
|
|
CP0673671
|
SID51085196
Show/Hide
|
C16H19ClN4O5S
|
1
|
1 |
AC50 = 1160 nM
|
|
|
CP0686770
|
(1R,2R,4R,8S,9R,10S,13S,16R)-2,8,16-trihydroxy-5,5,9-trimethyl-14-methylidenetetracyclo[11.2.1.0^{1,10}.0^{4,9}]hexadecan-15-one
Show/Hide
|
C20H30O4
|
1
|
1 |
AC50 = 1160 nM
|
|
|
CP0905179
|
SID144194047
Show/Hide
|
C22H21N3O
|
1
|
1 |
AC50 = 1160 nM
|
|
|
CP0942498
|
SID92763332
Show/Hide
|
C17H13N3O2
|
1
|
1 |
AC50 = 1170 nM
|
|
|
CP0075498
|
2-Amino-1,7-dihydro-purine-6-thione
Show/Hide
|
C5H5N5S
|
1
|
1 |
AC50 = 1180 nM
|
|
|
CP0699254
|
SID24813175
Show/Hide
|
C18H17N3O4S
|
1
|
1 |
AC50 = 1190 nM
|
|
|
CP0865134
|
SID87543717
Show/Hide
|
C29H36Cl2N4O6S
|
1
|
1 |
AC50 = 1190 nM
|
|
|
CP0907410
|
SID144194087
Show/Hide
|
C21H21FN2O
|
1
|
1 |
AC50 = 1200 nM
|
|
|
CP0010269
|
MLS001211083
Show/Hide
|
C23H26N2O2
|
1
|
1 |
AC50 = 1210 nM
|
|
|
CP0134143
|
6-amino-7-bromo-quinoline-5,8-quinone
Show/Hide
|
C9H5BrN2O2
|
1
|
1 |
AC50 = 1220 nM
|
|
|
CP0407999
|
2-bromo-N-(3-ethoxypropyl)-11-ethyldibenzo[b,f][1,4]thiazepine-8-carboxamide
Show/Hide
|
C21H23BrN2O2S
|
1
|
1 |
AC50 = 1220 nM
|
|
|
CP0152855
|
2-[[2-keto-2-(3-keto-2,4-dihydroquinoxalin-1-yl)ethyl]thio]-6,8-dimethyl-quinoline-3-carbonitrile
Show/Hide
|
C22H18N4O2S
|
1
|
1 |
AC50 = 1250 nM
|
|
|
CP0926614
|
SID144194095
Show/Hide
|
C22H21N3O
|
1
|
1 |
AC50 = 1250 nM
|
|
|
CP0332729
|
Furan-2-carboxylic acid [5-(2,2-dimethyl-propionylamino)-pyridin-2-yl]-amide
Show/Hide
|
C15H17N3O3
|
1
|
1 |
AC50 = 1260 nM
|
|
|
CP0489161
|
(3S)-2-(2-chloro-1-oxoethyl)-1,1-dimethyl-4,9-dihydro-3H-pyrido[3,4-b]indole-3-carboxylic acid methyl ester
Show/Hide
|
C17H19ClN2O3
|
1
|
1 |
AC50 = 1260 nM
|
|
|
CP0407261
|
4-(4-chlorophenyl)sulfanyl-1-(trifluoromethyl)-[1,2,4]triazolo[4,3-a]quinoxaline
Show/Hide
|
C16H8ClF3N4S
|
1
|
1 |
AC50 = 1270 nM
|
|
|
CP0698372
|
SID49678797
Show/Hide
|
C20H22N4O4S
|
1
|
1 |
AC50 = 1270 nM
|
|
|
CP0167829
|
MLS001140457
Show/Hide
|
C26H25N3O6S
|
1
|
1 |
AC50 = 1290 nM
|
|
|
CP0880917
|
SID99205795
Show/Hide
|
C22H26ClN3O3
|
1
|
1 |
AC50 = 1300 nM
|
|
|
CP0844824
|
SID24825554
Show/Hide
|
C13H13ClN2OS
|
1
|
1 |
AC50 = 1310 nM
|
|
|
CP0907800
|
SID124755249
Show/Hide
|
C30H33Cl2N3O6
|
1
|
1 |
AC50 = 1330 nM
|
|
|
CP0068790
|
2-chloranyl-N-(1-ethanoylindol-3-yl)-N-phenyl-ethanamide
Show/Hide
|
C18H15ClN2O2
|
1
|
1 |
AC50 = 1340 nM
|
|
|
CP0738005
|
SID24825651
Show/Hide
|
C12H9Cl3N2OS
|
1
|
1 |
AC50 = 1360 nM
|
|
|
CP0812816
|
SID849093
Show/Hide
|
C10H9BrN6
|
1
|
1 |
AC50 = 1360 nM
|
|
|
CP0882034
|
SID99495763
Show/Hide
|
C17H13F3N2O3
|
1
|
1 |
AC50 = 1370 nM
|
|
|
CP0090178
|
3-[(3S,5R,8R,9S,10S,13R,14S,17R)-10,13-dimethyl-3,14-bis(oxidanyl)-1,2,3,4,5,6,7,8,9,11,12,15,16,17-tetradecahydrocyclopenta[a]phenanthren-17-yl]-2H-furan-5-one
Show/Hide
|
C23H34O4
|
1
|
1 |
AC50 = 1380 nM
|
|
|
CP0891430
|
SID24835896
Show/Hide
|
C26H25N3O7S
|
1
|
1 |
AC50 = 1380 nM
|
|
|
CP0857038
|
SID121284983
Show/Hide
|
C29H31N7O
|
1
|
1 |
AC50 = 1400 nM
|
|
|
CP0658193
|
SID57264490
Show/Hide
|
C21H19ClN2O4
|
1
|
1 |
AC50 = 1410 nM
|
|
|
CP0885723
|
SID87543554
Show/Hide
|
C37H45F4N5O6
|
1
|
1 |
AC50 = 1410 nM
|
|
|
CP0447723
|
2-(N-(2-chloroacetyl)-4-fluoroanilino)-N-cyclohexyl-2-pyridin-3-ylacetamide
Show/Hide
|
C21H23ClFN3O2
|
1
|
1 |
AC50 = 1430 nM
|
|
|
CP0897221
|
SID92763835
Show/Hide
|
C22H30O5
|
1
|
1 |
AC50 = 1430 nM
|
|
|
CP0201524
|
7-amino-6-chloro-5,8-diketo-naphthalene-2-sulfonamide
Show/Hide
|
C10H7ClN2O4S
|
1
|
1 |
AC50 = 1470 nM
|
|
|
CP0419010
|
4-(4-acetamidophenyl)-N-(phenylmethyl)-2,3-dihydrofuro[2,3-b]pyridine-2-carboxamide
Show/Hide
|
C23H21N3O3
|
1
|
1 |
AC50 = 1500 nM
|
|
|
CP0879706
|
SID121283276
Show/Hide
|
C19H18N6O4
|
1
|
1 |
AC50 = 1500 nM
|
|
|
CP0905592
|
SID121284949
Show/Hide
|
C30H31N7O5
|
1
|
1 |
AC50 = 1520 nM
|
|
|
CP0924104
|
SID92763379
Show/Hide
|
C29H33NO10
|
1
|
1 |
AC50 = 1520 nM
|
|
|
CP0925849
|
SID17402854
Show/Hide
|
C16H8ClF3N4S
|
1
|
1 |
AC50 = 1520 nM
|
|
|
CP0908685
|
SID24830873
Show/Hide
|
C16H12N4O
|
1
|
1 |
AC50 = 1540 nM
|
|
|
CP0909180
|
SID121284950
Show/Hide
|
C30H31N7O3
|
1
|
1 |
AC50 = 1540 nM
|
|
|
CP0448623
|
MLS003124126
Show/Hide
|
C23H21N3O4
|
1
|
1 |
AC50 = 1550 nM
|
|
|
CP0642600
|
SID855543
Show/Hide
|
C27H30ClNO10
|
1
|
1 |
AC50 = 1550 nM
|
|
|
CP0752972
|
SID26671540
Show/Hide
|
C13H13BrN4O2S
|
1
|
1 |
AC50 = 1550 nM
|
|
|
CP0879950
|
SID131447130
Show/Hide
|
C23H28N2O2
|
1
|
1 |
AC50 = 1550 nM
|
|
|
CP0110873
|
(3E,5E)-3,5-bis(3,4,5-trimethoxybenzylidene)tetrahydropyran-4-one
Show/Hide
|
C25H28O8
|
1
|
1 |
AC50 = 1560 nM
|
|
|
CP0375795
|
2-chloranyl-N-(1-ethanoylindol-3-yl)-N-(2-methoxyphenyl)ethanamide
Show/Hide
|
C19H17ClN2O3
|
1
|
1 |
AC50 = 1560 nM
|
|
|
CP0900341
|
SID131451078
Show/Hide
|
C31H31Cl2N3O6
|
1
|
1 |
AC50 = 1570 nM
|
|
|
CP0751652
|
SID49820710
Show/Hide
|
C24H30N2O6
|
1
|
1 |
AC50 = 1580 nM
|
|
|
CP0907622
|
SID124755201
Show/Hide
|
C34H37N3O6
|
1
|
1 |
AC50 = 1590 nM
|
|
|
CP0881541
|
SID24789354
Show/Hide
|
C16H12N2OS
|
1
|
1 |
AC50 = 1600 nM
|
|
|
CP0886750
|
SID164339367
Show/Hide
|
C22H26N2O4S
|
1
|
1 |
AC50 = 1610 nM
|
|
|
CP0885698
|
SID124753415
Show/Hide
|
C13H10O4
|
1
|
1 |
AC50 = 1630 nM
|
|
|
CP0257597
|
2-[2-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-keto-ethyl]-1,1-diketo-1,2-benzothiazol-3-one
Show/Hide
|
C17H13NO6S
|
1
|
1 |
AC50 = 1640 nM
|
|
|
CP0886118
|
SID26657548
Show/Hide
|
C12H10Cl2N2OS
|
1
|
1 |
AC50 = 1640 nM
|
|
|
CP0327036
|
2-(1H-benzimidazol-2-yl)-1-phthalazinone
Show/Hide
|
C15H10N4O
|
1
|
1 |
AC50 = 1650 nM
|
|
|
CP0857586
|
SID99358994
Show/Hide
|
C32H37N3O4
|
1
|
1 |
AC50 = 1660 nM
|
|
|
CP0733346
|
SID51088957
Show/Hide
|
C14H15ClN4O5S
|
1
|
1 |
AC50 = 1670 nM
|
|
|
CP0923970
|
SID121286576
Show/Hide
|
C17H26ClNO4
|
1
|
1 |
AC50 = 1680 nM
|
|
|
CP0353291
|
4-amino-2-anilino-5-(4-fluorobenzoyl)-N-(4-methoxyphenyl)thiophene-3-carboxamide
Show/Hide
|
C25H20FN3O3S
|
1
|
1 |
AC50 = 1690 nM
|
|
|
CP0445599
|
(1S,4R,6S,6aR,9R,11bS)-methyl 1,6-dihydroxy-4,11b-dimethyl-8-methylene-7-oxotetradecahydro-6a,9-methanocyclohepta[a]naphthalene-4-carboxylate
Show/Hide
|
C21H30O5
|
1
|
1 |
AC50 = 1710 nM
|
|
|
CP0857581
|
SID87335577
Show/Hide
|
C18H21NO
|
1
|
1 |
AC50 = 1710 nM
|
|
|
CP0180639
|
MLS000520174
Show/Hide
|
C22H26N2O2S
|
1
|
1 |
AC50 = 1740 nM
|
|
|
CP0418194
|
4-(2-cyclopropyl-1,3-oxazol-5-yl)-N-(2,6-dimethylphenyl)benzenesulfonamide
Show/Hide
|
C20H20N2O3S
|
1
|
1 |
AC50 = 1740 nM
|
|
|
CP0874952
|
SID92764246
Show/Hide
|
C20H16O8
|
1
|
1 |
AC50 = 1740 nM
|
|
|
CP0912041
|
SID164339408
Show/Hide
|
C25H21FO5
|
1
|
1 |
AC50 = 1740 nM
|
|
|
CP0407992
|
(4R,6S,6aR,9R,11bS)-6-hydroxy-4,11b-dimethyl-8-methylene-7-oxotetradecahydro-6a,9-methanocyclohepta[a]naphthalene-4-carboxylic acid
Show/Hide
|
C20H28O4
|
1
|
1 |
AC50 = 1770 nM
|
|
|
CP0856388
|
SID121284955
Show/Hide
|
C26H25N7O3S
|
1
|
1 |
AC50 = 1780 nM
|
|
|
CP0866432
|
SID92764156
Show/Hide
|
C24H24O9
|
1
|
1 |
AC50 = 1780 nM
|
|
|
CP0852415
|
N'-(2-(trifluoromethyl)quinazolin-4-yl)-4-methoxy-N'-methylbenzohydrazide
Show/Hide
|
C18H15F3N4O2
|
1
|
1 |
AC50 = 1790 nM
|
|
|
CP0008433
|
MLS001205299
Show/Hide
|
C20H20N2O2
|
1
|
1 |
AC50 = 1810 nM
|
|
|
CP0926625
|
SID125306647
Show/Hide
|
C31H37N3O6
|
1
|
1 |
AC50 = 1810 nM
|
|
|
CP0210915
|
7-bromanyl-5-[[4-(2-methoxyphenyl)piperazin-1-yl]methyl]quinolin-8-ol
Show/Hide
|
C21H22BrN3O2
|
1
|
1 |
AC50 = 1820 nM
|
|
|
CP0517958
|
(3Z,5Z)-1-acryloyl-3,5-bis(4-chlorobenzylidene)-4-piperidone
Show/Hide
|
C22H17Cl2NO2
|
1
|
1 |
AC50 = 1820 nM
|
|
|
CP0336974
|
MLS000591280
Show/Hide
|
C16H9F6N5O3S
|
1
|
1 |
AC50 = 1860 nM
|
|
|
CP0392853
|
MLS002701540
Show/Hide
|
C22H30O7
|
1
|
1 |
AC50 = 1860 nM
|
|
|
CP0876247
|
SID49716130
Show/Hide
|
C23H18N2O5S
|
1
|
1 |
AC50 = 1860 nM
|
|
|
CP0886255
|
SID92763383
Show/Hide
|
C8H17N3O4
|
1
|
1 |
AC50 = 1860 nM
|
|
|
CP0908037
|
SID56463667
Show/Hide
|
C16H18ClNO4
|
1
|
1 |
AC50 = 1880 nM
|
|
|
CP0010278
|
MLS001163495
Show/Hide
|
C22H18N2O2
|
1
|
1 |
AC50 = 1890 nM
|
|
|
CP0862095
|
SID87540787
Show/Hide
|
C38H45F6N5O6
|
1
|
1 |
AC50 = 1890 nM
|
|
|
CP0884742
|
SID87543518
Show/Hide
|
C37H46F3N5O6
|
1
|
1 |
AC50 = 1890 nM
|
|
|
CP0906102
|
SID99360807
Show/Hide
|
C18H22N4O8S
|
1
|
1 |
AC50 = 1890 nM
|
|
|
CP0260685
|
2-(dichloromethyl)-4-(ethylthio)-6-phenyl-1,3,5-triazine
Show/Hide
|
C12H11Cl2N3S
|
1
|
1 |
AC50 = 1950 nM
|
|
|
CP0944760
|
SID131443540
Show/Hide
|
C28H30N2O7S
|
1
|
1 |
AC50 = 1950 nM
|
|
|
CP0732728
|
SID49733776
Show/Hide
|
C20H18N4O5S
|
1
|
1 |
AC50 = 1960 nM
|
|
|
CP0880254
|
SID14729694
Show/Hide
|
C21H26ClNO3
|
1
|
1 |
AC50 = 1960 nM
|
|
|
CP0177764
|
2-methyl-4,5-dioxo-3-(phenylmethyl)-1-benzo[e]indolecarboxylic acid ethyl ester
Show/Hide
|
C23H19NO4
|
1
|
1 |
AC50 = 1980 nM
|
|
|
CP0856922
|
SID92763930
Show/Hide
|
C48H74O20
|
1
|
1 |
AC50 = 1980 nM
|
|
|
CP0386929
|
4-(2-cyclopropyl-1,3-oxazol-5-yl)-N-methyl-N-(3-methylphenyl)benzenesulfonamide
Show/Hide
|
C20H20N2O3S
|
1
|
1 |
AC50 = 1990 nM
|
|
|
CP0828846
|
SID89856098
Show/Hide
|
C26H24BrClN6O5S2
|
1
|
1 |
AC50 = 1990 nM
|
|
|
CP0011400
|
MLS001211315
Show/Hide
|
C21H22N2O2
|
1
|
1 |
AC50 = 2030 nM
|
|
|
CP0088502
|
5-(3-methylsulfonylphenyl)-4-(1-methyltetrazol-5-yl)sulfanylthieno[2,3-d]pyrimidine
Show/Hide
|
C15H12N6O2S3
|
1
|
1 |
AC50 = 2030 nM
|
|
|
CP0881140
|
SID49667106
Show/Hide
|
C16H14ClNO3S2
|
1
|
1 |
AC50 = 2030 nM
|
|
|
CP0818772
|
SID49673524
Show/Hide
|
C15H13N3O2
|
1
|
1 |
AC50 = 2040 nM
|
|
|
CP0942893
|
SID131413419
Show/Hide
|
C30H35N3O5S
|
1
|
1 |
AC50 = 2040 nM
|
|
|
CP0712544
|
SID26671321
Show/Hide
|
C16H12N4O2
|
1
|
1 |
AC50 = 2070 nM
|
|
|
CP0900320
|
SID131443480
Show/Hide
|
C30H30F3N3O5
|
1
|
1 |
AC50 = 2070 nM
|
|
|
CP0846298
|
SID99360857
Show/Hide
|
C18H17Cl2NO3
|
1
|
1 |
AC50 = 2080 nM
|
|
|
CP0389536
|
MLS001204199
Show/Hide
|
C18H15ClN2O2
|
1
|
1 |
AC50 = 2090 nM
|
|
|
CP0860634
|
SID92763810
Show/Hide
|
C23H34O4
|
1
|
1 |
AC50 = 2090 nM
|
|
|
CP0797640
|
SID17410182
Show/Hide
|
C24H18N4O5S2
|
1
|
1 |
AC50 = 2100 nM
|
|
|
CP0865350
|
SID17508418
Show/Hide
|
C25H20N2O2
|
1
|
1 |
AC50 = 2100 nM
|
|
|
CP0851528
|
SID131412496
Show/Hide
|
C35H46FN3O8S2
|
1
|
1 |
AC50 = 2110 nM
|
|
|
CP0681219
|
C10322355
Show/Hide
|
C14H15N3O2S
|
1
|
1 |
AC50 = 2140 nM
|
|
|
CP0881645
|
SID121284958
Show/Hide
|
C25H29N7O3S
|
1
|
1 |
AC50 = 2140 nM
|
|
|
CP0855013
|
SID24818981
Show/Hide
|
C20H17NO5
|
1
|
1 |
AC50 = 2150 nM
|
|
|
CP0952397
|
SID131423342
Show/Hide
|
C29H34N4O5S
|
1
|
1 |
AC50 = 2160 nM
|
|
|
CP0295761
|
6-[(7-nitro-2,1,3-benzoxadiazol-4-yl)sulfanyl]-9H-purin-2-amine
Show/Hide
|
C11H6N8O3S
|
1
|
1 |
AC50 = 2170 nM
|
|
|
CP0810768
|
SID51088040
Show/Hide
|
C22H22N4O3
|
1
|
1 |
AC50 = 2180 nM
|
|
|
CP0851386
|
SID49672328
Show/Hide
|
C17H16FNO3
|
1
|
1 |
AC50 = 2180 nM
|
|
|
CP0695737
|
SID24841212
Show/Hide
|
C14H10Cl2N4O3
|
1
|
1 |
AC50 = 2190 nM
|
|
|
CP0852866
|
SID49648722
Show/Hide
|
C27H41NO5
|
1
|
1 |
AC50 = 2190 nM
|
|
|
CP0883098
|
SID92764806
Show/Hide
|
C28H45BrN2O2
|
1
|
1 |
AC50 = 2200 nM
|
|
|
CP0419067
|
CHEBI:38178
Show/Hide
|
C23H32O6
|
1
|
1 |
AC50 = 2220 nM
|
|
|
CP0884554
|
SID49647303
Show/Hide
|
C23H31NO5
|
1
|
1 |
AC50 = 2220 nM
|
|
|
CP0905829
|
SID87540114
Show/Hide
|
C36H45F3N4O7S
|
1
|
1 |
AC50 = 2230 nM
|
|
|
CP0128793
|
(2R,3R,4S,5R)-2-(6-(furan-2-ylmethylamino)-9H-purin-9-yl)-5-(hydroxymethyl)-tetrahydrofuran-3,4-diol
Show/Hide
|
C15H17N5O5
|
1
|
1 |
AC50 = 2250 nM
|
|
|
CP0195117
|
2-(dichloromethyl)-4-(methylthio)-6-phenyl-1,3,5-triazine
Show/Hide
|
C11H9Cl2N3S
|
1
|
1 |
AC50 = 2260 nM
|
|
|
CP0287180
|
4-(3,4-dihydro-1H-isoquinolin-2-ylsulfonyl)-N'-(5,7-dimethyl-1,3-benzothiazol-2-yl)benzohydrazide
Show/Hide
|
C25H24N4O3S2
|
1
|
1 |
AC50 = 2270 nM
|
|
|
CP0947580
|
SID121283020
Show/Hide
|
C16H14N4
|
1
|
1 |
AC50 = 2270 nM
|
|
|
CP0665224
|
SID87337590
Show/Hide
|
C29H24N2O4S
|
1
|
1 |
AC50 = 2280 nM
|
|
|
CP0389423
|
3-[2-(2-methylphenoxy)ethanoylamino]benzoic acid
Show/Hide
|
C16H15NO4
|
1
|
1 |
AC50 = 2300 nM
|
|
|
CP0908721
|
SID87540255
Show/Hide
|
C38H45F6N5O6
|
1
|
1 |
AC50 = 2310 nM
|
|
|
CP0943301
|
SID87541885
Show/Hide
|
C38H45F6N5O6
|
1
|
1 |
AC50 = 2320 nM
|
|
|
CP0001363
|
(E)-N-[(salicyloylamino)thiocarbamoyl]-3-(2-thienyl)acrylamide
Show/Hide
|
C15H13N3O3S2
|
1
|
1 |
AC50 = 2350 nM
|
|
|
CP0311200
|
CS337
Show/Hide
|
C23H34O5
|
1
|
1 |
AC50 = 2350 nM
|
|
|
CP0480964
|
(3Z,5Z)-1-acryloyl-3,5-bis(4-fluorobenzylidene)-4-piperidone
Show/Hide
|
C22H17F2NO2
|
1
|
1 |
AC50 = 2360 nM
|
|
|
CP0814939
|
4-octyl-2,3,5,6,7,8-hexahydro-1H-cyclopenta[b]quinolin-9-imine;hydrobromide
Show/Hide
|
C20H33BrN2
|
1
|
1 |
AC50 = 2360 nM
|
|
|
CP0907445
|
SID49721444
Show/Hide
|
C21H22F3N3O4S
|
1
|
1 |
AC50 = 2360 nM
|
|
|
CP0472654
|
MLS001175788
Show/Hide
|
C18H19NO3
|
1
|
1 |
AC50 = 2380 nM
|
|
|
CP0886265
|
SID87541150
Show/Hide
|
C37H45Cl2F3N4O5
|
1
|
1 |
AC50 = 2390 nM
|
|
|
CP0965808
|
SID131425909
Show/Hide
|
C30H35N3O5S
|
1
|
1 |
AC50 = 2390 nM
|
|
|
CP0862119
|
SID104170388
Show/Hide
|
C36H44ClF3N4O7S
|
1
|
1 |
AC50 = 2410 nM
|
|
|
CP0865836
|
SID92763934
Show/Hide
|
C29H38O4
|
1
|
1 |
AC50 = 2410 nM
|
|
|
CP0871668
|
SID50107430
Show/Hide
|
C15H17N5O5
|
1
|
1 |
AC50 = 2410 nM
|
|
|
CP0942505
|
SID131446404
Show/Hide
|
C26H21N3O3
|
1
|
1 |
AC50 = 2410 nM
|
|
|
CP0413234
|
1-[4-(5-chloranylthiophen-2-yl)-1,3-thiazol-2-yl]-3-(4-nitrophenyl)urea
Show/Hide
|
C14H9ClN4O3S2
|
1
|
1 |
AC50 = 2420 nM
|
|
|
CP0841097
|
SID85146192
Show/Hide
|
C14H9ClN6S2
|
1
|
1 |
AC50 = 2420 nM
|
|
|
CP0862096
|
SID87218847
Show/Hide
|
C30H35Cl2N3O5S
|
1
|
1 |
AC50 = 2420 nM
|
|
|
CP0957466
|
SID87543402
Show/Hide
|
C34H45F6N3O5
|
1
|
1 |
AC50 = 2430 nM
|
|
|
CP0345718
|
MLS000715346
Show/Hide
|
C22H24N2O3
|
1
|
1 |
AC50 = 2440 nM
|
|
|
CP0465834
|
2-(N-(2-chloro-1-oxoethyl)-4-methoxyanilino)-N-(2-phenylethyl)-2-thiophen-2-ylacetamide
Show/Hide
|
C23H23ClN2O3S
|
1
|
1 |
AC50 = 2440 nM
|
|
|
CP0881653
|
SID131414045
Show/Hide
|
C30H32N4O7S
|
1
|
1 |
AC50 = 2440 nM
|
|
|
CP0908006
|
SID125306694
Show/Hide
|
C29H35N3O7
|
1
|
1 |
AC50 = 2440 nM
|
|
|
CP0906902
|
SID87543553
Show/Hide
|
C34H43ClFN3O8S2
|
1
|
1 |
AC50 = 2460 nM
|
|
|
CP0949671
|
SID131447931
Show/Hide
|
C24H27FN2O2
|
1
|
1 |
AC50 = 2470 nM
|
|
|
CP0011641
|
MLS000950003
Show/Hide
|
C18H12ClN3O5
|
1
|
1 |
AC50 = 2480 nM
|
|
|
CP0882466
|
SID121282997
Show/Hide
|
C10H5NO4
|
1
|
1 |
AC50 = 2490 nM
|
|
|
CP0188609
|
4,5-bis(chloranyl)-2-[2-(4-naphthalen-2-ylsulfonylpiperazin-1-yl)-2-oxidanylidene-ethyl]pyridazin-3-one
Show/Hide
|
C20H18Cl2N4O4S
|
1
|
1 |
AC50 = 2510 nM
|
|
|
CP0966332
|
SID131414016
Show/Hide
|
C29H33N3O6S2
|
1
|
1 |
AC50 = 2510 nM
|
|
|
CP0908699
|
SID131413846
Show/Hide
|
C29H33N3O6S2
|
1
|
1 |
AC50 = 2520 nM
|
|
|
CP0158826
|
MLS002701980
Show/Hide
|
C14H12ClNO3
|
1
|
1 |
AC50 = 2540 nM
|
|
|
CP0926618
|
SID131412849
Show/Hide
|
C37H52F3N5O6
|
1
|
1 |
AC50 = 2540 nM
|
|
|
CP0767123
|
SID89650088
Show/Hide
|
C12H8N6S3
|
1
|
1 |
AC50 = 2560 nM
|
|
|
CP0858060
|
SID85146195
Show/Hide
|
C14H9N7O2S2
|
1
|
1 |
AC50 = 2570 nM
|
|
|
CP0897511
|
SID131411631
Show/Hide
|
C37H45F4N5O6
|
1
|
1 |
AC50 = 2580 nM
|
|
|
CP0180992
|
2-(4-aminophenyl)-1,3-benzothiazole-6-carboxylic acid
Show/Hide
|
C14H10N2O2S
|
1
|
1 |
AC50 = 2600 nM
|
|
|
CP0217397
|
2-(7-Methoxy-4-methyl-quinazolin-2-ylamino)-6-phenyl-pyrimidin-4-ol
Show/Hide
|
C20H17N5O2
|
1
|
1 |
AC50 = 2610 nM
|
|
|
CP0125193
|
2-[(3,4-difluorophenyl)sulfonylamino]-N-[4-(4-methoxyphenyl)-1,3-thiazol-2-yl]benzamide
Show/Hide
|
C23H17F2N3O4S2
|
1
|
1 |
AC50 = 2640 nM
|
|
|
CP0651040
|
SID85146185
Show/Hide
|
C14H9FN6S2
|
1
|
1 |
AC50 = 2640 nM
|
|
|
CP0851434
|
SID92764765
Show/Hide
|
C26H25Cl5N2O3
|
1
|
1 |
AC50 = 2650 nM
|
|
|
CP0068873
|
4,5-bis(bromanyl)-2-(4,6-dimethoxypyrimidin-2-yl)pyridazin-3-one
Show/Hide
|
C10H8Br2N4O3
|
1
|
1 |
AC50 = 2660 nM
|
|
|
CP0220342
|
3-(4-Methoxy-phenyl)-2,4-dimethylene-1,5-diphenyl-pentane-1,5-dione
Show/Hide
|
C26H22O3
|
1
|
1 |
AC50 = 2660 nM
|
|
|
CP0345717
|
2-(trichloromethyl)-4-benzo[h][1]benzopyranone
Show/Hide
|
C14H7Cl3O2
|
1
|
1 |
AC50 = 2660 nM
|
|
|
CP0882381
|
SID134215387
Show/Hide
|
C36H46FN3O3
|
1
|
1 |
AC50 = 2660 nM
|
|
|
CP0907391
|
SID131423449
Show/Hide
|
C29H37N3O5S
|
1
|
1 |
AC50 = 2680 nM
|
|
|
CP0040187
|
CHEBI:8241
Show/Hide
|
C17H19NO5
|
1
|
1 |
AC50 = 2690 nM
|
|
|
CP0111416
|
3-[[4-[6-(3-chloroanilino)-4-pyrimidinyl]-2-pyrimidinyl]amino]-1-propanol
Show/Hide
|
C17H17ClN6O
|
1
|
1 |
AC50 = 2700 nM
|
|
|
CP0646258
|
SID47201962
Show/Hide
|
C18H16N6O2
|
1
|
1 |
AC50 = 2700 nM
|
|
|
CP0036293
|
Racemic
Show/Hide
|
C23H24N4O5S
|
1
|
1 |
AC50 = 2710 nM
|
|
|
CP0691324
|
SID24824109
Show/Hide
|
C15H12N4O5S
|
1
|
1 |
AC50 = 2710 nM
|
|
|
CP0910438
|
SID144191552
Show/Hide
|
C32H36N4O7S
|
1
|
1 |
AC50 = 2720 nM
|
|
|
CP0906894
|
SID17415149
Show/Hide
|
C18H17BrN2O3
|
1
|
1 |
AC50 = 2730 nM
|
|
|
CP0053259
|
MLS001029919
Show/Hide
|
C18H18ClNO3
|
1
|
1 |
AC50 = 2740 nM
|
|
|
CP0865945
|
SID89650068
Show/Hide
|
C14H9BrN6S2
|
1
|
1 |
AC50 = 2750 nM
|
|
|
CP0721150
|
SID99494286
Show/Hide
|
C15H13BrN6S
|
1
|
1 |
AC50 = 2780 nM
|
|
|
CP0858473
|
SID49668084
Show/Hide
|
C20H20FNO5
|
1
|
1 |
AC50 = 2780 nM
|
|
|
CP0886264
|
SID131412953
Show/Hide
|
C34H43Cl2N3O8S2
|
1
|
1 |
AC50 = 2780 nM
|
|
|
CP0885257
|
SID103073844
Show/Hide
|
C23H21N3O4
|
1
|
1 |
AC50 = 2790 nM
|
|
|
CP0908693
|
SID104170737
Show/Hide
|
C37H52F3N5O6
|
1
|
1 |
AC50 = 2800 nM
|
|
|
CP0330167
|
2-[(E)-1-(benzenesulfonyl)-2-[4-(trifluoromethyl)phenyl]ethenyl]-1H-benzimidazole
Show/Hide
|
C22H15F3N2O2S
|
1
|
1 |
AC50 = 2820 nM
|
|
|
CP0100749
|
2-(4-chloro-N-(2-chloro-1-oxoethyl)anilino)-N-(2-phenylethyl)-2-thiophen-2-ylacetamide
Show/Hide
|
C22H20Cl2N2O2S
|
1
|
1 |
AC50 = 2840 nM
|
|
|
CP0860399
|
SID131425908
Show/Hide
|
C30H35N3O5S
|
1
|
1 |
AC50 = 2840 nM
|
|
|
CP0882469
|
SID56320908
Show/Hide
|
C27H30ClNO10
|
1
|
1 |
AC50 = 2840 nM
|
|
|
CP0418024
|
2-[4,5-bis(chloranyl)-6-oxidanylidene-pyridazin-1-yl]-N-(cyclohexylcarbamoyl)ethanamide
Show/Hide
|
C13H16Cl2N4O3
|
1
|
1 |
AC50 = 2850 nM
|
|
|
CP0885255
|
SID87539824
Show/Hide
|
C38H47F3N4O6
|
1
|
1 |
AC50 = 2850 nM
|
|
|
CP0826479
|
SID49735130
Show/Hide
|
C20H27N9O3
|
1
|
1 |
AC50 = 2860 nM
|
|
|
CP0908033
|
SID87542529
Show/Hide
|
C36H44ClF3N4O7S
|
1
|
1 |
AC50 = 2860 nM
|
|
|
CP0852416
|
SID131410419
Show/Hide
|
C36H44ClF3N4O7S
|
1
|
1 |
AC50 = 2870 nM
|
|
|
CP0882032
|
SID99494427
Show/Hide
|
C25H24N4O5
|
1
|
1 |
AC50 = 2880 nM
|
|
|
CP0857095
|
SID47202224
Show/Hide
|
C22H25N3O5
|
1
|
1 |
AC50 = 2890 nM
|
|
|
CP0881649
|
SID131448107
Show/Hide
|
C24H25N3O2
|
1
|
1 |
AC50 = 2890 nM
|
|
|
CP0888836
|
SID49669494
Show/Hide
|
C24H32N2O4
|
1
|
1 |
AC50 = 2900 nM
|
|
|
CP0039514
|
3-Amino-4,6-dimethyl-thieno[2,3-b]pyridine-2-carboxylic acid (5-methyl-thiazol-2-yl)-amide
Show/Hide
|
C14H14N4OS2
|
1
|
1 |
AC50 = 2920 nM
|
|
|
CP0230319
|
(1Z)-1-(1,3-thiazol-2-ylhydrazinylidene)naphthalen-2-one
Show/Hide
|
C13H9N3OS
|
1
|
1 |
AC50 = 2920 nM
|
|
|
CP0447724
|
2-[2-(1,3-benzodioxol-5-yl)ethenyl]quinoxaline
Show/Hide
|
C17H12N2O2
|
1
|
1 |
AC50 = 2920 nM
|
|
|
CP0078802
|
2-[2-(2,4-dichlorophenyl)-2-keto-ethyl]-1,1-diketo-1,2-benzothiazol-3-one
Show/Hide
|
C15H9Cl2NO4S
|
1
|
1 |
AC50 = 2930 nM
|
|
|
CP0304221
|
(Z)-4,4-Dimethyl-1-(3-nitro-phenyl)-2-[1,2,4]triazol-1-yl-pent-1-en-3-one
Show/Hide
|
C15H16N4O3
|
1
|
1 |
AC50 = 2930 nM
|
|
|
CP0905961
|
SID103162960
Show/Hide
|
C23H21N3O4
|
1
|
1 |
AC50 = 2930 nM
|
|
|
CP0881628
|
SID121286225
Show/Hide
|
C15H12N4
|
1
|
1 |
AC50 = 2950 nM
|
|
|
CP0700391
|
SID85146202
Show/Hide
|
C12H9N7S2
|
1
|
1 |
AC50 = 2960 nM
|
|
|
CP0394351
|
1-(3-Chloro-phenyl)-3-(5-pyridin-4-yl-[1,3,4]thiadiazol-2-yl)-urea
Show/Hide
|
C14H10ClN5OS
|
1
|
1 |
AC50 = 2970 nM
|
|
|
CP0874834
|
SID144194108
Show/Hide
|
C20H21N3O
|
1
|
1 |
AC50 = 2980 nM
|
|
|
CP0329072
|
4-(3,4-dihydro-1H-isoquinolin-2-ylsulfonyl)-N'-(6-methyl-1,3-benzothiazol-2-yl)benzohydrazide
Show/Hide
|
C24H22N4O3S2
|
1
|
1 |
AC50 = 3010 nM
|
|
|
CP0885905
|
SID56322302
Show/Hide
|
C13H14Cl2N4O2
|
1
|
1 |
AC50 = 3010 nM
|
|
|
CP0411509
|
5-(diethylsulfamoyl)-N-[2-(2,6-difluoroanilino)-2-keto-ethyl]-N-ethyl-2-piperidino-benzamide
Show/Hide
|
C26H34F2N4O4S
|
1
|
1 |
AC50 = 3020 nM
|
|
|
CP0864560
|
SID131413949
Show/Hide
|
C30H32N4O7S
|
1
|
1 |
AC50 = 3020 nM
|
|
|
CP0918067
|
SID87539809
Show/Hide
|
C37H46F3N5O6
|
1
|
1 |
AC50 = 3020 nM
|
|
|
CP0395818
|
MLS003107615
Show/Hide
|
C35H47N5O8S
|
1
|
1 |
AC50 = 3030 nM
|
|
|
CP0712403
|
SID24801057
Show/Hide
|
C15H12N2O4
|
1
|
1 |
AC50 = 3040 nM
|
|
|
CP0732997
|
SID49676635
Show/Hide
|
C17H17F3N4O
|
1
|
1 |
AC50 = 3040 nM
|
|
|
CP0856556
|
SID92763919
Show/Hide
|
C18H15N3O2
|
1
|
1 |
AC50 = 3040 nM
|
|
|
CP0446895
|
4-[(6,7,10-trimethylbenzo[b][1,4]benzothiazepine-3-carbonyl)amino]piperidine-1-carboxylic acid ethyl ester
Show/Hide
|
C25H29N3O3S
|
1
|
1 |
AC50 = 3050 nM
|
|
|
CP0885766
|
SID144194092
Show/Hide
|
C22H24N2O2
|
1
|
1 |
AC50 = 3060 nM
|
|
|
CP0909791
|
SID85808922
Show/Hide
|
C32H37F3N4O6S
|
1
|
1 |
AC50 = 3060 nM
|
|
|
CP0966628
|
SID144190999
Show/Hide
|
C26H24F3N3O
|
1
|
1 |
AC50 = 3060 nM
|
|
|
CP0942495
|
SID144198556
Show/Hide
|
C37H46F3N5O6
|
1
|
1 |
AC50 = 3070 nM
|
|
|
CP0912881
|
SID87542413
Show/Hide
|
C37H46F3N3O5
|
1
|
1 |
AC50 = 3090 nM
|
|
|
CP0950344
|
SID131446920
Show/Hide
|
C26H25FN2O2
|
1
|
1 |
AC50 = 3090 nM
|
|
|
CP0841100
|
SID89650081
Show/Hide
|
C16H12N6OS2
|
1
|
1 |
AC50 = 3100 nM
|
|
|
CP0663179
|
SID85146200
Show/Hide
|
C16H10N6OS2
|
1
|
1 |
AC50 = 3120 nM
|
|
|
CP0942503
|
SID87218853
Show/Hide
|
C30H34Cl2FN3O5S
|
1
|
1 |
AC50 = 3120 nM
|
|
|
CP0856877
|
SID131423444
Show/Hide
|
C29H37N3O5S
|
1
|
1 |
AC50 = 3130 nM
|
|
|
CP0881601
|
SID87541743
Show/Hide
|
C37H47F3N4O7S
|
1
|
1 |
AC50 = 3140 nM
|
|
|
CP0860341
|
SID131413851
Show/Hide
|
C29H33N3O6S2
|
1
|
1 |
AC50 = 3150 nM
|
|
|
CP0862639
|
SID92763408
Show/Hide
|
C29H37NO5
|
1
|
1 |
AC50 = 3150 nM
|
|
|
CP0907183
|
SID144196939
Show/Hide
|
C26H26N2O3
|
1
|
1 |
AC50 = 3150 nM
|
|
|
CP0729919
|
SID164339401
Show/Hide
|
C18H20N2O4S2
|
1
|
1 |
AC50 = 3160 nM
|
|
|
CP0744196
|
SID104219503
Show/Hide
|
C15H14N2O3S
|
1
|
1 |
AC50 = 3160 nM
|
|
|
CP0856709
|
SID87539608
Show/Hide
|
C34H43F3N4O7S2
|
1
|
1 |
AC50 = 3170 nM
|
|
|
CP0378386
|
2-Chloro-N-(5-chloro-3-methyl-1-phenyl-1H-pyrazol-4-ylmethyl)-N-(4-chloro-phenyl)-acetamide
Show/Hide
|
C19H16Cl3N3O
|
1
|
1 |
AC50 = 3190 nM
|
|
|
CP0881650
|
SID87539708
Show/Hide
|
C35H46ClN3O8S2
|
1
|
1 |
AC50 = 3200 nM
|
|
|
CP0930556
|
SID131412039
Show/Hide
|
C32H43ClF3N3O7S
|
1
|
1 |
AC50 = 3200 nM
|
|
|
CP0966333
|
SID131444678
Show/Hide
|
C28H30N2O6S
|
1
|
1 |
AC50 = 3200 nM
|
|
|
CP0221748
|
(4-methoxyphenyl)-(2-morpholin-4-yl-5-nitro-phenyl)methanone
Show/Hide
|
C18H18N2O5
|
1
|
1 |
AC50 = 3210 nM
|
|
|
CP0004490
|
MLS001204081
Show/Hide
|
C21H22N2O2
|
1
|
1 |
AC50 = 3240 nM
|
|
|
CP0884748
|
SID131412105
Show/Hide
|
C36H45F3N4O7S
|
1
|
1 |
AC50 = 3240 nM
|
|
|
CP0345249
|
3-acenaphthen-5-yl-N-[(4-chloro-3-nitro-benzylidene)amino]-1H-pyrazole-5-carboxamide
Show/Hide
|
C23H16ClN5O3
|
1
|
1 |
AC50 = 3250 nM
|
|
|
CP0700688
|
SID24786849
Show/Hide
|
C19H21ClN4O5
|
1
|
1 |
AC50 = 3250 nM
|
|
|
CP0882380
|
SID87542791
Show/Hide
|
C36H44ClF3N4O7S
|
1
|
1 |
AC50 = 3250 nM
|
|
|
CP0908897
|
SID131412955
Show/Hide
|
C34H43Cl2N3O8S2
|
1
|
1 |
AC50 = 3270 nM
|
|
|
CP0966604
|
SID51086862
Show/Hide
|
C21H25ClN4O4S
|
1
|
1 |
AC50 = 3270 nM
|
|
|
CP0856751
|
SID131409965
Show/Hide
|
C30H44ClN3O6S
|
1
|
1 |
AC50 = 3280 nM
|
|
|
CP0048396
|
HEXACHLOROPHENE
Show/Hide
|
C13H6Cl6O2
|
1
|
1 |
AC50 = 3300 nM
|
|
|
CP0907194
|
SID131413959
Show/Hide
|
C29H33N3O6S2
|
1
|
1 |
AC50 = 3300 nM
|
|
|
CP0188290
|
1,2-Dione-Based Compound, 17
Show/Hide
|
C12H6N2O2
|
1
|
1 |
AC50 = 3320 nM
|
|
|
CP0637400
|
2'-(2-((pyridin-2-yl)methylene)hydrazinyl)-1',3'-benzothiazole
Show/Hide
|
C13H10N4S
|
1
|
1 |
AC50 = 3320 nM
|
|
|
CP0865829
|
SID92764016
Show/Hide
|
C15H12F4N4
|
1
|
1 |
AC50 = 3320 nM
|
|
|
CP0891493
|
SID87542390
Show/Hide
|
C35H46FN3O8S2
|
1
|
1 |
AC50 = 3320 nM
|
|
|
CP0891767
|
SID57266362
Show/Hide
|
C16H12BrN3O3S2
|
1
|
1 |
AC50 = 3320 nM
|
|
|
CP0886268
|
SID87540967
Show/Hide
|
C38H47F3N4O7
|
1
|
1 |
AC50 = 3340 nM
|
|
|
CP0943342
|
SID121282541
Show/Hide
|
C28H29ClN2O7S
|
1
|
1 |
AC50 = 3360 nM
|
|
|
CP0259162
|
2,2,2-trifluoro-N-[3-[6-(4-methyl-1-piperidinyl)-3-pyridazinyl]phenyl]acetamide
Show/Hide
|
C18H19F3N4O
|
1
|
1 |
AC50 = 3370 nM
|
|
|
CP0856553
|
SID17504722
Show/Hide
|
C20H30O5
|
1
|
1 |
AC50 = 3370 nM
|
|
|
CP0952674
|
SID87543033
Show/Hide
|
C37H46F4N4O5
|
1
|
1 |
AC50 = 3370 nM
|
|
|
CP0885131
|
SID17432820
Show/Hide
|
C19H20N2O3
|
1
|
1 |
AC50 = 3390 nM
|
|
|
CP0894294
|
SID92763950
Show/Hide
|
C23H32O6
|
1
|
1 |
AC50 = 3390 nM
|
|
|
CP0907619
|
SID131446804
Show/Hide
|
C27H28N2O3
|
1
|
1 |
AC50 = 3390 nM
|
|
|
CP0086865
|
(4E)-4-[(5-chloro-2,4-dimethoxyphenyl)imino]-2-hydroxynaphthalen-1(4H)-one
Show/Hide
|
C18H14ClNO4
|
1
|
1 |
AC50 = 3400 nM
|
|
|
CP0900574
|
SID131414261
Show/Hide
|
C29H32FN3O4S
|
1
|
1 |
AC50 = 3400 nM
|
|
|
CP0942496
|
SID131447309
Show/Hide
|
C27H28N2O3
|
1
|
1 |
AC50 = 3400 nM
|
|
|
CP0669540
|
SID89650065
Show/Hide
|
C15H9F3N6S2
|
1
|
1 |
AC50 = 3410 nM
|
|
|
CP0889305
|
SID92764343
Show/Hide
|
C28H31N3O14
|
1
|
1 |
AC50 = 3410 nM
|
|
|
CP0912292
|
SID87539857
Show/Hide
|
C34H43ClFN3O8S2
|
1
|
1 |
AC50 = 3410 nM
|
|
|
CP0935293
|
SID131413140
Show/Hide
|
C38H48F3N5O7
|
1
|
1 |
AC50 = 3410 nM
|
|
|
CP0942605
|
SID131413968
Show/Hide
|
C32H38N2O5S
|
1
|
1 |
AC50 = 3420 nM
|
|
|
CP0736989
|
SID22405802
Show/Hide
|
C20H25N3O6
|
1
|
1 |
AC50 = 3430 nM
|
|
|
CP0857040
|
SID87541362
Show/Hide
|
C37H48F3N3O7S
|
1
|
1 |
AC50 = 3430 nM
|
|
|
CP0851527
|
MMV1509658
Show/Hide
|
C13H7F3N6
|
1
|
1 |
AC50 = 3440 nM
|
|
|
CP0889187
|
SID131444802
Show/Hide
|
C33H31FN2O6S
|
1
|
1 |
AC50 = 3440 nM
|
|
|
CP0897520
|
SID87542798
Show/Hide
|
C36H45F3N4O7S
|
1
|
1 |
AC50 = 3440 nM
|
|
|
CP0926615
|
SID87543014
Show/Hide
|
C36H44ClF3N4O7S
|
1
|
1 |
AC50 = 3440 nM
|
|
|
CP0370678
|
5-chloranyl-2-ethylsulfonyl-N-[4-(4-methylpiperidin-1-yl)sulfonylphenyl]pyrimidine-4-carboxamide
Show/Hide
|
C19H23ClN4O5S2
|
1
|
1 |
AC50 = 3450 nM
|
|
|
CP0404964
|
2-chloranyl-N-(3-methylphenyl)-N-(phenylmethyl)ethanamide
Show/Hide
|
C16H16ClNO
|
1
|
1 |
AC50 = 3460 nM
|
|
|
CP0908898
|
SID136348308
Show/Hide
|
C15H14N2
|
1
|
1 |
AC50 = 3460 nM
|
|
|
CP0930585
|
SID131447882
Show/Hide
|
C22H33N3O2
|
1
|
1 |
AC50 = 3470 nM
|
|
|
CP0879940
|
SID131410837
Show/Hide
|
C34H43F3N4O7S2
|
1
|
1 |
AC50 = 3480 nM
|
|
|
CP0274206
|
triazolothiadiazine, 6
Show/Hide
|
C24H26N4O4S
|
1
|
1 |
AC50 = 3490 nM
|
|
|
CP0872578
|
SID57267384
Show/Hide
|
C13H12N2O3S
|
1
|
1 |
AC50 = 3490 nM
|
|
|
CP0886293
|
SID99456595
Show/Hide
|
C24H22FN3O5
|
1
|
1 |
AC50 = 3490 nM
|
|
|
CP0753507
|
SID22401243
Show/Hide
|
C24H17BrN4O
|
1
|
1 |
AC50 = 3500 nM
|
|
|
CP0881113
|
SID131412850
Show/Hide
|
C37H52F3N5O6
|
1
|
1 |
AC50 = 3500 nM
|
|
|
CP0077816
|
LASALOCID A SODIUM
Show/Hide
|
C34H53NaO8
|
1
|
1 |
AC50 = 3520 nM
|
|
|
CP0873861
|
SID26726873
Show/Hide
|
C16H13NO5S
|
1
|
1 |
AC50 = 3530 nM
|
|
|
CP0907569
|
SID131411339
Show/Hide
|
C37H45F3N4O6
|
1
|
1 |
AC50 = 3530 nM
|
|
|
CP0860347
|
SID51088780
Show/Hide
|
C16H13FN2O3S2
|
1
|
1 |
AC50 = 3550 nM
|
|
|
CP0915685
|
SID103059968
Show/Hide
|
C18H20N2O4S
|
1
|
1 |
AC50 = 3550 nM
|
|
|
CP0850665
|
SID89650069
Show/Hide
|
C14H9BrN6S2
|
1
|
1 |
AC50 = 3560 nM
|
|
|
CP0258431
|
4-methyl-N-(3-quinolinyl)benzamide
Show/Hide
|
C17H14N2O
|
1
|
1 |
AC50 = 3570 nM
|
|
|
CP0366335
|
2-(4,5-dichloro-6-keto-pyridazin-1-yl)-N-[2-keto-2-(p-toluidino)ethyl]-N-methyl-acetamide
Show/Hide
|
C16H16Cl2N4O3
|
1
|
1 |
AC50 = 3570 nM
|
|
|
CP0449295
|
MLS002920361
Show/Hide
|
C19H14ClNO4
|
1
|
1 |
AC50 = 3590 nM
|
|
|
CP0907570
|
SID134962105
Show/Hide
|
C30H35N3O5S2
|
1
|
1 |
AC50 = 3600 nM
|
|
|
CP0930593
|
SID85793938
Show/Hide
|
C39H47N5O6
|
1
|
1 |
AC50 = 3610 nM
|
|
|
CP0404293
|
3,5-bis(3-pyridinylmethyl)-1,3,5-thiadiazinane-2-thione
Show/Hide
|
C15H16N4S2
|
1
|
1 |
AC50 = 3620 nM
|
|
|
CP0489813
|
(1S,4R,4aS,6S,6aR,9R,11aS,11bS)-4-(methoxycarbonyl)-4,11b-dimethyl-8-methylene-7-oxotetradecahydro-6a,9-methanocyclohepta[a]naphthalene-1,6-diyl diacetate
Show/Hide
|
C25H34O7
|
1
|
1 |
AC50 = 3620 nM
|
|
|
CP0874985
|
SID87540471
Show/Hide
|
C37H45F4N5O6
|
1
|
1 |
AC50 = 3620 nM
|
|
|
CP0856879
|
SID131412872
Show/Hide
|
C39H48N4O7S
|
1
|
1 |
AC50 = 3660 nM
|
|
|
CP0189438
|
3,4,5,6-tetramethylphenanthrene-9,10-dione
Show/Hide
|
C18H16O2
|
1
|
1 |
AC50 = 3670 nM
|
|
|
CP0965721
|
SID131413896
Show/Hide
|
C30H32N4O7S
|
1
|
1 |
AC50 = 3680 nM
|
|
|
CP0662708
|
N-(1,3-benzothiazol-2-yl)-2-methoxybenzamide
Show/Hide
|
C15H12N2O2S
|
1
|
1 |
AC50 = 3690 nM
|
|
|
CP0935290
|
SID144191555
Show/Hide
|
C33H36F3N3O5S
|
1
|
1 |
AC50 = 3690 nM
|
|
|
CP0966823
|
SID87540991
Show/Hide
|
C37H45F3N4O6
|
1
|
1 |
AC50 = 3720 nM
|
|
|
CP0875941
|
SID26660762
Show/Hide
|
C17H31BrN2
|
1
|
1 |
AC50 = 3740 nM
|
|
|
CP0007525
|
MLS001146578
Show/Hide
|
C17H13N3O7
|
1
|
1 |
AC50 = 3750 nM
|
|
|
CP0868347
|
SID144190662
Show/Hide
|
C25H23N3O2S
|
1
|
1 |
AC50 = 3750 nM
|
|
|
CP0445810
|
(2-morpholin-4-yl-5-nitro-phenyl)-(4-phenylpiperazin-1-yl)methanone
Show/Hide
|
C21H24N4O4
|
1
|
1 |
AC50 = 3760 nM
|
|
|
CP0900395
|
SID87543601
Show/Hide
|
C37H45F3N4O6
|
1
|
1 |
AC50 = 3760 nM
|
|
|
CP0053500
|
(7R,9R)-7-[(2R,4S,5S,6S)-4-azanyl-6-methyl-5-oxidanyl-oxan-2-yl]oxy-9-ethanoyl-6,9,11-tris(oxidanyl)-8,10-dihydro-7H-tetracene-5,12-dione
Show/Hide
|
C26H27NO9
|
1
|
1 |
AC50 = 3770 nM
|
|
|
CP0941652
|
SID121284957
Show/Hide
|
C32H29N7O3
|
1
|
1 |
AC50 = 3780 nM
|
|
|
CP0431168
|
7-(3,4-dihydroxy-5-methylol-tetrahydrofuran-2-yl)-4-(3-methylbut-2-enylamino)pyrrolo[2,3-d]pyrimidine-5-carbonitrile
Show/Hide
|
C17H21N5O4
|
1
|
1 |
AC50 = 3790 nM
|
|
|
CP0456178
|
3-(2,3-dihydro-1H-inden-5-yloxymethyl)benzoic acid
Show/Hide
|
C17H16O3
|
1
|
1 |
AC50 = 3790 nM
|
|
|
CP0862106
|
SID99359887
Show/Hide
|
C23H18ClN5O2
|
1
|
1 |
AC50 = 3790 nM
|
|
|
CP0442083
|
MLS002246639
Show/Hide
|
C10H7N3O5S
|
1
|
1 |
AC50 = 3800 nM
|
|
|
CP0669456
|
SID164339394
Show/Hide
|
C18H16BrNO3
|
1
|
1 |
AC50 = 3800 nM
|
|
|
CP0869059
|
SID121284987
Show/Hide
|
C23H27N7O
|
1
|
1 |
AC50 = 3800 nM
|
|
|
CP0047178
|
4-[2-[(5E)-5-(4-chlorobenzylidene)-4-keto-2-thioxo-thiazolidin-3-yl]ethyl]benzenesulfonamide
Show/Hide
|
C18H15ClN2O3S3
|
1
|
1 |
AC50 = 3810 nM
|
|
|
CP0194694
|
3-methyl-8-nitro-7-(phenylmethyl)purine-2,6-dione
Show/Hide
|
C13H11N5O4
|
1
|
1 |
AC50 = 3810 nM
|
|
|
CP0779348
|
SID24812872
Show/Hide
|
C11H9BrN4
|
1
|
1 |
AC50 = 3840 nM
|
|
|
CP0857030
|
SID24791955
Show/Hide
|
C16H16N2O4
|
1
|
1 |
AC50 = 3850 nM
|
|
|
CP0865126
|
SID87541116
Show/Hide
|
C32H42ClN3O8S3
|
1
|
1 |
AC50 = 3860 nM
|
|
|
CP0915297
|
SID131442360
Show/Hide
|
C29H29FN2O6S
|
1
|
1 |
AC50 = 3860 nM
|
|
|
CP0205884
|
5-(4-dibenzothiophenyl)-4-[(1-methyl-5-tetrazolyl)thio]thieno[2,3-d]pyrimidine
Show/Hide
|
C20H12N6S3
|
1
|
1 |
AC50 = 3890 nM
|
|
|
CP0934881
|
SID85805524
Show/Hide
|
C37H53F3N4O5
|
1
|
1 |
AC50 = 3900 nM
|
|
|
CP0396874
|
MLS003107618
Show/Hide
|
C39H43N5O12S
|
1
|
1 |
AC50 = 3910 nM
|
|
|
CP0064465
|
5-nitro-N-[4-[4-(phenylcarbonyl)piperazin-1-yl]phenyl]furan-2-carboxamide
Show/Hide
|
C22H20N4O5
|
1
|
1 |
AC50 = 3920 nM
|
|
|
CP0307648
|
(Z)-2-(1,3-benzothiazol-2-yl)-N-(4-chlorophenyl)-3-(3-hydroxyphenyl)-2-propenamide
Show/Hide
|
C22H15ClN2O2S
|
1
|
1 |
AC50 = 3920 nM
|
|
|
CP0862126
|
SID131461588
Show/Hide
|
C25H25FN2O4S
|
1
|
1 |
AC50 = 3920 nM
|
|
|
CP0719734
|
SID49667402
Show/Hide
|
C19H17ClN2O2
|
1
|
1 |
AC50 = 3930 nM
|
|
|
CP0930683
|
SID87541275
Show/Hide
|
C37H48F3N3O6S
|
1
|
1 |
AC50 = 3930 nM
|
|
|
CP0428211
|
MLS002248660
Show/Hide
|
C16H17N3O6S2
|
1
|
1 |
AC50 = 3940 nM
|
|
|
CP0753872
|
SID24841193
Show/Hide
|
C9H7BrClN3O2
|
1
|
1 |
AC50 = 3950 nM
|
|
|
CP0887204
|
N-benzyl-2-chloro-N-phenylacetamide
Show/Hide
|
C15H14ClNO
|
1
|
1 |
AC50 = 3950 nM
|
|
|
CP0905831
|
SID87540768
Show/Hide
|
C35H46FN3O9S2
|
1
|
1 |
AC50 = 3960 nM
|
|
|
CP0248880
|
2-chloranyl-N-cyclohexyl-N-phenyl-ethanamide
Show/Hide
|
C14H18ClNO
|
1
|
1 |
AC50 = 3980 nM
|
|
|
CP0959683
|
SID104170460
Show/Hide
|
C38H48F3N3O5
|
1
|
1 |
AC50 = 3980 nM
|
|
|
CP0940506
|
SID104170750
Show/Hide
|
C35H46ClN3O9S2
|
1
|
1 |
AC50 = 3990 nM
|
|
|
CP0950773
|
SID99357416
Show/Hide
|
C28H37N5O5S
|
1
|
1 |
AC50 = 3990 nM
|
|
|
CP0821827
|
SID26725217
Show/Hide
|
C20H24O6
|
1
|
1 |
AC50 = 4030 nM
|
|
|
CP0883670
|
SID131414023
Show/Hide
|
C29H33N3O6S2
|
1
|
1 |
AC50 = 4030 nM
|
|
|
CP0342064
|
5-nitro-N-[3-(2-thenoylamino)phenyl]-2-furamide
Show/Hide
|
C16H11N3O5S
|
1
|
1 |
AC50 = 4040 nM
|
|
|
CP0436833
|
3-[[(E)-1-oxo-3-phenylprop-2-enyl]amino]benzoic acid
Show/Hide
|
C16H13NO3
|
1
|
1 |
AC50 = 4060 nM
|
|
|
CP0407187
|
(1S,4R,4aS,6S,6aR,9R,11aS,11bS)-1-acetoxy-6-hydroxy-4,11b-dimethyl-8-methylene-7-oxotetradecahydro-6a,9-methanocyclohepta[a]naphthalene-4-carboxylic acid
Show/Hide
|
C22H30O6
|
1
|
1 |
AC50 = 4070 nM
|
|
|
CP0498572
|
MLS002170809
Show/Hide
|
C13H9Cl2N3O4
|
1
|
1 |
AC50 = 4070 nM
|
|
|
CP0856880
|
SID85805571
Show/Hide
|
C36H51FN4O6
|
1
|
1 |
AC50 = 4070 nM
|
|
|
CP0862124
|
SID131413134
Show/Hide
|
C35H46ClN3O8S2
|
1
|
1 |
AC50 = 4090 nM
|
|
|
CP0889239
|
SID131460966
Show/Hide
|
C24H22F2N2O3S
|
1
|
1 |
AC50 = 4090 nM
|
|
|
CP0195353
|
2-[(E)-1-(benzenesulfonyl)-2-(3-methylphenyl)ethenyl]-1H-benzimidazole
Show/Hide
|
C22H18N2O2S
|
1
|
1 |
AC50 = 4100 nM
|
|
|
CP0944038
|
SID131442203
Show/Hide
|
C31H30F3N3O5
|
1
|
1 |
AC50 = 4100 nM
|
|
|
CP0202116
|
2-[[2-(2,4-diketo-6-methyl-1,3-diazaspiro[4.5]decan-3-yl)acetyl]amino]-4-(4-fluorophenyl)thiophene-3-carboxylic acid ethyl ester
Show/Hide
|
C24H26FN3O5S
|
1
|
1 |
AC50 = 4110 nM
|
|
|
CP0912951
|
SID131411633
Show/Hide
|
C37H45F4N5O6
|
1
|
1 |
AC50 = 4110 nM
|
|
|
CP0707580
|
SID24808858
Show/Hide
|
C18H19ClN4O5
|
1
|
1 |
AC50 = 4120 nM
|
|
|
CP0900535
|
SID104170611
Show/Hide
|
C37H46F4N4O5
|
1
|
1 |
AC50 = 4130 nM
|
|
|
CP0386936
|
3-[(4-methoxyphenoxy)methyl]-N-(5-methyl-1,2-oxazol-3-yl)benzamide
Show/Hide
|
C19H18N2O4
|
1
|
1 |
AC50 = 4140 nM
|
|
|
CP0043874
|
5-(4-fluorophenyl)-4-(1-methyltetrazol-5-yl)sulfanylthieno[2,3-d]pyrimidine
Show/Hide
|
C14H9FN6S2
|
1
|
1 |
AC50 = 4150 nM
|
|
|
CP0377810
|
(5E)-5-[[2-(trifluoromethyl)phenyl]hydrazinylidene]-8-quinolinone
Show/Hide
|
C16H10F3N3O
|
1
|
1 |
AC50 = 4150 nM
|
|
|
CP0899486
|
SID131412525
Show/Hide
|
C40H50N4O7S
|
1
|
1 |
AC50 = 4150 nM
|
|
|
CP0908038
|
SID87542764
Show/Hide
|
C37H45Cl2F3N4O5
|
1
|
1 |
AC50 = 4170 nM
|
|
|
CP0912656
|
SID131412381
Show/Hide
|
C36H46F3N3O6S
|
1
|
1 |
AC50 = 4170 nM
|
|
|
CP0375868
|
MLS003107612
Show/Hide
|
C33H47N5O8S
|
1
|
1 |
AC50 = 4180 nM
|
|
|
CP0926404
|
SID131412705
Show/Hide
|
C37H48F3N3O6S
|
1
|
1 |
AC50 = 4180 nM
|
|
|
CP0944779
|
SID131412616
Show/Hide
|
C32H42ClN3O8S3
|
1
|
1 |
AC50 = 4180 nM
|
|
|
CP0884590
|
SID131410333
Show/Hide
|
C37H45Cl2F3N4O5
|
1
|
1 |
AC50 = 4200 nM
|
|
|
CP0240471
|
1-ethyl-6-methyl-3-[(E)-2-phenylethenyl]pyrimido[5,4-e][1,2,4]triazine-5,7-dione
Show/Hide
|
C16H15N5O2
|
1
|
1 |
AC50 = 4210 nM
|
|
|
CP0408003
|
MLS000056567
Show/Hide
|
C19H19N7O2S2
|
1
|
1 |
AC50 = 4210 nM
|
|
|
CP0946014
|
SID131411671
Show/Hide
|
C36H46F3N5O5
|
1
|
1 |
AC50 = 4210 nM
|
|
|
CP0408002
|
MLS003107617
Show/Hide
|
C29H27N5O8S3
|
1
|
1 |
AC50 = 4220 nM
|
|
|
CP0918114
|
SID131412603
Show/Hide
|
C33H45N3O8S3
|
1
|
1 |
AC50 = 4230 nM
|
|
|
CP0900323
|
SID87218862
Show/Hide
|
C30H34Cl3N3O5S
|
1
|
1 |
AC50 = 4260 nM
|
|
|
CP0944043
|
SID144190512
Show/Hide
|
C21H21FN4O2S
|
1
|
1 |
AC50 = 4260 nM
|
|
|
CP0856869
|
SID87349674
Show/Hide
|
C28H41ClN2O4
|
1
|
1 |
AC50 = 4270 nM
|
|
|
CP0889186
|
SID87542263
Show/Hide
|
C36H46Cl2N4O5
|
1
|
1 |
AC50 = 4290 nM
|
|
|
CP0851408
|
SID85198584
Show/Hide
|
C18H20Cl2N4O4S
|
1
|
1 |
AC50 = 4300 nM
|
|
|
CP0908891
|
SID87543881
Show/Hide
|
C34H43ClFN3O8S2
|
1
|
1 |
AC50 = 4330 nM
|
|
|
CP0879865
|
SID99360397
Show/Hide
|
C16H22O2
|
1
|
1 |
AC50 = 4340 nM
|
|
|
CP0882420
|
SID131412951
Show/Hide
|
C34H43Cl2N3O8S2
|
1
|
1 |
AC50 = 4340 nM
|
|
|
CP0908027
|
SID131410687
Show/Hide
|
C38H47F3N4O6
|
1
|
1 |
AC50 = 4340 nM
|
|
|
CP0760503
|
SID49822477
Show/Hide
|
C22H21N3O2S2
|
1
|
1 |
AC50 = 4370 nM
|
|
|
CP0831902
|
SID24837680
Show/Hide
|
C26H32ClF3N2
|
1
|
1 |
AC50 = 4370 nM
|
|
|
CP0862100
|
SID144194774
Show/Hide
|
C26H26N2O3
|
1
|
1 |
AC50 = 4380 nM
|
|
|
CP0932671
|
SID131447111
Show/Hide
|
C26H19F2N3O2
|
1
|
1 |
AC50 = 4380 nM
|
|
|
CP0337238
|
MLS001163735
Show/Hide
|
C15H18N2O4
|
1
|
1 |
AC50 = 4390 nM
|
|
|
CP0908904
|
SID87543333
Show/Hide
|
C36H45ClF3N3O6S
|
1
|
1 |
AC50 = 4390 nM
|
|
|
CP0907921
|
SID87540665
Show/Hide
|
C35H46ClN3O8S2
|
1
|
1 |
AC50 = 4400 nM
|
|
|
CP0781464
|
SID26732655
Show/Hide
|
C32H48N6O8
|
1
|
1 |
AC50 = 4410 nM
|
|
|
CP0809518
|
SID24815344
Show/Hide
|
C13H12N2O2S
|
1
|
1 |
AC50 = 4410 nM
|
|
|
CP0915517
|
SID131421177
Show/Hide
|
C27H37N3O4S
|
1
|
1 |
AC50 = 4410 nM
|
|
|
CP0916969
|
SID131444803
Show/Hide
|
C33H31FN2O6S
|
1
|
1 |
AC50 = 4410 nM
|
|
|
CP0941952
|
SID144191494
Show/Hide
|
C33H36F3N3O5S
|
1
|
1 |
AC50 = 4410 nM
|
|
|
CP0852372
|
SID144190595
Show/Hide
|
C18H20N2O2S
|
1
|
1 |
AC50 = 4420 nM
|
|
|
CP0933801
|
SID131464572
Show/Hide
|
C30H33N3O2
|
1
|
1 |
AC50 = 4420 nM
|
|
|
CP0039752
|
MLS002693850
Show/Hide
|
C17H11NO3
|
1
|
1 |
AC50 = 4430 nM
|
|
|
CP0408001
|
5-Bromo-3-phenyl-1H-indole-2-carboxylic acid [1-(4-hydroxy-phenyl)-meth-(E)-ylidene]-hydrazide
Show/Hide
|
C22H16BrN3O2
|
1
|
1 |
AC50 = 4430 nM
|
|
|
CP0880368
|
SID57261345
Show/Hide
|
C14H15ClN2O2
|
1
|
1 |
AC50 = 4430 nM
|
|
|
CP0906234
|
SID131411588
Show/Hide
|
C35H45Cl2N3O6S
|
1
|
1 |
AC50 = 4440 nM
|
|
|
CP0864559
|
SID131411725
Show/Hide
|
C36H46Cl2N4O5
|
1
|
1 |
AC50 = 4450 nM
|
|
|
CP0934608
|
SID131413159
Show/Hide
|
C34H43ClFN3O8S2
|
1
|
1 |
AC50 = 4450 nM
|
|
|
CP0856712
|
SID131412846
Show/Hide
|
C37H52F3N5O6
|
1
|
1 |
AC50 = 4460 nM
|
|
|
CP0942472
|
SID131410361
Show/Hide
|
C35H46ClN3O8S2
|
1
|
1 |
AC50 = 4470 nM
|
|
|
CP0012388
|
MLS000708339
Show/Hide
|
C19H22N4O5
|
1
|
1 |
AC50 = 4480 nM
|
|
|
CP0858471
|
SID89852970
Show/Hide
|
C16H13NO
|
1
|
1 |
AC50 = 4480 nM
|
|
|
CP0454032
|
4-(2-chloro-4,6-dimethoxy-anilino)-1,2-naphthoquinone
Show/Hide
|
C18H14ClNO4
|
1
|
1 |
AC50 = 4490 nM
|
|
|
CP0915291
|
SID131411785
Show/Hide
|
C39H47ClN4O7S
|
1
|
1 |
AC50 = 4510 nM
|
|
|
CP0239508
|
3-[1-[[1-(2,3-dihydro-1,4-benzodioxin-6-yl)-1,2,3,4-tetrazol-5-yl]-[2-(trifluoromethyloxy)phenyl]methyl]piperidin-4-yl]-1H-benzimidazol-2-one
Show/Hide
|
C29H26F3N7O4
|
1
|
1 |
AC50 = 4520 nM
|
|
|
CP0912291
|
SID87543219
Show/Hide
|
C36H44ClF3N4O7S
|
1
|
1 |
AC50 = 4520 nM
|
|
|
CP0685363
|
SID17507180
Show/Hide
|
C19H18N4O3
|
1
|
1 |
AC50 = 4540 nM
|
|
|
CP0940409
|
SID87541135
Show/Hide
|
C37H47Cl2N3O5
|
1
|
1 |
AC50 = 4540 nM
|
|
|
CP0847472
|
SID92764813
Show/Hide
|
C18H22IN3S2
|
1
|
1 |
AC50 = 4550 nM
|
|
|
CP0857094
|
SID131410784
Show/Hide
|
C34H44F3N3O6S2
|
1
|
1 |
AC50 = 4550 nM
|
|
|
CP0256447
|
1-(N-(2-chloro-1-oxoethyl)anilino)-3-phenylurea
Show/Hide
|
C15H14ClN3O2
|
1
|
1 |
AC50 = 4570 nM
|
|
|
CP0856710
|
SID131413828
Show/Hide
|
C32H38N2O5S
|
1
|
1 |
AC50 = 4570 nM
|
|
|
CP0890221
|
SID49642974
Show/Hide
|
C18H17ClN2O4S
|
1
|
1 |
AC50 = 4570 nM
|
|
|
CP0890545
|
SID49823076
Show/Hide
|
C22H22N2O4S2
|
1
|
1 |
AC50 = 4570 nM
|
|
|
CP0003832
|
N'-hydroxy-N-phenyloctanediamide
Show/Hide
|
C14H20N2O3
|
1
|
1 |
AC50 = 4580 nM
|
|
|
CP0014682
|
2-(4,5-dichloro-6-keto-pyridazin-1-yl)-N-(4-methyl-3-piperidinosulfonyl-phenyl)acetamide
Show/Hide
|
C18H20Cl2N4O4S
|
1
|
1 |
AC50 = 4580 nM
|
|
|
CP0395948
|
5-(2-methylquinolin-4-yl)sulfanyl-1,3,4-thiadiazol-2-amine
Show/Hide
|
C12H10N4S2
|
1
|
1 |
AC50 = 4580 nM
|
|
|
CP0864558
|
SID144188544
Show/Hide
|
C28H32N2O4S
|
1
|
1 |
AC50 = 4580 nM
|
|
|
CP0143443
|
3-(2-thienylsulfonyl)pyrazine-2-carbonitrile
Show/Hide
|
C9H5N3O2S2
|
1
|
1 |
AC50 = 4590 nM
|
|
|
CP0853619
|
SID844866
Show/Hide
|
C16H16O5S
|
1
|
1 |
AC50 = 4590 nM
|
|
|
CP0885785
|
SID131411728
Show/Hide
|
C36H46Cl2N4O5
|
1
|
1 |
AC50 = 4600 nM
|
|
|
CP0912882
|
SID49732953
Show/Hide
|
C15H19N3O3S2
|
1
|
1 |
AC50 = 4600 nM
|
|
|
CP0016685
|
3-(2,4-dichlorophenyl)-4-(1-methyl-1H-indol-3-yl)-2,5-dihydro-1H-pyrrole-2,5-dione
Show/Hide
|
C19H12Cl2N2O2
|
1
|
1 |
AC50 = 4610 nM
|
|
|
CP0882379
|
SID87542174
Show/Hide
|
C37H47F3N4O5
|
1
|
1 |
AC50 = 4610 nM
|
|
|
CP0047365
|
2-(4,5-dichloro-6-keto-pyridazin-1-yl)-N-(5-methoxy-2-methyl-4-nitro-phenyl)acetamide
Show/Hide
|
C14H12Cl2N4O5
|
1
|
1 |
AC50 = 4620 nM
|
|
|
CP0890220
|
SID131410267
Show/Hide
|
C38H48F3N3O5
|
1
|
1 |
AC50 = 4620 nM
|
|
|
CP0912885
|
SID131412706
Show/Hide
|
C37H48F3N3O6S
|
1
|
1 |
AC50 = 4620 nM
|
|
|
CP0462461
|
(3E,5E)-1-benzyl-3,5-bis(3-hydroxy-4-methoxy-benzylidene)-4-piperidone
Show/Hide
|
C28H27NO5
|
1
|
1 |
AC50 = 4630 nM
|
|
|
CP0884818
|
SID87539815
Show/Hide
|
C36H44F4N4O7S
|
1
|
1 |
AC50 = 4630 nM
|
|
|
CP0900322
|
SID85799757
Show/Hide
|
C32H37F3N4O7S
|
1
|
1 |
AC50 = 4640 nM
|
|
|
CP0908684
|
SID144192109
Show/Hide
|
C28H25FN2O4S
|
1
|
1 |
AC50 = 4640 nM
|
|
|
CP0908030
|
SID104170743
Show/Hide
|
C35H46FN3O9S2
|
1
|
1 |
AC50 = 4650 nM
|
|
|
CP0377553
|
(E)-2-(benzenesulfonyl)-3-[5-(3,4-dichlorophenyl)-2-furanyl]-N-(3-pyridinylmethyl)-2-propenamide
Show/Hide
|
C25H18Cl2N2O4S
|
1
|
1 |
AC50 = 4660 nM
|
|
|
CP0900524
|
SID87540250
Show/Hide
|
C36H46F3N3O6S
|
1
|
1 |
AC50 = 4660 nM
|
|
|
CP0940737
|
SID144192299
Show/Hide
|
C25H26N2O4S
|
1
|
1 |
AC50 = 4660 nM
|
|
|
CP0886576
|
SID131413116
Show/Hide
|
C35H46FN3O9S2
|
1
|
1 |
AC50 = 4670 nM
|
|
|
CP0907265
|
SID87218848
Show/Hide
|
C37H43N3O6S
|
1
|
1 |
AC50 = 4670 nM
|
|
|
CP0966625
|
SID87540619
Show/Hide
|
C36H44ClF3N4O7S
|
1
|
1 |
AC50 = 4680 nM
|
|
|
CP0868092
|
SID57269093
Show/Hide
|
C20H23F3N4O3
|
1
|
1 |
AC50 = 4700 nM
|
|
|
CP0869055
|
SID87543890
Show/Hide
|
C35H46ClN3O6S
|
1
|
1 |
AC50 = 4700 nM
|
|
|
CP0865417
|
SID164339411
Show/Hide
|
C20H32N2O2S
|
1
|
1 |
AC50 = 4720 nM
|
|
|
CP0873976
|
SID92764122
Show/Hide
|
C34H33Cl2N3O10
|
1
|
1 |
AC50 = 4720 nM
|
|
|
CP0864733
|
SID87539566
Show/Hide
|
C36H45ClF3N3O6S
|
1
|
1 |
AC50 = 4730 nM
|
|
|
CP0256394
|
MLS000588796
Show/Hide
|
C23H22N2O3
|
1
|
1 |
AC50 = 4740 nM
|
|
|
CP0862193
|
SID131409529
Show/Hide
|
C31H35F4N3O5S
|
1
|
1 |
AC50 = 4760 nM
|
|
|
CP0906230
|
SID104170713
Show/Hide
|
C34H43Cl2N3O8S2
|
1
|
1 |
AC50 = 4760 nM
|
|
|
CP0864735
|
SID51090004
Show/Hide
|
C23H30ClN3O5S2
|
1
|
1 |
AC50 = 4770 nM
|
|
|
CP0907294
|
SID131410334
Show/Hide
|
C37H45Cl2F3N4O5
|
1
|
1 |
AC50 = 4770 nM
|
|
|
CP0886263
|
SID87543866
Show/Hide
|
C35H46FN3O9S2
|
1
|
1 |
AC50 = 4780 nM
|
|
|
CP0935289
|
SID144199866
Show/Hide
|
C34H39N3O5
|
1
|
1 |
AC50 = 4780 nM
|
|
|
CP0862117
|
SID131411092
Show/Hide
|
C33H50N4O7S2
|
1
|
1 |
AC50 = 4790 nM
|
|
|
CP0864563
|
SID87540315
Show/Hide
|
C35H46ClN3O9S2
|
1
|
1 |
AC50 = 4800 nM
|
|
|
CP0851435
|
SID87335818
Show/Hide
|
C21H15ClN2O3S2
|
1
|
1 |
AC50 = 4820 nM
|
|
|
CP0909617
|
SID104170401
Show/Hide
|
C35H45FN4O7S
|
1
|
1 |
AC50 = 4820 nM
|
|
|
CP0846191
|
SID99358637
Show/Hide
|
C30H40N2O7S2
|
1
|
1 |
AC50 = 4830 nM
|
|
|
CP0308667
|
2-(4,5-dichloro-6-keto-pyridazin-1-yl)-N-[3-(diethylsulfamoyl)-4-methyl-phenyl]acetamide
Show/Hide
|
C17H20Cl2N4O4S
|
1
|
1 |
AC50 = 4840 nM
|
|
|
CP0862953
|
SID104170382
Show/Hide
|
C35H44Cl3N3O6S
|
1
|
1 |
AC50 = 4840 nM
|
|
|
CP0900423
|
SID131414068
Show/Hide
|
C32H38N2O5S
|
1
|
1 |
AC50 = 4840 nM
|
|
|
CP0952399
|
SID131412342
Show/Hide
|
C35H44ClFN4O7S
|
1
|
1 |
AC50 = 4840 nM
|
|
|
CP0881162
|
SID131412024
Show/Hide
|
C35H44Cl2FN3O6S
|
1
|
1 |
AC50 = 4850 nM
|
|
|
CP0445625
|
MLS003129868
Show/Hide
|
C32H36ClN3O5S
|
1
|
1 |
AC50 = 4860 nM
|
|
|
CP0913849
|
SID87541535
Show/Hide
|
C37H47F3N4O5
|
1
|
1 |
AC50 = 4860 nM
|
|
|
CP0075432
|
5,7-DIIODO-8-HYDROXYQUINOLINE
Show/Hide
|
C9H5I2NO
|
1
|
1 |
AC50 = 4870 nM
|
|
|
CP0862123
|
SID87542580
Show/Hide
|
C38H47F3N4O6
|
1
|
1 |
AC50 = 4870 nM
|
|
|
CP0900396
|
SID131461232
Show/Hide
|
C26H24FN3O3S
|
1
|
1 |
AC50 = 4870 nM
|
|
|
CP0213593
|
2-(2-indolin-1-yl-2-keto-ethyl)-1,1-diketo-1,2-benzothiazol-3-one
Show/Hide
|
C17H14N2O4S
|
1
|
1 |
AC50 = 4880 nM
|
|
|
CP0796946
|
SID22414029
Show/Hide
|
C19H22ClNO
|
1
|
1 |
AC50 = 4880 nM
|
|
|
CP0868348
|
SID131415030
Show/Hide
|
C31H31FN2O7S
|
1
|
1 |
AC50 = 4880 nM
|
|
|
CP0942413
|
SID87541378
Show/Hide
|
C36H44F4N4O7S
|
1
|
1 |
AC50 = 4880 nM
|
|
|
CP0864688
|
SID131464142
Show/Hide
|
C31H33N3O3
|
1
|
1 |
AC50 = 4900 nM
|
|
|
CP0907408
|
SID87543373
Show/Hide
|
C33H43Cl2N3O6S2
|
1
|
1 |
AC50 = 4910 nM
|
|
|
CP0851534
|
SID87543664
Show/Hide
|
C35H46F3N5O8S
|
1
|
1 |
AC50 = 4920 nM
|
|
|
CP0888885
|
SID89650061
Show/Hide
|
C15H12N6OS2
|
1
|
1 |
AC50 = 4920 nM
|
|
|
CP0856557
|
SID99356266
Show/Hide
|
C19H18O5
|
1
|
1 |
AC50 = 4950 nM
|
|
|
CP0856714
|
SID131411914
Show/Hide
|
C37H47F3N4O5
|
1
|
1 |
AC50 = 4950 nM
|
|
|
CP0862097
|
SID87543793
Show/Hide
|
C34H43ClFN3O8S2
|
1
|
1 |
AC50 = 4970 nM
|
|
|
CP0942508
|
SID87542761
Show/Hide
|
C37H52F3N5O6
|
1
|
1 |
AC50 = 4980 nM
|
|
|
CP0848114
|
SID87539610
Show/Hide
|
C35H50ClN3O7S
|
1
|
1 |
AC50 = 4990 nM
|
|
|
CP0188611
|
3-[(4-Nitro-phenylaminooxalyl)-amino]-benzoic acid
Show/Hide
|
C15H11N3O6
|
1
|
1 |
AC50 = 5000 nM
|
|
|
CP0311113
|
1-[[5-[5-(4-methylphenyl)thieno[2,3-d]pyrimidin-4-yl]sulfanyl-1,3,4-oxadiazol-2-yl]methyl]azepan-2-one
Show/Hide
|
C22H21N5O2S2
|
1
|
1 |
AC50 = 5000 nM
|
|
|
CP0857042
|
SID131410332
Show/Hide
|
C37H45Cl2F3N4O5
|
1
|
1 |
AC50 = 5000 nM
|
|
|
CP0908715
|
SID87544028
Show/Hide
|
C35H45Cl2N3O6S
|
1
|
1 |
AC50 = 5000 nM
|
|
|
CP0281587
|
4-(2,2-difluoroethylamino)-6-(3,5-difluorophenylamino)-1,3,5-triazine-2-carbonitrile
Show/Hide
|
C12H8F4N6
|
1
|
1 |
AC50 = 5010 nM
|
|
|
CP0846337
|
SID51087203
Show/Hide
|
C15H15ClN2O4S2
|
1
|
1 |
AC50 = 5010 nM
|
|
|
CP0709991
|
SID49828905
Show/Hide
|
C22H20FN3O2S2
|
1
|
1 |
AC50 = 5040 nM
|
|
|
CP0864578
|
SID131412182
Show/Hide
|
C34H43ClFN3O8S2
|
1
|
1 |
AC50 = 5050 nM
|
|
|
CP0909153
|
SID131411911
Show/Hide
|
C37H47F3N4O5
|
1
|
1 |
AC50 = 5050 nM
|
|
|
CP0942468
|
SID131414517
Show/Hide
|
C32H37N3O4
|
1
|
1 |
AC50 = 5050 nM
|
|
|
CP0865940
|
SID24830222
Show/Hide
|
C14H15Cl2F3N2O2
|
1
|
1 |
AC50 = 5060 nM
|
|
|
CP0908126
|
SID87543057
Show/Hide
|
C36H45Cl2FN4O5
|
1
|
1 |
AC50 = 5060 nM
|
|
|
CP0912631
|
SID131463011
Show/Hide
|
C29H35N3O2
|
1
|
1 |
AC50 = 5070 nM
|
|
|
CP0211482
|
MLS000707627
Show/Hide
|
C24H23ClFN3O5S2
|
1
|
1 |
AC50 = 5080 nM
|
|
|
CP0852369
|
SID87541153
Show/Hide
|
C36H45F4N3O6S
|
1
|
1 |
AC50 = 5080 nM
|
|
|
CP0943350
|
SID131410335
Show/Hide
|
C37H45Cl2F3N4O5
|
1
|
1 |
AC50 = 5080 nM
|
|
|
CP0447171
|
MLS003124134
Show/Hide
|
C23H22N4O5S
|
1
|
1 |
AC50 = 5090 nM
|
|
|
CP0950365
|
SID144194030
Show/Hide
|
C25H24FN3O2
|
1
|
1 |
AC50 = 5090 nM
|
|
|
CP0249481
|
cid_779573
Show/Hide
|
C11H8Cl2N2O
|
1
|
1 |
AC50 = 5110 nM
|
|
|
CP0196797
|
5-chloranyl-2-ethylsulfonyl-N-[4-[methyl(phenyl)sulfamoyl]phenyl]pyrimidine-4-carboxamide
Show/Hide
|
C20H19ClN4O5S2
|
1
|
1 |
AC50 = 5120 nM
|
|
|
CP0444263
|
1-(4-chlorophenyl)-3-[3-[(2-chlorophenyl)sulfamoyl]-4-(1-pyrrolidinyl)phenyl]urea
Show/Hide
|
C23H22Cl2N4O3S
|
1
|
1 |
AC50 = 5130 nM
|
|
|
CP0851524
|
SID49823832
Show/Hide
|
C15H12N2O5
|
1
|
1 |
AC50 = 5130 nM
|
|
|
CP0912771
|
SID22408831
Show/Hide
|
C24H22N2O2S
|
1
|
1 |
AC50 = 5150 nM
|
|
|
CP0912916
|
SID104170793
Show/Hide
|
C35H47N3O9S2
|
1
|
1 |
AC50 = 5150 nM
|
|
|
CP0666075
|
SID24809040
Show/Hide
|
C19H22N4O5
|
1
|
1 |
AC50 = 5170 nM
|
|
|
CP0942507
|
SID131426088
Show/Hide
|
C30H33N3O6S
|
1
|
1 |
AC50 = 5170 nM
|
|
|
CP0959673
|
SID87543477
Show/Hide
|
C36H45F4N3O6S
|
1
|
1 |
AC50 = 5170 nM
|
|
|
CP0879954
|
SID87541129
Show/Hide
|
C37H45F3N4O6
|
1
|
1 |
AC50 = 5180 nM
|
|
|
CP0196339
|
1,4,5,6-Tetrahydro-cyclopentapyrazole-3-carboxylic acid [1-thiophen-2-yl-eth-(E)-ylidene]-hydrazide
Show/Hide
|
C13H14N4OS
|
1
|
1 |
AC50 = 5190 nM
|
|
|
CP0181010
|
MLS000707959
Show/Hide
|
C17H13N3O6
|
1
|
1 |
AC50 = 5200 nM
|
|
|
CP0423983
|
5-Nitro-furan-2-carboxylic acid {3-[(furan-2-carbonyl)-amino]-phenyl}-amide
Show/Hide
|
C16H11N3O6
|
1
|
1 |
AC50 = 5200 nM
|
|
|
CP0886462
|
SID144190809
Show/Hide
|
C31H33FN4O5S
|
1
|
1 |
AC50 = 5200 nM
|
|
|
CP0454310
|
(3aS,5S,9aS)-5-[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]-2-phenylhexahydro-7H-pyrrolo[3,4-g]pyrrolizin-1(2H)-one
Show/Hide
|
C25H26N4O2
|
1
|
1 |
AC50 = 5210 nM
|
|
|
CP0906890
|
SID131413001
Show/Hide
|
C35H52ClN3O6S
|
1
|
1 |
AC50 = 5210 nM
|
|
|
CP0857034
|
SID87539575
Show/Hide
|
C36H47Cl2N3O6S
|
1
|
1 |
AC50 = 5220 nM
|
|
|
CP0881652
|
SID87543040
Show/Hide
|
C37H45F4N5O6
|
1
|
1 |
AC50 = 5230 nM
|
|
|
CP0930588
|
SID131412501
Show/Hide
|
C34H44ClN3O8S2
|
1
|
1 |
AC50 = 5230 nM
|
|
|
CP0864552
|
SID144191409
Show/Hide
|
C33H36F3N3O5S
|
1
|
1 |
AC50 = 5240 nM
|
|
|
CP0906897
|
SID7970999
Show/Hide
|
C27H27N5O2S
|
1
|
1 |
AC50 = 5250 nM
|
|
|
CP0874781
|
SID131412255
Show/Hide
|
C37H46F4N4O5
|
1
|
1 |
AC50 = 5260 nM
|
|
|
CP0897518
|
SID87543988
Show/Hide
|
C37H45F3N4O6
|
1
|
1 |
AC50 = 5260 nM
|
|
|
CP0942477
|
SID144188742
Show/Hide
|
C21H23FN2O4S
|
1
|
1 |
AC50 = 5260 nM
|
|
|
CP0006902
|
N'-hydroxy-N-[1-[2-(hydroxymethyl)pyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]-2-pentylbutanediamide
Show/Hide
|
C19H35N3O5
|
1
|
1 |
AC50 = 5270 nM
|
|
|
CP0299127
|
4,6-Dimethyl-3-(3-naphthalen-1-yl-acryloyl)-1H-pyridin-2-one
Show/Hide
|
C20H17NO2
|
1
|
1 |
AC50 = 5270 nM
|
|
|
CP0873857
|
SID131414074
Show/Hide
|
C32H38N2O5S
|
1
|
1 |
AC50 = 5270 nM
|
|
|
CP0895550
|
(4-benzhydrylpiperazin-1-yl)(5-methyl-4-nitroisoxazol-3-yl)methanone
Show/Hide
|
C22H22N4O4
|
1
|
1 |
AC50 = 5280 nM
|
|
|
CP0959675
|
SID87542541
Show/Hide
|
C39H47ClN4O7S
|
1
|
1 |
AC50 = 5290 nM
|
|
|
CP0779227
|
SID85147444
Show/Hide
|
C28H24ClF3N4O6S
|
1
|
1 |
AC50 = 5300 nM
|
|
|
CP0875589
|
SID56316401
Show/Hide
|
C17H18N4O5S2
|
1
|
1 |
AC50 = 5300 nM
|
|
|
CP0885652
|
SID131410336
Show/Hide
|
C37H45Cl2F3N4O5
|
1
|
1 |
AC50 = 5300 nM
|
|
|
CP0196877
|
2-(4-propan-2-ylphenyl)-1,3-benzothiazole
Show/Hide
|
C16H15NS
|
1
|
1 |
AC50 = 5310 nM
|
|
|
CP0286110
|
5-nitro-N-[4-(4-propanoylpiperazin-1-yl)phenyl]furan-2-carboxamide
Show/Hide
|
C18H20N4O5
|
1
|
1 |
AC50 = 5310 nM
|
|
|
CP0827100
|
SID24833101
Show/Hide
|
C26H30N4O4
|
1
|
1 |
AC50 = 5320 nM
|
|
|
CP0884586
|
SID87218860
Show/Hide
|
C36H40FN3O6S
|
1
|
1 |
AC50 = 5320 nM
|
|
|
CP0121968
|
(2,6-dimethyl-4-quinolyl)-(4-nitrophenyl)amine
Show/Hide
|
C17H15N3O2
|
1
|
1 |
AC50 = 5330 nM
|
|
|
CP0885846
|
SID131409313
Show/Hide
|
C29H34F3N3O5S2
|
1
|
1 |
AC50 = 5330 nM
|
|
|
CP0338169
|
5-chloranyl-2-ethylsulfonyl-N-[4-(3-methylpiperidin-1-yl)sulfonylphenyl]pyrimidine-4-carboxamide
Show/Hide
|
C19H23ClN4O5S2
|
1
|
1 |
AC50 = 5340 nM
|
|
|
CP0898937
|
SID57260110
Show/Hide
|
C6H10N6O
|
1
|
1 |
AC50 = 5340 nM
|
|
|
CP0879115
|
SID92763673
Show/Hide
|
C42H55N5O3S2
|
1
|
1 |
AC50 = 5350 nM
|
|
|
CP0891365
|
SID87540874
Show/Hide
|
C37H46F4N4O5
|
1
|
1 |
AC50 = 5360 nM
|
|
|
CP0381122
|
(E)-N-[2-(cyclohexylamino)-2-keto-ethyl]-4-(2-hydroxy-4-methoxy-phenyl)-4-keto-N-(2-methoxyethyl)but-2-enamide
Show/Hide
|
C22H30N2O6
|
1
|
1 |
AC50 = 5380 nM
|
|
|
CP0854901
|
SID56422465
Show/Hide
|
C29H46O12
|
1
|
1 |
AC50 = 5380 nM
|
|
|
CP0178237
|
2-hydroxy-N-(4-methoxyphenyl)-5-nitro-benzamide
Show/Hide
|
C14H12N2O5
|
1
|
1 |
AC50 = 5390 nM
|
|
|
CP0908125
|
SID85797536
Show/Hide
|
C36H52N4O6
|
1
|
1 |
AC50 = 5390 nM
|
|
|
CP0944063
|
SID87543075
Show/Hide
|
C31H41Cl2N3O4
|
1
|
1 |
AC50 = 5390 nM
|
|
|
CP0950341
|
SID131411783
Show/Hide
|
C39H47ClN4O7S
|
1
|
1 |
AC50 = 5390 nM
|
|
|
CP0905181
|
SID87540264
Show/Hide
|
C39H47FN4O7S
|
1
|
1 |
AC50 = 5400 nM
|
|
|
CP0477521
|
MLS002701874
Show/Hide
|
C18H14O5
|
1
|
1 |
AC50 = 5410 nM
|
|
|
CP0873653
|
SID57263481
Show/Hide
|
C23H27N3O7S
|
1
|
1 |
AC50 = 5420 nM
|
|
|
CP0891370
|
SID87541470
Show/Hide
|
C36H54N4O5
|
1
|
1 |
AC50 = 5420 nM
|
|
|
CP0891778
|
SID131411336
Show/Hide
|
C37H45F3N4O6
|
1
|
1 |
AC50 = 5420 nM
|
|
|
CP0908901
|
SID87542458
Show/Hide
|
C38H47F3N4O7
|
1
|
1 |
AC50 = 5420 nM
|
|
|
CP0897515
|
SID49647125
Show/Hide
|
C15H20O4
|
1
|
1 |
AC50 = 5430 nM
|
|
|
CP0912515
|
SID131412210
Show/Hide
|
C35H46ClN3O6S
|
1
|
1 |
AC50 = 5430 nM
|
|
|
CP0915300
|
SID131409441
Show/Hide
|
C38H42N4O6
|
1
|
1 |
AC50 = 5450 nM
|
|
|
CP0945689
|
SID87540331
Show/Hide
|
C36H45ClF3N3O6S
|
1
|
1 |
AC50 = 5450 nM
|
|
|
CP0439662
|
MLS001172197
Show/Hide
|
C19H18ClNO4
|
1
|
1 |
AC50 = 5460 nM
|
|
|
CP0664710
|
SID49681823
Show/Hide
|
C27H30ClNO11
|
1
|
1 |
AC50 = 5460 nM
|
|
|
CP0912638
|
SID87543635
Show/Hide
|
C37H45Cl2F3N4O5
|
1
|
1 |
AC50 = 5490 nM
|
|
|
CP0821788
|
SID24800864
Show/Hide
|
C19H18N4O3
|
1
|
1 |
AC50 = 5500 nM
|
|
|
CP0862956
|
SID121284982
Show/Hide
|
C29H31N7O3
|
1
|
1 |
AC50 = 5500 nM
|
|
|
CP0890212
|
SID87541270
Show/Hide
|
C35H46FN3O8S2
|
1
|
1 |
AC50 = 5500 nM
|
|
|
CP0906899
|
SID87540394
Show/Hide
|
C35H52ClN3O6S
|
1
|
1 |
AC50 = 5500 nM
|
|
|
CP0864576
|
SID87542870
Show/Hide
|
C36H55N3O6S
|
1
|
1 |
AC50 = 5510 nM
|
|
|
CP0411508
|
MLS003107619
Show/Hide
|
C35H33F2N5O8S
|
1
|
1 |
AC50 = 5520 nM
|
|
|
CP0885769
|
SID87543806
Show/Hide
|
C36H46F3N5O5
|
1
|
1 |
AC50 = 5520 nM
|
|
|
CP0912918
|
SID87543248
Show/Hide
|
C34H43Cl2N3O8S2
|
1
|
1 |
AC50 = 5520 nM
|
|
|
CP0926606
|
SID144188466
Show/Hide
|
C29H29N3O4
|
1
|
1 |
AC50 = 5520 nM
|
|
|
CP0966624
|
SID87541920
Show/Hide
|
C36H45F4N3O6S
|
1
|
1 |
AC50 = 5540 nM
|
|
|
CP0890215
|
SID87541918
Show/Hide
|
C36H51FN4O6
|
1
|
1 |
AC50 = 5550 nM
|
|
|
CP0949361
|
SID131447484
Show/Hide
|
C25H24N2O3
|
1
|
1 |
AC50 = 5550 nM
|
|
|
CP0846809
|
SID144199879
Show/Hide
|
C34H37F3N4O4
|
1
|
1 |
AC50 = 5560 nM
|
|
|
CP0888946
|
SID92763805
Show/Hide
|
C15H21NO4
|
1
|
1 |
AC50 = 5560 nM
|
|
|
CP0930557
|
SID131411245
Show/Hide
|
C38H47F3N4O7
|
1
|
1 |
AC50 = 5560 nM
|
|
|
CP0930587
|
SID87543003
Show/Hide
|
C37H48F3N3O6S
|
1
|
1 |
AC50 = 5570 nM
|
|
|
CP0950780
|
SID131446864
Show/Hide
|
C22H21FN2O3S
|
1
|
1 |
AC50 = 5570 nM
|
|
|
CP0420391
|
1-[2-(4-methoxyphenyl)-3,4-dimethyl-7-pyrazolo[3,4-d]pyridazinyl]-N-[(3-methylphenyl)methyl]-4-piperidinecarboxamide
Show/Hide
|
C28H32N6O2
|
1
|
1 |
AC50 = 5580 nM
|
|
|
CP0909154
|
SID87540293
Show/Hide
|
C37H48F3N3O7S
|
1
|
1 |
AC50 = 5590 nM
|
|
|
CP0932245
|
SID131446654
Show/Hide
|
C25H24FN3O2
|
1
|
1 |
AC50 = 5590 nM
|
|
|
CP0827516
|
SID24819479
Show/Hide
|
C11H8Cl2N2O2
|
1
|
1 |
AC50 = 5620 nM
|
|
|
CP0884740
|
SID131412736
Show/Hide
|
C36H44F4N4O7S
|
1
|
1 |
AC50 = 5620 nM
|
|
|
CP0906233
|
SID131454588
Show/Hide
|
C28H32F3N3O5
|
1
|
1 |
AC50 = 5620 nM
|
|
|
CP0907412
|
SID87543225
Show/Hide
|
C38H47F3N4O7
|
1
|
1 |
AC50 = 5640 nM
|
|
|
CP0728770
|
SID24823447
Show/Hide
|
C21H22N8O4
|
1
|
1 |
AC50 = 5650 nM
|
|
|
CP0167831
|
5-chloranyl-N-[4-(2-ethylpiperidin-1-yl)sulfonylphenyl]-2-methylsulfonyl-pyrimidine-4-carboxamide
Show/Hide
|
C19H23ClN4O5S2
|
1
|
1 |
AC50 = 5670 nM
|
|
|
CP0879867
|
SID131464910
Show/Hide
|
C31H33N3O3
|
1
|
1 |
AC50 = 5670 nM
|
|
|
CP0942473
|
SID131454052
Show/Hide
|
C31H34N2O6
|
1
|
1 |
AC50 = 5670 nM
|
|
|
CP0966334
|
SID87218864
Show/Hide
|
C31H37Cl2N3O5S
|
1
|
1 |
AC50 = 5670 nM
|
|
|
CP0864700
|
SID134962038
Show/Hide
|
C34H38N4O6
|
1
|
1 |
AC50 = 5680 nM
|
|
|
CP0046285
|
(1E)-2-[6-[[amino-[(E)-[amino-(4-chloroanilino)methylene]amino]methylene]amino]hexyl]-1-[amino-(4-chloroanilino)methylene]guanidine;hydrochloride
Show/Hide
|
C22H30Cl2N10
|
1
|
1 |
AC50 = 5690 nM
|
|
|
CP0865129
|
SID85799724
Show/Hide
|
C33H35ClN4O6S
|
1
|
1 |
AC50 = 5690 nM
|
|
|
CP0892939
|
SID85803792
Show/Hide
|
C31H36F3N5O4
|
1
|
1 |
AC50 = 5690 nM
|
|
|
CP0757065
|
SID17403358
Show/Hide
|
C19H16BrN3O2S2
|
1
|
1 |
AC50 = 5710 nM
|
|
|
CP0879866
|
SID87541708
Show/Hide
|
C36H46F3N3O6S
|
1
|
1 |
AC50 = 5710 nM
|
|
|
CP0930590
|
SID87542170
Show/Hide
|
C38H49F3N4O6
|
1
|
1 |
AC50 = 5710 nM
|
|
|
CP0001364
|
1,3-dihydrobenzo[f]benzimidazole-2,4,9-trione
Show/Hide
|
C11H6N2O3
|
1
|
1 |
AC50 = 5720 nM
|
|
|
CP0137427
|
1-[2-(dimethylamino)ethylamino]-4-(hydroxymethyl)-7-oxidanyl-thioxanthen-9-one
Show/Hide
|
C18H20N2O3S
|
1
|
1 |
AC50 = 5720 nM
|
|
|
CP0884744
|
SID144188468
Show/Hide
|
C29H29N3O4
|
1
|
1 |
AC50 = 5720 nM
|
|
|
CP0884746
|
SID87541940
Show/Hide
|
C31H35Cl2FN4O4
|
1
|
1 |
AC50 = 5720 nM
|
|
|
CP0010841
|
1-(3-Ethylsulfanyl-[1,2,4]thiadiazol-5-yl)-3-(3-fluoro-phenyl)-urea
Show/Hide
|
C11H11FN4OS2
|
1
|
1 |
AC50 = 5730 nM
|
|
|
CP0378735
|
MLS001125540
Show/Hide
|
C16H14N2O2S
|
1
|
1 |
AC50 = 5740 nM
|
|
|
CP0942412
|
SID131412379
Show/Hide
|
C36H46F3N3O6S
|
1
|
1 |
AC50 = 5740 nM
|
|
|
CP0862125
|
SID131414963
Show/Hide
|
C31H31FN2O7S
|
1
|
1 |
AC50 = 5760 nM
|
|
|
CP0890213
|
SID131412933
Show/Hide
|
C36H49N3O8S2
|
1
|
1 |
AC50 = 5760 nM
|
|
|
CP0966626
|
SID144192342
Show/Hide
|
C28H22F2N2O3
|
1
|
1 |
AC50 = 5770 nM
|
|
|
CP0879951
|
SID131412531
Show/Hide
|
C40H50N4O7S
|
1
|
1 |
AC50 = 5780 nM
|
|
|
CP0891606
|
SID858166
Show/Hide
|
C16H15NO5
|
1
|
1 |
AC50 = 5790 nM
|
|
|
CP0864684
|
SID85809239
Show/Hide
|
C37H48N4O4
|
1
|
1 |
AC50 = 5800 nM
|
|
|
CP0865837
|
SID121284948
Show/Hide
|
C30H27N7O4
|
1
|
1 |
AC50 = 5800 nM
|
|
|
CP0940510
|
SID131434103
Show/Hide
|
C33H39N3O6S
|
1
|
1 |
AC50 = 5800 nM
|
|
|
CP0890223
|
SID87540516
Show/Hide
|
C36H46F3N3O6S
|
1
|
1 |
AC50 = 5820 nM
|
|
|
CP0176768
|
5-Nitro-furan-2-carboxylic acid [4-(4-acetyl-piperazin-1-yl)-3-chloro-phenyl]-amide
Show/Hide
|
C17H17ClN4O5
|
1
|
1 |
AC50 = 5830 nM
|
|
|
CP0957475
|
SID131410529
Show/Hide
|
C36H45F4N3O6S
|
1
|
1 |
AC50 = 5830 nM
|
|
|
CP0908890
|
SID87542969
Show/Hide
|
C34H43Cl2N3O8S2
|
1
|
1 |
AC50 = 5860 nM
|
|
|
CP0888892
|
SID131413980
Show/Hide
|
C32H38N2O5S
|
1
|
1 |
AC50 = 5870 nM
|
|
|
CP0852172
|
SID87550751
Show/Hide
|
C21H26N2O7S
|
1
|
1 |
AC50 = 5880 nM
|
|
|
CP0883291
|
SID85805553
Show/Hide
|
C39H47FN4O7S
|
1
|
1 |
AC50 = 5880 nM
|
|
|
CP0906901
|
SID134961993
Show/Hide
|
C32H36FN3O5S
|
1
|
1 |
AC50 = 5880 nM
|
|
|
CP0942587
|
SID131425986
Show/Hide
|
C31H33FN2O5S
|
1
|
1 |
AC50 = 5880 nM
|
|
|
CP0878201
|
SID49826806
Show/Hide
|
C21H26N4O2S
|
1
|
1 |
AC50 = 5890 nM
|
|
|
CP0879870
|
SID87539664
Show/Hide
|
C34H45F6N3O5
|
1
|
1 |
AC50 = 5890 nM
|
|
|
CP0129110
|
3-Phenyl-1H-naphtho[2,1-b]pyran-1-one
Show/Hide
|
C19H12O2
|
1
|
1 |
AC50 = 5900 nM
|
|
|
CP0862954
|
SID87541725
Show/Hide
|
C36H45ClF3N3O6S
|
1
|
1 |
AC50 = 5900 nM
|
|
|
CP0864736
|
SID92764237
Show/Hide
|
C22H17ClO5
|
1
|
1 |
AC50 = 5900 nM
|
|
|
CP0930592
|
SID99356410
Show/Hide
|
C32H40N4O4
|
1
|
1 |
AC50 = 5900 nM
|
|
|
CP0104284
|
4-[(3-allyl-4-oxo-2-thioxo-1,3-thiazolidin-5-ylidene)methyl]-2-ethoxy-3-nitrophenyl acetate
Show/Hide
|
C17H16N2O6S2
|
1
|
1 |
AC50 = 5910 nM
|
|
|
CP0468757
|
2-chloro-N-heptyl-N-(3-methylphenyl)acetamide
Show/Hide
|
C16H24ClNO
|
1
|
1 |
AC50 = 5910 nM
|
|
|
CP0890222
|
SID87540064
Show/Hide
|
C37H46F4N4O5
|
1
|
1 |
AC50 = 5910 nM
|
|
|
CP0910496
|
SID87539806
Show/Hide
|
C34H43ClFN3O8S2
|
1
|
1 |
AC50 = 5920 nM
|
|
|
CP0303163
|
4-propylbenzoic acid [(Z)-[amino(2-pyridinyl)methylidene]amino] ester
Show/Hide
|
C16H17N3O2
|
1
|
1 |
AC50 = 5930 nM
|
|
|
CP0926608
|
SID131443807
Show/Hide
|
C27H26ClFN2O6S
|
1
|
1 |
AC50 = 5930 nM
|
|
|
CP0855583
|
SID164339397
Show/Hide
|
C18H16Cl2N4O2S2
|
1
|
1 |
AC50 = 5940 nM
|
|
|
CP0875021
|
SID85272359
Show/Hide
|
C34H38N4O6S
|
1
|
1 |
AC50 = 5940 nM
|
|
|
CP0691829
|
SID49722558
Show/Hide
|
C27H30N6O
|
1
|
1 |
AC50 = 5950 nM
|
|
|
CP0771382
|
SID17507447
Show/Hide
|
C11H9NO2S
|
1
|
1 |
AC50 = 5950 nM
|
|
|
CP0944036
|
SID131410786
Show/Hide
|
C34H44F3N3O6S2
|
1
|
1 |
AC50 = 5950 nM
|
|
|
CP0908889
|
SID131446863
Show/Hide
|
C22H21FN2O3S
|
1
|
1 |
AC50 = 5960 nM
|
|
|
CP0395879
|
3-[6-[4-(2,5-dimethylphenyl)-1-piperazinyl]-6-oxohexyl]-6-(4-morpholinyl)-2-sulfanylidene-1H-quinazolin-4-one
Show/Hide
|
C30H39N5O3S
|
1
|
1 |
AC50 = 5970 nM
|
|
|
CP0860522
|
SID131421176
Show/Hide
|
C27H37N3O4S
|
1
|
1 |
AC50 = 5970 nM
|
|
|
CP0881740
|
SID144190858
Show/Hide
|
C32H35FN4O5S
|
1
|
1 |
AC50 = 5970 nM
|
|
|
CP0885695
|
SID85807677
Show/Hide
|
C32H33F6N5O5
|
1
|
1 |
AC50 = 5970 nM
|
|
|
CP0890224
|
SID144197423
Show/Hide
|
C22H28N2O4S
|
1
|
1 |
AC50 = 5980 nM
|
|
|
CP0900573
|
SID131413096
Show/Hide
|
C38H49F3N4O6
|
1
|
1 |
AC50 = 5980 nM
|
|
|
CP0942497
|
SID87540342
Show/Hide
|
C37H48F3N3O6S
|
1
|
1 |
AC50 = 5990 nM
|
|
|
CP0884815
|
SID144190990
Show/Hide
|
C31H33FN4O5S
|
1
|
1 |
AC50 = 6000 nM
|
|
|
CP0912917
|
SID131447132
Show/Hide
|
C23H28N2O2
|
1
|
1 |
AC50 = 6020 nM
|
|
|
CP0864689
|
SID131413902
Show/Hide
|
C29H33N3O6S2
|
1
|
1 |
AC50 = 6030 nM
|
|
|
CP0960190
|
SID131408963
Show/Hide
|
C31H36F3N3O5S
|
1
|
1 |
AC50 = 6030 nM
|
|
|
CP0297405
|
MLS000707180
Show/Hide
|
C13H12ClN3O4S2
|
1
|
1 |
AC50 = 6050 nM
|
|
|
CP0846810
|
SID131447312
Show/Hide
|
C27H28N2O3
|
1
|
1 |
AC50 = 6050 nM
|
|
|
CP0873856
|
SID17509635
Show/Hide
|
C21H23Cl2N3O2
|
1
|
1 |
AC50 = 6050 nM
|
|
|
CP0411347
|
5-dibenzo[1,2-d:1',2'-g][7]annulenone
Show/Hide
|
C15H10O
|
1
|
1 |
AC50 = 6070 nM
|
|
|
CP0113920
|
cid_72813
Show/Hide
|
C10H6Cl2N2O
|
1
|
1 |
AC50 = 6100 nM
|
|
|
CP0882533
|
SID131411822
Show/Hide
|
C37H48F3N3O7S
|
1
|
1 |
AC50 = 6100 nM
|
|
|
CP0966630
|
SID121282591
Show/Hide
|
C35H44ClFN4O7S
|
1
|
1 |
AC50 = 6110 nM
|
|
|
CP0398869
|
MLS003107613
Show/Hide
|
C31H39N5O8S
|
1
|
1 |
AC50 = 6120 nM
|
|
|
CP0966619
|
SID131461120
Show/Hide
|
C24H27FN2O3S
|
1
|
1 |
AC50 = 6120 nM
|
|
|
CP0448584
|
2-methylene-6-(2-methylpropoxy)-4,9-dihydro-3H-carbazol-1-one
Show/Hide
|
C17H19NO2
|
1
|
1 |
AC50 = 6140 nM
|
|
|
CP0700418
|
SID22410794
Show/Hide
|
C12H10N2O2S
|
1
|
1 |
AC50 = 6140 nM
|
|
|
CP0862127
|
SID131412385
Show/Hide
|
C36H46F3N3O6S
|
1
|
1 |
AC50 = 6140 nM
|
|
|
CP0872670
|
SID92764451
Show/Hide
|
C21H23NO4S
|
1
|
1 |
AC50 = 6140 nM
|
|
|
CP0907414
|
SID131462625
Show/Hide
|
C27H34N2O4S
|
1
|
1 |
AC50 = 6140 nM
|
|
|
CP0942414
|
SID87540574
Show/Hide
|
C37H52F3N5O6
|
1
|
1 |
AC50 = 6150 nM
|
|
|
CP0942604
|
SID85799028
Show/Hide
|
C38H39N5O5
|
1
|
1 |
AC50 = 6150 nM
|
|
|
CP0943303
|
SID131442891
Show/Hide
|
C33H31FN2O7S
|
1
|
1 |
AC50 = 6150 nM
|
|
|
CP0898774
|
SID131414194
Show/Hide
|
C30H40N2O7S2
|
1
|
1 |
AC50 = 6160 nM
|
|
|
CP0907540
|
SID131412707
Show/Hide
|
C37H48F3N3O6S
|
1
|
1 |
AC50 = 6160 nM
|
|
|
CP0908036
|
SID131434102
Show/Hide
|
C33H39N3O6S
|
1
|
1 |
AC50 = 6160 nM
|
|
|
CP0912878
|
SID85804191
Show/Hide
|
C38H48F3N3O5
|
1
|
1 |
AC50 = 6160 nM
|
|
|
CP0909181
|
SID131448024
Show/Hide
|
C23H27N3O2
|
1
|
1 |
AC50 = 6170 nM
|
|
|
CP0442210
|
3-(benzenesulfonyl)-N-[3-(dimethylamino)propyl]-N-(4-methyl-1,3-benzothiazol-2-yl)propanamide
Show/Hide
|
C22H27N3O3S2
|
1
|
1 |
AC50 = 6180 nM
|
|
|
CP0885643
|
SID87542109
Show/Hide
|
C34H44ClN3O8S2
|
1
|
1 |
AC50 = 6180 nM
|
|
|
CP0889188
|
SID131414402
Show/Hide
|
C30H38FN3O5S
|
1
|
1 |
AC50 = 6200 nM
|
|
|
CP0907784
|
SID104170763
Show/Hide
|
C36H47Cl2N3O6S
|
1
|
1 |
AC50 = 6200 nM
|
|
|
CP0886508
|
SID85802255
Show/Hide
|
C32H38F3N3O6S
|
1
|
1 |
AC50 = 6210 nM
|
|
|
CP0864574
|
SID131412344
Show/Hide
|
C35H44ClFN4O7S
|
1
|
1 |
AC50 = 6230 nM
|
|
|
CP0335212
|
2-chloranyl-N-hexyl-N-phenyl-ethanamide
Show/Hide
|
C14H20ClNO
|
1
|
1 |
AC50 = 6260 nM
|
|
|
CP0883316
|
SID87218834
Show/Hide
|
C36H40ClN3O6S
|
1
|
1 |
AC50 = 6270 nM
|
|
|
CP0907787
|
SID131412290
Show/Hide
|
C36H49N3O9S2
|
1
|
1 |
AC50 = 6270 nM
|
|
|
CP0912880
|
SID87540361
Show/Hide
|
C36H45F4N3O6S
|
1
|
1 |
AC50 = 6280 nM
|
|
|
CP0874891
|
SID57262891
Show/Hide
|
C19H16N4O7S
|
1
|
1 |
AC50 = 6290 nM
|
|
|
CP0965811
|
SID87218863
Show/Hide
|
C37H43N3O6S
|
1
|
1 |
AC50 = 6290 nM
|
|
|
CP0908005
|
SID121284981
Show/Hide
|
C29H27N7O2
|
1
|
1 |
AC50 = 6310 nM
|
|
|
CP0851526
|
SID131426922
Show/Hide
|
C30H38FN3O5S
|
1
|
1 |
AC50 = 6320 nM
|
|
|
CP0941620
|
SID144192256
Show/Hide
|
C26H23F2N3O3
|
1
|
1 |
AC50 = 6320 nM
|
|
|
CP0908786
|
SID87544032
Show/Hide
|
C36H45Cl2FN4O5
|
1
|
1 |
AC50 = 6330 nM
|
|
|
CP0905180
|
SID87543124
Show/Hide
|
C37H47F3N4O5
|
1
|
1 |
AC50 = 6350 nM
|
|
|
CP0934880
|
SID87540528
Show/Hide
|
C32H35Cl2F3N4O4
|
1
|
1 |
AC50 = 6350 nM
|
|
|
CP0942510
|
SID87543594
Show/Hide
|
C34H41N3O4
|
1
|
1 |
AC50 = 6350 nM
|
|
|
CP0907783
|
SID131446486
Show/Hide
|
C24H22N2O3
|
1
|
1 |
AC50 = 6370 nM
|
|
|
CP0359466
|
1-(2,4-dimethylphenyl)-4-[4-(3-methoxyphenyl)-1-piperazinyl]pyrazolo[3,4-d]pyrimidine
Show/Hide
|
C24H26N6O
|
1
|
1 |
AC50 = 6380 nM
|
|
|
CP0940507
|
SID144190663
Show/Hide
|
C21H21FN2O
|
1
|
1 |
AC50 = 6380 nM
|
|
|
CP0947582
|
SID87543158
Show/Hide
|
C37H48F3N3O6S
|
1
|
1 |
AC50 = 6380 nM
|
|
|
CP0286631
|
MLS000392833
Show/Hide
|
C21H18N2O5S
|
1
|
1 |
AC50 = 6400 nM
|
|
|
CP0890230
|
SID131443542
Show/Hide
|
C28H30N2O7S
|
1
|
1 |
AC50 = 6400 nM
|
|
|
CP0919690
|
SID87541862
Show/Hide
|
C37H47F3N4O5
|
1
|
1 |
AC50 = 6400 nM
|
|
|
CP0637766
|
SID49667232
Show/Hide
|
C13H12N4O4
|
1
|
1 |
AC50 = 6410 nM
|
|
|
CP0810838
|
SID22411045
Show/Hide
|
C24H22ClF3N4O3S
|
1
|
1 |
AC50 = 6410 nM
|
|
|
CP0869058
|
SID49734422
Show/Hide
|
C16H17ClN4O4
|
1
|
1 |
AC50 = 6410 nM
|
|
|
CP0952400
|
SID144189669
Show/Hide
|
C32H37N3O4S
|
1
|
1 |
AC50 = 6410 nM
|
|
|
CP0966606
|
SID131410265
Show/Hide
|
C38H48F3N3O5
|
1
|
1 |
AC50 = 6420 nM
|
|
|
CP0875003
|
SID85813713
Show/Hide
|
C37H46F3N5O5
|
1
|
1 |
AC50 = 6430 nM
|
|
|
CP0959680
|
SID87543879
Show/Hide
|
C35H52ClN3O6S
|
1
|
1 |
AC50 = 6430 nM
|
|
|
CP0890226
|
SID92763672
Show/Hide
|
C41H53N5O3S2
|
1
|
1 |
AC50 = 6440 nM
|
|
|
CP0031043
|
N-quinolin-8-ylbenzenesulfonamide
Show/Hide
|
C15H12N2O2S
|
1
|
1 |
AC50 = 6460 nM
|
|
|
CP0856876
|
SID164339399
Show/Hide
|
C14H18N2OS
|
1
|
1 |
AC50 = 6460 nM
|
|
|
CP0881127
|
SID87218840
Show/Hide
|
C36H40FN3O6S
|
1
|
1 |
AC50 = 6470 nM
|
|
|
CP0940508
|
SID131411676
Show/Hide
|
C36H46F3N5O5
|
1
|
1 |
AC50 = 6480 nM
|
|
|
CP0406470
|
MLS003107001
Show/Hide
|
C23H32O5
|
1
|
1 |
AC50 = 6490 nM
|
|
|
CP0431715
|
5-bromanyl-1-[[4-methylidene-5-oxidanylidene-2-(4-phenylphenyl)oxolan-2-yl]methyl]pyrimidine-2,4-dione
Show/Hide
|
C22H17BrN2O4
|
1
|
1 |
AC50 = 6490 nM
|
|
|
CP0930591
|
SID131426930
Show/Hide
|
C29H38N2O7S2
|
1
|
1 |
AC50 = 6490 nM
|
|
|
CP0936522
|
SID144190379
Show/Hide
|
C33H33FN4O6
|
1
|
1 |
AC50 = 6510 nM
|
|
|
CP0862952
|
SID144198634
Show/Hide
|
C34H44ClN3O8S2
|
1
|
1 |
AC50 = 6520 nM
|
|
|
CP0891494
|
SID104170668
Show/Hide
|
C36H44F4N4O7S
|
1
|
1 |
AC50 = 6530 nM
|
|
|
CP0959676
|
SID104170442
Show/Hide
|
C36H52FN5O6
|
1
|
1 |
AC50 = 6550 nM
|
|
|
CP0771297
|
SID17387367
Show/Hide
|
C25H28N8O3
|
1
|
1 |
AC50 = 6570 nM
|
|
|
CP0856719
|
SID49825053
Show/Hide
|
C20H23ClN4O2S
|
1
|
1 |
AC50 = 6570 nM
|
|
|
CP0891360
|
SID87541097
Show/Hide
|
C34H44F6N4O6
|
1
|
1 |
AC50 = 6570 nM
|
|
|
CP0926612
|
SID87541102
Show/Hide
|
C37H46F3N3O5
|
1
|
1 |
AC50 = 6570 nM
|
|
|
CP0950343
|
SID131411335
Show/Hide
|
C37H45F3N4O6
|
1
|
1 |
AC50 = 6570 nM
|
|
|
CP0860342
|
SID85804240
Show/Hide
|
C33H45N3O8S3
|
1
|
1 |
AC50 = 6600 nM
|
|
|
CP0910442
|
SID131412028
Show/Hide
|
C36H45F3N4O7S
|
1
|
1 |
AC50 = 6600 nM
|
|
|
CP0848113
|
SID131413863
Show/Hide
|
C32H38N2O5S
|
1
|
1 |
AC50 = 6610 nM
|
|
|
CP0851432
|
SID49819758
Show/Hide
|
C20H24N4O2S
|
1
|
1 |
AC50 = 6610 nM
|
|
|
CP0966629
|
SID131460370
Show/Hide
|
C25H22FN3O3S
|
1
|
1 |
AC50 = 6610 nM
|
|
|
CP0909794
|
SID104170687
Show/Hide
|
C36H45ClF3N3O6S
|
1
|
1 |
AC50 = 6620 nM
|
|
|
CP0926405
|
SID87543392
Show/Hide
|
C34H43F3N4O7S2
|
1
|
1 |
AC50 = 6630 nM
|
|
|
CP0314996
|
4-[[2-(4,5-dichloro-6-keto-pyridazin-1-yl)acetyl]amino]benzoic acid ethyl ester
Show/Hide
|
C15H13Cl2N3O4
|
1
|
1 |
AC50 = 6640 nM
|
|
|
CP0007375
|
4-chloranyl-1-methyl-3-nitro-quinolin-2-one
Show/Hide
|
C10H7ClN2O3
|
1
|
1 |
AC50 = 6650 nM
|
|
|
CP0920058
|
SID144194946
Show/Hide
|
C26H30N2O2
|
1
|
1 |
AC50 = 6670 nM
|
|
|
CP0259647
|
3-butyl-8-[(4,5-dichloro-6-keto-pyridazin-1-yl)methyl]-7-propyl-xanthine
Show/Hide
|
C17H20Cl2N6O3
|
1
|
1 |
AC50 = 6680 nM
|
|
|
CP0873860
|
SID99495631
Show/Hide
|
C24H32F3N3O9S
|
1
|
1 |
AC50 = 6680 nM
|
|
|
CP0337980
|
2-[(E)-2-(4-methoxyphenyl)ethenyl]-1-methyl-benzimidazole
Show/Hide
|
C17H16N2O
|
1
|
1 |
AC50 = 6690 nM
|
|
|
CP0918116
|
SID131412106
Show/Hide
|
C36H45F3N4O7S
|
1
|
1 |
AC50 = 6700 nM
|
|
|
CP0961308
|
SID87539807
Show/Hide
|
C35H46ClN3O8S2
|
1
|
1 |
AC50 = 6700 nM
|
|
|
CP0024809
|
MLS001111235
Show/Hide
|
C14H11F3N6O
|
1
|
1 |
AC50 = 6710 nM
|
|
|
CP0942502
|
SID131410525
Show/Hide
|
C36H45F4N3O6S
|
1
|
1 |
AC50 = 6710 nM
|
|
|
CP0391455
|
4,5-bis(chloranyl)-6-methoxy-2-phenyl-pyridazin-3-one
Show/Hide
|
C11H8Cl2N2O2
|
1
|
1 |
AC50 = 6720 nM
|
|
|
CP0910493
|
SID99358653
Show/Hide
|
C32H38N2O5S
|
1
|
1 |
AC50 = 6730 nM
|
|
|
CP0856717
|
SID87540499
Show/Hide
|
C37H46F4N4O5
|
1
|
1 |
AC50 = 6740 nM
|
|
|
CP0891496
|
SID87542786
Show/Hide
|
C37H45Cl2F3N4O5
|
1
|
1 |
AC50 = 6740 nM
|
|
|
CP0910495
|
SID131461375
Show/Hide
|
C27H34N2O3
|
1
|
1 |
AC50 = 6750 nM
|
|
|
CP0884745
|
N-(((2S,8R,9R)-14-(dimethylamino)-11-((S)-1-hydroxypropan-2-yl)-2,9-dimethyl-12-oxo-2,3,4,5,6,8,9,10,11,12-decahydrobenzo[b][1,9,5]dioxaazacyclotetradecin-8-yl)methyl)-4-fluoro-N-methylbenzenesulfonamide
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C30H44FN3O6S
|
1
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1 |
AC50 = 6760 nM
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CP0908026
|
SID131412851
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C35H44Cl3N3O6S
|
1
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1 |
AC50 = 6760 nM
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CP0188721
|
3-[[5-(2,4-dimethoxyphenyl)-6H-1,3,4-thiadiazin-2-yl]amino]-N,N,4-trimethyl-benzenesulfonamide
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C20H24N4O4S2
|
1
|
1 |
AC50 = 6770 nM
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CP0873947
|
SID17508981
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C15H18ClN3O
|
1
|
1 |
AC50 = 6770 nM
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CP0885640
|
SID85801925
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C32H38F3N3O6S
|
1
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1 |
AC50 = 6770 nM
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CP0886259
|
SID121286618
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C11H18N6O
|
1
|
1 |
AC50 = 6780 nM
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CP0959678
|
SID144194439
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C33H36F3N3O5S
|
1
|
1 |
AC50 = 6800 nM
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CP0398258
|
1-benzyl-6-(2-hydroxy-5-methoxy-benzoyl)-3-methyl-pyrido[2,3-d]pyrimidine-2,4-quinone
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|
C23H19N3O5
|
1
|
1 |
AC50 = 6810 nM
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CP0873494
|
SID49644456
Show/Hide
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C17H21N3O
|
1
|
1 |
AC50 = 6820 nM
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CP0882535
|
SID131412457
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C36H45ClF3N3O6S
|
1
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1 |
AC50 = 6820 nM
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CP0959681
|
SID87540553
Show/Hide
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C36H45F4N3O6S
|
1
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1 |
AC50 = 6820 nM
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CP0882033
|
SID131411823
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C37H48F3N3O7S
|
1
|
1 |
AC50 = 6830 nM
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CP0907190
|
SID104170606
Show/Hide
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C34H43ClFN3O8S2
|
1
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1 |
AC50 = 6830 nM
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CP0398868
|
MLS000086269
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C17H15F3N4O4S2
|
1
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1 |
AC50 = 6850 nM
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CP0852373
|
SID104170647
Show/Hide
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C37H53F3N4O5
|
1
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1 |
AC50 = 6850 nM
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CP0851525
|
SID85813808
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C38H48F3N5O5
|
1
|
1 |
AC50 = 6870 nM
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CP0907822
|
SID131461603
Show/Hide
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C25H25FN2O4S
|
1
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1 |
AC50 = 6870 nM
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CP0908716
|
SID131434101
Show/Hide
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C33H39N3O6S
|
1
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1 |
AC50 = 6870 nM
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CP0949672
|
SID131412378
Show/Hide
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C36H46F3N3O6S
|
1
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1 |
AC50 = 6880 nM
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CP0909155
|
SID131414993
Show/Hide
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C31H31FN2O7S
|
1
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1 |
AC50 = 6890 nM
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CP0202384
|
4-methyl-N-[4-[4-(4-nitrophenyl)piperazine-1-carbonyl]benzyl]benzenesulfonamide
Show/Hide
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C25H26N4O5S
|
1
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1 |
AC50 = 6910 nM
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CP0879604
|
SID92764824
Show/Hide
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C23H29ClN4O
|
1
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1 |
AC50 = 6910 nM
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CP0891771
|
SID121284986
Show/Hide
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C28H29N7O2
|
1
|
1 |
AC50 = 6910 nM
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CP0902480
|
SID131461003
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C28H27FN2O4S
|
1
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1 |
AC50 = 6920 nM
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CP0404623
|
1-[3,5-bis(2,2,2-trifluoroethoxy)phenyl]-3-phenyl-urea
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C17H14F6N2O3
|
1
|
1 |
AC50 = 6930 nM
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CP0845627
|
SID24793712
Show/Hide
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C19H15NO2
|
1
|
1 |
AC50 = 6930 nM
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CP0912661
|
SID87539863
Show/Hide
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C36H45F3N4O7S
|
1
|
1 |
AC50 = 6960 nM
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CP0728243
|
SID26659333
Show/Hide
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C16H17NO4S
|
1
|
1 |
AC50 = 6970 nM
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CP0898646
|
SID14731796
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C20H16N2O3S
|
1
|
1 |
AC50 = 6980 nM
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CP0926629
|
SID131412854
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C35H44Cl3N3O6S
|
1
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1 |
AC50 = 7000 nM
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CP0879751
|
SID49671892
Show/Hide
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C13H15NO3S2
|
1
|
1 |
AC50 = 7010 nM
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CP0881126
|
SID92764784
Show/Hide
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C18H22BrClN2O6
|
1
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1 |
AC50 = 7030 nM
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CP0950340
|
SID131412708
Show/Hide
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C37H48F3N3O6S
|
1
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1 |
AC50 = 7030 nM
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CP0224076
|
1-N-benzo[g]quinolin-4-yl-4-N-propan-2-ylbenzene-1,4-diamine
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C22H21N3
|
1
|
1 |
AC50 = 7040 nM
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CP0413323
|
3-(benzenesulfonyl)-N-[3-(dimethylamino)propyl]-N-(4-methoxy-1,3-benzothiazol-2-yl)propanamide
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C22H27N3O4S2
|
1
|
1 |
AC50 = 7040 nM
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CP0879939
|
SID85806166
Show/Hide
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C31H35F3N4O7S
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1
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1 |
AC50 = 7040 nM
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CP0942892
|
SID85807373
Show/Hide
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C31H35Cl2FN4O4
|
1
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1 |
AC50 = 7040 nM
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CP0046604
|
2-hydroxy-N-[4-(2,2,3,3-tetrafluoropropoxy)-3-(trifluoromethyl)phenyl]benzamide
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C17H12F7NO3
|
1
|
1 |
AC50 = 7060 nM
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CP0846123
|
SID49669711
Show/Hide
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C22H28ClN3O4S
|
1
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1 |
AC50 = 7060 nM
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CP0068943
|
4-(2-pyridinylsulfanyl)-1-(trifluoromethyl)[1,2,4]triazolo[4,3-a]quinoxaline
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C15H8F3N5S
|
1
|
1 |
AC50 = 7080 nM
|
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CP0966635
|
SID131412382
Show/Hide
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C36H46F3N3O6S
|
1
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1 |
AC50 = 7080 nM
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CP0846812
|
SID87539915
Show/Hide
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C35H44F2N4O7S
|
1
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1 |
AC50 = 7090 nM
|
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CP0862109
|
SID87542251
Show/Hide
|
C37H48F3N3O7S
|
1
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1 |
AC50 = 7090 nM
|
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CP0434618
|
2-benzylsulfonyl-5-chloro-N-(2-ethoxyphenyl)pyrimidine-4-carboxamide
Show/Hide
|
C20H18ClN3O4S
|
1
|
1 |
AC50 = 7100 nM
|
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CP0864555
|
SID87543088
Show/Hide
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C38H47F3N4O7
|
1
|
1 |
AC50 = 7110 nM
|
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CP0939545
|
SID85200863
Show/Hide
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C38H54O13
|
1
|
1 |
AC50 = 7140 nM
|
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CP0966599
|
SID131462224
Show/Hide
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C30H30FN3O2
|
1
|
1 |
AC50 = 7150 nM
|
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CP0910499
|
SID85804695
Show/Hide
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C38H48F3N3O5
|
1
|
1 |
AC50 = 7160 nM
|
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CP0799820
|
SID24816334
Show/Hide
|
C21H25ClFN3O2S
|
1
|
1 |
AC50 = 7170 nM
|
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CP0813403
|
SID104219453
Show/Hide
|
C14H10ClNO4
|
1
|
1 |
AC50 = 7170 nM
|
|
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CP0283084
|
2-[2-(2-chlorophenyl)-2-keto-ethyl]-1,1-diketo-1,2-benzothiazol-3-one
Show/Hide
|
C15H10ClNO4S
|
1
|
1 |
AC50 = 7180 nM
|
|
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CP0942469
|
SID85805577
Show/Hide
|
C36H46ClN3O7S
|
1
|
1 |
AC50 = 7180 nM
|
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CP0944759
|
SID131462790
Show/Hide
|
C26H32N2O4S
|
1
|
1 |
AC50 = 7180 nM
|
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CP0864564
|
SID85269712
Show/Hide
|
C20H17F2N3O3S2
|
1
|
1 |
AC50 = 7190 nM
|
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CP0919689
|
SID87540423
Show/Hide
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C34H44F3N3O6S2
|
1
|
1 |
AC50 = 7200 nM
|
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CP0938691
|
SID144198206
Show/Hide
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C30H29F3N4O4
|
1
|
1 |
AC50 = 7200 nM
|
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CP0891698
|
SID131412383
Show/Hide
|
C36H46F3N3O6S
|
1
|
1 |
AC50 = 7210 nM
|
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CP0912514
|
SID131461765
Show/Hide
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C27H30N2O5S
|
1
|
1 |
AC50 = 7210 nM
|
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CP0864582
|
SID131410263
Show/Hide
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C38H48F3N3O5
|
1
|
1 |
AC50 = 7220 nM
|
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CP0885546
|
SID131410266
Show/Hide
|
C38H48F3N3O5
|
1
|
1 |
AC50 = 7230 nM
|
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CP0210430
|
3-(7-Chloro-4-nitro-benzo[1,2,5]oxadiazol-5-ylamino)-phenol
Show/Hide
|
C12H7ClN4O4
|
1
|
1 |
AC50 = 7240 nM
|
|
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CP0905584
|
SID26731845
Show/Hide
|
C21H10Cl2N4O4S
|
1
|
1 |
AC50 = 7240 nM
|
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CP0907801
|
SID131442201
Show/Hide
|
C31H30F3N3O5
|
1
|
1 |
AC50 = 7260 nM
|
|
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CP0897523
|
SID87543296
Show/Hide
|
C35H46ClN3O8S2
|
1
|
1 |
AC50 = 7270 nM
|
|
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CP0906892
|
MMV568655
Show/Hide
|
C25H25N3O
|
1
|
1 |
AC50 = 7270 nM
|
|
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CP0936521
|
SID87541959
Show/Hide
|
C36H46F3N5O5
|
1
|
1 |
AC50 = 7300 nM
|
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CP0395730
|
1-[5-(2-Ethylsulfanyl-ethyl)-[1,3,4]thiadiazol-2-yl]-3-(3-trifluoromethyl-phenyl)-urea
Show/Hide
|
C14H15F3N4OS2
|
1
|
1 |
AC50 = 7310 nM
|
|
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CP0874953
|
SID85805095
Show/Hide
|
C35H46FN3O6S
|
1
|
1 |
AC50 = 7310 nM
|
|
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CP0907815
|
SID131444801
Show/Hide
|
C33H31FN2O6S
|
1
|
1 |
AC50 = 7310 nM
|
|
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CP0942500
|
SID131412458
Show/Hide
|
C36H45ClF3N3O6S
|
1
|
1 |
AC50 = 7310 nM
|
|
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CP0949670
|
SID131447059
Show/Hide
|
C24H21N3O3
|
1
|
1 |
AC50 = 7310 nM
|
|
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CP0899484
|
SID104170407
Show/Hide
|
C37H47F3N4O8S
|
1
|
1 |
AC50 = 7320 nM
|
|
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CP0912879
|
SID131442894
Show/Hide
|
C33H31FN2O7S
|
1
|
1 |
AC50 = 7320 nM
|
|
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CP0765183
|
SID49716863
Show/Hide
|
C23H27ClN6OS
|
1
|
1 |
AC50 = 7330 nM
|
|
|
CP0891782
|
SID131409545
Show/Hide
|
C32H37F3N4O6S
|
1
|
1 |
AC50 = 7340 nM
|
|
|
CP0411342
|
MLS002607898
Show/Hide
|
C12H10N2O4S
|
1
|
1 |
AC50 = 7360 nM
|
|
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CP0891820
|
SID103075184
Show/Hide
|
C33H36N6O5
|
1
|
1 |
AC50 = 7360 nM
|
|
|
CP0950778
|
SID131412456
Show/Hide
|
C36H45ClF3N3O6S
|
1
|
1 |
AC50 = 7370 nM
|
|
|
CP0912884
|
SID131412500
Show/Hide
|
C34H44ClN3O8S2
|
1
|
1 |
AC50 = 7400 nM
|
|
|
CP0918113
|
SID121283022
Show/Hide
|
C17H16N4
|
1
|
1 |
AC50 = 7400 nM
|
|
|
CP0942411
|
SID87541152
Show/Hide
|
C35H46F3N5O8S
|
1
|
1 |
AC50 = 7410 nM
|
|
|
CP0908718
|
SID104170415
Show/Hide
|
C36H46Cl2N4O5
|
1
|
1 |
AC50 = 7420 nM
|
|
|
CP0817264
|
SID47198474
Show/Hide
|
C15H15N3O3
|
1
|
1 |
AC50 = 7430 nM
|
|
|
CP0909444
|
SID131411672
Show/Hide
|
C36H46F3N5O5
|
1
|
1 |
AC50 = 7430 nM
|
|
|
CP0910489
|
SID87218869
Show/Hide
|
C36H40ClN3O6S
|
1
|
1 |
AC50 = 7430 nM
|
|
|
CP0868107
|
SID92764559
Show/Hide
|
C30H24N2O2
|
1
|
1 |
AC50 = 7450 nM
|
|
|
CP0882467
|
SID131409359
Show/Hide
|
C41H46N4O5
|
1
|
1 |
AC50 = 7450 nM
|
|
|
CP0889241
|
SID131464506
Show/Hide
|
C29H34N2O3S
|
1
|
1 |
AC50 = 7450 nM
|
|
|
CP0907571
|
SID87540974
Show/Hide
|
C33H44Cl2F3N3O5
|
1
|
1 |
AC50 = 7470 nM
|
|
|
CP0940512
|
SID131412014
Show/Hide
|
C37H46F3N3O5
|
1
|
1 |
AC50 = 7470 nM
|
|
|
CP0881655
|
SID85804669
Show/Hide
|
C37H48F3N3O6S
|
1
|
1 |
AC50 = 7480 nM
|
|
|
CP0884587
|
SID104170417
Show/Hide
|
C36H45F4N3O6S
|
1
|
1 |
AC50 = 7500 nM
|
|
|
CP0918065
|
SID87543727
Show/Hide
|
C29H32Cl3N3O5S
|
1
|
1 |
AC50 = 7500 nM
|
|
|
CP0283529
|
4-Methoxy-benzoic acid N'-(pyridine-2-carbonyl)-hydrazide
Show/Hide
|
C14H13N3O3
|
1
|
1 |
AC50 = 7510 nM
|
|
|
CP0872445
|
SID131413378
Show/Hide
|
C30H35N3O5S
|
1
|
1 |
AC50 = 7510 nM
|
|
|
CP0225784
|
7-chloranyl-3-phenyl-[1,3]thiazolo[4,5-d]pyrimidine-2-thione
Show/Hide
|
C11H6ClN3S2
|
1
|
1 |
AC50 = 7520 nM
|
|
|
CP0201064
|
2-({7-[(1-methyl-1H-imidazol-2-yl)thio]-4-nitro-2,1,3-benzoxadiazol-5-yl}amino)ethyl propionate
Show/Hide
|
C15H16N6O5S
|
1
|
1 |
AC50 = 7530 nM
|
|
|
CP0935307
|
SID121284971
Show/Hide
|
C29H31N7O2
|
1
|
1 |
AC50 = 7540 nM
|
|
|
CP0943283
|
SID131460344
Show/Hide
|
C27H27N3O3S
|
1
|
1 |
AC50 = 7550 nM
|
|
|
CP0790084
|
SID164339407
Show/Hide
|
C19H16BrN3O2S2
|
1
|
1 |
AC50 = 7560 nM
|
|
|
CP0885594
|
SID49722282
Show/Hide
|
C21H23N3O4S3
|
1
|
1 |
AC50 = 7560 nM
|
|
|
CP0900330
|
SID85805158
Show/Hide
|
C35H51ClN4O7S
|
1
|
1 |
AC50 = 7570 nM
|
|
|
CP0884721
|
SID49677812
Show/Hide
|
C18H14N2O2S
|
1
|
1 |
AC50 = 7580 nM
|
|
|
CP0907785
|
SID131414347
Show/Hide
|
C30H40N2O7S2
|
1
|
1 |
AC50 = 7590 nM
|
|
|
CP0826797
|
SID26732536
Show/Hide
|
C33H49N5O8
|
1
|
1 |
AC50 = 7600 nM
|
|
|
CP0952398
|
SID87541096
Show/Hide
|
C38H48F3N3O5
|
1
|
1 |
AC50 = 7600 nM
|
|
|
CP0868091
|
SID87539821
Show/Hide
|
C34H44F3N3O6S2
|
1
|
1 |
AC50 = 7620 nM
|
|
|
CP0176463
|
2-[[5-(2-bromophenyl)-1,3,4-oxadiazol-2-yl]methyl]-4,5-bis(chloranyl)pyridazin-3-one
Show/Hide
|
C13H7BrCl2N4O2
|
1
|
1 |
AC50 = 7630 nM
|
|
|
CP0844329
|
SID164339404
Show/Hide
|
C19H20BrNO3S
|
1
|
1 |
AC50 = 7630 nM
|
|
|
CP0874970
|
SID87543292
Show/Hide
|
C38H47F3N4O7
|
1
|
1 |
AC50 = 7630 nM
|
|
|
CP0897501
|
SID103050603
Show/Hide
|
C24H26N2O3S2
|
1
|
1 |
AC50 = 7650 nM
|
|
|
CP0900340
|
SID131413160
Show/Hide
|
C34H43ClFN3O8S2
|
1
|
1 |
AC50 = 7670 nM
|
|
|
CP0865132
|
SID131411824
Show/Hide
|
C37H48F3N3O7S
|
1
|
1 |
AC50 = 7680 nM
|
|
|
CP0966608
|
SID87543395
Show/Hide
|
C35H46ClN3O9S2
|
1
|
1 |
AC50 = 7700 nM
|
|
|
CP0143940
|
5-chloranyl-N-(2-ethoxyphenyl)-2-[(3-methylphenyl)methylsulfonyl]pyrimidine-4-carboxamide
Show/Hide
|
C21H20ClN3O4S
|
1
|
1 |
AC50 = 7710 nM
|
|
|
CP0907198
|
SID131410530
Show/Hide
|
C36H45F4N3O6S
|
1
|
1 |
AC50 = 7710 nM
|
|
|
CP0865133
|
SID144190859
Show/Hide
|
C32H35FN4O5S
|
1
|
1 |
AC50 = 7720 nM
|
|
|
CP0891359
|
SID56315011
Show/Hide
|
C23H28F2N4O4S
|
1
|
1 |
AC50 = 7720 nM
|
|
|
CP0885876
|
SID131410272
Show/Hide
|
C34H43F3N4O7S2
|
1
|
1 |
AC50 = 7750 nM
|
|
|
CP0890127
|
SID99357067
Show/Hide
|
C37H34F6N6O5
|
1
|
1 |
AC50 = 7760 nM
|
|
|
CP0940977
|
SID85805102
Show/Hide
|
C34H48N4O10S2
|
1
|
1 |
AC50 = 7760 nM
|
|
|
CP0881168
|
SID85795175
Show/Hide
|
C30H42ClN3O5S
|
1
|
1 |
AC50 = 7770 nM
|
|
|
CP0125189
|
5-chloranyl-2-methylsulfonyl-N-naphthalen-2-yl-pyrimidine-4-carboxamide
Show/Hide
|
C16H12ClN3O3S
|
1
|
1 |
AC50 = 7810 nM
|
|
|
CP0137403
|
4-bromanyl-2-[(E)-3-(2,5-dimethoxyphenyl)prop-2-enoyl]-7-(methylamino)cyclohepta-2,4,6-trien-1-one
Show/Hide
|
C19H18BrNO4
|
1
|
1 |
AC50 = 7830 nM
|
|
|
CP0217180
|
2,2-Di-m-tolyl-cyclopropanecarboxylic acid (2-hydroxy-4-nitro-phenyl)-amide
Show/Hide
|
C24H22N2O4
|
1
|
1 |
AC50 = 7830 nM
|
|
|
CP0862094
|
SID131426923
Show/Hide
|
C30H38FN3O5S
|
1
|
1 |
AC50 = 7830 nM
|
|
|
CP0883287
|
SID131409570
Show/Hide
|
C33H37F3N4O6
|
1
|
1 |
AC50 = 7850 nM
|
|
|
CP0885653
|
SID131443062
Show/Hide
|
C29H27ClF3N3O5
|
1
|
1 |
AC50 = 7850 nM
|
|
|
CP0883681
|
SID49673940
Show/Hide
|
C19H19N3O4S
|
1
|
1 |
AC50 = 7880 nM
|
|
|
CP0875015
|
SID131452382
Show/Hide
|
C29H34ClN3O5
|
1
|
1 |
AC50 = 7900 nM
|
|
|
CP0862113
|
SID131412395
Show/Hide
|
C36H47Cl2N3O6S
|
1
|
1 |
AC50 = 7920 nM
|
|
|
CP0908584
|
SID87540161
Show/Hide
|
C32H42ClN3O8S3
|
1
|
1 |
AC50 = 7930 nM
|
|
|
CP0965790
|
SID131426920
Show/Hide
|
C30H38FN3O5S
|
1
|
1 |
AC50 = 7930 nM
|
|
|
CP0882353
|
SID87543603
Show/Hide
|
C38H48F3N3O5
|
1
|
1 |
AC50 = 7940 nM
|
|
|
CP0952408
|
SID131411592
Show/Hide
|
C35H45Cl2N3O6S
|
1
|
1 |
AC50 = 7950 nM
|
|
|
CP0868349
|
SID131462665
Show/Hide
|
C30H32FN3O2
|
1
|
1 |
AC50 = 7960 nM
|
|
|
CP0912231
|
SID144190623
Show/Hide
|
C28H32N4O3
|
1
|
1 |
AC50 = 7960 nM
|
|
|
CP0862111
|
SID131426788
Show/Hide
|
C30H34F3N3O5S
|
1
|
1 |
AC50 = 8000 nM
|
|
|
CP0862107
|
SID87542876
Show/Hide
|
C37H52F3N5O6
|
1
|
1 |
AC50 = 8030 nM
|
|
|
CP0940735
|
SID104170642
Show/Hide
|
C35H47N3O8S2
|
1
|
1 |
AC50 = 8050 nM
|
|
|
CP0966627
|
SID131410686
Show/Hide
|
C38H47F3N4O6
|
1
|
1 |
AC50 = 8050 nM
|
|
|
CP0942586
|
SID87550752
Show/Hide
|
C22H28N2O7S
|
1
|
1 |
AC50 = 8070 nM
|
|
|
CP0857855
|
SID22401637
Show/Hide
|
C19H18F6N2O4
|
1
|
1 |
AC50 = 8080 nM
|
|
|
CP0886578
|
SID131426926
Show/Hide
|
C30H38FN3O5S
|
1
|
1 |
AC50 = 8090 nM
|
|
|
CP0890233
|
SID131411632
Show/Hide
|
C37H45F4N5O6
|
1
|
1 |
AC50 = 8090 nM
|
|
|
CP0946013
|
SID131447010
Show/Hide
|
C25H26N2O3S
|
1
|
1 |
AC50 = 8090 nM
|
|
|
CP0897058
|
SID85805118
Show/Hide
|
C36H51FN4O6
|
1
|
1 |
AC50 = 8100 nM
|
|
|
CP0908032
|
SID87541865
Show/Hide
|
C36H45Cl2FN4O5
|
1
|
1 |
AC50 = 8100 nM
|
|
|
CP0856720
|
SID131464869
Show/Hide
|
C29H34N2O3S
|
1
|
1 |
AC50 = 8110 nM
|
|
|
CP0868093
|
SID131413095
Show/Hide
|
C38H49F3N4O6
|
1
|
1 |
AC50 = 8110 nM
|
|
|
CP0934879
|
SID85800397
Show/Hide
|
C34H48F3N5O6
|
1
|
1 |
AC50 = 8110 nM
|
|
|
CP0936520
|
SID144192113
Show/Hide
|
C28H25FN2O4S
|
1
|
1 |
AC50 = 8120 nM
|
|
|
CP0966602
|
SID87543884
Show/Hide
|
C35H46FN3O8S2
|
1
|
1 |
AC50 = 8120 nM
|
|
|
CP0881165
|
SID87541143
Show/Hide
|
C35H46ClN3O8S2
|
1
|
1 |
AC50 = 8130 nM
|
|
|
CP0907804
|
SID85270718
Show/Hide
|
C20H27N5O7S
|
1
|
1 |
AC50 = 8140 nM
|
|
|
CP0864532
|
SID49819753
Show/Hide
|
C25H27ClN6O2S
|
1
|
1 |
AC50 = 8150 nM
|
|
|
CP0846751
|
SID49719633
Show/Hide
|
C17H14ClN3O3S2
|
1
|
1 |
AC50 = 8170 nM
|
|
|
CP0881648
|
SID164339398
Show/Hide
|
C21H19BrN2O3S2
|
1
|
1 |
AC50 = 8170 nM
|
|
|
CP0168755
|
2-(benzenesulfonyl)-6-methoxy-3-nitropyridine
Show/Hide
|
C12H10N2O5S
|
1
|
1 |
AC50 = 8180 nM
|
|
|
CP0395813
|
Chloro-acetic acid N'-(2-hydroxy-2,2-diphenyl-acetyl)-N-p-tolyl-hydrazide
Show/Hide
|
C23H21ClN2O3
|
1
|
1 |
AC50 = 8180 nM
|
|
|
CP0944040
|
SID87542353
Show/Hide
|
C38H49F3N4O6
|
1
|
1 |
AC50 = 8180 nM
|
|
|
CP0137296
|
3,3-bis(2-methyl-4-oxidanyl-5-propan-2-yl-phenyl)-2-benzofuran-1-one
Show/Hide
|
C28H30O4
|
1
|
1 |
AC50 = 8190 nM
|
|
|
CP0908004
|
SID87543488
Show/Hide
|
C35H47F3N4O7S
|
1
|
1 |
AC50 = 8190 nM
|
|
|
CP0966597
|
SID131412118
Show/Hide
|
C35H44Cl2FN3O6S
|
1
|
1 |
AC50 = 8200 nM
|
|
|
CP0862105
|
SID131412252
Show/Hide
|
C37H46F4N4O5
|
1
|
1 |
AC50 = 8210 nM
|
|
|
CP0948172
|
SID87540667
Show/Hide
|
C36H51FN4O6
|
1
|
1 |
AC50 = 8220 nM
|
|
|
CP0862102
|
SID131464505
Show/Hide
|
C29H34N2O3S
|
1
|
1 |
AC50 = 8230 nM
|
|
|
CP0905586
|
SID131412012
Show/Hide
|
C37H46F3N3O5
|
1
|
1 |
AC50 = 8240 nM
|
|
|
CP0196311
|
4,5-bis(bromanyl)-2-phenyl-pyridazin-3-one
Show/Hide
|
C10H6Br2N2O
|
1
|
1 |
AC50 = 8260 nM
|
|
|
CP0865903
|
SID49671543
Show/Hide
|
C15H12N2O2S
|
1
|
1 |
AC50 = 8260 nM
|
|
|
CP0912913
|
SID131460784
Show/Hide
|
C28H27FN2O3S
|
1
|
1 |
AC50 = 8270 nM
|
|
|
CP0950777
|
SID87540749
Show/Hide
|
C34H43ClFN3O8S2
|
1
|
1 |
AC50 = 8270 nM
|
|
|
CP0957467
|
SID131456925
Show/Hide
|
C29H31ClN2O6S
|
1
|
1 |
AC50 = 8280 nM
|
|
|
CP0941618
|
SID87543537
Show/Hide
|
C36H45ClF3N3O6S
|
1
|
1 |
AC50 = 8290 nM
|
|
|
CP0908892
|
SID131442889
Show/Hide
|
C33H31FN2O7S
|
1
|
1 |
AC50 = 8320 nM
|
|
|
CP0942509
|
SID131456922
Show/Hide
|
C29H31ClN2O6S
|
1
|
1 |
AC50 = 8330 nM
|
|
|
CP0944788
|
SID131426743
Show/Hide
|
C28H37N3O4S
|
1
|
1 |
AC50 = 8330 nM
|
|
|
CP0442706
|
2-(4-methylphenyl)sulfonyl-3-nitro-pyridine
Show/Hide
|
C12H10N2O4S
|
1
|
1 |
AC50 = 8340 nM
|
|
|
CP0908691
|
SID87543410
Show/Hide
|
C38H47F3N4O7
|
1
|
1 |
AC50 = 8350 nM
|
|
|
CP0890217
|
SID22403644
Show/Hide
|
C26H21NO3S2
|
1
|
1 |
AC50 = 8360 nM
|
|
|
CP0866399
|
SID87542749
Show/Hide
|
C38H49F3N4O6
|
1
|
1 |
AC50 = 8380 nM
|
|
|
CP0930584
|
SID131414294
Show/Hide
|
C30H38FN3O5S
|
1
|
1 |
AC50 = 8380 nM
|
|
|
CP0900397
|
SID131410609
Show/Hide
|
C37H53F3N4O5
|
1
|
1 |
AC50 = 8390 nM
|
|
|
CP0930555
|
SID144194245
Show/Hide
|
C26H21N3O3
|
1
|
1 |
AC50 = 8390 nM
|
|
|
CP0948166
|
SID85797649
Show/Hide
|
C32H42F3N5O5
|
1
|
1 |
AC50 = 8400 nM
|
|
|
CP0944037
|
SID104170846
Show/Hide
|
C36H46F3N5O5
|
1
|
1 |
AC50 = 8410 nM
|
|
|
CP0885767
|
SID87541352
Show/Hide
|
C36H46Cl2N4O5
|
1
|
1 |
AC50 = 8420 nM
|
|
|
CP0907920
|
SID131426924
Show/Hide
|
C30H38FN3O5S
|
1
|
1 |
AC50 = 8430 nM
|
|
|
CP0864529
|
SID87540841
Show/Hide
|
C37H47F3N4O5
|
1
|
1 |
AC50 = 8440 nM
|
|
|
CP0935267
|
SID131412704
Show/Hide
|
C37H48F3N3O6S
|
1
|
1 |
AC50 = 8450 nM
|
|
|
CP0932672
|
SID87543042
Show/Hide
|
C36H45ClF3N3O6S
|
1
|
1 |
AC50 = 8480 nM
|
|
|
CP0943349
|
SID131461605
Show/Hide
|
C25H25FN2O4S
|
1
|
1 |
AC50 = 8480 nM
|
|
|
CP0865130
|
SID131411839
Show/Hide
|
C35H50ClN3O7S
|
1
|
1 |
AC50 = 8510 nM
|
|
|
CP0912886
|
SID49716858
Show/Hide
|
C20H23BrN6OS
|
1
|
1 |
AC50 = 8510 nM
|
|
|
CP0908035
|
SID144191371
Show/Hide
|
C25H22F3N3O
|
1
|
1 |
AC50 = 8550 nM
|
|
|
CP0881155
|
SID131411248
Show/Hide
|
C38H47F3N4O7
|
1
|
1 |
AC50 = 8560 nM
|
|
|
CP0881125
|
SID131410527
Show/Hide
|
C36H45F4N3O6S
|
1
|
1 |
AC50 = 8570 nM
|
|
|
CP0864580
|
SID131446805
Show/Hide
|
C27H28N2O3
|
1
|
1 |
AC50 = 8610 nM
|
|
|
CP0888888
|
SID87540146
Show/Hide
|
C34H40F3N3O4
|
1
|
1 |
AC50 = 8610 nM
|
|
|
CP0863890
|
SID49727002
Show/Hide
|
C21H26N2O5S2
|
1
|
1 |
AC50 = 8620 nM
|
|
|
CP0935173
|
SID144191370
Show/Hide
|
C25H22F3N3O
|
1
|
1 |
AC50 = 8620 nM
|
|
|
CP0949414
|
SID104170839
Show/Hide
|
C35H44F2N4O7S
|
1
|
1 |
AC50 = 8620 nM
|
|
|
CP0909622
|
SID87540116
Show/Hide
|
C34H43F3N4O7S2
|
1
|
1 |
AC50 = 8640 nM
|
|
|
CP0438709
|
1-(4-chlorobenzyl)-4-(4-phenylpiperazino)pyrazolo[3,4-d]pyrimidine
Show/Hide
|
C22H21ClN6
|
1
|
1 |
AC50 = 8650 nM
|
|
|
CP0862122
|
SID131411727
Show/Hide
|
C36H46Cl2N4O5
|
1
|
1 |
AC50 = 8650 nM
|
|
|
CP0912230
|
SID131411752
Show/Hide
|
C34H45F6N3O5
|
1
|
1 |
AC50 = 8650 nM
|
|
|
CP0865128
|
SID85804725
Show/Hide
|
C37H48N4O4
|
1
|
1 |
AC50 = 8660 nM
|
|
|
CP0908091
|
SID87541921
Show/Hide
|
C34H44F3N3O6S2
|
1
|
1 |
AC50 = 8660 nM
|
|
|
CP0905827
|
SID131414292
Show/Hide
|
C29H32FN3O4S
|
1
|
1 |
AC50 = 8670 nM
|
|
|
CP0949417
|
SID131412855
Show/Hide
|
C35H44Cl3N3O6S
|
1
|
1 |
AC50 = 8680 nM
|
|
|
CP0906937
|
SID85201451
Show/Hide
|
C31H35F3N4O7S
|
1
|
1 |
AC50 = 8690 nM
|
|
|
CP0950303
|
SID131410528
Show/Hide
|
C36H45F4N3O6S
|
1
|
1 |
AC50 = 8700 nM
|
|
|
CP0915294
|
SID131461890
Show/Hide
|
C27H27FN2O3
|
1
|
1 |
AC50 = 8720 nM
|
|
|
CP0671680
|
SID50107233
Show/Hide
|
C28H30N2O6S
|
1
|
1 |
AC50 = 8770 nM
|
|
|
CP0883185
|
SID131411338
Show/Hide
|
C37H45F3N4O6
|
1
|
1 |
AC50 = 8770 nM
|
|
|
CP0647991
|
SID49645896
Show/Hide
|
C18H16BrN3O
|
1
|
1 |
AC50 = 8780 nM
|
|
|
CP0926607
|
SID144191247
Show/Hide
|
C26H24F3N3O
|
1
|
1 |
AC50 = 8800 nM
|
|
|
CP0042741
|
AURIN
Show/Hide
|
C19H14O3
|
1
|
1 |
AC50 = 8810 nM
|
|
|
CP0848115
|
SID87541350
Show/Hide
|
C30H44ClN3O6S
|
1
|
1 |
AC50 = 8810 nM
|
|
|
CP0952612
|
SID87218849
Show/Hide
|
C36H40FN3O5S
|
1
|
1 |
AC50 = 8820 nM
|
|
|
CP0875509
|
SID49731807
Show/Hide
|
C19H16ClN3O4S
|
1
|
1 |
AC50 = 8830 nM
|
|
|
CP0247735
|
(4S)-3-[2-(4-ethoxyphenyl)ethyl]-4-[(4-hydroxyphenyl)methyl]-1-[(2S)-1-(4-hydroxyphenyl)-3-[(2R)-2-[[(5S)-5-(2-methylpropyl)-2-sulfanylidene-1-imidazolidinyl]methyl]-1-pyrrolidinyl]propan-2-yl]-2-imidazolidinethione
Show/Hide
|
C41H55N5O3S2
|
1
|
1 |
AC50 = 8840 nM
|
|
|
CP0892613
|
SID17515789
Show/Hide
|
C18H18ClF2N3OS2
|
1
|
1 |
AC50 = 8860 nM
|
|
|
CP0883152
|
SID131456882
Show/Hide
|
C25H28Cl3N3O5
|
1
|
1 |
AC50 = 8870 nM
|
|
|
CP0900575
|
SID85805567
Show/Hide
|
C36H45Cl2N3O5
|
1
|
1 |
AC50 = 8870 nM
|
|
|
CP0950342
|
SID87543582
Show/Hide
|
C33H35F6N5O5
|
1
|
1 |
AC50 = 8870 nM
|
|
|
CP0243963
|
4-methoxybenzoic acid [(Z)-[amino(2-pyridinyl)methylidene]amino] ester
Show/Hide
|
C14H13N3O3
|
1
|
1 |
AC50 = 8880 nM
|
|
|
CP0245298
|
7-chloranyl-1,3,6-trimethyl-pteridine-2,4-dione
Show/Hide
|
C9H9ClN4O2
|
1
|
1 |
AC50 = 8880 nM
|
|
|
CP0827288
|
SID57260982
Show/Hide
|
C19H12O3
|
1
|
1 |
AC50 = 8880 nM
|
|
|
CP0864691
|
SID131447151
Show/Hide
|
C22H21FN2O2
|
1
|
1 |
AC50 = 8880 nM
|
|
|
CP0815877
|
SID87335296
Show/Hide
|
C17H19Cl2N5O5S
|
1
|
1 |
AC50 = 8910 nM
|
|
|
CP0712538
|
SID24808744
Show/Hide
|
C19H16BrN3O2S2
|
1
|
1 |
AC50 = 8920 nM
|
|
|
CP0957472
|
SID87543349
Show/Hide
|
C36H45F4N3O6S
|
1
|
1 |
AC50 = 8920 nM
|
|
|
CP0872444
|
SID87541101
Show/Hide
|
C37H46F3N3O5
|
1
|
1 |
AC50 = 8950 nM
|
|
|
CP0900525
|
SID124754746
Show/Hide
|
C36H29F3N6O3
|
1
|
1 |
AC50 = 8950 nM
|
|
|
CP0860400
|
SID85200285
Show/Hide
|
C39H44FN3O5
|
1
|
1 |
AC50 = 8960 nM
|
|
|
CP0279214
|
4-[(7-chloranyl-4-nitro-2,1,3-benzoxadiazol-5-yl)amino]-1,5-dimethyl-2-phenyl-pyrazol-3-one
Show/Hide
|
C17H13ClN6O4
|
1
|
1 |
AC50 = 8970 nM
|
|
|
CP0957477
|
SID131438440
Show/Hide
|
C22H24Cl2FN3O4
|
1
|
1 |
AC50 = 8970 nM
|
|
|
CP0890214
|
SID99357045
Show/Hide
|
C34H33F6N5O6
|
1
|
1 |
AC50 = 8980 nM
|
|
|
CP0942778
|
SID144193222
Show/Hide
|
C26H27FN2O4S
|
1
|
1 |
AC50 = 8980 nM
|
|
|
CP0947578
|
SID131413392
Show/Hide
|
C30H35N3O5S
|
1
|
1 |
AC50 = 8980 nM
|
|
|
CP0957474
|
SID131412710
Show/Hide
|
C37H48F3N3O6S
|
1
|
1 |
AC50 = 8980 nM
|
|
|
CP0886329
|
SID131412384
Show/Hide
|
C36H46F3N3O6S
|
1
|
1 |
AC50 = 9010 nM
|
|
|
CP0965723
|
SID131411675
Show/Hide
|
C36H46F3N5O5
|
1
|
1 |
AC50 = 9030 nM
|
|
|
CP0966607
|
SID134214409
Show/Hide
|
C35H29BrF3N5O2
|
1
|
1 |
AC50 = 9030 nM
|
|
|
CP0244118
|
2-methyl-2-propenoic acid [7-methyl-3-oxo-2-(trifluoromethyl)-4H-1,4-benzoxazin-2-yl] ester
Show/Hide
|
C14H12F3NO4
|
1
|
1 |
AC50 = 9050 nM
|
|
|
CP0912513
|
SID131411840
Show/Hide
|
C35H50ClN3O7S
|
1
|
1 |
AC50 = 9050 nM
|
|
|
CP0908905
|
SID131426793
Show/Hide
|
C30H34F3N3O5S
|
1
|
1 |
AC50 = 9060 nM
|
|
|
CP0910464
|
SID103050677
Show/Hide
|
C26H24F3N5O2
|
1
|
1 |
AC50 = 9070 nM
|
|
|
CP0933809
|
SID104170438
Show/Hide
|
C36H49N3O8S2
|
1
|
1 |
AC50 = 9070 nM
|
|
|
CP0698515
|
SID49641429
Show/Hide
|
C19H19N3O
|
1
|
1 |
AC50 = 9080 nM
|
|
|
CP0868094
|
SID87541280
Show/Hide
|
C34H44F3N3O6S2
|
1
|
1 |
AC50 = 9080 nM
|
|
|
CP0950372
|
SID104170772
Show/Hide
|
C38H48F3N3O5
|
1
|
1 |
AC50 = 9100 nM
|
|
|
CP0450711
|
(phenylmethyl) N-[4-[phenylmethoxycarbonyl-[3-[(phenylmethyl)amino]propyl]amino]butyl]-N-[3-[(phenylmethyl)amino]propyl]carbamate
Show/Hide
|
C40H50N4O4
|
1
|
1 |
AC50 = 9110 nM
|
|
|
CP0908896
|
SID131454051
Show/Hide
|
C31H34N2O6
|
1
|
1 |
AC50 = 9110 nM
|
|
|
CP0942781
|
SID87543361
Show/Hide
|
C37H47F3N4O5
|
1
|
1 |
AC50 = 9110 nM
|
|
|
CP0879952
|
SID131408798
Show/Hide
|
C32H44N4O6
|
1
|
1 |
AC50 = 9150 nM
|
|
|
CP0938692
|
SID131411249
Show/Hide
|
C38H47F3N4O7
|
1
|
1 |
AC50 = 9150 nM
|
|
|
CP0209442
|
6-(1H-Benzoimidazol-2-ylsulfanylmethyl)-2-(4-methyl-quinazolin-2-ylamino)-pyrimidin-4-ol
Show/Hide
|
C21H17N7OS
|
1
|
1 |
AC50 = 9160 nM
|
|
|
CP0890232
|
SID87542232
Show/Hide
|
C37H48F3N3O6S
|
1
|
1 |
AC50 = 9160 nM
|
|
|
CP0908582
|
SID87541727
Show/Hide
|
C38H49F3N4O6
|
1
|
1 |
AC50 = 9160 nM
|
|
|
CP0793499
|
SID49722406
Show/Hide
|
C28H32N6O
|
1
|
1 |
AC50 = 9170 nM
|
|
|
CP0862093
|
SID131412393
Show/Hide
|
C36H47Cl2N3O6S
|
1
|
1 |
AC50 = 9180 nM
|
|
|
CP0888887
|
SID104170558
Show/Hide
|
C33H43Cl2N3O6S2
|
1
|
1 |
AC50 = 9200 nM
|
|
|
CP0873859
|
SID131413002
Show/Hide
|
C35H52ClN3O6S
|
1
|
1 |
AC50 = 9230 nM
|
|
|
CP0907788
|
SID131410264
Show/Hide
|
C38H48F3N3O5
|
1
|
1 |
AC50 = 9250 nM
|
|
|
CP0852371
|
SID87539816
Show/Hide
|
C37H45Cl2F3N4O5
|
1
|
1 |
AC50 = 9260 nM
|
|
|
CP0857391
|
SID121283976
Show/Hide
|
C42H55N5O2S2
|
1
|
1 |
AC50 = 9270 nM
|
|
|
CP0933807
|
SID81066244
Show/Hide
|
C32H31FN2O4
|
1
|
1 |
AC50 = 9270 nM
|
|
|
CP0358944
|
5-chloranyl-N-(4-fluorophenyl)-2-[(3-methylphenyl)methylsulfonyl]pyrimidine-4-carboxamide
Show/Hide
|
C19H15ClFN3O3S
|
1
|
1 |
AC50 = 9280 nM
|
|
|
CP0045980
|
7-chloranyl-N-[2-(dimethylamino)ethyl]-4H-thieno[3,2-c]thiochromene-2-carboxamide
Show/Hide
|
C16H17ClN2OS2
|
1
|
1 |
AC50 = 9290 nM
|
|
|
CP0868108
|
SID131426791
Show/Hide
|
C30H34F3N3O5S
|
1
|
1 |
AC50 = 9300 nM
|
|
|
CP0912635
|
SID87541156
Show/Hide
|
C32H37F3N4O4
|
1
|
1 |
AC50 = 9300 nM
|
|
|
CP0409989
|
(2S)-2-amino-N-[(3S,10R,13S,17S)-3-hydroxy-10,13-dimethyl-2,3,4,7,8,9,11,12,14,15,16,17-dodecahydro-1H-cyclopenta[a]phenanthren-17-yl]-3,3-dimethyl-butyramide
Show/Hide
|
C25H42N2O2
|
1
|
1 |
AC50 = 9310 nM
|
|
|
CP0930558
|
SID87540016
Show/Hide
|
C38H43N3O4
|
1
|
1 |
AC50 = 9310 nM
|
|
|
CP0946011
|
SID131462187
Show/Hide
|
C27H35N3O2
|
1
|
1 |
AC50 = 9310 nM
|
|
|
CP0864729
|
SID87543200
Show/Hide
|
C33H44Cl2F3N3O5
|
1
|
1 |
AC50 = 9320 nM
|
|
|
CP0900521
|
SID131410855
Show/Hide
|
C38H49F3N4O6
|
1
|
1 |
AC50 = 9320 nM
|
|
|
CP0944035
|
SID87540043
Show/Hide
|
C37H46F3N3O5
|
1
|
1 |
AC50 = 9330 nM
|
|
|
CP0432832
|
MLS003122000
Show/Hide
|
C23H25F3N2O4S
|
1
|
1 |
AC50 = 9350 nM
|
|
|
CP0952081
|
SID87542183
Show/Hide
|
C38H43N3O4
|
1
|
1 |
AC50 = 9360 nM
|
|
|
CP0856878
|
SID131412254
Show/Hide
|
C37H46F4N4O5
|
1
|
1 |
AC50 = 9370 nM
|
|
|
CP0860395
|
SID87218833
Show/Hide
|
C31H34F4N4O6S
|
1
|
1 |
AC50 = 9390 nM
|
|
|
CP0908686
|
SID131461766
Show/Hide
|
C27H30N2O5S
|
1
|
1 |
AC50 = 9390 nM
|
|
|
CP0439301
|
1,2,3-Trimethyl-2-phenyl-2,3-dihydro-1H-benzoimidazole
Show/Hide
|
C16H18N2
|
1
|
1 |
AC50 = 9400 nM
|
|
|
CP0884584
|
SID87540637
Show/Hide
|
C35H46F3N5O8S
|
1
|
1 |
AC50 = 9400 nM
|
|
|
CP0907295
|
SID144192178
Show/Hide
|
C28H22F2N2O3
|
1
|
1 |
AC50 = 9400 nM
|
|
|
CP0912665
|
SID87218837
Show/Hide
|
C37H43N3O6S
|
1
|
1 |
AC50 = 9410 nM
|
|
|
CP0935274
|
SID87541080
Show/Hide
|
C34H44F3N3O6S2
|
1
|
1 |
AC50 = 9410 nM
|
|
|
CP0902685
|
SID87542342
Show/Hide
|
C34H43ClFN3O8S2
|
1
|
1 |
AC50 = 9430 nM
|
|
|
CP0908659
|
SID144194145
Show/Hide
|
C26H26N2O3S
|
1
|
1 |
AC50 = 9430 nM
|
|
|
CP0908658
|
SID131462624
Show/Hide
|
C27H34N2O4S
|
1
|
1 |
AC50 = 9440 nM
|
|
|
CP0885651
|
SID131412372
Show/Hide
|
C36H46ClN3O8S
|
1
|
1 |
AC50 = 9450 nM
|
|
|
CP0935175
|
SID85810268
Show/Hide
|
C32H37F3N4O6S
|
1
|
1 |
AC50 = 9450 nM
|
|
|
CP0957469
|
SID131414741
Show/Hide
|
C27H35FN2O6S2
|
1
|
1 |
AC50 = 9450 nM
|
|
|
CP0966893
|
SID87218855
Show/Hide
|
C30H35Cl2N3O5S
|
1
|
1 |
AC50 = 9450 nM
|
|
|
CP0966605
|
SID131412257
Show/Hide
|
C37H46F4N4O5
|
1
|
1 |
AC50 = 9460 nM
|
|
|
CP0908903
|
SID131426921
Show/Hide
|
C30H38FN3O5S
|
1
|
1 |
AC50 = 9470 nM
|
|
|
CP0959674
|
SID131411334
Show/Hide
|
C37H45F3N4O6
|
1
|
1 |
AC50 = 9480 nM
|
|
|
CP0938694
|
SID87540449
Show/Hide
|
C37H47F3N4O5
|
1
|
1 |
AC50 = 9490 nM
|
|
|
CP0881115
|
SID131442205
Show/Hide
|
C31H30F3N3O5
|
1
|
1 |
AC50 = 9500 nM
|
|
|
CP0961312
|
SID131414219
Show/Hide
|
C30H40N2O7S2
|
1
|
1 |
AC50 = 9500 nM
|
|
|
CP0883179
|
SID104170450
Show/Hide
|
C36H45Cl2FN4O5
|
1
|
1 |
AC50 = 9510 nM
|
|
|
CP0928969
|
SID131411825
Show/Hide
|
C37H48F3N3O7S
|
1
|
1 |
AC50 = 9510 nM
|
|
|
CP0089042
|
MLS000689772
Show/Hide
|
C18H14N4O3S2
|
1
|
1 |
AC50 = 9520 nM
|
|
|
CP0916970
|
SID131426919
Show/Hide
|
C30H38FN3O5S
|
1
|
1 |
AC50 = 9520 nM
|
|
|
CP0921054
|
SID131434104
Show/Hide
|
C33H39N3O6S
|
1
|
1 |
AC50 = 9530 nM
|
|
|
CP0860396
|
SID87542419
Show/Hide
|
C37H46F3N3O5
|
1
|
1 |
AC50 = 9550 nM
|
|
|
CP0936518
|
SID131414997
Show/Hide
|
C27H35FN2O6S2
|
1
|
1 |
AC50 = 9600 nM
|
|
|
CP0058175
|
1-(2-furanyl)-3-phenyl-2-propyn-1-one
Show/Hide
|
C13H8O2
|
1
|
1 |
AC50 = 9610 nM
|
|
|
CP0886437
|
SID134961947
Show/Hide
|
C30H33F3N2O5S
|
1
|
1 |
AC50 = 9620 nM
|
|
|
CP0942606
|
SID85805566
Show/Hide
|
C37H48F3N3O7S
|
1
|
1 |
AC50 = 9620 nM
|
|
|
CP0966892
|
SID131456926
Show/Hide
|
C29H31ClN2O6S
|
1
|
1 |
AC50 = 9620 nM
|
|
|
CP0947577
|
SID87543151
Show/Hide
|
C38H48F3N3O5
|
1
|
1 |
AC50 = 9660 nM
|
|
|
CP0965720
|
SID104170390
Show/Hide
|
C37H45Cl2F3N4O5
|
1
|
1 |
AC50 = 9660 nM
|
|
|
CP0864531
|
SID144192112
Show/Hide
|
C28H25FN2O4S
|
1
|
1 |
AC50 = 9680 nM
|
|
|
CP0860346
|
SID26661590
Show/Hide
|
C27H26N4O
|
1
|
1 |
AC50 = 9700 nM
|
|
|
CP0950779
|
SID99356700
Show/Hide
|
C25H30ClFN4O
|
1
|
1 |
AC50 = 9710 nM
|
|
|
CP0856713
|
SID131410526
Show/Hide
|
C36H45F4N3O6S
|
1
|
1 |
AC50 = 9730 nM
|
|
|
CP0907262
|
SID99359313
Show/Hide
|
C37H46F3N3O5
|
1
|
1 |
AC50 = 9740 nM
|
|
|
CP0942390
|
SID131446923
Show/Hide
|
C26H25FN2O2
|
1
|
1 |
AC50 = 9740 nM
|
|
|
CP0940403
|
SID131412178
Show/Hide
|
C34H43ClFN3O8S2
|
1
|
1 |
AC50 = 9750 nM
|
|
|
CP0912658
|
SID131460384
Show/Hide
|
C26H32N2O3
|
1
|
1 |
AC50 = 9800 nM
|
|
|
CP0865947
|
SID50085505
Show/Hide
|
C18H20O5S
|
1
|
1 |
AC50 = 9820 nM
|
|
|
CP0884817
|
SID87541425
Show/Hide
|
C37H42N4O5
|
1
|
1 |
AC50 = 9840 nM
|
|
|
CP0885563
|
SID103050557
Show/Hide
|
C26H25N5O2S
|
1
|
1 |
AC50 = 9840 nM
|
|
|
CP0176769
|
MLS001116215
Show/Hide
|
C20H17ClN4O4S
|
1
|
1 |
AC50 = 9860 nM
|
|
|
CP0862103
|
SID131412373
Show/Hide
|
C36H46ClN3O8S
|
1
|
1 |
AC50 = 9860 nM
|
|
|
CP0921255
|
SID92763670
Show/Hide
|
C42H55N5O2S2
|
1
|
1 |
AC50 = 9860 nM
|
|
|
CP0908092
|
SID131456923
Show/Hide
|
C29H31ClN2O6S
|
1
|
1 |
AC50 = 9870 nM
|
|
|
CP0411344
|
MLS003124149
Show/Hide
|
C27H29N5O2S
|
1
|
1 |
AC50 = 9880 nM
|
|
|
CP0857029
|
SID144194411
Show/Hide
|
C34H38F3N3O3
|
1
|
1 |
AC50 = 9890 nM
|
|
|
CP0874968
|
SID85805606
Show/Hide
|
C36H45ClF3N3O6S
|
1
|
1 |
AC50 = 9890 nM
|
|
|
CP0920056
|
SID131463064
Show/Hide
|
C31H32FN3O3
|
1
|
1 |
AC50 = 9890 nM
|
|
|
CP0965785
|
SID131464460
Show/Hide
|
C30H30FN3O2
|
1
|
1 |
AC50 = 9890 nM
|
|
|
CP0197844
|
(2S)-1-N-[(2R)-1-cyclohexyl-3-(methylamino)propan-2-yl]-4-methyl-2-N-[2-[3-(trifluoromethyl)phenyl]ethyl]pentane-1,2-diamine
Show/Hide
|
C25H42F3N3
|
1
|
1 |
AC50 = 9930 nM
|
|
|
CP0906226
|
SID104170636
Show/Hide
|
C35H45Cl2N3O6S
|
1
|
1 |
AC50 = 9930 nM
|
|
|
CP0388928
|
4-[4-(3,4-dimethoxyphenyl)-6-(trifluoromethyl)pyrimidin-2-yl]sulfonyl-N-(5-methyl-1,2-oxazol-3-yl)butanamide
Show/Hide
|
C21H21F3N4O6S
|
1
|
1 |
AC50 = 9940 nM
|
|
|
CP0439555
|
(2R,3R)-2-N-[(2R)-2-[2-[3,5-bis(trifluoromethyl)phenyl]ethylamino]pentyl]-1-N,3-dimethylpentane-1,2-diamine
Show/Hide
|
C22H35F6N3
|
1
|
1 |
AC50 = 9950 nM
|
|
|
CP0445623
|
2-Chloro-N-(5-chloro-3-methyl-1-phenyl-1H-pyrazol-4-ylmethyl)-N-naphthalen-1-yl-acetamide
Show/Hide
|
C23H19Cl2N3O
|
1
|
1 |
AC50 = 9950 nM
|
|
|
CP0856882
|
SID87541998
Show/Hide
|
C36H47FN4O8S
|
1
|
1 |
AC50 = 9960 nM
|
|
|
CP0885784
|
SID87541634
Show/Hide
|
C37H47F3N4O8S
|
1
|
1 |
AC50 = 9960 nM
|
|
|
CP0934611
|
SID131412709
Show/Hide
|
C37H48F3N3O6S
|
1
|
1 |
AC50 = 9980 nM
|
|
|
CP0886270
|
SID131464768
Show/Hide
|
C27H34N2O3S
|
1
|
1 |
AC50 = 9990 nM
|
|
|
CP0935285
|
SID131460486
Show/Hide
|
C25H30N2O4S
|
1
|
1 |
AC50 = 10010 nM
|
|
|
CP0897059
|
SID131412503
Show/Hide
|
C34H44ClN3O8S2
|
1
|
1 |
AC50 = 10060 nM
|
|
|
CP0950774
|
SID131461186
Show/Hide
|
C27H27N3O3S
|
1
|
1 |
AC50 = 10060 nM
|
|
|
CP0908580
|
SID87540899
Show/Hide
|
C31H36F3N3O5S
|
1
|
1 |
AC50 = 10080 nM
|
|
|
CP0158376
|
(2E)-N-[2-(1-azepanyl)ethyl]-2-[(3-methoxyphenyl)methylidene]-3-oxo-4H-1,4-benzothiazine-6-carboxamide
Show/Hide
|
C25H29N3O3S
|
1
|
1 |
AC50 = 10100 nM
|
|
|
CP0879938
|
SID131410608
Show/Hide
|
C37H53F3N4O5
|
1
|
1 |
AC50 = 10110 nM
|
|
|
CP0950480
|
SID144191157
Show/Hide
|
C27H30N2O3
|
1
|
1 |
AC50 = 10110 nM
|
|
|
CP0942475
|
SID131464462
Show/Hide
|
C30H30FN3O2
|
1
|
1 |
AC50 = 10120 nM
|
|
|
CP0897514
|
SID87541643
Show/Hide
|
C37H46F3N3O5
|
1
|
1 |
AC50 = 10130 nM
|
|
|
CP0908119
|
SID85808898
Show/Hide
|
C37H47F3N4O5
|
1
|
1 |
AC50 = 10130 nM
|
|
|
CP0908899
|
SID131412181
Show/Hide
|
C34H43ClFN3O8S2
|
1
|
1 |
AC50 = 10140 nM
|
|
|
CP0942585
|
SID131412011
Show/Hide
|
C37H46F3N3O5
|
1
|
1 |
AC50 = 10150 nM
|
|
|
CP0907411
|
SID134214420
Show/Hide
|
C36H38F3NO5
|
1
|
1 |
AC50 = 10160 nM
|
|
|
CP0908028
|
SID85804815
Show/Hide
|
C29H32ClFN4O6S
|
1
|
1 |
AC50 = 10160 nM
|
|
|
CP0908034
|
SID131412376
Show/Hide
|
C36H46ClN3O8S
|
1
|
1 |
AC50 = 10160 nM
|
|
|
CP0900526
|
SID131464558
Show/Hide
|
C28H29F2N3O2
|
1
|
1 |
AC50 = 10170 nM
|
|
|
CP0481883
|
5-(3,5-dichlorobenzyl)-4,6-dihydrotriazolo[1,5-a][1,4]benzodiazepine-6-carbonitrile
Show/Hide
|
C18H13Cl2N5
|
1
|
1 |
AC50 = 10180 nM
|
|
|
CP0872446
|
SID85810736
Show/Hide
|
C36H47Cl2N3O7S
|
1
|
1 |
AC50 = 10210 nM
|
|
|
CP0912290
|
SID131461102
Show/Hide
|
C27H27FN2O2
|
1
|
1 |
AC50 = 10230 nM
|
|
|
CP0864665
|
SID87542504
Show/Hide
|
C35H44Cl3N3O6S
|
1
|
1 |
AC50 = 10240 nM
|
|
|
CP0883682
|
SID85794589
Show/Hide
|
C32H42F3N5O5
|
1
|
1 |
AC50 = 10250 nM
|
|
|
CP0942427
|
SID131461219
Show/Hide
|
C27H30N2O5S
|
1
|
1 |
AC50 = 10260 nM
|
|
|
CP0864561
|
SID131447921
Show/Hide
|
C19H23FN2O3S
|
1
|
1 |
AC50 = 10270 nM
|
|
|
CP0917912
|
SID131414929
Show/Hide
|
C27H35FN2O6S2
|
1
|
1 |
AC50 = 10280 nM
|
|
|
CP0918066
|
SID131409347
Show/Hide
|
C38H41F3N4O5
|
1
|
1 |
AC50 = 10300 nM
|
|
|
CP0934610
|
SID131415237
Show/Hide
|
C29H37FN2O5S
|
1
|
1 |
AC50 = 10320 nM
|
|
|
CP0873978
|
SID85201720
Show/Hide
|
C31H34ClF3N4O6S
|
1
|
1 |
AC50 = 10350 nM
|
|
|
CP0891768
|
SID49645784
Show/Hide
|
C21H18ClN3O2
|
1
|
1 |
AC50 = 10350 nM
|
|
|
CP0885642
|
SID131410359
Show/Hide
|
C35H46ClN3O8S2
|
1
|
1 |
AC50 = 10360 nM
|
|
|
CP0352388
|
2-benzylsulfonyl-5-chloro-N-(4-fluorophenyl)pyrimidine-4-carboxamide
Show/Hide
|
C18H13ClFN3O3S
|
1
|
1 |
AC50 = 10370 nM
|
|
|
CP0115115
|
1-(4-methoxyphenyl)-3-[(5-phenyl-1,3,4-oxadiazol-2-yl)sulfanyl]pyrrolidine-2,5-dione
Show/Hide
|
C19H15N3O4S
|
1
|
1 |
AC50 = 10390 nM
|
|
|
CP0907182
|
SID131461874
Show/Hide
|
C27H30N2O4S
|
1
|
1 |
AC50 = 10390 nM
|
|
|
CP0908893
|
SID144192239
Show/Hide
|
C28H23F2N3O3
|
1
|
1 |
AC50 = 10390 nM
|
|
|
CP0932243
|
SID87541326
Show/Hide
|
C33H45ClN4O9S2
|
1
|
1 |
AC50 = 10420 nM
|
|
|
CP0891770
|
SID131462629
Show/Hide
|
C27H34N2O4S
|
1
|
1 |
AC50 = 10430 nM
|
|
|
CP0809722
|
SID17401429
Show/Hide
|
C30H31NO5
|
1
|
1 |
AC50 = 10440 nM
|
|
|
CP0898772
|
SID131415353
Show/Hide
|
C29H37FN2O5S
|
1
|
1 |
AC50 = 10440 nM
|
|
|
CP0882352
|
SID85813514
Show/Hide
|
C32H41N5O4
|
1
|
1 |
AC50 = 10460 nM
|
|
|
CP0950762
|
SID131446655
Show/Hide
|
C25H24FN3O2
|
1
|
1 |
AC50 = 10470 nM
|
|
|
CP0885256
|
SID131461118
Show/Hide
|
C24H27FN2O3S
|
1
|
1 |
AC50 = 10490 nM
|
|
|
CP0881161
|
SID131411861
Show/Hide
|
C35H51ClN4O7S
|
1
|
1 |
AC50 = 10500 nM
|
|
|
CP0934609
|
SID131464705
Show/Hide
|
C30H31N3O2
|
1
|
1 |
AC50 = 10500 nM
|
|
|
CP0263109
|
8-aminoquinoline-5,6-dione
Show/Hide
|
C9H6N2O2
|
1
|
1 |
AC50 = 10510 nM
|
|
|
CP0908637
|
SID131412778
Show/Hide
|
C33H45ClN4O9S2
|
1
|
1 |
AC50 = 10520 nM
|
|
|
CP0237388
|
MLS000911561
Show/Hide
|
C33H31F6N5O3
|
1
|
1 |
AC50 = 10570 nM
|
|
|
CP0860345
|
SID131461247
Show/Hide
|
C26H28N2O5S
|
1
|
1 |
AC50 = 10570 nM
|
|
|
CP0860507
|
SID144195157
Show/Hide
|
C27H35N3O3
|
1
|
1 |
AC50 = 10570 nM
|
|
|
CP0881739
|
SID87540147
Show/Hide
|
C34H40F3N3O5
|
1
|
1 |
AC50 = 10610 nM
|
|
|
CP0938689
|
SID131412253
Show/Hide
|
C37H46F4N4O5
|
1
|
1 |
AC50 = 10610 nM
|
|
|
CP0908124
|
SID144194869
Show/Hide
|
C26H25FN2O3
|
1
|
1 |
AC50 = 10630 nM
|
|
|
CP0858470
|
SID131454189
Show/Hide
|
C30H34N2O6S
|
1
|
1 |
AC50 = 10650 nM
|
|
|
CP0908041
|
SID144190778
Show/Hide
|
C26H24FN3O
|
1
|
1 |
AC50 = 10650 nM
|
|
|
CP0906225
|
SID87539803
Show/Hide
|
C37H46F4N4O5
|
1
|
1 |
AC50 = 10660 nM
|
|
|
CP0942478
|
SID131460392
Show/Hide
|
C27H35N3O3
|
1
|
1 |
AC50 = 10700 nM
|
|
|
CP0888858
|
SID131442206
Show/Hide
|
C31H30F3N3O5
|
1
|
1 |
AC50 = 10720 nM
|
|
|
CP0930560
|
SID87540723
Show/Hide
|
C33H50N4O7S2
|
1
|
1 |
AC50 = 10720 nM
|
|
|
CP0900528
|
SID131411836
Show/Hide
|
C35H50ClN3O7S
|
1
|
1 |
AC50 = 10770 nM
|
|
|
CP0952671
|
SID87543037
Show/Hide
|
C37H46F3N5O6
|
1
|
1 |
AC50 = 10770 nM
|
|
|
CP0862098
|
SID87540258
Show/Hide
|
C36H45F2N5O6
|
1
|
1 |
AC50 = 10790 nM
|
|
|
CP0865835
|
SID131461056
Show/Hide
|
C25H30N2O3S
|
1
|
1 |
AC50 = 10810 nM
|
|
|
CP0886579
|
SID104170692
Show/Hide
|
C37H48F3N3O7S
|
1
|
1 |
AC50 = 10810 nM
|
|
|
CP0943302
|
SID87540247
Show/Hide
|
C37H47F3N4O5
|
1
|
1 |
AC50 = 10840 nM
|
|
|
CP0189344
|
(2S)-2-(4-fluorobenzyl)hex-5-enoic acid [(2R)-2-[[(2R)-2-[2-[benzyl(2-hydroxyethyl)amino]-2-keto-ethyl]pent-4-enoyl]amino]-3-(1H-indol-3-yl)propyl] ester
Show/Hide
|
C40H46FN3O5
|
1
|
1 |
AC50 = 10860 nM
|
|
|
CP0884738
|
SID131412776
Show/Hide
|
C33H45ClN4O9S2
|
1
|
1 |
AC50 = 10860 nM
|
|
|
CP0930554
|
SID87540354
Show/Hide
|
C38H49F3N4O6
|
1
|
1 |
AC50 = 10860 nM
|
|
|
CP0949415
|
SID131425910
Show/Hide
|
C30H35N3O5S
|
1
|
1 |
AC50 = 10860 nM
|
|
|
CP0890219
|
SID131463062
Show/Hide
|
C31H32FN3O3
|
1
|
1 |
AC50 = 10870 nM
|
|
|
CP0912504
|
SID131411927
Show/Hide
|
C36H54N4O5
|
1
|
1 |
AC50 = 10880 nM
|
|
|
CP0942777
|
SID131462385
Show/Hide
|
C27H34N2O3S
|
1
|
1 |
AC50 = 10880 nM
|
|
|
CP0940509
|
SID104170451
Show/Hide
|
C37H47F3N4O5
|
1
|
1 |
AC50 = 10890 nM
|
|
|
CP0900527
|
SID144196897
Show/Hide
|
C27H35N3O3
|
1
|
1 |
AC50 = 10910 nM
|
|
|
CP0872442
|
SID131411774
Show/Hide
|
C37H47FN4O7
|
1
|
1 |
AC50 = 10930 nM
|
|
|
CP0884743
|
SID131461057
Show/Hide
|
C25H30N2O3S
|
1
|
1 |
AC50 = 10930 nM
|
|
|
CP0941654
|
SID81065978
Show/Hide
|
C31H28F4N2O4
|
1
|
1 |
AC50 = 10940 nM
|
|
|
CP0875012
|
SID131408816
Show/Hide
|
C32H44N4O6
|
1
|
1 |
AC50 = 10980 nM
|
|
|
CP0885555
|
SID131449099
Show/Hide
|
C24H22ClFN2O3S
|
1
|
1 |
AC50 = 10980 nM
|
|
|
CP0881111
|
SID131408792
Show/Hide
|
C32H41N3O4
|
1
|
1 |
AC50 = 11000 nM
|
|
|
CP0905830
|
SID87541805
Show/Hide
|
C32H35Cl2F3N4O4
|
1
|
1 |
AC50 = 11050 nM
|
|
|
CP0881654
|
SID134962141
Show/Hide
|
C32H36FN3O5S
|
1
|
1 |
AC50 = 11070 nM
|
|
|
CP0900522
|
SID131447425
Show/Hide
|
C24H21FN2O2
|
1
|
1 |
AC50 = 11090 nM
|
|
|
CP0885260
|
SID85815481
Show/Hide
|
C36H53N5O5
|
1
|
1 |
AC50 = 11100 nM
|
|
|
CP0874969
|
SID85802667
Show/Hide
|
C32H34F3N5O7
|
1
|
1 |
AC50 = 11120 nM
|
|
|
CP0942474
|
SID144194783
Show/Hide
|
C26H33N3O2
|
1
|
1 |
AC50 = 11120 nM
|
|
|
CP0908031
|
SID131461218
Show/Hide
|
C27H30N2O5S
|
1
|
1 |
AC50 = 11140 nM
|
|
|
CP0908713
|
SID131447015
Show/Hide
|
C25H26N2O3S
|
1
|
1 |
AC50 = 11140 nM
|
|
|
CP0889240
|
SID87541487
Show/Hide
|
C37H47Cl2N3O5
|
1
|
1 |
AC50 = 11170 nM
|
|
|
CP0915296
|
SID85804262
Show/Hide
|
C31H35ClF3N3O5S
|
1
|
1 |
AC50 = 11180 nM
|
|
|
CP0294729
|
2-[[2-(2,4-dichlorophenyl)-2-(1H-indol-3-yl)ethyl]amino]-1-phenyl-ethanol
Show/Hide
|
C24H22Cl2N2O
|
1
|
1 |
AC50 = 11200 nM
|
|
|
CP0347224
|
2-(4-Bromo-phenyl)-6-methyl-imidazo[1,2-a]pyridine
Show/Hide
|
C14H11BrN2
|
1
|
1 |
AC50 = 11200 nM
|
|
|
CP0907263
|
SID131449036
Show/Hide
|
C19H22N2O2
|
1
|
1 |
AC50 = 11210 nM
|
|
|
CP0865857
|
SID99358387
Show/Hide
|
C32H36FN3O5S
|
1
|
1 |
AC50 = 11300 nM
|
|
|
CP0907197
|
SID99359305
Show/Hide
|
C36H45Cl2FN4O5
|
1
|
1 |
AC50 = 11310 nM
|
|
|
CP0846305
|
SID50085521
Show/Hide
|
C16H15FO3S
|
1
|
1 |
AC50 = 11320 nM
|
|
|
CP0926613
|
SID87540182
Show/Hide
|
C35H53N5O5
|
1
|
1 |
AC50 = 11330 nM
|
|
|
CP0908888
|
SID131464468
Show/Hide
|
C29H34N2O3S
|
1
|
1 |
AC50 = 11360 nM
|
|
|
CP0926617
|
SID85810889
Show/Hide
|
C32H35F4N5O5
|
1
|
1 |
AC50 = 11410 nM
|
|
|
CP0934878
|
SID85811442
Show/Hide
|
C31H35F4N3O5S
|
1
|
1 |
AC50 = 11440 nM
|
|
|
CP0886575
|
SID144196926
Show/Hide
|
C26H33N3O2
|
1
|
1 |
AC50 = 11450 nM
|
|
|
CP0906898
|
SID104170571
Show/Hide
|
C37H53F3N4O5
|
1
|
1 |
AC50 = 11450 nM
|
|
|
CP0442869
|
(4S)-1-[(1S)-1-benzyl-2-[2-[[(5S)-5-(4-hydroxybenzyl)-2-thioxo-imidazolidin-1-yl]methyl]pyrrolidino]ethyl]-4-(4-hydroxybenzyl)-3-phenethyl-imidazolidine-2-thione
Show/Hide
|
C42H49N5O2S2
|
1
|
1 |
AC50 = 11490 nM
|
|
|
CP0907184
|
SID103076710
Show/Hide
|
C27H26F3N5O2
|
1
|
1 |
AC50 = 11490 nM
|
|
|
CP0857039
|
SID134215620
Show/Hide
|
C29H27F4N3O3
|
1
|
1 |
AC50 = 11500 nM
|
|
|
CP0890229
|
SID131411838
Show/Hide
|
C35H50ClN3O7S
|
1
|
1 |
AC50 = 11510 nM
|
|
|
CP0908906
|
SID85803063
Show/Hide
|
C30H35FN4O6S
|
1
|
1 |
AC50 = 11530 nM
|
|
|
CP0917909
|
SID131412853
Show/Hide
|
C35H44Cl3N3O6S
|
1
|
1 |
AC50 = 11530 nM
|
|
|
CP0875005
|
SID131410783
Show/Hide
|
C34H44F3N3O6S2
|
1
|
1 |
AC50 = 11540 nM
|
|
|
CP0966598
|
SID131413941
Show/Hide
|
C32H38N2O5S
|
1
|
1 |
AC50 = 11550 nM
|
|
|
CP0884585
|
SID87542072
Show/Hide
|
C37H47F3N4O5
|
1
|
1 |
AC50 = 11590 nM
|
|
|
CP0163339
|
1-(3-chlorophenyl)-3-(5-nitro-3-thienyl)urea
Show/Hide
|
C11H8ClN3O3S
|
1
|
1 |
AC50 = 11630 nM
|
|
|
CP0881129
|
SID87539725
Show/Hide
|
C36H46Cl2N4O5
|
1
|
1 |
AC50 = 11630 nM
|
|
|
CP0920033
|
SID134962092
Show/Hide
|
C32H36FN3O5S
|
1
|
1 |
AC50 = 11630 nM
|
|
|
CP0851520
|
SID131462082
Show/Hide
|
C30H32N4O3
|
1
|
1 |
AC50 = 11640 nM
|
|
|
CP0959685
|
SID131410712
Show/Hide
|
C36H52Cl2N4O5
|
1
|
1 |
AC50 = 11670 nM
|
|
|
CP0934882
|
SID85795185
Show/Hide
|
C30H42ClN3O5S
|
1
|
1 |
AC50 = 11680 nM
|
|
|
CP0920059
|
SID131412852
Show/Hide
|
C35H44Cl3N3O6S
|
1
|
1 |
AC50 = 11710 nM
|
|
|
CP0966601
|
SID131412470
Show/Hide
|
C42H52ClN5O7S
|
1
|
1 |
AC50 = 11710 nM
|
|
|
CP0882822
|
SID99360413
Show/Hide
|
C32H31ClF3N3O4S
|
1
|
1 |
AC50 = 11720 nM
|
|
|
CP0884589
|
SID17407962
Show/Hide
|
C28H28FN3O2S
|
1
|
1 |
AC50 = 11720 nM
|
|
|
CP0966825
|
SID85790285
Show/Hide
|
C33H38F3N3O4
|
1
|
1 |
AC50 = 11800 nM
|
|
|
CP0881123
|
SID87336743
Show/Hide
|
C33H43ClN4O4
|
1
|
1 |
AC50 = 11840 nM
|
|
|
CP0926403
|
SID87540438
Show/Hide
|
C36H46Cl2N4O5
|
1
|
1 |
AC50 = 11860 nM
|
|
|
CP0884596
|
SID85800281
Show/Hide
|
C30H41ClN4O6S
|
1
|
1 |
AC50 = 11870 nM
|
|
|
CP0201359
|
(2R,3R)-1-N,3-dimethyl-2-N-[(2R)-3-naphthalen-1-yl-2-[2-[3-(trifluoromethyl)phenyl]ethylamino]propyl]pentane-1,2-diamine
Show/Hide
|
C29H38F3N3
|
1
|
1 |
AC50 = 11930 nM
|
|
|
CP0900530
|
SID131409528
Show/Hide
|
C31H35F4N3O5S
|
1
|
1 |
AC50 = 11930 nM
|
|
|
CP0858468
|
SID131446406
Show/Hide
|
C26H21N3O3
|
1
|
1 |
AC50 = 11940 nM
|
|
|
CP0886262
|
SID85802394
Show/Hide
|
C32H37F3N4O7S
|
1
|
1 |
AC50 = 11940 nM
|
|
|
CP0907203
|
SID131411538
Show/Hide
|
C37H53F3N4O5
|
1
|
1 |
AC50 = 11970 nM
|
|
|
CP0933804
|
SID85805612
Show/Hide
|
C36H45F3N4O5
|
1
|
1 |
AC50 = 12020 nM
|
|
|
CP0338847
|
2-methoxy-6-[(E)-[(6-methoxy-2-methylquinolin-4-yl)hydrazinylidene]methyl]phenol
Show/Hide
|
C19H19N3O3
|
1
|
1 |
AC50 = 12050 nM
|
|
|
CP0851519
|
SID131462623
Show/Hide
|
C27H34N2O4S
|
1
|
1 |
AC50 = 12050 nM
|
|
|
CP0881167
|
SID49647702
Show/Hide
|
C32H31BrN4O2
|
1
|
1 |
AC50 = 12070 nM
|
|
|
CP0908687
|
SID104170445
Show/Hide
|
C37H45F3N4O6
|
1
|
1 |
AC50 = 12100 nM
|
|
|
CP0900335
|
SID864737
Show/Hide
|
C22H28N4O2S
|
1
|
1 |
AC50 = 12110 nM
|
|
|
CP0888205
|
SID49815767
Show/Hide
|
C34H33F6N5O5
|
1
|
1 |
AC50 = 12140 nM
|
|
|
CP0851518
|
SID87542164
Show/Hide
|
C37H47F3N4O5
|
1
|
1 |
AC50 = 12160 nM
|
|
|
CP0872441
|
SID85806897
Show/Hide
|
C36H41N3O6S
|
1
|
1 |
AC50 = 12160 nM
|
|
|
CP0907261
|
SID87543197
Show/Hide
|
C42H57Cl2N5O6
|
1
|
1 |
AC50 = 12190 nM
|
|
|
CP0920032
|
SID87341394
Show/Hide
|
C42H54N4O5
|
1
|
1 |
AC50 = 12190 nM
|
|
|
CP0932242
|
SID134215759
Show/Hide
|
C28H25ClF3N3O2
|
1
|
1 |
AC50 = 12260 nM
|
|
|
CP0884813
|
SID131461767
Show/Hide
|
C27H30N2O5S
|
1
|
1 |
AC50 = 12270 nM
|
|
|
CP0942506
|
SID131447112
Show/Hide
|
C26H19F2N3O2
|
1
|
1 |
AC50 = 12290 nM
|
|
|
CP0918115
|
SID144191412
Show/Hide
|
C31H35F3N2O3
|
1
|
1 |
AC50 = 12310 nM
|
|
|
CP0906207
|
SID131414088
Show/Hide
|
C32H38N2O5S
|
1
|
1 |
AC50 = 12330 nM
|
|
|
CP0944027
|
SID131460812
Show/Hide
|
C26H37N3O2
|
1
|
1 |
AC50 = 12340 nM
|
|
|
CP0883180
|
SID131462553
Show/Hide
|
C27H33FN2O3S
|
1
|
1 |
AC50 = 12360 nM
|
|
|
CP0856304
|
SID49681580
Show/Hide
|
C20H27N5O5
|
1
|
1 |
AC50 = 12410 nM
|
|
|
CP0874967
|
SID131463797
Show/Hide
|
C31H33N3O3
|
1
|
1 |
AC50 = 12480 nM
|
|
|
CP0908040
|
SID131411729
Show/Hide
|
C36H46Cl2N4O5
|
1
|
1 |
AC50 = 12480 nM
|
|
|
CP0907406
|
SID131426744
Show/Hide
|
C28H37N3O4S
|
1
|
1 |
AC50 = 12500 nM
|
|
|
CP0883671
|
SID85803790
Show/Hide
|
C34H48F3N5O6
|
1
|
1 |
AC50 = 12510 nM
|
|
|
CP0926626
|
SID85803973
Show/Hide
|
C31H35F3N4O6S
|
1
|
1 |
AC50 = 12600 nM
|
|
|
CP0411346
|
(E)-3-(4-chloranyl-3-nitro-phenyl)-N-[2-(4-methylpiperazin-1-yl)-5-piperidin-1-ylsulfonyl-phenyl]prop-2-enamide
Show/Hide
|
C25H30ClN5O5S
|
1
|
1 |
AC50 = 12620 nM
|
|
|
CP0920057
|
SID131447133
Show/Hide
|
C23H28N2O2
|
1
|
1 |
AC50 = 12690 nM
|
|
|
CP0883463
|
SID144194641
Show/Hide
|
C24H32N2O2
|
1
|
1 |
AC50 = 12740 nM
|
|
|
CP0327630
|
3-(4-fluorophenyl)-7,8-dimethoxy-5-[(4-methoxyphenyl)methyl]pyrazolo[4,3-c]quinoline
Show/Hide
|
C26H22FN3O3
|
1
|
1 |
AC50 = 12880 nM
|
|
|
CP0864588
|
SID131414872
Show/Hide
|
C27H35FN2O6S2
|
1
|
1 |
AC50 = 12890 nM
|
|
|
CP0189321
|
(2R)-2-(4-fluorobenzyl)hex-5-enoic acid [(2S)-2-[[(2R)-2-[2-[benzyl(2-hydroxyethyl)amino]-2-keto-ethyl]pent-4-enoyl]amino]-3-(1H-indol-3-yl)propyl] ester
Show/Hide
|
C40H46FN3O5
|
1
|
1 |
AC50 = 12940 nM
|
|
|
CP0864550
|
SID24794864
Show/Hide
|
C23H22N2O6S
|
1
|
1 |
AC50 = 12960 nM
|
|
|
CP0912920
|
SID87542115
Show/Hide
|
C35H52FN3O6S
|
1
|
1 |
AC50 = 12970 nM
|
|
|
CP0885768
|
SID131409577
Show/Hide
|
C33H35F6N5O5
|
1
|
1 |
AC50 = 12990 nM
|
|
|
CP0395983
|
2-[4-[2-(4-methoxyphenyl)-1-benzothiophen-3-yl]phenoxy]-N,N-dimethyl-ethanamine
Show/Hide
|
C25H25NO2S
|
1
|
1 |
AC50 = 13010 nM
|
|
|
CP0897524
|
SID99495630
Show/Hide
|
C20H26F3N3O9S
|
1
|
1 |
AC50 = 13040 nM
|
|
|
CP0857043
|
SID131409422
Show/Hide
|
C31H33F4N5O5
|
1
|
1 |
AC50 = 13100 nM
|
|
|
CP0883153
|
SID131411726
Show/Hide
|
C36H46Cl2N4O5
|
1
|
1 |
AC50 = 13100 nM
|
|
|
CP0926627
|
SID131414844
Show/Hide
|
C31H31FN2O7S
|
1
|
1 |
AC50 = 13160 nM
|
|
|
CP0916972
|
SID131442607
Show/Hide
|
C30H30F3N3O5
|
1
|
1 |
AC50 = 13190 nM
|
|
|
CP0966603
|
SID131464629
Show/Hide
|
C30H35N3O3
|
1
|
1 |
AC50 = 13210 nM
|
|
|
CP0930550
|
SID85805840
Show/Hide
|
C35H41N5O5
|
1
|
1 |
AC50 = 13220 nM
|
|
|
CP0857096
|
SID87542551
Show/Hide
|
C31H35Cl2FN4O4
|
1
|
1 |
AC50 = 13240 nM
|
|
|
CP0938693
|
SID144191046
Show/Hide
|
C25H21F4N3O
|
1
|
1 |
AC50 = 13240 nM
|
|
|
CP0851437
|
SID87542238
Show/Hide
|
C37H48F3N3O6S
|
1
|
1 |
AC50 = 13270 nM
|
|
|
CP0886463
|
SID131435469
Show/Hide
|
C27H34N2O5S
|
1
|
1 |
AC50 = 13290 nM
|
|
|
CP0907200
|
SID131443346
Show/Hide
|
C34H33N3O5
|
1
|
1 |
AC50 = 13300 nM
|
|
|
CP0897525
|
SID87218868
Show/Hide
|
C31H37Cl2N3O5S
|
1
|
1 |
AC50 = 13310 nM
|
|
|
CP0944787
|
SID131455689
Show/Hide
|
C29H37ClN2O6S
|
1
|
1 |
AC50 = 13340 nM
|
|
|
CP0947079
|
SID131447493
Show/Hide
|
C25H23FN2O2
|
1
|
1 |
AC50 = 13390 nM
|
|
|
CP0942501
|
SID131411590
Show/Hide
|
C35H45Cl2N3O6S
|
1
|
1 |
AC50 = 13420 nM
|
|
|
CP0480152
|
4-amyl-8-[1-(1,3-benzodioxol-5-yl)-3-piperidino-propyl]-5,7-dimethoxy-coumarin
Show/Hide
|
C31H39NO6
|
1
|
1 |
AC50 = 13440 nM
|
|
|
CP0942610
|
SID131456879
Show/Hide
|
C25H28Cl3N3O5
|
1
|
1 |
AC50 = 13480 nM
|
|
|
CP0864557
|
SID131414686
Show/Hide
|
C30H36N2O7S
|
1
|
1 |
AC50 = 13500 nM
|
|
|
CP0864699
|
SID131411913
Show/Hide
|
C37H47F3N4O5
|
1
|
1 |
AC50 = 13550 nM
|
|
|
CP0682046
|
SID24793277
Show/Hide
|
C18H14FN5O3S
|
1
|
1 |
AC50 = 13570 nM
|
|
|
CP0858467
|
SID131461831
Show/Hide
|
C25H25FN2O3S
|
1
|
1 |
AC50 = 13590 nM
|
|
|
CP0900331
|
SID131411673
Show/Hide
|
C36H46F3N5O5
|
1
|
1 |
AC50 = 13610 nM
|
|
|
CP0912950
|
SID85805294
Show/Hide
|
C29H32Cl3N3O5S
|
1
|
1 |
AC50 = 13650 nM
|
|
|
CP0909152
|
SID144194180
Show/Hide
|
C26H27N3O3
|
1
|
1 |
AC50 = 13680 nM
|
|
|
CP0890228
|
SID134961984
Show/Hide
|
C32H36FN3O5S
|
1
|
1 |
AC50 = 13720 nM
|
|
|
CP0966617
|
SID144194181
Show/Hide
|
C24H21F2N3O
|
1
|
1 |
AC50 = 13840 nM
|
|
|
CP0864734
|
SID85793709
Show/Hide
|
C32H37F3N4O5
|
1
|
1 |
AC50 = 13860 nM
|
|
|
CP0881110
|
SID131411937
Show/Hide
|
C36H45Cl2N3O5
|
1
|
1 |
AC50 = 13970 nM
|
|
|
CP0225799
|
6-phenyl-2-(2-pyridinyl)-3H-thieno[2,3-d]pyrimidin-4-one
Show/Hide
|
C17H11N3OS
|
1
|
1 |
AC50 = 13990 nM
|
|
|
CP0377375
|
4-mesyl-3-nitro-benzoic acid [2-keto-2-(2-thenylamino)ethyl] ester
Show/Hide
|
C15H14N2O7S2
|
1
|
1 |
AC50 = 14030 nM
|
|
|
CP0966821
|
SID87541724
Show/Hide
|
C37H48Cl2N4O6
|
1
|
1 |
AC50 = 14140 nM
|
|
|
CP0908894
|
SID144194916
Show/Hide
|
C26H32N2O3
|
1
|
1 |
AC50 = 14150 nM
|
|
|
CP0966621
|
SID87540704
Show/Hide
|
C35H46F3N5O8S
|
1
|
1 |
AC50 = 14190 nM
|
|
|
CP0900435
|
SID87541199
Show/Hide
|
C36H54N4O5
|
1
|
1 |
AC50 = 14220 nM
|
|
|
CP0912657
|
SID22407366
Show/Hide
|
C18H15ClN2O4
|
1
|
1 |
AC50 = 14240 nM
|
|
|
CP0333050
|
2-fluoranyl-5-nitro-N-(12-oxidanylidene-7,8,9,10-tetrahydro-6H-azepino[2,1-b]quinazolin-2-yl)benzamide
Show/Hide
|
C20H17FN4O4
|
1
|
1 |
AC50 = 14260 nM
|
|
|
CP0912637
|
SID104170518
Show/Hide
|
C38H47F3N4O7
|
1
|
1 |
AC50 = 14280 nM
|
|
|
CP0669270
|
SID24841640
Show/Hide
|
C29H35F3N2O4
|
1
|
1 |
AC50 = 14320 nM
|
|
|
CP0897519
|
SID131426745
Show/Hide
|
C28H37N3O4S
|
1
|
1 |
AC50 = 14390 nM
|
|
|
CP0465243
|
(2R,3R)-2-N-[(2S)-2-[(4-tert-butylcyclohexyl)methylamino]pentyl]-1-N,3-dimethylpentane-1,2-diamine
Show/Hide
|
C23H49N3
|
1
|
1 |
AC50 = 14410 nM
|
|
|
CP0897522
|
SID131413665
Show/Hide
|
C28H38N2O7S2
|
1
|
1 |
AC50 = 14470 nM
|
|
|
CP0875019
|
SID131460391
Show/Hide
|
C27H35N3O3
|
1
|
1 |
AC50 = 14480 nM
|
|
|
CP0947080
|
SID131414853
Show/Hide
|
C27H35FN2O6S2
|
1
|
1 |
AC50 = 14480 nM
|
|
|
CP0931529
|
SID87540185
Show/Hide
|
C37H56N4O6
|
1
|
1 |
AC50 = 14490 nM
|
|
|
CP0897060
|
SID131409384
Show/Hide
|
C37H48N4O4
|
1
|
1 |
AC50 = 14500 nM
|
|
|
CP0749665
|
SID22409699
Show/Hide
|
C23H19NO6
|
1
|
1 |
AC50 = 14510 nM
|
|
|
CP0906227
|
SID87457183
Show/Hide
|
C38H47F3N4O7
|
1
|
1 |
AC50 = 14550 nM
|
|
|
CP0856617
|
SID131461915
Show/Hide
|
C28H36N2O4S
|
1
|
1 |
AC50 = 14600 nM
|
|
|
CP0926624
|
SID131464628
Show/Hide
|
C30H35N3O3
|
1
|
1 |
AC50 = 14610 nM
|
|
|
CP0875017
|
SID87541900
Show/Hide
|
C38H49F3N4O6
|
1
|
1 |
AC50 = 14630 nM
|
|
|
CP0860343
|
SID85800737
Show/Hide
|
C35H36F3N5O5
|
1
|
1 |
AC50 = 14650 nM
|
|
|
CP0250533
|
1-[3-(diethylsulfamoyl)phenyl]-3-[3-(trifluoromethyl)phenyl]urea
Show/Hide
|
C18H20F3N3O3S
|
1
|
1 |
AC50 = 14860 nM
|
|
|
CP0959686
|
SID131464906
Show/Hide
|
C31H33N3O3
|
1
|
1 |
AC50 = 14870 nM
|
|
|
CP0881128
|
SID85200562
Show/Hide
|
C36H41FN2O5
|
1
|
1 |
AC50 = 14980 nM
|
|
|
CP0902496
|
SID131455760
Show/Hide
|
C29H38N2O5
|
1
|
1 |
AC50 = 14990 nM
|
|
|
CP0864554
|
SID131446407
Show/Hide
|
C26H21N3O3
|
1
|
1 |
AC50 = 15010 nM
|
|
|
CP0094831
|
5-[(2,3-dimethylanilino)methyl]-8-quinolinol
Show/Hide
|
C18H18N2O
|
1
|
1 |
AC50 = 15050 nM
|
|
|
CP0856555
|
SID85148905
Show/Hide
|
C31H31FN2O4
|
1
|
1 |
AC50 = 15130 nM
|
|
|
CP0933806
|
SID85798985
Show/Hide
|
C30H33F4N3O5S
|
1
|
1 |
AC50 = 15310 nM
|
|
|
CP0890231
|
SID87336011
Show/Hide
|
C27H21BrN4O2S
|
1
|
1 |
AC50 = 15390 nM
|
|
|
CP0884820
|
SID131446311
Show/Hide
|
C21H23N3OS
|
1
|
1 |
AC50 = 15430 nM
|
|
|
CP0957471
|
SID131464464
Show/Hide
|
C30H30FN3O2
|
1
|
1 |
AC50 = 15440 nM
|
|
|
CP0843536
|
SID22408552
Show/Hide
|
C18H14F2N4O4S
|
1
|
1 |
AC50 = 15460 nM
|
|
|
CP0856875
|
SID22408067
Show/Hide
|
C29H24ClN5O2S
|
1
|
1 |
AC50 = 15510 nM
|
|
|
CP0808238
|
SID49728465
Show/Hide
|
C14H13N3O2
|
1
|
1 |
AC50 = 15530 nM
|
|
|
CP0950481
|
SID131464394
Show/Hide
|
C31H32FN3O3
|
1
|
1 |
AC50 = 15530 nM
|
|
|
CP0912232
|
SID131412025
Show/Hide
|
C35H44Cl2FN3O6S
|
1
|
1 |
AC50 = 15560 nM
|
|
|
CP0247729
|
(8R)-3-[3-[2-(4-chloranylphenoxy)ethanoylamino]phenyl]-7-(2,2-diphenylethanoyl)-1-oxa-2,7-diazaspiro[4.4]non-2-ene-8-carboxamide
Show/Hide
|
C35H31ClN4O5
|
1
|
1 |
AC50 = 15700 nM
|
|
|
CP0907409
|
SID85792388
Show/Hide
|
C35H39N3O6S
|
1
|
1 |
AC50 = 15720 nM
|
|
|
CP0796027
|
SID24817667
Show/Hide
|
C16H12F3NO4
|
1
|
1 |
AC50 = 15810 nM
|
|
|
CP0942499
|
SID104170643
Show/Hide
|
C35H50ClN3O7S
|
1
|
1 |
AC50 = 15830 nM
|
|
|
CP0851535
|
SID131443481
Show/Hide
|
C30H30F3N3O5
|
1
|
1 |
AC50 = 15880 nM
|
|
|
CP0883461
|
SID134961958
Show/Hide
|
C30H36N2O6S
|
1
|
1 |
AC50 = 15900 nM
|
|
|
CP0952613
|
SID131414047
Show/Hide
|
C32H38N2O5S
|
1
|
1 |
AC50 = 15910 nM
|
|
|
CP0886570
|
SID85200367
Show/Hide
|
C38H49N3O7
|
1
|
1 |
AC50 = 15940 nM
|
|
|
CP0959677
|
SID131442684
Show/Hide
|
C28H29FN2O7S
|
1
|
1 |
AC50 = 16090 nM
|
|
|
CP0886574
|
SID85808340
Show/Hide
|
C31H35Cl2FN4O4
|
1
|
1 |
AC50 = 16220 nM
|
|
|
CP0906228
|
SID131415229
Show/Hide
|
C27H36N2O4S
|
1
|
1 |
AC50 = 16230 nM
|
|
|
CP0908720
|
SID87218838
Show/Hide
|
C31H37Cl2N3O6S
|
1
|
1 |
AC50 = 16250 nM
|
|
|
CP0792292
|
SID22409409
Show/Hide
|
C25H26F2N4O3S3
|
1
|
1 |
AC50 = 16380 nM
|
|
|
CP0882376
|
SID131433975
Show/Hide
|
C37H46N4O4
|
1
|
1 |
AC50 = 16420 nM
|
|
|
CP0898773
|
SID87543997
Show/Hide
|
C36H44ClF3N4O7S
|
1
|
1 |
AC50 = 16430 nM
|
|
|
CP0912293
|
SID131426756
Show/Hide
|
C29H37N3O5S
|
1
|
1 |
AC50 = 16530 nM
|
|
|
CP0864528
|
SID87541674
Show/Hide
|
C33H43N5O4
|
1
|
1 |
AC50 = 16620 nM
|
|
|
CP0926619
|
SID87539854
Show/Hide
|
C37H51N3O7S
|
1
|
1 |
AC50 = 16770 nM
|
|
|
CP0944025
|
SID131464703
Show/Hide
|
C30H31N3O2
|
1
|
1 |
AC50 = 16770 nM
|
|
|
CP0915292
|
SID92763382
Show/Hide
|
C18H19N3O3
|
1
|
1 |
AC50 = 16820 nM
|
|
|
CP0317486
|
4-[(Z)-[4-(4-chlorobenzyl)-3-keto-1,4-benzoxazin-2-ylidene]methyl]-N-[3-(4-methylpiperazino)propyl]benzamide
Show/Hide
|
C31H33ClN4O3
|
1
|
1 |
AC50 = 16940 nM
|
|
|
CP0966618
|
SID144200016
Show/Hide
|
C39H43N3O4
|
1
|
1 |
AC50 = 17070 nM
|
|
|
CP0907224
|
SID131411973
Show/Hide
|
C36H44F3N5O6
|
1
|
1 |
AC50 = 17090 nM
|
|
|
CP0912955
|
SID144190760
Show/Hide
|
C24H28FN3O
|
1
|
1 |
AC50 = 17150 nM
|
|
|
CP0965787
|
SID87539852
Show/Hide
|
C35H46FN3O6S
|
1
|
1 |
AC50 = 17150 nM
|
|
|
CP0876047
|
SID134215622
Show/Hide
|
C26H25F6N3O2
|
1
|
1 |
AC50 = 17160 nM
|
|
|
CP0188285
|
5-chloranyl-2-ethylsulfonyl-N-(4-methylphenyl)pyrimidine-4-carboxamide
Show/Hide
|
C14H14ClN3O3S
|
1
|
1 |
AC50 = 17170 nM
|
|
|
CP0944761
|
SID131456897
Show/Hide
|
C29H31FN2O6S
|
1
|
1 |
AC50 = 17190 nM
|
|
|
CP0795376
|
SID24797727
Show/Hide
|
C23H22Cl3N3O2
|
1
|
1 |
AC50 = 17210 nM
|
|
|
CP0917910
|
SID17516817
Show/Hide
|
C15H13N3
|
1
|
1 |
AC50 = 17250 nM
|
|
|
CP0944780
|
SID131411247
Show/Hide
|
C38H47F3N4O7
|
1
|
1 |
AC50 = 17250 nM
|
|
|
CP0926623
|
SID131446622
Show/Hide
|
C25H21FN2O2
|
1
|
1 |
AC50 = 17270 nM
|
|
|
CP0926616
|
SID131409583
Show/Hide
|
C36H41N3O5S
|
1
|
1 |
AC50 = 17430 nM
|
|
|
CP0413988
|
MLS000709318
Show/Hide
|
C26H28BrN3O3
|
1
|
1 |
AC50 = 17440 nM
|
|
|
CP0885553
|
SID131443063
Show/Hide
|
C29H27ClF3N3O5
|
1
|
1 |
AC50 = 17500 nM
|
|
|
CP0912663
|
SID131411589
Show/Hide
|
C35H45Cl2N3O6S
|
1
|
1 |
AC50 = 17530 nM
|
|
|
CP0897516
|
SID131461419
Show/Hide
|
C26H29N3O2
|
1
|
1 |
AC50 = 17780 nM
|
|
|
CP0875020
|
SID131410499
Show/Hide
|
C34H45F3N6O7S
|
1
|
1 |
AC50 = 17860 nM
|
|
|
CP0856926
|
2-piperidyl-[2-(trifluoromethyl)-6-[4-(trifluoromethyl)phenyl]-4-pyridyl]methanol
Show/Hide
|
C19H18F6N2O
|
1
|
1 |
AC50 = 17890 nM
|
|
|
CP0515974
|
MLS001214907
Show/Hide
|
C20H26N4O2
|
1
|
1 |
AC50 = 18080 nM
|
|
|
CP0889300
|
SID85148967
Show/Hide
|
C32H30FN3O4
|
1
|
1 |
AC50 = 18200 nM
|
|
|
CP0886581
|
SID85804015
Show/Hide
|
C33H36N4O6S2
|
1
|
1 |
AC50 = 18260 nM
|
|
|
CP0887141
|
SID144191105
Show/Hide
|
C24H20F2N2O
|
1
|
1 |
AC50 = 18320 nM
|
|
|
CP0917911
|
SID85809182
Show/Hide
|
C31H35Cl2FN4O4
|
1
|
1 |
AC50 = 18400 nM
|
|
|
CP0864732
|
SID85798995
Show/Hide
|
C35H38N4O6
|
1
|
1 |
AC50 = 18490 nM
|
|
|
CP0945690
|
SID131463815
Show/Hide
|
C30H30FN3O2
|
1
|
1 |
AC50 = 18690 nM
|
|
|
CP0897062
|
SID131433146
Show/Hide
|
C31H35N5O4S
|
1
|
1 |
AC50 = 18850 nM
|
|
|
CP0897513
|
SID87542144
Show/Hide
|
C37H48F3N3O7S
|
1
|
1 |
AC50 = 18910 nM
|
|
|
CP0299409
|
2-cyclobutyl-6,7-dimethoxy-4-[4-(2-methoxyphenyl)-1-piperazinyl]quinazoline
Show/Hide
|
C25H30N4O3
|
1
|
1 |
AC50 = 18920 nM
|
|
|
CP0908029
|
SID87542557
Show/Hide
|
C34H41N3O4
|
1
|
1 |
AC50 = 18920 nM
|
|
|
CP0959682
|
SID87543782
Show/Hide
|
C37H47F3N4O5
|
1
|
1 |
AC50 = 19020 nM
|
|
|
CP0874987
|
SID92764858
Show/Hide
|
C30H37ClN2O4
|
1
|
1 |
AC50 = 19060 nM
|
|
|
CP0862115
|
SID49714947
Show/Hide
|
C24H35N3O5S
|
1
|
1 |
AC50 = 19070 nM
|
|
|
CP0906208
|
SID131462323
Show/Hide
|
C26H31FN2O2
|
1
|
1 |
AC50 = 19090 nM
|
|
|
CP0944778
|
SID85798450
Show/Hide
|
C31H39N3O4
|
1
|
1 |
AC50 = 19090 nM
|
|
|
CP0950775
|
SID131412010
Show/Hide
|
C37H46F3N3O5
|
1
|
1 |
AC50 = 19110 nM
|
|
|
CP0912660
|
SID131434297
Show/Hide
|
C32H36FN3O5S
|
1
|
1 |
AC50 = 19230 nM
|
|
|
CP0897521
|
SID131415135
Show/Hide
|
C29H38N2O6S
|
1
|
1 |
AC50 = 19290 nM
|
|
|
CP0965722
|
SID85802367
Show/Hide
|
C32H38F3N3O6S
|
1
|
1 |
AC50 = 19300 nM
|
|
|
CP0917908
|
SID131412196
Show/Hide
|
C36H47N3O7S
|
1
|
1 |
AC50 = 19370 nM
|
|
|
CP0916974
|
SID144191280
Show/Hide
|
C24H21F2N3O
|
1
|
1 |
AC50 = 19500 nM
|
|
|
CP0885786
|
SID22410812
Show/Hide
|
C22H25N3O3S
|
1
|
1 |
AC50 = 19510 nM
|
|
|
CP0872443
|
SID131447174
Show/Hide
|
C26H24N2O3
|
1
|
1 |
AC50 = 19540 nM
|
|
|
CP0884811
|
SID131462446
Show/Hide
|
C29H32FN3O2
|
1
|
1 |
AC50 = 19550 nM
|
|
|
CP0864530
|
SID87544008
Show/Hide
|
C35H53N3O6S
|
1
|
1 |
AC50 = 19600 nM
|
|
|
CP0881160
|
SID131436519
Show/Hide
|
C23H31Cl2N5O3
|
1
|
1 |
AC50 = 19680 nM
|
|
|
CP0942504
|
SID144195125
Show/Hide
|
C27H32N4O2
|
1
|
1 |
AC50 = 19880 nM
|
|
|
CP0875013
|
SID17510268
Show/Hide
|
C22H19F2N3O5
|
1
|
1 |
AC50 = 20040 nM
|
|
|
CP0907786
|
SID87542119
Show/Hide
|
C35H53N3O6S
|
1
|
1 |
AC50 = 20100 nM
|
|
|
CP0881651
|
SID87540041
Show/Hide
|
C38H49F3N4O6
|
1
|
1 |
AC50 = 20130 nM
|
|
|
CP0941617
|
SID144190635
Show/Hide
|
C27H26N2O2
|
1
|
1 |
AC50 = 20210 nM
|
|
|
CP0865530
|
SID87539628
Show/Hide
|
C31H43FN4O4
|
1
|
1 |
AC50 = 20350 nM
|
|
|
CP0725828
|
SID104222616
Show/Hide
|
C19H24N6O4
|
1
|
1 |
AC50 = 20370 nM
|
|
|
CP0912664
|
SID131462383
Show/Hide
|
C27H34N2O3S
|
1
|
1 |
AC50 = 20540 nM
|
|
|
CP0864730
|
SID144194942
Show/Hide
|
C26H26FN3O2
|
1
|
1 |
AC50 = 20770 nM
|
|
|
CP0050781
|
5'-(N-ethyl-N-isopropyl)amiloride
Show/Hide
|
C11H18ClN7O
|
1
|
1 |
AC50 = 20940 nM
|
|
|
CP0864701
|
SID87540866
Show/Hide
|
C37H49N3O8S
|
1
|
1 |
AC50 = 20980 nM
|
|
|
CP0957473
|
SID131464559
Show/Hide
|
C28H29F2N3O2
|
1
|
1 |
AC50 = 21080 nM
|
|
|
CP0950776
|
SID121286619
Show/Hide
|
C12H14N6O
|
1
|
1 |
AC50 = 21250 nM
|
|
|
CP0900537
|
SID131463065
Show/Hide
|
C28H29F2N3O2
|
1
|
1 |
AC50 = 21330 nM
|
|
|
CP0909795
|
SID85810294
Show/Hide
|
C30H36FN3O7S2
|
1
|
1 |
AC50 = 21500 nM
|
|
|
CP0846198
|
SID131463369
Show/Hide
|
C28H37N3O2
|
1
|
1 |
AC50 = 21580 nM
|
|
|
CP0912948
|
SID144191277
Show/Hide
|
C27H24F3N3O
|
1
|
1 |
AC50 = 21680 nM
|
|
|
CP0926609
|
SID103050537
Show/Hide
|
C14H14N2O3
|
1
|
1 |
AC50 = 21680 nM
|
|
|
CP0885878
|
SID131411759
Show/Hide
|
C37H49FN4O6
|
1
|
1 |
AC50 = 21700 nM
|
|
|
CP0934874
|
SID131464017
Show/Hide
|
C29H32FN3O2
|
1
|
1 |
AC50 = 21730 nM
|
|
|
CP0881647
|
SID131411777
Show/Hide
|
C37H47FN4O7
|
1
|
1 |
AC50 = 21950 nM
|
|
|
CP0856620
|
SID103158992
Show/Hide
|
C25H27ClN2O4S
|
1
|
1 |
AC50 = 22000 nM
|
|
|
CP0886260
|
SID85795421
Show/Hide
|
C32H37F3N4O5
|
1
|
1 |
AC50 = 22030 nM
|
|
|
CP0890074
|
SID99357780
Show/Hide
|
C29H39N5O4
|
1
|
1 |
AC50 = 22090 nM
|
|
|
CP0856621
|
SID85797502
Show/Hide
|
C31H43F3N4O5
|
1
|
1 |
AC50 = 22150 nM
|
|
|
CP0908122
|
SID131446879
Show/Hide
|
C23H24FN3O2
|
1
|
1 |
AC50 = 22200 nM
|
|
|
CP0907624
|
SID85797915
Show/Hide
|
C30H33F4N3O5S
|
1
|
1 |
AC50 = 22240 nM
|
|
|
CP0907264
|
SID85807330
Show/Hide
|
C36H40N4O4
|
1
|
1 |
AC50 = 22340 nM
|
|
|
CP0851533
|
SID144191045
Show/Hide
|
C25H21F4N3O
|
1
|
1 |
AC50 = 22380 nM
|
|
|
CP0865946
|
SID131463399
Show/Hide
|
C26H31FN2O3S
|
1
|
1 |
AC50 = 22430 nM
|
|
|
CP0881166
|
SID131464730
Show/Hide
|
C28H30FN3O2
|
1
|
1 |
AC50 = 22580 nM
|
|
|
CP0882636
|
SID144194129
Show/Hide
|
C26H25N3O
|
1
|
1 |
AC50 = 22600 nM
|
|
|
CP0857097
|
SID131433184
Show/Hide
|
C30H35N3O4
|
1
|
1 |
AC50 = 22620 nM
|
|
|
CP0830716
|
SID162403654
Show/Hide
|
C19H26N6S
|
1
|
1 |
AC50 = 22930 nM
|
|
|
CP0682595
|
SID24794939
Show/Hide
|
C15H11NO2S
|
1
|
1 |
AC50 = 23070 nM
|
|
|
CP0950310
|
SID49734954
Show/Hide
|
C22H28FN3O2S
|
1
|
1 |
AC50 = 23070 nM
|
|
|
CP0886272
|
SID87541988
Show/Hide
|
C33H47F3N4O5
|
1
|
1 |
AC50 = 23100 nM
|
|
|
CP0900332
|
SID131426785
Show/Hide
|
C28H37FN2O4S
|
1
|
1 |
AC50 = 23130 nM
|
|
|
CP0941619
|
SID131464911
Show/Hide
|
C31H33N3O3
|
1
|
1 |
AC50 = 23160 nM
|
|
|
CP0885906
|
SID144194091
Show/Hide
|
C30H28N2O3S
|
1
|
1 |
AC50 = 23330 nM
|
|
|
CP0885649
|
SID144194192
Show/Hide
|
C24H22F2N2
|
1
|
1 |
AC50 = 23430 nM
|
|
|
CP0873977
|
SID85809622
Show/Hide
|
C38H44N4O6
|
1
|
1 |
AC50 = 23460 nM
|
|
|
CP0945142
|
SID131455649
Show/Hide
|
C25H30ClFN2O4
|
1
|
1 |
AC50 = 23690 nM
|
|
|
CP0934877
|
SID131455688
Show/Hide
|
C29H37ClN2O6S
|
1
|
1 |
AC50 = 23730 nM
|
|
|
CP0687288
|
SID24790402
Show/Hide
|
C23H22N2O6S
|
1
|
1 |
AC50 = 23900 nM
|
|
|
CP0908900
|
SID134962299
Show/Hide
|
C35H48N4O4S
|
1
|
1 |
AC50 = 24020 nM
|
|
|
CP0944041
|
SID144194765
Show/Hide
|
C27H28N2O3
|
1
|
1 |
AC50 = 24250 nM
|
|
|
CP0966600
|
SID134962114
Show/Hide
|
C33H37FN4O4
|
1
|
1 |
AC50 = 24570 nM
|
|
|
CP0882534
|
SID85804092
Show/Hide
|
C37H43N3O6S
|
1
|
1 |
AC50 = 24610 nM
|
|
|
CP0335726
|
3-bromanyl-N-[(2S)-1-[(3R,6R)-6-[(4-hydroxyphenyl)methyl]-3-(phenylmethyl)-2,3,5,6-tetrahydroimidazo[1,2-a]imidazol-7-yl]propan-2-yl]-4-methyl-benzamide
Show/Hide
|
C30H33BrN4O2
|
1
|
1 |
AC50 = 24790 nM
|
|
|
CP0857492
|
SID124754940
Show/Hide
|
C26H31F3N2O4
|
1
|
1 |
AC50 = 24930 nM
|
|
|
CP0938690
|
SID144199873
Show/Hide
|
C39H43N3O3
|
1
|
1 |
AC50 = 24940 nM
|
|
|
CP0966631
|
SID104170827
Show/Hide
|
C34H44F3N3O6S2
|
1
|
1 |
AC50 = 25210 nM
|
|
|
CP0857032
|
SID131414805
Show/Hide
|
C23H34N2O4S
|
1
|
1 |
AC50 = 25270 nM
|
|
|
CP0857854
|
SID85808600
Show/Hide
|
C30H36FN3O7S2
|
1
|
1 |
AC50 = 25300 nM
|
|
|
CP0887142
|
SID85807332
Show/Hide
|
C38H44N4O6
|
1
|
1 |
AC50 = 25300 nM
|
|
|
CP0919691
|
SID131433185
Show/Hide
|
C30H35N3O4
|
1
|
1 |
AC50 = 25340 nM
|
|
|
CP0720195
|
SID17432349
Show/Hide
|
C23H21ClN4O2S
|
1
|
1 |
AC50 = 25410 nM
|
|
|
CP0900523
|
SID131412250
Show/Hide
|
C36H45Cl2FN4O5
|
1
|
1 |
AC50 = 25910 nM
|
|
|
CP0897509
|
SID87540527
Show/Hide
|
C34H41N3O4
|
1
|
1 |
AC50 = 26080 nM
|
|
|
CP0699276
|
SID17515351
Show/Hide
|
C20H21N3O3S
|
1
|
1 |
AC50 = 26330 nM
|
|
|
CP0864692
|
SID85794270
Show/Hide
|
C35H38N4O6
|
1
|
1 |
AC50 = 26460 nM
|
|
|
CP0912654
|
SID131442875
Show/Hide
|
C25H28F3N3O6
|
1
|
1 |
AC50 = 26610 nM
|
|
|
CP0917915
|
SID134215760
Show/Hide
|
C28H25F4N3O2
|
1
|
1 |
AC50 = 26790 nM
|
|
|
CP0652494
|
SID17508683
Show/Hide
|
C24H20N4O2
|
1
|
1 |
AC50 = 26910 nM
|
|
|
CP0881644
|
SID24810201
Show/Hide
|
C15H10BrF3N2O3
|
1
|
1 |
AC50 = 27110 nM
|
|
|
CP0860506
|
SID85808205
Show/Hide
|
C36H40FN3O5S
|
1
|
1 |
AC50 = 27140 nM
|
|
|
CP0959684
|
SID85798007
Show/Hide
|
C30H36F3N5O5
|
1
|
1 |
AC50 = 27530 nM
|
|
|
CP0908692
|
SID87543362
Show/Hide
|
C30H42F3N3O7S2
|
1
|
1 |
AC50 = 27610 nM
|
|
|
CP0906224
|
SID131456584
Show/Hide
|
C26H30F4N2O4
|
1
|
1 |
AC50 = 27850 nM
|
|
|
CP0860340
|
SID131461119
Show/Hide
|
C24H27FN2O3S
|
1
|
1 |
AC50 = 28240 nM
|
|
|
CP0906903
|
SID131433048
Show/Hide
|
C33H42N4O4
|
1
|
1 |
AC50 = 28670 nM
|
|
|
CP0930589
|
SID131462384
Show/Hide
|
C27H34N2O3S
|
1
|
1 |
AC50 = 29220 nM
|
|
|
CP0865831
|
SID131434027
Show/Hide
|
C33H41N3O4
|
1
|
1 |
AC50 = 29510 nM
|
|
|
CP0908090
|
SID85797706
Show/Hide
|
C31H37N3O6S
|
1
|
1 |
AC50 = 29810 nM
|
|
|
CP0917914
|
SID131433084
Show/Hide
|
C33H43N5O4
|
1
|
1 |
AC50 = 30080 nM
|
|
|
CP0915293
|
SID85811561
Show/Hide
|
C32H37F3N4O6S
|
1
|
1 |
AC50 = 30380 nM
|
|
|
CP0876611
|
SID85804575
Show/Hide
|
C37H48N4O4
|
1
|
1 |
AC50 = 30600 nM
|
|
|
CP0885644
|
SID144191081
Show/Hide
|
C25H24FN3O
|
1
|
1 |
AC50 = 30740 nM
|
|
|
CP0882823
|
SID131411300
Show/Hide
|
C38H50N4O7
|
1
|
1 |
AC50 = 30950 nM
|
|
|
CP0926610
|
SID85804608
Show/Hide
|
C32H44N4O6
|
1
|
1 |
AC50 = 31180 nM
|
|
|
CP0884812
|
SID99359766
Show/Hide
|
C33H39N5O12S
|
1
|
1 |
AC50 = 31850 nM
|
|
|
CP0883206
|
SID131463507
Show/Hide
|
C27H29FN4O2
|
1
|
1 |
AC50 = 32200 nM
|
|
|
CP0908579
|
SID131433087
Show/Hide
|
C33H43N5O4
|
1
|
1 |
AC50 = 32880 nM
|
|
|
CP0908640
|
SID22402793
Show/Hide
|
C20H21F3N2S
|
1
|
1 |
AC50 = 33180 nM
|
|
|
CP0926611
|
SID85792258
Show/Hide
|
C34H46N4O5
|
1
|
1 |
AC50 = 33510 nM
|
|
|
CP0862108
|
SID131462424
Show/Hide
|
C27H29FN2O3S
|
1
|
1 |
AC50 = 33650 nM
|
|
|
CP0912241
|
SID131455664
Show/Hide
|
C25H37FN2O4
|
1
|
1 |
AC50 = 33960 nM
|
|
|
CP0952082
|
SID131442813
Show/Hide
|
C33H36N2O7
|
1
|
1 |
AC50 = 34260 nM
|
|
|
CP0966894
|
SID22409430
Show/Hide
|
C21H20Cl2N4O3S3
|
1
|
1 |
AC50 = 34850 nM
|
|
|
CP0906235
|
SID131464289
Show/Hide
|
C24H28F4N2O
|
1
|
1 |
AC50 = 34890 nM
|
|
|
CP0851521
|
SID85809458
Show/Hide
|
C29H34ClN3O7S2
|
1
|
1 |
AC50 = 35510 nM
|
|
|
CP0679569
|
SID17509398
Show/Hide
|
C22H20BrN5O
|
1
|
1 |
AC50 = 35760 nM
|
|
|
CP0862101
|
SID17510315
Show/Hide
|
C27H29FN4O3
|
1
|
1 |
AC50 = 35830 nM
|
|
|
CP0736361
|
SID4242957
Show/Hide
|
C18H21N5O2
|
1
|
1 |
AC50 = 36060 nM
|
|
|
CP0947579
|
SID17510497
Show/Hide
|
C21H27N5O
|
1
|
1 |
AC50 = 37150 nM
|
|
|
CP0944748
|
SID131460627
Show/Hide
|
C27H27N3O4S
|
1
|
1 |
AC50 = 38090 nM
|
|
|
CP0465767
|
(6E)-4-ethyl-3-hydroxy-6-[5-methyl-4-(1-methyl-2-benzimidazolyl)-1,2-dihydropyrazol-3-ylidene]-1-cyclohexa-2,4-dienone
Show/Hide
|
C20H20N4O2
|
1
|
1 |
AC50 = 40630 nM
|
|
|
CP0906893
|
SID131455650
Show/Hide
|
C25H30ClFN2O4
|
1
|
1 |
AC50 = 41160 nM
|
|
|
CP0858469
|
SID22414355
Show/Hide
|
C22H23N3O3S
|
1
|
1 |
AC50 = 41470 nM
|
|
|
CP0910494
|
SID131464147
Show/Hide
|
C30H34N2O3
|
1
|
1 |
AC50 = 41490 nM
|
|
|
CP0940511
|
SID17506494
Show/Hide
|
C20H24N2O3
|
1
|
1 |
AC50 = 41640 nM
|
|
|
CP0948167
|
SID144191134
Show/Hide
|
C30H25N3O2S
|
1
|
1 |
AC50 = 41900 nM
|
|
|
CP0900422
|
SID22416767
Show/Hide
|
C20H16O5
|
1
|
1 |
AC50 = 42430 nM
|
|
|
CP0856619
|
SID131434826
Show/Hide
|
C21H25ClFN3O5S
|
1
|
1 |
AC50 = 42730 nM
|
|
|
CP0692754
|
SID22401915
Show/Hide
|
C18H13ClN4O2S
|
1
|
1 |
AC50 = 43470 nM
|
|
|
CP0241079
|
2-(3-bromophenyl)-N-(5-nitro-2-pyridinyl)-4-quinolinecarboxamide
Show/Hide
|
C21H13BrN4O3
|
1
|
1 |
AC50 = 45550 nM
|
|
|
CP0889069
|
SID22414063
Show/Hide
|
C21H22N2O4S
|
1
|
1 |
AC50 = 47900 nM
|
|
|
CP0930559
|
SID131458696
Show/Hide
|
C27H33N3O4
|
1
|
1 |
AC50 = 48200 nM
|
|
|
CP0885907
|
SID17504545
Show/Hide
|
C24H26N2O
|
1
|
1 |
AC50 = 48210 nM
|
|
|
CP0908039
|
SID131448836
Show/Hide
|
C19H21ClN2O
|
1
|
1 |
AC50 = 50540 nM
|
|
|
CP0857789
|
SID17506165
Show/Hide
|
C20H17ClN4OS
|
1
|
1 |
AC50 = 50730 nM
|
|
|
CP0296804
|
MLS000336336
Show/Hide
|
C21H16N2OS3
|
1
|
1 |
AC50 = 51150 nM
|
|
|
CP0890218
|
SID22407983
Show/Hide
|
C19H13N3OS2
|
1
|
1 |
AC50 = 51750 nM
|
|
|
CP0865135
|
SID22405001
Show/Hide
|
C20H19NO3S
|
1
|
1 |
AC50 = 54100 nM
|
|
|
CP0912659
|
SID131462404
Show/Hide
|
C28H30FN3O2
|
1
|
1 |
AC50 = 57020 nM
|
|
|
CP0908697
|
SID131461267
Show/Hide
|
C27H26N4O2
|
1
|
1 |
AC50 = 57180 nM
|
|
|
CP0886258
|
SID131462646
Show/Hide
|
C25H32N2O3
|
1
|
1 |
AC50 = 58890 nM
|
|
|
CP0890225
|
SID87342026
Show/Hide
|
C20H23N3O4S
|
1
|
1 |
AC50 = 59150 nM
|
|
|
CP0165495
|
MLS000771265
Show/Hide
|
C14H13N3O5
|
1
|
1 |
AC50 = 59230 nM
|
|
|
CP0908895
|
SID103162580
Show/Hide
|
C17H18N2O7S
|
1
|
1 |
AC50 = 62080 nM
|
|
|
CP0864731
|
SID85800812
Show/Hide
|
C33H40N4O7
|
1
|
1 |
AC50 = 62320 nM
|
|
|
CP0660766
|
SID17432511
Show/Hide
|
C18H21F2NOS
|
1
|
1 |
AC50 = 62800 nM
|
|
|
CP0296888
|
2-[(5Z)-2,4-diketo-5-[(E)-2-methyl-3-phenyl-prop-2-enylidene]thiazolidin-3-yl]-N-(4-hydroxyphenyl)acetamide
Show/Hide
|
C21H18N2O4S
|
1
|
1 |
AC50 = 64280 nM
|
|
|
CP0886580
|
SID24800064
Show/Hide
|
C22H23N5O
|
1
|
1 |
AC50 = 64980 nM
|
|
|
CP0917638
|
SID22415174
Show/Hide
|
C24H31N3O2
|
1
|
1 |
AC50 = 65180 nM
|
|
|
CP0890216
|
SID22416446
Show/Hide
|
C18H21NOS
|
1
|
1 |
AC50 = 65370 nM
|
|
|
CP0949673
|
SID131434015
Show/Hide
|
C27H35N3O3
|
1
|
1 |
AC50 = 66120 nM
|
|
|
CP0864551
|
SID24801966
Show/Hide
|
C21H19ClN2O6
|
1
|
1 |
AC50 = 66400 nM
|
|
|
CP0029317
|
2-[[6-(hydroxymethyl)-2-(4-methoxyphenyl)-9-methyl-5H-pyrido[1,2]pyrano[2,4-b]pyrimidin-4-yl]sulfanyl]-N-(3-hydroxyphenyl)acetamide
Show/Hide
|
C27H24N4O5S
|
1
|
1 |
AC50 = 67580 nM
|
|
|
CP0959679
|
SID85805937
Show/Hide
|
C26H30N4O6S2
|
1
|
1 |
AC50 = 69490 nM
|
|
|
CP0916976
|
SID131409773
Show/Hide
|
C32H47N3O5
|
1
|
1 |
AC50 = 69510 nM
|
|
|
CP0909616
|
SID104170732
Show/Hide
|
C41H52N4O6
|
1
|
1 |
AC50 = 69590 nM
|
|
|
CP0013042
|
(5R,5aR,8aR,9R)-5-hydroxy-9-(3,4,5-trimethoxyphenyl)-5a,6,8a,9-tetrahydro-5H-[2]benzofuro[5,6-f][1,3]benzodioxol-8-one
Show/Hide
|
C22H22O8
|
1
|
1 |
AC50 < 260 nM
|
|
|
CP0037274
|
(S)-N-(5,6,7,9-tetrahydro-1,2,3,10-tetramethoxy-9-oxobenzo[a]heptalen-7-yl)acetamide
Show/Hide
|
C22H25NO6
|
1
|
1 |
AC50 < 260 nM
|
|
|
CP0077813
|
(-)-demecolcine
Show/Hide
|
C21H25NO5
|
1
|
1 |
AC50 < 260 nM
|
|
|
CP0079091
|
Anisomycin from Streptomyces griseolus
Show/Hide
|
C14H19NO4
|
1
|
1 |
AC50 < 260 nM
|
|
|
CP0103674
|
(S)-10-Amino-4-ethyl-4-hydroxy-1,12-dihydro-4H-2-oxa-6,12a-diaza-dibenzo[b,h]fluorene-3,13-dione
Show/Hide
|
C20H17N3O4
|
1
|
1 |
AC50 < 260 nM
|
|
|
CP0128167
|
4-(2-fluorophenyl)-2-methylimino-N-[(Z)-2-pyrrolylidenemethyl]-3-thiazolamine
Show/Hide
|
C15H13FN4S
|
1
|
1 |
AC50 < 260 nM
|
|
|
CP0160096
|
(1S,2E,7S,10E,12R,13R,15S)-12,15-dihydroxy-7-methyl-8-oxabicyclo[11.3.0]hexadeca-2,10-dien-9-one
Show/Hide
|
C16H24O4
|
1
|
1 |
AC50 < 260 nM
|
|
|
CP0336495
|
MLS000677248
Show/Hide
|
C22H24N2O4S
|
1
|
1 |
AC50 < 260 nM
|
|
|
CP0378346
|
(2E,10E)-12,15-dihydroxy-7-methyl-8-oxabicyclo[11.3.0]hexadeca-2,10-dien-9-one
Show/Hide
|
C16H24O4
|
1
|
1 |
AC50 < 260 nM
|
|
|
CP0396014
|
MLS003124330
Show/Hide
|
C24H23N3O4
|
1
|
1 |
AC50 < 260 nM
|
|
|
CP0408645
|
(3-fluoranyl-4-methoxy-phenyl)methyl 2-morpholin-4-yl-5-nitro-benzoate
Show/Hide
|
C19H19FN2O6
|
1
|
1 |
AC50 < 260 nM
|
|
|
CP0411307
|
4-amino-7-(3,4-dihydroxy-5-methylol-tetrahydrofuran-2-yl)pyrrolo[2,3-d]pyrimidine-5-carboxamide;hydrate
Show/Hide
|
C12H15N5O5
|
1
|
1 |
AC50 < 260 nM
|
|
|
CP0419016
|
MLS002701815
Show/Hide
|
C23H25NO7
|
1
|
1 |
AC50 < 260 nM
|
|
|
CP0423819
|
1-[(3-ethyl-9,10-dimethoxy-2,3,4,6,7,11b-hexahydro-1H-benzo[a]quinolizin-2-yl)methyl]-2,3,4,9-tetrahydro-1H-beta-carbolin-6-ol
Show/Hide
|
C29H37N3O3
|
1
|
1 |
AC50 < 260 nM
|
|
|
CP0427012
|
(20RS)-10-Amino-4-ethyl-4-hydroxy-1,12-dihydro-4H-2-oxa-6,12a-diaza-dibenzo[b,h]fluorene-3,13-dione
Show/Hide
|
C20H17N3O4
|
1
|
1 |
AC50 < 260 nM
|
|
|
CP0428588
|
MLS002702974
Show/Hide
|
C36H52O13
|
1
|
1 |
AC50 < 260 nM
|
|
|
CP0430099
|
2-ethoxyacetic acid [7-[(2-ethoxy-1-oxoethyl)amino]-1,2-dimethoxy-10-(methylthio)-9-oxo-6,7-dihydro-5H-benzo[a]heptalen-3-yl] ester
Show/Hide
|
C27H33NO8S
|
1
|
1 |
AC50 < 260 nM
|
|
|
CP0433892
|
4-[2-(3,5-dimethyl-5-oxidanyl-2-oxidanylidene-cyclohexyl)-2-oxidanyl-ethyl]piperidine-2,6-dione
Show/Hide
|
C15H23NO5
|
1
|
1 |
AC50 < 260 nM
|
|
|
CP0438388
|
1,2,3,4,7-pentahydroxy-2,3,4,4a,5,11b-hexahydro-1H-[1,3]dioxolo[4,5-j]phenanthridin-6-one
Show/Hide
|
C14H15NO8
|
1
|
1 |
AC50 < 260 nM
|
|
|
CP0445604
|
MLS001181432
Show/Hide
|
C32H48O8
|
1
|
1 |
AC50 < 260 nM
|
|
|
CP0447173
|
MLS000587490
Show/Hide
|
C18H16N4OS2
|
1
|
1 |
AC50 < 260 nM
|
|
|
CP0452846
|
DEOXYBOUVARDIN
Show/Hide
|
C40H48N6O9
|
1
|
1 |
AC50 < 260 nM
|
|
|
CP0468259
|
MLS000335164
Show/Hide
|
C18H19FN4S
|
1
|
1 |
AC50 < 260 nM
|
|
|
CP0480149
|
2-[7-(dimethylamino)-3-triazolo[4,5-d]pyrimidinyl]-5-(hydroxymethyl)oxolane-3,4-diol
Show/Hide
|
C11H16N6O4
|
1
|
1 |
AC50 < 260 nM
|
|
|
CP0480360
|
4-cycloheptyl-N-(1-pyridin-2-ylethylideneamino)piperazine-1-carbothioamide
Show/Hide
|
C19H29N5S
|
1
|
1 |
AC50 < 260 nM
|
|
|
CP0488680
|
MLS002702060
Show/Hide
|
C26H32O11
|
1
|
1 |
AC50 < 260 nM
|
|
|
CP0678329
|
SID49681835
Show/Hide
|
C23H24ClN3O5
|
1
|
1 |
AC50 < 260 nM
|
|
|
CP0707939
|
SID121285144
Show/Hide
|
C29H40Cl2N4O7S2
|
1
|
1 |
AC50 < 260 nM
|
|
|
CP0711111
|
SID855758
Show/Hide
|
C46H60N4O13S
|
1
|
1 |
AC50 < 260 nM
|
|
|
CP0725066
|
SID24831169
Show/Hide
|
C15H23ClN4OS
|
1
|
1 |
AC50 < 260 nM
|
|
|
CP0763465
|
SID26753779
Show/Hide
|
C22H22O8
|
1
|
1 |
AC50 < 260 nM
|
|
|
CP0767459
|
(E)-N-Allyl-2-(1-(pyridin-2-yl)ethylidene)hydrazinecarbothioamide
Show/Hide
|
C11H14N4S
|
1
|
1 |
AC50 < 260 nM
|
|
|
CP0792595
|
SID22410530
Show/Hide
|
C15H13N3OS2
|
1
|
1 |
AC50 < 260 nM
|
|
|
CP0849486
|
SID92763868
Show/Hide
|
C28H28O9
|
1
|
1 |
AC50 < 260 nM
|
|
|
CP0852370
|
SID49734122
Show/Hide
|
C19H19N3O4
|
1
|
1 |
AC50 < 260 nM
|
|
|
CP0858472
|
SID92763344
Show/Hide
|
C11H14N4O4
|
1
|
1 |
AC50 < 260 nM
|
|
|
CP0862099
|
SID49671357
Show/Hide
|
C22H25NO6
|
1
|
1 |
AC50 < 260 nM
|
|
|
CP0863442
|
SID92763420
Show/Hide
|
C28H36O11
|
1
|
1 |
AC50 < 260 nM
|
|
|
CP0863563
|
SID56463137
Show/Hide
|
C30H42O8
|
1
|
1 |
AC50 < 260 nM
|
|
|
CP0864577
|
SID92763446
Show/Hide
|
C57H89N7O15
|
1
|
1 |
AC50 < 260 nM
|
|
|
CP0865087
|
SID121285140
Show/Hide
|
C56H94N6O13
|
1
|
1 |
AC50 < 260 nM
|
|
|
CP0871397
|
SID92763343
Show/Hide
|
C22H26N4O5
|
1
|
1 |
AC50 < 260 nM
|
|
|
CP0873847
|
SID92763435
Show/Hide
|
C29H49N7O5
|
1
|
1 |
AC50 < 260 nM
|
|
|
CP0875014
|
SID85149103
Show/Hide
|
C30H42O8
|
1
|
1 |
AC50 < 260 nM
|
|
|
CP0878794
|
SID22403915
Show/Hide
|
C19H20N2O5
|
1
|
1 |
AC50 < 260 nM
|
|
|
CP0880472
|
SID92763425
Show/Hide
|
C28H43NO6
|
1
|
1 |
AC50 < 260 nM
|
|
|
CP0883001
|
SID92763360
Show/Hide
|
C36H45BrN4O6
|
1
|
1 |
AC50 < 260 nM
|
|
|
CP0884405
|
SID92763432
Show/Hide
|
C40H48N6O10
|
1
|
1 |
AC50 < 260 nM
|
|
|
CP0885650
|
SID92763352
Show/Hide
|
C21H23NO5S
|
1
|
1 |
AC50 < 260 nM
|
|
|
CP0886277
|
SID92763357
Show/Hide
|
C30H42O7
|
1
|
1 |
AC50 < 260 nM
|
|
|
CP0888889
|
SID99357477
Show/Hide
|
C27H36N6O4S
|
1
|
1 |
AC50 < 260 nM
|
|
|
CP0888980
|
SID92763369
Show/Hide
|
C11H13N3O4S
|
1
|
1 |
AC50 < 260 nM
|
|
|
CP0889738
|
SID92763370
Show/Hide
|
C20H31NO5
|
1
|
1 |
AC50 < 260 nM
|
|
|
CP0890227
|
SID99357801
Show/Hide
|
C27H36N6O4S
|
1
|
1 |
AC50 < 260 nM
|
|
|
CP0890588
|
SID49726715
Show/Hide
|
C19H19N3O3
|
1
|
1 |
AC50 < 260 nM
|
|
|
CP0897424
|
SID92763445
Show/Hide
|
C22H22F3NO5S
|
1
|
1 |
AC50 < 260 nM
|
|
|
CP0898193
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SID92763401
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C32H46O8
|
1
|
1 |
AC50 < 260 nM
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CP0900558
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SID92764053
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C12H14N6O4
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1
|
1 |
AC50 < 260 nM
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|
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CP0900991
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SID92763376
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C12H14N2O3
|
1
|
1 |
AC50 < 260 nM
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|
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CP0945691
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SID92763444
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C11H14N4S
|
1
|
1 |
AC50 < 260 nM
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CP0411294
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2-(3-chloro-N-(2-chloro-1-oxoethyl)anilino)-N-cyclohexyl-2-(4-methoxyphenyl)acetamide
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C23H26Cl2N2O3
|
1
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1 |
AC50 < 500 nM
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|
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CP0886269
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SID87345638
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C23H18BrN3O2
|
1
|
1 |
AC50 < 500 nM
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