All Bioactivity

Brief Information of the Cell Line and Protein

Cell Line ID: CL000006 , HEK293

Cell Line Info

Synonyms	Hek293 HEK-293 HEK/293 HEK 293 HEK;293 293 293 HEK 293 Ad5 Graham 293 Graham-293 Human Embryonic Kidney 293
Category	Transformed cell line
Organism	Homo sapiens (Human)
Cellosaurus ID	CVCL_0045

Protein ID: PT00943 , D(3) dopamine receptor

Protein Info

Gene Name	DRD3
Organism	Homo sapiens, Human
Protein Classification	Membrane receptor
Uniprot ID	P35462

Table of Molecular Bioactivities Related to the Cell Line and Protein

Cell Line ID: CL000006

Cell Line Info

Protein ID: PT00943

Protein Info

Compound ID	Compound Name	Compound Formula
CP0869682 Compound Info	N-(4-(4-(2,3-dichlorophenyl)piperazin-1-yl)butyl)-1H-indole-2-carboxamide hydrochloride Show/Hide	C23H27Cl3N4O	2
1	EC50 = 0.026 nM Bioactivity Info	TI LI LO TS
2	Ki = 15.6 nM Bioactivity Info	TI LI LO TS
CP0460373 Compound Info	(S)-N-(4-(4-Phenylbenzoylamino)butyl)-N-propyl-5-amino-4,5,6,7-tetrahydropyrazolo[1,5-a]pyridine Show/Hide	C27H34N4O	7
1	EC50 = 0.056 nM Bioactivity Info	TI LI LO TS
2	Ki = 0.058 nM Bioactivity Info	TI LI LO TS
3	Ki = 0.076 nM Bioactivity Info	TI LI LO TS
4	Ki = 0.98 nM Bioactivity Info	TI LI LO TS
5	Ki = 2.3 nM Bioactivity Info	TI LI LO TS
6	Ki = 170 nM Bioactivity Info	TI LI LO TS
7	Ki = 850 nM Bioactivity Info	TI LI LO TS
CP0006107 Compound Info	CAS_85760-74-3 Show/Hide	C13H21N3	6
1	EC50 = 0.097 nM Bioactivity Info	TI LI LO TS
2	EC50 = 2.4 nM Bioactivity Info	TI LI LO TS
3	EC50 = 10 nM Bioactivity Info	TI LI LO TS
4	Ki = 6.76 nM Bioactivity Info	TI LI LO TS
5	Ki = 8.01 nM Bioactivity Info	TI LI LO TS
6	Ki = 29.3 nM Bioactivity Info	TI LI LO TS
CP0137322 Compound Info	1H-indol-2-yl-[4-[2-(4-methoxyphenoxy)ethyl]piperazin-1-yl]methanone Show/Hide	C22H25N3O3	12
1	EC50 = 0.18 nM Bioactivity Info	TI LI LO TS
2	EC50 = 1.2 nM Bioactivity Info	TI LI LO TS
3	EC50 = 17 nM Bioactivity Info	TI LI LO TS
4	EC50 = 86 nM Bioactivity Info	TI LI LO TS
5	EC50 = 520 nM Bioactivity Info	TI LI LO TS
6	Ki = 12.5 nM Bioactivity Info	TI LI LO TS
7	Ki = 22 nM Bioactivity Info	TI LI LO TS
8	Ki = 94 nM Bioactivity Info	TI LI LO TS
9	Ki = 350 nM Bioactivity Info	TI LI LO TS
10	Ki = 720 nM Bioactivity Info	TI LI LO TS
11	Ki = 1500 nM Bioactivity Info	TI LI LO TS
12	Ki = 3700 nM Bioactivity Info	TI LI LO TS
CP0041034 Compound Info	US8748608, 16 Show/Hide	C26H28Cl2N4O2	3
1	EC50 = 1 nM Bioactivity Info	TI LI LO TS
2	IC50 = 1 nM Bioactivity Info	TI LI LO TS
3	Ki = 3 nM Bioactivity Info	TI LI LO TS
CP0876922 Compound Info	N-(4-(4-(2,4-dichlorophenyl)piperazin-1-yl)butyl)-1H-indole-2-carboxamide hydrochloride Show/Hide	C23H27Cl3N4O	2
1	EC50 = 1.1 nM Bioactivity Info	TI LI LO TS
2	Ki = 407.2 nM Bioactivity Info	TI LI LO TS
CP0036921 Compound Info	3-HYDROXYTYRAMINE HYDROCHLORIDE Show/Hide	C8H11NO2	14
1	EC50 = 1.1 nM Bioactivity Info	TI LI LO TS
2	EC50 = 2.1 nM Bioactivity Info	TI LI LO TS
3	EC50 = 2.3 nM Bioactivity Info	TI LI LO TS
4	EC50 = 3.5 nM Bioactivity Info	TI LI LO TS
5	EC50 = 33 nM Bioactivity Info	TI LI LO TS
6	EC50 = 55 nM Bioactivity Info	TI LI LO TS
7	EC50 = 820 nM Bioactivity Info	TI LI LO TS
8	Ki = 2.97 nM Bioactivity Info	TI LI LO TS
9	Ki = 7.58 nM Bioactivity Info	TI LI LO TS
10	Ki = 15 nM Bioactivity Info	TI LI LO TS
11	Ki = 72 nM Bioactivity Info	TI LI LO TS
12	Ki = 293 nM Bioactivity Info	TI LI LO TS
13	Ki = 1100 nM Bioactivity Info	TI LI LO TS
14	Ki > 80000 nM Bioactivity Info	TI LI LO TS
CP0382046 Compound Info	1-[4-[2,3-dihydro-1H-inden-2-yl(propyl)amino]butyl]-3-(4-fluorophenyl)iminourea Show/Hide	C23H29FN4O	2
1	EC50 = 2.6 nM Bioactivity Info	TI LI LO TS
2	EC50 = 68 nM Bioactivity Info	TI LI LO TS
CP0167371 Compound Info	US8748608, 21 Show/Hide	C26H28Cl2N4O2	3
1	EC50 = 3.4 nM Bioactivity Info	TI LI LO TS
2	IC50 = 5.4 nM Bioactivity Info	TI LI LO TS
3	Ki = 0.5 nM Bioactivity Info	TI LI LO TS
CP0167372 Compound Info	US8748608, 20 Show/Hide	C28H30Cl2N4O3	3
1	EC50 = 3.9 nM Bioactivity Info	TI LI LO TS
2	IC50 = 5.4 nM Bioactivity Info	TI LI LO TS
3	Ki = 11.7 nM Bioactivity Info	TI LI LO TS
CP0388832 Compound Info	1-(3,4-difluorophenyl)imino-3-[4-[2,3-dihydro-1H-inden-2-yl(propyl)amino]butyl]urea Show/Hide	C23H28F2N4O	2
1	EC50 = 6.1 nM Bioactivity Info	TI LI LO TS
2	EC50 = 79 nM Bioactivity Info	TI LI LO TS
CP0049308 Compound Info	N-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butyl]-4-pyridin-2-ylbenzamide Show/Hide	C26H28Cl2N4O	2
1	EC50 = 6.3 nM Bioactivity Info	TI LI LO TS
2	Ki = 0.4 nM Bioactivity Info	TI LI LO TS
CP0376123 Compound Info	1-[4-[2,3-dihydro-1H-inden-2-yl(propyl)amino]butyl]-3-(3,4,5-trifluorophenyl)iminourea Show/Hide	C23H27F3N4O	2
1	EC50 = 11 nM Bioactivity Info	TI LI LO TS
2	EC50 = 114 nM Bioactivity Info	TI LI LO TS
CP0197219 Compound Info	N-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]-3-hydroxybutyl]-1-benzofuran-2-carboxamide Show/Hide	C23H25Cl2N3O3	4
1	EC50 = 22.8 nM Bioactivity Info	TI LI LO TS
2	IC50 = 13.7 nM Bioactivity Info	TI LI LO TS
3	Ki = 0.98 nM Bioactivity Info	TI LI LO TS
4	Ki = 6.11 nM Bioactivity Info	TI LI LO TS
CP0065116 Compound Info	US8748608, 17 Show/Hide	C28H29Cl2N3O2	3
1	EC50 = 42 nM Bioactivity Info	TI LI LO TS
2	IC50 = 42 nM Bioactivity Info	TI LI LO TS
3	Ki = 1.8 nM Bioactivity Info	TI LI LO TS
CP0436005 Compound Info	(R)-N-(4-(4-Phenylbenzoylamino)butyl)-N-propyl-5-amino-4,5,6,7-tetrahydropyrazolo[1,5-a]pyridine Show/Hide	C27H34N4O	7
1	EC50 = 51 nM Bioactivity Info	TI LI LO TS
2	Ki = 15 nM Bioactivity Info	TI LI LO TS
3	Ki = 19 nM Bioactivity Info	TI LI LO TS
4	Ki = 43 nM Bioactivity Info	TI LI LO TS
5	Ki = 240 nM Bioactivity Info	TI LI LO TS
6	Ki = 1400 nM Bioactivity Info	TI LI LO TS
7	Ki = 3700 nM Bioactivity Info	TI LI LO TS
CP0288360 Compound Info	N-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]-3-hydroxybutyl]-5-iodo-1-benzofuran-2-carboxamide Show/Hide	C23H24Cl2IN3O3	4
1	EC50 = 84 nM Bioactivity Info	TI LI LO TS
2	IC50 = 217 nM Bioactivity Info	TI LI LO TS
3	Ki = 3.5 nM Bioactivity Info	TI LI LO TS
4	Ki = 7.71 nM Bioactivity Info	TI LI LO TS
CP0065124 Compound Info	9H-Fluorene-2-carboxylic acid {(E)-4-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-but-2-enyl}-amide Show/Hide	C28H27Cl2N3O	3
1	EC50 = 173 nM Bioactivity Info	TI LI LO TS
2	Ki = 1.5 nM Bioactivity Info	TI LI LO TS
3	Ki = 5.9 nM Bioactivity Info	TI LI LO TS
CP0104676 Compound Info	Benzo[b]thiophene-2-carboxylic acid {4-[4-(2-methoxy-phenyl)-piperazin-1-yl]-butyl}-amide Show/Hide	C24H29N3O2S	2
1	IC50 = 0.22 nM Bioactivity Info	TI LI LO TS
2	Ki = 0.19 nM Bioactivity Info	TI LI LO TS
CP0049309 Compound Info	N-[(E)-4-[4-(2,3-dichlorophenyl)piperazin-1-yl]but-2-enyl]-4-(6-oxo-1H-pyridin-2-yl)benzamide Show/Hide	C26H26Cl2N4O2	2
1	IC50 = 1 nM Bioactivity Info	TI LI LO TS
2	Ki = 0.6 nM Bioactivity Info	TI LI LO TS
CP0127237 Compound Info	N-[(E)-4-[4-(2-methoxyphenyl)piperazin-1-yl]but-2-enyl]-1-benzothiophene-2-carboxamide Show/Hide	C24H27N3O2S	2
1	IC50 = 1.09 nM Bioactivity Info	TI LI LO TS
2	Ki = 2.61 nM Bioactivity Info	TI LI LO TS
CP0065125 Compound Info	N-[(E)-4-[4-(2,3-dichlorophenyl)piperazin-1-yl]but-2-enyl]-4-(1-oxidopyridin-1-ium-2-yl)benzamide Show/Hide	C26H26Cl2N4O2	2
1	IC50 = 1.2 nM Bioactivity Info	TI LI LO TS
2	Ki = 1.1 nM Bioactivity Info	TI LI LO TS
CP0197218 Compound Info	N-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]-3-hydroxybutyl]-5-methoxy-1H-indole-2-carboxamide Show/Hide	C24H28Cl2N4O3	3
1	IC50 = 1.51 nM Bioactivity Info	TI LI LO TS
2	Ki = 0.92 nM Bioactivity Info	TI LI LO TS
3	Ki = 1.2 nM Bioactivity Info	TI LI LO TS
CP0369518 Compound Info	N-[3-hydroxy-4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]-5-methoxy-1H-indole-2-carboxamide Show/Hide	C25H32N4O4	2
1	IC50 = 1.58 nM Bioactivity Info	TI LI LO TS
2	Ki = 2.32 nM Bioactivity Info	TI LI LO TS
CP0096655 Compound Info	5-fluoro-N-[3-hydroxy-4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]-1H-indole-2-carboxamide Show/Hide	C24H29FN4O3	2
1	IC50 = 1.76 nM Bioactivity Info	TI LI LO TS
2	Ki = 2.41 nM Bioactivity Info	TI LI LO TS
CP0261925 Compound Info	N-[4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]-9H-fluorene-2-carboxamide Show/Hide	C29H33N3O2	2
1	IC50 = 2.2 nM Bioactivity Info	TI LI LO TS
2	Ki = 0.3 nM Bioactivity Info	TI LI LO TS
CP0045037 Compound Info	Benzofuran-2-carboxylic acid {4-[4-(2-methoxy-phenyl)-piperazin-1-yl]-butyl}-amide Show/Hide	C24H29N3O3	2
1	IC50 = 2.39 nM Bioactivity Info	TI LI LO TS
2	Ki = 0.92 nM Bioactivity Info	TI LI LO TS
CP0224357 Compound Info	N-[4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]-4-pyridin-2-ylbenzamide Show/Hide	C27H32N4O2	2
1	IC50 = 2.9 nM Bioactivity Info	TI LI LO TS
2	Ki = 0.4 nM Bioactivity Info	TI LI LO TS
CP0061556 Compound Info	N-[(E)-4-[4-(2,3-dichlorophenyl)piperazin-1-yl]but-2-enyl]-4-pyridin-2-ylbenzamide Show/Hide	C26H26Cl2N4O	3
1	IC50 = 3 nM Bioactivity Info	TI LI LO TS
2	Ki = 0.316 nM Bioactivity Info	TI LI LO TS
3	Ki = 0.7 nM Bioactivity Info	TI LI LO TS
CP0377890 Compound Info	US8748608, 19 Show/Hide	C29H33N3O3	2
1	IC50 = 3.9 nM Bioactivity Info	TI LI LO TS
2	Ki = 1.8 nM Bioactivity Info	TI LI LO TS
CP0043442 Compound Info	Benzo[b]thiophene-2-carboxylic acid {4-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-butyl}-amide Show/Hide	C23H25Cl2N3OS	3
1	IC50 = 4.94 nM Bioactivity Info	TI LI LO TS
2	Ki = 0.5 nM Bioactivity Info	TI LI LO TS
3	Ki = 0.81 nM Bioactivity Info	TI LI LO TS
CP0333371 Compound Info	N-[3-hydroxy-4-[4-(2-propoxyphenyl)piperazin-1-yl]butyl]-1H-indole-2-carboxamide Show/Hide	C26H34N4O3	2
1	IC50 = 6.51 nM Bioactivity Info	TI LI LO TS
2	Ki = 62.1 nM Bioactivity Info	TI LI LO TS
CP0293888 Compound Info	N-[(3S)-4-[4-(2,3-dichlorophenyl)piperazin-1-yl]-3-hydroxybutyl]-1H-indole-2-carboxamide Show/Hide	C23H26Cl2N4O2	3
1	IC50 = 6.6 nM Bioactivity Info	TI LI LO TS
2	Ki = 3.9 nM Bioactivity Info	TI LI LO TS
3	Ki = 16.6 nM Bioactivity Info	TI LI LO TS
CP0202185 Compound Info	N-[(E)-4-[4-(2,3-dichlorophenyl)piperazin-1-yl]but-2-enyl]-4-(6-methylpyridin-2-yl)benzamide Show/Hide	C27H28Cl2N4O	2
1	IC50 = 6.7 nM Bioactivity Info	TI LI LO TS
2	Ki = 1.4 nM Bioactivity Info	TI LI LO TS
CP0288362 Compound Info	N-[(E)-4-[4-(2,3-dichlorophenyl)piperazin-1-yl]but-2-enyl]-1H-indole-2-carboxamide Show/Hide	C23H24Cl2N4O	2
1	IC50 = 7 nM Bioactivity Info	TI LI LO TS
2	Ki = 0.44 nM Bioactivity Info	TI LI LO TS
CP0041389 Compound Info	Benzofuran-2-carboxylic acid {4-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-butyl}-amide Show/Hide	C23H25Cl2N3O2	3
1	IC50 = 9.01 nM Bioactivity Info	TI LI LO TS
2	Ki = 0.8 nM Bioactivity Info	TI LI LO TS
3	Ki = 0.81 nM Bioactivity Info	TI LI LO TS
CP0047599 Compound Info	Benzo[b]thiophene-2-carboxylic acid {4-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-but-2-enyl}-amide Show/Hide	C23H23Cl2N3OS	2
1	IC50 = 9.62 nM Bioactivity Info	TI LI LO TS
2	Ki = 1.11 nM Bioactivity Info	TI LI LO TS
CP0369519 Compound Info	N-[3-hydroxy-4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]-1-benzofuran-2-carboxamide Show/Hide	C24H29N3O4	3
1	IC50 = 11.2 nM Bioactivity Info	TI LI LO TS
2	Ki = 5.4 nM Bioactivity Info	TI LI LO TS
3	Ki = 7.51 nM Bioactivity Info	TI LI LO TS
CP0288363 Compound Info	N-[3-hydroxy-4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]-1H-indole-2-carboxamide Show/Hide	C24H30N4O3	3
1	IC50 = 12.1 nM Bioactivity Info	TI LI LO TS
2	Ki = 1.37 nM Bioactivity Info	TI LI LO TS
3	Ki = 1.4 nM Bioactivity Info	TI LI LO TS
CP0277136 Compound Info	US8748608, 18 Show/Hide	C27H32N4O3	3
1	IC50 = 12.8 nM Bioactivity Info	TI LI LO TS
2	Ki = 2.8 nM Bioactivity Info	TI LI LO TS
3	Ki = 6.7 nM Bioactivity Info	TI LI LO TS
CP0185379 Compound Info	N-[[(1S,2S)-2-[[4-(2,3-dichlorophenyl)piperazin-1-yl]methyl]cyclopropyl]methyl]-4-pyridin-2-ylbenzamide Show/Hide	C27H28Cl2N4O	2
1	IC50 = 14.3 nM Bioactivity Info	TI LI LO TS
2	Ki = 1 nM Bioactivity Info	TI LI LO TS
CP0079495 Compound Info	9H-Fluorene-2-carboxylic acid {4-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-butyl}-amide Show/Hide	C28H29Cl2N3O	4
1	IC50 = 14.4 nM Bioactivity Info	TI LI LO TS
2	Ki = 0.233 nM Bioactivity Info	TI LI LO TS
3	Ki = 1.4 nM Bioactivity Info	TI LI LO TS
4	Ki = 2 nM Bioactivity Info	TI LI LO TS
CP0288361 Compound Info	N-[3-hydroxy-4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]-5-iodo-1-benzofuran-2-carboxamide Show/Hide	C24H28IN3O4	3
1	IC50 = 14.5 nM Bioactivity Info	TI LI LO TS
2	Ki = 2.2 nM Bioactivity Info	TI LI LO TS
3	Ki = 7.5 nM Bioactivity Info	TI LI LO TS
CP0267025 Compound Info	N-[(E)-4-[4-(2-methoxyphenyl)piperazin-1-yl]but-2-enyl]-1-benzofuran-2-carboxamide Show/Hide	C24H27N3O3	2
1	IC50 = 14.9 nM Bioactivity Info	TI LI LO TS
2	Ki = 11.3 nM Bioactivity Info	TI LI LO TS
CP0122857 Compound Info	(R)-N-(4-(4-(2,3-dichlorophenyl)piperazin-1-yl)-3-hydroxybutyl)-1H-indole-2-carboxamide Show/Hide	C23H26Cl2N4O2	3
1	IC50 = 18.2 nM Bioactivity Info	TI LI LO TS
2	Ki = 0.53 nM Bioactivity Info	TI LI LO TS
3	Ki = 1.12 nM Bioactivity Info	TI LI LO TS
CP0044765 Compound Info	Benzofuran-2-carboxylic acid {4-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-but-2-enyl}-amide Show/Hide	C23H23Cl2N3O2	2
1	IC50 = 18.7 nM Bioactivity Info	TI LI LO TS
2	Ki = 2.11 nM Bioactivity Info	TI LI LO TS
CP0167369 Compound Info	N-[(E)-4-[4-(2-methoxyphenyl)piperazin-1-yl]but-2-enyl]-9H-fluorene-2-carboxamide Show/Hide	C29H31N3O2	3
1	IC50 = 18.9 nM Bioactivity Info	TI LI LO TS
2	Ki = 1.2 nM Bioactivity Info	TI LI LO TS
3	Ki = 12 nM Bioactivity Info	TI LI LO TS
CP0197217 Compound Info	5-Iodo-benzofuran-2-carboxylic acid {4-[4-(2-methoxy-phenyl)-piperazin-1-yl]-butyl}-amide Show/Hide	C24H28IN3O3	2
1	IC50 = 22.9 nM Bioactivity Info	TI LI LO TS
2	Ki = 0.72 nM Bioactivity Info	TI LI LO TS
CP0156829 Compound Info	N-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]-3-hydroxybutyl]-5-fluoro-1H-indole-2-carboxamide Show/Hide	C23H25Cl2FN4O2	3
1	IC50 = 23.9 nM Bioactivity Info	TI LI LO TS
2	Ki = 1.61 nM Bioactivity Info	TI LI LO TS
3	Ki = 1.8 nM Bioactivity Info	TI LI LO TS
CP0065126 Compound Info	N-[(E)-4-[4-(2,3-dichlorophenyl)piperazin-1-yl]but-2-enyl]-4-(3-methylpyridin-2-yl)benzamide Show/Hide	C27H28Cl2N4O	2
1	IC50 = 25.6 nM Bioactivity Info	TI LI LO TS
2	Ki = 1.6 nM Bioactivity Info	TI LI LO TS
CP0218398 Compound Info	6-[5-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]pentanoyl]-1-azatricyclo[6.3.1.04,12]dodeca-4,6,8(12)-trien-11-one Show/Hide	C28H30FN3O3	1
1	IC50 = 25.6 nM Bioactivity Info	TI LI LO TS
CP0096659 Compound Info	N-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]-2-hydroxybutyl]-1H-indole-2-carboxamide Show/Hide	C23H26Cl2N4O2	2
1	IC50 = 25.7 nM Bioactivity Info	TI LI LO TS
2	Ki = 0.26 nM Bioactivity Info	TI LI LO TS
CP0057840 Compound Info	US8748608, 34 Show/Hide	C23H26Cl2N4O2	4
1	IC50 = 29.9 nM Bioactivity Info	TI LI LO TS
2	Ki = 1.39 nM Bioactivity Info	TI LI LO TS
3	Ki = 1.88 nM Bioactivity Info	TI LI LO TS
4	Ki = 1.9 nM Bioactivity Info	TI LI LO TS
CP0091917 Compound Info	N-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]-3-hydroxybutyl]-5-iodo-1H-indole-2-carboxamide Show/Hide	C23H25Cl2IN4O2	2
1	IC50 = 38 nM Bioactivity Info	TI LI LO TS
2	Ki = 5.21 nM Bioactivity Info	TI LI LO TS
CP0096658 Compound Info	N-[3-hydroxy-4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]-1-benzothiophene-2-carboxamide Show/Hide	C24H29N3O3S	2
1	IC50 = 39.1 nM Bioactivity Info	TI LI LO TS
2	Ki = 4.6 nM Bioactivity Info	TI LI LO TS
CP0252256 Compound Info	N-[(E)-4-[4-(2-methoxyphenyl)piperazin-1-yl]but-2-enyl]-4-pyridin-2-ylbenzamide Show/Hide	C27H30N4O2	2
1	IC50 = 42.6 nM Bioactivity Info	TI LI LO TS
2	Ki = 2.9 nM Bioactivity Info	TI LI LO TS
CP0040671 Compound Info	8-[4-(4-fluorophenyl)-4-keto-butyl]-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one Show/Hide	C23H26FN3O2	3
1	IC50 = 93.2 nM Bioactivity Info	TI LI LO TS
2	Ki = 0.33 nM Bioactivity Info	TI LI LO TS
3	Ki = 0.48 nM Bioactivity Info	TI LI LO TS
CP0327018 Compound Info	N-[3-hydroxy-4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]-5-iodo-1H-indole-2-carboxamide Show/Hide	C24H29IN4O3	2
1	IC50 = 173 nM Bioactivity Info	TI LI LO TS
2	Ki = 3.6 nM Bioactivity Info	TI LI LO TS
CP0253779 Compound Info	5-Iodo-benzofuran-2-carboxylic acid {4-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-butyl}-amide Show/Hide	C23H24Cl2IN3O2	2
1	IC50 = 520 nM Bioactivity Info	TI LI LO TS
2	Ki = 1.59 nM Bioactivity Info	TI LI LO TS
CP0382963 Compound Info	MLS001173843 Show/Hide	C21H26N2O4	1
1	IC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0243806 Compound Info	N-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]-3-fluorobutyl]-1-benzofuran-2-carboxamide Show/Hide	C23H24Cl2FN3O2	6
1	Kd = 0.03 nM Bioactivity Info	TI LI LO TS
2	Kd = 0.04 nM Bioactivity Info	TI LI LO TS
3	Ki = 5.4 nM Bioactivity Info	TI LI LO TS
4	Ki = 6.1 nM Bioactivity Info	TI LI LO TS
5	Ki = 10 nM Bioactivity Info	TI LI LO TS
6	Ki = 31.5 nM Bioactivity Info	TI LI LO TS
CP0053105 Compound Info	(S)-3-chloro-5-ethyl-N-((1-ethylpyrrolidin-2-yl)methyl)-6-hydroxy-2-methoxybenzamide Show/Hide	C17H25ClN2O3	2
1	Ki = 0.11 nM Bioactivity Info	TI LI LO TS
2	Ki = 0.134 nM Bioactivity Info	TI LI LO TS
CP0057834 Compound Info	N-[4-(4-naphthalen-1-ylpiperazin-1-yl)butyl]-1H-indole-2-carboxamide Show/Hide	C27H30N4O	1
1	Ki = 0.118 nM Bioactivity Info	TI LI LO TS
CP0427965 Compound Info	N-[4-(4-naphthalen-1-ylpiperazin-1-yl)butyl]-1-benzothiophene-2-carboxamide Show/Hide	C27H29N3OS	1
1	Ki = 0.128 nM Bioactivity Info	TI LI LO TS
CP0224535 Compound Info	N-[4-[4-(2-chloro-3-ethylphenyl)piperazin-1-yl]butyl]-1H-indole-2-carboxamide Show/Hide	C25H31ClN4O	1
1	Ki = 0.142 nM Bioactivity Info	TI LI LO TS
CP0224534 Compound Info	N-[4-[4-(2-chloro-3-ethylphenyl)piperazin-1-yl]butyl]-1-benzofuran-2-carboxamide Show/Hide	C25H30ClN3O2	1
1	Ki = 0.153 nM Bioactivity Info	TI LI LO TS
CP0460372 Compound Info	Biphenyl-4-carboxylic acid {4-[4-(2-methoxy-phenyl)-piperazin-1-yl]-butyl}-amide; oxalic acid Show/Hide	C28H33N3O2	6
1	Ki = 0.16 nM Bioactivity Info	TI LI LO TS
2	Ki = 0.58 nM Bioactivity Info	TI LI LO TS
3	Ki = 0.9 nM Bioactivity Info	TI LI LO TS
4	Ki = 2.8 nM Bioactivity Info	TI LI LO TS
5	Ki = 180 nM Bioactivity Info	TI LI LO TS
6	Ki = 790 nM Bioactivity Info	TI LI LO TS
CP0786649 Compound Info	4-(Thiophen-3-yl)-N-(4-(4-(2-(2-fluoroethoxy)phenyl)piperazin-1-yl)butyl)benzamide oxalic acid salt Show/Hide	C29H34FN3O6S	1
1	Ki = 0.17 nM Bioactivity Info	TI LI LO TS
CP0538829 Compound Info	N-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butyl]quinoline-3-carboxamide Show/Hide	C24H26Cl2N4O	1
1	Ki = 0.172 nM Bioactivity Info	TI LI LO TS
CP0381583 Compound Info	5-methoxy-N-[4-(4-naphthalen-1-ylpiperazin-1-yl)butyl]-1H-indole-2-carboxamide Show/Hide	C28H32N4O2	1
1	Ki = 0.173 nM Bioactivity Info	TI LI LO TS
CP0850773 Compound Info	5-Hydroxy-N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)-1H-indole-2-carboxamide oxalic acid Show/Hide	C26H32N4O7	1
1	Ki = 0.18 nM Bioactivity Info	TI LI LO TS
CP0375619 Compound Info	(S)-6-(propyl(2-(4-(quinolin-4-yl)piperazin-1-yl)ethyl)amino)-5,6,7,8-tetrahydronaphthalen-1-ol Show/Hide	C28H36N4O	1
1	Ki = 0.186 nM Bioactivity Info	TI LI LO TS
CP0419149 Compound Info	(-)-(S)-6-(Propyl(2-(4-(quinolin-4-yl)piperazin-1-yl)ethyl)amino)-5,6,7,8-tetrahydronaphthalen-1-ol Show/Hide	C29H38N4O	1
1	Ki = 0.19 nM Bioactivity Info	TI LI LO TS
CP0435436 Compound Info	N-[4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]-4-thiophen-3-ylbenzamide Show/Hide	C26H31N3O2S	1
1	Ki = 0.2 nM Bioactivity Info	TI LI LO TS
CP0480201 Compound Info	N-[4-[4-(2-chloro-3-ethylphenyl)piperazin-1-yl]-2-hydroxybutyl]-1H-indole-2-carboxamide Show/Hide	C25H31ClN4O2	1
1	Ki = 0.2 nM Bioactivity Info	TI LI LO TS
CP0381742 Compound Info	N-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]-3-hydroxybutyl]-9H-fluorene-3-carboxamide Show/Hide	C28H29Cl2N3O2	1
1	Ki = 0.233 nM Bioactivity Info	TI LI LO TS
CP0550061 Compound Info	N-[4-(4-naphthalen-1-ylpiperazin-1-yl)butyl]-1-benzofuran-2-carboxamide Show/Hide	C27H29N3O2	1
1	Ki = 0.244 nM Bioactivity Info	TI LI LO TS
CP0435434 Compound Info	N-[4-[4-(2-cyanophenyl)piperazin-1-yl]butyl]-4-thiophen-3-ylbenzamide Show/Hide	C26H28N4OS	1
1	Ki = 0.25 nM Bioactivity Info	TI LI LO TS
CP0337664 Compound Info	8-[4-(4-Fluoro-phenyl)-4-oxo-butyl]-3-methyl-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one Show/Hide	C24H28FN3O2	1
1	Ki = 0.265 nM Bioactivity Info	TI LI LO TS
CP0109326 Compound Info	5-Fluoro-1H-indole-2-carboxylic acid {4-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-butyl}-amide Show/Hide	C23H25Cl2FN4O	2
1	Ki = 0.28 nM Bioactivity Info	TI LI LO TS
2	Ki = 0.52 nM Bioactivity Info	TI LI LO TS
CP0063621 Compound Info	N-[(3R)-4-[4-(2-chloro-3-ethylphenyl)piperazin-1-yl]-3-hydroxybutyl]-1H-indole-2-carboxamide Show/Hide	C25H31ClN4O2	1
1	Ki = 0.29 nM Bioactivity Info	TI LI LO TS
CP0071762 Compound Info	N-[4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]naphthalene-2-carboxamide Show/Hide	C26H31N3O2	1
1	Ki = 0.3 nM Bioactivity Info	TI LI LO TS
CP0410602 Compound Info	N-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butyl]imidazo[1,2-a]pyridine-2-carboxamide Show/Hide	C22H25Cl2N5O	1
1	Ki = 0.3 nM Bioactivity Info	TI LI LO TS
CP0314424 Compound Info	1H-Indole-2-carboxylic acid {4-[4-(2-methoxy-phenyl)-piperazin-1-yl]-butyl}-amide Show/Hide	C24H30N4O2	1
1	Ki = 0.32 nM Bioactivity Info	TI LI LO TS
CP0424340 Compound Info	N-[4-[4-(2-chloro-3-ethylphenyl)piperazin-1-yl]butyl]imidazo[1,2-a]pyridine-2-carboxamide Show/Hide	C24H30ClN5O	1
1	Ki = 0.331 nM Bioactivity Info	TI LI LO TS
CP0888512 Compound Info	endo-8-(Benzofur-3-ylmethyl)-3-(3,4-dichlorophenyl)-8-azabicyclo[3.2.1]octan-3-ol Show/Hide	C22H21Cl2NO2	1
1	Ki = 0.34 nM Bioactivity Info	TI LI LO TS
CP0135680 Compound Info	N-[4-[4-(3-chloro-5-ethyl-2-methoxyphenyl)piperazin-1-yl]butyl]-1H-indole-2-carboxamide Show/Hide	C26H33ClN4O2	1
1	Ki = 0.341 nM Bioactivity Info	TI LI LO TS
CP0045182 Compound Info	N-[4-(4-naphthalen-1-ylpiperazin-1-yl)butyl]quinoline-3-carboxamide Show/Hide	C28H30N4O	1
1	Ki = 0.351 nM Bioactivity Info	TI LI LO TS
CP0157764 Compound Info	N-[4-[4-(2-chloro-3-ethylphenyl)piperazin-1-yl]-3-hydroxybutyl]-1H-indole-2-carboxamide Show/Hide	C25H31ClN4O2	2
1	Ki = 0.362 nM Bioactivity Info	TI LI LO TS
2	Ki = 0.433 nM Bioactivity Info	TI LI LO TS
CP0158026 Compound Info	1-butyl-4-(2-chloro-3-ethylphenyl)piperazine Show/Hide	C16H25ClN2	1
1	Ki = 0.363 nM Bioactivity Info	TI LI LO TS
CP0869617 Compound Info	endo-8-(5-Fluorobenzofur-3-ylmethyl)-3-(4-chlorophenyl)-8-azabicyclo[3.2.1]octan-3-ol Show/Hide	C22H21ClFNO2	1
1	Ki = 0.37 nM Bioactivity Info	TI LI LO TS
CP0463676 Compound Info	N-[(3R)-4-[4-(2-chloro-3-ethylphenyl)piperazin-1-yl]-3-fluorobutyl]-1H-indole-2-carboxamide Show/Hide	C25H30ClFN4O	1
1	Ki = 0.373 nM Bioactivity Info	TI LI LO TS
CP0860173 Compound Info	N-(4-(4-(2-(2-fluoroethoxy)phenyl)piperazin-1-yl)butyl)-5-methoxy-1H-indole-3-carboxamide oxalic acid Show/Hide	C28H35FN4O7	1
1	Ki = 0.39 nM Bioactivity Info	TI LI LO TS
CP0494803 Compound Info	N-[4-[4-(3-chloro-2-methoxyphenyl)piperazin-1-yl]butyl]-1H-indole-2-carboxamide Show/Hide	C24H29ClN4O2	1
1	Ki = 0.392 nM Bioactivity Info	TI LI LO TS
CP0894766 Compound Info	6-(Propyl(2-(4-(quinolin-4-yl)piperazin-1-yl)ethyl)amino)-5,6,7,8-tetrahydronaphthalen-1-ol Show/Hide	C29H38N4O	1
1	Ki = 0.4 nM Bioactivity Info	TI LI LO TS
CP0519086 Compound Info	4-thiophen-3-yl-N-[4-[4-[3-(trifluoromethyl)phenyl]piperazin-1-yl]butyl]benzamide Show/Hide	C26H28F3N3OS	1
1	Ki = 0.41 nM Bioactivity Info	TI LI LO TS
CP0869493 Compound Info	5-(2-fluoroethoxy)-N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)-1H-indole-2-carboxamide oxalic acid Show/Hide	C28H35FN4O7	1
1	Ki = 0.43 nM Bioactivity Info	TI LI LO TS
CP0419143 Compound Info	7-((2-(4-(Naphthalen-1-yl)-piperazin-1-yl)ethyl)(propyl)amino)-5,6,7,8-tetrahydronaphthalen-2-ol Show/Hide	C29H37N3O	1
1	Ki = 0.435 nM Bioactivity Info	TI LI LO TS
CP0075581 Compound Info	N-[4-[4-(3,5-dichlorophenyl)piperazin-1-yl]butyl]-4-thiophen-3-ylbenzamide Show/Hide	C25H27Cl2N3OS	1
1	Ki = 0.44 nM Bioactivity Info	TI LI LO TS
CP0452360 Compound Info	7-((2-(4-(Isoquinolin-1-yl)piperazin-1-yl)ethyl)(propyl)amino)-5,6,7,8-tetrahydronaphthalen-2-ol Show/Hide	C28H36N4O	1
1	Ki = 0.441 nM Bioactivity Info	TI LI LO TS
CP0434348 Compound Info	6-[(2-(4-(2,3-dichlorophenyl)piperazin-1-yl)ethyl)(propyl)amino]-5,6,7,8-tetrahydronaphthalen-1-ol Show/Hide	C25H33Cl2N3O	1
1	Ki = 0.45 nM Bioactivity Info	TI LI LO TS
CP0455628 Compound Info	N-[[(1R,2R)-2-[[4-(2,3-dichlorophenyl)piperazin-1-yl]methyl]cyclopropyl]methyl]-1H-indole-2-carboxamide Show/Hide	C24H26Cl2N4O	1
1	Ki = 0.45 nM Bioactivity Info	TI LI LO TS
CP0466448 Compound Info	N-[4-[4-(3-hydroxyphenyl)piperazin-1-yl]butyl]-4-thiophen-3-ylbenzamide Show/Hide	C25H29N3O2S	1
1	Ki = 0.47 nM Bioactivity Info	TI LI LO TS
CP0375779 Compound Info	N-[4-[4-(2-methylsulfanylphenyl)piperazin-1-yl]butyl]pyrazolo[1,5-a]pyridine-2-carboxamide Show/Hide	C23H29N5OS	8
1	Ki = 0.5 nM Bioactivity Info	TI LI LO TS
2	Ki = 0.76 nM Bioactivity Info	TI LI LO TS
3	Ki = 18 nM Bioactivity Info	TI LI LO TS
4	Ki = 33 nM Bioactivity Info	TI LI LO TS
5	Ki = 40 nM Bioactivity Info	TI LI LO TS
6	Ki = 58 nM Bioactivity Info	TI LI LO TS
7	Ki = 160 nM Bioactivity Info	TI LI LO TS
8	Ki = 230 nM Bioactivity Info	TI LI LO TS
CP0450101 Compound Info	N-[2-hydroxy-4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]-1H-indole-2-carboxamide Show/Hide	C24H30N4O3	2
1	Ki = 0.5 nM Bioactivity Info	TI LI LO TS
2	Ki = 0.51 nM Bioactivity Info	TI LI LO TS
CP0159265 Compound Info	N-[4-[4-(3-cyanophenyl)piperazin-1-yl]butyl]-4-thiophen-3-ylbenzamide Show/Hide	C26H28N4OS	1
1	Ki = 0.5 nM Bioactivity Info	TI LI LO TS
CP0785530 Compound Info	4-(2-Fluoroethoxy)-N-(4-(4-(2-(2-fluoroethoxy)phenyl)piperazin-1-yl)butyl)benzamide oxalic acid salt Show/Hide	C27H35F2N3O7	1
1	Ki = 0.52 nM Bioactivity Info	TI LI LO TS
CP0881590 Compound Info	endo-8-(5-Fluorobenzofur-3-ylmethyl)-3-(3,4-dichlorophenyl)-8-azabicyclo[3.2.1]octan-3-ol Show/Hide	C22H20Cl2FNO2	1
1	Ki = 0.53 nM Bioactivity Info	TI LI LO TS
CP0520078 Compound Info	N-[4-[4-(2-chlorophenyl)piperazin-1-yl]butyl]-4-thiophen-3-ylbenzamide Show/Hide	C25H28ClN3OS	1
1	Ki = 0.55 nM Bioactivity Info	TI LI LO TS
CP0469532 Compound Info	(S)-(4-(2-((5-hydroxy-1,2,3,4-tetrahydronaphthalen-2-yl)(propyl)amino)ethyl)piperazin-1-yl)(1H-indol-2-yl)methanone Show/Hide	C28H36N4O2	1
1	Ki = 0.57 nM Bioactivity Info	TI LI LO TS
CP0504692 Compound Info	N-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butyl]-6-fluoroquinoline-3-carboxamide Show/Hide	C24H25Cl2FN4O	1
1	Ki = 0.57 nM Bioactivity Info	TI LI LO TS
CP0488182 Compound Info	N-[4-[4-(2-chloro-3-ethylphenyl)piperazin-1-yl]butyl]-5-methyl-1H-imidazole-2-carboxamide Show/Hide	C21H30ClN5O	1
1	Ki = 0.621 nM Bioactivity Info	TI LI LO TS
CP0653272 Compound Info	4-(Dimethylamino)-N-(4-(4-(2-(2-fluoroethoxy)phenyl)piperazin-1-yl)butyl)benzamide oxalic acid salt Show/Hide	C27H37FN4O6	1
1	Ki = 0.65 nM Bioactivity Info	TI LI LO TS
CP0551018 Compound Info	US8748608, 47 Show/Hide	C24H28FN3O4	1
1	Ki = 0.65 nM Bioactivity Info	TI LI LO TS
CP0391046 Compound Info	N-[4-[4-(2-methylphenyl)piperazin-1-yl]butyl]-4-thiophen-3-ylbenzamide Show/Hide	C26H31N3OS	1
1	Ki = 0.68 nM Bioactivity Info	TI LI LO TS
CP0439252 Compound Info	7-((2-(4-(Naphthalen-2-yl)piperazin-1-yl)ethyl)(propyl)amino)-5,6,7,8-tetrahydronaphthalen-2-ol Show/Hide	C29H37N3O	1
1	Ki = 0.685 nM Bioactivity Info	TI LI LO TS
CP0393853 Compound Info	N-[4-[[(10R)-2-oxo-3-propyl-1,3-diazatricyclo[6.3.1.04,12]dodeca-4,6,8(12)-trien-10-yl]-propylamino]butyl]-1H-indole-2-carboxamide Show/Hide	C29H37N5O2	1
1	Ki = 0.69 nM Bioactivity Info	TI LI LO TS
CP0469462 Compound Info	N-[4-[4-(2-methoxyphenyl)-1,4-diazepan-1-yl]butyl]-4-thiophen-3-ylbenzamide Show/Hide	C27H33N3O2S	1
1	Ki = 0.7 nM Bioactivity Info	TI LI LO TS
CP0701083 Compound Info	endo-8-(Benzofur-3-ylmethyl)-3-(4-chlorophenyl)-8-azabicyclo[3.2.1]octan-3-ol Show/Hide	C22H22ClNO2	1
1	Ki = 0.71 nM Bioactivity Info	TI LI LO TS
CP0126478 Compound Info	N-[4-[4-(2-chloro-3-ethylphenyl)piperazin-1-yl]-3-fluorobutyl]-1H-indole-2-carboxamide Show/Hide	C25H30ClFN4O	1
1	Ki = 0.756 nM Bioactivity Info	TI LI LO TS
CP0266686 Compound Info	N-[4-[(4-ethynylcyclohex-3-en-1-yl)-propylamino]butyl]-4-phenylbenzamide Show/Hide	C28H34N2O	3
1	Ki = 0.78 nM Bioactivity Info	TI LI LO TS
2	Ki = 20 nM Bioactivity Info	TI LI LO TS
3	Ki = 870 nM Bioactivity Info	TI LI LO TS
CP0181036 Compound Info	4-(dimethylamino)-N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)benzamide Show/Hide	C24H34N4O2	1
1	Ki = 0.8 nM Bioactivity Info	TI LI LO TS
CP0478203 Compound Info	N-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butyl]-1-benzothiophene-3-carboxamide Show/Hide	C23H25Cl2N3OS	1
1	Ki = 0.8 nM Bioactivity Info	TI LI LO TS
CP0452361 Compound Info	(R)-6-((2-(4-phenylpiperazin-1-yl)ethyl)(propyl)amino)-5,6,7,8-tetrahydronaphthalen-1-ol Show/Hide	C25H35N3O	1
1	Ki = 0.825 nM Bioactivity Info	TI LI LO TS
CP0376400 Compound Info	(-)-(S)-6-((2-(4-phenylpiperazin-1-yl)ethyl)(propyl)amino)-5,6,7,8-tetrahydronaphthalen-1-ol Show/Hide	C25H35N3O	1
1	Ki = 0.825 nM Bioactivity Info	TI LI LO TS
CP0565212 Compound Info	N-[(3S)-4-[4-(2-chloro-3-ethylphenyl)piperazin-1-yl]-3-fluorobutyl]-1H-indole-2-carboxamide Show/Hide	C25H30ClFN4O	1
1	Ki = 0.84 nM Bioactivity Info	TI LI LO TS
CP0063623 Compound Info	N-[(3S)-4-[4-(2-chloro-3-ethylphenyl)piperazin-1-yl]-3-hydroxybutyl]-1H-indole-2-carboxamide Show/Hide	C25H31ClN4O2	1
1	Ki = 0.886 nM Bioactivity Info	TI LI LO TS
CP0481572 Compound Info	N-[2-[(1S,2R)-2-[(7-cyano-3,4-dihydro-1H-isoquinolin-2-yl)methyl]cyclopropyl]ethyl]-1H-indole-2-carboxamide Show/Hide	C25H26N4O	1
1	Ki = 0.89 nM Bioactivity Info	TI LI LO TS
CP0554781 Compound Info	N-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butyl]-4-thiophen-3-ylbenzamide Show/Hide	C25H27Cl2N3OS	1
1	Ki = 0.89 nM Bioactivity Info	TI LI LO TS
CP0902370 Compound Info	8-(Benzofuran-3-ylmethyl)-3-((1-(2-fluoroethyl)-1H-1,2,3-triazol-4-yl)methyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one oxalate Show/Hide	C29H31FN6O6	1
1	Ki = 0.9 nM Bioactivity Info	TI LI LO TS
CP0772206 Compound Info	SID56463240 Show/Hide	C26H32ClN3O2	1
1	Ki = 0.9 nM Bioactivity Info	TI LI LO TS
CP0860172 Compound Info	N-(4-(4-(2-(2-fluoroethoxy)phenyl)piperazin-1-yl)butyl)-1H-indole-3-carboxamide oxalic acid Show/Hide	C27H33FN4O6	1
1	Ki = 0.9 nM Bioactivity Info	TI LI LO TS
CP0376253 Compound Info	N-[4-[4-(3-chloro-2-methoxyphenyl)piperazin-1-yl]butyl]-1-benzofuran-2-carboxamide Show/Hide	C24H28ClN3O3	1
1	Ki = 0.907 nM Bioactivity Info	TI LI LO TS
CP0918928 Compound Info	endo-8-(Benzofur-3-ylmethyl)-3-(4-bromophenyl)-8-azabicyclo-[3.2.1]octan-3-ol Show/Hide	C22H22BrNO2	1
1	Ki = 0.92 nM Bioactivity Info	TI LI LO TS
CP0402710 Compound Info	(S)-N6-[2-(4-Biphenyl-4-yl-piperazin-1-yl)-ethyl]-N6-propyl-4,5,6,7-tetrahydro-benzothiazole-2,6-diamine Show/Hide	C28H37N5S	1
1	Ki = 0.92 nM Bioactivity Info	TI LI LO TS
CP0127400 Compound Info	(-)-Pramipexole Show/Hide	C10H17N3S	7
1	Ki = 0.94 nM Bioactivity Info	TI LI LO TS
2	Ki = 1.1 nM Bioactivity Info	TI LI LO TS
3	Ki = 1.32 nM Bioactivity Info	TI LI LO TS
4	Ki = 5.6 nM Bioactivity Info	TI LI LO TS
5	Ki = 8.2 nM Bioactivity Info	TI LI LO TS
6	Ki = 13 nM Bioactivity Info	TI LI LO TS
7	Ki = 17 nM Bioactivity Info	TI LI LO TS
CP0561496 Compound Info	N-[4-[4-(2-chloro-3-ethylphenyl)piperazin-1-yl]butyl]-5-methylimidazo[2,1-b][1,3]thiazole-6-carboxamide Show/Hide	C23H30ClN5OS	1
1	Ki = 0.941 nM Bioactivity Info	TI LI LO TS
CP0250704 Compound Info	N-[4-[4-(2-chloro-3-ethylphenyl)piperazin-1-yl]-3-hydroxybutyl]-1-benzofuran-2-carboxamide Show/Hide	C25H30ClN3O3	1
1	Ki = 0.985 nM Bioactivity Info	TI LI LO TS
CP0508620 Compound Info	N-[4-[2,3-dihydro-1H-inden-2-yl(propyl)amino]butyl]-2-phenylbenzamide Show/Hide	C29H34N2O	2
1	Ki = 1 nM Bioactivity Info	TI LI LO TS
2	Ki = 230 nM Bioactivity Info	TI LI LO TS
CP0400385 Compound Info	5-[4-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butyl]triazol-1-yl]-1H-indole Show/Hide	C24H26Cl2N6	1
1	Ki = 1 nM Bioactivity Info	TI LI LO TS
CP0042927 Compound Info	7-{4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butoxy}-3,4-dihydroquinolin-2(1H)-one Show/Hide	C23H27Cl2N3O2	4
1	Ki = 1 nM Bioactivity Info	TI LI LO TS
2	Ki = 3.57 nM Bioactivity Info	TI LI LO TS
3	Ki = 6.8 nM Bioactivity Info	TI LI LO TS
4	Ki = 9.7 nM Bioactivity Info	TI LI LO TS
CP0546535 Compound Info	US8748608, 49 Show/Hide	C25H31N3O5	1
1	Ki = 1 nM Bioactivity Info	TI LI LO TS
CP0722004 Compound Info	4-(2-Fluoroethyl)-N-(4-(4-(2-(2-Fluoroethoxy)phenyl)piperazin-1-yl)-trans-butyl-2-enyl)benzamide oxalic acid salt Show/Hide	C27H33F2N3O6	1
1	Ki = 1.1 nM Bioactivity Info	TI LI LO TS
CP0786650 Compound Info	4-(2-Fluoroethoxy)-N-(4-(4-(2-methoxyphenyl)-piperazin-1-yl)-butyl)benzamide oxalic acid salt Show/Hide	C26H34FN3O7	1
1	Ki = 1.1 nM Bioactivity Info	TI LI LO TS
CP0844267 Compound Info	4-(Thiophen-3-yl)-N-(4-(4-(2-(2-fluoroethoxy)phenyl)piperazin-1-yl)-trans-but-2-enyl)benzamides oxalic acid salt Show/Hide	C29H32FN3O6S	1
1	Ki = 1.1 nM Bioactivity Info	TI LI LO TS
CP0883761 Compound Info	(2S,4aR,10bR)-2-(4-hydroxyphenyl)-4-propyl-1,2,3,4,4a,5,6,10b-octahydrobenzo[f]quinoline-8,9-diol hydrobromide Show/Hide	C22H28BrNO3	1
1	Ki = 1.1 nM Bioactivity Info	TI LI LO TS
CP0869497 Compound Info	5-(2-(2-Fluoroethoxy)ethoxy)-N-(4-(4-(2-methoxyphenyl)-piperazin-1-yl)butyl)-1H-indole-2-carboxamide oxalic acid Show/Hide	C30H39FN4O8	1
1	Ki = 1.1 nM Bioactivity Info	TI LI LO TS
CP0422348 Compound Info	7-({2-[4-(2,3-Dichloro-phenyl)-piperazin-1-yl]-ethyl}-propyl-amino)-5,6,7,8-tetrahydro-naphthalen-2-ol Show/Hide	C25H33Cl2N3O	1
1	Ki = 1.13 nM Bioactivity Info	TI LI LO TS
CP0847582 Compound Info	(+/-)-11-(3-(4-((4-(2-Methoxyphenyl)piperazin-1-yl)ethyl)-1H-1,2,3-triazol-1-yl)propoxy)-N-propylnoraporphine Show/Hide	C37H46N6O2	1
1	Ki = 1.14 nM Bioactivity Info	TI LI LO TS
CP0421285 Compound Info	N-[4-[4-(2-chloro-3-ethylphenyl)piperazin-1-yl]butyl]-5-ethyl-1H-imidazole-2-carboxamide Show/Hide	C22H32ClN5O	1
1	Ki = 1.14 nM Bioactivity Info	TI LI LO TS
CP0881592 Compound Info	endo-8-(Benzofur-3-ylmethyl)-3-(4-fluorophenyl)-8-azabicyclo[3.2.1]octan-3-ol Show/Hide	C22H22FNO2	1
1	Ki = 1.2 nM Bioactivity Info	TI LI LO TS
CP0402682 Compound Info	(-)-(S)-N6-Propyl-N6-(2-(4-(quinolin-5-yl)piperazin-1-yl)ethyl)-4,5,6,7-tetrahydrobenzo[d]thiazole-2,6-diamine Show/Hide	C25H34N6S	1
1	Ki = 1.21 nM Bioactivity Info	TI LI LO TS
CP0452975 Compound Info	7-(Propyl(2-(4-(quinolin-5-yl)piperazin-1-yl)ethyl)amino)-5,6,7,8-tetrahydronaphthalen-2-ol Show/Hide	C28H36N4O	1
1	Ki = 1.27 nM Bioactivity Info	TI LI LO TS
CP0424341 Compound Info	N-[(E)-4-[4-(2-chloro-3-ethylphenyl)piperazin-1-yl]but-2-enyl]-5-methyl-1H-imidazole-2-carboxamide Show/Hide	C21H28ClN5O	1
1	Ki = 1.28 nM Bioactivity Info	TI LI LO TS
CP0510175 Compound Info	US8748608, 23 Show/Hide	C29H33N3O3	1
1	Ki = 1.3 nM Bioactivity Info	TI LI LO TS
CP0480941 Compound Info	US8748608, 48 Show/Hide	C24H27Cl2N3O4	1
1	Ki = 1.3 nM Bioactivity Info	TI LI LO TS
CP0909483 Compound Info	6-(1-(4-(4-(2,3-Dichlorophenyl)piperazin-1-yl)butyl)-1H-1,2,3-triazol-4-yl)quinoline Show/Hide	C25H26Cl2N6	1
1	Ki = 1.35 nM Bioactivity Info	TI LI LO TS
CP0103545 Compound Info	(-)-5-hydroxy-2-(dipropylamino)tetralin Show/Hide	C16H25NO	1
1	Ki = 1.36 nM Bioactivity Info	TI LI LO TS
CP0384350 Compound Info	6-[(2-(4-phenylpiperazin-1-yl)ethyl)(propyl)amino]-5,6,7,8-tetrahydronaphthalene-2,3-diol Show/Hide	C25H35N3O2	1
1	Ki = 1.39 nM Bioactivity Info	TI LI LO TS
CP0394596 Compound Info	(+)-7-{[4-(4-phenylpiperazin-1-yl)butyl]prop-2-ynylamino}-5,6,7,8-tetrahydronaphthalen-2-ol Show/Hide	C27H35N3O	1
1	Ki = 1.4 nM Bioactivity Info	TI LI LO TS
CP0042204 Compound Info	1H-Indole-2-carboxylic acid {4-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-butyl}-amide Show/Hide	C23H26Cl2N4O	1
1	Ki = 1.4 nM Bioactivity Info	TI LI LO TS
CP0456795 Compound Info	N-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butyl]-9-oxofluorene-2-carboxamide Show/Hide	C28H27Cl2N3O2	1
1	Ki = 1.4 nM Bioactivity Info	TI LI LO TS
CP0443217 Compound Info	5-[1-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butyl]triazol-4-yl]-1H-indole Show/Hide	C24H26Cl2N6	1
1	Ki = 1.47 nM Bioactivity Info	TI LI LO TS
CP0162854 Compound Info	(+/-)-7-(dipropylamino)-5,6,7,8-tetrahydronaphthalen-2-ol Show/Hide	C16H25NO	6
1	Ki = 1.49 nM Bioactivity Info	TI LI LO TS
2	Ki = 1.75 nM Bioactivity Info	TI LI LO TS
3	Ki = 2.35 nM Bioactivity Info	TI LI LO TS
4	Ki = 3.6 nM Bioactivity Info	TI LI LO TS
5	Ki = 270 nM Bioactivity Info	TI LI LO TS
6	Ki = 1400 nM Bioactivity Info	TI LI LO TS
CP0190973 Compound Info	N-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]-3-fluorobutyl]-5-methoxy-1H-indole-2-carboxamide Show/Hide	C24H27Cl2FN4O2	1
1	Ki = 1.5 nM Bioactivity Info	TI LI LO TS
CP0381642 Compound Info	N-[4-[4-(2-methoxyphenyl)-1,4-diazepan-1-yl]butyl]-1-benzothiophene-2-carboxamide Show/Hide	C25H31N3O2S	1
1	Ki = 1.5 nM Bioactivity Info	TI LI LO TS
CP0898479 Compound Info	5-(2-(2-(2-Fluoroethoxy)ethoxy)ethoxy)-N-(4-(4-(2-methoxy-phenyl)piperazin-1-yl)butyl)-1H-indole-2-carboxamide oxalic acid Show/Hide	C32H43FN4O9	1
1	Ki = 1.5 nM Bioactivity Info	TI LI LO TS
CP0554865 Compound Info	4-thiophen-3-yl-N-[4-[4-[2-(trifluoromethyl)phenyl]piperazin-1-yl]butyl]benzamide Show/Hide	C26H28F3N3OS	1
1	Ki = 1.5 nM Bioactivity Info	TI LI LO TS
CP0396214 Compound Info	N-[[(1R,2R)-2-[[4-(2,3-dichlorophenyl)piperazin-1-yl]methyl]cyclopropyl]methyl]quinoline-4-carboxamide Show/Hide	C25H26Cl2N4O	1
1	Ki = 1.51 nM Bioactivity Info	TI LI LO TS
CP0378423 Compound Info	7-((2-(4-phenylpiperazin-1-yl)ethyl)(propyl)amino)-5,6,7,8-tetrahydronaphthalen-2-ol Show/Hide	C25H35N3O	2
1	Ki = 1.56 nM Bioactivity Info	TI LI LO TS
2	Ki = 1.75 nM Bioactivity Info	TI LI LO TS
CP0410742 Compound Info	1-[4-[1-(9H-fluoren-2-yl)triazol-4-yl]butyl]-4-(2-methoxyphenyl)piperazine Show/Hide	C30H33N5O	1
1	Ki = 1.59 nM Bioactivity Info	TI LI LO TS
CP0548699 Compound Info	US8748608, 46 Show/Hide	C23H24Cl2FN3O3	1
1	Ki = 1.6 nM Bioactivity Info	TI LI LO TS
CP0053493 Compound Info	(+)-1-Propyl-2,3,10,10a-tetrahydro-1H,4aH-4,9-dioxa-1-aza-phenanthren-6-ol Show/Hide	C14H19NO3	2
1	Ki = 1.67 nM Bioactivity Info	TI LI LO TS
2	Ki = 1.69 nM Bioactivity Info	TI LI LO TS
CP0439502 Compound Info	(+)-(R)-7-((2-(4-phenylpiperazin-1-yl)ethyl)(propyl)amino)-5,6,7,8-tetrahydronaphthalen-2-ol Show/Hide	C25H35N3O	1
1	Ki = 1.77 nM Bioactivity Info	TI LI LO TS
CP0397773 Compound Info	4-ethenyl-N-[4-[4-(2-methoxyphenyl)-1,4-diazepan-1-yl]butyl]benzamide Show/Hide	C25H33N3O2	1
1	Ki = 1.8 nM Bioactivity Info	TI LI LO TS
CP0410571 Compound Info	5-[4-[5-[4-(2-methoxyphenyl)piperazin-1-yl]pentyl]triazol-1-yl]isoquinoline Show/Hide	C27H32N6O	1
1	Ki = 1.8 nM Bioactivity Info	TI LI LO TS
CP0473216 Compound Info	(-)-S-11-(3-(4-((4-(2-Methoxyphenyl)piperazin-1-yl)ethyl)-1H-1,2,3-triazol-1-yl)propoxy)-N-propylnoraporphine Show/Hide	C37H46N6O2	1
1	Ki = 1.82 nM Bioactivity Info	TI LI LO TS
CP0444479 Compound Info	N-[2-[(1R,2S)-2-[[(2S,5S)-2-(6-aminopyridin-3-yl)-5-methylmorpholin-4-yl]methyl]cyclopropyl]ethyl]-1H-indole-2-carboxamide Show/Hide	C25H31N5O2	2
1	Ki = 1.85 nM Bioactivity Info	TI LI LO TS
2	Ki = 5.36 nM Bioactivity Info	TI LI LO TS
CP0424070 Compound Info	1-butyl-4-(2,3-dichlorophenyl)piperazine Show/Hide	C14H20Cl2N2	1
1	Ki = 1.9 nM Bioactivity Info	TI LI LO TS
CP0059097 Compound Info	N-[4-[4-(3-chloro-2-methoxyphenyl)piperazin-1-yl]butyl]quinoline-3-carboxamide Show/Hide	C25H29ClN4O2	1
1	Ki = 1.99 nM Bioactivity Info	TI LI LO TS
CP0008601 Compound Info	4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1-(4-fluoro-phenyl)-butan-1-one;propionate(HCl) Show/Hide	C21H23ClFNO2	3
1	Ki = 2 nM Bioactivity Info	TI LI LO TS
2	Ki = 12.7 nM Bioactivity Info	TI LI LO TS
3	Ki = 29 nM Bioactivity Info	TI LI LO TS
CP0879780 Compound Info	endo-8-(Naphtho[1,2-b]fur-3-ylmethyl)-3-(4-chlorophenyl)-8-azabicyclo[3.2.1]octan-3-ol Show/Hide	C26H24ClNO2	1
1	Ki = 2 nM Bioactivity Info	TI LI LO TS
CP0869500 Compound Info	(E)-N-(4-(4-(2-(2-Fluoroethoxy)phenyl)piperazin-1-yl)but-2-en-1-yl)-1H-indole-2-carboxamide oxalic acid Show/Hide	C27H31FN4O6	1
1	Ki = 2 nM Bioactivity Info	TI LI LO TS
CP0869616 Compound Info	endo-8-(5-Methoxybenzofur-3-ylmethyl)-3-(4-chlorophenyl)-8-azabicyclo[3.2.1]octan-3-ol Show/Hide	C23H24ClNO3	1
1	Ki = 2.1 nM Bioactivity Info	TI LI LO TS
CP0919567 Compound Info	8-(Benzofuran-3-ylmethyl)-3-methyl-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one oxalate Show/Hide	C25H27N3O6	1
1	Ki = 2.1 nM Bioactivity Info	TI LI LO TS
CP0116811 Compound Info	5-Bromo-N-{4-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-butyl}-2,3-dimethoxy-benzamide Show/Hide	C23H28BrCl2N3O3	1
1	Ki = 2.1 nM Bioactivity Info	TI LI LO TS
CP0362283 Compound Info	1-(2-methoxyphenyl)-4-[4-[1-(4-methylsulfanylphenyl)triazol-4-yl]butyl]piperazine Show/Hide	C24H31N5OS	1
1	Ki = 2.1 nM Bioactivity Info	TI LI LO TS
CP0156136 Compound Info	N-[4-[4-(2-chloro-5-methylphenyl)piperazin-1-yl]butyl]-2-oxo-3H-1,3-benzoxazole-5-carboxamide Show/Hide	C23H27ClN4O3	2
1	Ki = 2.11 nM Bioactivity Info	TI LI LO TS
2	Ki = 3.04 nM Bioactivity Info	TI LI LO TS
CP0494802 Compound Info	6-fluoro-N-[4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]quinoline-3-carboxamide Show/Hide	C25H29FN4O2	1
1	Ki = 2.14 nM Bioactivity Info	TI LI LO TS
CP0411950 Compound Info	(-)-(S)-N6-(2-(4-(Isoquinolin-1-yl)piperazin-1-yl)ethyl)-N6-propyl-4,5,6,7-tetrahydrobenzo[d]-thiazole-2,6-diamine Show/Hide	C25H34N6S	1
1	Ki = 2.23 nM Bioactivity Info	TI LI LO TS
CP0438793 Compound Info	7-({4-[4-(2,3-Dichloro-phenyl)-piperazin-1-yl]-butyl}-propyl-amino)-5,6,7,8-tetrahydro-naphthalen-2-ol Show/Hide	C27H37Cl2N3O	1
1	Ki = 2.26 nM Bioactivity Info	TI LI LO TS
CP0234732 Compound Info	1-(2-methoxyphenyl)-4-[5-[1-(4-methylsulfanylphenyl)triazol-4-yl]pentyl]piperazine Show/Hide	C25H33N5OS	1
1	Ki = 2.3 nM Bioactivity Info	TI LI LO TS
CP0044536 Compound Info	(2R)-7-Dipropylamino-5,6,7,8-tetrahydro-naphthalen-2-ol Show/Hide	C16H25NO	1
1	Ki = 2.35 nM Bioactivity Info	TI LI LO TS
CP0231075 Compound Info	4-(2-fluoroethyl)-N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)benzamide Show/Hide	C24H32FN3O2	1
1	Ki = 2.4 nM Bioactivity Info	TI LI LO TS
CP0467853 Compound Info	7-[4-[4-(2-chloro-3-ethylphenyl)piperazin-1-yl]butoxy]-3,4-dihydro-1H-quinolin-2-one Show/Hide	C25H32ClN3O2	1
1	Ki = 2.42 nM Bioactivity Info	TI LI LO TS
CP0463698 Compound Info	N-[4-[methyl-[(10R)-2-oxo-3-propyl-1,3-diazatricyclo[6.3.1.04,12]dodeca-4,6,8(12)-trien-10-yl]amino]butyl]-1H-indole-2-carboxamide Show/Hide	C27H33N5O2	1
1	Ki = 2.45 nM Bioactivity Info	TI LI LO TS
CP0063614 Compound Info	N-[4-[4-(2-chloro-3-ethylphenyl)piperazin-1-yl]-3-fluorobutyl]-1-benzofuran-2-carboxamide Show/Hide	C25H29ClFN3O2	1
1	Ki = 2.45 nM Bioactivity Info	TI LI LO TS
CP0473012 Compound Info	N-[2-[(1S,2R)-2-[(7-cyano-3,4-dihydro-1H-isoquinolin-2-yl)methyl]cyclopropyl]ethyl]-1H-pyrrolo[2,3-b]pyridine-2-carboxamide Show/Hide	C24H25N5O	1
1	Ki = 2.47 nM Bioactivity Info	TI LI LO TS
CP0389512 Compound Info	4-ethynyl-N-[4-[4-(4-phenylphenyl)triazol-1-yl]butyl]-N-propylcyclohex-3-en-1-amine Show/Hide	C29H34N4	3
1	Ki = 2.5 nM Bioactivity Info	TI LI LO TS
2	Ki = 33 nM Bioactivity Info	TI LI LO TS
3	Ki = 1500 nM Bioactivity Info	TI LI LO TS
CP0384905 Compound Info	US8748608, 22 Show/Hide	C28H29Cl2N3O2	1
1	Ki = 2.5 nM Bioactivity Info	TI LI LO TS
CP0856731 Compound Info	4-(2-(2-Fluoroethoxy)ethoxy)-N-(4-(4-(2-(2-fluoroethoxy)phenyl)piperazin-1-yl)butyl)benzamide oxalic acid salt Show/Hide	C29H39F2N3O8	1
1	Ki = 2.5 nM Bioactivity Info	TI LI LO TS
CP0397772 Compound Info	N-[4-[4-(2-methoxyphenyl)-1,4-diazepan-1-yl]butyl]-1H-indole-2-carboxamide Show/Hide	C25H32N4O2	1
1	Ki = 2.5 nM Bioactivity Info	TI LI LO TS
CP0528747 Compound Info	6-fluoro-N-[4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]quinoline-2-carboxamide Show/Hide	C25H29FN4O2	1
1	Ki = 2.51 nM Bioactivity Info	TI LI LO TS
CP0329850 Compound Info	N-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]-3-fluorobutyl]-9H-fluorene-2-carboxamide Show/Hide	C28H28Cl2FN3O	1
1	Ki = 2.6 nM Bioactivity Info	TI LI LO TS
CP0402681 Compound Info	(-)-(S)-N6-Propyl-N6-(2-(4-(quinolin-4-yl)piperazin-1-yl)ethyl)-4,5,6,7-tetrahydrobenzo[d]thiazole-2,6-diamine Show/Hide	C25H34N6S	1
1	Ki = 2.61 nM Bioactivity Info	TI LI LO TS
CP0060505 Compound Info	N-[3-[2-[[2-(4-chlorophenyl)cyclopropyl]-propylamino]ethyl]-3-hydroxycyclobutyl]naphthalene-2-carboxamide Show/Hide	C29H33ClN2O2	1
1	Ki = 2.61 nM Bioactivity Info	TI LI LO TS
CP0452974 Compound Info	7-(Propyl(2-(4-(quinolin-4-yl)piperazin-1-yl)ethyl)amino)-5,6,7,8-tetrahydronaphthalen-2-ol Show/Hide	C28H36N4O	1
1	Ki = 2.65 nM Bioactivity Info	TI LI LO TS
CP0906113 Compound Info	(+/-)-11-((1-(3-(4-(2-Methoxyphenyl)piperazin-1-yl)butyl)-1H-1,2,3-triazol-4-yl)methoxy)-N-propylnoraporphine Show/Hide	C37H46N6O2	1
1	Ki = 2.67 nM Bioactivity Info	TI LI LO TS
CP0501590 Compound Info	N-[4-[2,3-dihydro-1H-inden-2-yl(propyl)amino]butyl]-2-phenylacetamide Show/Hide	C24H32N2O	2
1	Ki = 2.7 nM Bioactivity Info	TI LI LO TS
2	Ki = 250 nM Bioactivity Info	TI LI LO TS
CP0887640 Compound Info	7-(4-(4-(2-(2-Fluoroethoxy)phenyl)piperazin-1-yl)butoxy)quinolin-2(1H)-one oxalate Show/Hide	C27H32FN3O7	1
1	Ki = 2.7 nM Bioactivity Info	TI LI LO TS
CP0434739 Compound Info	N-[3-[2-[[(1R,2S)-2-(4-chlorophenyl)cyclopropyl]-propylamino]ethyl]-3-hydroxycyclobutyl]naphthalene-2-carboxamide Show/Hide	C29H33ClN2O2	1
1	Ki = 2.8 nM Bioactivity Info	TI LI LO TS
CP0434349 Compound Info	6-[(4-(4-phenylpiperazin-1-yl)butyl)(propyl)amino]-5,6,7,8-tetrahydronaphthalene-2,3-diol Show/Hide	C27H39N3O2	1
1	Ki = 2.89 nM Bioactivity Info	TI LI LO TS
CP0038047 Compound Info	N-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]-3-fluorobutyl]-1-benzothiophene-2-carboxamide Show/Hide	C23H24Cl2FN3OS	1
1	Ki = 2.9 nM Bioactivity Info	TI LI LO TS
CP0396653 Compound Info	N-[4-[4-(2-methoxyphenyl)-1,4-diazepan-1-yl]butyl]-4-methylsulfanylbenzamide Show/Hide	C24H33N3O2S	1
1	Ki = 2.9 nM Bioactivity Info	TI LI LO TS
CP0386825 Compound Info	N-[4-[4-[3-(trifluoromethyl)phenyl]piperazin-1-yl]butyl]imidazo[1,2-a]pyridine-2-carboxamide Show/Hide	C23H26F3N5O	1
1	Ki = 2.9 nM Bioactivity Info	TI LI LO TS
CP0555052 Compound Info	2-[4-[4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]triazol-1-yl]phenol Show/Hide	C23H29N5O2	1
1	Ki = 2.9 nM Bioactivity Info	TI LI LO TS
CP0417544 Compound Info	N-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]-3-hydroxybutyl]quinoline-3-carboxamide Show/Hide	C24H26Cl2N4O2	2
1	Ki = 2.91 nM Bioactivity Info	TI LI LO TS
2	Ki = 4.26 nM Bioactivity Info	TI LI LO TS
CP0400383 Compound Info	1-(2-methoxyphenyl)-4-[4-(1-naphthalen-2-yltriazol-4-yl)butyl]piperazine Show/Hide	C27H31N5O	1
1	Ki = 2.93 nM Bioactivity Info	TI LI LO TS
CP0861001 Compound Info	1-(1-(Benzofuran-3-ylmethyl)piperidin-4-yl)-1Hbenzo[d]imidazol-2-(3H)-one oxalate Show/Hide	C23H23N3O6	1
1	Ki = 3 nM Bioactivity Info	TI LI LO TS
CP0898311 Compound Info	(E)-5-Methoxy-N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)but-2-en-1-yl)-1H-indole-3-carboxamide oxalic acid Show/Hide	C27H32N4O7	1
1	Ki = 3 nM Bioactivity Info	TI LI LO TS
CP0530038 Compound Info	N-[4-[4-(2-chloro-3-ethylphenyl)piperazin-1-yl]-3-hydroxybutyl]-1,3-benzodioxole-5-carboxamide Show/Hide	C24H30ClN3O4	1
1	Ki = 3.02 nM Bioactivity Info	TI LI LO TS
CP0869499 Compound Info	(E)-N-(4-(4-(2-(2-Fluoroethoxy)phenyl)piperazin-1-yl)but-2-en-1-yl)-5-methoxy-1H-indole-2-carboxamide oxalic acid Show/Hide	C28H33FN4O7	1
1	Ki = 3.1 nM Bioactivity Info	TI LI LO TS
CP0410572 Compound Info	1-(2-methoxyphenyl)-4-[5-(1-phenyltriazol-4-yl)pentyl]piperazine Show/Hide	C24H31N5O	1
1	Ki = 3.1 nM Bioactivity Info	TI LI LO TS
CP0444621 Compound Info	5-[4-[4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]triazol-1-yl]-1H-indole Show/Hide	C25H30N6O	1
1	Ki = 3.1 nM Bioactivity Info	TI LI LO TS
CP0456678 Compound Info	5-[5-[3-[(1S,5R)-1-[2-fluoro-4-(trifluoromethyl)phenyl]-3-azabicyclo[3.1.0]hexan-3-yl]propylsulfanyl]-4-methyl-1,2,4-triazol-3-yl]-4-methyl-1,3-oxazole Show/Hide	C22H23F4N5OS	1
1	Ki = 3.15 nM Bioactivity Info	TI LI LO TS
CP0224533 Compound Info	N-[4-[4-(3-chloro-5-ethyl-2-methoxyphenyl)piperazin-1-yl]butyl]-1-benzofuran-2-carboxamide Show/Hide	C26H32ClN3O3	1
1	Ki = 3.19 nM Bioactivity Info	TI LI LO TS
CP0869498 Compound Info	(E)-N-(4-(4-(2-(2-fluoroethoxy)phenyl)piperazin-1-yl)but-2-en-1-yl)-5-methoxy-1H-indole-3-carboxamide oxalic acid Show/Hide	C28H33FN4O7	1
1	Ki = 3.2 nM Bioactivity Info	TI LI LO TS
CP0397121 Compound Info	1-[5-[1-(4-fluorophenyl)triazol-4-yl]pentyl]-4-(2-methoxyphenyl)piperazine Show/Hide	C24H30FN5O	1
1	Ki = 3.2 nM Bioactivity Info	TI LI LO TS
CP0477399 Compound Info	3-(2-methoxyphenyl)-9-[3-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]propyl]-3,9-diazaspiro[5.5]undec-4-ene Show/Hide	C28H35N5OS	1
1	Ki = 3.2 nM Bioactivity Info	TI LI LO TS
CP0393847 Compound Info	(10R)-10-(dipropylamino)-3-propyl-1,3-diazatricyclo[6.3.1.04,12]dodeca-4,6,8(12)-trien-2-one Show/Hide	C19H29N3O	2
1	Ki = 3.39 nM Bioactivity Info	TI LI LO TS
2	Ki = 6.05 nM Bioactivity Info	TI LI LO TS
CP0375780 Compound Info	N-[3-[4-(2-methylsulfanylphenyl)piperazin-1-yl]propyl]pyrazolo[1,5-a]pyridine-3-carboxamide Show/Hide	C22H27N5OS	8
1	Ki = 3.4 nM Bioactivity Info	TI LI LO TS
2	Ki = 8 nM Bioactivity Info	TI LI LO TS
3	Ki = 17 nM Bioactivity Info	TI LI LO TS
4	Ki = 26 nM Bioactivity Info	TI LI LO TS
5	Ki = 320 nM Bioactivity Info	TI LI LO TS
6	Ki = 430 nM Bioactivity Info	TI LI LO TS
7	Ki = 650 nM Bioactivity Info	TI LI LO TS
8	Ki = 740 nM Bioactivity Info	TI LI LO TS
CP0407878 Compound Info	N-[4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]quinoline-2-carboxamide Show/Hide	C25H30N4O2	1
1	Ki = 3.46 nM Bioactivity Info	TI LI LO TS
CP0386823 Compound Info	N-[4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]imidazo[1,2-a]pyridine-2-carboxamide Show/Hide	C23H29N5O2	1
1	Ki = 3.5 nM Bioactivity Info	TI LI LO TS
CP0438619 Compound Info	7-({4-[4-(2,3-Dichloro-phenyl)-piperazin-1-yl]-butyl}-prop-2-ynyl-amino)-5,6,7,8-tetrahydro-naphthalen-2-ol Show/Hide	C27H33Cl2N3O	1
1	Ki = 3.59 nM Bioactivity Info	TI LI LO TS
CP0847307 Compound Info	4-(Dimethylamino)-N-(4-(4-(2-(2-fluoroethoxy)phenyl)piperazin-1-yl)-trans-butyl-2-enyl)benzamide oxalic acid salt Show/Hide	C27H35FN4O6	1
1	Ki = 3.6 nM Bioactivity Info	TI LI LO TS
CP0701087 Compound Info	endo-8-(Benzothien-3-ylmethyl)-3-(4-chlorophenyl)-8-azabicyclo[3.2.1]octan-3-ol Show/Hide	C22H22ClNOS	1
1	Ki = 3.62 nM Bioactivity Info	TI LI LO TS
CP0109608 Compound Info	N-[3-hydroxy-4-(4-naphthalen-1-ylpiperazin-1-yl)butyl]quinoline-3-carboxamide Show/Hide	C28H30N4O2	1
1	Ki = 3.63 nM Bioactivity Info	TI LI LO TS
CP0397169 Compound Info	4-chloro-N-[4-[4-(2-methoxyphenyl)-1,4-diazepan-1-yl]butyl]benzamide Show/Hide	C23H30ClN3O2	1
1	Ki = 3.7 nM Bioactivity Info	TI LI LO TS
CP0869495 Compound Info	(E)-N-(4-(4-(2-(2-Fluoroethoxy)phenyl)piperazin-1-yl)but-2-en-1-yl)-6-methoxy-1H-indole-3-carboxamide oxalic acid Show/Hide	C28H33FN4O7	1
1	Ki = 3.7 nM Bioactivity Info	TI LI LO TS
CP0906704 Compound Info	(E)-5-(2-fluoroethoxy)-N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)but-2-en-1-yl)-1H-indole-2-carboxamide oxalic acid Show/Hide	C28H33FN4O7	1
1	Ki = 3.7 nM Bioactivity Info	TI LI LO TS
CP0362281 Compound Info	5-[4-[4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]triazol-1-yl]isoquinoline Show/Hide	C26H30N6O	1
1	Ki = 3.7 nM Bioactivity Info	TI LI LO TS
CP0375620 Compound Info	5-((4-(2-((5-Hydroxy-1,2,3,4-tetrahydronaphthalen-2-yl)(propyl)amino)ethyl)piperazin-1-yl)methyl)quinolin-8-ol Show/Hide	C28H36N4O2	1
1	Ki = 3.71 nM Bioactivity Info	TI LI LO TS
CP0402972 Compound Info	(+)-7-[(4-(4-phenylpiperazin-1-yl)butyl)(propyl)amino]-5,6,7,8-tetrahydronaphthalen-2-ol Show/Hide	C27H39N3O	1
1	Ki = 3.79 nM Bioactivity Info	TI LI LO TS
CP0294038 Compound Info	N-[3-fluoro-4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]-1-benzothiophene-2-carboxamide Show/Hide	C24H28FN3O2S	1
1	Ki = 3.8 nM Bioactivity Info	TI LI LO TS
CP0920165 Compound Info	7-(5-(4-(2-Methoxyphenyl)piperazin-1-yl)pentyloxy)quinolin-2(1H)-one oxalate Show/Hide	C27H33N3O7	1
1	Ki = 3.8 nM Bioactivity Info	TI LI LO TS
CP0033479 Compound Info	(chloropromazine) [3-(2-Chloro-phenothiazin-10-yl)-propyl]-dimethyl-amine Show/Hide	C17H19ClN2S	1
1	Ki = 3.8 nM Bioactivity Info	TI LI LO TS
CP0860158 Compound Info	(E)-5-(2-(2-Fluoroethoxy)ethoxy)-N-(4-(4-(2-methoxyphenyl)-piperazin-1-yl)but-2-en-1-yl)-1H-indole-2-carboxamide oxalic acid Show/Hide	C30H37FN4O8	1
1	Ki = 3.8 nM Bioactivity Info	TI LI LO TS
CP0389180 Compound Info	1-(2,3-dichlorophenyl)-4-[4-(1-naphthalen-2-yltriazol-4-yl)butyl]piperazine Show/Hide	C26H27Cl2N5	1
1	Ki = 3.8 nM Bioactivity Info	TI LI LO TS
CP0478827 Compound Info	N-[4-[4-(2,4-dichlorophenyl)piperazin-1-yl]butyl]-4-thiophen-3-ylbenzamide Show/Hide	C25H27Cl2N3OS	1
1	Ki = 3.8 nM Bioactivity Info	TI LI LO TS
CP0381617 Compound Info	4-(dimethylamino)-N-[4-[4-(2-methoxyphenyl)-1,4-diazepan-1-yl]butyl]benzamide Show/Hide	C25H36N4O2	1
1	Ki = 3.9 nM Bioactivity Info	TI LI LO TS
CP0115686 Compound Info	N-[4-[2-(7-cyano-3,4-dihydro-1H-isoquinolin-2-yl)ethyl]cyclohexyl]-1H-indole-2-carboxamide Show/Hide	C27H30N4O	1
1	Ki = 3.9 nM Bioactivity Info	TI LI LO TS
CP0847873 Compound Info	N-(Benzothiazol-2-yl)-5-(4-(2-fluorophenyl)piperazin-1-yl)pentanamide Show/Hide	C22H25FN4OS	1
1	Ki = 3.9 nM Bioactivity Info	TI LI LO TS
CP0258057 Compound Info	N-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]-3-fluorobutyl]-1H-indole-2-carboxamide Show/Hide	C23H25Cl2FN4O	1
1	Ki = 4 nM Bioactivity Info	TI LI LO TS
CP0906705 Compound Info	(E)-N-(4-(4-(2-(2-Fluoroethoxy)phenyl)piperazin-1-yl)but-2-en-1-yl)-5-hydroxy-1H-indole-2-carboxamide oxalic acid Show/Hide	C27H31FN4O7	1
1	Ki = 4 nM Bioactivity Info	TI LI LO TS
CP0471596 Compound Info	N-[(3R)-4-[4-(2,3-dichlorophenyl)piperazin-1-yl]-3-hydroxybutyl]quinoline-3-carboxamide Show/Hide	C24H26Cl2N4O2	1
1	Ki = 4.12 nM Bioactivity Info	TI LI LO TS
CP0771814 Compound Info	4-(2-(2-(2-Fluoroethoxy)ethoxy)ethoxy)-N-(4-(4-(2-methoxyphenyl)piperazin-1-l)butyl)benzamide oxalic acid salt Show/Hide	C30H42FN3O9	1
1	Ki = 4.2 nM Bioactivity Info	TI LI LO TS
CP0379465 Compound Info	N-[4-[4-[2-tert-butyl-6-(trifluoromethyl)pyrimidin-4-yl]piperazin-1-yl]butyl]imidazo[1,2-a]pyridine-2-carboxamide Show/Hide	C25H32F3N7O	6
1	Ki = 4.2 nM Bioactivity Info	TI LI LO TS
2	Ki = 8.4 nM Bioactivity Info	TI LI LO TS
3	Ki = 12 nM Bioactivity Info	TI LI LO TS
4	Ki = 13 nM Bioactivity Info	TI LI LO TS
5	Ki = 20 nM Bioactivity Info	TI LI LO TS
6	Ki = 40 nM Bioactivity Info	TI LI LO TS
CP0434495 Compound Info	N-[4-[4-(2-chloro-3-ethylphenyl)piperazin-1-yl]-3-hydroxybutyl]imidazo[1,2-a]pyridine-2-carboxamide Show/Hide	C24H30ClN5O2	1
1	Ki = 4.23 nM Bioactivity Info	TI LI LO TS
CP0386830 Compound Info	N-[4-[4-[2-tert-butyl-6-(trifluoromethyl)pyrimidin-4-yl]piperazin-1-yl]butyl]-1H-benzimidazole-2-carboxamide Show/Hide	C25H32F3N7O	1
1	Ki = 4.3 nM Bioactivity Info	TI LI LO TS
CP0565213 Compound Info	N-[4-[4-(6-ethyl-1,3-benzodioxol-5-yl)piperazin-1-yl]-3-hydroxybutyl]-1H-indole-2-carboxamide Show/Hide	C26H32N4O4	1
1	Ki = 4.31 nM Bioactivity Info	TI LI LO TS
CP0869494 Compound Info	(E)-5-Methoxy-N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)but-2-en-1-yl)-1H-indole-2-carboxamide oxalic acid Show/Hide	C27H32N4O7	1
1	Ki = 4.4 nM Bioactivity Info	TI LI LO TS
CP0273714 Compound Info	N-[3-fluoro-4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]-5-methoxy-1H-indole-2-carboxamide Show/Hide	C25H31FN4O3	1
1	Ki = 4.6 nM Bioactivity Info	TI LI LO TS
CP0410743 Compound Info	1-(2-methoxyphenyl)-4-[4-(1-phenyltriazol-4-yl)butyl]piperazine Show/Hide	C23H29N5O	2
1	Ki = 4.7 nM Bioactivity Info	TI LI LO TS
2	Ki = 5.42 nM Bioactivity Info	TI LI LO TS
CP0402706 Compound Info	(-)-(S)-N6-Propyl-N6-(2-(4-(4-(pyridin-4-yl)phenyl)piperazin-1-yl)-ethyl)-4,5,6,7-tetrahydrobenzo[d]-thiazole-2,6-diamine Show/Hide	C27H36N6S	1
1	Ki = 4.78 nM Bioactivity Info	TI LI LO TS
CP0488181 Compound Info	N-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butyl]propanamide Show/Hide	C17H25Cl2N3O	1
1	Ki = 4.8 nM Bioactivity Info	TI LI LO TS
CP0396657 Compound Info	5-bromo-N-[4-[4-(2-methoxyphenyl)-1,4-diazepan-1-yl]butyl]thiophene-2-carboxamide Show/Hide	C21H28BrN3O2S	1
1	Ki = 4.8 nM Bioactivity Info	TI LI LO TS
CP0433590 Compound Info	1-(2,3-dichlorophenyl)-4-[4-[1-(9H-fluoren-2-yl)triazol-4-yl]butyl]piperazine Show/Hide	C29H29Cl2N5	1
1	Ki = 5.05 nM Bioactivity Info	TI LI LO TS
CP0860667 Compound Info	4-(2-(2-(2-Fluoroethoxy)ethoxy)ethoxy)-N-(4-(4-(2-(2-fluoroethoxy)phenyl)piperazin-1-yl)butyl)benzamide oxalic acid salt Show/Hide	C31H43F2N3O9	1
1	Ki = 5.2 nM Bioactivity Info	TI LI LO TS
CP0913681 Compound Info	7-(4-(4-(2-Methoxyphenyl)piperazin-1-yl)butoxy)quinolin-2(1H)-one oxalate Show/Hide	C26H31N3O7	1
1	Ki = 5.4 nM Bioactivity Info	TI LI LO TS
CP0389480 Compound Info	5-[1-[4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]triazol-4-yl]-1H-indole Show/Hide	C25H30N6O	1
1	Ki = 5.48 nM Bioactivity Info	TI LI LO TS
CP0375438 Compound Info	N-[4-[4-(2-methoxyphenyl)-1,4-diazepan-1-yl]butyl]-1-benzofuran-2-carboxamide Show/Hide	C25H31N3O3	1
1	Ki = 5.5 nM Bioactivity Info	TI LI LO TS
CP0410746 Compound Info	1-[4-[4-(9H-fluoren-2-yl)triazol-1-yl]butyl]-4-(2-methoxyphenyl)piperazine Show/Hide	C30H33N5O	1
1	Ki = 5.55 nM Bioactivity Info	TI LI LO TS
CP0430951 Compound Info	5-((4-(2-((7-Hydroxy-1,2,3,4-tetrahydronaphthalen-2-yl)(propyl)amino)ethyl)piperazin-1-yl)methyl)quinolin-8-ol Show/Hide	C28H36N4O2	1
1	Ki = 5.57 nM Bioactivity Info	TI LI LO TS
CP0129619 Compound Info	N-[3-[2-[[(6S)-2-amino-4,5,6,7-tetrahydro-1,3-benzothiazol-6-yl]-propylamino]ethyl]-3-hydroxycyclobutyl]naphthalene-2-carboxamide Show/Hide	C27H34N4O2S	1
1	Ki = 5.6 nM Bioactivity Info	TI LI LO TS
CP0913682 Compound Info	7-(3-(4-(2-Methoxyphenyl)piperazin-1-yl)propoxy)quinolin-2(1H)-one oxalate Show/Hide	C25H29N3O7	1
1	Ki = 5.7 nM Bioactivity Info	TI LI LO TS
CP0852589 Compound Info	(rac)-4-(4-(1H-Indol-5-yl)-1H-1,2,3-triazol-1-yl)-1-(4-(2,3-dichlorophenyl)piperazin-1-yl)butan-2-ol Show/Hide	C24H26Cl2N6O	1
1	Ki = 5.85 nM Bioactivity Info	TI LI LO TS
CP0452963 Compound Info	1-(2-methoxyphenyl)-4-[4-[4-(4-phenylphenyl)triazol-1-yl]butyl]piperazine Show/Hide	C29H33N5O	1
1	Ki = 5.88 nM Bioactivity Info	TI LI LO TS
CP0382695 Compound Info	N-[4-[(2S,5S)-2-(6-aminopyridin-3-yl)-5-methylmorpholin-4-yl]butyl]-1H-indole-2-carboxamide Show/Hide	C23H29N5O2	2
1	Ki = 5.96 nM Bioactivity Info	TI LI LO TS
2	Ki = 182 nM Bioactivity Info	TI LI LO TS
CP0260081 Compound Info	N-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]-3-fluorobutyl]naphthalene-2-carboxamide Show/Hide	C25H26Cl2FN3O	1
1	Ki = 6.1 nM Bioactivity Info	TI LI LO TS
CP0847579 Compound Info	4-(2-Fluoroethoxy)-N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)-transbutyl-2-enyl)benzamide oxalic acid salt Show/Hide	C26H32FN3O7	1
1	Ki = 6.2 nM Bioactivity Info	TI LI LO TS
CP0890281 Compound Info	4-(2-(2-Fluoroethoxy)ethoxy)-N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)benzamide oxalic acid salt Show/Hide	C28H38FN3O8	1
1	Ki = 6.2 nM Bioactivity Info	TI LI LO TS
CP0190972 Compound Info	N-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]-3-fluorobutyl]-4-pyridin-2-ylbenzamide Show/Hide	C26H27Cl2FN4O	1
1	Ki = 6.2 nM Bioactivity Info	TI LI LO TS
CP0496628 Compound Info	1-(2,3-dichlorophenyl)-4-propylpiperazine Show/Hide	C13H18Cl2N2	1
1	Ki = 6.3 nM Bioactivity Info	TI LI LO TS
CP0093141 Compound Info	1-(2-methoxyphenyl)-4-[5-[1-(4-thiophen-3-ylphenyl)triazol-4-yl]pentyl]piperazine Show/Hide	C28H33N5OS	1
1	Ki = 6.3 nM Bioactivity Info	TI LI LO TS
CP0666613 Compound Info	endo-8-(1H-Indol-3-ylmethyl)-3-(3,4-dichlorophenyl)-8-azabicyclo[3.2.1]octan-3-ol Show/Hide	C22H22Cl2N2O	1
1	Ki = 6.35 nM Bioactivity Info	TI LI LO TS
CP0049047 Compound Info	(+)butaclamol Show/Hide	C25H31NO	1
1	Ki = 6.39 nM Bioactivity Info	TI LI LO TS
CP0513106 Compound Info	N-[4-[4-[3-cyano-5-(trifluoromethyl)phenyl]piperazin-1-yl]butyl]imidazo[1,2-a]pyridine-2-carboxamide Show/Hide	C24H25F3N6O	1
1	Ki = 6.4 nM Bioactivity Info	TI LI LO TS
CP0397122 Compound Info	1-[4-[1-(4-fluorophenyl)triazol-4-yl]butyl]-4-(2-methoxyphenyl)piperazine Show/Hide	C23H28FN5O	1
1	Ki = 6.5 nM Bioactivity Info	TI LI LO TS
CP0001212 Compound Info	1-(2-methoxyphenyl)-4-[3-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]propyl]piperazine Show/Hide	C23H29N5OS	1
1	Ki = 6.5 nM Bioactivity Info	TI LI LO TS
CP0474295 Compound Info	4-[4-[5-[4-(2-methoxyphenyl)piperazin-1-yl]pentyl]triazol-1-yl]-N,N-dimethylaniline Show/Hide	C26H36N6O	1
1	Ki = 6.7 nM Bioactivity Info	TI LI LO TS
CP0433591 Compound Info	6-[1-[4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]triazol-4-yl]quinoline Show/Hide	C26H30N6O	1
1	Ki = 6.73 nM Bioactivity Info	TI LI LO TS
CP0410554 Compound Info	2-[4-[3-[4-(2-methoxyphenyl)piperazin-1-yl]propyl]triazol-1-yl]phenol Show/Hide	C22H27N5O2	1
1	Ki = 6.8 nM Bioactivity Info	TI LI LO TS
CP0157762 Compound Info	N-[4-[4-(3-chloro-5-ethyl-2-methoxyphenyl)piperazin-1-yl]-3-hydroxybutyl]-1H-indole-2-carboxamide Show/Hide	C26H33ClN4O3	2
1	Ki = 6.84 nM Bioactivity Info	TI LI LO TS
2	Ki = 7.61 nM Bioactivity Info	TI LI LO TS
CP0857031 Compound Info	4-(2-Fluoroethyl)-N-(4-(4-(2-(2-fluoroethoxy)phenyl)piperazin-1-yl)-butyl)benzamide oxalic acid salt Show/Hide	C27H35F2N3O6	1
1	Ki = 6.9 nM Bioactivity Info	TI LI LO TS
CP0693927 Compound Info	SID50106425 Show/Hide	C16H26BrNO	1
1	Ki = 6.9 nM Bioactivity Info	TI LI LO TS
CP0410937 Compound Info	N-[(3R)-4-[4-(2,3-dichlorophenyl)piperazin-1-yl]-3-fluorobutyl]-1-benzofuran-2-carboxamide Show/Hide	C23H24Cl2FN3O2	1
1	Ki = 6.9 nM Bioactivity Info	TI LI LO TS
CP0871789 Compound Info	7-(5-(4-(2-Methoxyphenyl)piperazin-1-yl)pentyloxy)-3,4-dihydroquinolin-2(1H)-one oxalate Show/Hide	C27H35N3O7	1
1	Ki = 7 nM Bioactivity Info	TI LI LO TS
CP0397770 Compound Info	N-[4-[4-(2-methoxyphenyl)-1,4-diazepan-1-yl]butyl]-4-(methylamino)benzamide Show/Hide	C24H34N4O2	1
1	Ki = 7.2 nM Bioactivity Info	TI LI LO TS
CP0045034 Compound Info	N-[4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]pyrazolo[1,5-a]pyridine-2-carboxamide Show/Hide	C23H29N5O2	8
1	Ki = 7.4 nM Bioactivity Info	TI LI LO TS
2	Ki = 7.6 nM Bioactivity Info	TI LI LO TS
3	Ki = 93 nM Bioactivity Info	TI LI LO TS
4	Ki = 97 nM Bioactivity Info	TI LI LO TS
5	Ki = 130 nM Bioactivity Info	TI LI LO TS
6	Ki = 290 nM Bioactivity Info	TI LI LO TS
7	Ki = 340 nM Bioactivity Info	TI LI LO TS
8	Ki = 500 nM Bioactivity Info	TI LI LO TS
CP0891096 Compound Info	7-(3-(4-(2-Methoxyphenyl)piperazin-1-yl)propoxy)-3,4-dihydroquinolin-2(1H)-one oxalate Show/Hide	C25H31N3O7	1
1	Ki = 7.4 nM Bioactivity Info	TI LI LO TS
CP0239897 Compound Info	N-[(3R)-4-[4-(3-chloro-5-ethyl-2-methoxyphenyl)piperazin-1-yl]-3-hydroxybutyl]-1H-indole-2-carboxamide Show/Hide	C26H33ClN4O3	1
1	Ki = 7.4 nM Bioactivity Info	TI LI LO TS
CP0477829 Compound Info	N-[4-[4-(2-methoxyphenyl)-1,4-diazepan-1-yl]butyl]-5-methylthiophene-2-carboxamide Show/Hide	C22H31N3O2S	1
1	Ki = 7.5 nM Bioactivity Info	TI LI LO TS
CP0381017 Compound Info	(+)-R-11-(3-(4-((4-(2-Methoxyphenyl)piperazin-1-yl)ethyl)-1H-1,2,3-triazol-1-yl)propoxy)-N-propylnoraporphine Show/Hide	C37H46N6O2	1
1	Ki = 7.7 nM Bioactivity Info	TI LI LO TS
CP0547198 Compound Info	1-(2,3-dichlorophenyl)-4-[4-(4-naphthalen-2-yltriazol-1-yl)butyl]piperazine Show/Hide	C26H27Cl2N5	1
1	Ki = 7.7 nM Bioactivity Info	TI LI LO TS
CP0475836 Compound Info	(-)-S-11-((1-(3-(4-(2-Methoxyphenyl)piperazin-1-yl)butyl)-1H-1,2,3-triazol-4-yl)methoxy)-N-propylnoraporphine Show/Hide	C37H46N6O2	1
1	Ki = 8 nM Bioactivity Info	TI LI LO TS
CP0273713 Compound Info	N-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]-3-fluorobutyl]-5-methoxy-1-benzofuran-2-carboxamide Show/Hide	C24H26Cl2FN3O3	1
1	Ki = 8 nM Bioactivity Info	TI LI LO TS
CP0052483 Compound Info	4-Bromo-1-methoxy-naphthalene-2-carboxylic acid {2-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-ethyl}-amide Show/Hide	C24H24BrCl2N3O2	1
1	Ki = 8 nM Bioactivity Info	TI LI LO TS
CP0407660 Compound Info	5-(4-fluorophenyl)-N-[4-[4-(2-methoxyphenyl)-1,4-diazepan-1-yl]butyl]thiophene-2-carboxamide Show/Hide	C27H32FN3O2S	1
1	Ki = 8 nM Bioactivity Info	TI LI LO TS
CP0378578 Compound Info	N-[4-[4-[2-tert-butyl-6-(trifluoromethyl)pyrimidin-4-yl]piperazin-1-yl]butyl]imidazo[1,2-a]pyrazine-2-carboxamide Show/Hide	C24H31F3N8O	1
1	Ki = 8 nM Bioactivity Info	TI LI LO TS
CP0489688 Compound Info	N-[4-(4-phenylpiperazin-1-yl)butyl]-4-thiophen-3-ylbenzamide Show/Hide	C25H29N3OS	1
1	Ki = 8 nM Bioactivity Info	TI LI LO TS
CP0542701 Compound Info	N-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]-3-hydroxybutyl]-6-fluoroquinoline-3-carboxamide Show/Hide	C24H25Cl2FN4O2	1
1	Ki = 8.05 nM Bioactivity Info	TI LI LO TS
CP0395781 Compound Info	(+/-)-11-(3-(4-((4-(2-Methoxyphenyl)piperazin-1-yl)butyl)-1H-1,2,3-triazol-1-yl)propoxy)-N-propylnoraporphine Show/Hide	C39H50N6O2	1
1	Ki = 8.14 nM Bioactivity Info	TI LI LO TS
CP0471346 Compound Info	(+/-)-11-(3-(4-((4-(2-Methoxyphenyl)piperazin-1-yl)propyl)-1H-1,2,3-triazol-1-yl)propoxy)-N-propylnoraporphine Show/Hide	C38H48N6O2	1
1	Ki = 8.16 nM Bioactivity Info	TI LI LO TS
CP0093139 Compound Info	1-(2-methoxyphenyl)-4-[4-[1-(4-thiophen-3-ylphenyl)triazol-4-yl]butyl]piperazine Show/Hide	C27H31N5OS	1
1	Ki = 8.2 nM Bioactivity Info	TI LI LO TS
CP0438434 Compound Info	N-[4-[4-(3-chlorophenyl)piperazin-1-yl]butyl]-4-thiophen-3-ylbenzamide Show/Hide	C25H28ClN3OS	1
1	Ki = 8.3 nM Bioactivity Info	TI LI LO TS
CP0864137 Compound Info	1-(4-(4-([1,10-Biphenyl]-4-yl)-1H-1,2,3-triazol-1-yl)-butyl)-4-(2,3-dichlorophenyl)piperazine Show/Hide	C28H29Cl2N5	1
1	Ki = 8.32 nM Bioactivity Info	TI LI LO TS
CP0847346 Compound Info	endo-8-(Naphtho[2,1-b]fur-1-ylmethyl)-3-(4-chlorophenyl)-8-azabicyclo[3.2.1]octan-3-ol Show/Hide	C26H24ClNO2	1
1	Ki = 8.4 nM Bioactivity Info	TI LI LO TS
CP0847308 Compound Info	4-(2-Fluoroethoxy)-N-(4-(4-(2-(2-fluoroethoxy)phenyl)piperazin-1-yl)-trans-butyl-2-enyl)benzamide oxalic acid salt Show/Hide	C27H33F2N3O7	1
1	Ki = 8.4 nM Bioactivity Info	TI LI LO TS
CP0869496 Compound Info	(E)-5-(2-(2-(2-fluoroethoxy)ethoxy)ethoxy)-N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)but-2-en-1-yl)-1H-indole-2-carboxamide oxalic acid Show/Hide	C32H41FN4O9	1
1	Ki = 8.4 nM Bioactivity Info	TI LI LO TS
CP0425930 Compound Info	N-[4-[4-(2-tert-butyl-6-cyclopropylpyrimidin-4-yl)piperazin-1-yl]butyl]imidazo[1,2-a]pyridine-2-carboxamide Show/Hide	C27H37N7O	1
1	Ki = 8.4 nM Bioactivity Info	TI LI LO TS
CP0440174 Compound Info	4-fluoro-N-[4-[4-(2-methoxyphenyl)-1,4-diazepan-1-yl]butyl]benzamide Show/Hide	C23H30FN3O2	1
1	Ki = 8.8 nM Bioactivity Info	TI LI LO TS
CP0367294 Compound Info	1-(2-methoxyphenyl)-4-[3-[1-(4-thiophen-3-ylphenyl)triazol-4-yl]propyl]piperazine Show/Hide	C26H29N5OS	1
1	Ki = 8.9 nM Bioactivity Info	TI LI LO TS
CP0375440 Compound Info	4-(2-fluoroethyl)-N-[4-[4-(2-methoxyphenyl)-1,4-diazepan-1-yl]butyl]benzamide Show/Hide	C25H34FN3O2	1
1	Ki = 9 nM Bioactivity Info	TI LI LO TS
CP0380992 Compound Info	N-[4-[4-(2-methoxyphenyl)-1,4-diazepan-1-yl]butyl]-5-phenylthiophene-2-carboxamide Show/Hide	C27H33N3O2S	1
1	Ki = 9 nM Bioactivity Info	TI LI LO TS
CP0400253 Compound Info	N-[4-[4-[2-tert-butyl-6-(trifluoromethyl)pyrimidin-4-yl]piperazin-1-yl]butyl]-3-[(dimethylamino)methyl]imidazo[1,2-a]pyridine-2-carboxamide Show/Hide	C28H39F3N8O	5
1	Ki = 9.1 nM Bioactivity Info	TI LI LO TS
2	Ki = 16 nM Bioactivity Info	TI LI LO TS
3	Ki = 19 nM Bioactivity Info	TI LI LO TS
4	Ki = 27 nM Bioactivity Info	TI LI LO TS
5	Ki = 29 nM Bioactivity Info	TI LI LO TS
CP0500980 Compound Info	(+)-R-11-((1-(3-(4-(2-Methoxyphenyl)piperazin-1-yl)butyl)-1H-1,2,3-triazol-4-yl)methoxy)-N-propylnoraporphine Show/Hide	C37H46N6O2	1
1	Ki = 9.18 nM Bioactivity Info	TI LI LO TS
CP0860998 Compound Info	8-(Benzofuran-3-ylmethyl)-3-(2-fluoroethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one oxalate Show/Hide	C26H28FN3O6	1
1	Ki = 9.3 nM Bioactivity Info	TI LI LO TS
CP0386820 Compound Info	N-[4-[4-(2-tert-butyl-6-methylpyrimidin-4-yl)piperazin-1-yl]butyl]imidazo[1,2-a]pyridine-2-carboxamide Show/Hide	C25H35N7O	1
1	Ki = 9.3 nM Bioactivity Info	TI LI LO TS
CP0386829 Compound Info	N-[4-[4-[2-tert-butyl-6-(trifluoromethyl)pyrimidin-4-yl]piperazin-1-yl]butyl]-4-phenylcyclohexane-1-carboxamide Show/Hide	C30H42F3N5O	1
1	Ki = 9.4 nM Bioactivity Info	TI LI LO TS
CP0190971 Compound Info	N-[3-fluoro-4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]-1H-indole-2-carboxamide Show/Hide	C24H29FN4O2	1
1	Ki = 9.5 nM Bioactivity Info	TI LI LO TS
CP0400278 Compound Info	1-(2-methoxyphenyl)-4-[3-[1-(4-methylsulfanylphenyl)triazol-4-yl]propyl]piperazine Show/Hide	C23H29N5OS	1
1	Ki = 9.6 nM Bioactivity Info	TI LI LO TS
CP0520091 Compound Info	N-[[(1R,2S)-2-[2-(7-cyano-3,4-dihydro-1H-isoquinolin-2-yl)ethyl]cyclopropyl]methyl]-1H-indole-2-carboxamide Show/Hide	C25H26N4O	1
1	Ki = 9.81 nM Bioactivity Info	TI LI LO TS
CP0042751 Compound Info	(6aR)-6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline-10,11-diol;hydrate;hydrochloride Show/Hide	C17H17NO2	2
1	Ki = 10 nM Bioactivity Info	TI LI LO TS
2	Ki = 17 nM Bioactivity Info	TI LI LO TS
CP0386828 Compound Info	N-[4-[4-[2-tert-butyl-6-(trifluoromethyl)pyrimidin-4-yl]piperazin-1-yl]butyl]-6-chloroimidazo[1,2-b]pyridazine-2-carboxamide Show/Hide	C24H30ClF3N8O	1
1	Ki = 10 nM Bioactivity Info	TI LI LO TS
CP0553536 Compound Info	N-[4-(4-phenylpiperazin-1-yl)butyl]imidazo[1,2-a]pyridine-2-carboxamide Show/Hide	C22H27N5O	1
1	Ki = 10 nM Bioactivity Info	TI LI LO TS
CP0294037 Compound Info	N-[3-fluoro-4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]-9H-fluorene-2-carboxamide Show/Hide	C29H32FN3O2	1
1	Ki = 10.1 nM Bioactivity Info	TI LI LO TS
CP0501917 Compound Info	7-[(3-(4-phenylpiperazin-1-yl)propyl)(propyl)amino]-5,6,7,8-tetrahydronaphthalen-2-ol Show/Hide	C26H37N3O	1
1	Ki = 10.3 nM Bioactivity Info	TI LI LO TS
CP0398936 Compound Info	(10R)-3-butyl-10-(methylamino)-1,3-diazatricyclo[6.3.1.04,12]dodeca-4,6,8(12)-trien-2-one Show/Hide	C15H21N3O	2
1	Ki = 10.3 nM Bioactivity Info	TI LI LO TS
2	Ki = 142 nM Bioactivity Info	TI LI LO TS
CP0417214 Compound Info	8-[(2-(4-phenylpiperazin-1-yl)ethyl)(propyl)amino]-6,7,8,9-tetrahydro-1H-benzo[e]indol-2(3H)-one Show/Hide	C27H36N4O	1
1	Ki = 10.9 nM Bioactivity Info	TI LI LO TS
CP0912199 Compound Info	1-(Benzofuran-3-ylmethyl)-4-(4-bromophenyl)piperidin-4-ol oxalate Show/Hide	C22H22BrNO6	1
1	Ki = 10.9 nM Bioactivity Info	TI LI LO TS
CP0903618 Compound Info	2-(2-Fluoroethoxy)-5-iodo-N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)-trans-butyl-2-enyl)benzamide oxalic acid salt Show/Hide	C26H31FIN3O7	1
1	Ki = 10.9 nM Bioactivity Info	TI LI LO TS
CP0386826 Compound Info	N-[4-[4-[2-tert-butyl-6-(trifluoromethyl)pyrimidin-4-yl]piperazin-1-yl]butyl]-1H-indole-2-carboxamide Show/Hide	C26H33F3N6O	1
1	Ki = 11 nM Bioactivity Info	TI LI LO TS
CP0200768 Compound Info	N-[4-[2-(6-cyano-3,4-dihydro-1H-isoquinolin-2-yl)ethyl]cyclohexyl]quinoline-4-carboxamide Show/Hide	C28H30N4O	1
1	Ki = 11 nM Bioactivity Info	TI LI LO TS
CP0449146 Compound Info	1-(2-methoxyphenyl)-4-[4-(4-naphthalen-2-yltriazol-1-yl)butyl]piperazine Show/Hide	C27H31N5O	1
1	Ki = 11.1 nM Bioactivity Info	TI LI LO TS
CP0378422 Compound Info	6-[(2-(4-phenylpiperazin-1-yl)ethyl)(propyl)amino]-5,6,7,8-tetrahydronaphthalen-2-ol Show/Hide	C25H35N3O	1
1	Ki = 11.2 nM Bioactivity Info	TI LI LO TS
CP0860992 Compound Info	1-(Benzofuran-3-ylmethyl)-4-(4-iodophenyl)piperidin-4-ol oxalate Show/Hide	C22H22INO6	1
1	Ki = 11.2 nM Bioactivity Info	TI LI LO TS
CP0480200 Compound Info	N-[4-[4-(2-chloro-3-ethylphenyl)piperazin-1-yl]-3-hydroxybutyl]-5-methyl-1H-imidazole-2-carboxamide Show/Hide	C21H30ClN5O2	1
1	Ki = 11.2 nM Bioactivity Info	TI LI LO TS
CP0397771 Compound Info	N-[4-[4-(2-methoxyphenyl)-1,4-diazepan-1-yl]butyl]-9-oxofluorene-4-carboxamide Show/Hide	C30H33N3O3	1
1	Ki = 11.6 nM Bioactivity Info	TI LI LO TS
CP0386822 Compound Info	N-[4-[4-[2-tert-butyl-6-(trifluoromethyl)pyrimidin-4-yl]piperazin-1-yl]butyl]imidazo[1,2-a]pyrimidine-2-carboxamide Show/Hide	C24H31F3N8O	1
1	Ki = 12 nM Bioactivity Info	TI LI LO TS
CP0379464 Compound Info	N-[4-[4-[2-tert-butyl-6-(trifluoromethyl)pyrimidin-4-yl]piperazin-1-yl]butyl]-5-[(dimethylamino)methyl]imidazo[1,2-a]pyridine-2-carboxamide Show/Hide	C28H39F3N8O	5
1	Ki = 12 nM Bioactivity Info	TI LI LO TS
2	Ki = 16 nM Bioactivity Info	TI LI LO TS
3	Ki = 24 nM Bioactivity Info	TI LI LO TS
4	Ki = 27 nM Bioactivity Info	TI LI LO TS
5	Ki = 44 nM Bioactivity Info	TI LI LO TS
CP0003459 Compound Info	3-(2-methoxyphenyl)-9-[3-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]propyl]-3,9-diazaspiro[5.5]undecane Show/Hide	C28H37N5OS	1
1	Ki = 12 nM Bioactivity Info	TI LI LO TS
CP0455926 Compound Info	N-[4-[methyl-[(10R)-2-oxo-1,3-diazatricyclo[6.3.1.04,12]dodeca-4,6,8(12)-trien-10-yl]amino]butyl]-9H-fluorene-2-carboxamide Show/Hide	C29H30N4O2	2
1	Ki = 12.5 nM Bioactivity Info	TI LI LO TS
2	Ki = 1090 nM Bioactivity Info	TI LI LO TS
CP0468878 Compound Info	N-[(3R)-4-[4-(3-chloro-5-ethyl-2-methoxyphenyl)piperazin-1-yl]-3-fluorobutyl]-1H-indole-2-carboxamide Show/Hide	C26H32ClFN4O2	1
1	Ki = 13 nM Bioactivity Info	TI LI LO TS
CP0847130 Compound Info	7-(4-(4-(2-Methoxyphenyl)piperazin-1-yl)butoxy)-3,4-dihydroquinolin-2(1H)-one oxalate Show/Hide	C26H33N3O7	1
1	Ki = 13.1 nM Bioactivity Info	TI LI LO TS
CP0410750 Compound Info	6-[4-[4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]triazol-1-yl]isoquinoline Show/Hide	C26H30N6O	1
1	Ki = 13.1 nM Bioactivity Info	TI LI LO TS
CP0414228 Compound Info	N-[(6,6-diphenyl-1,4-dioxan-2-yl)methyl]-2-(2-methoxyphenoxy)ethanamine Show/Hide	C26H29NO4	1
1	Ki = 13.18 nM Bioactivity Info	TI LI LO TS
CP0375439 Compound Info	4-(2-hydroxyethyl)-N-[4-[4-(2-methoxyphenyl)-1,4-diazepan-1-yl]butyl]benzamide Show/Hide	C25H35N3O3	1
1	Ki = 13.2 nM Bioactivity Info	TI LI LO TS
CP0036333 Compound Info	(S)-3,5-Dichloro-N-(1-ethyl-pyrrolidin-2-ylmethyl)-2-hydroxy-6-methoxy-benzamide Show/Hide	C15H20Cl2N2O3	1
1	Ki = 13.4 nM Bioactivity Info	TI LI LO TS
CP0847131 Compound Info	7-(4-(4-(2-(2-Fluoroethoxy)phenyl)piperazin-1-yl)butoxy)-3,4-dihydroquinolin-2(1H)-one oxalate Show/Hide	C27H34FN3O7	1
1	Ki = 13.5 nM Bioactivity Info	TI LI LO TS
CP0847306 Compound Info	5-Bromo-2-(2-fluoroethoxy)-N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)-trans-butyl-2-enyl)benzamide oxalic acid salt Show/Hide	C26H31BrFN3O7	1
1	Ki = 13.6 nM Bioactivity Info	TI LI LO TS
CP0489689 Compound Info	N-[4-[4-(4-hydroxyphenyl)piperazin-1-yl]butyl]-4-thiophen-3-ylbenzamide Show/Hide	C25H29N3O2S	1
1	Ki = 13.6 nM Bioactivity Info	TI LI LO TS
CP0224532 Compound Info	1-(2-chloro-3-ethylphenyl)-4-methylpiperazine Show/Hide	C13H19ClN2	1
1	Ki = 13.6 nM Bioactivity Info	TI LI LO TS
CP0847769 Compound Info	5-Bromo-2-(2-fluoroethoxy)-3-methoxy-N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)-trans-butyl-2-enyl)benzamide oxalic acid salt Show/Hide	C27H33BrFN3O8	1
1	Ki = 13.8 nM Bioactivity Info	TI LI LO TS
CP0207473 Compound Info	N-[3-fluoro-4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]-5-methoxy-1-benzofuran-2-carboxamide Show/Hide	C25H30FN3O4	1
1	Ki = 13.9 nM Bioactivity Info	TI LI LO TS
CP0234731 Compound Info	4-[4-[4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]triazol-1-yl]-N,N-dimethylaniline Show/Hide	C25H34N6O	1
1	Ki = 13.9 nM Bioactivity Info	TI LI LO TS
CP0389182 Compound Info	1-(2,3-dichlorophenyl)-4-[4-[4-(9H-fluoren-2-yl)triazol-1-yl]butyl]piperazine Show/Hide	C29H29Cl2N5	1
1	Ki = 14 nM Bioactivity Info	TI LI LO TS
CP0377326 Compound Info	7-{[2-(4-Phenyl-piperazin-1-yl)-ethyl]-prop-2-ynyl-amino}-5,6,7,8-tetrahydro-naphthalen-2-ol Show/Hide	C25H31N3O	1
1	Ki = 14.2 nM Bioactivity Info	TI LI LO TS
CP0435435 Compound Info	1-butyl-4-[2-(2-fluoroethoxy)phenyl]piperazine Show/Hide	C16H25FN2O	2
1	Ki = 14.7 nM Bioactivity Info	TI LI LO TS
2	Ki = 22.3 nM Bioactivity Info	TI LI LO TS
CP0392993 Compound Info	1-(1-Benzyl-piperidin-4-yl)-5-methyl-3,4-diphenyl-1,3-dihydro-imidazol-2-one Show/Hide	C28H29N3O	1
1	Ki = 15 nM Bioactivity Info	TI LI LO TS
CP0381618 Compound Info	6-chloro-N-[4-[4-(2-methoxyphenyl)-1,4-diazepan-1-yl]butyl]pyridine-3-carboxamide Show/Hide	C22H29ClN4O2	1
1	Ki = 15 nM Bioactivity Info	TI LI LO TS
CP0772878 Compound Info	endo-8-(1H-Indol-3-ylmethyl)-3-(4-chlorophenyl)-8-azabicyclo-[3.2.1]octan-3-ol Show/Hide	C22H23ClN2O	1
1	Ki = 15.5 nM Bioactivity Info	TI LI LO TS
CP0100739 Compound Info	N-[3-[4-(2-methoxyphenyl)piperazin-1-yl]propyl]pyrazolo[1,5-a]pyridine-3-carboxamide Show/Hide	C22H27N5O2	8
1	Ki = 16 nM Bioactivity Info	TI LI LO TS
2	Ki = 34 nM Bioactivity Info	TI LI LO TS
3	Ki = 69 nM Bioactivity Info	TI LI LO TS
4	Ki = 320 nM Bioactivity Info	TI LI LO TS
5	Ki = 390 nM Bioactivity Info	TI LI LO TS
6	Ki = 630 nM Bioactivity Info	TI LI LO TS
7	Ki = 640 nM Bioactivity Info	TI LI LO TS
8	Ki = 1030 nM Bioactivity Info	TI LI LO TS
CP0476734 Compound Info	N-[4-[4-(2-hydroxyphenyl)piperazin-1-yl]butyl]-4-thiophen-3-ylbenzamide Show/Hide	C25H29N3O2S	1
1	Ki = 16.7 nM Bioactivity Info	TI LI LO TS
CP0848870 Compound Info	1-(Hydroxymethyl)-apomorphine Hydrochloride Show/Hide	C18H20ClNO3	1
1	Ki = 17 nM Bioactivity Info	TI LI LO TS
CP0879779 Compound Info	endo-8-(Benzothien-3-ylmethyl)-3-(3,4-dichlorophenyl)-8-azabicyclo[3.2.1]octan-3-ol Show/Hide	C22H21Cl2NOS	1
1	Ki = 17.9 nM Bioactivity Info	TI LI LO TS
CP0465278 Compound Info	6-bromo-N-[4-[4-(2-methoxyphenyl)-1,4-diazepan-1-yl]butyl]pyridine-3-carboxamide Show/Hide	C22H29BrN4O2	1
1	Ki = 17.9 nM Bioactivity Info	TI LI LO TS
CP0410752 Compound Info	1-[4-(2,3-dichlorophenyl)piperazin-1-yl]-4-(4-quinolin-6-yltriazol-1-yl)butan-2-ol Show/Hide	C25H26Cl2N6O	1
1	Ki = 18 nM Bioactivity Info	TI LI LO TS
CP0519605 Compound Info	N-[4-[4-(3-methoxyphenyl)piperazin-1-yl]butyl]-4-thiophen-3-ylbenzamide Show/Hide	C26H31N3O2S	1
1	Ki = 18 nM Bioactivity Info	TI LI LO TS
CP0905141 Compound Info	4-(2-(2-Fluoroethoxy)ethoxy)-N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)-trans-butyl-2-enyl)benzamide oxalic acid salt Show/Hide	C28H36FN3O8	1
1	Ki = 18.2 nM Bioactivity Info	TI LI LO TS
CP0857036 Compound Info	2-(2-Fluoroethoxy)-5-methyl-N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)-trans-butyl-2-enyl)benzamide oxalic acid salt Show/Hide	C27H34FN3O7	1
1	Ki = 18.5 nM Bioactivity Info	TI LI LO TS
CP0410751 Compound Info	4-[4-(9H-fluoren-2-yl)triazol-1-yl]-1-[4-(2-methoxyphenyl)piperazin-1-yl]butan-2-ol Show/Hide	C30H33N5O2	1
1	Ki = 18.5 nM Bioactivity Info	TI LI LO TS
CP0410601 Compound Info	N-[4-[4-(2,6-ditert-butylpyrimidin-4-yl)piperazin-1-yl]butyl]imidazo[1,2-a]pyridine-2-carboxamide Show/Hide	C28H41N7O	1
1	Ki = 19 nM Bioactivity Info	TI LI LO TS
CP0869680 Compound Info	2-(4-(4-(2,3-difluorophenyl)piperazin-1-yl)butyl)isoindoline-1,3-dione Show/Hide	C22H23F2N3O2	1
1	Ki = 19.3 nM Bioactivity Info	TI LI LO TS
CP0856728 Compound Info	4-(2-(2-Fluoroethoxy)ethoxy)-N-(4-(4-(2-(2-fluoroethoxy)phenyl)piperazin-1-yl)-trans-but-2-enyl)benzamide oxalic acid salt Show/Hide	C29H37F2N3O8	1
1	Ki = 19.6 nM Bioactivity Info	TI LI LO TS
CP0098320 Compound Info	2-(2-methoxyphenyl)-8-[3-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]propyl]-2,8-diazaspiro[4.5]decane Show/Hide	C27H35N5OS	1
1	Ki = 19.6 nM Bioactivity Info	TI LI LO TS
CP0521214 Compound Info	N-[4-[4-(4-methoxyphenyl)piperazin-1-yl]butyl]-4-thiophen-3-ylbenzamide Show/Hide	C26H31N3O2S	1
1	Ki = 19.8 nM Bioactivity Info	TI LI LO TS
CP0377980 Compound Info	(+/-)-11-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butoxy)-N-propylnoraporphine Show/Hide	C34H43N3O2	1
1	Ki = 19.9 nM Bioactivity Info	TI LI LO TS
CP0386824 Compound Info	N-[4-(4-quinolin-4-ylpiperazin-1-yl)butyl]imidazo[1,2-a]pyridine-2-carboxamide Show/Hide	C25H28N6O	1
1	Ki = 20 nM Bioactivity Info	TI LI LO TS
CP0207472 Compound Info	N-[3-fluoro-4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]-4-pyridin-2-ylbenzamide Show/Hide	C27H31FN4O2	1
1	Ki = 20.5 nM Bioactivity Info	TI LI LO TS
CP0395780 Compound Info	(+/-)-11-((1-(3-(4-(2-Methoxyphenyl)piperazin-1-yl)propyl)-1H-1,2,3-triazol-4-yl)methoxy)-N-propylnoraporphine Show/Hide	C36H44N6O2	1
1	Ki = 21 nM Bioactivity Info	TI LI LO TS
CP0416962 Compound Info	3-(4-fluoro-2-methoxyphenyl)-9-[3-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]propyl]-3,9-diazaspiro[5.5]undecane Show/Hide	C28H36FN5OS	1
1	Ki = 21 nM Bioactivity Info	TI LI LO TS
CP0490608 Compound Info	1-(2-methoxyphenyl)-4-[5-[1-(2-methoxyphenyl)triazol-4-yl]pentyl]piperazine Show/Hide	C25H33N5O2	1
1	Ki = 21.1 nM Bioactivity Info	TI LI LO TS
CP0880729 Compound Info	endo-8-(5-Methoxy-1H-indol-3-ylmethyl)-3-(4-chlorophenyl)-8-azabicyclo[3.2.1]octan-3-ol Show/Hide	C23H25ClN2O2	1
1	Ki = 21.2 nM Bioactivity Info	TI LI LO TS
CP0871615 Compound Info	N-((1S,4r)-4-(2-((2S,5S)-2-(6-aminopyridin-3-yl)-5-methylmorpholino)ethyl)cyclohexyl)-1H-indole-2-carboxamide Show/Hide	C27H35N5O2	1
1	Ki = 21.6 nM Bioactivity Info	TI LI LO TS
CP0401191 Compound Info	(10R)-3-propyl-10-(propylamino)-1,3-diazatricyclo[6.3.1.04,12]dodeca-4,6,8(12)-trien-2-one Show/Hide	C16H23N3O	2
1	Ki = 21.7 nM Bioactivity Info	TI LI LO TS
2	Ki = 47.9 nM Bioactivity Info	TI LI LO TS
CP0435437 Compound Info	N-[4-[4-(3-methylphenyl)piperazin-1-yl]butyl]-4-thiophen-3-ylbenzamide Show/Hide	C26H31N3OS	1
1	Ki = 21.9 nM Bioactivity Info	TI LI LO TS
CP0341205 Compound Info	N-[3-[2-[[(1S,2R)-2-(2-chlorophenyl)cyclopropyl]-propylamino]ethyl]-3-hydroxycyclobutyl]naphthalene-2-carboxamide Show/Hide	C29H33ClN2O2	1
1	Ki = 22.1 nM Bioactivity Info	TI LI LO TS
CP0434347 Compound Info	2-N-[2-(4-phenylpiperazin-1-yl)ethyl]-2-N-propyl-1,2,3,4-tetrahydronaphthalene-2,7-diamine Show/Hide	C25H36N4	1
1	Ki = 22.2 nM Bioactivity Info	TI LI LO TS
CP0555051 Compound Info	1-(2-methoxyphenyl)-4-[3-(1-phenyltriazol-4-yl)propyl]piperazine Show/Hide	C22H27N5O	1
1	Ki = 22.2 nM Bioactivity Info	TI LI LO TS
CP0135682 Compound Info	1-butyl-4-(3-chloro-5-ethyl-2-methoxyphenyl)piperazine Show/Hide	C17H27ClN2O	1
1	Ki = 22.5 nM Bioactivity Info	TI LI LO TS
CP0266687 Compound Info	1-(2-methoxyphenyl)-4-[4-(4-phenyltriazol-1-yl)butyl]piperazine Show/Hide	C23H29N5O	1
1	Ki = 22.9 nM Bioactivity Info	TI LI LO TS
CP0255950 Compound Info	2-[1-(benzenesulfonyl)indol-3-yl]-N,N-dimethylethanamine Show/Hide	C18H20N2O2S	1
1	Ki = 23 nM Bioactivity Info	TI LI LO TS
CP0860429 Compound Info	1-Methylapomorphine Hydrochloride Show/Hide	C18H20ClNO2	1
1	Ki = 23 nM Bioactivity Info	TI LI LO TS
CP0454412 Compound Info	(+)-R-11-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butoxy)-N-propylnoraporphine Show/Hide	C34H43N3O2	1
1	Ki = 23.4 nM Bioactivity Info	TI LI LO TS
CP0417545 Compound Info	N-[(3S)-4-[4-(2,3-dichlorophenyl)piperazin-1-yl]-3-hydroxybutyl]quinoline-3-carboxamide Show/Hide	C24H26Cl2N4O2	1
1	Ki = 23.4 nM Bioactivity Info	TI LI LO TS
CP0396209 Compound Info	N-[[(1R,2S)-2-[2-(7-cyano-3,4-dihydro-1H-isoquinolin-2-yl)ethyl]cyclopropyl]methyl]-1H-pyrrolo[2,3-b]pyridine-2-carboxamide Show/Hide	C24H25N5O	1
1	Ki = 23.4 nM Bioactivity Info	TI LI LO TS
CP0417011 Compound Info	N-[4-[4-(6-ethyl-1,3-benzodioxol-5-yl)piperazin-1-yl]-3-hydroxybutyl]-1-benzofuran-2-carboxamide Show/Hide	C26H31N3O5	1
1	Ki = 23.6 nM Bioactivity Info	TI LI LO TS
CP0384351 Compound Info	7-[(2-(4-phenylpiperazin-1-yl)ethyl)(2-(thiophen-2-yl)ethyl)amino]-5,6,7,8-tetrahydronaphthalen-2-ol Show/Hide	C28H35N3OS	1
1	Ki = 23.9 nM Bioactivity Info	TI LI LO TS
CP0266478 Compound Info	1-Butyl-4-(2-methoxy-phenyl)-piperazine Show/Hide	C15H24N2O	1
1	Ki = 23.9 nM Bioactivity Info	TI LI LO TS
CP0547879 Compound Info	2-(2-methoxyphenyl)-7-[3-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]propyl]-2,7-diazaspiro[4.4]nonane Show/Hide	C26H33N5OS	1
1	Ki = 24.2 nM Bioactivity Info	TI LI LO TS
CP0556695 Compound Info	N-[4-[4-(3-chloro-5-ethyl-2-methoxyphenyl)piperazin-1-yl]-3-hydroxybutyl]-1,3-benzodioxole-5-carboxamide Show/Hide	C25H32ClN3O5	1
1	Ki = 24.5 nM Bioactivity Info	TI LI LO TS
CP0903635 Compound Info	4-(2-Fluoroethyl)-N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)-transbutyl-2-enyl)benzamide oxalic acid salt Show/Hide	C26H32FN3O6	1
1	Ki = 24.9 nM Bioactivity Info	TI LI LO TS
CP0378576 Compound Info	N-[4-[4-[2-tert-butyl-6-(trifluoromethyl)pyrimidin-4-yl]piperazin-1-yl]butyl]-3-[(dimethylamino)methyl]-1H-indole-2-carboxamide Show/Hide	C29H40F3N7O	1
1	Ki = 25 nM Bioactivity Info	TI LI LO TS
CP0397790 Compound Info	1-[4-(2,3-dichlorophenyl)piperazin-1-yl]-4-(4-naphthalen-2-yltriazol-1-yl)butan-2-ol Show/Hide	C26H27Cl2N5O	1
1	Ki = 25.2 nM Bioactivity Info	TI LI LO TS
CP0375299 Compound Info	1-(2-methoxyphenyl)-4-[4-[1-(2-methoxyphenyl)triazol-4-yl]butyl]piperazine Show/Hide	C24H31N5O2	1
1	Ki = 25.4 nM Bioactivity Info	TI LI LO TS
CP0483103 Compound Info	2-[4-[5-[3-[3-(2-methoxyphenyl)-3,9-diazaspiro[5.5]undecan-9-yl]propylsulfanyl]-4-methyl-1,2,4-triazol-3-yl]phenyl]-1,3-oxazole Show/Hide	C31H38N6O2S	1
1	Ki = 25.4 nM Bioactivity Info	TI LI LO TS
CP0084819 Compound Info	(R)-5-Propylamino-5,6-dihydro-1H,4H-imidazo[4,5,1-ij]quinolin-2-one Show/Hide	C13H17N3O	2
1	Ki = 25.5 nM Bioactivity Info	TI LI LO TS
2	Ki = 410 nM Bioactivity Info	TI LI LO TS
CP0162156 Compound Info	3-(4-fluorophenyl)-9-[3-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]propyl]-3,9-diazaspiro[5.5]undecane Show/Hide	C27H34FN5S	1
1	Ki = 25.6 nM Bioactivity Info	TI LI LO TS
CP0411136 Compound Info	9-[3-[[5-(2-fluorophenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanyl]propyl]-3-(2-methoxyphenyl)-3,9-diazaspiro[5.5]undecane Show/Hide	C28H36FN5OS	1
1	Ki = 25.9 nM Bioactivity Info	TI LI LO TS
CP0375407 Compound Info	1-[3-[1-(4-fluorophenyl)triazol-4-yl]propyl]-4-(2-methoxyphenyl)piperazine Show/Hide	C22H26FN5O	1
1	Ki = 26.5 nM Bioactivity Info	TI LI LO TS
CP0409653 Compound Info	(R)-5-Dipropylamino-5,6-dihydro-1H,4H-imidazo[4,5,1-ij]quinolin-2-one Show/Hide	C16H23N3O	1
1	Ki = 27.1 nM Bioactivity Info	TI LI LO TS
CP0489687 Compound Info	4-(Thiophen-3-yl)-N-(4-(4-(2-(2-fluoroethoxy)phenyl)piperazin-1-yl)butyl)benzamide oxalic acid salt Show/Hide	C27H32FN3O2S	1
1	Ki = 27.7 nM Bioactivity Info	TI LI LO TS
CP0416958 Compound Info	8-(2-methoxyphenyl)-2-[3-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]propyl]-2,8-diazaspiro[4.5]decane Show/Hide	C27H35N5OS	1
1	Ki = 27.8 nM Bioactivity Info	TI LI LO TS
CP0063606 Compound Info	N-[4-[4-(3-chloro-5-ethyl-2-methoxyphenyl)piperazin-1-yl]-3-fluorobutyl]-1H-indole-2-carboxamide Show/Hide	C26H32ClFN4O2	1
1	Ki = 27.9 nM Bioactivity Info	TI LI LO TS
CP0375516 Compound Info	1-Benzyl-4-(3-methyl-4-phenyl-pyrazol-1-yl)-piperidine Show/Hide	C22H25N3	1
1	Ki = 28 nM Bioactivity Info	TI LI LO TS
CP0409143 Compound Info	1-(benzofuran-3-ylmethyl)-4-(3,4-dichlorophenyl)piperidin-4-ol Show/Hide	C20H19Cl2NO2	1
1	Ki = 28 nM Bioactivity Info	TI LI LO TS
CP0845763 Compound Info	1-(4-Hydroxybenzyl)-apomorphine Hydrochloride Show/Hide	C24H24ClNO3	1
1	Ki = 28 nM Bioactivity Info	TI LI LO TS
CP0038049 Compound Info	N-[3-fluoro-4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]-1-benzofuran-2-carboxamide Show/Hide	C24H28FN3O3	1
1	Ki = 28.6 nM Bioactivity Info	TI LI LO TS
CP0414817 Compound Info	N-[(3S)-4-[4-(2,3-dichlorophenyl)piperazin-1-yl]-3-fluorobutyl]-1-benzofuran-2-carboxamide Show/Hide	C23H24Cl2FN3O2	1
1	Ki = 29 nM Bioactivity Info	TI LI LO TS
CP0513108 Compound Info	N-[4-[4-(7-chloroquinolin-4-yl)piperazin-1-yl]butyl]imidazo[1,2-a]pyridine-2-carboxamide Show/Hide	C25H27ClN6O	1
1	Ki = 29 nM Bioactivity Info	TI LI LO TS
CP0474296 Compound Info	4-[4-[3-[4-(2-methoxyphenyl)piperazin-1-yl]propyl]triazol-1-yl]-N,N-dimethylaniline Show/Hide	C24H32N6O	1
1	Ki = 29.6 nM Bioactivity Info	TI LI LO TS
CP0433565 Compound Info	1-[4-(2-methoxyphenyl)piperazin-1-yl]-4-[4-(4-phenylphenyl)triazol-1-yl]butan-2-ol Show/Hide	C29H33N5O2	1
1	Ki = 30.5 nM Bioactivity Info	TI LI LO TS
CP0880731 Compound Info	endo-8-(1H-Indol-3-ylmethyl)-3-(4-fluorophenyl)-8-azabicyclo[3.2.1]octan-3-ol Show/Hide	C22H23FN2O	1
1	Ki = 31 nM Bioactivity Info	TI LI LO TS
CP0157763 Compound Info	1-(2-chloro-3-ethylphenyl)piperazine Show/Hide	C12H17ClN2	1
1	Ki = 31.1 nM Bioactivity Info	TI LI LO TS
CP0382715 Compound Info	7-[4-[(2S,5S)-2-(6-aminopyridin-3-yl)-5-methylmorpholin-4-yl]butoxy]-3,4-dihydro-1H-quinolin-2-one Show/Hide	C23H30N4O3	1
1	Ki = 31.2 nM Bioactivity Info	TI LI LO TS
CP0376256 Compound Info	N-[4-[4-(3-chloro-2-methoxyphenyl)piperazin-1-yl]-3-hydroxybutyl]quinoline-3-carboxamide Show/Hide	C25H29ClN4O3	1
1	Ki = 31.6 nM Bioactivity Info	TI LI LO TS
CP0902371 Compound Info	1-(Benzofuran-2-ylmethyl)-4-(4-bromophenyl)piperidin-4-ol oxalate Show/Hide	C22H22BrNO6	1
1	Ki = 31.8 nM Bioactivity Info	TI LI LO TS
CP0399511 Compound Info	N-[4-[4-[2-tert-butyl-6-(trifluoromethyl)pyrimidin-4-yl]piperazin-1-yl]butyl]thieno[2,3-b]pyridine-2-carboxamide Show/Hide	C25H31F3N6OS	1
1	Ki = 32 nM Bioactivity Info	TI LI LO TS
CP0400252 Compound Info	N-[4-[4-[2-tert-butyl-6-(trifluoromethyl)pyrimidin-4-yl]piperazin-1-yl]butyl]-1-phenylpiperidine-4-carboxamide Show/Hide	C29H41F3N6O	1
1	Ki = 32 nM Bioactivity Info	TI LI LO TS
CP0396210 Compound Info	N-[[(1R,2R)-2-[(7-cyano-3,4-dihydro-1H-isoquinolin-2-yl)methyl]cyclopropyl]methyl]-1H-indole-2-carboxamide Show/Hide	C24H24N4O	1
1	Ki = 32 nM Bioactivity Info	TI LI LO TS
CP0852046 Compound Info	endo-8-(Benzofur-3-ylmethyl)-3-(2,3-dichlorophenyl)-8-azabicyclo[3.2.1]octan-3-ol Show/Hide	C22H21Cl2NO2	1
1	Ki = 32.2 nM Bioactivity Info	TI LI LO TS
CP0468994 Compound Info	3-(2-methoxyphenyl)-9-[3-[(5-phenyl-1H-1,2,4-triazol-3-yl)sulfanyl]propyl]-3,9-diazaspiro[5.5]undecane Show/Hide	C27H35N5OS	1
1	Ki = 32.5 nM Bioactivity Info	TI LI LO TS
CP0466447 Compound Info	N-[4-[4-(4-chlorophenyl)piperazin-1-yl]butyl]-4-thiophen-3-ylbenzamide Show/Hide	C25H28ClN3OS	1
1	Ki = 32.7 nM Bioactivity Info	TI LI LO TS
CP0416957 Compound Info	3-[2-(2-fluoroethoxy)phenyl]-9-[3-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]propyl]-3,9-diazaspiro[5.5]undecane Show/Hide	C29H38FN5OS	1
1	Ki = 33.3 nM Bioactivity Info	TI LI LO TS
CP0852588 Compound Info	(rac)-4-(4-(1H-Indol-5-yl)-1H-1,2,3-triazol-1-yl)-1-(4-(2-methoxyphenyl)piperazin-1-yl)butan-2-ol Show/Hide	C25H30N6O2	1
1	Ki = 33.6 nM Bioactivity Info	TI LI LO TS
CP0072089 Compound Info	N-[3-hydroxy-4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]quinoline-3-carboxamide Show/Hide	C25H30N4O3	1
1	Ki = 33.8 nM Bioactivity Info	TI LI LO TS
CP0396051 Compound Info	2-[2-[(6,6-diphenyl-1,4-dioxan-2-yl)methylamino]ethoxy]phenol Show/Hide	C25H27NO4	1
1	Ki = 33.88 nM Bioactivity Info	TI LI LO TS
CP0382710 Compound Info	N-[2-[2-[[(2S,5S)-2-(6-aminopyridin-3-yl)-5-methylmorpholin-4-yl]methyl]cyclopropyl]ethyl]-1H-indole-2-carboxamide Show/Hide	C25H31N5O2	2
1	Ki = 34 nM Bioactivity Info	TI LI LO TS
2	Ki = 284 nM Bioactivity Info	TI LI LO TS
CP0417546 Compound Info	(2S)-1-[4-(2,3-dichlorophenyl)piperazin-1-yl]butan-2-ol Show/Hide	C14H20Cl2N2O	1
1	Ki = 34.3 nM Bioactivity Info	TI LI LO TS
CP0139957 Compound Info	3-[Bis-(4-fluoro-phenyl)-methoxy]-8-butyl-8-aza-bicyclo[3.2.1]octane Show/Hide	C24H29F2NO	1
1	Ki = 34.4 nM Bioactivity Info	TI LI LO TS
CP0396168 Compound Info	3-(4-butylpiperazin-1-yl)benzonitrile Show/Hide	C15H21N3	1
1	Ki = 34.7 nM Bioactivity Info	TI LI LO TS
CP0381018 Compound Info	(+/-)-11-((1-(3-(4-(2,3-Dichlorophenyl)piperazin-1-yl)propyl)-1H-1,2,3-triazol-4-yl)methoxy)-N-propylnoraporphine Show/Hide	C35H40Cl2N6O	1
1	Ki = 35 nM Bioactivity Info	TI LI LO TS
CP0520591 Compound Info	3-amino-N-[4-[4-[2-tert-butyl-6-(trifluoromethyl)pyrimidin-4-yl]piperazin-1-yl]butyl]thieno[2,3-b]pyridine-2-carboxamide Show/Hide	C25H32F3N7OS	1
1	Ki = 35 nM Bioactivity Info	TI LI LO TS
CP0417010 Compound Info	N-[(3S)-4-[4-(3-chloro-5-ethyl-2-methoxyphenyl)piperazin-1-yl]-3-fluorobutyl]-1H-indole-2-carboxamide Show/Hide	C26H32ClFN4O2	1
1	Ki = 35.3 nM Bioactivity Info	TI LI LO TS
CP0400251 Compound Info	1-benzyl-N-[4-[4-[2-tert-butyl-6-(trifluoromethyl)pyrimidin-4-yl]piperazin-1-yl]butyl]piperidine-4-carboxamide Show/Hide	C30H43F3N6O	1
1	Ki = 36 nM Bioactivity Info	TI LI LO TS
CP0519088 Compound Info	N-[4-[4-(4-methylphenyl)piperazin-1-yl]butyl]-4-thiophen-3-ylbenzamide Show/Hide	C26H31N3OS	1
1	Ki = 36.1 nM Bioactivity Info	TI LI LO TS
CP0443872 Compound Info	N-[4-[4-(3-chloro-5-ethyl-2-methoxyphenyl)piperazin-1-yl]-3-hydroxybutyl]-1-benzofuran-2-carboxamide Show/Hide	C26H32ClN3O4	1
1	Ki = 36.1 nM Bioactivity Info	TI LI LO TS
CP0449717 Compound Info	2-[4-(2,3-dichlorophenyl)piperazin-1-yl]ethanol Show/Hide	C12H16Cl2N2O	1
1	Ki = 36.3 nM Bioactivity Info	TI LI LO TS
CP0375302 Compound Info	5-[4-[3-[4-(2-methoxyphenyl)piperazin-1-yl]propyl]triazol-1-yl]isoquinoline Show/Hide	C25H28N6O	1
1	Ki = 36.3 nM Bioactivity Info	TI LI LO TS
CP0427966 Compound Info	N-[3-hydroxy-4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]quinoline-7-carboxamide Show/Hide	C25H30N4O3	1
1	Ki = 37.7 nM Bioactivity Info	TI LI LO TS
CP0260574 Compound Info	CHEMBL3265065 Show/Hide	C29H33ClN2O2	1
1	Ki = 37.9 nM Bioactivity Info	TI LI LO TS
CP0063619 Compound Info	N-[(3S)-4-[4-(3-chloro-5-ethyl-2-methoxyphenyl)piperazin-1-yl]-3-hydroxybutyl]-1H-indole-2-carboxamide Show/Hide	C26H33ClN4O3	1
1	Ki = 37.9 nM Bioactivity Info	TI LI LO TS
CP0378670 Compound Info	1-(1-Benzyl-piperidin-4-yl)-5-methyl-4-thiophen-2-yl-1,3-dihydro-imidazol-2-one Show/Hide	C20H23N3OS	1
1	Ki = 38 nM Bioactivity Info	TI LI LO TS
CP0500313 Compound Info	N-[4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]propanamide Show/Hide	C18H29N3O2	1
1	Ki = 38.6 nM Bioactivity Info	TI LI LO TS
CP0492205 Compound Info	9-[3-[[5-(4-fluorophenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanyl]propyl]-3-(2-methoxyphenyl)-3,9-diazaspiro[5.5]undecane Show/Hide	C28H36FN5OS	1
1	Ki = 39.8 nM Bioactivity Info	TI LI LO TS
CP0410753 Compound Info	1-[4-(2-methoxyphenyl)piperazin-1-yl]-4-(4-naphthalen-2-yltriazol-1-yl)butan-2-ol Show/Hide	C27H31N5O2	1
1	Ki = 40.7 nM Bioactivity Info	TI LI LO TS
CP0535496 Compound Info	7-[4-[4-(3-chloro-5-ethyl-2-methoxyphenyl)piperazin-1-yl]butoxy]-3,4-dihydro-1H-quinolin-2-one Show/Hide	C26H34ClN3O3	1
1	Ki = 40.9 nM Bioactivity Info	TI LI LO TS
CP0373714 Compound Info	6-Methyl-5,6,7,8,13,15-hexahydro-4H-indolo[4,3a,3-fg][3]benzazacycloundecene Show/Hide	C20H22N2	1
1	Ki = 42.9 nM Bioactivity Info	TI LI LO TS
CP0427419 Compound Info	2-((4-(2-methoxyphenyl)piperazin-1-yl)methyl)H-pyrazolo[1,5-a]pyridine Show/Hide	C19H22N4O	8
1	Ki = 44 nM Bioactivity Info	TI LI LO TS
2	Ki = 51 nM Bioactivity Info	TI LI LO TS
3	Ki = 61 nM Bioactivity Info	TI LI LO TS
4	Ki = 340 nM Bioactivity Info	TI LI LO TS
5	Ki = 680 nM Bioactivity Info	TI LI LO TS
6	Ki = 720 nM Bioactivity Info	TI LI LO TS
7	Ki = 770 nM Bioactivity Info	TI LI LO TS
8	Ki = 2300 nM Bioactivity Info	TI LI LO TS
CP0503261 Compound Info	(+/-)-11-((1-(3-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)-1H-1,2,3-triazol-4-yl)methoxy)-N-propylnoraporphine Show/Hide	C35H42N6O2	1
1	Ki = 44 nM Bioactivity Info	TI LI LO TS
CP0478838 Compound Info	N-[4-[2,3-dihydro-1H-inden-2-yl(propyl)amino]butyl]pentanamide Show/Hide	C21H34N2O	2
1	Ki = 44 nM Bioactivity Info	TI LI LO TS
2	Ki = 760 nM Bioactivity Info	TI LI LO TS
CP0427930 Compound Info	4-(4-chlorophenyl)-1-((2-methyl-1H-indol-3-yl)methyl)piperidin-4-ol Show/Hide	C21H23ClN2O	1
1	Ki = 44.1 nM Bioactivity Info	TI LI LO TS
CP0396656 Compound Info	2,3-dimethoxy-N-[4-[4-(2-methoxyphenyl)-1,4-diazepan-1-yl]butyl]benzamide Show/Hide	C25H35N3O4	1
1	Ki = 44.2 nM Bioactivity Info	TI LI LO TS
CP0534583 Compound Info	6-fluoro-N-[3-hydroxy-4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]quinoline-3-carboxamide Show/Hide	C25H29FN4O3	1
1	Ki = 44.8 nM Bioactivity Info	TI LI LO TS
CP0051912 Compound Info	(5S)-N,N-dipropyl-4,5,6,7-tetrahydropyrazolo[1,5-a]pyridin-5-amine Show/Hide	C13H23N3	5
1	Ki = 45 nM Bioactivity Info	TI LI LO TS
2	Ki = 150 nM Bioactivity Info	TI LI LO TS
3	Ki = 420 nM Bioactivity Info	TI LI LO TS
4	Ki = 840 nM Bioactivity Info	TI LI LO TS
5	Ki = 8100 nM Bioactivity Info	TI LI LO TS
CP0482020 Compound Info	N-[4-[4-[2-tert-butyl-6-(trifluoromethyl)pyrimidin-4-yl]piperazin-1-yl]butyl]-5-(hydroxymethyl)imidazo[1,2-a]pyridine-2-carboxamide Show/Hide	C26H34F3N7O2	1
1	Ki = 45 nM Bioactivity Info	TI LI LO TS
CP0416956 Compound Info	3-(2-ethoxyphenyl)-9-[3-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]propyl]-3,9-diazaspiro[5.5]undecane Show/Hide	C29H39N5OS	1
1	Ki = 45.1 nM Bioactivity Info	TI LI LO TS
CP0393890 Compound Info	1-Benzyl-4-[5-(4-chloro-phenyl)-4-ethyl-1H-pyrazol-3-yl]-piperidine Show/Hide	C23H26ClN3	1
1	Ki = 46 nM Bioactivity Info	TI LI LO TS
CP0052067 Compound Info	2-((4-(4-chlorophenyl)piperazin-1-yl)methyl)-pyrazolo[1,5-a]pyridine Show/Hide	C18H19ClN4	8
1	Ki = 46 nM Bioactivity Info	TI LI LO TS
2	Ki = 76 nM Bioactivity Info	TI LI LO TS
3	Ki = 730 nM Bioactivity Info	TI LI LO TS
4	Ki = 1600 nM Bioactivity Info	TI LI LO TS
5	Ki = 2500 nM Bioactivity Info	TI LI LO TS
6	Ki = 8300 nM Bioactivity Info	TI LI LO TS
7	Ki = 9200 nM Bioactivity Info	TI LI LO TS
8	Ki = 12000 nM Bioactivity Info	TI LI LO TS
CP0861000 Compound Info	1-(1-(Benzo[b]thiophen-3-ylmethyl)piperidin-4-yl)-1Hbenzo[d]imidazol-2-(3H)-one oxalate Show/Hide	C23H23N3O5S	1
1	Ki = 46.7 nM Bioactivity Info	TI LI LO TS
CP0175178 Compound Info	11-methyl-11-aza-tricyclo[12.4.0.03,8]octadeca-1(18),3(8),4,6,14,16-hexaene Show/Hide	C18H21N	1
1	Ki = 47.5 nM Bioactivity Info	TI LI LO TS
CP0041232 Compound Info	1-((1H-indol-3-yl)methyl)-4-(4-chlorophenyl)piperidin-4-ol Show/Hide	C20H21ClN2O	3
1	Ki = 48.6 nM Bioactivity Info	TI LI LO TS
2	Ki = 104 nM Bioactivity Info	TI LI LO TS
3	Ki = 163 nM Bioactivity Info	TI LI LO TS
CP0416960 Compound Info	9-[3-[(4-ethyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]propyl]-3-(2-methoxyphenyl)-3,9-diazaspiro[5.5]undecane Show/Hide	C29H39N5OS	1
1	Ki = 48.7 nM Bioactivity Info	TI LI LO TS
CP0912200 Compound Info	1-(Benzofuran-2-ylmethyl)-4-(4-iodophenyl)piperidin-4-ol oxalate Show/Hide	C22H22INO6	1
1	Ki = 49 nM Bioactivity Info	TI LI LO TS
CP0167370 Compound Info	4-(2,3-dichlorophenyl)-1-(4-(4-(pyridin-2-yl)benzamido)-transbut-2-enyl)piperazine 1-oxide Show/Hide	C26H26Cl2N4O2	1
1	Ki = 49.2 nM Bioactivity Info	TI LI LO TS
CP0883762 Compound Info	(+/-)-trans-2-(4-Hydroxyphenyl)-1,2,3,4,4a,5,6,10b-octahydrobenzo[f]quinoline-8,9-diol Hydrobromide Show/Hide	C19H22BrNO3	1
1	Ki = 50 nM Bioactivity Info	TI LI LO TS
CP0383352 Compound Info	4-{(7-Hydroxy-1,2,3,4-tetrahydro-naphthalen-2-yl)-[3-(4-phenyl-piperazin-1-yl)-propyl]-amino}-butyronitrile Show/Hide	C27H36N4O	1
1	Ki = 50.2 nM Bioactivity Info	TI LI LO TS
CP0460520 Compound Info	N-[[(1R,2R)-2-[[4-(3-cyanophenyl)piperazin-1-yl]methyl]cyclopropyl]methyl]quinoline-4-carboxamide Show/Hide	C26H27N5O	1
1	Ki = 51.7 nM Bioactivity Info	TI LI LO TS
CP0853848 Compound Info	3-hydroxy-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine hydrobromide Show/Hide	C18H22BrNO	1
1	Ki = 52.5 nM Bioactivity Info	TI LI LO TS
CP0376254 Compound Info	N-[3-hydroxy-4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]-6-methylquinoline-3-carboxamide Show/Hide	C26H32N4O3	1
1	Ki = 52.9 nM Bioactivity Info	TI LI LO TS
CP0449024 Compound Info	1-(benzofuran-3-ylmethyl)-4-(4-chlorophenyl)piperidin-4-ol Show/Hide	C20H20ClNO2	1
1	Ki = 53 nM Bioactivity Info	TI LI LO TS
CP0861963 Compound Info	1-[4-(N,N-Dimethylamino)-benzyl]-apomorphine Dihydrochloride Show/Hide	C26H30Cl2N2O2	1
1	Ki = 53 nM Bioactivity Info	TI LI LO TS
CP0381584 Compound Info	6-fluoro-N-[3-hydroxy-4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]quinoline-2-carboxamide Show/Hide	C25H29FN4O3	1
1	Ki = 53.1 nM Bioactivity Info	TI LI LO TS
CP0482432 Compound Info	1-(2,3-dichlorophenyl)-4-methylpiperazine Show/Hide	C11H14Cl2N2	1
1	Ki = 54.6 nM Bioactivity Info	TI LI LO TS
CP0857932 Compound Info	1-Benzylapomorphine Hydrochloride Show/Hide	C24H24ClNO2	1
1	Ki = 55 nM Bioactivity Info	TI LI LO TS
CP0377602 Compound Info	N-[2-[(7-hydroxy-1,2,3,4-tetrahydronaphthalen-2-yl)-[3-(4-phenylpiperazin-1-yl)propyl]amino]ethyl]benzamide Show/Hide	C32H40N4O2	1
1	Ki = 55.7 nM Bioactivity Info	TI LI LO TS
CP0389447 Compound Info	1-[4-(2,3-dichlorophenyl)piperazin-1-yl]-4-[4-(4-phenylphenyl)triazol-1-yl]butan-2-ol Show/Hide	C28H29Cl2N5O	1
1	Ki = 55.8 nM Bioactivity Info	TI LI LO TS
CP0483049 Compound Info	9-[3-[(5-cyclohexyl-4-methyl-1,2,4-triazol-3-yl)sulfanyl]propyl]-3-(2-methoxyphenyl)-3,9-diazaspiro[5.5]undecane Show/Hide	C28H43N5OS	1
1	Ki = 57 nM Bioactivity Info	TI LI LO TS
CP0536765 Compound Info	3-(2-methoxyphenyl)-9-[4-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]butyl]-3,9-diazaspiro[5.5]undecane Show/Hide	C29H39N5OS	1
1	Ki = 59.2 nM Bioactivity Info	TI LI LO TS
CP0912198 Compound Info	8-(Benzo[b]thiophen-3-ylmethyl)-3-methyl-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one oxalate Show/Hide	C25H27N3O5S	1
1	Ki = 60.1 nM Bioactivity Info	TI LI LO TS
CP0574554 Compound Info	4-(dimethylamino)-N-[4-[3-(2-methoxyphenyl)-3,9-diazaspiro[5.5]undecan-9-yl]butyl]benzamide Show/Hide	C29H42N4O2	1
1	Ki = 61.5 nM Bioactivity Info	TI LI LO TS
CP0492204 Compound Info	3-(2-methoxyphenyl)-9-[3-[[5-(2-methoxyphenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanyl]propyl]-3,9-diazaspiro[5.5]undecane Show/Hide	C29H39N5O2S	1
1	Ki = 63 nM Bioactivity Info	TI LI LO TS
CP0517043 Compound Info	7-[(1R)-2-[[(1S,2S)-2-cyclohexylcyclopentyl]amino]-1-hydroxyethyl]-4-hydroxy-3H-1,3-benzothiazol-2-one Show/Hide	C20H28N2O3S	1
1	Ki = 64 nM Bioactivity Info	TI LI LO TS
CP0451508 Compound Info	N-[2-[bis(4-fluorophenyl)methylsulfanyl]ethyl]-3-phenylpropan-1-amine Show/Hide	C24H25F2NS	1
1	Ki = 65.9 nM Bioactivity Info	TI LI LO TS
CP0418991 Compound Info	[1-(benzenesulfonyl)-4-[2-(dimethylamino)ethyl]indol-2-yl]-phenylmethanone Show/Hide	C25H24N2O3S	1
1	Ki = 66 nM Bioactivity Info	TI LI LO TS
CP0389448 Compound Info	N-[(6,6-diphenyl-1,4-dioxan-2-yl)methyl]-2-[2-(methoxymethoxy)phenoxy]ethanamine Show/Hide	C27H31NO5	1
1	Ki = 66.07 nM Bioactivity Info	TI LI LO TS
CP0375617 Compound Info	N-(1-benzothiophen-3-ylmethyl)-4-[4-(2-methoxyphenyl)piperazin-1-yl]-N-propylbutan-1-amine Show/Hide	C27H37N3OS	1
1	Ki = 67.9 nM Bioactivity Info	TI LI LO TS
CP0919398 Compound Info	1-(1-((5-Methoxy-1H-indol-3-yl)methyl)piperidin-4-yl)-1H-benzo[d]imidazol-2(3H)-one oxalate Show/Hide	C24H26N4O6	1
1	Ki = 68.2 nM Bioactivity Info	TI LI LO TS
CP0381747 Compound Info	1-[4-(2-methoxyphenyl)piperazin-1-yl]-4-(4-quinolin-6-yltriazol-1-yl)butan-2-ol Show/Hide	C26H30N6O2	1
1	Ki = 68.2 nM Bioactivity Info	TI LI LO TS
CP0376255 Compound Info	N-[3-hydroxy-4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]-6-methoxyquinoline-3-carboxamide Show/Hide	C26H32N4O4	1
1	Ki = 69.9 nM Bioactivity Info	TI LI LO TS
CP0473557 Compound Info	N-(9H-fluoren-2-ylmethyl)-4-[4-(2-methoxyphenyl)piperazin-1-yl]-N-propylbutan-1-amine Show/Hide	C32H41N3O	1
1	Ki = 71.5 nM Bioactivity Info	TI LI LO TS
CP0058651 Compound Info	7-[(1R)-2-[2-(3-butylphenyl)ethylamino]-1-hydroxyethyl]-4-hydroxy-3H-1,3-benzothiazol-2-one Show/Hide	C21H26N2O3S	1
1	Ki = 73 nM Bioactivity Info	TI LI LO TS
CP0416961 Compound Info	3-[3-[3-(2-methoxyphenyl)-3,9-diazaspiro[5.5]undecan-9-yl]propylsulfanyl]-5-phenyl-1,2,4-triazol-4-amine Show/Hide	C27H36N6OS	1
1	Ki = 75 nM Bioactivity Info	TI LI LO TS
CP0485739 Compound Info	(2S)-1-[4-(2,3-dichlorophenyl)piperazin-1-yl]propan-2-ol Show/Hide	C13H18Cl2N2O	1
1	Ki = 75.2 nM Bioactivity Info	TI LI LO TS
CP0240206 Compound Info	N-[4-[methyl-[(10R)-2-oxo-1,3-diazatricyclo[6.3.1.04,12]dodeca-4,6,8(12)-trien-10-yl]amino]butyl]-1H-indole-2-carboxamide Show/Hide	C24H27N5O2	2
1	Ki = 76.9 nM Bioactivity Info	TI LI LO TS
2	Ki = 337 nM Bioactivity Info	TI LI LO TS
CP0482018 Compound Info	N-[4-(4-quinolin-2-ylpiperazin-1-yl)butyl]imidazo[1,2-a]pyridine-2-carboxamide Show/Hide	C25H28N6O	1
1	Ki = 77 nM Bioactivity Info	TI LI LO TS
CP0393851 Compound Info	(10R)-10-(methylamino)-3-[8-(4-phenylbutoxy)octyl]-1,3-diazatricyclo[6.3.1.04,12]dodeca-4,6,8(12)-trien-2-one Show/Hide	C29H41N3O2	1
1	Ki = 77.7 nM Bioactivity Info	TI LI LO TS
CP0513107 Compound Info	N-[4-[4-(2-tert-butylquinazolin-4-yl)piperazin-1-yl]butyl]imidazo[1,2-a]pyridine-2-carboxamide Show/Hide	C28H35N7O	1
1	Ki = 78 nM Bioactivity Info	TI LI LO TS
CP0391044 Compound Info	4-thiophen-3-yl-N-[4-[4-[4-(trifluoromethyl)phenyl]piperazin-1-yl]butyl]benzamide Show/Hide	C26H28F3N3OS	1
1	Ki = 78.3 nM Bioactivity Info	TI LI LO TS
CP0393889 Compound Info	1-(4-Chloro-benzyl)-4-[3-(4-chloro-phenyl)-isoxazol-5-yl]-piperidine Show/Hide	C21H20Cl2N2O	1
1	Ki = 80 nM Bioactivity Info	TI LI LO TS
CP0045069 Compound Info	2-[1-(benzenesulfonyl)-5-methoxyindol-3-yl]-N,N-dimethylethanamine Show/Hide	C19H22N2O3S	1
1	Ki = 80 nM Bioactivity Info	TI LI LO TS
CP0463700 Compound Info	(10R)-3-[6-(4-phenylbutoxy)hexyl]-10-(propylamino)-1,3-diazatricyclo[6.3.1.04,12]dodeca-4,6,8(12)-trien-2-one Show/Hide	C29H41N3O2	1
1	Ki = 80.6 nM Bioactivity Info	TI LI LO TS
CP0460211 Compound Info	4-(4-(2-Methoxyphenyl)piperazin-1-yl)-N-(naphthalen-2-ylmethyl)-N-propylbutan-1-amine Show/Hide	C29H39N3O	1
1	Ki = 80.8 nM Bioactivity Info	TI LI LO TS
CP0566757 Compound Info	3-(2,3-dichlorophenyl)-9-[3-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]propyl]-3,9-diazaspiro[5.5]undecane Show/Hide	C27H33Cl2N5S	1
1	Ki = 82.4 nM Bioactivity Info	TI LI LO TS
CP0447260 Compound Info	N-[4-[(10R)-10-(dipropylamino)-2-oxo-1,3-diazatricyclo[6.3.1.04,12]dodeca-4,6,8(12)-trien-3-yl]butyl]-1H-indole-2-carboxamide Show/Hide	C29H37N5O2	1
1	Ki = 83.9 nM Bioactivity Info	TI LI LO TS
CP0880730 Compound Info	endo-8-(1H-Indazol-3-ylmethyl)-3-(4-chlorophenyl)-8-azabicyclo[3.2.1]octan-3-ol Show/Hide	C21H22ClN3O	1
1	Ki = 84.7 nM Bioactivity Info	TI LI LO TS
CP0544829 Compound Info	4-(4-Iodophenyl)-1-((4-methoxy-1H-indol-3-yl)methyl)-piperidin-4-ol oxalate Show/Hide	C21H23IN2O2	1
1	Ki = 87.6 nM Bioactivity Info	TI LI LO TS
CP0889346 Compound Info	N-(Benzothiazol-2-yl)-5-(4-(2,4-dichlorophenyl)piperazin-1-yl)pentanamide hydrochloride Show/Hide	C22H25Cl3N4OS	1
1	Ki = 87.6 nM Bioactivity Info	TI LI LO TS
CP0468995 Compound Info	3-(2-methoxyphenyl)-9-[2-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]ethyl]-3,9-diazaspiro[5.5]undecane Show/Hide	C27H35N5OS	1
1	Ki = 89.7 nM Bioactivity Info	TI LI LO TS
CP0468996 Compound Info	N-[4-[3-(2-methoxyphenyl)-3,9-diazaspiro[5.5]undecan-9-yl]butyl]-4-thiophen-3-ylbenzamide Show/Hide	C31H39N3O2S	1
1	Ki = 92.9 nM Bioactivity Info	TI LI LO TS
CP0483747 Compound Info	1-(2-methoxyphenyl)-4-[3-[1-(2-methoxyphenyl)triazol-4-yl]propyl]piperazine Show/Hide	C23H29N5O2	1
1	Ki = 93.1 nM Bioactivity Info	TI LI LO TS
CP0393846 Compound Info	(10R)-3-[4-(4-phenylbutoxy)butyl]-10-(propylamino)-1,3-diazatricyclo[6.3.1.04,12]dodeca-4,6,8(12)-trien-2-one Show/Hide	C27H37N3O2	1
1	Ki = 94.2 nM Bioactivity Info	TI LI LO TS
CP0901061 Compound Info	1-((1H-Indol-3-yl)methyl)-4-(4-iodophenyl)piperidin-4-ol oxalate Show/Hide	C22H23IN2O5	1
1	Ki = 94.4 nM Bioactivity Info	TI LI LO TS
CP0506201 Compound Info	4-(4-bromophenyl)-1-((5-methoxy-1H-indol-3-yl)methyl)piperidin-4-ol Show/Hide	C21H23BrN2O2	1
1	Ki = 96.9 nM Bioactivity Info	TI LI LO TS
CP0411137 Compound Info	3-(4-methoxyphenyl)-9-[3-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]propyl]-3,9-diazaspiro[5.5]undecane Show/Hide	C28H37N5OS	1
1	Ki = 97.7 nM Bioactivity Info	TI LI LO TS
CP0382164 Compound Info	N-[3-hydroxy-4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]quinoline-2-carboxamide Show/Hide	C25H30N4O3	1
1	Ki = 97.9 nM Bioactivity Info	TI LI LO TS
CP0482019 Compound Info	N-[4-[4-[7-(trifluoromethyl)quinolin-4-yl]piperazin-1-yl]butyl]imidazo[1,2-a]pyridine-2-carboxamide Show/Hide	C26H27F3N6O	1
1	Ki = 99 nM Bioactivity Info	TI LI LO TS
CP0398934 Compound Info	(10R)-10-(methylamino)-3-propyl-1,3-diazatricyclo[6.3.1.04,12]dodeca-4,6,8(12)-trien-2-one Show/Hide	C14H19N3O	2
1	Ki = 99.5 nM Bioactivity Info	TI LI LO TS
2	Ki = 187 nM Bioactivity Info	TI LI LO TS
CP0063610 Compound Info	N-[4-[4-(3-chloro-5-ethyl-2-methoxyphenyl)piperazin-1-yl]-3-fluorobutyl]-1-benzofuran-2-carboxamide Show/Hide	C26H31ClFN3O3	1
1	Ki = 99.9 nM Bioactivity Info	TI LI LO TS
CP0902372 Compound Info	4-(4-Iodophenyl)-1-((5-methoxy-1H-indol-3-yl)methyl)-piperidin-4-ol oxalate Show/Hide	C23H25IN2O6	1
1	Ki = 100 nM Bioactivity Info	TI LI LO TS
CP0487362 Compound Info	N-(1-benzothiophen-3-ylmethyl)-4-[4-(2,3-dichlorophenyl)piperazin-1-yl]-N-propylbutan-1-amine Show/Hide	C26H33Cl2N3S	1
1	Ki = 101 nM Bioactivity Info	TI LI LO TS
CP0573032 Compound Info	3-(2-methoxyphenyl)-9-[3-[[4-methyl-5-(4-thiophen-3-ylphenyl)-1,2,4-triazol-3-yl]sulfanyl]propyl]-3,9-diazaspiro[5.5]undecane Show/Hide	C32H39N5OS2	1
1	Ki = 101 nM Bioactivity Info	TI LI LO TS
CP0454411 Compound Info	(+/-)-N-(3-(4-(2-methoxyphenyl)piperazin-1-yl)propyl)-N-(3-(N-propylnoraporphin-11-yloxy)-propyl)methanesulfonamide Show/Hide	C37H50N4O4S	1
1	Ki = 102 nM Bioactivity Info	TI LI LO TS
CP0495123 Compound Info	4-(4-(2,3-Dichlorophenyl)piperazin-1-yl)-N-(naphthalen-2-ylmethyl)-N-propylbutan-1-amine Show/Hide	C28H35Cl2N3	1
1	Ki = 104 nM Bioactivity Info	TI LI LO TS
CP0409654 Compound Info	(10R)-10-[methyl(propyl)amino]-1,3-diazatricyclo[6.3.1.04,12]dodeca-4,6,8(12)-trien-2-one Show/Hide	C14H19N3O	2
1	Ki = 104 nM Bioactivity Info	TI LI LO TS
2	Ki = 290 nM Bioactivity Info	TI LI LO TS
CP0449019 Compound Info	(1-((1H-indol-3-yl)methyl)-4-(4-chlorophenyl)piperidin-4-yl)methanol Show/Hide	C21H23ClN2O	1
1	Ki = 106 nM Bioactivity Info	TI LI LO TS
CP0318039 Compound Info	3-(2-Dimethylamino-ethyl)-1H-indole-2-carboxylic acid ethyl ester Show/Hide	C15H20N2O2	1
1	Ki = 110 nM Bioactivity Info	TI LI LO TS
CP0406019 Compound Info	1-((1H-indol-3-yl)methyl)-4-(4-bromophenyl)piperidin-4-ol Show/Hide	C20H21BrN2O	1
1	Ki = 110 nM Bioactivity Info	TI LI LO TS
CP0421766 Compound Info	1-((1H-indol-3-yl)methyl)-4-(3,4-dichlorophenyl)piperidin-4-ol Show/Hide	C20H20Cl2N2O	1
1	Ki = 111 nM Bioactivity Info	TI LI LO TS
CP0403227 Compound Info	3-(2,4-dimethoxyphenyl)-9-[3-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]propyl]-3,9-diazaspiro[5.5]undecane Show/Hide	C29H39N5O2S	1
1	Ki = 112 nM Bioactivity Info	TI LI LO TS
CP0393850 Compound Info	(10R)-10-(methylamino)-3-[10-(4-phenylbutoxy)decyl]-1,3-diazatricyclo[6.3.1.04,12]dodeca-4,6,8(12)-trien-2-one Show/Hide	C31H45N3O2	1
1	Ki = 113 nM Bioactivity Info	TI LI LO TS
CP0379809 Compound Info	4-hydroxy-7-[(1R)-1-hydroxy-2-[2-[4-(2-methylpropyl)phenyl]ethylamino]ethyl]-3H-1,3-benzothiazol-2-one Show/Hide	C21H26N2O3S	1
1	Ki = 115 nM Bioactivity Info	TI LI LO TS
CP0508464 Compound Info	N-[4-[(10R)-2-oxo-10-(propylamino)-1,3-diazatricyclo[6.3.1.04,12]dodeca-4,6,8(12)-trien-3-yl]butyl]-1H-indole-2-carboxamide Show/Hide	C26H31N5O2	1
1	Ki = 115 nM Bioactivity Info	TI LI LO TS
CP0463440 Compound Info	(2R)-1-[4-(2,3-dichlorophenyl)piperazin-1-yl]butan-2-ol Show/Hide	C14H20Cl2N2O	1
1	Ki = 119 nM Bioactivity Info	TI LI LO TS
CP0506670 Compound Info	1-(3-Chloro-benzyl)-4-(3-methyl-4-phenyl-pyrazol-1-yl)-piperidine Show/Hide	C22H24ClN3	1
1	Ki = 120 nM Bioactivity Info	TI LI LO TS
CP0548583 Compound Info	4-hydroxy-7-[(1R)-1-hydroxy-2-[[(1R,2R)-2-(2-phenylethyl)cyclopentyl]amino]ethyl]-3H-1,3-benzothiazol-2-one Show/Hide	C22H26N2O3S	1
1	Ki = 120 nM Bioactivity Info	TI LI LO TS
CP0861004 Compound Info	4-(4-Iodophenyl)-1-((4-methoxy-1H-indol-3-yl)methyl)-piperidin-4-ol oxalate Show/Hide	C23H25IN2O6	1
1	Ki = 122 nM Bioactivity Info	TI LI LO TS
CP0400250 Compound Info	N-[4-[4-(3,5-ditert-butylphenyl)piperazin-1-yl]butyl]imidazo[1,2-a]pyridine-2-carboxamide Show/Hide	C30H43N5O	1
1	Ki = 124 nM Bioactivity Info	TI LI LO TS
CP0478474 Compound Info	4-[4-(2,3-dichlorophenyl)piperazin-1-yl]-N-(9H-fluoren-2-ylmethyl)-N-propylbutan-1-amine Show/Hide	C31H37Cl2N3	1
1	Ki = 129 nM Bioactivity Info	TI LI LO TS
CP0517044 Compound Info	7-[(1R)-2-[2-(4-butoxyphenyl)ethylamino]-1-hydroxyethyl]-4-hydroxy-3H-1,3-benzothiazol-2-one Show/Hide	C21H26N2O4S	1
1	Ki = 129 nM Bioactivity Info	TI LI LO TS
CP0378625 Compound Info	1-(1-Benzyl-piperidin-4-yl)-5-ethyl-4-phenyl-1,3-dihydro-imidazol-2-one Show/Hide	C23H27N3O	1
1	Ki = 130 nM Bioactivity Info	TI LI LO TS
CP0860438 Compound Info	1-(4-Hydroxynaphthylmethyl)-apomorphine Hydrochloride Show/Hide	C28H26ClNO3	1
1	Ki = 130 nM Bioactivity Info	TI LI LO TS
CP0411141 Compound Info	(11S)-N-[(4-cyanophenyl)methyl]-5-ethyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide Show/Hide	C24H19N3O3S	1
1	Ki = 130 nM Bioactivity Info	TI LI LO TS
CP0861003 Compound Info	1-(1-((4-Methoxy-1H-indol-3-yl)methyl)piperidin-4-yl)-1H-benzo[d]imidazol-2(3H)-one oxalate Show/Hide	C24H26N4O6	1
1	Ki = 132 nM Bioactivity Info	TI LI LO TS
CP0482239 Compound Info	4-(((9H-Fluoren-2-yl)methyl)amino)-1-(4-(2,3-dichlorophenyl)piperazin-1-yl)butan-2-ol Show/Hide	C28H31Cl2N3O	1
1	Ki = 134 nM Bioactivity Info	TI LI LO TS
CP0482017 Compound Info	N-[4-[4-(6-tert-butyl-2-methylpyrimidin-4-yl)piperazin-1-yl]butyl]imidazo[1,2-a]pyridine-2-carboxamide Show/Hide	C25H35N7O	1
1	Ki = 134 nM Bioactivity Info	TI LI LO TS
CP0492203 Compound Info	4-[5-[3-[3-(2-methoxyphenyl)-3,9-diazaspiro[5.5]undecan-9-yl]propylsulfanyl]-4-methyl-1,2,4-triazol-3-yl]-N,N-dimethylaniline Show/Hide	C30H42N6OS	1
1	Ki = 138 nM Bioactivity Info	TI LI LO TS
CP0372385 Compound Info	1-(benzofuran-3-ylmethyl)-4-(4-(methylthio)phenyl)piperidin-4-ol Show/Hide	C21H23NO2S	1
1	Ki = 139 nM Bioactivity Info	TI LI LO TS
CP0463699 Compound Info	(10R)-10-(methylamino)-3-[6-(4-phenylbutoxy)hexyl]-1,3-diazatricyclo[6.3.1.04,12]dodeca-4,6,8(12)-trien-2-one Show/Hide	C27H37N3O2	1
1	Ki = 139 nM Bioactivity Info	TI LI LO TS
CP0420764 Compound Info	4-(1-Benzyl-piperidin-4-yl)-6-(4-chloro-phenyl)-pyrimidin-2-ylamine Show/Hide	C22H23ClN4	1
1	Ki = 140 nM Bioactivity Info	TI LI LO TS
CP0512281 Compound Info	1-(1-Benzyl-piperidin-4-yl)-3,5-dimethyl-4-phenyl-1,3-dihydro-imidazol-2-one Show/Hide	C23H27N3O	1
1	Ki = 140 nM Bioactivity Info	TI LI LO TS
CP0472714 Compound Info	(10R)-10-(methylamino)-3-[12-(4-phenylbutoxy)dodecyl]-1,3-diazatricyclo[6.3.1.04,12]dodeca-4,6,8(12)-trien-2-one Show/Hide	C33H49N3O2	1
1	Ki = 141 nM Bioactivity Info	TI LI LO TS
CP0927947 Compound Info	1-(Benzo[b]thiophen-2-ylmethyl)-4-(4-bromophenyl)-piperidin-4-ol oxalate Show/Hide	C22H23NO5S	1
1	Ki = 142 nM Bioactivity Info	TI LI LO TS
CP0064477 Compound Info	7-[(1R)-2-[2-(3-butoxyphenyl)ethylamino]-1-hydroxyethyl]-4-hydroxy-3H-1,3-benzothiazol-2-one Show/Hide	C21H26N2O4S	1
1	Ki = 144 nM Bioactivity Info	TI LI LO TS
CP0386821 Compound Info	N-[4-[4-[6-methyl-2-(trifluoromethyl)pyrimidin-4-yl]piperazin-1-yl]butyl]imidazo[1,2-a]pyridine-2-carboxamide Show/Hide	C22H26F3N7O	1
1	Ki = 148 nM Bioactivity Info	TI LI LO TS
CP0259163 Compound Info	4-hydroxy-7-[(1R)-1-hydroxy-2-[2-(4-propylphenyl)ethylamino]ethyl]-3H-1,3-benzothiazol-2-one Show/Hide	C20H24N2O3S	1
1	Ki = 149 nM Bioactivity Info	TI LI LO TS
CP0408800 Compound Info	2-butyl-3,4-dihydro-1H-isoquinoline-7-carbonitrile Show/Hide	C14H18N2	1
1	Ki = 149 nM Bioactivity Info	TI LI LO TS
CP0449085 Compound Info	1-(1-Benzyl-piperidin-4-yl)-3-methyl-4-phenyl-1,3-dihydro-imidazol-2-one Show/Hide	C22H25N3O	1
1	Ki = 150 nM Bioactivity Info	TI LI LO TS
CP0322398 Compound Info	4-hydroxy-7-[(1R)-1-hydroxy-2-[2-(3-propylphenyl)ethylamino]ethyl]-3H-1,3-benzothiazol-2-one Show/Hide	C20H24N2O3S	1
1	Ki = 152 nM Bioactivity Info	TI LI LO TS
CP0449018 Compound Info	1-((1H-indazol-3-yl)methyl)-4-(3,4-dichlorophenyl)piperidin-4-ol Show/Hide	C19H19Cl2N3O	1
1	Ki = 156 nM Bioactivity Info	TI LI LO TS
CP0406327 Compound Info	1-Benzyl-4-[5-(4-chloro-phenyl)-1H-pyrazol-3-yl]-piperidine Show/Hide	C21H22ClN3	1
1	Ki = 160 nM Bioactivity Info	TI LI LO TS
CP0277135 Compound Info	N-[[(1S,2R)-2-[[4-(2,3-dichlorophenyl)piperazin-1-yl]methyl]cyclopropyl]methyl]-4-pyridin-2-ylbenzamide Show/Hide	C27H28Cl2N4O	1
1	Ki = 160 nM Bioactivity Info	TI LI LO TS
CP0460213 Compound Info	4-(((9H-Fluoren-2-yl)methyl)(methyl)amino)-1-(4-(2,3-dichlorophenyl)piperazin-1-yl)butan-2-ol Show/Hide	C29H33Cl2N3O	1
1	Ki = 162 nM Bioactivity Info	TI LI LO TS
CP0384374 Compound Info	2-(3',4',-5',6'-tetrahydro-2'H-[2,4'-bipyridine]-1'-yl)-N-(m-tolyl)acetamide Show/Hide	C19H23N3O	2
1	Ki = 167 nM Bioactivity Info	TI LI LO TS
2	Ki = 1680 nM Bioactivity Info	TI LI LO TS
CP0437100 Compound Info	1-(2-methoxyphenyl)-7-[3-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]propyl]-1,7-diazaspiro[3.5]nonane Show/Hide	C26H33N5OS	1
1	Ki = 169 nM Bioactivity Info	TI LI LO TS
CP0381741 Compound Info	1-[4-(2-methoxyphenyl)piperazin-1-yl]-4-(4-phenyltriazol-1-yl)butan-2-ol Show/Hide	C23H29N5O2	1
1	Ki = 173 nM Bioactivity Info	TI LI LO TS
CP0382713 Compound Info	7-[4-[(5S)-2-(6-aminopyridin-3-yl)-5-methylmorpholin-4-yl]butoxy]-3,4-dihydro-1H-quinolin-2-one Show/Hide	C23H30N4O3	1
1	Ki = 173 nM Bioactivity Info	TI LI LO TS
CP0167921 Compound Info	1-(3-chloro-5-ethyl-2-methoxyphenyl)-4-methylpiperazine Show/Hide	C14H21ClN2O	1
1	Ki = 179 nM Bioactivity Info	TI LI LO TS
CP0448500 Compound Info	1-[1-(4-Chloro-benzyl)-piperidin-4-yl]-5-methyl-4-phenyl-1,3-dihydro-imidazol-2-one Show/Hide	C22H24ClN3O	1
1	Ki = 180 nM Bioactivity Info	TI LI LO TS
CP0425631 Compound Info	5-[(5S)-5-methyl-4-propylmorpholin-2-yl]pyridin-2-amine Show/Hide	C13H21N3O	1
1	Ki = 185 nM Bioactivity Info	TI LI LO TS
CP0902374 Compound Info	4-(4-Bromophenyl)-1-((5-(2-fluoroethoxy)-1H-indol-3-yl)-methyl)piperidin-4-ol oxalate Show/Hide	C24H26BrFN2O6	1
1	Ki = 188 nM Bioactivity Info	TI LI LO TS
CP0454413 Compound Info	(-)-S-11-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butoxy)-N-propylnoraporphine Show/Hide	C34H43N3O2	1
1	Ki = 189 nM Bioactivity Info	TI LI LO TS
CP0129799 Compound Info	(4-Ethynyl-cyclohex-3-enyl)-dipropyl-amine Show/Hide	C14H23N	3
1	Ki = 190 nM Bioactivity Info	TI LI LO TS
2	Ki = 5700 nM Bioactivity Info	TI LI LO TS
3	Ki > 10000 nM Bioactivity Info	TI LI LO TS
CP0377177 Compound Info	4-(4-bromophenyl)-1-((4-methoxy-1H-indol-3-yl)methyl)piperidin-4-ol Show/Hide	C21H23BrN2O2	1
1	Ki = 190 nM Bioactivity Info	TI LI LO TS
CP0377128 Compound Info	(+/-)-11-((1-(3-(4-Phenylpiperazin-1-yl)propyl)-1H-1,2,3-triazol-4-yl)methoxy)-N-propylnoraporphine Show/Hide	C35H42N6O	1
1	Ki = 191 nM Bioactivity Info	TI LI LO TS
CP0547876 Compound Info	7-(2-methoxyphenyl)-2-[3-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]propyl]-2,7-diazaspiro[3.4]octane Show/Hide	C25H31N5OS	1
1	Ki = 192 nM Bioactivity Info	TI LI LO TS
CP0409195 Compound Info	N-[4-(4-chlorophenyl)-1-(1H-indol-3-ylmethyl)piperidin-4-yl]acetamide Show/Hide	C22H24ClN3O	1
1	Ki = 193 nM Bioactivity Info	TI LI LO TS
CP0364794 Compound Info	1-(2,3-dichlorophenyl)piperazine Show/Hide	C10H12Cl2N2	1
1	Ki = 197.4 nM Bioactivity Info	TI LI LO TS
CP0025667 Compound Info	2-[4-(4-Methyl-benzyl)-piperazin-1-yl]-1-(2-methyl-2,3-dihydro-indol-1-yl)-ethanone Show/Hide	C18H19ClN4	1
1	Ki = 200 nM Bioactivity Info	TI LI LO TS
CP0504160 Compound Info	4-(4-chlorophenyl)-1-((5-methoxy-1H-indol-3-yl)methyl)piperidin-4-ol Show/Hide	C21H23ClN2O2	1
1	Ki = 204 nM Bioactivity Info	TI LI LO TS
CP0384492 Compound Info	3-(2-fluorophenyl)-9-[3-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]propyl]-3,9-diazaspiro[5.5]undecane Show/Hide	C27H34FN5S	1
1	Ki = 208 nM Bioactivity Info	TI LI LO TS
CP0038689 Compound Info	(4aS,5R,10bR)-5-phenyl-1,2,3,4,4a,5,6,10b-octahydrobenzo[h]isoquinoline-7,8-diol Show/Hide	C19H21NO2	1
1	Ki = 210 nM Bioactivity Info	TI LI LO TS
CP0445424 Compound Info	3-((4-(4-chlorophenyl)-4-fluoropiperidin-1-yl)methyl)-1H-indole Show/Hide	C20H20ClFN2	1
1	Ki = 211 nM Bioactivity Info	TI LI LO TS
CP0384491 Compound Info	3-(2-methoxyphenyl)-9-[3-[(4-methyl-5-pyridin-3-yl-1,2,4-triazol-3-yl)sulfanyl]propyl]-3,9-diazaspiro[5.5]undecane Show/Hide	C27H36N6OS	1
1	Ki = 213 nM Bioactivity Info	TI LI LO TS
CP0455116 Compound Info	1-(1-Benzyl-piperidin-4-yl)-5-methyl-4-p-tolyl-1,3-dihydro-imidazol-2-one Show/Hide	C23H27N3O	1
1	Ki = 220 nM Bioactivity Info	TI LI LO TS
CP0455407 Compound Info	1-(1-Benzyl-piperidin-4-yl)-4-(2-chloro-phenyl)-5-methyl-1,3-dihydro-imidazol-2-one Show/Hide	C22H24ClN3O	1
1	Ki = 220 nM Bioactivity Info	TI LI LO TS
CP0496624 Compound Info	2-[5-[4-(4-Chlorophenyl)piperazin-1-yl]pentyl]pyrazolo[1,5-a]-pyridine Show/Hide	C22H27ClN4	4
1	Ki = 220 nM Bioactivity Info	TI LI LO TS
2	Ki = 530 nM Bioactivity Info	TI LI LO TS
3	Ki = 1100 nM Bioactivity Info	TI LI LO TS
4	Ki = 1900 nM Bioactivity Info	TI LI LO TS
CP0914958 Compound Info	endo-8-(1H-Indol-3-ylmethyl)-3-(2-naphthyl)-8-azabicyclo[3.2.1]octan-3-ol Show/Hide	C26H26N2O	1
1	Ki = 224 nM Bioactivity Info	TI LI LO TS
CP0393860 Compound Info	(10R)-10-(methylamino)-3-[2-[2-(4-phenylbutoxy)ethoxy]ethyl]-1,3-diazatricyclo[6.3.1.04,12]dodeca-4,6,8(12)-trien-2-one Show/Hide	C25H33N3O3	1
1	Ki = 227 nM Bioactivity Info	TI LI LO TS
CP0494338 Compound Info	2-N,N-dipropylaminoindane Show/Hide	C15H23N	2
1	Ki = 230 nM Bioactivity Info	TI LI LO TS
2	Ki = 350 nM Bioactivity Info	TI LI LO TS
CP0530680 Compound Info	(11S)-5-ethyl-N-[(4-fluorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide Show/Hide	C23H19FN2O3S	1
1	Ki = 230 nM Bioactivity Info	TI LI LO TS
CP0407283 Compound Info	2-(2-methoxyphenyl)-7-[3-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]propyl]-2,7-diazaspiro[3.5]nonane Show/Hide	C26H33N5OS	1
1	Ki = 235 nM Bioactivity Info	TI LI LO TS
CP0449015 Compound Info	4-(4-chlorophenyl)-1-((1-methyl-1H-indol-3-yl)methyl)piperidin-4-ol Show/Hide	C21H23ClN2O	1
1	Ki = 238 nM Bioactivity Info	TI LI LO TS
CP0508564 Compound Info	1-Benzyl-3-[5-(4-chloro-phenyl)-1H-pyrazol-3-yl]-piperidine Show/Hide	C21H22ClN3	1
1	Ki = 240 nM Bioactivity Info	TI LI LO TS
CP0467016 Compound Info	1-(1-Benzyl-piperidin-4-yl)-5-methyl-4-phenyl-1,3-dihydro-imidazol-2-one Show/Hide	C22H25N3O	1
1	Ki = 240 nM Bioactivity Info	TI LI LO TS
CP0403521 Compound Info	1-(1-Benzyl-piperidin-4-yl)-4-(3-chloro-phenyl)-5-methyl-1,3-dihydro-imidazol-2-one Show/Hide	C22H24ClN3O	1
1	Ki = 250 nM Bioactivity Info	TI LI LO TS
CP0504457 Compound Info	4-(4-chlorophenyl)-1-((4-methoxy-1H-indol-3-yl)methyl)piperidin-4-ol Show/Hide	C21H23ClN2O2	1
1	Ki = 250 nM Bioactivity Info	TI LI LO TS
CP0913527 Compound Info	7-(4-(4-(2-Methoxy-4-methylphenyl)piperazin-1-yl)butoxy)-3,4-dihydroquinolin-2(1H)-one oxalate Show/Hide	C27H35N3O7	1
1	Ki = 251 nM Bioactivity Info	TI LI LO TS
CP0379466 Compound Info	N-[4-(4-quinazolin-4-ylpiperazin-1-yl)butyl]imidazo[1,2-a]pyridine-2-carboxamide Show/Hide	C24H27N7O	1
1	Ki = 253 nM Bioactivity Info	TI LI LO TS
CP0398933 Compound Info	N-[4-[methyl-[(10R)-2-oxo-1,3-diazatricyclo[6.3.1.04,12]dodeca-4,6,8(12)-trien-10-yl]amino]butyl]-1-benzofuran-2-carboxamide Show/Hide	C24H26N4O3	2
1	Ki = 256 nM Bioactivity Info	TI LI LO TS
2	Ki = 2610 nM Bioactivity Info	TI LI LO TS
CP0396213 Compound Info	N-[[(1R,2R)-2-[(7-cyano-3,4-dihydro-1H-isoquinolin-2-yl)methyl]cyclopropyl]methyl]quinoline-4-carboxamide Show/Hide	C25H24N4O	1
1	Ki = 256 nM Bioactivity Info	TI LI LO TS
CP0421822 Compound Info	1-[(6,6-diphenyl-1,4-dioxan-2-yl)methyl]-4-(2-methoxyphenyl)piperazine Show/Hide	C28H32N2O3	1
1	Ki = 257.04 nM Bioactivity Info	TI LI LO TS
CP0492442 Compound Info	3-[4-(3-Methyl-4-phenyl-pyrazol-1-yl)-piperidin-1-ylmethyl]-benzonitrile Show/Hide	C23H24N4	1
1	Ki = 260 nM Bioactivity Info	TI LI LO TS
CP0495774 Compound Info	3-((4-(4-chlorophenyl)-4-methoxypiperidin-1-yl)methyl)-1H-indole Show/Hide	C21H23ClN2O	1
1	Ki = 262 nM Bioactivity Info	TI LI LO TS
CP0409196 Compound Info	1-((1H-indol-3-yl)methyl)-4-(2,3-dichlorophenyl)piperidin-4-ol Show/Hide	C20H20Cl2N2O	1
1	Ki = 273 nM Bioactivity Info	TI LI LO TS
CP0123458 Compound Info	4-hydroxy-7-[(1R)-1-hydroxy-2-[[(1R,2R)-2-(3-methylphenyl)cyclopentyl]amino]ethyl]-3H-1,3-benzothiazol-2-one Show/Hide	C21H24N2O3S	1
1	Ki = 279 nM Bioactivity Info	TI LI LO TS
CP0461813 Compound Info	[(1S,2R,5R,6R,7R)-3-benzyl-2-phenyl-7-pyrrolidin-1-yl-3-azabicyclo[3.2.0]heptan-6-yl]methanol Show/Hide	C24H30N2O	1
1	Ki = 280 nM Bioactivity Info	TI LI LO TS
CP0395778 Compound Info	(+/-)-11-(3-(4-((4-(2-Methoxyphenyl)piperazin-1-yl)methyl)-1H-1,2,3-triazol-1-yl)propoxy)-N-propylnoraporphine Show/Hide	C36H44N6O2	1
1	Ki = 281 nM Bioactivity Info	TI LI LO TS
CP0411640 Compound Info	1-[3-(4-pentylpiperidin-1-yl)propyl]-3,4-dihydroquinolin-2-one Show/Hide	C22H34N2O	1
1	Ki = 281.84 nM Bioactivity Info	TI LI LO TS
CP0438521 Compound Info	N-[2-[(1S,2R)-2-[[(2S,5S)-2-(6-aminopyridin-3-yl)-5-methylmorpholin-4-yl]methyl]cyclopropyl]ethyl]-1H-indole-2-carboxamide Show/Hide	C25H31N5O2	2
1	Ki = 282 nM Bioactivity Info	TI LI LO TS
2	Ki = 2900 nM Bioactivity Info	TI LI LO TS
CP0330654 Compound Info	2-[1-(benzenesulfonyl)indol-4-yl]-N,N-dimethylethanamine Show/Hide	C18H20N2O2S	1
1	Ki = 300 nM Bioactivity Info	TI LI LO TS
CP0431322 Compound Info	(12S)-11,12-dimethyl-11,21-diazatetracyclo[12.7.0.03,8.015,20]henicosa-1(14),3,5,7,15,17,19-heptaene Show/Hide	C21H24N2	1
1	Ki = 304 nM Bioactivity Info	TI LI LO TS
CP0429805 Compound Info	5-Methyl-1-[1-(3-methyl-benzyl)-piperidin-4-yl]-4-phenyl-1,3-dihydro-imidazol-2-one Show/Hide	C23H27N3O	1
1	Ki = 320 nM Bioactivity Info	TI LI LO TS
CP0478649 Compound Info	N-[4-[2,3-dihydro-1H-inden-2-yl(propyl)amino]butyl]acetamide Show/Hide	C18H28N2O	2
1	Ki = 330 nM Bioactivity Info	TI LI LO TS
2	Ki = 410 nM Bioactivity Info	TI LI LO TS
CP0382130 Compound Info	(11S)-5-methyl-6,11-dioxo-N-(2-pyrrolidin-1-ylethyl)benzo[b][1,4]benzothiazepine-3-carboxamide Show/Hide	C21H23N3O3S	1
1	Ki = 350 nM Bioactivity Info	TI LI LO TS
CP0437037 Compound Info	1-(1-Benzyl-piperidin-4-yl)-4-(4-methoxy-phenyl)-5-methyl-1,3-dihydro-imidazol-2-one Show/Hide	C23H27N3O2	1
1	Ki = 360 nM Bioactivity Info	TI LI LO TS
CP0411142 Compound Info	(11S)-N-[(4-bromophenyl)methyl]-5-methyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide Show/Hide	C22H17BrN2O3S	1
1	Ki = 370 nM Bioactivity Info	TI LI LO TS
CP0416710 Compound Info	3-[2-fluoro-4-(trifluoromethyl)phenyl]-9-[3-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]propyl]-3,9-diazaspiro[5.5]undecane Show/Hide	C28H33F4N5S	1
1	Ki = 370 nM Bioactivity Info	TI LI LO TS
CP0560050 Compound Info	(2R)-1-[4-(2,3-dichlorophenyl)piperazin-1-yl]propan-2-ol Show/Hide	C13H18Cl2N2O	1
1	Ki = 373 nM Bioactivity Info	TI LI LO TS
CP0455784 Compound Info	(10R)-10-(methylamino)-3-[4-(4-phenylbutoxy)butyl]-1,3-diazatricyclo[6.3.1.04,12]dodeca-4,6,8(12)-trien-2-one Show/Hide	C25H33N3O2	1
1	Ki = 377 nM Bioactivity Info	TI LI LO TS
CP0424155 Compound Info	1-(1-Benzyl-piperidin-4-yl)-4-(4-chloro-phenyl)-5-methyl-1,3-dihydro-imidazol-2-one Show/Hide	C22H24ClN3O	1
1	Ki = 380 nM Bioactivity Info	TI LI LO TS
CP0046420 Compound Info	CAS_3853 Show/Hide	C18H19ClN4	1
1	Ki = 380.19 nM Bioactivity Info	TI LI LO TS
CP0427783 Compound Info	1-((1H-indol-3-yl)methyl)-4-(4-chlorophenyl)piperidin-4-amine Show/Hide	C20H22ClN3	1
1	Ki = 382 nM Bioactivity Info	TI LI LO TS
CP0393849 Compound Info	(10R)-10-[methyl-[4-[(2-oxo-3,4-dihydro-1H-quinolin-7-yl)oxy]butyl]amino]-1,3-diazatricyclo[6.3.1.04,12]dodeca-4,6,8(12)-trien-2-one Show/Hide	C24H28N4O3	1
1	Ki = 382 nM Bioactivity Info	TI LI LO TS
CP0416955 Compound Info	3-(2-methoxyphenyl)-9-[3-[(5-phenyl-1H-imidazol-2-yl)sulfanyl]propyl]-3,9-diazaspiro[5.5]undecane Show/Hide	C28H36N4OS	1
1	Ki = 383 nM Bioactivity Info	TI LI LO TS
CP0206600 Compound Info	4-[4-(2,3-dichlorophenyl)piperazin-1-yl]-N-(9H-fluoren-2-ylmethyl)-3-fluoro-N-methylbutan-1-amine Show/Hide	C29H32Cl2FN3	1
1	Ki = 393 nM Bioactivity Info	TI LI LO TS
CP0384496 Compound Info	2-[9-[3-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]propyl]-3,9-diazaspiro[5.5]undecan-3-yl]phenol Show/Hide	C27H35N5OS	1
1	Ki = 396 nM Bioactivity Info	TI LI LO TS
CP0471920 Compound Info	(4aR,10bR)-2,3,4,4a,5,10b-hexahydrochromeno[4,3-b][1,4]oxazin-9-ol Show/Hide	C11H13NO3	1
1	Ki = 403 nM Bioactivity Info	TI LI LO TS
CP0393635 Compound Info	1-[3-[4-(2-phenylethyl)piperidin-1-yl]propyl]-3,4-dihydroquinolin-2-one Show/Hide	C25H32N2O	1
1	Ki = 407.38 nM Bioactivity Info	TI LI LO TS
CP0384711 Compound Info	3-(2-methoxyphenyl)-9-[3-(1-methyl-5-phenylimidazol-2-yl)sulfanylpropyl]-3,9-diazaspiro[5.5]undecane Show/Hide	C29H38N4OS	1
1	Ki = 418 nM Bioactivity Info	TI LI LO TS
CP0944914 Compound Info	N-(4-((2S,5S)-2-(6-aminopyridin-3-yl)-5-methylmorpholino)-3-hydroxybutyl)-1H-indole-2-carboxamide Show/Hide	C23H29N5O3	1
1	Ki = 423 nM Bioactivity Info	TI LI LO TS
CP0451512 Compound Info	1-[4-[2-[bis(4-fluorophenyl)methylsulfanyl]ethyl]piperazin-1-yl]propan-2-ol Show/Hide	C22H28F2N2OS	1
1	Ki = 424 nM Bioactivity Info	TI LI LO TS
CP0440942 Compound Info	5-[(2S,5S)-5-methylmorpholin-2-yl]pyridin-2-amine Show/Hide	C10H15N3O	1
1	Ki = 424 nM Bioactivity Info	TI LI LO TS
CP0887642 Compound Info	7-(4-(3-Methyl-4-oxo-1-phenyl-1,3,8-triazaspiro[4.5]decan-8-yl)butoxy)-3,4-dihydro-quinolin-2(1H)-one oxalate Show/Hide	C29H36N4O7	1
1	Ki = 427 nM Bioactivity Info	TI LI LO TS
CP0394248 Compound Info	1-Benzyl-4-[5-(4-chloro-phenyl)-4-methyl-1H-pyrazol-3-yl]-piperidine Show/Hide	C22H24ClN3	1
1	Ki = 430 nM Bioactivity Info	TI LI LO TS
CP0460885 Compound Info	1-(4-Chloro-benzyl)-4-[5-(4-chloro-phenyl)-isoxazol-3-yl]-piperidine Show/Hide	C21H20Cl2N2O	1
1	Ki = 430 nM Bioactivity Info	TI LI LO TS
CP0852047 Compound Info	endo-8-(Benzothien-3-ylmethyl)-3-(2,3-dichlorophenyl)-8-azabicyclo[3.2.1]octan-3-ol Show/Hide	C22H21Cl2NOS	1
1	Ki = 431 nM Bioactivity Info	TI LI LO TS
CP0384369 Compound Info	2-(4-phenylpiperidin-1-yl)-N-(m-tolyl)acetamide Show/Hide	C20H24N2O	2
1	Ki = 433 nM Bioactivity Info	TI LI LO TS
2	Ki = 777 nM Bioactivity Info	TI LI LO TS
CP0407284 Compound Info	3-[9-[3-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]propyl]-3,9-diazaspiro[5.5]undecan-3-yl]benzonitrile Show/Hide	C28H34N6S	1
1	Ki = 438 nM Bioactivity Info	TI LI LO TS
CP0467820 Compound Info	1-((1H-indazol-3-yl)methyl)-4-(4-chlorophenyl)piperidin-4-ol Show/Hide	C19H20ClN3O	1
1	Ki = 440 nM Bioactivity Info	TI LI LO TS
CP0135681 Compound Info	1-(3-chloro-5-ethyl-2-methoxyphenyl)piperazine Show/Hide	C13H19ClN2O	1
1	Ki = 446 nM Bioactivity Info	TI LI LO TS
CP0375430 Compound Info	1-Benzyl-4-(5-methyl-4-phenyl-pyrazol-1-yl)-piperidine Show/Hide	C22H25N3	1
1	Ki = 450 nM Bioactivity Info	TI LI LO TS
CP0461030 Compound Info	1-Benzyl-4-(4-methyl-5-phenyl-1H-pyrazol-3-yl)-piperidine Show/Hide	C22H25N3	1
1	Ki = 450 nM Bioactivity Info	TI LI LO TS
CP0435244 Compound Info	1-((1H-indol-3-yl)methyl)-4-(3-chlorophenyl)piperidin-4-ol Show/Hide	C20H21ClN2O	1
1	Ki = 450 nM Bioactivity Info	TI LI LO TS
CP0449016 Compound Info	4-biphenyl-4-yl-1-(1H-indol-3-ylmethyl)-piperidin-4-ol Show/Hide	C26H26N2O	1
1	Ki = 467 nM Bioactivity Info	TI LI LO TS
CP0460212 Compound Info	4-[4-(2,3-dichlorophenyl)piperazin-1-yl]-N-(9H-fluoren-2-ylmethyl)-3-fluorobutan-1-amine Show/Hide	C28H30Cl2FN3	1
1	Ki = 467 nM Bioactivity Info	TI LI LO TS
CP0093802 Compound Info	7-[(1R)-2-[[(1R,2R)-2-(3-ethylphenyl)cyclopentyl]amino]-1-hydroxyethyl]-4-hydroxy-3H-1,3-benzothiazol-2-one Show/Hide	C22H26N2O3S	1
1	Ki = 477 nM Bioactivity Info	TI LI LO TS
CP0081150 Compound Info	4-[3-(4-Chloro-phenyl)-4-methyl-isoxazol-5-yl]-1-phenethyl-piperidine Show/Hide	C23H25ClN2O	1
1	Ki = 480 nM Bioactivity Info	TI LI LO TS
CP0935609 Compound Info	endo-8-(1H-Indol-3-ylmethyl)-3-(2,3-dichlorophenyl)-8-azabicyclo[3.2.1]octan-3-ol Show/Hide	C22H22Cl2N2O	1
1	Ki = 480 nM Bioactivity Info	TI LI LO TS
CP0464096 Compound Info	US10913711, Compound 10d Show/Hide	C22H28F2N2O2S	1
1	Ki = 480 nM Bioactivity Info	TI LI LO TS
CP0372388 Compound Info	4-(4-chlorophenyl)-1-((1-hexyl-1H-indol-3-yl)methyl)piperidin-4-ol Show/Hide	C26H33ClN2O	1
1	Ki = 488 nM Bioactivity Info	TI LI LO TS
CP0449026 Compound Info	1-((1H-indol-3-yl)methyl)-4-(4-fluorophenyl)piperidin-4-ol Show/Hide	C20H21FN2O	1
1	Ki = 490 nM Bioactivity Info	TI LI LO TS
CP0443218 Compound Info	1-[4-(2-methoxyphenyl)piperazin-1-yl]-4-[4-(2-methoxyphenyl)triazol-1-yl]butan-2-ol Show/Hide	C24H31N5O3	1
1	Ki = 493 nM Bioactivity Info	TI LI LO TS
CP0384677 Compound Info	N-(3-ethylphenyl)-2-(4-pyridin-2-ylpiperidin-1-yl)acetamide Show/Hide	C20H25N3O	1
1	Ki = 496 nM Bioactivity Info	TI LI LO TS
CP0517042 Compound Info	4-hydroxy-7-[(1R)-1-hydroxy-2-[[(1R,2R)-2-(4-methylphenyl)cyclopentyl]amino]ethyl]-3H-1,3-benzothiazol-2-one Show/Hide	C21H24N2O3S	1
1	Ki = 502 nM Bioactivity Info	TI LI LO TS
CP0394250 Compound Info	(Z)-1-(1-benzylpiperidin-4-yl)-3-(4-chlorophenyl)-3-hydroxyprop-2-en-1-one Show/Hide	C21H22ClNO2	1
1	Ki = 510 nM Bioactivity Info	TI LI LO TS
CP0454998 Compound Info	(Z)-1-(1-benzyl-4-methylpiperidin-4-yl)-3-(4-chlorophenyl)-3-hydroxyprop-2-en-1-one Show/Hide	C22H24ClNO2	1
1	Ki = 510 nM Bioactivity Info	TI LI LO TS
CP0384679 Compound Info	N-(3-methylphenyl)-3-(4-pyridin-2-ylpiperidin-1-yl)propanamide Show/Hide	C20H25N3O	2
1	Ki = 510 nM Bioactivity Info	TI LI LO TS
2	Ki = 3040 nM Bioactivity Info	TI LI LO TS
CP0115242 Compound Info	4-hydroxy-7-[(1R)-1-hydroxy-2-[[(1R,2R)-2-phenylcyclopentyl]amino]ethyl]-3H-1,3-benzothiazol-2-one Show/Hide	C20H22N2O3S	1
1	Ki = 512 nM Bioactivity Info	TI LI LO TS
CP0245845 Compound Info	4-hydroxy-7-[(1R)-1-hydroxy-2-[[(1R,2R)-2-propan-2-ylcyclopentyl]amino]ethyl]-3H-1,3-benzothiazol-2-one Show/Hide	C17H24N2O3S	1
1	Ki = 512 nM Bioactivity Info	TI LI LO TS
CP0400351 Compound Info	7-Methyl-6,7,8,9,10,15-hexahydroindolo[2,3-f][3]benzazecine Show/Hide	C20H22N2	1
1	Ki = 513 nM Bioactivity Info	TI LI LO TS
CP0425933 Compound Info	N-[4-[4-[2-(trifluoromethyl)quinolin-4-yl]piperazin-1-yl]butyl]imidazo[1,2-a]pyridine-2-carboxamide Show/Hide	C26H27F3N6O	1
1	Ki = 524 nM Bioactivity Info	TI LI LO TS
CP0535381 Compound Info	N-[(3,3-diphenyl-1,4-dioxan-2-yl)methyl]-2-(2-methoxyphenoxy)ethanamine Show/Hide	C26H29NO4	1
1	Ki = 537.03 nM Bioactivity Info	TI LI LO TS
CP0438184 Compound Info	(+/-)-11-((1-(3-(4-Pyrimidinpiperazin-2-yl)propyl)-1H-1,2,3-triazol-4-yl)methoxy)-N-propylnoraporphine Show/Hide	C33H40N8O	1
1	Ki = 539 nM Bioactivity Info	TI LI LO TS
CP0870327 Compound Info	endo-8-(1H-Indol-3-ylmethyl)-3-(4-(methylthio)phenyl)-8-azabicyclo[3.2.1]octan-3-ol Show/Hide	C23H26N2OS	1
1	Ki = 541 nM Bioactivity Info	TI LI LO TS
CP0467821 Compound Info	methyl 4-(4-chlorophenyl)-1-(1H-indol-3-ylmethyl)piperidine-4-carboxylate Show/Hide	C22H23ClN2O2	1
1	Ki = 544 nM Bioactivity Info	TI LI LO TS
CP0178363 Compound Info	(R)-5-Methylamino-5,6-dihydro-1H,4H-imidazo[4,5,1-ij]quinolin-2-one Show/Hide	C11H13N3O	3
1	Ki = 546 nM Bioactivity Info	TI LI LO TS
2	Ki = 573 nM Bioactivity Info	TI LI LO TS
3	Ki = 6330 nM Bioactivity Info	TI LI LO TS
CP0393856 Compound Info	(10R)-10-(methylamino)-3-[2-[2-[2-(4-phenylbutoxy)ethoxy]ethoxy]ethyl]-1,3-diazatricyclo[6.3.1.04,12]dodeca-4,6,8(12)-trien-2-one Show/Hide	C27H37N3O4	1
1	Ki = 558 nM Bioactivity Info	TI LI LO TS
CP0410131 Compound Info	N-[3-[4-(2,3-dichlorophenyl)piperazin-1-yl]-4-fluorobutyl]-1-benzofuran-2-carboxamide Show/Hide	C23H24Cl2FN3O2	1
1	Ki = 560 nM Bioactivity Info	TI LI LO TS
CP0501761 Compound Info	1-((1H-indol-3-yl)methyl)-4-(3-(trifluoromethyl)phenyl)piperidin-4-ol Show/Hide	C21H21F3N2O	1
1	Ki = 570 nM Bioactivity Info	TI LI LO TS
CP0416755 Compound Info	2-[4-[4-(4-bromoanilino)quinazolin-2-yl]piperazin-1-yl]ethanol Show/Hide	C20H22BrN5O	1
1	Ki = 570.88 nM Bioactivity Info	TI LI LO TS
CP0891094 Compound Info	7-(4-(4-(5-Chloro-2-oxo-2,3-dihydro-1H-benzo[d]imidazol-1-yl)piperidin-1-yl)butoxy)-3,4-dihydroquinolin-2(1H)-one oxalate Show/Hide	C27H31ClN4O7	1
1	Ki = 574 nM Bioactivity Info	TI LI LO TS
CP0463313 Compound Info	4-hydroxy-7-[(1R)-1-hydroxy-2-[[(1R,2R)-2-(2-methylphenyl)cyclopentyl]amino]ethyl]-3H-1,3-benzothiazol-2-one Show/Hide	C21H24N2O3S	1
1	Ki = 575 nM Bioactivity Info	TI LI LO TS
CP0409144 Compound Info	1-((5-methoxy-1H-indol-3-yl)methyl)-4-(4-(methylthio)phenyl)piperidin-4-ol Show/Hide	C22H26N2O2S	1
1	Ki = 580 nM Bioactivity Info	TI LI LO TS
CP0396167 Compound Info	3-piperazin-1-ylbenzonitrile Show/Hide	C11H13N3	1
1	Ki = 581 nM Bioactivity Info	TI LI LO TS
CP0379138 Compound Info	1-[3-[4-(3-hydroxypropyl)piperidin-1-yl]propyl]-3,4-dihydroquinolin-2-one Show/Hide	C20H30N2O2	1
1	Ki = 588.84 nM Bioactivity Info	TI LI LO TS
CP0476869 Compound Info	1-(2-methoxyphenyl)-4-methylpiperazine Show/Hide	C12H18N2O	1
1	Ki = 589.9 nM Bioactivity Info	TI LI LO TS
CP0447259 Compound Info	(10R)-10-(methylamino)-3-[12-[(2-oxo-3,4-dihydro-1H-quinolin-7-yl)oxy]dodecyl]-1,3-diazatricyclo[6.3.1.04,12]dodeca-4,6,8(12)-trien-2-one Show/Hide	C32H44N4O3	1
1	Ki = 598 nM Bioactivity Info	TI LI LO TS
CP0380731 Compound Info	1'-phenethyl-3-phenylspiro[2,4,5,6-tetrahydrocyclopenta[c]pyrazole-6,4'-(hexahydropyridine)] Show/Hide	C24H27N3	1
1	Ki = 600 nM Bioactivity Info	TI LI LO TS
CP0438518 Compound Info	N-[4-[[(4aR,10bR)-4-propyl-3,4a,5,10b-tetrahydro-2H-chromeno[4,3-b][1,4]oxazin-9-yl]oxy]butyl]-1H-indole-2-carboxamide Show/Hide	C27H33N3O4	1
1	Ki = 613 nM Bioactivity Info	TI LI LO TS
CP0232092 Compound Info	1-[3-(4-butylpiperidin-1-yl)propyl]-3,4-dihydroquinolin-2-one Show/Hide	C21H32N2O	1
1	Ki = 616.6 nM Bioactivity Info	TI LI LO TS
CP0441597 Compound Info	1-(1-Benzyl-piperidin-4-yl)-4-phenyl-1,3-dihydro-imidazol-2-one Show/Hide	C21H23N3O	1
1	Ki = 630 nM Bioactivity Info	TI LI LO TS
CP0559802 Compound Info	4,4-dimethyl-1-[3-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]propyl]piperidine Show/Hide	C19H28N4S	1
1	Ki = 631 nM Bioactivity Info	TI LI LO TS
CP0467837 Compound Info	1-((1H-indol-3-yl)methyl)-4-(4-(methylthio)phenyl)piperidin-4-ol Show/Hide	C21H24N2OS	1
1	Ki = 638 nM Bioactivity Info	TI LI LO TS
CP0412938 Compound Info	(10R)-10-(methylamino)-3-[2-[2-[2-[2-[(2-oxo-3,4-dihydro-1H-quinolin-7-yl)oxy]ethoxy]ethoxy]ethoxy]ethyl]-1,3-diazatricyclo[6.3.1.04,12]dodeca-4,6,8(12)-trien-2-one Show/Hide	C28H36N4O6	1
1	Ki = 640 nM Bioactivity Info	TI LI LO TS
CP0385310 Compound Info	US10913711, Compound 10j Show/Hide	C28H32F2N2O2S	1
1	Ki = 652 nM Bioactivity Info	TI LI LO TS
CP0378647 Compound Info	1-[3-[4-(5-hydroxypentyl)piperidin-1-yl]propyl]-3,4-dihydroquinolin-2-one Show/Hide	C22H34N2O2	1
1	Ki = 676.08 nM Bioactivity Info	TI LI LO TS
CP0392875 Compound Info	[(12R)-11-methyl-11,21-diazatetracyclo[12.7.0.03,8.015,20]henicosa-1(14),3,5,7,15,17,19-heptaen-12-yl]methanol Show/Hide	C21H24N2O	1
1	Ki = 681 nM Bioactivity Info	TI LI LO TS
CP0421765 Compound Info	1-((1H-indol-3-yl)methyl)-4-(4-chlorophenyl)piperidine-4-carbonitrile Show/Hide	C21H20ClN3	1
1	Ki = 684 nM Bioactivity Info	TI LI LO TS
CP0429530 Compound Info	1-(1-Benzyl-piperidin-4-yl)-3-phenyl-urea Show/Hide	C19H23N3O	1
1	Ki = 700 nM Bioactivity Info	TI LI LO TS
CP0489929 Compound Info	1-[3-(4-phenylpiperidin-1-yl)propyl]-3,4-dihydroquinolin-2-one Show/Hide	C23H28N2O	1
1	Ki = 707.95 nM Bioactivity Info	TI LI LO TS
CP0449025 Compound Info	3-((4-(allyloxy)-4-(4-chlorophenyl)piperidin-1-yl)methyl)-1H-indole Show/Hide	C23H25ClN2O	1
1	Ki = 718 nM Bioactivity Info	TI LI LO TS
CP0374265 Compound Info	4-[5-(4-Chloro-phenyl)-1H-pyrazol-3-yl]-1-cyclohexylmethyl-piperidine Show/Hide	C21H28ClN3	1
1	Ki = 720 nM Bioactivity Info	TI LI LO TS
CP0409198 Compound Info	ethyl 4-(4-chlorophenyl)-1-(1H-indol-3-ylmethyl)piperidine-4-carboxylate Show/Hide	C23H25ClN2O2	1
1	Ki = 724 nM Bioactivity Info	TI LI LO TS
CP0429850 Compound Info	1-Benzyl-4-(4-phenyl-imidazol-1-yl)-piperidine Show/Hide	C21H23N3	1
1	Ki = 740 nM Bioactivity Info	TI LI LO TS
CP0454594 Compound Info	N-[4-[(7-hydroxy-1,2,3,4-tetrahydronaphthalen-2-yl)-[3-(4-phenylpiperazin-1-yl)propyl]amino]butyl]benzamide Show/Hide	C34H44N4O2	1
1	Ki = 756 nM Bioactivity Info	TI LI LO TS
CP0099174 Compound Info	4-[5-(4-Chloro-phenyl)-4-methyl-isoxazol-3-yl]-1-phenethyl-piperidine Show/Hide	C23H25ClN2O	1
1	Ki = 770 nM Bioactivity Info	TI LI LO TS
CP0384372 Compound Info	N-(3-methylphenyl)-3-(4-pyridin-2-ylpiperazin-1-yl)propanamide Show/Hide	C19H24N4O	2
1	Ki = 781 nM Bioactivity Info	TI LI LO TS
2	Ki = 3790 nM Bioactivity Info	TI LI LO TS
CP0891095 Compound Info	7-(4-(4-(2,4-Dimethoxyphenyl)piperazin-1-yl)butoxy)-3,4-dihydroquinolin-2(1H)-one oxalate Show/Hide	C27H35N3O8	1
1	Ki = 785 nM Bioactivity Info	TI LI LO TS
CP0382711 Compound Info	N-[4-[[(4aR,10bR)-4-propyl-3,4a,5,10b-tetrahydro-2H-chromeno[4,3-b][1,4]oxazin-9-yl]oxy]butyl]-9H-fluorene-2-carboxamide Show/Hide	C32H36N2O4	1
1	Ki = 806 nM Bioactivity Info	TI LI LO TS
CP0448976 Compound Info	1-Benzyl-4-(5-phenyl-pyrazol-1-yl)-piperidine Show/Hide	C21H23N3	1
1	Ki = 810 nM Bioactivity Info	TI LI LO TS
CP0183485 Compound Info	1-(4-Chloro-benzyl)-4-[5-(4-chloro-phenyl)-1H-pyrazol-3-yl]-piperidine Show/Hide	C21H21Cl2N3	1
1	Ki = 820 nM Bioactivity Info	TI LI LO TS
CP0437126 Compound Info	1-(3-Chloro-benzyl)-4-(5-methyl-4-phenyl-pyrazol-1-yl)-piperidine Show/Hide	C22H24ClN3	1
1	Ki = 820 nM Bioactivity Info	TI LI LO TS
CP0393905 Compound Info	4-(4-Methyl-5-phenyl-1H-pyrazol-3-yl)-1-phenethyl-1,2,3,6-tetrahydro-pyridine Show/Hide	C23H25N3	1
1	Ki = 830 nM Bioactivity Info	TI LI LO TS
CP0547878 Compound Info	2-(2-methoxyphenyl)-6-[3-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]propyl]-2,6-diazaspiro[3.3]heptane Show/Hide	C24H29N5OS	1
1	Ki = 833 nM Bioactivity Info	TI LI LO TS
CP0258990 Compound Info	7-((R)-2-((cis)-bi(cyclopentan)-2-ylamino)-1-hydroxyethyl)-4-hydroxybenzo[d]thiazol-2(3H)-one Show/Hide	C19H26N2O3S	1
1	Ki = 842 nM Bioactivity Info	TI LI LO TS
CP0904688 Compound Info	4-(4-Bromophenyl)-1-((4-(2-fluoroethoxy)-1H-indol-3-yl)-methyl)piperidin-4-ol oxalate Show/Hide	C24H26BrFN2O6	1
1	Ki = 849 nM Bioactivity Info	TI LI LO TS
CP0453528 Compound Info	4-[5-(4-Chloro-phenyl)-1H-pyrazol-3-yl]-1-(3-phenyl-propyl)-piperidine Show/Hide	C23H26ClN3	1
1	Ki = 870 nM Bioactivity Info	TI LI LO TS
CP0573634 Compound Info	9-[3-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]propyl]-3-pyridin-2-yl-3,9-diazaspiro[5.5]undecane Show/Hide	C26H34N6S	1
1	Ki = 871 nM Bioactivity Info	TI LI LO TS
CP0887641 Compound Info	7-(4-(4-(2-Oxo-2,3-dihydro-1H-benzo[d]imidazol-1-yl)-piperidin-1-yl)butoxy)-3,4-dihydroquinolin-2(1H)-one oxalate Show/Hide	C27H32N4O7	1
1	Ki = 879 nM Bioactivity Info	TI LI LO TS
CP0480949 Compound Info	(11S)-N-[(1R)-1-(4-bromophenyl)ethyl]-5-ethyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide Show/Hide	C24H21BrN2O3S	1
1	Ki = 880 nM Bioactivity Info	TI LI LO TS
CP0187238 Compound Info	7-((R)-2-((1S,2S)-2-(benzyloxy)cyclopentylamino)-1-hydroxyethyl)-4-hydroxybenzo[d]thiazol-2(3H)-one Show/Hide	C21H24N2O4S	1
1	Ki = 895 nM Bioactivity Info	TI LI LO TS
CP0374292 Compound Info	3-(1-Benzyl-pyrrolidin-3-yl)-5-(4-chloro-phenyl)-1H-pyrazole Show/Hide	C20H20ClN3	1
1	Ki = 920 nM Bioactivity Info	TI LI LO TS
CP0373007 Compound Info	1-(1-Benzyl-piperidin-4-yl)-4-(4-fluoro-phenyl)-5-methyl-1,3-dihydro-imidazol-2-one Show/Hide	C22H24FN3O	1
1	Ki = 930 nM Bioactivity Info	TI LI LO TS
CP0891097 Compound Info	7-(4-(4-(4-Methoxyphenyl)piperazin-1-yl)butoxy)-3,4-dihydroquinolin-2(1H)-one oxalate Show/Hide	C26H33N3O7	1
1	Ki = 930 nM Bioactivity Info	TI LI LO TS
CP0379189 Compound Info	2-(1-Benzenesulfonyl-1H-indol-4-yl)-ethylamine Show/Hide	C16H16N2O2S	1
1	Ki = 940 nM Bioactivity Info	TI LI LO TS
CP0378380 Compound Info	1-(1-Benzyl-piperidin-4-yl)-3-pyridin-2-yl-urea Show/Hide	C18H22N4O	1
1	Ki = 950 nM Bioactivity Info	TI LI LO TS
CP0393625 Compound Info	1-[3-[4-(7-hydroxyheptyl)piperidin-1-yl]propyl]-3,4-dihydroquinolin-2-one Show/Hide	C24H38N2O2	1
1	Ki = 954.99 nM Bioactivity Info	TI LI LO TS
CP0396212 Compound Info	N-[[(1R,2R)-2-[(6-cyano-3,4-dihydro-1H-isoquinolin-2-yl)methyl]cyclopropyl]methyl]quinoline-4-carboxamide Show/Hide	C25H24N4O	1
1	Ki = 1040 nM Bioactivity Info	TI LI LO TS
CP0159295 Compound Info	8-Hydroxy-5-[(R)-1-hydroxy-2-(5,6-diethylindan-2-ylamino)-ethyl]-1H-quinolin-2-one Show/Hide	C24H28N2O3	1
1	Ki = 1048 nM Bioactivity Info	TI LI LO TS
CP0065062 Compound Info	1-hydroxy-2-naphthoic acid;4-[1-hydroxy-2-[6-(4-phenylbutoxy)hexylamino]ethyl]-2-methylol-phenol Show/Hide	C25H37NO4	1
1	Ki = 1049 nM Bioactivity Info	TI LI LO TS
CP0396211 Compound Info	2-butyl-3,4-dihydro-1H-isoquinoline-6-carbonitrile Show/Hide	C14H18N2	1
1	Ki = 1090 nM Bioactivity Info	TI LI LO TS
CP0562951 Compound Info	1-[3-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]propyl]piperidine Show/Hide	C17H24N4S	1
1	Ki = 1098 nM Bioactivity Info	TI LI LO TS
CP0430826 Compound Info	1-Phenethyl-4-(5-thiophen-2-yl-1H-pyrazol-3-yl)-piperidine Show/Hide	C20H23N3S	1
1	Ki = 1100 nM Bioactivity Info	TI LI LO TS
CP0453196 Compound Info	4-(4-Chloro-phenyl)-5-methyl-6-(1-phenethyl-piperidin-4-yl)-pyrimidin-2-ylamine Show/Hide	C24H27ClN4	1
1	Ki = 1100 nM Bioactivity Info	TI LI LO TS
CP0460142 Compound Info	1-(1-Cyclohexylmethyl-piperidin-4-yl)-5-methyl-4-phenyl-1,3-dihydro-imidazol-2-one Show/Hide	C22H31N3O	1
1	Ki = 1100 nM Bioactivity Info	TI LI LO TS
CP0093810 Compound Info	7-[(1R)-2-[[(1R,2R)-2-cyclohexylcyclopentyl]amino]-1-hydroxyethyl]-4-hydroxy-3H-1,3-benzothiazol-2-one Show/Hide	C20H28N2O3S	1
1	Ki = 1100 nM Bioactivity Info	TI LI LO TS
CP0416761 Compound Info	2-[4-[4-(4-propan-2-ylanilino)quinazolin-2-yl]piperazin-1-yl]ethanol Show/Hide	C23H29N5O	1
1	Ki = 1140.65 nM Bioactivity Info	TI LI LO TS
CP0459850 Compound Info	7-[(1R)-2-[[(1S,2R)-2-cyclopentylcyclopentyl]amino]-1-hydroxyethyl]-4-hydroxy-3H-1,3-benzothiazol-2-one Show/Hide	C19H26N2O3S	1
1	Ki = 1141 nM Bioactivity Info	TI LI LO TS
CP0416959 Compound Info	3-[3-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]propyl]-3,9-diazaspiro[5.5]undecane Show/Hide	C21H31N5S	1
1	Ki = 1145 nM Bioactivity Info	TI LI LO TS
CP0438516 Compound Info	7-[(E)-4-[(2S,5S)-2-(6-aminopyridin-3-yl)-5-methylmorpholin-4-yl]but-2-enoxy]-3,4-dihydro-1H-quinolin-2-one Show/Hide	C23H28N4O3	1
1	Ki = 1150 nM Bioactivity Info	TI LI LO TS
CP0535796 Compound Info	N-[1-[(3,4-difluorophenyl)methyl]piperidin-4-yl]-6-(trifluoromethyl)pyridazin-3-amine Show/Hide	C17H17F5N4	1
1	Ki = 1159 nM Bioactivity Info	TI LI LO TS
CP0382704 Compound Info	2-[4-[[(4aR,10bR)-4-propyl-3,4a,5,10b-tetrahydro-2H-chromeno[4,3-b][1,4]oxazin-9-yl]oxy]butyl]isoindole-1,3-dione Show/Hide	C26H30N2O5	1
1	Ki = 1190 nM Bioactivity Info	TI LI LO TS
CP0372647 Compound Info	4-[5-(4-Chloro-phenyl)-4-methyl-1H-pyrazol-3-yl]-1-phenethyl-piperidine Show/Hide	C23H26ClN3	1
1	Ki = 1200 nM Bioactivity Info	TI LI LO TS
CP0419180 Compound Info	1-Phenethyl-4-(5-phenyl-1H-pyrazol-3-yl)-piperazine Show/Hide	C21H24N4	1
1	Ki = 1200 nM Bioactivity Info	TI LI LO TS
CP0487032 Compound Info	4-(5-Cyclohexyl-1H-pyrazol-3-yl)-1-phenethyl-piperidine Show/Hide	C22H31N3	1
1	Ki = 1200 nM Bioactivity Info	TI LI LO TS
CP0406711 Compound Info	1-(1-Benzyl-piperidin-4-yl)-5-methyl-4-pyridin-2-yl-1,3-dihydro-imidazol-2-one Show/Hide	C21H24N4O	1
1	Ki = 1200 nM Bioactivity Info	TI LI LO TS
CP0919167 Compound Info	endo-8-(5-Methoxy-1H-indol-3-ylmethyl)-3-(4-methylthiophenyl)-8-azabicyclo[3.2.1]octan-3-ol Show/Hide	C24H28N2O2S	1
1	Ki = 1210 nM Bioactivity Info	TI LI LO TS
CP0384375 Compound Info	N-(3-methylphenyl)-2-(4-naphthalen-1-ylpiperazin-1-yl)acetamide Show/Hide	C23H25N3O	2
1	Ki = 1246 nM Bioactivity Info	TI LI LO TS
2	Ki = 11459 nM Bioactivity Info	TI LI LO TS
CP0420812 Compound Info	1-Benzyl-4-[5-(4-chloro-phenyl)-1H-pyrazol-3-yl]-4-methyl-piperidine Show/Hide	C22H24ClN3	1
1	Ki = 1300 nM Bioactivity Info	TI LI LO TS
CP0432438 Compound Info	1-(2-Chloro-benzyl)-4-[5-(4-chloro-phenyl)-1H-pyrazol-3-yl]-piperidine Show/Hide	C21H21Cl2N3	1
1	Ki = 1300 nM Bioactivity Info	TI LI LO TS
CP0492208 Compound Info	1-Benzyl-4-(4-phenyl-[1,2,3]triazol-1-yl)-piperidine Show/Hide	C20H22N4	1
1	Ki = 1300 nM Bioactivity Info	TI LI LO TS
CP0429032 Compound Info	[(1S,2R,5R,6R,7R)-3-benzyl-7-(diethylamino)-2-phenyl-3-azabicyclo[3.2.0]heptan-6-yl]methanol Show/Hide	C24H32N2O	1
1	Ki = 1300 nM Bioactivity Info	TI LI LO TS
CP0232093 Compound Info	1-[3-(4-phenylpiperazin-1-yl)propyl]-3,4-dihydroquinolin-2-one Show/Hide	C22H27N3O	1
1	Ki = 1318.26 nM Bioactivity Info	TI LI LO TS
CP0519118 Compound Info	N-[4-[[(4aR,10bR)-4-propyl-3,4a,5,10b-tetrahydro-2H-chromeno[4,3-b][1,4]oxazin-9-yl]oxy]butyl]-1,3-benzothiazole-2-carboxamide Show/Hide	C26H31N3O4S	1
1	Ki = 1330 nM Bioactivity Info	TI LI LO TS
CP0432721 Compound Info	(10R)-10-(methylamino)-3-[4-[(2-oxo-3,4-dihydro-1H-quinolin-7-yl)oxy]butyl]-1,3-diazatricyclo[6.3.1.04,12]dodeca-4,6,8(12)-trien-2-one Show/Hide	C24H28N4O3	1
1	Ki = 1350 nM Bioactivity Info	TI LI LO TS
CP0375428 Compound Info	1-Benzyl-4-(5-phenyl-1H-pyrazol-3-yl)-piperidine Show/Hide	C21H23N3	1
1	Ki = 1400 nM Bioactivity Info	TI LI LO TS
CP0436445 Compound Info	1-Benzyl-4-(5-phenyl-tetrazol-2-yl)-piperidine Show/Hide	C19H21N5	1
1	Ki = 1400 nM Bioactivity Info	TI LI LO TS
CP0416758 Compound Info	2-[4-[4-(benzylamino)quinazolin-2-yl]piperazin-1-yl]ethanol Show/Hide	C21H25N5O	1
1	Ki = 1435.7 nM Bioactivity Info	TI LI LO TS
CP0384370 Compound Info	N-(3-ethylphenyl)-2-(4-pyridin-2-ylpiperazin-1-yl)acetamide Show/Hide	C19H24N4O	2
1	Ki = 1490 nM Bioactivity Info	TI LI LO TS
2	Ki > 50000 nM Bioactivity Info	TI LI LO TS
CP0509754 Compound Info	[(1S,2R,5R,6R,7R)-3-benzyl-2-phenyl-7-piperidin-1-yl-3-azabicyclo[3.2.0]heptan-6-yl]methanol Show/Hide	C25H32N2O	1
1	Ki = 1500 nM Bioactivity Info	TI LI LO TS
CP0043573 Compound Info	1,2,3,4-Tetrahydro-isoquinoline-7-carbonitrile Show/Hide	C10H10N2	1
1	Ki = 1520 nM Bioactivity Info	TI LI LO TS
CP0382705 Compound Info	5-[(2R,5S)-5-methylmorpholin-2-yl]pyridin-2-amine Show/Hide	C10H15N3O	1
1	Ki = 1520 nM Bioactivity Info	TI LI LO TS
CP0891093 Compound Info	7-(4-(4-(4-Chlorophenyl)-4-hydroxypiperidin-1-yl)butoxy)-3,4-dihydroquinolin-2(1H)-one oxalate Show/Hide	C26H31ClN2O7	1
1	Ki = 1536 nM Bioactivity Info	TI LI LO TS
CP0393633 Compound Info	1-[3-(4-propylpiperidin-1-yl)propyl]-3,4-dihydroquinolin-2-one Show/Hide	C20H30N2O	1
1	Ki = 1548.82 nM Bioactivity Info	TI LI LO TS
CP0861002 Compound Info	1-((1H-Pyrrolo[2,3-b]pyridine-3-yl)methyl)-4-(4-iodophenyl)piperidin-4-ol oxalate Show/Hide	C21H22IN3O5	1
1	Ki = 1585 nM Bioactivity Info	TI LI LO TS
CP0471921 Compound Info	7-[4-[[(4aR,10bR)-4-propyl-3,4a,5,10b-tetrahydro-2H-chromeno[4,3-b][1,4]oxazin-9-yl]oxy]butoxy]-3,4-dihydro-1H-quinolin-2-one Show/Hide	C27H34N2O5	1
1	Ki = 1590 nM Bioactivity Info	TI LI LO TS
CP0066323 Compound Info	CAS_73573-87-2 Show/Hide	C19H24N2O4	1
1	Ki = 1626 nM Bioactivity Info	TI LI LO TS
CP0458244 Compound Info	[(1R,2S,5R,6R,7R)-3-benzyl-7-(diethylamino)-2-methyl-3-azabicyclo[3.2.0]heptan-6-yl]methanol Show/Hide	C19H30N2O	1
1	Ki = 1770 nM Bioactivity Info	TI LI LO TS
CP0449653 Compound Info	1-Benzyl-2-[5-(4-chloro-phenyl)-1H-pyrazol-3-yl]-piperidine Show/Hide	C21H22ClN3	1
1	Ki = 1800 nM Bioactivity Info	TI LI LO TS
CP0116478 Compound Info	1-[3-(4-benzylpiperidin-1-yl)propyl]-3,4-dihydroquinolin-2-one Show/Hide	C24H30N2O	1
1	Ki = 1819.7 nM Bioactivity Info	TI LI LO TS
CP0449014 Compound Info	1-((1H-indol-3-yl)methyl)-4-(2-chlorophenyl)piperidin-4-ol Show/Hide	C20H21ClN2O	1
1	Ki = 1860 nM Bioactivity Info	TI LI LO TS
CP0448388 Compound Info	5-Methyl-4-phenyl-1-[1-(3-phenyl-propyl)-piperidin-4-yl]-1,3-dihydro-imidazol-2-one Show/Hide	C24H29N3O	1
1	Ki = 1900 nM Bioactivity Info	TI LI LO TS
CP0377527 Compound Info	5-ethyl-6,11-diketo-N-p-anisyl-benzo[b][1,4]benzothiazepine-3-carboxamide Show/Hide	C24H22N2O4S	1
1	Ki = 1900 nM Bioactivity Info	TI LI LO TS
CP0449021 Compound Info	1-((1H-indol-3-yl)methyl)-4-(4-(hexyloxy)phenyl)piperidin-4-ol Show/Hide	C26H34N2O2	1
1	Ki = 1950 nM Bioactivity Info	TI LI LO TS
CP0035276 Compound Info	1-(4-fluorophenyl)-4-(4-hydroxy-5-azahexacyclo[5.4.1.02,6.03,10.04,8.09,12]dodecan-5-yl)butan-1-one Show/Hide	C21H22FNO2	1
1	Ki = 1958 nM Bioactivity Info	TI LI LO TS
CP0416338 Compound Info	1-(1-Benzyl-piperidin-4-yl)-3-isoquinolin-1-yl-urea Show/Hide	C22H24N4O	1
1	Ki = 2000 nM Bioactivity Info	TI LI LO TS
CP0400254 Compound Info	N-[4-[4-[2-methyl-6-(trifluoromethyl)pyrimidin-4-yl]piperazin-1-yl]butyl]imidazo[1,2-a]pyridine-2-carboxamide Show/Hide	C22H26F3N7O	1
1	Ki = 2014 nM Bioactivity Info	TI LI LO TS
CP0439296 Compound Info	1-Benzyl-4-(5-benzyl-1H-pyrazol-3-yl)-piperidine Show/Hide	C22H25N3	1
1	Ki = 2100 nM Bioactivity Info	TI LI LO TS
CP0445423 Compound Info	3-((4-(4-chlorophenyl)-4-methylpiperidin-1-yl)methyl)-1H-indole Show/Hide	C21H23ClN2	1
1	Ki = 2100 nM Bioactivity Info	TI LI LO TS
CP0467819 Compound Info	1-((1H-indol-3-yl)methyl)-4-(4-chlorophenyl)azepan-4-ol Show/Hide	C21H23ClN2O	1
1	Ki = 2100 nM Bioactivity Info	TI LI LO TS
CP0449017 Compound Info	1-((1H-indol-3-yl)methyl)-4-(4-methoxyphenyl)piperidin-4-ol Show/Hide	C21H24N2O2	1
1	Ki = 2130 nM Bioactivity Info	TI LI LO TS
CP0382714 Compound Info	N-[4-[[(4aR,10bR)-4-propyl-3,4a,5,10b-tetrahydro-2H-chromeno[4,3-b][1,4]oxazin-9-yl]oxy]butyl]-1,3-benzothiazole-5-carboxamide Show/Hide	C26H31N3O4S	1
1	Ki = 2130 nM Bioactivity Info	TI LI LO TS
CP0502925 Compound Info	[(1S,2R,5R,6R,7R)-3-benzyl-2-(4-bromophenyl)-7-(diethylamino)-3-azabicyclo[3.2.0]heptan-6-yl]methanol Show/Hide	C24H31BrN2O	1
1	Ki = 2140 nM Bioactivity Info	TI LI LO TS
CP0432236 Compound Info	1-Benzyl-4-(4-methyl-5-phenyl-[1,2,3]triazol-1-yl)-piperidine Show/Hide	C21H24N4	1
1	Ki = 2200 nM Bioactivity Info	TI LI LO TS
CP0046762 Compound Info	(N-(o-methoxyphenyl)piperazine)1-(2-Methoxy-phenyl)-piperazine Show/Hide	C11H16N2O	1
1	Ki = 2262 nM Bioactivity Info	TI LI LO TS
CP0519090 Compound Info	N-[4-[4-(4-cyanophenyl)piperazin-1-yl]butyl]-4-thiophen-3-ylbenzamide Show/Hide	C26H28N4OS	1
1	Ki = 2378 nM Bioactivity Info	TI LI LO TS
CP0847583 Compound Info	(+/-)-11-prop-2-ynyloxy N-propylnoraporphine Show/Hide	C22H23NO	1
1	Ki = 2400 nM Bioactivity Info	TI LI LO TS
CP0495061 Compound Info	1-Benzyl-4-(5-methyl-4-phenyl-[1,2,3]triazol-1-yl)-piperidine Show/Hide	C21H24N4	1
1	Ki = 2500 nM Bioactivity Info	TI LI LO TS
CP0472845 Compound Info	1-[3-(4-benzylpiperazin-1-yl)propyl]-3,4-dihydroquinolin-2-one Show/Hide	C23H29N3O	1
1	Ki = 2630.27 nM Bioactivity Info	TI LI LO TS
CP0541816 Compound Info	9-butyl-3-(2-methoxyphenyl)-3,9-diazaspiro[5.5]undecane Show/Hide	C20H32N2O	1
1	Ki = 2773 nM Bioactivity Info	TI LI LO TS
CP0426667 Compound Info	1-[[(2R)-3,3-diphenyl-1,4-dioxan-2-yl]methyl]-4-(2-methoxyphenyl)piperazine Show/Hide	C28H32N2O3	1
1	Ki = 2884.03 nM Bioactivity Info	TI LI LO TS
CP0919396 Compound Info	1-((5-Methoxy-1H-indol-3-yl)methyl)-4-phenylpiperidin-4-ol oxalate Show/Hide	C23H26N2O6	1
1	Ki = 2927 nM Bioactivity Info	TI LI LO TS
CP0919397 Compound Info	1-((1H-Pyrrolo[2,3-b]pyridine-3-yl)methyl)-4-(4-bromophenyl)piperidin-4-ol oxalate Show/Hide	C21H22BrN3O5	1
1	Ki = 2983 nM Bioactivity Info	TI LI LO TS
CP0509616 Compound Info	1-Benzyl-4-(3-methyl-5-phenyl-pyrazol-1-yl)-piperidine Show/Hide	C22H25N3	1
1	Ki = 3000 nM Bioactivity Info	TI LI LO TS
CP0401190 Compound Info	(10R)-10-amino-1,3-diazatricyclo[6.3.1.04,12]dodeca-4,6,8(12)-trien-2-one Show/Hide	C10H11N3O	2
1	Ki = 3390 nM Bioactivity Info	TI LI LO TS
2	Ki = 11800 nM Bioactivity Info	TI LI LO TS
CP0441507 Compound Info	1-Benzyl-4-(5-methyl-1H-pyrazol-3-yl)-piperidine Show/Hide	C16H21N3	1
1	Ki = 3400 nM Bioactivity Info	TI LI LO TS
CP0380862 Compound Info	(11S)-5-ethyl-N-[(1R)-1-naphthalen-2-ylethyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide Show/Hide	C28H24N2O3S	1
1	Ki = 3400 nM Bioactivity Info	TI LI LO TS
CP0424550 Compound Info	2-[5-(1-Phenethyl-piperidin-4-yl)-2H-pyrazol-3-yl]-pyridine Show/Hide	C21H24N4	1
1	Ki = 3600 nM Bioactivity Info	TI LI LO TS
CP0404224 Compound Info	1-(1-Benzyl-piperidin-4-yl)-4-methyl-5-phenyl-1,3-dihydro-imidazol-2-one Show/Hide	C22H25N3O	1
1	Ki = 3600 nM Bioactivity Info	TI LI LO TS
CP0384675 Compound Info	N-(3-methylphenyl)-2-[4-(4-methylphenyl)piperidin-1-yl]acetamide Show/Hide	C21H26N2O	1
1	Ki = 3681 nM Bioactivity Info	TI LI LO TS
CP0186950 Compound Info	(4S,5S)-4-Dimethylamino-1-(toluene-4-sulfonyl)-1,3,4,5-tetrahydro-benzo[cd]indol-5-ol Show/Hide	C20H22N2O3S	1
1	Ki = 3700 nM Bioactivity Info	TI LI LO TS
CP0393627 Compound Info	1-[3-(4-methylpiperidin-1-yl)propyl]-3,4-dihydroquinolin-2-one Show/Hide	C18H26N2O	1
1	Ki = 3715.35 nM Bioactivity Info	TI LI LO TS
CP0055980 Compound Info	N-[2-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl]-2-methoxy-5-methylbenzamide Show/Hide	C22H28N2O4	1
1	Ki = 3760 nM Bioactivity Info	TI LI LO TS
CP0411642 Compound Info	1-[3-(4-butylpiperazin-1-yl)propyl]-3,4-dihydroquinolin-2-one Show/Hide	C20H31N3O	1
1	Ki = 3890.45 nM Bioactivity Info	TI LI LO TS
CP0393626 Compound Info	1-[3-[4-(2-phenylethyl)piperazin-1-yl]propyl]-3,4-dihydroquinolin-2-one Show/Hide	C24H31N3O	1
1	Ki = 3981.07 nM Bioactivity Info	TI LI LO TS
CP0382131 Compound Info	(11S)-5-methyl-6,11-dioxo-N-(2-thiophen-2-ylethyl)benzo[b][1,4]benzothiazepine-3-carboxamide Show/Hide	C21H18N2O3S2	1
1	Ki = 4100 nM Bioactivity Info	TI LI LO TS
CP0372387 Compound Info	1-((1H-indol-3-yl)methyl)-3-(4-chlorophenyl)piperidin-3-ol Show/Hide	C20H21ClN2O	1
1	Ki = 4270 nM Bioactivity Info	TI LI LO TS
CP0377724 Compound Info	1-(3-Chloro-benzyl)-4-[5-(4-chloro-phenyl)-1H-pyrazol-3-yl]-piperidine Show/Hide	C21H21Cl2N3	1
1	Ki = 4300 nM Bioactivity Info	TI LI LO TS
CP0409440 Compound Info	3-[4-(5-Methyl-4-phenyl-pyrazol-1-yl)-piperidin-1-ylmethyl]-benzonitrile Show/Hide	C23H24N4	1
1	Ki = 4400 nM Bioactivity Info	TI LI LO TS
CP0395779 Compound Info	(+/-)-3-(3-(N-propylnoraporphin-11-yloxy)propylamino)propan-1-ol Show/Hide	C25H34N2O2	1
1	Ki = 4514 nM Bioactivity Info	TI LI LO TS
CP0384371 Compound Info	N-(3-methylphenyl)-3-(4-pyrimidin-2-ylpiperazin-1-yl)propanamide Show/Hide	C18H23N5O	2
1	Ki = 4530 nM Bioactivity Info	TI LI LO TS
2	Ki = 9350 nM Bioactivity Info	TI LI LO TS
CP0431323 Compound Info	[(12S)-11-methyl-11,21-diazatetracyclo[12.7.0.03,8.015,20]henicosa-1(14),3,5,7,15,17,19-heptaen-12-yl]methanol Show/Hide	C21H24N2O	1
1	Ki = 4676 nM Bioactivity Info	TI LI LO TS
CP0566758 Compound Info	1-(2-methoxyphenyl)-6-[3-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]propyl]-1,6-diazaspiro[3.3]heptane Show/Hide	C24H29N5OS	1
1	Ki = 4790 nM Bioactivity Info	TI LI LO TS
CP0919407 Compound Info	1-((1H-Pyrrolo[2,3-b]pyridine-3-yl)methyl)-4-(4-(methylthio)phenyl)piperidin-4-ol oxalate Show/Hide	C22H25N3O5S	1
1	Ki = 4938 nM Bioactivity Info	TI LI LO TS
CP0423854 Compound Info	[(1R,2S,5S,6S,7S)-3-benzyl-2-phenyl-7-piperidin-1-yl-3-azabicyclo[3.2.0]heptan-6-yl]methanol Show/Hide	C25H32N2O	1
1	Ki = 5300 nM Bioactivity Info	TI LI LO TS
CP0372344 Compound Info	1-((1H-indol-3-yl)methyl)-4-(4-chlorobenzyl)piperidin-4-ol Show/Hide	C21H23ClN2O	1
1	Ki = 5480 nM Bioactivity Info	TI LI LO TS
CP0922740 Compound Info	N-(4-((4aS,10bS)-9-hydroxy-2,3,4a,5-tetrahydrochromeno[4,3-b][1,4]oxazin-4(10bH)-yl)butyl)-1H-indole-2-carboxamide Show/Hide	C24H27N3O4	1
1	Ki = 5540 nM Bioactivity Info	TI LI LO TS
CP0405332 Compound Info	(-)-1-Propyl-2,3,10,10a-tetrahydro-1H,4aH-4,9-dioxa-1-aza-phenanthren-6-ol Show/Hide	C14H19NO3	1
1	Ki = 5620 nM Bioactivity Info	TI LI LO TS
CP0396205 Compound Info	1,2,3,4-tetrahydroisoquinoline-6-carbonitrile Show/Hide	C10H10N2	1
1	Ki = 5890 nM Bioactivity Info	TI LI LO TS
CP0384667 Compound Info	N-(3-methylphenyl)-2-(4-pyrimidin-2-ylpiperazin-1-yl)acetamide Show/Hide	C17H21N5O	2
1	Ki = 5990 nM Bioactivity Info	TI LI LO TS
2	Ki > 10000 nM Bioactivity Info	TI LI LO TS
CP0438519 Compound Info	N-[4-[[(4aR,10bR)-4-propyl-3,4a,5,10b-tetrahydro-2H-chromeno[4,3-b][1,4]oxazin-9-yl]oxy]butyl]-1-benzofuran-2-carboxamide Show/Hide	C27H32N2O5	1
1	Ki = 6010 nM Bioactivity Info	TI LI LO TS
CP0908362 Compound Info	endo-8-(1H-Indol-3-ylmethyl)-3-(2-methoxyphenyl)-8-azabicyclo[3.2.1]octan-3-ol Show/Hide	C23H26N2O2	1
1	Ki = 6410 nM Bioactivity Info	TI LI LO TS
CP0382707 Compound Info	N-[4-[(2R,5S)-2-(6-aminopyridin-3-yl)-5-methylmorpholin-4-yl]butyl]-1H-indole-2-carboxamide Show/Hide	C23H29N5O2	1
1	Ki = 6470 nM Bioactivity Info	TI LI LO TS
CP0384672 Compound Info	N-(3-methylphenyl)-2-(4-pyridin-2-ylpiperazin-1-yl)acetamide Show/Hide	C18H22N4O	2
1	Ki = 6480 nM Bioactivity Info	TI LI LO TS
2	Ki > 10000 nM Bioactivity Info	TI LI LO TS
CP0535809 Compound Info	8-butyl-2-(2-methoxyphenyl)-2,8-diazaspiro[4.5]decane Show/Hide	C19H30N2O	1
1	Ki = 6647 nM Bioactivity Info	TI LI LO TS
CP0409126 Compound Info	[(1R,2S,5S,6S,7S)-3-benzyl-2-(4-bromophenyl)-7-(diethylamino)-3-azabicyclo[3.2.0]heptan-6-yl]methanol Show/Hide	C24H31BrN2O	1
1	Ki = 7930 nM Bioactivity Info	TI LI LO TS
CP0462359 Compound Info	N-[4-[[(4aR,10bR)-4-propyl-3,4a,5,10b-tetrahydro-2H-chromeno[4,3-b][1,4]oxazin-9-yl]oxy]butyl]-1H-pyrrolo[2,3-b]pyridine-2-carboxamide Show/Hide	C26H32N4O4	1
1	Ki = 8660 nM Bioactivity Info	TI LI LO TS
CP0423855 Compound Info	[(1S,2R,5R,6R,7R)-3-benzyl-7-(diethylamino)-2-pyridin-2-yl-3-azabicyclo[3.2.0]heptan-6-yl]methanol Show/Hide	C23H31N3O	1
1	Ki = 8800 nM Bioactivity Info	TI LI LO TS
CP0490048 Compound Info	5-methyl-6,11-dioxo-N-(2-thiophen-2-ylethyl)benzo[b][1,4]benzothiazepine-3-carboxamide Show/Hide	C21H18N2O3S2	1
1	Ki = 9200 nM Bioactivity Info	TI LI LO TS
CP0373716 Compound Info	5-Methyl-4,5,6,7-tetrahydroindolo[4,3a,3-ef][3]benzazecine Show/Hide	C19H20N2	1
1	Ki > 10000 nM Bioactivity Info	TI LI LO TS
CP0400347 Compound Info	2,6,7,9,10,14b-Hexahydroindolo[3',4':3,4,5]azepino[2,1-a]-isoquinoline Show/Hide	C19H18N2	1
1	Ki > 10000 nM Bioactivity Info	TI LI LO TS
CP0401522 Compound Info	5,6,8,9,10,14c-Hexahydroindolo[3',2':3,4,]pyrido[2,1-a]isoquinoline Show/Hide	C19H18N2	1
1	Ki > 10000 nM Bioactivity Info	TI LI LO TS
CP0429881 Compound Info	2,8,9,13b-Tetrahydro-6H-isoquino[2,1-b]pyrrolo[4,3,2-de]-isoquinoline Show/Hide	C18H16N2	1
1	Ki > 10000 nM Bioactivity Info	TI LI LO TS
CP0057703 Compound Info	N-[2-(4-hydroxy-5-azahexacyclo[5.4.1.02,6.03,10.04,8.09,12]dodecan-5-yl)ethyl]-2-methoxy-5-methylbenzamide Show/Hide	C22H26N2O3	1
1	Ki > 10000 nM Bioactivity Info	TI LI LO TS
CP0392876 Compound Info	(12R)-11,12-dimethyl-11,21-diazatetracyclo[12.7.0.03,8.015,20]henicosa-1(14),3,5,7,15,17,19-heptaene Show/Hide	C21H24N2	1
1	Ki > 10000 nM Bioactivity Info	TI LI LO TS
CP0392877 Compound Info	11-methyl-11,21-diazatetracyclo[12.7.0.03,8.015,20]henicosa-1(14),3,5,7,15,17,19-heptaene-12-carboxylic acid Show/Hide	C21H22N2O2	1
1	Ki > 10000 nM Bioactivity Info	TI LI LO TS
CP0002070 Compound Info	1-(1H-Indol-3-yl)-2-propanamine Show/Hide	C11H14N2	1
1	Ki > 10000 nM Bioactivity Info	TI LI LO TS
CP0384376 Compound Info	N-(3-methylphenyl)-2-[4-(5-methylpyridin-2-yl)piperidin-1-yl]acetamide Show/Hide	C20H25N3O	2
1	Ki > 10000 nM Bioactivity Info	TI LI LO TS
2	Ki > 50000 nM Bioactivity Info	TI LI LO TS
CP0416633 Compound Info	2-[4-(5-chloropyridin-2-yl)piperazin-1-yl]-N-(3-methylphenyl)acetamide Show/Hide	C18H21ClN4O	2
1	Ki > 10000 nM Bioactivity Info	TI LI LO TS
2	Ki > 50000 nM Bioactivity Info	TI LI LO TS
CP0458243 Compound Info	[(1R,2S,5R,6R,7R)-3-benzyl-2-methyl-7-pyrrolidin-1-yl-3-azabicyclo[3.2.0]heptan-6-yl]methanol Show/Hide	C19H28N2O	1
1	Ki = 11000 nM Bioactivity Info	TI LI LO TS
CP0470560 Compound Info	[(1R,2S,5S,6S,7S)-3-benzyl-2-phenyl-7-pyrrolidin-1-yl-3-azabicyclo[3.2.0]heptan-6-yl]methanol Show/Hide	C24H30N2O	1
1	Ki = 11000 nM Bioactivity Info	TI LI LO TS
CP0382712 Compound Info	7-[4-[(4aR,10bR)-9-hydroxy-3,4a,5,10b-tetrahydro-2H-chromeno[4,3-b][1,4]oxazin-4-yl]butoxy]-3,4-dihydro-1H-quinolin-2-one Show/Hide	C24H28N2O5	1
1	Ki = 11300 nM Bioactivity Info	TI LI LO TS
CP0449020 Compound Info	N-[[4-(4-chlorophenyl)-1-(1H-indol-3-ylmethyl)piperidin-4-yl]methyl]acetamide Show/Hide	C23H26ClN3O	1
1	Ki = 12500 nM Bioactivity Info	TI LI LO TS
CP0475616 Compound Info	[(1R,2S,5S,6S,7S)-3-benzyl-7-(diethylamino)-2-phenyl-3-azabicyclo[3.2.0]heptan-6-yl]methanol Show/Hide	C24H32N2O	1
1	Ki = 13200 nM Bioactivity Info	TI LI LO TS
CP0946433 Compound Info	N-(4-((4aS,10bR)-9-hydroxy-2,3,4a,5-tetrahydrochromeno[4,3-b][1,4]oxazin-4(10bH)-yl)butyl)-1H-indole-2-carboxamide Show/Hide	C24H27N3O4	1
1	Ki = 13800 nM Bioactivity Info	TI LI LO TS
CP0548208 Compound Info	7-[3-[3-(2-methoxyphenyl)-3,9-diazaspiro[5.5]undecan-9-yl]propoxy]-3,4-dihydro-1H-quinolin-2-one Show/Hide	C28H37N3O3	1
1	Ki = 14587 nM Bioactivity Info	TI LI LO TS
CP0296558 Compound Info	[1-[(3S,4S)-1-[(4-fluorophenyl)methyl]-3-hydroxypiperidin-4-yl]piperidin-4-yl]-(4-methoxyphenyl)methanone Show/Hide	C25H31FN2O3	1
1	Ki > 15000 nM Bioactivity Info	TI LI LO TS
CP0464320 Compound Info	1-((1H-indol-3-yl)methyl)-4-(4-hydroxyphenyl)piperidin-4-ol Show/Hide	C20H22N2O2	1
1	Ki = 16800 nM Bioactivity Info	TI LI LO TS
CP0272134 Compound Info	(4-fluorophenyl)-[1-[(3S,4S)-1-[(4-fluorophenyl)methyl]-3-hydroxypiperidin-4-yl]piperidin-4-yl]methanone Show/Hide	C24H28F2N2O2	1
1	Ki > 20000 nM Bioactivity Info	TI LI LO TS
CP0429033 Compound Info	[(1S,2R,5S,6S,7S)-3-benzyl-7-(diethylamino)-2-methyl-3-azabicyclo[3.2.0]heptan-6-yl]methanol Show/Hide	C19H30N2O	1
1	Ki = 21000 nM Bioactivity Info	TI LI LO TS
CP0411140 Compound Info	(11S)-5-methyl-6,11-dioxo-N-(pyridin-3-ylmethyl)benzo[b][1,4]benzothiazepine-3-carboxamide Show/Hide	C21H17N3O3S	1
1	Ki = 21000 nM Bioactivity Info	TI LI LO TS
CP0467854 Compound Info	5-[(5S)-5-methyl-4-propylmorpholin-2-yl]-N,N-dipropylpyridin-2-amine Show/Hide	C19H33N3O	1
1	Ki = 21100 nM Bioactivity Info	TI LI LO TS
CP0208172 Compound Info	N-butyl-1H-indole-2-carboxamide Show/Hide	C13H16N2O	1
1	Ki = 21542 nM Bioactivity Info	TI LI LO TS
CP0477400 Compound Info	7-butyl-2-(2-methoxyphenyl)-2,7-diazaspiro[4.4]nonane Show/Hide	C18H28N2O	1
1	Ki = 23256 nM Bioactivity Info	TI LI LO TS
CP0422924 Compound Info	7-[4-[(2R,5S)-2-(6-aminopyridin-3-yl)-5-methylmorpholin-4-yl]butoxy]-3,4-dihydro-1H-quinolin-2-one Show/Hide	C23H30N4O3	1
1	Ki = 24200 nM Bioactivity Info	TI LI LO TS
CP0384366 Compound Info	2-[4-(4-chlorophenyl)piperidin-1-yl]-N-(3-methylphenyl)acetamide Show/Hide	C20H23ClN2O	1
1	Ki = 26320 nM Bioactivity Info	TI LI LO TS
CP0447952 Compound Info	(10R)-10-(methylamino)-2-oxo-1,3-diazatricyclo[6.3.1.04,12]dodeca-4,6,8(12)-triene-6-carbonitrile Show/Hide	C12H12N4O	1
1	Ki = 27200 nM Bioactivity Info	TI LI LO TS
CP0478825 Compound Info	N-butyl-4-thiophen-3-ylbenzamide Show/Hide	C15H17NOS	1
1	Ki > 30000 nM Bioactivity Info	TI LI LO TS
CP0409127 Compound Info	[(1R,2S,5S,6S,7S)-3-benzyl-7-(diethylamino)-2-pyridin-2-yl-3-azabicyclo[3.2.0]heptan-6-yl]methanol Show/Hide	C23H31N3O	1
1	Ki = 36000 nM Bioactivity Info	TI LI LO TS
CP0423853 Compound Info	[(1S,2R,5S,6S,7S)-3-benzyl-2-methyl-7-pyrrolidin-1-yl-3-azabicyclo[3.2.0]heptan-6-yl]methanol Show/Hide	C19H28N2O	1
1	Ki = 36000 nM Bioactivity Info	TI LI LO TS
CP0390315 Compound Info	(R)-Modafinil Show/Hide	C15H15NO2S	1
1	Ki = 39000 nM Bioactivity Info	TI LI LO TS
CP0548209 Compound Info	3-(2-methoxyphenyl)-3,9-diazaspiro[5.5]undecane Show/Hide	C16H24N2O	1
1	Ki > 39319 nM Bioactivity Info	TI LI LO TS
CP0411143 Compound Info	(11R)-5-methyl-6,11-dioxo-N-(2-thiophen-2-ylethyl)benzo[b][1,4]benzothiazepine-3-carboxamide Show/Hide	C21H18N2O3S2	1
1	Ki > 50000 nM Bioactivity Info	TI LI LO TS
CP0396207 Compound Info	N-pentan-2-yl-1H-indole-2-carboxamide Show/Hide	C14H18N2O	1
1	Ki > 50000 nM Bioactivity Info	TI LI LO TS
CP0384367 Compound Info	2-[4-(5-chloropyridin-2-yl)piperazin-1-yl]-N-(3-ethylphenyl)acetamide Show/Hide	C19H23ClN4O	1
1	Ki > 50000 nM Bioactivity Info	TI LI LO TS
CP0384381 Compound Info	N-pyridin-3-yl-2-(4-pyridin-2-ylpiperazin-1-yl)acetamide Show/Hide	C16H19N5O	1
1	Ki > 50000 nM Bioactivity Info	TI LI LO TS
CP0384383 Compound Info	2-(4-pyridin-2-ylpiperazin-1-yl)-N-pyrimidin-5-ylacetamide Show/Hide	C15H18N6O	1
1	Ki > 50000 nM Bioactivity Info	TI LI LO TS
CP0384678 Compound Info	2-[4-(5-chloropyridin-2-yl)piperazin-1-yl]-N-pyrimidin-5-ylacetamide Show/Hide	C15H17ClN6O	1
1	Ki > 50000 nM Bioactivity Info	TI LI LO TS
CP0421988 Compound Info	2-[4-(5-chloropyridin-2-yl)piperazin-1-yl]-N-pyridin-3-ylacetamide Show/Hide	C16H18ClN5O	1
1	Ki > 50000 nM Bioactivity Info	TI LI LO TS
CP0416963 Compound Info	4-methyl-3-phenyl-5-propylsulfanyl-1,2,4-triazole Show/Hide	C12H15N3S	1
1	Ki > 50316 nM Bioactivity Info	TI LI LO TS
CP0384478 Compound Info	1-[3-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]propyl]piperazine Show/Hide	C16H23N5S	1
1	Ki = 72753 nM Bioactivity Info	TI LI LO TS
CP0519115 Compound Info	7-[(E)-4-[(2R,5S)-2-(6-aminopyridin-3-yl)-5-methylmorpholin-4-yl]but-2-enoxy]-3,4-dihydro-1H-quinolin-2-one Show/Hide	C23H28N4O3	1
1	Ki = 73000 nM Bioactivity Info	TI LI LO TS
CP0396215 Compound Info	N-propan-2-yl-1H-indole-2-carboxamide Show/Hide	C12H14N2O	1
1	Ki > 100000 nM Bioactivity Info	TI LI LO TS
CP0463359 Compound Info	N-heptan-4-yl-1H-indole-2-carboxamide Show/Hide	C16H22N2O	1
1	Ki > 100000 nM Bioactivity Info	TI LI LO TS
CP0470556 Compound Info	N-(cyclopropylmethyl)-1H-indole-2-carboxamide Show/Hide	C13H14N2O	1
1	Ki > 100000 nM Bioactivity Info	TI LI LO TS
CP0400240 Compound Info	7-(aminomethyl)-3-methyl-5-phenyl-1,2,4,5-tetrahydro-3-benzazepin-8-ol Show/Hide	C18H22N2O	1
1	Ki > 1000 nM Bioactivity Info	TI LI LO TS
CP0410524 Compound Info	8-(diethylamino)-3-methyl-5-phenyl-1,2,4,5-tetrahydro-3-benzazepin-7-ol Show/Hide	C21H28N2O	1
1	Ki > 1000 nM Bioactivity Info	TI LI LO TS
CP0410526 Compound Info	3-methyl-5-phenyl-1,2,4,5-tetrahydro-3-benzazepin-7-amine Show/Hide	C17H20N2	1
1	Ki > 1000 nM Bioactivity Info	TI LI LO TS
CP0410530 Compound Info	8-amino-3-methyl-5-phenyl-1,2,4,5-tetrahydro-3-benzazepin-7-ol Show/Hide	C17H20N2O	1
1	Ki > 1000 nM Bioactivity Info	TI LI LO TS
CP0424270 Compound Info	3-methyl-5-phenyl-1,2,4,5-tetrahydro-3-benzazepin-8-amine Show/Hide	C17H20N2	1
1	Ki > 1000 nM Bioactivity Info	TI LI LO TS
CP0426632 Compound Info	3-methyl-8-(3-methylphenyl)-5-phenyl-1,2,4,5-tetrahydro-3-benzazepin-7-ol Show/Hide	C24H25NO	1
1	Ki > 1000 nM Bioactivity Info	TI LI LO TS
CP0443430 Compound Info	3-methyl-8-(4-methylphenyl)-5-phenyl-1,2,4,5-tetrahydro-3-benzazepin-7-ol Show/Hide	C24H25NO	1
1	Ki > 1000 nM Bioactivity Info	TI LI LO TS
CP0443432 Compound Info	7-amino-3-methyl-5-phenyl-1,2,4,5-tetrahydro-3-benzazepin-8-ol Show/Hide	C17H20N2O	1
1	Ki > 1000 nM Bioactivity Info	TI LI LO TS
CP0443434 Compound Info	8-(benzylamino)-3-methyl-5-phenyl-1,2,4,5-tetrahydro-3-benzazepin-7-ol Show/Hide	C24H26N2O	1
1	Ki > 1000 nM Bioactivity Info	TI LI LO TS
CP0509154 Compound Info	3-methyl-5-phenyl-1,2,4,5-tetrahydro-3-benzazepin-7-ol Show/Hide	C17H19NO	1
1	Ki > 1000 nM Bioactivity Info	TI LI LO TS
CP0509157 Compound Info	3-methyl-5-phenyl-1,2,4,5-tetrahydro-3-benzazepin-8-ol Show/Hide	C17H19NO	1
1	Ki > 1000 nM Bioactivity Info	TI LI LO TS
CP0529531 Compound Info	7-(hydroxymethyl)-3-methyl-5-phenyl-1,2,4,5-tetrahydro-3-benzazepin-8-ol Show/Hide	C18H21NO2	1
1	Ki > 1000 nM Bioactivity Info	TI LI LO TS
CP0487134 Compound Info	4-[5-(4-Chloro-phenyl)-1H-pyrazol-3-yl]-1-methyl-piperidine Show/Hide	C15H18ClN3	1
1	Ki > 1900 nM Bioactivity Info	TI LI LO TS
CP0374884 Compound Info	5-Methyl-1-(1-phenethyl-piperidin-4-yl)-4-phenyl-1,3-dihydro-imidazol-2-one Show/Hide	C23H27N3O	1
1	Ki > 3200 nM Bioactivity Info	TI LI LO TS
CP0409092 Compound Info	[3-[2-(dimethylamino)ethyl]-5-hydroxyindol-1-yl]-phenylmethanone Show/Hide	C19H20N2O2	1
1	Ki > 3500 nM Bioactivity Info	TI LI LO TS
CP0377325 Compound Info	1-[1-(3-Methoxy-benzyl)-piperidin-4-yl]-5-methyl-4-phenyl-1,3-dihydro-imidazol-2-one Show/Hide	C23H27N3O2	1
1	Ki > 3900 nM Bioactivity Info	TI LI LO TS
CP0169831 Compound Info	4-[5-(4-Chloro-phenyl)-1H-pyrazol-3-yl]-1-phenethyl-piperidine Show/Hide	C22H24ClN3	1
1	Ki > 4000 nM Bioactivity Info	TI LI LO TS
CP0455488 Compound Info	4-[5-(1-Phenethyl-piperidin-4-yl)-2H-pyrazol-3-yl]-pyridine Show/Hide	C21H24N4	1
1	Ki > 4000 nM Bioactivity Info	TI LI LO TS
CP0404428 Compound Info	1-[1-(2-Chloro-benzyl)-piperidin-4-yl]-5-methyl-4-phenyl-1,3-dihydro-imidazol-2-one Show/Hide	C22H24ClN3O	1
1	Ki > 4000 nM Bioactivity Info	TI LI LO TS
CP0404174 Compound Info	3-[5-(1-Phenethyl-piperidin-4-yl)-2H-pyrazol-3-yl]-pyridine Show/Hide	C21H24N4	1
1	Ki > 4200 nM Bioactivity Info	TI LI LO TS
CP0414849 Compound Info	1-Benzyl-3-(1-benzyl-piperidin-4-yl)-urea Show/Hide	C20H25N3O	1
1	Ki > 4200 nM Bioactivity Info	TI LI LO TS
CP0442957 Compound Info	4-[3-(4-CHLOROPHENYL)-1H-PYRAZOL-5-YL]PIPERIDINE Show/Hide	C14H16ClN3	1
1	Ki > 4400 nM Bioactivity Info	TI LI LO TS
CP0460824 Compound Info	1-Benzyl-4-(5-phenyl-tetrazol-1-yl)-piperidine Show/Hide	C19H21N5	1
1	Ki > 4400 nM Bioactivity Info	TI LI LO TS
CP0378669 Compound Info	1-Benzoyl-3-(1-benzyl-piperidin-4-yl)-urea Show/Hide	C20H23N3O2	1
1	Ki > 4400 nM Bioactivity Info	TI LI LO TS
CP0380824 Compound Info	5-Methyl-1-(1-methyl-piperidin-4-yl)-4-phenyl-1,3-dihydro-imidazol-2-one Show/Hide	C16H21N3O	1
1	Ki > 4400 nM Bioactivity Info	TI LI LO TS
CP0437134 Compound Info	1-[1-(3-Chloro-benzyl)-piperidin-4-yl]-5-methyl-4-phenyl-1,3-dihydro-imidazol-2-one Show/Hide	C22H24ClN3O	1
1	Ki > 4700 nM Bioactivity Info	TI LI LO TS
CP0383198 Compound Info	3-[4-(5-Methyl-2-oxo-4-phenyl-2,3-dihydro-imidazol-1-yl)-piperidin-1-ylmethyl]-benzonitrile Show/Hide	C23H24N4O	1
1	Ki > 4800 nM Bioactivity Info	TI LI LO TS
CP0372386 Compound Info	(1-((1H-indol-3-yl)methyl)-4-(4-chlorophenyl)piperidin-4-yl)methanamine Show/Hide	C21H24ClN3	1
1	Ki > 5000 nM Bioactivity Info	TI LI LO TS

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About MolBiC

Correspondence

Prof. Feng ZHU

Prof. Leo, Lianyi Han