General Information of the Cell Line
Cell Line ID
CL000814
Cell Line Name
Mt2-4
Category
Induced pluripotent stem cell
Organism
Homo sapiens (Human)
Tissue Information
Skin
Disease
Mitochondrial diabetes (NCIt: C131859)
Maternally-inherited diabetes and deafness (ORDO: Orphanet_225)
Map of Molecular Bioactivity Related to the Cell Line
Map of Molecular Bioactivity Related to the Cell Line

Cell Line
Protein
Compound

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Cell Line
Protein ID: PT00840, Adenosine receptor A1
Compound ID Compound Name Compound Formula
CP0536816
US9181253, 121
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C18H22ClN5O2
 1
1
Ki = 47.9 nM
   TI
   LI
   LO
   TS
CP0406830
US9181253, 109
   Show/Hide
C15H18ClN5O2
 1
1
Ki = 51.6 nM
   TI
   LI
   LO
   TS
CP0436167
US9181253, 119
   Show/Hide
C15H18ClN5O2
 1
1
Ki = 68.4 nM
   TI
   LI
   LO
   TS
CP0438910
US9181253, 117
   Show/Hide
C14H18ClN5O2
 1
1
Ki = 72.2 nM
   TI
   LI
   LO
   TS
CP0441098
US9181253, 116
   Show/Hide
C13H15ClFN5O2
 1
1
Ki = 72.7 nM
   TI
   LI
   LO
   TS
CP0479874
US9181253, 118
   Show/Hide
C16H22ClN5O2
 1
1
Ki = 78.8 nM
   TI
   LI
   LO
   TS
CP0441097
US9181253, 120c
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C16H20ClN5O2
 1
1
Ki = 86.8 nM
   TI
   LI
   LO
   TS
CP0436166
US9181253, 110
   Show/Hide
C17H22ClN5O2
 1
1
Ki = 140 nM
   TI
   LI
   LO
   TS
CP0470684
US9181253, 108
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C14H16ClN5O2
 1
1
Ki = 210 nM
   TI
   LI
   LO
   TS
CP0423749
US9181253, 111
   Show/Hide
C18H24ClN5O2
 1
1
Ki = 230 nM
   TI
   LI
   LO
   TS
CP0545707
US9181253, 107
   Show/Hide
C11H12ClN5O2
 1
1
Ki = 350 nM
   TI
   LI
   LO
   TS
CP0504111
US9181253, 112
   Show/Hide
C19H26ClN5O2
 1
1
Ki = 760 nM
   TI
   LI
   LO
   TS
CP0530381
US9181253, 115
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C13H16ClN5O2
 1
1
Ki = 930 nM
   TI
   LI
   LO
   TS
CP0479875
US9181253, 126
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C18H16ClF2N5O2
 1
1
Ki = 1260 nM
   TI
   LI
   LO
   TS
CP0529184
US9181253, 128
   Show/Hide
C19H18ClF2N5O3
 1
1
Ki = 1910 nM
   TI
   LI
   LO
   TS
CP0528985
US9181253, 125
   Show/Hide
C20H21ClFN5O3
 1
1
Ki = 3580 nM
   TI
   LI
   LO
   TS
CP0545706
US9181253, 122
   Show/Hide
C18H17ClFN5O2
 1
1
Ki = 4790 nM
   TI
   LI
   LO
   TS
Protein family and CMB statistics Related to the Cell Line
Cell Lines Derived from the same Tissue Source (Skin)
Cell Line Name Organism Disease
A-375 Homo sapiens (Human) Amelanotic melanoma
A375-P Homo sapiens (Human) Amelanotic melanoma
A375-SM Homo sapiens (Human) Amelanotic melanoma
SK-MEL-28 Homo sapiens (Human) Cutaneous melanoma
EBC-1 Homo sapiens (Human) Lung squamous cell carcinoma
WM115 Homo sapiens (Human) Melanoma
WM266-4 Homo sapiens (Human) Melanoma
G-361 Homo sapiens (Human) Melanoma
UACC-62 Homo sapiens (Human) Melanoma
SK-MEL-2 Homo sapiens (Human) Melanoma
NMIi005-A Homo sapiens (Human) Schizophrenia
A-431 Homo sapiens (Human) Skin squamous cell carcinoma
FF Mesocricetus auratus (Golden hamster) Hamster melanoma
B16-F10 Mus musculus (Mouse) Mouse melanoma
B16 Mus musculus (Mouse) Mouse melanoma
B16-BL6 Mus musculus (Mouse) Mouse melanoma
B16-F1 Mus musculus (Mouse) Mouse melanoma
B16-F0 Mus musculus (Mouse) Mouse melanoma
HaCaT Homo sapiens (Human) -
HFF Homo sapiens (Human) -
S12 [Human keratinocyte] Homo sapiens (Human) -
Malme-3 Homo sapiens (Human) -
BJ [Human fibroblast] Homo sapiens (Human) -
HMEC-1 Homo sapiens (Human) -
297L1 Homo sapiens (Human) -
HaCaT-ARE-Luc Homo sapiens (Human) -
Melan-a Mus musculus (Mouse) -
JB6 Cl 41-5a Mus musculus (Mouse) -