Brief Information of the Cell Line and Protein
Cell Line ID: CL000006 , HEK293
Synonyms
Hek293
HEK-293
HEK/293
HEK 293
HEK;293
293
293 HEK
293 Ad5
Graham 293
Graham-293
Human Embryonic Kidney 293
Category Transformed cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_0045
Protein ID: PT00864 , Vascular endothelial growth factor receptor 2
Gene Name KDR
Organism Homo sapiens, Human
Protein Classification Kinase
Uniprot ID P35968
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000006  Protein ID: PT00864
 
Compound ID Compound Name Compound Formula
CP0276883
2-Methoxy-5-{[6-methoxy-7-(3-pyrrolidin-1-ylpropoxy)quinazolin-4-yl]amino}benzo-1,4-quinone
   Show/Hide
C23H26N4O5
 1
1
IC50 = 3 nM
   TI
   LI
   LO
   TS
CP0287174
2-Methoxy-5-({6-methoxy-7-[(1-methylpiperidin-4-yl)methoxy]quinazolin-4-yl}amino)benzo-1,4-quinone
   Show/Hide
C23H26N4O5
 1
1
IC50 = 5 nM
   TI
   LI
   LO
   TS
CP0111076
2-(6-(4-(2-(pyrrolidin-1-yl)ethyl)piperazin-1-yl)pyrimidin-4-ylamino)thiazole-5-carbonitrile
   Show/Hide
C18H24N8S
 1
1
IC50 = 11 nM
   TI
   LI
   LO
   TS
CP0376346
1-methanesulfonyl-4-[(4-{3-phenylimidazo[1,2-a]pyridin-7-yl}phenyl)methyl]piperazine
   Show/Hide
C25H26N4O2S
 1
1
IC50 = 13 nM
   TI
   LI
   LO
   TS
CP0038986
2-(4-Piperazin-1-ylmethylpyridin-2-ylamino)thiazole-5-carbonitrile
   Show/Hide
C14H16N6S
 2
1
IC50 = 13 nM
   TI
   LI
   LO
   TS
2
IC50 = 24 nM
   TI
   LI
   LO
   TS
CP0141029
2-(6-(4-aminoazepan-1-yl)pyrimidin-4-ylamino)thiazole-5-carbonitrile
   Show/Hide
C14H17N7S
 1
1
IC50 = 15 nM
   TI
   LI
   LO
   TS
CP0037980
(4-chlorophenyl)-[4-(4-pyridylmethyl)phthalazin-1-yl]amine
   Show/Hide
C20H15ClN4
 2
1
IC50 < 15 nM
   TI
   LI
   LO
   TS
2
IC50 = 21 nM
   TI
   LI
   LO
   TS
CP0037988
N-(4-bromo-2-fluorophenyl)-6-methoxy-7-[(1-methylpiperidin-4-yl)methoxy]quinazolin-4-amine
   Show/Hide
C22H24BrFN4O2
 2
1
IC50 < 15 nM
   TI
   LI
   LO
   TS
2
IC50 = 1660 nM
   TI
   LI
   LO
   TS
CP0659535
2-{[6-Methoxy-7-(2-methoxyethoxy)-4-quinazolinyl]amino}-5-methylbenzo-1,4-quinone
   Show/Hide
C19H19N3O5
 1
1
IC50 < 15 nM
   TI
   LI
   LO
   TS
CP0144564
(5-Phenylthiazol-2-yl)(4-pyrrolidin-1-ylmethylpyridin-2-yl)amine
   Show/Hide
C19H20N4S
 2
1
IC50 = 15 nM
   TI
   LI
   LO
   TS
2
IC50 = 24 nM
   TI
   LI
   LO
   TS
CP0146007
4-({2-[(5-cyano-1,3-thiazol-2-yl)amino]-3-methylpyridin-4-yl}methyl)-N-methylpiperazine-1-carboxamide
   Show/Hide
C17H21N7OS
 2
1
IC50 = 16 nM
   TI
   LI
   LO
   TS
2
IC50 = 38 nM
   TI
   LI
   LO
   TS
CP0133219
4-{[4-(Methylsulfonyl)piperazin-1-yl]methyl}-N-(5-phenyl-1,3-thiazol-2-yl)pyridin-2-amine
   Show/Hide
C20H23N5O2S2
 2
1
IC50 = 17 nM
   TI
   LI
   LO
   TS
2
IC50 = 29 nM
   TI
   LI
   LO
   TS
CP0092730
1-(2-(pyridin-4-yl)ethyl)-N-(4-(trifluoromethoxy)phenyl)-1H-pyrazole-5-carboxamide
   Show/Hide
C18H15F3N4O2
 1
1
IC50 = 18 nM
   TI
   LI
   LO
   TS
CP0074851
2-(6-(4-(2-morpholinoethyl)piperazin-1-yl)pyrimidin-4-ylamino)thiazole-5-carbonitrile
   Show/Hide
C18H24N8OS
 1
1
IC50 = 19 nM
   TI
   LI
   LO
   TS
CP0205190
(rac)-2-(6-(3-aminopyrrolidin-1-yl)pyrimidin-4-ylamino)thiazole-5-carbonitrile
   Show/Hide
C12H13N7S
 1
1
IC50 = 21 nM
   TI
   LI
   LO
   TS
CP0104347
N-[3-[chloro(difluoro)methoxy]phenyl]-2-(2-pyridin-4-ylethyl)pyrazole-3-carboxamide
   Show/Hide
C18H15ClF2N4O2
 1
1
IC50 = 21 nM
   TI
   LI
   LO
   TS
CP0155086
2-(6-(4-(2-methoxyethyl)piperazin-1-yl)pyrimidin-4-ylamino)thiazole-5-carbonitrile
   Show/Hide
C15H19N7OS
 1
1
IC50 = 22 nM
   TI
   LI
   LO
   TS
CP0074847
2-(6-(4-methylpiperazin-1-yl)pyrimidin-4-ylamino)thiazole-5-carbonitrile
   Show/Hide
C13H15N7S
 1
1
IC50 = 23 nM
   TI
   LI
   LO
   TS
CP0155085
2-(6-(4-(3-morpholinopropyl)piperazin-1-yl)pyrimidin-4-ylamino)thiazole-5-carbonitrile
   Show/Hide
C19H26N8OS
 1
1
IC50 = 23 nM
   TI
   LI
   LO
   TS
CP0038985
4-({2-[(5-Cyano-1,3-thiazol-2-yl)amino]-4-pyridinyl}-methyl)-1-piperazinecarboxamide
   Show/Hide
C15H17N7OS
 2
1
IC50 = 24 nM
   TI
   LI
   LO
   TS
2
IC50 = 47 nM
   TI
   LI
   LO
   TS
CP0133199
5-phenyl-N-[5-(pyrrolidin-1-ylmethyl)pyridin-2-yl]-1,3-thiazol-2-amine
   Show/Hide
C19H20N4S
 2
1
IC50 = 24 nM
   TI
   LI
   LO
   TS
2
IC50 = 28 nM
   TI
   LI
   LO
   TS
CP0659537
2-methoxy-5-{[6-methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino}benzo-1,4-quinone
   Show/Hide
C19H19N3O6
 1
1
IC50 = 25 nM
   TI
   LI
   LO
   TS
CP0162412
4-({2-[(5-cyano-1,3-thiazol-2-yl)amino]pyridin-4-yl}methyl)-N-methylpiperazine-1-carboxamide
   Show/Hide
C16H19N7OS
 2
1
IC50 = 27 nM
   TI
   LI
   LO
   TS
2
IC50 = 31 nM
   TI
   LI
   LO
   TS
CP0453005
4-{3-phenylimidazo[1,2-a]pyridin-7-yl}-1-[3-(piperidin-1-yl)propyl]-1,2-dihydropyridin-2-one
   Show/Hide
C26H28N4O
 1
1
IC50 = 28 nM
   TI
   LI
   LO
   TS
CP0104182
4-({2-[(5-Cyano-1,3-thiazol-2-yl)amino]-4-pyridinyl}-methyl)-N,N-dimethyl-1-piperazinecarboxamide
   Show/Hide
C17H21N7OS
 2
1
IC50 = 28 nM
   TI
   LI
   LO
   TS
2
IC50 = 40 nM
   TI
   LI
   LO
   TS
CP0104183
1-[4-({2-[(5-phenyl-1,3-thiazol-2-yl)amino]pyridin-4-yl}methyl)piperazin-1-yl]ethan-1-one
   Show/Hide
C21H23N5OS
 2
1
IC50 = 28 nM
   TI
   LI
   LO
   TS
2
IC50 = 43 nM
   TI
   LI
   LO
   TS
CP0339626
2-(4-Morpholin-4-ylmethylpyridin-2-ylamino)thiazole-5-carbonitrile
   Show/Hide
C14H15N5OS
 2
1
IC50 = 28 nM
   TI
   LI
   LO
   TS
2
IC50 = 43 nM
   TI
   LI
   LO
   TS
CP0058668
2-(dimethylamino)-5-[[6-methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino]cyclohexa-2,5-diene-1,4-dione
   Show/Hide
C20H22N4O5
 1
1
IC50 = 31 nM
   TI
   LI
   LO
   TS
CP0275018
2-({4-[(4-methanesulfonylpiperidin-1-yl)methyl]pyridin-2-yl}amino)-1,3-thiazole-5-carbonitrile
   Show/Hide
C16H19N5O2S2
 2
1
IC50 = 31 nM
   TI
   LI
   LO
   TS
2
IC50 = 48 nM
   TI
   LI
   LO
   TS
CP0046140
2-(6-(1,4-diazepan-1-yl)pyrimidin-4-ylamino)thiazole-5-carbonitrile
   Show/Hide
C13H15N7S
 1
1
IC50 = 32 nM
   TI
   LI
   LO
   TS
CP0104334
N-(4-tert-butylphenyl)-2-(2-pyridin-4-ylethyl)pyrazole-3-carboxamide
   Show/Hide
C21H24N4O
 1
1
IC50 = 33 nM
   TI
   LI
   LO
   TS
CP0046151
2-(6-(piperazin-1-yl)pyrimidin-4-ylamino)thiazole-5-carbonitrile
   Show/Hide
C12H13N7S
 1
1
IC50 = 34 nM
   TI
   LI
   LO
   TS
CP0144563
2-[(4-{[4-(2-hydroxyacetyl)piperazin-1-yl]methyl}pyridin-2-yl)amino]-1,3-thiazole-5-carbonitrile
   Show/Hide
C16H18N6O2S
 2
1
IC50 = 35 nM
   TI
   LI
   LO
   TS
2
IC50 = 39 nM
   TI
   LI
   LO
   TS
CP0141416
2-({4-[(4-acetylpiperazin-1-yl)methyl]pyridin-2-yl}amino)-1,3-thiazole-5-carbonitrile
   Show/Hide
C16H18N6OS
 2
1
IC50 = 36 nM
   TI
   LI
   LO
   TS
2
IC50 = 41 nM
   TI
   LI
   LO
   TS
CP0037347
4-(pyridin-4-ylmethylamino)-N-(3-(trifluoromethoxy)phenyl)isothiazole-3-carboxamide
   Show/Hide
C17H13F3N4O2S
 1
1
IC50 = 41 nM
   TI
   LI
   LO
   TS
CP0166793
2-{7-phenylimidazo[1,2-a]pyridin-3-yl}-1,3-thiazole
   Show/Hide
C16H11N3S
 1
1
IC50 = 42 nM
   TI
   LI
   LO
   TS
CP0059956
2-(6-(4-acetylpiperazin-1-yl)pyrimidin-4-ylamino)thiazole-5-carbonitrile
   Show/Hide
C14H15N7OS
 1
1
IC50 = 44 nM
   TI
   LI
   LO
   TS
CP0044880
((pyridin-4-yl)ethyl)pyridine 25
   Show/Hide
C21H16ClF2N5O2
 1
1
IC50 = 44 nM
   TI
   LI
   LO
   TS
CP0092718
1-(2-(pyridin-4-yl)ethyl)-N-(4-(trifluoromethyl)phenyl)-1Hpyrazole-5-carboxamide
   Show/Hide
C18H15F3N4O
 1
1
IC50 = 48 nM
   TI
   LI
   LO
   TS
CP0053328
2-[(pyridin-4-ylmethyl)amino]-N-(quinolin-3-yl)benzamide
   Show/Hide
C22H18N4O
 1
1
IC50 = 50 nM
   TI
   LI
   LO
   TS
CP0496664
4-{7-phenylimidazo[1,2-a]pyridin-3-yl}-1,2-thiazole
   Show/Hide
C16H11N3S
 1
1
IC50 = 50 nM
   TI
   LI
   LO
   TS
CP0046078
((pyridin-4-yl)ethyl)pyridine 26
   Show/Hide
C21H16F3N5O2
 1
1
IC50 = 51 nM
   TI
   LI
   LO
   TS
CP0509172
N-methyl-4-[(4-{3-phenylimidazo[1,2-a]pyridin-7-yl}phenyl)methyl]piperazine-1-carboxamide
   Show/Hide
C26H27N5O
 1
1
IC50 = 52 nM
   TI
   LI
   LO
   TS
CP0092729
N-(4-propan-2-ylphenyl)-2-(2-pyridin-4-ylethyl)pyrazole-3-carboxamide
   Show/Hide
C20H22N4O
 1
1
IC50 = 53 nM
   TI
   LI
   LO
   TS
CP0049078
4-(pyridin-4-ylmethylamino)-N-(3-(trifluoromethyl)phenyl)isothiazole-3-carboxamide
   Show/Hide
C17H13F3N4OS
 1
1
IC50 = 54 nM
   TI
   LI
   LO
   TS
CP0037353
N-[4-methyl-3-(trifluoromethyl)phenyl]-4-(pyridin-4-ylmethylamino)-1,2-thiazole-3-carboxamide
   Show/Hide
C18H15F3N4OS
 1
1
IC50 = 56 nM
   TI
   LI
   LO
   TS
CP0074846
2-(6-(4-aminopiperidin-1-yl)pyrimidin-4-ylamino)thiazole-5-carbonitrile
   Show/Hide
C13H15N7S
 1
1
IC50 = 59 nM
   TI
   LI
   LO
   TS
CP0068325
((pyridin-4-yl)ethyl)pyridine 19
   Show/Hide
C24H25N5O
 1
1
IC50 = 63 nM
   TI
   LI
   LO
   TS
CP0161326
N-(3-methoxyphenyl)-5-[3-methyl-5-(pyridin-4-ylmethylamino)imidazol-4-yl]-1,3,4-oxadiazol-2-amine
   Show/Hide
C19H19N7O2
 1
1
IC50 = 64 nM
   TI
   LI
   LO
   TS
CP0077687
5-(1-methyl-4-(pyridin-4-ylmethylamino)-1H-imidazol-5-yl)-N-(4-(trifluoromethoxy)phenyl)-1,3,4-oxadiazol-2-amine
   Show/Hide
C19H16F3N7O2
 1
1
IC50 = 66 nM
   TI
   LI
   LO
   TS
CP0506752
1-(3-{3-[(dimethylamino)methyl]piperidin-1-yl}propyl)-4-{3-phenylimidazo[1,2-a]pyridin-7-yl}-1,2-dihydropyridin-2-one
   Show/Hide
C29H35N5O
 1
1
IC50 = 67 nM
   TI
   LI
   LO
   TS
CP0498122
4-[(4-{3-phenylimidazo[1,2-a]pyridin-7-yl}phenyl)methyl]piperazine-1-carboxamide
   Show/Hide
C25H25N5O
 1
1
IC50 = 69 nM
   TI
   LI
   LO
   TS
CP0079002
3,6-diarylpyrazolo[1,5-a]pyrimidine 1
   Show/Hide
C19H15N3O
 1
1
IC50 = 71 nM
   TI
   LI
   LO
   TS
CP0172259
N-(4-tert-butylphenyl)-4-[2-(pyridin-4-yl)ethyl]-1,3-thiazole-5-carboxamide
   Show/Hide
C21H23N3OS
 1
1
IC50 = 73 nM
   TI
   LI
   LO
   TS
CP0154872
((pyridin-4-yl)ethyl)pyridine 20
   Show/Hide
C23H23N5O
 1
1
IC50 = 75 nM
   TI
   LI
   LO
   TS
CP0044879
((pyridin-4-yl)ethyl)pyridine 27
   Show/Hide
C21H16F3N5O
 1
1
IC50 = 76 nM
   TI
   LI
   LO
   TS
CP0508598
1-{4-[(4-{3-phenylimidazo[1,2-a]pyridin-7-yl}phenyl)methyl]piperazin-1-yl}ethan-1-one
   Show/Hide
C26H26N4O
 1
1
IC50 = 77 nM
   TI
   LI
   LO
   TS
CP0083122
2-[3-(Ethylamino)phenoxy]-5-{[6-methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino}benzo-1,4-quinone
   Show/Hide
C26H26N4O6
 1
1
IC50 = 78 nM
   TI
   LI
   LO
   TS
CP0048979
N-(3-tert-butylphenyl)-4-(pyridin-4-ylmethylamino)-1,2-thiazole-3-carboxamide
   Show/Hide
C20H22N4OS
 1
1
IC50 = 82 nM
   TI
   LI
   LO
   TS
CP0154766
5-(1-methyl-4-(pyridin-4-ylmethylamino)-1H-imidazol-5-yl)-N-(4-(trifluoromethyl)phenyl)-1,3,4-oxadiazol-2-amine
   Show/Hide
C19H16F3N7O
 1
1
IC50 = 82 nM
   TI
   LI
   LO
   TS
CP0154666
N-(Aryl)-thiazole-5-carboxamide 17
   Show/Hide
C18H14ClF2N3O2S
 1
1
IC50 = 85 nM
   TI
   LI
   LO
   TS
CP0176477
N-(4-ethylphenyl)-2-(2-pyridin-4-ylethyl)pyrazole-3-carboxamide
   Show/Hide
C19H20N4O
 1
1
IC50 = 86 nM
   TI
   LI
   LO
   TS
CP0037106
2-[(pyridin-4-ylmethyl)amino]-N-[3-(trifluoromethyl)phenyl]benzamide
   Show/Hide
C20H16F3N3O
 1
1
IC50 = 90 nM
   TI
   LI
   LO
   TS
CP0144490
N-(3,4-dimethoxyphenyl)-2-(2-pyridin-4-ylethyl)pyrazole-3-carboxamide
   Show/Hide
C19H20N4O3
 1
1
IC50 = 90 nM
   TI
   LI
   LO
   TS
CP0144613
N-(4-chlorophenyl)-2-(2-pyridin-4-ylethyl)pyrazole-3-carboxamide
   Show/Hide
C17H15ClN4O
 1
1
IC50 = 90 nM
   TI
   LI
   LO
   TS
CP0198306
((pyridin-4-yl)ethyl)pyridine 43
   Show/Hide
C22H18F3N5O
 1
1
IC50 = 92 nM
   TI
   LI
   LO
   TS
CP0154793
N-(3,4-dimethoxyphenyl)-5-[3-methyl-5-(pyridin-4-ylmethylamino)imidazol-4-yl]-1,3,4-oxadiazol-2-amine
   Show/Hide
C20H21N7O3
 1
1
IC50 = 93 nM
   TI
   LI
   LO
   TS
CP0187168
N-(3,4-dichlorophenyl)-4-[2-(pyridin-4-yl)ethyl]-1,3-thiazole-5-carboxamide
   Show/Hide
C17H13Cl2N3OS
 1
1
IC50 = 93 nM
   TI
   LI
   LO
   TS
CP0198307
((pyridin-4-yl)ethyl)pyridine 41
   Show/Hide
C20H15Cl2N5O
 1
1
IC50 = 94 nM
   TI
   LI
   LO
   TS
CP0081011
N-(4-chlorophenyl)-4-[2-(pyridin-4-yl)ethyl]-1,3-thiazole-5-carboxamide
   Show/Hide
C17H14ClN3OS
 1
1
IC50 = 95 nM
   TI
   LI
   LO
   TS
CP0156059
N-[3-chloro-4-(trifluoromethyl)phenyl]-2-(2-pyridin-4-ylethyl)pyrazole-3-carboxamide
   Show/Hide
C18H14ClF3N4O
 1
1
IC50 = 95 nM
   TI
   LI
   LO
   TS
CP0095083
N-[4-[chloro(difluoro)methoxy]phenyl]-5-[3-methyl-5-(pyridin-4-ylmethylamino)imidazol-4-yl]-1,3,4-oxadiazol-2-amine
   Show/Hide
C19H16ClF2N7O2
 1
1
IC50 = 96 nM
   TI
   LI
   LO
   TS
CP0487511
1-{3-[(2-methoxyethyl)(methyl)amino]propyl}-4-{3-phenylimidazo[1,2-a]pyridin-7-yl}-1,2-dihydropyridin-2-one
   Show/Hide
C25H28N4O2
 1
1
IC50 = 96 nM
   TI
   LI
   LO
   TS
CP0520350
3,7-diphenylimidazo[1,2-a]pyridine
   Show/Hide
C19H14N2
 1
1
IC50 = 98 nM
   TI
   LI
   LO
   TS
CP0430391
5-{7-phenylimidazo[1,2-a]pyridin-3-yl}-1,3-thiazole
   Show/Hide
C16H11N3S
 1
1
IC50 = 99 nM
   TI
   LI
   LO
   TS
CP0167046
N-[4-chloro-3-(trifluoromethyl)phenyl]-5-[3-methyl-5-(pyridin-4-ylmethylamino)imidazol-4-yl]-1,3,4-oxadiazol-2-amine
   Show/Hide
C19H15ClF3N7O
 1
1
IC50 = 100 nM
   TI
   LI
   LO
   TS
CP0057908
((pyridin-4-yl)ethyl)pyridine 5
   Show/Hide
C21H16F3N5O
 1
1
IC50 = 110 nM
   TI
   LI
   LO
   TS
CP0171348
((pyridin-4-yl)ethyl)pyridine 42
   Show/Hide
C22H21N5O3
 1
1
IC50 = 110 nM
   TI
   LI
   LO
   TS
CP0283886
((pyridin-4-yl)ethyl)pyridine 34
   Show/Hide
C21H16F3N5O2
 1
1
IC50 = 110 nM
   TI
   LI
   LO
   TS
CP0085415
2-(2-((4-Pyridyl)methyl)aminophenyl)-5-(3,4-ethylenedioxy)phenylamino-1,3,4-oxadiazole
   Show/Hide
C22H19N5O3
 1
1
IC50 = 110 nM
   TI
   LI
   LO
   TS
CP0203643
5-(4-methoxyphenyl)-1-phenyl-1H-1,3-benzodiazole
   Show/Hide
C20H16N2O
 1
1
IC50 = 113 nM
   TI
   LI
   LO
   TS
CP0505701
1-(3-hydroxypropyl)-4-{3-phenylimidazo[1,2-a]pyridin-7-yl}-1,2-dihydropyridin-2-one
   Show/Hide
C21H19N3O2
 1
1
IC50 = 120 nM
   TI
   LI
   LO
   TS
CP0166883
N-(Aryl)-thiazole-5-carboxamide 15
   Show/Hide
C20H21N3OS
 1
1
IC50 = 120 nM
   TI
   LI
   LO
   TS
CP0176479
N-(3,4-dichlorophenyl)-2-(2-pyridin-4-ylethyl)pyrazole-3-carboxamide
   Show/Hide
C17H14Cl2N4O
 1
1
IC50 = 120 nM
   TI
   LI
   LO
   TS
CP0154800
5-(1-methyl-4-(pyridin-4-ylmethylamino)-1H-imidazol-5-yl)-N-(3-(trifluoromethoxy)phenyl)-1,3,4-oxadiazol-2-amine
   Show/Hide
C19H16F3N7O2
 1
1
IC50 = 130 nM
   TI
   LI
   LO
   TS
CP0504761
4-{7-phenylimidazo[1,2-a]pyridin-3-yl}pyridine
   Show/Hide
C18H13N3
 1
1
IC50 = 145 nM
   TI
   LI
   LO
   TS
CP0255544
2-[[6-methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino]-5-phenoxycyclohexa-2,5-diene-1,4-dione
   Show/Hide
C24H21N3O6
 1
1
IC50 = 184 nM
   TI
   LI
   LO
   TS
CP0776051
2-[2-Fluoro-1-(fluoromethyl)ethoxy]-5-({6-methoxy-7-[(1-methylpiperidin-4-yl)methoxy]quinazolin-4-yl}amino)benzo-1,4-quinone
   Show/Hide
C25H28F2N4O5
 1
1
IC50 = 189 nM
   TI
   LI
   LO
   TS
CP0083110
N-(Aryl)-thiazole-5-carboxamide 27
   Show/Hide
C18H13ClF3N3OS
 1
1
IC50 = 190 nM
   TI
   LI
   LO
   TS
CP0058680
2-[[6-methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino]-5-(pyridin-3-ylmethoxy)cyclohexa-2,5-diene-1,4-dione
   Show/Hide
C24H22N4O6
 1
1
IC50 = 193 nM
   TI
   LI
   LO
   TS
CP0922988
2-{[6-Methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino}-5-(2-methylaziridin-1-yl)benzo-1,4-quinone
   Show/Hide
C21H22N4O5
 1
1
IC50 = 206 nM
   TI
   LI
   LO
   TS
CP0070472
N-(3-bromophenyl)-4-(pyridin-4-ylmethylamino)-1,2-thiazole-3-carboxamide
   Show/Hide
C16H13BrN4OS
 1
1
IC50 = 210 nM
   TI
   LI
   LO
   TS
CP0058678
2-(1,3-difluoropropan-2-yloxy)-5-[[6-methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino]cyclohexa-2,5-diene-1,4-dione
   Show/Hide
C21H21F2N3O6
 1
1
IC50 = 212 nM
   TI
   LI
   LO
   TS
CP0085419
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-[2-(quinolin-6-ylmethylamino)pyridin-3-yl]-1,3,4-oxadiazol-2-amine
   Show/Hide
C25H20N6O3
 1
1
IC50 = 220 nM
   TI
   LI
   LO
   TS
CP0255372
N-(2-fluoro-4-methylphenyl)-4-[2-(pyridin-4-yl)ethyl]-1,3-thiazole-5-carboxamide
   Show/Hide
C18H16FN3OS
 1
1
IC50 = 230 nM
   TI
   LI
   LO
   TS
CP0533052
2-methoxy-6-{7-phenylimidazo[1,2-a]pyridin-3-yl}pyridine
   Show/Hide
C19H15N3O
 1
1
IC50 = 242 nM
   TI
   LI
   LO
   TS
CP0077686
N-(3,4-dichlorophenyl)-5-[3-methyl-5-(pyridin-4-ylmethylamino)imidazol-4-yl]-1,3,4-oxadiazol-2-amine
   Show/Hide
C18H15Cl2N7O
 1
1
IC50 = 260 nM
   TI
   LI
   LO
   TS
CP0114690
N-(3-bromophenyl)-4-(quinolin-4-ylmethylamino)-1,2-thiazole-3-carboxamide
   Show/Hide
C20H15BrN4OS
 1
1
IC50 = 270 nM
   TI
   LI
   LO
   TS
CP0131800
N-(1,3-benzodioxol-5-ylmethyl)-5-[3-methyl-5-(pyridin-4-ylmethylamino)imidazol-4-yl]-1,3,4-oxadiazol-2-amine
   Show/Hide
C20H19N7O3
 1
1
IC50 = 270 nM
   TI
   LI
   LO
   TS
CP0104348
1-(2-(pyridin-4-yl)ethyl)-N-(3-(trifluoromethoxy)phenyl)-1H-pyrazole-5-carboxamide
   Show/Hide
C18H15F3N4O2
 1
1
IC50 = 280 nM
   TI
   LI
   LO
   TS
CP0154933
((pyridin-4-yl)ethyl)pyridine 44
   Show/Hide
C22H19N5O3
 1
1
IC50 = 290 nM
   TI
   LI
   LO
   TS
CP0161222
((pyridin-4-yl)ethyl)pyridine 38
   Show/Hide
C21H19N5O2
 1
1
IC50 = 290 nM
   TI
   LI
   LO
   TS
CP0166949
2-(4-imidazol-1-ylphenoxy)-5-[[6-methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino]cyclohexa-2,5-diene-1,4-dione
   Show/Hide
C27H23N5O6
 1
1
IC50 = 310 nM
   TI
   LI
   LO
   TS
CP0428214
2-[[6-methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino]-5-piperidin-1-ylcyclohexa-2,5-diene-1,4-dione
   Show/Hide
C23H26N4O5
 1
1
IC50 = 310 nM
   TI
   LI
   LO
   TS
CP0154871
((pyridin-4-yl)ethyl)pyridine 21
   Show/Hide
C24H25N5O
 1
1
IC50 = 320 nM
   TI
   LI
   LO
   TS
CP0276881
2-[[6-methoxy-7-[(1-methylpiperidin-4-yl)methoxy]quinazolin-4-yl]amino]-5-[2-(N-methylanilino)ethoxy]cyclohexa-2,5-diene-1,4-dione
   Show/Hide
C31H35N5O5
 1
1
IC50 = 329 nM
   TI
   LI
   LO
   TS
CP0186425
N-(2H-1,3-benzodioxol-5-yl)-4-[2-(pyridin-4-yl)ethyl]-1,3-thiazole-5-carboxamide
   Show/Hide
C18H15N3O3S
 1
1
IC50 = 330 nM
   TI
   LI
   LO
   TS
CP0048988
4-(quinolin-4-ylmethylamino)-N-(3-(trifluoromethyl)phenyl)isothiazole-3-carboxamide
   Show/Hide
C21H15F3N4OS
 1
1
IC50 = 390 nM
   TI
   LI
   LO
   TS
CP0155091
((pyridin-4-yl)ethyl)pyridine 22
   Show/Hide
C23H23N5O
 1
1
IC50 = 390 nM
   TI
   LI
   LO
   TS
CP0048991
N-(4-chlorophenyl)-4-(pyridin-4-ylmethylamino)-1,2-thiazole-3-carboxamide
   Show/Hide
C16H13ClN4OS
 1
1
IC50 = 420 nM
   TI
   LI
   LO
   TS
CP0156055
N-[4-chloro-3-(trifluoromethyl)phenyl]-2-(2-pyridin-4-ylethyl)pyrazole-3-carboxamide
   Show/Hide
C18H14ClF3N4O
 1
1
IC50 = 450 nM
   TI
   LI
   LO
   TS
CP0739703
2-{[6-Methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino}-5-(methylthio)benzo-1,4-quinone
   Show/Hide
C19H19N3O5S
 1
1
IC50 = 456 nM
   TI
   LI
   LO
   TS
CP0287201
3-chloro-2-methoxy-5-[[6-methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino]cyclohexa-2,5-diene-1,4-dione
   Show/Hide
C19H18ClN3O6
 1
1
IC50 = 466 nM
   TI
   LI
   LO
   TS
CP0146175
2-[[6-methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino]-5-propan-2-yloxycyclohexa-2,5-diene-1,4-dione
   Show/Hide
C21H23N3O6
 1
1
IC50 = 481 nM
   TI
   LI
   LO
   TS
CP0334180
((pyridin-4-yl)ethyl)pyridine 32
   Show/Hide
C21H16F3N5O2
 1
1
IC50 = 510 nM
   TI
   LI
   LO
   TS
CP0257151
((pyridin-4-yl)ethyl)pyridine 23
   Show/Hide
C24H25N5O
 1
1
IC50 = 520 nM
   TI
   LI
   LO
   TS
CP0146720
N-[4-chloro-3-(trifluoromethyl)phenyl]-4-(pyridin-4-ylmethylamino)-1,2-thiazole-3-carboxamide
   Show/Hide
C17H12ClF3N4OS
 1
1
IC50 = 530 nM
   TI
   LI
   LO
   TS
CP0154935
((pyridin-4-yl)ethyl)pyridine 28
   Show/Hide
C21H16ClF2N5O2
 1
1
IC50 = 530 nM
   TI
   LI
   LO
   TS
CP0776052
2-(Benzyloxy)-5-({6-methoxy-7-[(1-methylpiperidin-4-yl)methoxy]quinazolin-4-yl}amino)benzo-1,4-quinone
   Show/Hide
C29H30N4O5
 1
1
IC50 = 536 nM
   TI
   LI
   LO
   TS
CP0140586
N-(4-chlorophenyl)-5-[3-methyl-5-(pyridin-4-ylmethylamino)imidazol-4-yl]-1,3,4-oxadiazol-2-amine
   Show/Hide
C18H16ClN7O
 1
1
IC50 = 570 nM
   TI
   LI
   LO
   TS
CP0205353
N-(Aryl)-thiazole-5-carboxamide 23
   Show/Hide
C21H22N4O2S
 1
1
IC50 = 580 nM
   TI
   LI
   LO
   TS
CP0167079
((pyridin-4-yl)ethyl)pyridine 31
   Show/Hide
C21H16ClF2N5O2
 1
1
IC50 = 590 nM
   TI
   LI
   LO
   TS
CP0154799
N-(2-fluoro-4-methylphenyl)-5-[3-methyl-5-(pyridin-4-ylmethylamino)imidazol-4-yl]-1,3,4-oxadiazol-2-amine
   Show/Hide
C19H18FN7O
 1
1
IC50 = 640 nM
   TI
   LI
   LO
   TS
CP0029006
4-[4-[7-amino-2-(1,2,3-benzothiadiazol-7-yl)furo[2,3-c]pyridin-4-yl]pyrazol-1-yl]cyclohexan-1-ol
   Show/Hide
C22H20N6O2S
 1
1
IC50 = 650 nM
   TI
   LI
   LO
   TS
CP0154927
((pyridin-4-yl)ethyl)pyridine 29
   Show/Hide
C21H16F3N5O2
 1
1
IC50 = 660 nM
   TI
   LI
   LO
   TS
CP0048977
N-[3-methyl-4-(trifluoromethyl)phenyl]-4-(pyridin-4-ylmethylamino)-1,2-thiazole-3-carboxamide
   Show/Hide
C18H15F3N4OS
 1
1
IC50 = 710 nM
   TI
   LI
   LO
   TS
CP0059884
((pyridin-4-yl)ethyl)pyridine 30
   Show/Hide
C21H16F3N5O
 1
1
IC50 = 720 nM
   TI
   LI
   LO
   TS
CP0046077
((pyridin-4-yl)ethyl)pyridine 33
   Show/Hide
C21H16F3N5O
 1
1
IC50 = 740 nM
   TI
   LI
   LO
   TS
CP0167080
((pyridin-4-yl)ethyl)pyridine 36
   Show/Hide
C21H16F3N5O2
 1
1
IC50 = 760 nM
   TI
   LI
   LO
   TS
CP0018308
4-[4-[7-amino-2-(1,2,3-benzothiadiazol-7-yl)-3-(1,3-thiazol-5-yl)furo[2,3-c]pyridin-4-yl]pyrazol-1-yl]cyclohexan-1-ol
   Show/Hide
C25H21N7O2S2
 1
1
IC50 = 760 nM
   TI
   LI
   LO
   TS
CP0037337
4-(pyridin-4-ylmethylamino)-N-(4-(trifluoromethoxy)phenyl)isothiazole-3-carboxamide
   Show/Hide
C17H13F3N4O2S
 1
1
IC50 = 770 nM
   TI
   LI
   LO
   TS
CP0070468
4-(pyridin-4-ylmethylamino)-N-(quinolin-2-yl)isothiazole-3-carboxamide
   Show/Hide
C19H15N5OS
 1
1
IC50 = 770 nM
   TI
   LI
   LO
   TS
CP0048983
N-(1,3-benzodioxol-5-ylmethyl)-4-(pyridin-4-ylmethylamino)-1,2-thiazole-3-carboxamide
   Show/Hide
C18H16N4O3S
 1
1
IC50 = 790 nM
   TI
   LI
   LO
   TS
CP0206502
3-chloro-2-(1,3-difluoropropan-2-yloxy)-5-[[6-methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino]cyclohexa-2,5-diene-1,4-dione
   Show/Hide
C21H20ClF2N3O6
 1
1
IC50 = 792 nM
   TI
   LI
   LO
   TS
CP0503935
5-(2-((1H-imidazol-5-yl)methylamino)pyridin-3-yl)-N-(2,3-dihydrobenzo[b][1,4]dioxin-6-yl)-1,3,4-oxadiazol-2-amine
   Show/Hide
C19H17N7O3
 1
1
IC50 = 830 nM
   TI
   LI
   LO
   TS
CP0154895
((pyridin-4-yl)ethyl)pyridine 35
   Show/Hide
C21H16F3N5O2
 1
1
IC50 = 860 nM
   TI
   LI
   LO
   TS
CP0735137
2-(2,2-Difluoroethoxy)-5-{[6-methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino}benzo-1,4-quinone
   Show/Hide
C20H19F2N3O6
 1
1
IC50 = 870 nM
   TI
   LI
   LO
   TS
CP0524550
3-{7-phenylimidazo[1,2-a]pyridin-3-yl}pyridine
   Show/Hide
C18H13N3
 1
1
IC50 = 930 nM
   TI
   LI
   LO
   TS
CP0465691
3-(5-(2,3-dihydrobenzo[b][1,4]dioxin-6-ylamino)-1,3,4-oxadiazol-2-yl)-N-(pyridin-4-ylmethyl)pyridin-2-amine
   Show/Hide
C21H18N6O3
 1
1
IC50 = 1000 nM
   TI
   LI
   LO
   TS
CP0510126
N-(pyridin-4-ylmethyl)-3-[3-[3-(trifluoromethyl)phenyl]-1H-1,2,4-triazol-5-yl]pyridin-2-amine
   Show/Hide
C20H15F3N6
 1
1
IC50 = 1000 nM
   TI
   LI
   LO
   TS
CP0171305
N-(4-bromophenyl)-4-[2-(pyridin-4-yl)ethyl]-1,3-thiazole-5-carboxamide
   Show/Hide
C17H14BrN3OS
 1
1
IC50 = 1020 nM
   TI
   LI
   LO
   TS
CP0070471
N-(4-bromophenyl)-4-(pyridin-4-ylmethylamino)-1,2-thiazole-3-carboxamide
   Show/Hide
C16H13BrN4OS
 1
1
IC50 = 1040 nM
   TI
   LI
   LO
   TS
CP0154791
N-(4-tert-butylphenyl)-5-[3-methyl-5-(pyridin-4-ylmethylamino)imidazol-4-yl]-1,3,4-oxadiazol-2-amine
   Show/Hide
C22H25N7O
 1
1
IC50 = 1050 nM
   TI
   LI
   LO
   TS
CP0144485
1-(2-(pyridin-4-yl)ethyl)-N-(4-(trifluoromethoxy)phenyl)-1H-imidazole-2-carboxamide
   Show/Hide
C18H15F3N4O2
 1
1
IC50 = 1050 nM
   TI
   LI
   LO
   TS
CP0037354
N-(3,4-dichlorophenyl)-4-(pyridin-4-ylmethylamino)-1,2-thiazole-3-carboxamide
   Show/Hide
C16H12Cl2N4OS
 1
1
IC50 = 1110 nM
   TI
   LI
   LO
   TS
CP0057927
((pyridin-4-yl)ethyl)pyridine 6
   Show/Hide
C21H16F3N5O
 1
1
IC50 = 1110 nM
   TI
   LI
   LO
   TS
CP0037346
N-(4-tert-butylphenyl)-4-(pyridin-4-ylmethylamino)-1,2-thiazole-3-carboxamide
   Show/Hide
C20H22N4OS
 1
1
IC50 = 1150 nM
   TI
   LI
   LO
   TS
CP0154794
5-[3-methyl-5-(pyridin-4-ylmethylamino)imidazol-4-yl]-N-(4-propan-2-ylphenyl)-1,3,4-oxadiazol-2-amine
   Show/Hide
C21H23N7O
 1
1
IC50 = 1150 nM
   TI
   LI
   LO
   TS
CP0092719
1-(2-(pyridin-4-yl)ethyl)-N-(quinolin-3-yl)-1H-pyrazole-5-carboxamide
   Show/Hide
C20H17N5O
 1
1
IC50 = 1220 nM
   TI
   LI
   LO
   TS
CP0104336
N-(4-chlorophenyl)-1-(2-pyridin-4-ylethyl)imidazole-2-carboxamide
   Show/Hide
C17H15ClN4O
 1
1
IC50 = 1320 nM
   TI
   LI
   LO
   TS
CP0104337
3-methyl-1-(2-(pyridin-4-yl)ethyl)-N-(4-(trifluoromethoxy)phenyl)-1H-pyrazole-5-carboxamide
   Show/Hide
C19H17F3N4O2
 1
1
IC50 = 1340 nM
   TI
   LI
   LO
   TS
CP0138150
4-(pyridin-4-ylmethylamino)-N-(4-(trifluoromethyl)phenyl)isothiazole-3-carboxamide
   Show/Hide
C17H13F3N4OS
 1
1
IC50 = 1530 nM
   TI
   LI
   LO
   TS
CP0144472
2-(2-pyridin-4-yl-ethyl)-2H-pyrazole-3-carboxylic acid biphenyl-4-ylamide
   Show/Hide
C23H20N4O
 1
1
IC50 = 1560 nM
   TI
   LI
   LO
   TS
CP0205352
N-(4-tert-butylphenyl)-4-[2-(1,2-oxazol-4-yl)ethyl]-1,3-thiazole-5-carboxamide
   Show/Hide
C19H21N3O2S
 1
1
IC50 = 1630 nM
   TI
   LI
   LO
   TS
CP0215330
1-(2-(pyridin-4-yl)ethyl)-N-(4-(trifluoromethyl)phenyl)-1H-imidazole-2-carboxamide
   Show/Hide
C18H15F3N4O
 1
1
IC50 = 1660 nM
   TI
   LI
   LO
   TS
CP0037344
N-(2-fluoro-4-methylphenyl)-4-(pyridin-4-ylmethylamino)-1,2-thiazole-3-carboxamide
   Show/Hide
C17H15FN4OS
 1
1
IC50 = 1890 nM
   TI
   LI
   LO
   TS
CP0092884
N-(4-chlorophenyl)-1-(2-pyridin-4-ylethyl)tetrazole-5-carboxamide
   Show/Hide
C15H13ClN6O
 1
1
IC50 = 2030 nM
   TI
   LI
   LO
   TS
CP0037350
N-[3-chloro-4-(trifluoromethyl)phenyl]-4-(pyridin-4-ylmethylamino)-1,2-thiazole-3-carboxamide
   Show/Hide
C17H12ClF3N4OS
 1
1
IC50 = 2050 nM
   TI
   LI
   LO
   TS
CP0154934
((pyridin-4-yl)ethyl)pyridine 37
   Show/Hide
C21H19N5O
 1
1
IC50 = 2140 nM
   TI
   LI
   LO
   TS
CP0081010
N-(Aryl)-thiazole-5-carboxamide 16
   Show/Hide
C16H12ClF2N3O3S
 1
1
IC50 = 2250 nM
   TI
   LI
   LO
   TS
CP0104344
N-(4-tert-butylphenyl)-1-(2-pyridin-4-ylethyl)imidazole-2-carboxamide
   Show/Hide
C21H24N4O
 1
1
IC50 = 2250 nM
   TI
   LI
   LO
   TS
CP0171304
N-(4-chlorophenyl)-4-[2-(1,2-oxazol-4-yl)ethyl]-1,3-thiazole-5-carboxamide
   Show/Hide
C15H12ClN3O2S
 1
1
IC50 = 2300 nM
   TI
   LI
   LO
   TS
CP0171517
((pyridin-4-yl)ethyl)pyridine 7
   Show/Hide
C21H16F3N5O
 1
1
IC50 = 2540 nM
   TI
   LI
   LO
   TS
CP0144476
N-(4-chlorophenyl)-5-methyl-2-(2-pyridin-4-ylethyl)pyrazole-3-carboxamide
   Show/Hide
C18H17ClN4O
 1
1
IC50 = 2540 nM
   TI
   LI
   LO
   TS
CP0186427
N-(2-fluoro-4-methylphenyl)-4-[2-(1,2-oxazol-4-yl)ethyl]-1,3-thiazole-5-carboxamide
   Show/Hide
C16H14FN3O2S
 1
1
IC50 = 2750 nM
   TI
   LI
   LO
   TS
CP0085417
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-[2-(pyridin-3-ylmethylamino)phenyl]-1H-1,2,4-triazol-3-amine
   Show/Hide
C22H20N6O2
 1
1
IC50 = 2800 nM
   TI
   LI
   LO
   TS
CP0144488
1-(2-(pyridin-4-yl)ethyl)-N-(4-(trifluoromethyl)phenyl)-1H-tetrazole-5-carboxamide
   Show/Hide
C16H13F3N6O
 1
1
IC50 = 2960 nM
   TI
   LI
   LO
   TS
CP0039110
1-(2-(pyridin-4-yl)ethyl)-N-(4-(trifluoromethoxy)phenyl)-1H-tetrazole-5-carboxamide
   Show/Hide
C16H13F3N6O2
 1
1
IC50 = 2970 nM
   TI
   LI
   LO
   TS
CP0029005
4-(1-methylpyrazol-4-yl)-2-thieno[2,3-c]pyridin-3-ylfuro[2,3-c]pyridin-7-amine
   Show/Hide
C18H13N5OS
 1
1
IC50 = 3400 nM
   TI
   LI
   LO
   TS
CP0104335
N-[3-chloro-4-(trifluoromethyl)phenyl]-1-(2-pyridin-4-ylethyl)imidazole-2-carboxamide
   Show/Hide
C18H14ClF3N4O
 1
1
IC50 = 4950 nM
   TI
   LI
   LO
   TS
CP0154792
5-(4-(3,4-difluorobenzylamino)-1-methyl-1H-imidazol-5-yl)-N-(4-chlorophenyl)-1,3,4-oxadiazol-2-amine
   Show/Hide
C19H15ClF2N6O
 1
1
IC50 = 5650 nM
   TI
   LI
   LO
   TS
CP0474411
5-(2-((1H-indazol-5-yl)methylamino)phenyl)-N-(2,3-dihydrobenzo[b][1,4]dioxin-6-yl)-4H-1,2,4-triazol-3-amine
   Show/Hide
C24H21N7O2
 1
1
IC50 = 7300 nM
   TI
   LI
   LO
   TS
CP0018195
4-[4-[7-amino-2-(1,2,3-benzothiadiazol-7-yl)-3-pyridin-3-ylfuro[2,3-c]pyridin-4-yl]pyrazol-1-yl]cyclohexan-1-ol
   Show/Hide
C27H23N7O2S
 1
1
IC50 = 8200 nM
   TI
   LI
   LO
   TS
CP0037332
N-(3-bromophenyl)-4-(1,2-oxazol-4-ylmethylamino)-1,2-thiazole-3-carboxamide
   Show/Hide
C14H11BrN4O2S
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0037333
4-(pyridin-2-ylmethylamino)-N-(3-(trifluoromethyl)phenyl)isothiazole-3-carboxamide
   Show/Hide
C17H13F3N4OS
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0037339
4-(pyridin-2-ylmethylamino)-N-(4-(trifluoromethyl)phenyl)isothiazole-3-carboxamide
   Show/Hide
C17H13F3N4OS
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0037342
N-(3-bromophenyl)-4-(quinolin-2-ylmethylamino)-1,2-thiazole-3-carboxamide
   Show/Hide
C20H15BrN4OS
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0037348
4-(2-(benzo[d][1,3]dioxol-5-yl)ethylamino)-N-(3-bromophenyl)isothiazole-3-carboxamide
   Show/Hide
C19H16BrN3O3S
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0037351
4-(pyridin-3-ylmethylamino)-N-(3-(trifluoromethyl)phenyl)isothiazole-3-carboxamide
   Show/Hide
C17H13F3N4OS
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0048975
4-(pyridin-3-ylmethylamino)-N-(4-(trifluoromethyl)phenyl)isothiazole-3-carboxamide
   Show/Hide
C17H13F3N4OS
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0048987
N-(2-bromophenyl)-4-(pyridin-4-ylmethylamino)-1,2-thiazole-3-carboxamide
   Show/Hide
C16H13BrN4OS
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0048990
4-(3,4-difluorobenzylamino)-N-(3-(trifluoromethyl)phenyl)isothiazole-3-carboxamide
   Show/Hide
C18H12F5N3OS
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0147380
4-(2-(benzo[d][1,3]dioxol-5-yl)ethylamino)-N-(3-(trifluoromethyl)phenyl)isothiazole-3-carboxamide
   Show/Hide
C20H16F3N3O3S
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0713299
N-(3a,7a-dihydro-1H-indazol-5-yl)-4-(pyridin-4-ylmethylamino)isothiazole-3-carboxamide
   Show/Hide
C17H16N6OS
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0077684
5-(4-((1H-indazol-5-yl)methylamino)-1-methyl-1H-imidazol-5-yl)-N-(4-chlorophenyl)-1,3,4-oxadiazol-2-amine
   Show/Hide
C20H17ClN8O
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0131798
5-(4-(2-(benzo[d][1,3]dioxol-5-yl)ethylamino)-1-methyl-1H-imidazol-5-yl)-N-(4-chlorophenyl)-1,3,4-oxadiazol-2-amine
   Show/Hide
C21H19ClN6O3
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0154788
N-(4-chlorophenyl)-5-[3-methyl-5-(pyridin-3-ylmethylamino)imidazol-4-yl]-1,3,4-oxadiazol-2-amine
   Show/Hide
C18H16ClN7O
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0154796
N-(4-chlorophenyl)-5-[3-methyl-5-(quinolin-2-ylmethylamino)imidazol-4-yl]-1,3,4-oxadiazol-2-amine
   Show/Hide
C22H18ClN7O
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0161325
N-(4-chlorophenyl)-5-[3-methyl-5-(pyridin-2-ylmethylamino)imidazol-4-yl]-1,3,4-oxadiazol-2-amine
   Show/Hide
C18H16ClN7O
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0166917
N-(4-chlorophenyl)-5-[3-methyl-5-(quinolin-5-ylmethylamino)imidazol-4-yl]-1,3,4-oxadiazol-2-amine
   Show/Hide
C22H18ClN7O
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0044892
((pyridin-2-yl)ethyl)pyridine 10
   Show/Hide
C21H16F3N5O
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0044893
((pyridin-4-yl)ethyl)quinoline 8
   Show/Hide
C25H18F3N5O
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0046076
5-{2-[2-(3,4-difluorophenyl)ethyl]pyridin-3-yl}-N-[3-(trifluoromethyl)phenyl]-1,3,4-oxadiazol-2-amine
   Show/Hide
C22H15F5N4O
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0046080
((indazole)ethyl)pyridine 14
   Show/Hide
C23H17F3N6O
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0068322
5-{3-[3-(2H-1,3-benzodioxol-5-yl)propyl]pyridin-4-yl}-N-[3-(trifluoromethyl)phenyl]-1,3,4-oxadiazol-2-amine
   Show/Hide
C24H19F3N4O3
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0140781
((quinoline)ethyl)pyridine 16
   Show/Hide
C25H18F3N5O
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0171340
5-{2-[3-(2H-1,3-benzodioxol-5-yl)propyl]pyridin-3-yl}-N-[3-(trifluoromethyl)phenyl]-1,3,4-oxadiazol-2-amine
   Show/Hide
C24H19F3N4O3
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0171476
((pyridin-3-yl)ethyl)pyridine 9
   Show/Hide
C21H16F3N5O
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0171558
((quinoline)ethyl)pyridine 15
   Show/Hide
C25H18F3N5O
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0081009
N-(3-methylphenyl)-4-[2-(1,2-oxazol-4-yl)ethyl]-1,3-thiazole-5-carboxamide
   Show/Hide
C16H15N3O2S
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0083107
N-(4-tert-butylphenyl)-4-[2-(quinolin-4-yl)ethyl]-1,3-thiazole-5-carboxamide
   Show/Hide
C25H25N3OS
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0166123
N-(4-chlorophenyl)-4-[2-(quinolin-2-yl)ethyl]-1,3-thiazole-5-carboxamide
   Show/Hide
C21H16ClN3OS
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0166884
4-[2-(1,2-benzoxazol-3-yl)ethyl]-N-(4-tert-butylphenyl)-1,3-thiazole-5-carboxamide
   Show/Hide
C23H23N3O2S
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0171307
N-(4-tert-butylphenyl)-4-[2-(quinolin-2-yl)ethyl]-1,3-thiazole-5-carboxamide
   Show/Hide
C25H25N3OS
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0186423
N-(4-chlorophenyl)-4-[2-(quinolin-4-yl)ethyl]-1,3-thiazole-5-carboxamide
   Show/Hide
C21H16ClN3OS
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0205354
4-[2-(1,2-benzoxazol-3-yl)ethyl]-N-(4-chlorophenyl)-1,3-thiazole-5-carboxamide
   Show/Hide
C19H14ClN3O2S
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0039085
N-(4-chlorophenyl)-2-(2-pyridin-2-ylethyl)pyrazole-3-carboxamide
   Show/Hide
C17H15ClN4O
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0039106
N-(4-phenoxyphenyl)-2-(2-pyridin-4-ylethyl)pyrazole-3-carboxamide
   Show/Hide
C23H20N4O2
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0092725
N-(4-chlorophenyl)-2-[2-(1,2-oxazol-4-yl)ethyl]pyrazole-3-carboxamide
   Show/Hide
C15H13ClN4O2
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0092726
N-[3-chloro-4-(trifluoromethyl)phenyl]-1-(2-pyridin-4-ylethyl)benzimidazole-2-carboxamide
   Show/Hide
C22H16ClF3N4O
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0092887
3,4-dimethyl-1-(2-(pyridin-4-yl)ethyl)-N-(4-(trifluoromethoxy)phenyl)-1H-pyrazole-5-carboxamide
   Show/Hide
C20H19F3N4O2
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0104342
N-(4-chlorophenyl)-1-(2-pyridin-4-ylethyl)benzimidazole-2-carboxamide
   Show/Hide
C21H17ClN4O
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0104345
N-(4-chlorophenyl)-1-(2-pyridin-4-ylethyl)indole-2-carboxamide
   Show/Hide
C22H18ClN3O
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0104346
N-(1H-indazol-5-yl)-2-(2-pyridin-4-ylethyl)pyrazole-3-carboxamide
   Show/Hide
C18H16N6O
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0144468
N-[3-chloro-4-(trifluoromethyl)phenyl]-1-(2-pyridin-4-ylethyl)tetrazole-5-carboxamide
   Show/Hide
C16H12ClF3N6O
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0144470
N-(4-chlorophenyl)-4,5-dimethyl-2-(2-pyridin-4-ylethyl)pyrazole-3-carboxamide
   Show/Hide
C19H19ClN4O
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0144473
1-(3,4-dimethoxyphenethyl)-N-(4-chlorophenyl)-1H-pyrazole-5-carboxamide
   Show/Hide
C20H20ClN3O3
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0144479
N-(1H-indazol-6-yl)-2-(2-pyridin-4-ylethyl)pyrazole-3-carboxamide
   Show/Hide
C18H16N6O
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0144481
1-(2-(benzo[d]isoxazol-3-yl)ethyl)-N-(4-chlorophenyl)-1H-pyrazole-5-carboxamide
   Show/Hide
C19H15ClN4O2
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0144483
1-(3,4-difluorophenethyl)-N-(4-chlorophenyl)-1H-pyrazole-5-carboxamide
   Show/Hide
C18H14ClF2N3O
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0144484
N-(4-tert-butylphenyl)-1-(2-pyridin-4-ylethyl)tetrazole-5-carboxamide
   Show/Hide
C19H22N6O
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0144492
1-(2-(1H-imidazol-4-yl)ethyl)-N-(4-chlorophenyl)-1H-pyrazole-5-carboxamide
   Show/Hide
C15H14ClN5O
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0144495
N-(4-chlorophenyl)-2-(2-pyridin-3-ylethyl)pyrazole-3-carboxamide
   Show/Hide
C17H15ClN4O
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0144498
N-(4-phenylmethoxyphenyl)-2-(2-pyridin-4-ylethyl)pyrazole-3-carboxamide
   Show/Hide
C24H22N4O2
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0172690
N-(4-chlorophenyl)-2-[2-(6-methyl-5,6-dihydro-1,3-benzodioxol-4-yl)ethyl]pyrazole-3-carboxamide
   Show/Hide
C20H20ClN3O3
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0210499
1-(2-(pyridin-4-yl)ethyl)-N-(4-(trifluoromethoxy)phenyl)-1H-benzo[d]imidazole-2-carboxamide
   Show/Hide
C22H17F3N4O2
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0212724
1-(2-(pyridin-4-yl)ethyl)-N-(4-(trifluoromethoxy)phenyl)-1H-indole-2-carboxamide
   Show/Hide
C23H18F3N3O2
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0051595
3-(5-(2,3-dihydrobenzo[b][1,4]dioxin-6-ylamino)-1,3,4-oxadiazol-2-yl)-N-(pyridin-3-ylmethyl)pyridin-2-amine
   Show/Hide
C21H18N6O3
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0085416
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-[2-(2-pyridin-3-ylethylamino)pyridin-3-yl]-1,3,4-oxadiazol-2-amine
   Show/Hide
C22H20N6O3
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0085418
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-[2-(quinolin-6-ylmethylamino)phenyl]-1H-1,2,4-triazol-3-amine
   Show/Hide
C26H22N6O2
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0103329
N-(2,2-difluoro-1,3-benzodioxol-5-yl)-5-[2-(pyridin-4-ylmethylamino)pyridin-3-yl]-1,3,4-oxadiazol-2-amine
   Show/Hide
C20H14F2N6O3
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0218509
5-(2-((1H-indazol-5-yl)methylamino)pyridin-3-yl)-N-(2,3-dihydrobenzo[b][1,4]dioxin-6-yl)-1,3,4-oxadiazol-2-amine
   Show/Hide
C23H19N7O3
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0234933
N-(1,4-dioxan-2-ylmethyl)-3-[3-(4-methylsulfonylphenyl)-1H-1,2,4-triazol-5-yl]pyridin-2-amine
   Show/Hide
C19H21N5O4S
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0234934
3-(5-(benzo[d][1,3]dioxol-5-ylamino)-1,3,4-oxadiazol-2-yl)-N-(pyridin-3-ylmethyl)pyridin-2-amine
   Show/Hide
C20H16N6O3
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0257946
N-(1,3-benzodioxol-5-yl)-5-[2-(1,3-benzodioxol-5-ylmethylamino)pyridin-3-yl]-1,3,4-oxadiazol-2-amine
   Show/Hide
C22H17N5O5
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0297397
N-(1H-pyrazol-4-ylmethyl)-3-[3-[3-(trifluoromethyl)phenyl]-1H-1,2,4-triazol-5-yl]pyridin-2-amine
   Show/Hide
C18H14F3N7
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0297398
N-(pyridin-4-ylmethyl)-3-[5-[3-(trifluoromethyl)phenyl]-1,3,4-oxadiazol-2-yl]pyridin-2-amine
   Show/Hide
C20H14F3N5O
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0297399
N-(1,3-benzodioxol-5-yl)-5-[2-(2-pyridin-4-ylethylamino)pyridin-3-yl]-1,3,4-oxadiazol-2-amine
   Show/Hide
C21H18N6O3
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0297400
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-[2-(pyridin-4-ylmethylamino)phenyl]-1H-1,2,4-triazol-3-amine
   Show/Hide
C22H20N6O2
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0297660
2-(2-((4-Pyridyl)methyl)aminophenyl)-5-(3,4-methylenedioxy)phenylamino-1,3,4-oxadiazole
   Show/Hide
C21H17N5O3
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0297661
3-(5-(benzo[d][1,3]dioxol-5-ylamino)-1,3,4-oxadiazol-2-yl)-N-(pyridin-2-ylmethyl)pyridin-2-amine
   Show/Hide
C20H16N6O3
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0297662
5-[2-(1,3-benzodioxol-5-ylmethylamino)pyridin-3-yl]-N-(2,3-dihydro-1,4-benzodioxin-6-yl)-1,3,4-oxadiazol-2-amine
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C23H19N5O5
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0297665
5-(2-((1H-imidazol-5-yl)methylamino)phenyl)-N-(2,3-dihydrobenzo[b][1,4]dioxin-6-yl)-4H-1,2,4-triazol-3-amine
   Show/Hide
C20H19N7O2
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0307728
3-(5-(benzo[d][1,3]dioxol-5-yl)-4H-1,2,4-triazol-3-yl)-N-(pyridin-4-ylmethyl)pyridin-2-amine
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C20H16N6O2
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0313290
N-(1,3-benzodioxol-5-yl)-5-[2-(2-pyridin-3-ylethylamino)pyridin-3-yl]-1,3,4-oxadiazol-2-amine
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C21H18N6O3
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0313292
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-[2-(2-pyridin-4-ylethylamino)pyridin-3-yl]-1,3,4-oxadiazol-2-amine
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C22H20N6O3
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0321542
3-(5-(benzo[d][1,3]dioxol-5-ylamino)-1,3,4-oxadiazol-2-yl)-N-(pyridin-4-ylmethyl)pyridin-2-amine
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C20H16N6O3
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0543671
3-(5-(2,3-dihydrobenzo[b][1,4]dioxin-6-ylamino)-1,3,4-oxadiazol-2-yl)-N-(pyridin-2-ylmethyl)pyridin-2-amine
   Show/Hide
C21H18N6O3
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0017901
4-[4-[7-amino-2-(1,2,3-benzothiadiazol-7-yl)-3-(fluoromethyl)furo[2,3-c]pyridin-4-yl]pyrazol-1-yl]cyclohexan-1-ol
   Show/Hide
C23H21FN6O2S
 1
1
IC50 = 18300 nM
   TI
   LI
   LO
   TS
CP0031772
4-(1,5-dimethylpyrazol-4-yl)-2-thieno[2,3-c]pyridin-3-ylfuro[2,3-c]pyridin-7-amine
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C19H15N5OS
 1
1
IC50 = 19900 nM
   TI
   LI
   LO
   TS
CP0018196
4-[4-[7-amino-2-(1,2,3-benzothiadiazol-7-yl)-3-(difluoromethyl)furo[2,3-c]pyridin-4-yl]pyrazol-1-yl]cyclohexan-1-ol
   Show/Hide
C23H20F2N6O2S
 1
1
IC50 > 20000 nM
   TI
   LI
   LO
   TS
CP0018592
4-[4-[7-amino-2-(1,2,3-benzothiadiazol-7-yl)-3-chlorofuro[2,3-c]pyridin-4-yl]pyrazol-1-yl]cyclohexan-1-ol
   Show/Hide
C22H19ClN6O2S
 1
1
IC50 > 20000 nM
   TI
   LI
   LO
   TS
CP0025123
7-amino-2-(1,2,3-benzothiadiazol-7-yl)-4-[1-(4-hydroxycyclohexyl)pyrazol-4-yl]furo[2,3-c]pyridine-3-carbonitrile
   Show/Hide
C23H19N7O2S
 1
1
IC50 > 20000 nM
   TI
   LI
   LO
   TS
CP0031773
4-(1,3-dimethylpyrazol-4-yl)-2-thieno[2,3-c]pyridin-3-ylfuro[2,3-c]pyridin-7-amine
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C19H15N5OS
 1
1
IC50 > 20000 nM
   TI
   LI
   LO
   TS
CP0031774
4-(3-methoxy-1-methylpyrazol-4-yl)-2-thieno[2,3-c]pyridin-3-ylfuro[2,3-c]pyridin-7-amine
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C19H15N5O2S
 1
1
IC50 > 20000 nM
   TI
   LI
   LO
   TS
CP0058676
2-(4-benzylpiperazin-1-yl)-5-[[6-methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino]cyclohexa-2,5-diene-1,4-dione
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C29H31N5O5
 1
1
IC50 > 1000 nM
   TI
   LI
   LO
   TS
CP0058682
2-[(4-fluorophenyl)methoxy]-5-[[6-methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino]cyclohexa-2,5-diene-1,4-dione
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C25H22FN3O6
 1
1
IC50 > 1000 nM
   TI
   LI
   LO
   TS
CP0146169
2-[[6-methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino]-5-morpholin-4-ylcyclohexa-2,5-diene-1,4-dione
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C22H24N4O6
 1
1
IC50 > 1000 nM
   TI
   LI
   LO
   TS
CP0154729
2-chloro-5-[[6-methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino]cyclohexa-2,5-diene-1,4-dione
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C18H16ClN3O5
 1
1
IC50 > 1000 nM
   TI
   LI
   LO
   TS
CP0166952
3-Chloro-2-ethoxy-5-{[6-methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino}benzo-1,4-quinone
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C20H20ClN3O6
 1
1
IC50 > 1000 nM
   TI
   LI
   LO
   TS
CP0206503
2-[[6-methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino]-5-(2,2,2-trifluoro-1-phenylethoxy)cyclohexa-2,5-diene-1,4-dione
   Show/Hide
C26H22F3N3O6
 1
1
IC50 > 1000 nM
   TI
   LI
   LO
   TS
CP0212509
2-Ethoxy-5-{[6-methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino}benzo-1,4-quinone
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C20H21N3O6
 1
1
IC50 > 1000 nM
   TI
   LI
   LO
   TS
CP0250096
2-(4-Ethylpiperazin-1-yl)-5-{[6-methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino}benzo-1,4-quinone
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C24H29N5O5
 1
1
IC50 > 1000 nM
   TI
   LI
   LO
   TS
CP0309154
2-[[6-methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino]cyclohexa-2,5-diene-1,4-dione
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C18H17N3O5
 1
1
IC50 > 1000 nM
   TI
   LI
   LO
   TS
CP0659536
2-{[6-Methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino}-5-[methyl(phenyl) amino] benzo-1,4-quinon
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C25H24N4O5
 1
1
IC50 > 1000 nM
   TI
   LI
   LO
   TS
CP0659539
2-{[6-Methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino}-5-(2-phenoxyethoxy)benzo-1,4-quinone
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C26H25N3O7
 1
1
IC50 > 1000 nM
   TI
   LI
   LO
   TS
CP0704450
2-{[-6-methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino}-5-(5-methyl-2-oxo-1,3-oxazolidin-3-yl)benzo-1,4-quinone
   Show/Hide
C22H22N4O7
 1
1
IC50 > 1000 nM
   TI
   LI
   LO
   TS
CP0113988
CEP-32496
   Show/Hide
C24H22F3N5O5
 1
1
Kd = 8 nM
   TI
   LI
   LO
   TS