Compound ID |
Compound Name |
Compound Formula |
CP0391607
|
US10047092, 13
Show/Hide
|
C17H14Cl2N6O
|
1
|
1 |
Ki = 1.4 nM
|
|
|
CP0484511
|
US10047092, 21
Show/Hide
|
C17H13ClF3N5O2
|
1
|
1 |
Ki = 1.4 nM
|
|
|
CP0056677
|
US10047092, 16
Show/Hide
|
C18H14ClF3N6O
|
1
|
1 |
Ki = 1.6 nM
|
|
|
CP0385599
|
BDBM160086
Show/Hide
|
C18H14ClF3N6O
|
1
|
1 |
Ki = 2 nM
|
|
|
CP0417275
|
US10047092, 32
Show/Hide
|
C17H13ClF3N5OS
|
1
|
1 |
Ki = 2 nM
|
|
|
CP0419739
|
US10047092, 35
Show/Hide
|
C20H17ClF3N5O2
|
1
|
1 |
Ki = 2 nM
|
|
|
CP0541424
|
US10047092, 37
Show/Hide
|
C17H13ClF3N5OS
|
1
|
1 |
Ki = 2 nM
|
|
|
CP0380496
|
US10047092, 76
Show/Hide
|
C20H16ClF4N5O
|
1
|
1 |
Ki = 2.5 nM
|
|
|
CP0381007
|
US10047092, 30
Show/Hide
|
C19H14ClF4N5O
|
1
|
1 |
Ki = 2.5 nM
|
|
|
CP0384906
|
US10047092, 34
Show/Hide
|
C18H13ClF4N6O
|
1
|
1 |
Ki = 2.5 nM
|
|
|
CP0512552
|
US10047092, 11
Show/Hide
|
C17H14Cl2N6O
|
1
|
1 |
Ki = 2.5 nM
|
|
|
CP0403649
|
US10047092, 75
Show/Hide
|
C19H15ClF4N6O
|
1
|
1 |
Ki = 3.2 nM
|
|
|
CP0408299
|
US10047092, 23
Show/Hide
|
C18H16ClF3N6O
|
1
|
1 |
Ki = 3.2 nM
|
|
|
CP0422528
|
US10047092, 63
Show/Hide
|
C20H16ClF3N6O
|
1
|
1 |
Ki = 3.2 nM
|
|
|
CP0429645
|
US10047092, 19
Show/Hide
|
C19H16ClF3N6O
|
1
|
1 |
Ki = 3.2 nM
|
|
|
CP0846069
|
US9040534, 28
Show/Hide
|
C17H14ClF3N6O
|
1
|
1 |
Ki = 3.2 nM
|
|
|
CP0877279
|
US9040534, 26
Show/Hide
|
C18H16ClF3N6O
|
1
|
1 |
Ki = 3.2 nM
|
|
|
CP0385598
|
US10047092, 29
Show/Hide
|
C19H15ClF3N5O
|
1
|
1 |
Ki = 4 nM
|
|
|
CP0397177
|
US10047092, 14
Show/Hide
|
C18H14ClF3N6O
|
1
|
1 |
Ki = 4 nM
|
|
|
CP0407689
|
US10047092, 20
Show/Hide
|
C17H13ClF3N5O2
|
1
|
1 |
Ki = 4 nM
|
|
|
CP0508728
|
US10047092, 31
Show/Hide
|
C17H13ClF3N5OS
|
1
|
1 |
Ki = 4 nM
|
|
|
CP0880953
|
US9040534, 68
Show/Hide
|
C19H16ClF3N6O
|
1
|
1 |
Ki = 4 nM
|
|
|
CP0472424
|
US10053462, 61
Show/Hide
|
C19H14ClF3N4OS
|
1
|
1 |
Ki = 4 nM
|
|
|
CP0385042
|
US10047092, 18
Show/Hide
|
C19H15ClF3N5O
|
1
|
1 |
Ki = 5 nM
|
|
|
CP0385597
|
US10047092, 33
Show/Hide
|
C18H14ClF3N6O
|
1
|
1 |
Ki = 5 nM
|
|
|
CP0385625
|
US10047092, 85
Show/Hide
|
C19H17F3N6O
|
1
|
1 |
Ki = 5 nM
|
|
|
CP0427095
|
US10047092, 66
Show/Hide
|
C20H16ClF3N6O
|
1
|
1 |
Ki = 5 nM
|
|
|
CP0456896
|
US10047092, 88
Show/Hide
|
C18H15F3N6O
|
1
|
1 |
Ki = 5 nM
|
|
|
CP0389368
|
US10047092, 64
Show/Hide
|
C20H16ClF3N6O
|
1
|
1 |
Ki = 6.3 nM
|
|
|
CP0416388
|
US10047092, 56
Show/Hide
|
C19H14Cl2F3N5O
|
1
|
1 |
Ki = 6.3 nM
|
|
|
CP0460008
|
US10047092, 22
Show/Hide
|
C17H13ClF3N5O2
|
1
|
1 |
Ki = 6.3 nM
|
|
|
CP0527398
|
US10047092, 45
Show/Hide
|
C19H14ClF4N5O
|
1
|
1 |
Ki = 6.3 nM
|
|
|
CP0539442
|
US10047092, 3
Show/Hide
|
C17H12ClF3N6O
|
1
|
1 |
Ki = 6.3 nM
|
|
|
CP0931107
|
US9096596, 75
Show/Hide
|
C20H17F4N5O
|
1
|
1 |
Ki = 6.3 nM
|
|
|
CP0945719
|
US9102686, 62
Show/Hide
|
C19H15ClF3N5O
|
1
|
1 |
Ki = 6.3 nM
|
|
|
CP0375375
|
US10047092, 17
Show/Hide
|
C20H15ClF4N4O
|
1
|
1 |
Ki = 7.9 nM
|
|
|
CP0389315
|
US10047092, 61
Show/Hide
|
C20H16ClF3N6O
|
1
|
1 |
Ki = 7.9 nM
|
|
|
CP0403042
|
US10047092, 70
Show/Hide
|
C20H15ClF4N6O
|
1
|
1 |
Ki = 7.9 nM
|
|
|
CP0407144
|
US10047092, 52
Show/Hide
|
C19H14Cl2F3N5O
|
1
|
1 |
Ki = 7.9 nM
|
|
|
CP0524290
|
US10047092, 42
Show/Hide
|
C18H13BrClF3N6O
|
1
|
1 |
Ki = 7.9 nM
|
|
|
CP0546701
|
US10047092, 67
Show/Hide
|
C21H17ClF3N5O
|
1
|
1 |
Ki = 7.9 nM
|
|
|
CP0863315
|
US9096596, 78
Show/Hide
|
C21H20F3N5O
|
1
|
1 |
Ki = 7.9 nM
|
|
|
CP0896590
|
US9096596, 113
Show/Hide
|
C19H15ClF3N5O
|
1
|
1 |
Ki = 7.9 nM
|
|
|
CP0935337
|
US9096596, 81
Show/Hide
|
C19H16Cl2FN5O
|
1
|
1 |
Ki = 7.9 nM
|
|
|
CP0462829
|
US10047092, 54
Show/Hide
|
C19H13ClF6N6O
|
1
|
1 |
Ki = 10 nM
|
|
|
CP0513238
|
US10047092, 9
Show/Hide
|
C18H13ClF3N5O
|
1
|
1 |
Ki = 10 nM
|
|
|
CP0860077
|
US9040534, 74
Show/Hide
|
C18H16ClF3N6O
|
1
|
1 |
Ki = 10 nM
|
|
|
CP0903792
|
US9096596, 84
Show/Hide
|
C19H17Cl2N5O
|
1
|
1 |
Ki = 10 nM
|
|
|
CP0388923
|
US10053462, 47
Show/Hide
|
C18H13Cl2FN6O
|
1
|
1 |
Ki = 10 nM
|
|
|
CP0407681
|
US10053462, 8
Show/Hide
|
C19H15ClF3N5OS
|
1
|
1 |
Ki = 10 nM
|
|
|
CP0470360
|
US10053462, 58
Show/Hide
|
C19H14ClF3N4OS
|
1
|
1 |
Ki = 10 nM
|
|
|
CP0400904
|
US10053462, 33
Show/Hide
|
C21H17ClF3N5O
|
1
|
1 |
Ki = 10.5 nM
|
|
|
CP0414577
|
US10053462, 36
Show/Hide
|
C19H15ClF3N5OS
|
1
|
1 |
Ki = 10.7 nM
|
|
|
CP0863273
|
US9096596, 89
Show/Hide
|
C19H17ClFN5O
|
1
|
1 |
Ki = 11.5 nM
|
|
|
CP0409905
|
US10047092, 73
Show/Hide
|
C20H17ClF3N5O
|
1
|
1 |
Ki = 12.6 nM
|
|
|
CP0420025
|
US10047092, 41
Show/Hide
|
C17H13ClF3N5O2
|
1
|
1 |
Ki = 12.6 nM
|
|
|
CP0434339
|
US10047092, 46
Show/Hide
|
C20H17ClF3N5O
|
1
|
1 |
Ki = 12.6 nM
|
|
|
CP0462711
|
US10047092, 48
Show/Hide
|
C20H17ClF3N5O
|
1
|
1 |
Ki = 12.6 nM
|
|
|
CP0509221
|
US10323032, Example 109
Show/Hide
|
C17H12ClF3N6O
|
1
|
1 |
Ki = 12.6 nM
|
|
|
CP0850616
|
US9096596, 118
Show/Hide
|
C18H14Cl2FN5O
|
1
|
1 |
Ki = 12.6 nM
|
|
|
CP0866477
|
US9096596, 119
Show/Hide
|
C18H14Cl2FN5O
|
1
|
1 |
Ki = 12.6 nM
|
|
|
CP0866681
|
US9096596, 71
Show/Hide
|
C19H16Cl2FN5O
|
1
|
1 |
Ki = 12.6 nM
|
|
|
CP0894646
|
US9096596, 67
Show/Hide
|
C19H17Cl2N5O
|
1
|
1 |
Ki = 12.6 nM
|
|
|
CP0384797
|
US10053462, 41
Show/Hide
|
C20H15ClF3N5O
|
1
|
1 |
Ki = 12.6 nM
|
|
|
CP0385435
|
US10053462, 7
Show/Hide
|
C19H15ClF3N5OS
|
1
|
1 |
Ki = 12.6 nM
|
|
|
CP0385779
|
US10053462, 44
Show/Hide
|
C21H18F3N5O
|
1
|
1 |
Ki = 12.6 nM
|
|
|
CP0396418
|
US10053462, 12
Show/Hide
|
C21H16ClF4N5O
|
1
|
1 |
Ki = 12.6 nM
|
|
|
CP0407607
|
US10053462, 45
Show/Hide
|
C20H14ClF4N5O
|
1
|
1 |
Ki = 12.6 nM
|
|
|
CP0414717
|
US10053462, 42
Show/Hide
|
C19H14ClF3N6O
|
1
|
1 |
Ki = 12.6 nM
|
|
|
CP0425425
|
US10053462, 5
Show/Hide
|
C22H17ClF4N4O
|
1
|
1 |
Ki = 12.6 nM
|
|
|
CP0456491
|
US10053462, 53
Show/Hide
|
C19H16F3N5OS
|
1
|
1 |
Ki = 12.6 nM
|
|
|
CP0422523
|
US10053462, 43
Show/Hide
|
C20H14ClF4N5O
|
1
|
1 |
Ki = 12.9 nM
|
|
|
CP0468095
|
US10053462, 18
Show/Hide
|
C20H15ClF4N6O
|
1
|
1 |
Ki = 13.8 nM
|
|
|
CP0411939
|
US10047092, 94
Show/Hide
|
C18H18N6O
|
1
|
1 |
Ki = 14.1 nM
|
|
|
CP0407563
|
US10323032, Example 7
Show/Hide
|
C17H13Cl2N5O
|
1
|
1 |
Ki = 15.4 nM
|
|
|
CP0389346
|
US10047092, 47
Show/Hide
|
C19H15ClF3N5O
|
1
|
1 |
Ki = 15.8 nM
|
|
|
CP0434796
|
US10047092, 78
Show/Hide
|
C17H14ClFN6O
|
1
|
1 |
Ki = 15.8 nM
|
|
|
CP0868205
|
US9096596, 68
Show/Hide
|
C19H17Cl2N5O
|
1
|
1 |
Ki = 15.8 nM
|
|
|
CP0879023
|
US9096596, 58
Show/Hide
|
C20H17ClF3N5O
|
1
|
1 |
Ki = 15.8 nM
|
|
|
CP0420624
|
US10053462, 50
Show/Hide
|
C19H13ClF4N6O
|
1
|
1 |
Ki = 15.8 nM
|
|
|
CP0541397
|
US10053462, 46
Show/Hide
|
C19H14ClF3N6O
|
1
|
1 |
Ki = 15.8 nM
|
|
|
CP0403398
|
US10323032, Example 33
Show/Hide
|
C19H15ClF3N5O
|
1
|
1 |
Ki = 16.4 nM
|
|
|
CP0861656
|
US9096596, 99
Show/Hide
|
C21H19ClF3N5O
|
1
|
1 |
Ki = 17.4 nM
|
|
|
CP0515335
|
US10053462, 14
Show/Hide
|
C21H17ClF3N5O
|
1
|
1 |
Ki = 17.4 nM
|
|
|
CP0470140
|
US10323032, Example 55
Show/Hide
|
C18H14ClF3N6O
|
1
|
1 |
Ki = 17.8 nM
|
|
|
CP0408165
|
US10047092, 40
Show/Hide
|
C18H15ClF3N5OS
|
1
|
1 |
Ki = 20 nM
|
|
|
CP0469293
|
US10047092, 8
Show/Hide
|
C17H13Cl2N5O
|
1
|
1 |
Ki = 20 nM
|
|
|
CP0469296
|
US10323032, Example 18
Show/Hide
|
C18H13ClF3N5O
|
1
|
1 |
Ki = 20 nM
|
|
|
CP0880632
|
US9096596, 122
Show/Hide
|
C18H14Cl2FN5O
|
1
|
1 |
Ki = 20 nM
|
|
|
CP0902249
|
US9096596, 102
Show/Hide
|
C22H21ClF3N5O
|
1
|
1 |
Ki = 20 nM
|
|
|
CP0902265
|
US9096596, 121
Show/Hide
|
C18H14Cl2FN5O
|
1
|
1 |
Ki = 20 nM
|
|
|
CP0397123
|
US10053462, 49
Show/Hide
|
C18H13ClF3N5OS
|
1
|
1 |
Ki = 20 nM
|
|
|
CP0491218
|
US10053462, 4
Show/Hide
|
C22H17ClF4N4O
|
1
|
1 |
Ki = 20 nM
|
|
|
CP0407608
|
US10053462, 40
Show/Hide
|
C21H15ClF4N4O
|
1
|
1 |
Ki = 21.9 nM
|
|
|
CP0408243
|
US10053462, 60
Show/Hide
|
C18H12Cl2F3N5OS
|
1
|
1 |
Ki = 21.9 nM
|
|
|
CP0913936
|
US9096596, 63
Show/Hide
|
C19H16ClF3N6O
|
1
|
1 |
Ki = 22.4 nM
|
|
|
CP0473488
|
US10053462, 23
Show/Hide
|
C22H19ClF3N5O
|
1
|
1 |
Ki = 24 nM
|
|
|
CP0456513
|
US10047092, 24
Show/Hide
|
C18H16ClF3N6O
|
1
|
1 |
Ki = 25.1 nM
|
|
|
CP0540780
|
US10047092, 36
Show/Hide
|
C18H15ClF3N5OS
|
1
|
1 |
Ki = 25.1 nM
|
|
|
CP0865045
|
US9040534, 25
Show/Hide
|
C17H14ClF3N6O
|
1
|
1 |
Ki = 25.1 nM
|
|
|
CP0385544
|
US10323032, Example 124
Show/Hide
|
C22H20ClF4N5O
|
1
|
1 |
Ki = 25.1 nM
|
|
|
CP0420230
|
US10323032, Example 19
Show/Hide
|
C19H15ClF3N5O
|
1
|
1 |
Ki = 25.1 nM
|
|
|
CP0440539
|
US10323032, Example 20
Show/Hide
|
C17H12Cl2FN5O
|
1
|
1 |
Ki = 25.1 nM
|
|
|
CP0860052
|
US9096596, 91
Show/Hide
|
C19H17ClFN5O
|
1
|
1 |
Ki = 25.1 nM
|
|
|
CP0861884
|
US9096596, 112
Show/Hide
|
C19H15ClF3N5O
|
1
|
1 |
Ki = 25.1 nM
|
|
|
CP0874169
|
US9096596, 74
Show/Hide
|
C20H17F4N5O
|
1
|
1 |
Ki = 25.1 nM
|
|
|
CP0892017
|
US9096596, 80
Show/Hide
|
C19H16Cl2FN5O
|
1
|
1 |
Ki = 25.1 nM
|
|
|
CP0911517
|
US9096596, 62
Show/Hide
|
C19H15ClF3N5O
|
1
|
1 |
Ki = 25.1 nM
|
|
|
CP0420629
|
US10053462, 39
Show/Hide
|
C20H17ClF3N5OS
|
1
|
1 |
Ki = 25.1 nM
|
|
|
CP0474346
|
US10053462, 55
Show/Hide
|
C19H13Cl2F3N4OS
|
1
|
1 |
Ki = 25.1 nM
|
|
|
CP0487012
|
US10053462, 54
Show/Hide
|
C17H12Cl2FN5OS
|
1
|
1 |
Ki = 25.1 nM
|
|
|
CP0385693
|
US10047092, 39
Show/Hide
|
C19H17ClF3N5OS
|
1
|
1 |
Ki = 27.5 nM
|
|
|
CP0414124
|
US10047092, 2
Show/Hide
|
C16H12Cl2N6O
|
1
|
1 |
Ki = 28.8 nM
|
|
|
CP0524252
|
US10053462, 26
Show/Hide
|
C22H19ClF3N5O2
|
1
|
1 |
Ki = 30.4 nM
|
|
|
CP0385144
|
US10323032, Example 10
Show/Hide
|
C19H16F3N5O
|
1
|
1 |
Ki = 30.9 nM
|
|
|
CP0385776
|
US10047092, 92
Show/Hide
|
C18H18N6O
|
1
|
1 |
Ki = 31.6 nM
|
|
|
CP0407605
|
US10047092, 69
Show/Hide
|
C21H16ClF4N5O
|
1
|
1 |
Ki = 31.6 nM
|
|
|
CP0509249
|
US10047092, 87
Show/Hide
|
C19H20N6O
|
1
|
1 |
Ki = 31.6 nM
|
|
|
CP0531138
|
US10047092, 80
Show/Hide
|
C17H15ClN6O
|
1
|
1 |
Ki = 31.6 nM
|
|
|
CP0487017
|
US10323032, Example 128
Show/Hide
|
C23H23ClF3N5O2
|
1
|
1 |
Ki = 31.6 nM
|
|
|
CP0850480
|
US9096596, 77
Show/Hide
|
C21H20F3N5O
|
1
|
1 |
Ki = 31.6 nM
|
|
|
CP0852696
|
US9096596, 87
Show/Hide
|
C19H17ClFN5O
|
1
|
1 |
Ki = 31.6 nM
|
|
|
CP0867838
|
US9096596, 95
Show/Hide
|
C19H17F2N5O
|
1
|
1 |
Ki = 31.6 nM
|
|
|
CP0869093
|
US9096596, 116
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C19H14ClF4N5O
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1
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1 |
Ki = 31.6 nM
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CP0880918
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US9096596, 115
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C19H14ClF4N5O
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1
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1 |
Ki = 31.6 nM
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CP0895816
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US9096596, 83
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C19H17Cl2N5O
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1
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1 |
Ki = 31.6 nM
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CP0407838
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US10053462, 52
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C18H12ClF4N5OS
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1
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1 |
Ki = 31.6 nM
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CP0389387
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US10053462, 57
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C18H13ClF3N5OS
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1
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1 |
Ki = 35.5 nM
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CP0472506
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US10053462, 30
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C21H16Cl2F3N5O
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1
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1 |
Ki = 35.5 nM
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CP0417817
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US10323032, Example 11
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C19H14Cl2N4O
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1
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1 |
Ki = 37.2 nM
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CP0846324
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US9096596, 56
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C20H17ClF3N5O
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1
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1 |
Ki = 37.2 nM
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CP0375674
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US10323032, Example 129
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C19H12Cl2F2N4O
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1
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1 |
Ki = 39.8 nM
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CP0403429
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US10323032, Example 21
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C17H13ClFN5O
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1
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1 |
Ki = 39.8 nM
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CP0406949
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US10323032, Example 35
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C19H14ClF4N5O
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1
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1 |
Ki = 39.8 nM
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CP0407229
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US10323032, Example 47
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C18H14ClF3N6O
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1
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1 |
Ki = 39.8 nM
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CP0861572
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US9096596, 70
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C19H16Cl2FN5O
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1
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1 |
Ki = 39.8 nM
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CP0863311
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US9096596, 104
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C20H18Cl2FN5O
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1
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1 |
Ki = 39.8 nM
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CP0375035
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US10053462, 3
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C20H16ClF3N6O
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1
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1 |
Ki = 39.8 nM
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CP0407675
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US10053462, 48
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C20H15ClF3N5O
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1
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1 |
Ki = 39.8 nM
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CP0456469
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US10053462, 56
Show/Hide
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C19H15ClF3N5OS
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1
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1 |
Ki = 39.8 nM
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CP0863244
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US9102686, 51
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C19H16ClF3N6O
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1
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1 |
Ki = 39.8 nM
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CP0546809
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US10047092, 57
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C20H17ClF3N5O
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1
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1 |
Ki = 50.1 nM
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CP0388932
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US10323032, Example 39
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C20H14ClF6N5O
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1
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1 |
Ki = 50.1 nM
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CP0403003
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US10323032, Example 43
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C18H12ClF3N4OS
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1
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1 |
Ki = 50.1 nM
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CP0524278
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US10323032, Example 37
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C18H12ClF3N4OS
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1
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1 |
Ki = 50.1 nM
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CP0544596
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US10323032, Example 111
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C18H13F4N5O
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1
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1 |
Ki = 50.1 nM
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CP0690977
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US9096596, 66
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C20H16ClF4N5O
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1
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1 |
Ki = 50.1 nM
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CP0375684
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US10053462, 1
Show/Hide
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C20H16ClF3N6O
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1
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1 |
Ki = 50.1 nM
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CP0411350
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US10053462, 21
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C19H15Cl2FN6O
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1
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1 |
Ki = 50.1 nM
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CP0848326
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US9096596, 98
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C21H19ClF3N5O
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1
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1 |
Ki = 55 nM
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CP0305154
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US10323032, Example 12
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C20H14ClF3N4O
|
1
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1 |
Ki = 58.9 nM
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CP0425315
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US10047092, 86
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C17H14Cl2N6O
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1
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1 |
Ki = 63.1 nM
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CP0457552
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US10047092, 82
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C18H17ClN6O3S
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1
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1 |
Ki = 63.1 nM
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CP0474497
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US10047092, 1
Show/Hide
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C19H13ClF4N4O
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1
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1 |
Ki = 63.1 nM
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CP0385845
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US10323032, Example 14
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C18H13Cl2N5O
|
1
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1 |
Ki = 63.1 nM
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CP0396423
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US10323032, Example 44
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C19H14ClF3N4OS
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1
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1 |
Ki = 63.1 nM
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CP0403490
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US10323032, Example 57
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C21H17ClF3N5O
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1
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1 |
Ki = 63.1 nM
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CP0409865
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US10323032, Example 53
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C18H14Cl2FN5O
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1
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1 |
Ki = 63.1 nM
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CP0411397
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US10323032, Example 34
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C18H15Cl2N5O
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1
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1 |
Ki = 63.1 nM
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CP0435051
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US10323032, Example 130
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C20H13ClF4N4O
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1
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1 |
Ki = 63.1 nM
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CP0382526
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US10323032, Example 38
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C17H12Cl2N4OS
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1
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1 |
Ki = 77.6 nM
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CP0382104
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US10323032, Example 42
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C19H14ClF3N4O
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1
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1 |
Ki = 79.4 nM
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CP0409841
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US10323032, Example 60
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C19H12ClF6N5O
|
1
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1 |
Ki = 79.4 nM
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CP0462690
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US10323032, Example 15
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C20H16F3N5O
|
1
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1 |
Ki = 79.4 nM
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CP0516657
|
US10323032, Example 36
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C18H14Cl2FN5O
|
1
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1 |
Ki = 79.4 nM
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CP0896500
|
US9096596, 64
Show/Hide
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C20H16ClF4N5O
|
1
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1 |
Ki = 79.4 nM
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CP0414028
|
US10323032, Example 2
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C20H15Cl2N3O
|
1
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1 |
Ki = 95.5 nM
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CP0413783
|
US10047092, 65
Show/Hide
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C20H16ClF3N6O
|
1
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1 |
Ki = 100 nM
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CP0407210
|
US10323032, Example 54
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C20H18ClF3N6O
|
1
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1 |
Ki = 100 nM
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CP0866306
|
US9096596, 101
Show/Hide
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C22H21ClF3N5O
|
1
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1 |
Ki = 100 nM
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CP0545289
|
US10323032, Example 73
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C21H19ClF3N5O
|
1
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1 |
Ki = 125.9 nM
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CP0420519
|
US10053462, 59
Show/Hide
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C19H15ClF3N5OS
|
1
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1 |
Ki = 125.9 nM
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CP0385627
|
US10047092, 93
Show/Hide
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C19H16ClF3N6O
|
1
|
1 |
Ki = 158.5 nM
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CP0863136
|
US9096596, 93
Show/Hide
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C19H17F2N5O
|
1
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1 |
Ki = 199.5 nM
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CP0866497
|
US9096596, 97
Show/Hide
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C19H18ClN5O
|
1
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1 |
Ki = 199.5 nM
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CP0400901
|
US10323032, Example 1
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C21H15ClF3N3O
|
1
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1 |
Ki = 223.9 nM
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CP0509255
|
US10047092, 58
Show/Hide
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C23H27ClF3N5O3
|
1
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1 |
Ki = 398.1 nM
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CP0470020
|
US10053462, 9
Show/Hide
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C19H15ClF3N5OS
|
1
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1 |
Ki = 398.1 nM
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CP0560290
|
US10323032, Example 27
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C21H17Cl2N3O
|
1
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1 |
Ki = 426.6 nM
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CP0951045
|
US9096596, 85
Show/Hide
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C19H17Cl2N5O
|
1
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1 |
Ki = 457.1 nM
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CP0375413
|
US10047092, 55
Show/Hide
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C20H14ClF6N5O
|
1
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1 |
Ki = 501.2 nM
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CP0937121
|
US9096596, 123
Show/Hide
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C18H14Cl2FN5O
|
1
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1 |
Ki = 501.2 nM
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CP0429635
|
US10047092, 60
Show/Hide
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C19H21ClF3N5O
|
1
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1 |
Ki = 631 nM
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CP0864614
|
US9096596, 114
Show/Hide
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C19H15ClF3N5O
|
1
|
1 |
Ki = 631 nM
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CP0904284
|
US9096596, 96
Show/Hide
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C19H18ClN5O
|
1
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1 |
Ki = 631 nM
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CP0408298
|
US10047092, 15
Show/Hide
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C18H14ClF3N6O
|
1
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1 |
Ki = 912 nM
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CP0384829
|
US10047092, 12
Show/Hide
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C17H14Cl2N6O
|
1
|
1 |
Ki = 1584.9 nM
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CP0384846
|
US10323032, Example 48
Show/Hide
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C18H14ClF3N6O
|
1
|
1 |
Ki = 1995.3 nM
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