Compound ID |
Compound Name |
Compound Formula |
CP0276883
|
2-Methoxy-5-{[6-methoxy-7-(3-pyrrolidin-1-ylpropoxy)quinazolin-4-yl]amino}benzo-1,4-quinone
Show/Hide
|
C23H26N4O5
|
1
|
1 |
IC50 = 3 nM
|
|
|
CP0287174
|
2-Methoxy-5-({6-methoxy-7-[(1-methylpiperidin-4-yl)methoxy]quinazolin-4-yl}amino)benzo-1,4-quinone
Show/Hide
|
C23H26N4O5
|
1
|
1 |
IC50 = 5 nM
|
|
|
CP0111076
|
2-(6-(4-(2-(pyrrolidin-1-yl)ethyl)piperazin-1-yl)pyrimidin-4-ylamino)thiazole-5-carbonitrile
Show/Hide
|
C18H24N8S
|
1
|
1 |
IC50 = 11 nM
|
|
|
CP0376346
|
1-methanesulfonyl-4-[(4-{3-phenylimidazo[1,2-a]pyridin-7-yl}phenyl)methyl]piperazine
Show/Hide
|
C25H26N4O2S
|
1
|
1 |
IC50 = 13 nM
|
|
|
CP0038986
|
2-(4-Piperazin-1-ylmethylpyridin-2-ylamino)thiazole-5-carbonitrile
Show/Hide
|
C14H16N6S
|
2
|
1 |
IC50 = 13 nM
|
|
|
2 |
IC50 = 24 nM
|
|
|
CP0141029
|
2-(6-(4-aminoazepan-1-yl)pyrimidin-4-ylamino)thiazole-5-carbonitrile
Show/Hide
|
C14H17N7S
|
1
|
1 |
IC50 = 15 nM
|
|
|
CP0037980
|
(4-chlorophenyl)-[4-(4-pyridylmethyl)phthalazin-1-yl]amine
Show/Hide
|
C20H15ClN4
|
2
|
1 |
IC50 < 15 nM
|
|
|
2 |
IC50 = 21 nM
|
|
|
CP0037988
|
N-(4-bromo-2-fluorophenyl)-6-methoxy-7-[(1-methylpiperidin-4-yl)methoxy]quinazolin-4-amine
Show/Hide
|
C22H24BrFN4O2
|
2
|
1 |
IC50 < 15 nM
|
|
|
2 |
IC50 = 1660 nM
|
|
|
CP0659535
|
2-{[6-Methoxy-7-(2-methoxyethoxy)-4-quinazolinyl]amino}-5-methylbenzo-1,4-quinone
Show/Hide
|
C19H19N3O5
|
1
|
1 |
IC50 < 15 nM
|
|
|
CP0144564
|
(5-Phenylthiazol-2-yl)(4-pyrrolidin-1-ylmethylpyridin-2-yl)amine
Show/Hide
|
C19H20N4S
|
2
|
1 |
IC50 = 15 nM
|
|
|
2 |
IC50 = 24 nM
|
|
|
CP0146007
|
4-({2-[(5-cyano-1,3-thiazol-2-yl)amino]-3-methylpyridin-4-yl}methyl)-N-methylpiperazine-1-carboxamide
Show/Hide
|
C17H21N7OS
|
2
|
1 |
IC50 = 16 nM
|
|
|
2 |
IC50 = 38 nM
|
|
|
CP0133219
|
4-{[4-(Methylsulfonyl)piperazin-1-yl]methyl}-N-(5-phenyl-1,3-thiazol-2-yl)pyridin-2-amine
Show/Hide
|
C20H23N5O2S2
|
2
|
1 |
IC50 = 17 nM
|
|
|
2 |
IC50 = 29 nM
|
|
|
CP0092730
|
1-(2-(pyridin-4-yl)ethyl)-N-(4-(trifluoromethoxy)phenyl)-1H-pyrazole-5-carboxamide
Show/Hide
|
C18H15F3N4O2
|
1
|
1 |
IC50 = 18 nM
|
|
|
CP0074851
|
2-(6-(4-(2-morpholinoethyl)piperazin-1-yl)pyrimidin-4-ylamino)thiazole-5-carbonitrile
Show/Hide
|
C18H24N8OS
|
1
|
1 |
IC50 = 19 nM
|
|
|
CP0205190
|
(rac)-2-(6-(3-aminopyrrolidin-1-yl)pyrimidin-4-ylamino)thiazole-5-carbonitrile
Show/Hide
|
C12H13N7S
|
1
|
1 |
IC50 = 21 nM
|
|
|
CP0104347
|
N-[3-[chloro(difluoro)methoxy]phenyl]-2-(2-pyridin-4-ylethyl)pyrazole-3-carboxamide
Show/Hide
|
C18H15ClF2N4O2
|
1
|
1 |
IC50 = 21 nM
|
|
|
CP0155086
|
2-(6-(4-(2-methoxyethyl)piperazin-1-yl)pyrimidin-4-ylamino)thiazole-5-carbonitrile
Show/Hide
|
C15H19N7OS
|
1
|
1 |
IC50 = 22 nM
|
|
|
CP0074847
|
2-(6-(4-methylpiperazin-1-yl)pyrimidin-4-ylamino)thiazole-5-carbonitrile
Show/Hide
|
C13H15N7S
|
1
|
1 |
IC50 = 23 nM
|
|
|
CP0155085
|
2-(6-(4-(3-morpholinopropyl)piperazin-1-yl)pyrimidin-4-ylamino)thiazole-5-carbonitrile
Show/Hide
|
C19H26N8OS
|
1
|
1 |
IC50 = 23 nM
|
|
|
CP0038985
|
4-({2-[(5-Cyano-1,3-thiazol-2-yl)amino]-4-pyridinyl}-methyl)-1-piperazinecarboxamide
Show/Hide
|
C15H17N7OS
|
2
|
1 |
IC50 = 24 nM
|
|
|
2 |
IC50 = 47 nM
|
|
|
CP0133199
|
5-phenyl-N-[5-(pyrrolidin-1-ylmethyl)pyridin-2-yl]-1,3-thiazol-2-amine
Show/Hide
|
C19H20N4S
|
2
|
1 |
IC50 = 24 nM
|
|
|
2 |
IC50 = 28 nM
|
|
|
CP0659537
|
2-methoxy-5-{[6-methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino}benzo-1,4-quinone
Show/Hide
|
C19H19N3O6
|
1
|
1 |
IC50 = 25 nM
|
|
|
CP0162412
|
4-({2-[(5-cyano-1,3-thiazol-2-yl)amino]pyridin-4-yl}methyl)-N-methylpiperazine-1-carboxamide
Show/Hide
|
C16H19N7OS
|
2
|
1 |
IC50 = 27 nM
|
|
|
2 |
IC50 = 31 nM
|
|
|
CP0453005
|
4-{3-phenylimidazo[1,2-a]pyridin-7-yl}-1-[3-(piperidin-1-yl)propyl]-1,2-dihydropyridin-2-one
Show/Hide
|
C26H28N4O
|
1
|
1 |
IC50 = 28 nM
|
|
|
CP0104182
|
4-({2-[(5-Cyano-1,3-thiazol-2-yl)amino]-4-pyridinyl}-methyl)-N,N-dimethyl-1-piperazinecarboxamide
Show/Hide
|
C17H21N7OS
|
2
|
1 |
IC50 = 28 nM
|
|
|
2 |
IC50 = 40 nM
|
|
|
CP0104183
|
1-[4-({2-[(5-phenyl-1,3-thiazol-2-yl)amino]pyridin-4-yl}methyl)piperazin-1-yl]ethan-1-one
Show/Hide
|
C21H23N5OS
|
2
|
1 |
IC50 = 28 nM
|
|
|
2 |
IC50 = 43 nM
|
|
|
CP0339626
|
2-(4-Morpholin-4-ylmethylpyridin-2-ylamino)thiazole-5-carbonitrile
Show/Hide
|
C14H15N5OS
|
2
|
1 |
IC50 = 28 nM
|
|
|
2 |
IC50 = 43 nM
|
|
|
CP0058668
|
2-(dimethylamino)-5-[[6-methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino]cyclohexa-2,5-diene-1,4-dione
Show/Hide
|
C20H22N4O5
|
1
|
1 |
IC50 = 31 nM
|
|
|
CP0275018
|
2-({4-[(4-methanesulfonylpiperidin-1-yl)methyl]pyridin-2-yl}amino)-1,3-thiazole-5-carbonitrile
Show/Hide
|
C16H19N5O2S2
|
2
|
1 |
IC50 = 31 nM
|
|
|
2 |
IC50 = 48 nM
|
|
|
CP0046140
|
2-(6-(1,4-diazepan-1-yl)pyrimidin-4-ylamino)thiazole-5-carbonitrile
Show/Hide
|
C13H15N7S
|
1
|
1 |
IC50 = 32 nM
|
|
|
CP0104334
|
N-(4-tert-butylphenyl)-2-(2-pyridin-4-ylethyl)pyrazole-3-carboxamide
Show/Hide
|
C21H24N4O
|
1
|
1 |
IC50 = 33 nM
|
|
|
CP0046151
|
2-(6-(piperazin-1-yl)pyrimidin-4-ylamino)thiazole-5-carbonitrile
Show/Hide
|
C12H13N7S
|
1
|
1 |
IC50 = 34 nM
|
|
|
CP0144563
|
2-[(4-{[4-(2-hydroxyacetyl)piperazin-1-yl]methyl}pyridin-2-yl)amino]-1,3-thiazole-5-carbonitrile
Show/Hide
|
C16H18N6O2S
|
2
|
1 |
IC50 = 35 nM
|
|
|
2 |
IC50 = 39 nM
|
|
|
CP0141416
|
2-({4-[(4-acetylpiperazin-1-yl)methyl]pyridin-2-yl}amino)-1,3-thiazole-5-carbonitrile
Show/Hide
|
C16H18N6OS
|
2
|
1 |
IC50 = 36 nM
|
|
|
2 |
IC50 = 41 nM
|
|
|
CP0037347
|
4-(pyridin-4-ylmethylamino)-N-(3-(trifluoromethoxy)phenyl)isothiazole-3-carboxamide
Show/Hide
|
C17H13F3N4O2S
|
1
|
1 |
IC50 = 41 nM
|
|
|
CP0166793
|
2-{7-phenylimidazo[1,2-a]pyridin-3-yl}-1,3-thiazole
Show/Hide
|
C16H11N3S
|
1
|
1 |
IC50 = 42 nM
|
|
|
CP0059956
|
2-(6-(4-acetylpiperazin-1-yl)pyrimidin-4-ylamino)thiazole-5-carbonitrile
Show/Hide
|
C14H15N7OS
|
1
|
1 |
IC50 = 44 nM
|
|
|
CP0044880
|
((pyridin-4-yl)ethyl)pyridine 25
Show/Hide
|
C21H16ClF2N5O2
|
1
|
1 |
IC50 = 44 nM
|
|
|
CP0092718
|
1-(2-(pyridin-4-yl)ethyl)-N-(4-(trifluoromethyl)phenyl)-1Hpyrazole-5-carboxamide
Show/Hide
|
C18H15F3N4O
|
1
|
1 |
IC50 = 48 nM
|
|
|
CP0053328
|
2-[(pyridin-4-ylmethyl)amino]-N-(quinolin-3-yl)benzamide
Show/Hide
|
C22H18N4O
|
1
|
1 |
IC50 = 50 nM
|
|
|
CP0496664
|
4-{7-phenylimidazo[1,2-a]pyridin-3-yl}-1,2-thiazole
Show/Hide
|
C16H11N3S
|
1
|
1 |
IC50 = 50 nM
|
|
|
CP0046078
|
((pyridin-4-yl)ethyl)pyridine 26
Show/Hide
|
C21H16F3N5O2
|
1
|
1 |
IC50 = 51 nM
|
|
|
CP0509172
|
N-methyl-4-[(4-{3-phenylimidazo[1,2-a]pyridin-7-yl}phenyl)methyl]piperazine-1-carboxamide
Show/Hide
|
C26H27N5O
|
1
|
1 |
IC50 = 52 nM
|
|
|
CP0092729
|
N-(4-propan-2-ylphenyl)-2-(2-pyridin-4-ylethyl)pyrazole-3-carboxamide
Show/Hide
|
C20H22N4O
|
1
|
1 |
IC50 = 53 nM
|
|
|
CP0049078
|
4-(pyridin-4-ylmethylamino)-N-(3-(trifluoromethyl)phenyl)isothiazole-3-carboxamide
Show/Hide
|
C17H13F3N4OS
|
1
|
1 |
IC50 = 54 nM
|
|
|
CP0037353
|
N-[4-methyl-3-(trifluoromethyl)phenyl]-4-(pyridin-4-ylmethylamino)-1,2-thiazole-3-carboxamide
Show/Hide
|
C18H15F3N4OS
|
1
|
1 |
IC50 = 56 nM
|
|
|
CP0074846
|
2-(6-(4-aminopiperidin-1-yl)pyrimidin-4-ylamino)thiazole-5-carbonitrile
Show/Hide
|
C13H15N7S
|
1
|
1 |
IC50 = 59 nM
|
|
|
CP0068325
|
((pyridin-4-yl)ethyl)pyridine 19
Show/Hide
|
C24H25N5O
|
1
|
1 |
IC50 = 63 nM
|
|
|
CP0161326
|
N-(3-methoxyphenyl)-5-[3-methyl-5-(pyridin-4-ylmethylamino)imidazol-4-yl]-1,3,4-oxadiazol-2-amine
Show/Hide
|
C19H19N7O2
|
1
|
1 |
IC50 = 64 nM
|
|
|
CP0077687
|
5-(1-methyl-4-(pyridin-4-ylmethylamino)-1H-imidazol-5-yl)-N-(4-(trifluoromethoxy)phenyl)-1,3,4-oxadiazol-2-amine
Show/Hide
|
C19H16F3N7O2
|
1
|
1 |
IC50 = 66 nM
|
|
|
CP0506752
|
1-(3-{3-[(dimethylamino)methyl]piperidin-1-yl}propyl)-4-{3-phenylimidazo[1,2-a]pyridin-7-yl}-1,2-dihydropyridin-2-one
Show/Hide
|
C29H35N5O
|
1
|
1 |
IC50 = 67 nM
|
|
|
CP0498122
|
4-[(4-{3-phenylimidazo[1,2-a]pyridin-7-yl}phenyl)methyl]piperazine-1-carboxamide
Show/Hide
|
C25H25N5O
|
1
|
1 |
IC50 = 69 nM
|
|
|
CP0079002
|
3,6-diarylpyrazolo[1,5-a]pyrimidine 1
Show/Hide
|
C19H15N3O
|
1
|
1 |
IC50 = 71 nM
|
|
|
CP0172259
|
N-(4-tert-butylphenyl)-4-[2-(pyridin-4-yl)ethyl]-1,3-thiazole-5-carboxamide
Show/Hide
|
C21H23N3OS
|
1
|
1 |
IC50 = 73 nM
|
|
|
CP0154872
|
((pyridin-4-yl)ethyl)pyridine 20
Show/Hide
|
C23H23N5O
|
1
|
1 |
IC50 = 75 nM
|
|
|
CP0044879
|
((pyridin-4-yl)ethyl)pyridine 27
Show/Hide
|
C21H16F3N5O
|
1
|
1 |
IC50 = 76 nM
|
|
|
CP0508598
|
1-{4-[(4-{3-phenylimidazo[1,2-a]pyridin-7-yl}phenyl)methyl]piperazin-1-yl}ethan-1-one
Show/Hide
|
C26H26N4O
|
1
|
1 |
IC50 = 77 nM
|
|
|
CP0083122
|
2-[3-(Ethylamino)phenoxy]-5-{[6-methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino}benzo-1,4-quinone
Show/Hide
|
C26H26N4O6
|
1
|
1 |
IC50 = 78 nM
|
|
|
CP0048979
|
N-(3-tert-butylphenyl)-4-(pyridin-4-ylmethylamino)-1,2-thiazole-3-carboxamide
Show/Hide
|
C20H22N4OS
|
1
|
1 |
IC50 = 82 nM
|
|
|
CP0154766
|
5-(1-methyl-4-(pyridin-4-ylmethylamino)-1H-imidazol-5-yl)-N-(4-(trifluoromethyl)phenyl)-1,3,4-oxadiazol-2-amine
Show/Hide
|
C19H16F3N7O
|
1
|
1 |
IC50 = 82 nM
|
|
|
CP0154666
|
N-(Aryl)-thiazole-5-carboxamide 17
Show/Hide
|
C18H14ClF2N3O2S
|
1
|
1 |
IC50 = 85 nM
|
|
|
CP0176477
|
N-(4-ethylphenyl)-2-(2-pyridin-4-ylethyl)pyrazole-3-carboxamide
Show/Hide
|
C19H20N4O
|
1
|
1 |
IC50 = 86 nM
|
|
|
CP0037106
|
2-[(pyridin-4-ylmethyl)amino]-N-[3-(trifluoromethyl)phenyl]benzamide
Show/Hide
|
C20H16F3N3O
|
1
|
1 |
IC50 = 90 nM
|
|
|
CP0144490
|
N-(3,4-dimethoxyphenyl)-2-(2-pyridin-4-ylethyl)pyrazole-3-carboxamide
Show/Hide
|
C19H20N4O3
|
1
|
1 |
IC50 = 90 nM
|
|
|
CP0144613
|
N-(4-chlorophenyl)-2-(2-pyridin-4-ylethyl)pyrazole-3-carboxamide
Show/Hide
|
C17H15ClN4O
|
1
|
1 |
IC50 = 90 nM
|
|
|
CP0198306
|
((pyridin-4-yl)ethyl)pyridine 43
Show/Hide
|
C22H18F3N5O
|
1
|
1 |
IC50 = 92 nM
|
|
|
CP0154793
|
N-(3,4-dimethoxyphenyl)-5-[3-methyl-5-(pyridin-4-ylmethylamino)imidazol-4-yl]-1,3,4-oxadiazol-2-amine
Show/Hide
|
C20H21N7O3
|
1
|
1 |
IC50 = 93 nM
|
|
|
CP0187168
|
N-(3,4-dichlorophenyl)-4-[2-(pyridin-4-yl)ethyl]-1,3-thiazole-5-carboxamide
Show/Hide
|
C17H13Cl2N3OS
|
1
|
1 |
IC50 = 93 nM
|
|
|
CP0198307
|
((pyridin-4-yl)ethyl)pyridine 41
Show/Hide
|
C20H15Cl2N5O
|
1
|
1 |
IC50 = 94 nM
|
|
|
CP0081011
|
N-(4-chlorophenyl)-4-[2-(pyridin-4-yl)ethyl]-1,3-thiazole-5-carboxamide
Show/Hide
|
C17H14ClN3OS
|
1
|
1 |
IC50 = 95 nM
|
|
|
CP0156059
|
N-[3-chloro-4-(trifluoromethyl)phenyl]-2-(2-pyridin-4-ylethyl)pyrazole-3-carboxamide
Show/Hide
|
C18H14ClF3N4O
|
1
|
1 |
IC50 = 95 nM
|
|
|
CP0095083
|
N-[4-[chloro(difluoro)methoxy]phenyl]-5-[3-methyl-5-(pyridin-4-ylmethylamino)imidazol-4-yl]-1,3,4-oxadiazol-2-amine
Show/Hide
|
C19H16ClF2N7O2
|
1
|
1 |
IC50 = 96 nM
|
|
|
CP0487511
|
1-{3-[(2-methoxyethyl)(methyl)amino]propyl}-4-{3-phenylimidazo[1,2-a]pyridin-7-yl}-1,2-dihydropyridin-2-one
Show/Hide
|
C25H28N4O2
|
1
|
1 |
IC50 = 96 nM
|
|
|
CP0520350
|
3,7-diphenylimidazo[1,2-a]pyridine
Show/Hide
|
C19H14N2
|
1
|
1 |
IC50 = 98 nM
|
|
|
CP0430391
|
5-{7-phenylimidazo[1,2-a]pyridin-3-yl}-1,3-thiazole
Show/Hide
|
C16H11N3S
|
1
|
1 |
IC50 = 99 nM
|
|
|
CP0167046
|
N-[4-chloro-3-(trifluoromethyl)phenyl]-5-[3-methyl-5-(pyridin-4-ylmethylamino)imidazol-4-yl]-1,3,4-oxadiazol-2-amine
Show/Hide
|
C19H15ClF3N7O
|
1
|
1 |
IC50 = 100 nM
|
|
|
CP0057908
|
((pyridin-4-yl)ethyl)pyridine 5
Show/Hide
|
C21H16F3N5O
|
1
|
1 |
IC50 = 110 nM
|
|
|
CP0171348
|
((pyridin-4-yl)ethyl)pyridine 42
Show/Hide
|
C22H21N5O3
|
1
|
1 |
IC50 = 110 nM
|
|
|
CP0283886
|
((pyridin-4-yl)ethyl)pyridine 34
Show/Hide
|
C21H16F3N5O2
|
1
|
1 |
IC50 = 110 nM
|
|
|
CP0085415
|
2-(2-((4-Pyridyl)methyl)aminophenyl)-5-(3,4-ethylenedioxy)phenylamino-1,3,4-oxadiazole
Show/Hide
|
C22H19N5O3
|
1
|
1 |
IC50 = 110 nM
|
|
|
CP0203643
|
5-(4-methoxyphenyl)-1-phenyl-1H-1,3-benzodiazole
Show/Hide
|
C20H16N2O
|
1
|
1 |
IC50 = 113 nM
|
|
|
CP0505701
|
1-(3-hydroxypropyl)-4-{3-phenylimidazo[1,2-a]pyridin-7-yl}-1,2-dihydropyridin-2-one
Show/Hide
|
C21H19N3O2
|
1
|
1 |
IC50 = 120 nM
|
|
|
CP0166883
|
N-(Aryl)-thiazole-5-carboxamide 15
Show/Hide
|
C20H21N3OS
|
1
|
1 |
IC50 = 120 nM
|
|
|
CP0176479
|
N-(3,4-dichlorophenyl)-2-(2-pyridin-4-ylethyl)pyrazole-3-carboxamide
Show/Hide
|
C17H14Cl2N4O
|
1
|
1 |
IC50 = 120 nM
|
|
|
CP0154800
|
5-(1-methyl-4-(pyridin-4-ylmethylamino)-1H-imidazol-5-yl)-N-(3-(trifluoromethoxy)phenyl)-1,3,4-oxadiazol-2-amine
Show/Hide
|
C19H16F3N7O2
|
1
|
1 |
IC50 = 130 nM
|
|
|
CP0504761
|
4-{7-phenylimidazo[1,2-a]pyridin-3-yl}pyridine
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C18H13N3
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1
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1 |
IC50 = 145 nM
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CP0255544
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2-[[6-methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino]-5-phenoxycyclohexa-2,5-diene-1,4-dione
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C24H21N3O6
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1
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1 |
IC50 = 184 nM
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CP0776051
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2-[2-Fluoro-1-(fluoromethyl)ethoxy]-5-({6-methoxy-7-[(1-methylpiperidin-4-yl)methoxy]quinazolin-4-yl}amino)benzo-1,4-quinone
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C25H28F2N4O5
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1
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1 |
IC50 = 189 nM
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CP0083110
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N-(Aryl)-thiazole-5-carboxamide 27
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C18H13ClF3N3OS
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1
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1 |
IC50 = 190 nM
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CP0058680
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2-[[6-methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino]-5-(pyridin-3-ylmethoxy)cyclohexa-2,5-diene-1,4-dione
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C24H22N4O6
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1
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1 |
IC50 = 193 nM
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CP0922988
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2-{[6-Methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino}-5-(2-methylaziridin-1-yl)benzo-1,4-quinone
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C21H22N4O5
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1
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1 |
IC50 = 206 nM
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CP0070472
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N-(3-bromophenyl)-4-(pyridin-4-ylmethylamino)-1,2-thiazole-3-carboxamide
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C16H13BrN4OS
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1
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1 |
IC50 = 210 nM
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CP0058678
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2-(1,3-difluoropropan-2-yloxy)-5-[[6-methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino]cyclohexa-2,5-diene-1,4-dione
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C21H21F2N3O6
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1
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1 |
IC50 = 212 nM
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CP0085419
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N-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-[2-(quinolin-6-ylmethylamino)pyridin-3-yl]-1,3,4-oxadiazol-2-amine
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C25H20N6O3
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1
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1 |
IC50 = 220 nM
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CP0255372
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N-(2-fluoro-4-methylphenyl)-4-[2-(pyridin-4-yl)ethyl]-1,3-thiazole-5-carboxamide
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C18H16FN3OS
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1
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1 |
IC50 = 230 nM
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CP0533052
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2-methoxy-6-{7-phenylimidazo[1,2-a]pyridin-3-yl}pyridine
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C19H15N3O
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1
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1 |
IC50 = 242 nM
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CP0077686
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N-(3,4-dichlorophenyl)-5-[3-methyl-5-(pyridin-4-ylmethylamino)imidazol-4-yl]-1,3,4-oxadiazol-2-amine
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C18H15Cl2N7O
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1
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1 |
IC50 = 260 nM
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CP0114690
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N-(3-bromophenyl)-4-(quinolin-4-ylmethylamino)-1,2-thiazole-3-carboxamide
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C20H15BrN4OS
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1
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1 |
IC50 = 270 nM
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CP0131800
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N-(1,3-benzodioxol-5-ylmethyl)-5-[3-methyl-5-(pyridin-4-ylmethylamino)imidazol-4-yl]-1,3,4-oxadiazol-2-amine
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C20H19N7O3
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1
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1 |
IC50 = 270 nM
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CP0104348
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1-(2-(pyridin-4-yl)ethyl)-N-(3-(trifluoromethoxy)phenyl)-1H-pyrazole-5-carboxamide
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C18H15F3N4O2
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1
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1 |
IC50 = 280 nM
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CP0154933
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((pyridin-4-yl)ethyl)pyridine 44
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C22H19N5O3
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1
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1 |
IC50 = 290 nM
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CP0161222
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((pyridin-4-yl)ethyl)pyridine 38
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C21H19N5O2
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1
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1 |
IC50 = 290 nM
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CP0166949
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2-(4-imidazol-1-ylphenoxy)-5-[[6-methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino]cyclohexa-2,5-diene-1,4-dione
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C27H23N5O6
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1
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1 |
IC50 = 310 nM
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CP0428214
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2-[[6-methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino]-5-piperidin-1-ylcyclohexa-2,5-diene-1,4-dione
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C23H26N4O5
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1
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1 |
IC50 = 310 nM
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CP0154871
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((pyridin-4-yl)ethyl)pyridine 21
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C24H25N5O
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1
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1 |
IC50 = 320 nM
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CP0276881
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2-[[6-methoxy-7-[(1-methylpiperidin-4-yl)methoxy]quinazolin-4-yl]amino]-5-[2-(N-methylanilino)ethoxy]cyclohexa-2,5-diene-1,4-dione
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C31H35N5O5
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1
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1 |
IC50 = 329 nM
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CP0186425
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N-(2H-1,3-benzodioxol-5-yl)-4-[2-(pyridin-4-yl)ethyl]-1,3-thiazole-5-carboxamide
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C18H15N3O3S
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1
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1 |
IC50 = 330 nM
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CP0048988
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4-(quinolin-4-ylmethylamino)-N-(3-(trifluoromethyl)phenyl)isothiazole-3-carboxamide
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C21H15F3N4OS
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1
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1 |
IC50 = 390 nM
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CP0155091
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((pyridin-4-yl)ethyl)pyridine 22
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C23H23N5O
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1
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1 |
IC50 = 390 nM
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CP0048991
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N-(4-chlorophenyl)-4-(pyridin-4-ylmethylamino)-1,2-thiazole-3-carboxamide
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C16H13ClN4OS
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1
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1 |
IC50 = 420 nM
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CP0156055
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N-[4-chloro-3-(trifluoromethyl)phenyl]-2-(2-pyridin-4-ylethyl)pyrazole-3-carboxamide
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C18H14ClF3N4O
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1
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1 |
IC50 = 450 nM
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CP0739703
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2-{[6-Methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino}-5-(methylthio)benzo-1,4-quinone
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C19H19N3O5S
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1
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1 |
IC50 = 456 nM
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CP0287201
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3-chloro-2-methoxy-5-[[6-methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino]cyclohexa-2,5-diene-1,4-dione
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C19H18ClN3O6
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1
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1 |
IC50 = 466 nM
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CP0146175
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2-[[6-methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino]-5-propan-2-yloxycyclohexa-2,5-diene-1,4-dione
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C21H23N3O6
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1
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1 |
IC50 = 481 nM
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CP0334180
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((pyridin-4-yl)ethyl)pyridine 32
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C21H16F3N5O2
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1
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1 |
IC50 = 510 nM
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CP0257151
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((pyridin-4-yl)ethyl)pyridine 23
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C24H25N5O
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1
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1 |
IC50 = 520 nM
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CP0146720
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N-[4-chloro-3-(trifluoromethyl)phenyl]-4-(pyridin-4-ylmethylamino)-1,2-thiazole-3-carboxamide
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C17H12ClF3N4OS
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1
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1 |
IC50 = 530 nM
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CP0154935
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((pyridin-4-yl)ethyl)pyridine 28
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C21H16ClF2N5O2
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1
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1 |
IC50 = 530 nM
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CP0776052
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2-(Benzyloxy)-5-({6-methoxy-7-[(1-methylpiperidin-4-yl)methoxy]quinazolin-4-yl}amino)benzo-1,4-quinone
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C29H30N4O5
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1
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1 |
IC50 = 536 nM
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CP0140586
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N-(4-chlorophenyl)-5-[3-methyl-5-(pyridin-4-ylmethylamino)imidazol-4-yl]-1,3,4-oxadiazol-2-amine
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C18H16ClN7O
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1
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1 |
IC50 = 570 nM
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CP0205353
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N-(Aryl)-thiazole-5-carboxamide 23
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C21H22N4O2S
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1
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1 |
IC50 = 580 nM
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CP0167079
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((pyridin-4-yl)ethyl)pyridine 31
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C21H16ClF2N5O2
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1
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1 |
IC50 = 590 nM
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CP0154799
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N-(2-fluoro-4-methylphenyl)-5-[3-methyl-5-(pyridin-4-ylmethylamino)imidazol-4-yl]-1,3,4-oxadiazol-2-amine
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C19H18FN7O
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1
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1 |
IC50 = 640 nM
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CP0029006
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4-[4-[7-amino-2-(1,2,3-benzothiadiazol-7-yl)furo[2,3-c]pyridin-4-yl]pyrazol-1-yl]cyclohexan-1-ol
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C22H20N6O2S
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1
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1 |
IC50 = 650 nM
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CP0154927
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((pyridin-4-yl)ethyl)pyridine 29
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C21H16F3N5O2
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1
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1 |
IC50 = 660 nM
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CP0048977
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N-[3-methyl-4-(trifluoromethyl)phenyl]-4-(pyridin-4-ylmethylamino)-1,2-thiazole-3-carboxamide
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C18H15F3N4OS
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1
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1 |
IC50 = 710 nM
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CP0059884
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((pyridin-4-yl)ethyl)pyridine 30
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C21H16F3N5O
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1
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1 |
IC50 = 720 nM
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CP0046077
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((pyridin-4-yl)ethyl)pyridine 33
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C21H16F3N5O
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1
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1 |
IC50 = 740 nM
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CP0167080
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((pyridin-4-yl)ethyl)pyridine 36
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C21H16F3N5O2
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1
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1 |
IC50 = 760 nM
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CP0018308
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4-[4-[7-amino-2-(1,2,3-benzothiadiazol-7-yl)-3-(1,3-thiazol-5-yl)furo[2,3-c]pyridin-4-yl]pyrazol-1-yl]cyclohexan-1-ol
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C25H21N7O2S2
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1
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1 |
IC50 = 760 nM
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CP0037337
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4-(pyridin-4-ylmethylamino)-N-(4-(trifluoromethoxy)phenyl)isothiazole-3-carboxamide
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C17H13F3N4O2S
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1
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1 |
IC50 = 770 nM
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CP0070468
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4-(pyridin-4-ylmethylamino)-N-(quinolin-2-yl)isothiazole-3-carboxamide
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C19H15N5OS
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1
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1 |
IC50 = 770 nM
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CP0048983
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N-(1,3-benzodioxol-5-ylmethyl)-4-(pyridin-4-ylmethylamino)-1,2-thiazole-3-carboxamide
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C18H16N4O3S
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1
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1 |
IC50 = 790 nM
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CP0206502
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3-chloro-2-(1,3-difluoropropan-2-yloxy)-5-[[6-methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino]cyclohexa-2,5-diene-1,4-dione
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C21H20ClF2N3O6
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1
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1 |
IC50 = 792 nM
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CP0503935
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5-(2-((1H-imidazol-5-yl)methylamino)pyridin-3-yl)-N-(2,3-dihydrobenzo[b][1,4]dioxin-6-yl)-1,3,4-oxadiazol-2-amine
Show/Hide
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C19H17N7O3
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1
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1 |
IC50 = 830 nM
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CP0154895
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((pyridin-4-yl)ethyl)pyridine 35
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C21H16F3N5O2
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1
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1 |
IC50 = 860 nM
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CP0735137
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2-(2,2-Difluoroethoxy)-5-{[6-methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino}benzo-1,4-quinone
Show/Hide
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C20H19F2N3O6
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1
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1 |
IC50 = 870 nM
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CP0524550
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3-{7-phenylimidazo[1,2-a]pyridin-3-yl}pyridine
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C18H13N3
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1
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1 |
IC50 = 930 nM
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CP0465691
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3-(5-(2,3-dihydrobenzo[b][1,4]dioxin-6-ylamino)-1,3,4-oxadiazol-2-yl)-N-(pyridin-4-ylmethyl)pyridin-2-amine
Show/Hide
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C21H18N6O3
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1
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1 |
IC50 = 1000 nM
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CP0510126
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N-(pyridin-4-ylmethyl)-3-[3-[3-(trifluoromethyl)phenyl]-1H-1,2,4-triazol-5-yl]pyridin-2-amine
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C20H15F3N6
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1
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1 |
IC50 = 1000 nM
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CP0171305
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N-(4-bromophenyl)-4-[2-(pyridin-4-yl)ethyl]-1,3-thiazole-5-carboxamide
Show/Hide
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C17H14BrN3OS
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1
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1 |
IC50 = 1020 nM
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CP0070471
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N-(4-bromophenyl)-4-(pyridin-4-ylmethylamino)-1,2-thiazole-3-carboxamide
Show/Hide
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C16H13BrN4OS
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1
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1 |
IC50 = 1040 nM
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CP0154791
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N-(4-tert-butylphenyl)-5-[3-methyl-5-(pyridin-4-ylmethylamino)imidazol-4-yl]-1,3,4-oxadiazol-2-amine
Show/Hide
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C22H25N7O
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1
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1 |
IC50 = 1050 nM
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CP0144485
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1-(2-(pyridin-4-yl)ethyl)-N-(4-(trifluoromethoxy)phenyl)-1H-imidazole-2-carboxamide
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C18H15F3N4O2
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1
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1 |
IC50 = 1050 nM
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CP0037354
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N-(3,4-dichlorophenyl)-4-(pyridin-4-ylmethylamino)-1,2-thiazole-3-carboxamide
Show/Hide
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C16H12Cl2N4OS
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1
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1 |
IC50 = 1110 nM
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CP0057927
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((pyridin-4-yl)ethyl)pyridine 6
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C21H16F3N5O
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1
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1 |
IC50 = 1110 nM
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CP0037346
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N-(4-tert-butylphenyl)-4-(pyridin-4-ylmethylamino)-1,2-thiazole-3-carboxamide
Show/Hide
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C20H22N4OS
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1
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1 |
IC50 = 1150 nM
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CP0154794
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5-[3-methyl-5-(pyridin-4-ylmethylamino)imidazol-4-yl]-N-(4-propan-2-ylphenyl)-1,3,4-oxadiazol-2-amine
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C21H23N7O
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1
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1 |
IC50 = 1150 nM
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CP0092719
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1-(2-(pyridin-4-yl)ethyl)-N-(quinolin-3-yl)-1H-pyrazole-5-carboxamide
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C20H17N5O
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1
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1 |
IC50 = 1220 nM
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CP0104336
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N-(4-chlorophenyl)-1-(2-pyridin-4-ylethyl)imidazole-2-carboxamide
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C17H15ClN4O
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1
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1 |
IC50 = 1320 nM
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CP0104337
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3-methyl-1-(2-(pyridin-4-yl)ethyl)-N-(4-(trifluoromethoxy)phenyl)-1H-pyrazole-5-carboxamide
Show/Hide
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C19H17F3N4O2
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1
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1 |
IC50 = 1340 nM
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CP0138150
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4-(pyridin-4-ylmethylamino)-N-(4-(trifluoromethyl)phenyl)isothiazole-3-carboxamide
Show/Hide
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C17H13F3N4OS
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1
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1 |
IC50 = 1530 nM
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CP0144472
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2-(2-pyridin-4-yl-ethyl)-2H-pyrazole-3-carboxylic acid biphenyl-4-ylamide
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C23H20N4O
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1
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1 |
IC50 = 1560 nM
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CP0205352
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N-(4-tert-butylphenyl)-4-[2-(1,2-oxazol-4-yl)ethyl]-1,3-thiazole-5-carboxamide
Show/Hide
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C19H21N3O2S
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1
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1 |
IC50 = 1630 nM
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CP0215330
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1-(2-(pyridin-4-yl)ethyl)-N-(4-(trifluoromethyl)phenyl)-1H-imidazole-2-carboxamide
Show/Hide
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C18H15F3N4O
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1
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1 |
IC50 = 1660 nM
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CP0037344
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N-(2-fluoro-4-methylphenyl)-4-(pyridin-4-ylmethylamino)-1,2-thiazole-3-carboxamide
Show/Hide
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C17H15FN4OS
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1
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1 |
IC50 = 1890 nM
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CP0092884
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N-(4-chlorophenyl)-1-(2-pyridin-4-ylethyl)tetrazole-5-carboxamide
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C15H13ClN6O
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1
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1 |
IC50 = 2030 nM
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CP0037350
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N-[3-chloro-4-(trifluoromethyl)phenyl]-4-(pyridin-4-ylmethylamino)-1,2-thiazole-3-carboxamide
Show/Hide
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C17H12ClF3N4OS
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1
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1 |
IC50 = 2050 nM
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CP0154934
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((pyridin-4-yl)ethyl)pyridine 37
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C21H19N5O
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1
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1 |
IC50 = 2140 nM
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CP0081010
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N-(Aryl)-thiazole-5-carboxamide 16
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C16H12ClF2N3O3S
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1
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1 |
IC50 = 2250 nM
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CP0104344
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N-(4-tert-butylphenyl)-1-(2-pyridin-4-ylethyl)imidazole-2-carboxamide
Show/Hide
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C21H24N4O
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1
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1 |
IC50 = 2250 nM
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CP0171304
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N-(4-chlorophenyl)-4-[2-(1,2-oxazol-4-yl)ethyl]-1,3-thiazole-5-carboxamide
Show/Hide
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C15H12ClN3O2S
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1
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1 |
IC50 = 2300 nM
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CP0171517
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((pyridin-4-yl)ethyl)pyridine 7
Show/Hide
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C21H16F3N5O
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1
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1 |
IC50 = 2540 nM
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CP0144476
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N-(4-chlorophenyl)-5-methyl-2-(2-pyridin-4-ylethyl)pyrazole-3-carboxamide
Show/Hide
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C18H17ClN4O
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1
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1 |
IC50 = 2540 nM
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CP0186427
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N-(2-fluoro-4-methylphenyl)-4-[2-(1,2-oxazol-4-yl)ethyl]-1,3-thiazole-5-carboxamide
Show/Hide
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C16H14FN3O2S
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1
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1 |
IC50 = 2750 nM
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CP0085417
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N-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-[2-(pyridin-3-ylmethylamino)phenyl]-1H-1,2,4-triazol-3-amine
Show/Hide
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C22H20N6O2
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1
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1 |
IC50 = 2800 nM
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CP0144488
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1-(2-(pyridin-4-yl)ethyl)-N-(4-(trifluoromethyl)phenyl)-1H-tetrazole-5-carboxamide
Show/Hide
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C16H13F3N6O
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1
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1 |
IC50 = 2960 nM
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CP0039110
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1-(2-(pyridin-4-yl)ethyl)-N-(4-(trifluoromethoxy)phenyl)-1H-tetrazole-5-carboxamide
Show/Hide
|
C16H13F3N6O2
|
1
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1 |
IC50 = 2970 nM
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CP0029005
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4-(1-methylpyrazol-4-yl)-2-thieno[2,3-c]pyridin-3-ylfuro[2,3-c]pyridin-7-amine
Show/Hide
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C18H13N5OS
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1
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1 |
IC50 = 3400 nM
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CP0104335
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N-[3-chloro-4-(trifluoromethyl)phenyl]-1-(2-pyridin-4-ylethyl)imidazole-2-carboxamide
Show/Hide
|
C18H14ClF3N4O
|
1
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1 |
IC50 = 4950 nM
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CP0154792
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5-(4-(3,4-difluorobenzylamino)-1-methyl-1H-imidazol-5-yl)-N-(4-chlorophenyl)-1,3,4-oxadiazol-2-amine
Show/Hide
|
C19H15ClF2N6O
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1
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1 |
IC50 = 5650 nM
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CP0474411
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5-(2-((1H-indazol-5-yl)methylamino)phenyl)-N-(2,3-dihydrobenzo[b][1,4]dioxin-6-yl)-4H-1,2,4-triazol-3-amine
Show/Hide
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C24H21N7O2
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1
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1 |
IC50 = 7300 nM
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CP0018195
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4-[4-[7-amino-2-(1,2,3-benzothiadiazol-7-yl)-3-pyridin-3-ylfuro[2,3-c]pyridin-4-yl]pyrazol-1-yl]cyclohexan-1-ol
Show/Hide
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C27H23N7O2S
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1
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1 |
IC50 = 8200 nM
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CP0037332
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N-(3-bromophenyl)-4-(1,2-oxazol-4-ylmethylamino)-1,2-thiazole-3-carboxamide
Show/Hide
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C14H11BrN4O2S
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1
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1 |
IC50 > 10000 nM
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CP0037333
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4-(pyridin-2-ylmethylamino)-N-(3-(trifluoromethyl)phenyl)isothiazole-3-carboxamide
Show/Hide
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C17H13F3N4OS
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1
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1 |
IC50 > 10000 nM
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CP0037339
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4-(pyridin-2-ylmethylamino)-N-(4-(trifluoromethyl)phenyl)isothiazole-3-carboxamide
Show/Hide
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C17H13F3N4OS
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1
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1 |
IC50 > 10000 nM
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CP0037342
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N-(3-bromophenyl)-4-(quinolin-2-ylmethylamino)-1,2-thiazole-3-carboxamide
Show/Hide
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C20H15BrN4OS
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1
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1 |
IC50 > 10000 nM
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CP0037348
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4-(2-(benzo[d][1,3]dioxol-5-yl)ethylamino)-N-(3-bromophenyl)isothiazole-3-carboxamide
Show/Hide
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C19H16BrN3O3S
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1
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1 |
IC50 > 10000 nM
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CP0037351
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4-(pyridin-3-ylmethylamino)-N-(3-(trifluoromethyl)phenyl)isothiazole-3-carboxamide
Show/Hide
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C17H13F3N4OS
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1
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1 |
IC50 > 10000 nM
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CP0048975
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4-(pyridin-3-ylmethylamino)-N-(4-(trifluoromethyl)phenyl)isothiazole-3-carboxamide
Show/Hide
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C17H13F3N4OS
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1
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1 |
IC50 > 10000 nM
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CP0048987
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N-(2-bromophenyl)-4-(pyridin-4-ylmethylamino)-1,2-thiazole-3-carboxamide
Show/Hide
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C16H13BrN4OS
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1
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1 |
IC50 > 10000 nM
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CP0048990
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4-(3,4-difluorobenzylamino)-N-(3-(trifluoromethyl)phenyl)isothiazole-3-carboxamide
Show/Hide
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C18H12F5N3OS
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1
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1 |
IC50 > 10000 nM
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CP0147380
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4-(2-(benzo[d][1,3]dioxol-5-yl)ethylamino)-N-(3-(trifluoromethyl)phenyl)isothiazole-3-carboxamide
Show/Hide
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C20H16F3N3O3S
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1
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1 |
IC50 > 10000 nM
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CP0713299
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N-(3a,7a-dihydro-1H-indazol-5-yl)-4-(pyridin-4-ylmethylamino)isothiazole-3-carboxamide
Show/Hide
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C17H16N6OS
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1
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1 |
IC50 > 10000 nM
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CP0077684
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5-(4-((1H-indazol-5-yl)methylamino)-1-methyl-1H-imidazol-5-yl)-N-(4-chlorophenyl)-1,3,4-oxadiazol-2-amine
Show/Hide
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C20H17ClN8O
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1
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1 |
IC50 > 10000 nM
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CP0131798
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5-(4-(2-(benzo[d][1,3]dioxol-5-yl)ethylamino)-1-methyl-1H-imidazol-5-yl)-N-(4-chlorophenyl)-1,3,4-oxadiazol-2-amine
Show/Hide
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C21H19ClN6O3
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1
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1 |
IC50 > 10000 nM
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CP0154788
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N-(4-chlorophenyl)-5-[3-methyl-5-(pyridin-3-ylmethylamino)imidazol-4-yl]-1,3,4-oxadiazol-2-amine
Show/Hide
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C18H16ClN7O
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1
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1 |
IC50 > 10000 nM
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CP0154796
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N-(4-chlorophenyl)-5-[3-methyl-5-(quinolin-2-ylmethylamino)imidazol-4-yl]-1,3,4-oxadiazol-2-amine
Show/Hide
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C22H18ClN7O
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1
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1 |
IC50 > 10000 nM
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CP0161325
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N-(4-chlorophenyl)-5-[3-methyl-5-(pyridin-2-ylmethylamino)imidazol-4-yl]-1,3,4-oxadiazol-2-amine
Show/Hide
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C18H16ClN7O
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1
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1 |
IC50 > 10000 nM
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CP0166917
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N-(4-chlorophenyl)-5-[3-methyl-5-(quinolin-5-ylmethylamino)imidazol-4-yl]-1,3,4-oxadiazol-2-amine
Show/Hide
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C22H18ClN7O
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1
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1 |
IC50 > 10000 nM
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CP0044892
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((pyridin-2-yl)ethyl)pyridine 10
Show/Hide
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C21H16F3N5O
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1
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1 |
IC50 > 10000 nM
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CP0044893
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((pyridin-4-yl)ethyl)quinoline 8
Show/Hide
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C25H18F3N5O
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1
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1 |
IC50 > 10000 nM
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CP0046076
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5-{2-[2-(3,4-difluorophenyl)ethyl]pyridin-3-yl}-N-[3-(trifluoromethyl)phenyl]-1,3,4-oxadiazol-2-amine
Show/Hide
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C22H15F5N4O
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1
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1 |
IC50 > 10000 nM
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CP0046080
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((indazole)ethyl)pyridine 14
Show/Hide
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C23H17F3N6O
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1
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1 |
IC50 > 10000 nM
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CP0068322
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5-{3-[3-(2H-1,3-benzodioxol-5-yl)propyl]pyridin-4-yl}-N-[3-(trifluoromethyl)phenyl]-1,3,4-oxadiazol-2-amine
Show/Hide
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C24H19F3N4O3
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1
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1 |
IC50 > 10000 nM
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CP0140781
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((quinoline)ethyl)pyridine 16
Show/Hide
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C25H18F3N5O
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1
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1 |
IC50 > 10000 nM
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CP0171340
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5-{2-[3-(2H-1,3-benzodioxol-5-yl)propyl]pyridin-3-yl}-N-[3-(trifluoromethyl)phenyl]-1,3,4-oxadiazol-2-amine
Show/Hide
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C24H19F3N4O3
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1
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1 |
IC50 > 10000 nM
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CP0171476
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((pyridin-3-yl)ethyl)pyridine 9
Show/Hide
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C21H16F3N5O
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1
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1 |
IC50 > 10000 nM
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CP0171558
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((quinoline)ethyl)pyridine 15
Show/Hide
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C25H18F3N5O
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1
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1 |
IC50 > 10000 nM
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CP0081009
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N-(3-methylphenyl)-4-[2-(1,2-oxazol-4-yl)ethyl]-1,3-thiazole-5-carboxamide
Show/Hide
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C16H15N3O2S
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1
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1 |
IC50 > 10000 nM
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CP0083107
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N-(4-tert-butylphenyl)-4-[2-(quinolin-4-yl)ethyl]-1,3-thiazole-5-carboxamide
Show/Hide
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C25H25N3OS
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1
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1 |
IC50 > 10000 nM
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CP0166123
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N-(4-chlorophenyl)-4-[2-(quinolin-2-yl)ethyl]-1,3-thiazole-5-carboxamide
Show/Hide
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C21H16ClN3OS
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1
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1 |
IC50 > 10000 nM
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CP0166884
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4-[2-(1,2-benzoxazol-3-yl)ethyl]-N-(4-tert-butylphenyl)-1,3-thiazole-5-carboxamide
Show/Hide
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C23H23N3O2S
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1
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1 |
IC50 > 10000 nM
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CP0171307
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N-(4-tert-butylphenyl)-4-[2-(quinolin-2-yl)ethyl]-1,3-thiazole-5-carboxamide
Show/Hide
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C25H25N3OS
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1
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1 |
IC50 > 10000 nM
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CP0186423
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N-(4-chlorophenyl)-4-[2-(quinolin-4-yl)ethyl]-1,3-thiazole-5-carboxamide
Show/Hide
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C21H16ClN3OS
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1
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1 |
IC50 > 10000 nM
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CP0205354
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4-[2-(1,2-benzoxazol-3-yl)ethyl]-N-(4-chlorophenyl)-1,3-thiazole-5-carboxamide
Show/Hide
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C19H14ClN3O2S
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1
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1 |
IC50 > 10000 nM
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CP0039085
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N-(4-chlorophenyl)-2-(2-pyridin-2-ylethyl)pyrazole-3-carboxamide
Show/Hide
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C17H15ClN4O
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1
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1 |
IC50 > 10000 nM
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CP0039106
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N-(4-phenoxyphenyl)-2-(2-pyridin-4-ylethyl)pyrazole-3-carboxamide
Show/Hide
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C23H20N4O2
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1
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1 |
IC50 > 10000 nM
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CP0092725
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N-(4-chlorophenyl)-2-[2-(1,2-oxazol-4-yl)ethyl]pyrazole-3-carboxamide
Show/Hide
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C15H13ClN4O2
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1
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1 |
IC50 > 10000 nM
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CP0092726
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N-[3-chloro-4-(trifluoromethyl)phenyl]-1-(2-pyridin-4-ylethyl)benzimidazole-2-carboxamide
Show/Hide
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C22H16ClF3N4O
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1
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1 |
IC50 > 10000 nM
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CP0092887
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3,4-dimethyl-1-(2-(pyridin-4-yl)ethyl)-N-(4-(trifluoromethoxy)phenyl)-1H-pyrazole-5-carboxamide
Show/Hide
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C20H19F3N4O2
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1
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1 |
IC50 > 10000 nM
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CP0104342
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N-(4-chlorophenyl)-1-(2-pyridin-4-ylethyl)benzimidazole-2-carboxamide
Show/Hide
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C21H17ClN4O
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1
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1 |
IC50 > 10000 nM
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CP0104345
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N-(4-chlorophenyl)-1-(2-pyridin-4-ylethyl)indole-2-carboxamide
Show/Hide
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C22H18ClN3O
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1
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1 |
IC50 > 10000 nM
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CP0104346
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N-(1H-indazol-5-yl)-2-(2-pyridin-4-ylethyl)pyrazole-3-carboxamide
Show/Hide
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C18H16N6O
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1
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1 |
IC50 > 10000 nM
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CP0144468
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N-[3-chloro-4-(trifluoromethyl)phenyl]-1-(2-pyridin-4-ylethyl)tetrazole-5-carboxamide
Show/Hide
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C16H12ClF3N6O
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1
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1 |
IC50 > 10000 nM
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CP0144470
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N-(4-chlorophenyl)-4,5-dimethyl-2-(2-pyridin-4-ylethyl)pyrazole-3-carboxamide
Show/Hide
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C19H19ClN4O
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1
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1 |
IC50 > 10000 nM
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CP0144473
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1-(3,4-dimethoxyphenethyl)-N-(4-chlorophenyl)-1H-pyrazole-5-carboxamide
Show/Hide
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C20H20ClN3O3
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1
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1 |
IC50 > 10000 nM
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CP0144479
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N-(1H-indazol-6-yl)-2-(2-pyridin-4-ylethyl)pyrazole-3-carboxamide
Show/Hide
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C18H16N6O
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1
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1 |
IC50 > 10000 nM
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CP0144481
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1-(2-(benzo[d]isoxazol-3-yl)ethyl)-N-(4-chlorophenyl)-1H-pyrazole-5-carboxamide
Show/Hide
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C19H15ClN4O2
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1
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1 |
IC50 > 10000 nM
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CP0144483
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1-(3,4-difluorophenethyl)-N-(4-chlorophenyl)-1H-pyrazole-5-carboxamide
Show/Hide
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C18H14ClF2N3O
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1
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1 |
IC50 > 10000 nM
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CP0144484
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N-(4-tert-butylphenyl)-1-(2-pyridin-4-ylethyl)tetrazole-5-carboxamide
Show/Hide
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C19H22N6O
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1
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1 |
IC50 > 10000 nM
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CP0144492
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1-(2-(1H-imidazol-4-yl)ethyl)-N-(4-chlorophenyl)-1H-pyrazole-5-carboxamide
Show/Hide
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C15H14ClN5O
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1
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1 |
IC50 > 10000 nM
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CP0144495
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N-(4-chlorophenyl)-2-(2-pyridin-3-ylethyl)pyrazole-3-carboxamide
Show/Hide
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C17H15ClN4O
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1
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1 |
IC50 > 10000 nM
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CP0144498
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N-(4-phenylmethoxyphenyl)-2-(2-pyridin-4-ylethyl)pyrazole-3-carboxamide
Show/Hide
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C24H22N4O2
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1
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1 |
IC50 > 10000 nM
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CP0172690
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N-(4-chlorophenyl)-2-[2-(6-methyl-5,6-dihydro-1,3-benzodioxol-4-yl)ethyl]pyrazole-3-carboxamide
Show/Hide
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C20H20ClN3O3
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1
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1 |
IC50 > 10000 nM
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CP0210499
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1-(2-(pyridin-4-yl)ethyl)-N-(4-(trifluoromethoxy)phenyl)-1H-benzo[d]imidazole-2-carboxamide
Show/Hide
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C22H17F3N4O2
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1
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1 |
IC50 > 10000 nM
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CP0212724
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1-(2-(pyridin-4-yl)ethyl)-N-(4-(trifluoromethoxy)phenyl)-1H-indole-2-carboxamide
Show/Hide
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C23H18F3N3O2
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1
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1 |
IC50 > 10000 nM
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CP0051595
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3-(5-(2,3-dihydrobenzo[b][1,4]dioxin-6-ylamino)-1,3,4-oxadiazol-2-yl)-N-(pyridin-3-ylmethyl)pyridin-2-amine
Show/Hide
|
C21H18N6O3
|
1
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1 |
IC50 > 10000 nM
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CP0085416
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N-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-[2-(2-pyridin-3-ylethylamino)pyridin-3-yl]-1,3,4-oxadiazol-2-amine
Show/Hide
|
C22H20N6O3
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1
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1 |
IC50 > 10000 nM
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CP0085418
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N-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-[2-(quinolin-6-ylmethylamino)phenyl]-1H-1,2,4-triazol-3-amine
Show/Hide
|
C26H22N6O2
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1
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1 |
IC50 > 10000 nM
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CP0103329
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N-(2,2-difluoro-1,3-benzodioxol-5-yl)-5-[2-(pyridin-4-ylmethylamino)pyridin-3-yl]-1,3,4-oxadiazol-2-amine
Show/Hide
|
C20H14F2N6O3
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1
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1 |
IC50 > 10000 nM
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CP0218509
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5-(2-((1H-indazol-5-yl)methylamino)pyridin-3-yl)-N-(2,3-dihydrobenzo[b][1,4]dioxin-6-yl)-1,3,4-oxadiazol-2-amine
Show/Hide
|
C23H19N7O3
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1
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1 |
IC50 > 10000 nM
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CP0234933
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N-(1,4-dioxan-2-ylmethyl)-3-[3-(4-methylsulfonylphenyl)-1H-1,2,4-triazol-5-yl]pyridin-2-amine
Show/Hide
|
C19H21N5O4S
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1
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1 |
IC50 > 10000 nM
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CP0234934
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3-(5-(benzo[d][1,3]dioxol-5-ylamino)-1,3,4-oxadiazol-2-yl)-N-(pyridin-3-ylmethyl)pyridin-2-amine
Show/Hide
|
C20H16N6O3
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1
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1 |
IC50 > 10000 nM
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CP0257946
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N-(1,3-benzodioxol-5-yl)-5-[2-(1,3-benzodioxol-5-ylmethylamino)pyridin-3-yl]-1,3,4-oxadiazol-2-amine
Show/Hide
|
C22H17N5O5
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1
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1 |
IC50 > 10000 nM
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CP0297397
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N-(1H-pyrazol-4-ylmethyl)-3-[3-[3-(trifluoromethyl)phenyl]-1H-1,2,4-triazol-5-yl]pyridin-2-amine
Show/Hide
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C18H14F3N7
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1
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1 |
IC50 > 10000 nM
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CP0297398
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N-(pyridin-4-ylmethyl)-3-[5-[3-(trifluoromethyl)phenyl]-1,3,4-oxadiazol-2-yl]pyridin-2-amine
Show/Hide
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C20H14F3N5O
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1
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1 |
IC50 > 10000 nM
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CP0297399
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N-(1,3-benzodioxol-5-yl)-5-[2-(2-pyridin-4-ylethylamino)pyridin-3-yl]-1,3,4-oxadiazol-2-amine
Show/Hide
|
C21H18N6O3
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1
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1 |
IC50 > 10000 nM
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CP0297400
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N-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-[2-(pyridin-4-ylmethylamino)phenyl]-1H-1,2,4-triazol-3-amine
Show/Hide
|
C22H20N6O2
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1
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1 |
IC50 > 10000 nM
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CP0297660
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2-(2-((4-Pyridyl)methyl)aminophenyl)-5-(3,4-methylenedioxy)phenylamino-1,3,4-oxadiazole
Show/Hide
|
C21H17N5O3
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1
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1 |
IC50 > 10000 nM
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CP0297661
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3-(5-(benzo[d][1,3]dioxol-5-ylamino)-1,3,4-oxadiazol-2-yl)-N-(pyridin-2-ylmethyl)pyridin-2-amine
Show/Hide
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C20H16N6O3
|
1
|
1 |
IC50 > 10000 nM
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CP0297662
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5-[2-(1,3-benzodioxol-5-ylmethylamino)pyridin-3-yl]-N-(2,3-dihydro-1,4-benzodioxin-6-yl)-1,3,4-oxadiazol-2-amine
Show/Hide
|
C23H19N5O5
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1
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1 |
IC50 > 10000 nM
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CP0297665
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5-(2-((1H-imidazol-5-yl)methylamino)phenyl)-N-(2,3-dihydrobenzo[b][1,4]dioxin-6-yl)-4H-1,2,4-triazol-3-amine
Show/Hide
|
C20H19N7O2
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1
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1 |
IC50 > 10000 nM
|
|
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CP0307728
|
3-(5-(benzo[d][1,3]dioxol-5-yl)-4H-1,2,4-triazol-3-yl)-N-(pyridin-4-ylmethyl)pyridin-2-amine
Show/Hide
|
C20H16N6O2
|
1
|
1 |
IC50 > 10000 nM
|
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CP0313290
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N-(1,3-benzodioxol-5-yl)-5-[2-(2-pyridin-3-ylethylamino)pyridin-3-yl]-1,3,4-oxadiazol-2-amine
Show/Hide
|
C21H18N6O3
|
1
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1 |
IC50 > 10000 nM
|
|
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CP0313292
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N-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-[2-(2-pyridin-4-ylethylamino)pyridin-3-yl]-1,3,4-oxadiazol-2-amine
Show/Hide
|
C22H20N6O3
|
1
|
1 |
IC50 > 10000 nM
|
|
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CP0321542
|
3-(5-(benzo[d][1,3]dioxol-5-ylamino)-1,3,4-oxadiazol-2-yl)-N-(pyridin-4-ylmethyl)pyridin-2-amine
Show/Hide
|
C20H16N6O3
|
1
|
1 |
IC50 > 10000 nM
|
|
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CP0543671
|
3-(5-(2,3-dihydrobenzo[b][1,4]dioxin-6-ylamino)-1,3,4-oxadiazol-2-yl)-N-(pyridin-2-ylmethyl)pyridin-2-amine
Show/Hide
|
C21H18N6O3
|
1
|
1 |
IC50 > 10000 nM
|
|
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CP0017901
|
4-[4-[7-amino-2-(1,2,3-benzothiadiazol-7-yl)-3-(fluoromethyl)furo[2,3-c]pyridin-4-yl]pyrazol-1-yl]cyclohexan-1-ol
Show/Hide
|
C23H21FN6O2S
|
1
|
1 |
IC50 = 18300 nM
|
|
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CP0031772
|
4-(1,5-dimethylpyrazol-4-yl)-2-thieno[2,3-c]pyridin-3-ylfuro[2,3-c]pyridin-7-amine
Show/Hide
|
C19H15N5OS
|
1
|
1 |
IC50 = 19900 nM
|
|
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CP0018196
|
4-[4-[7-amino-2-(1,2,3-benzothiadiazol-7-yl)-3-(difluoromethyl)furo[2,3-c]pyridin-4-yl]pyrazol-1-yl]cyclohexan-1-ol
Show/Hide
|
C23H20F2N6O2S
|
1
|
1 |
IC50 > 20000 nM
|
|
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CP0018592
|
4-[4-[7-amino-2-(1,2,3-benzothiadiazol-7-yl)-3-chlorofuro[2,3-c]pyridin-4-yl]pyrazol-1-yl]cyclohexan-1-ol
Show/Hide
|
C22H19ClN6O2S
|
1
|
1 |
IC50 > 20000 nM
|
|
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CP0025123
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7-amino-2-(1,2,3-benzothiadiazol-7-yl)-4-[1-(4-hydroxycyclohexyl)pyrazol-4-yl]furo[2,3-c]pyridine-3-carbonitrile
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C23H19N7O2S
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1
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1 |
IC50 > 20000 nM
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CP0031773
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4-(1,3-dimethylpyrazol-4-yl)-2-thieno[2,3-c]pyridin-3-ylfuro[2,3-c]pyridin-7-amine
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C19H15N5OS
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1
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1 |
IC50 > 20000 nM
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CP0031774
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4-(3-methoxy-1-methylpyrazol-4-yl)-2-thieno[2,3-c]pyridin-3-ylfuro[2,3-c]pyridin-7-amine
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C19H15N5O2S
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1
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1 |
IC50 > 20000 nM
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CP0058676
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2-(4-benzylpiperazin-1-yl)-5-[[6-methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino]cyclohexa-2,5-diene-1,4-dione
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C29H31N5O5
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1
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1 |
IC50 > 1000 nM
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CP0058682
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2-[(4-fluorophenyl)methoxy]-5-[[6-methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino]cyclohexa-2,5-diene-1,4-dione
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C25H22FN3O6
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1
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1 |
IC50 > 1000 nM
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CP0146169
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2-[[6-methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino]-5-morpholin-4-ylcyclohexa-2,5-diene-1,4-dione
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C22H24N4O6
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1
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1 |
IC50 > 1000 nM
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CP0154729
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2-chloro-5-[[6-methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino]cyclohexa-2,5-diene-1,4-dione
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C18H16ClN3O5
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1
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1 |
IC50 > 1000 nM
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CP0166952
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3-Chloro-2-ethoxy-5-{[6-methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino}benzo-1,4-quinone
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C20H20ClN3O6
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1
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1 |
IC50 > 1000 nM
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CP0206503
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2-[[6-methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino]-5-(2,2,2-trifluoro-1-phenylethoxy)cyclohexa-2,5-diene-1,4-dione
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C26H22F3N3O6
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1
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1 |
IC50 > 1000 nM
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CP0212509
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2-Ethoxy-5-{[6-methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino}benzo-1,4-quinone
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C20H21N3O6
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1
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1 |
IC50 > 1000 nM
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CP0250096
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2-(4-Ethylpiperazin-1-yl)-5-{[6-methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino}benzo-1,4-quinone
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C24H29N5O5
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1
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1 |
IC50 > 1000 nM
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CP0309154
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2-[[6-methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino]cyclohexa-2,5-diene-1,4-dione
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C18H17N3O5
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1
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1 |
IC50 > 1000 nM
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CP0659536
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2-{[6-Methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino}-5-[methyl(phenyl) amino] benzo-1,4-quinon
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C25H24N4O5
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1
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1 |
IC50 > 1000 nM
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CP0659539
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2-{[6-Methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino}-5-(2-phenoxyethoxy)benzo-1,4-quinone
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C26H25N3O7
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1
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1 |
IC50 > 1000 nM
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CP0704450
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2-{[-6-methoxy-7-(2-methoxyethoxy)quinazolin-4-yl]amino}-5-(5-methyl-2-oxo-1,3-oxazolidin-3-yl)benzo-1,4-quinone
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C22H22N4O7
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1
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1 |
IC50 > 1000 nM
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CP0113988
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CEP-32496
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C24H22F3N5O5
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1
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1 |
Kd = 8 nM
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