Brief Information of the Compound and Protein
Compound Name
 Compound Info 
(R)-N-(4-(4-Phenylbenzoylamino)butyl)-N-propyl-5-amino-4,5,6,7-tetrahydropyrazolo[1,5-a]pyridine
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 PubChem ID
CID: 52937875
SID: 123077946
Canonical SMILES
CCCN(CCCCNC(=O)c1ccc(cc1)-c1ccccc1)[C@@H]1CCn2nccc2C1
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Compound Formula C27H34N4O
Compound Structure
Protein Name
 Protein Info 
D(3) dopamine receptor
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
>
Small molecule receptor (family A GPCR)
>
Monoamine receptor
>
Dopamine receptor
Uniprot ID
P35462
Gene Name
DRD3
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO
 Cell Line Info 
Cricetulus griseus (Chinese hamster)  2
1
Ki = 6.3 nM
   TI
   LI
   LO
   TS
2
Ki = 15 nM
   TI
   LI
   LO
   TS
CL000006 HEK293
 Cell Line Info 
Homo sapiens (Human)  7
1
EC50 = 51 nM
   TI
   LI
   LO
   TS
2
Ki = 15 nM
   TI
   LI
   LO
   TS
3
Ki = 19 nM
   TI
   LI
   LO
   TS
4
Ki = 43 nM
   TI
   LI
   LO
   TS
5
Ki = 240 nM
   TI
   LI
   LO
   TS
6
Ki = 1400 nM
   TI
   LI
   LO
   TS
7
Ki = 3700 nM
   TI
   LI
   LO
   TS