Brief Information of the Cell Line and Protein
Cell Line ID: CL000814 , Mt2-4
Category Induced pluripotent stem cell
Organism
Homo sapiens (Human)
Protein ID: PT00862 , Adenosine receptor A2a
Gene Name ADORA2A
Organism Homo sapiens, Human
Protein Classification Membrane receptor
Uniprot ID P29274
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000814  Protein ID: PT00862
 
Compound ID Compound Name Compound Formula
CP0436166
US9181253, 110
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C17H22ClN5O2
 1
1
Ki = 2720 nM
   TI
   LI
   LO
   TS
CP0406830
US9181253, 109
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C15H18ClN5O2
 1
1
Ki = 3020 nM
   TI
   LI
   LO
   TS
CP0545707
US9181253, 107
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C11H12ClN5O2
 1
1
Ki = 3140 nM
   TI
   LI
   LO
   TS
CP0470684
US9181253, 108
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C14H16ClN5O2
 1
1
Ki = 3700 nM
   TI
   LI
   LO
   TS
CP0479874
US9181253, 118
   Show/Hide
C16H22ClN5O2
 1
1
Ki = 3700 nM
   TI
   LI
   LO
   TS
CP0423749
US9181253, 111
   Show/Hide
C18H24ClN5O2
 1
1
Ki = 3930 nM
   TI
   LI
   LO
   TS
CP0536816
US9181253, 121
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C18H22ClN5O2
 1
1
Ki = 3950 nM
   TI
   LI
   LO
   TS
CP0436167
US9181253, 119
   Show/Hide
C15H18ClN5O2
 1
1
Ki = 4410 nM
   TI
   LI
   LO
   TS
CP0529184
US9181253, 128
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C19H18ClF2N5O3
 1
1
Ki = 7510 nM
   TI
   LI
   LO
   TS