Brief Information of the Cell Line and Protein
Cell Line ID: CL000814 , Mt2-4
Category Induced pluripotent stem cell
Organism
Homo sapiens (Human)
Protein ID: PT01279 , Adenosine receptor A3
Gene Name ADORA3
Organism Homo sapiens, Human
Protein Classification Membrane receptor
Uniprot ID P0DMS8
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000814  Protein ID: PT01279
 
Compound ID Compound Name Compound Formula
CP0406830
US9181253, 109
   Show/Hide
C15H18ClN5O2
 1
1
Ki = 5.9 nM
   TI
   LI
   LO
   TS
CP0530381
US9181253, 115
   Show/Hide
C13H16ClN5O2
 1
1
Ki = 6.6 nM
   TI
   LI
   LO
   TS
CP0436167
US9181253, 119
   Show/Hide
C15H18ClN5O2
 1
1
Ki = 8.9 nM
   TI
   LI
   LO
   TS
CP0504112
US9181253, 123
   Show/Hide
C20H21ClFN5O3
 1
1
Ki = 10.3 nM
   TI
   LI
   LO
   TS
CP0438910
US9181253, 117
   Show/Hide
C14H18ClN5O2
 1
1
Ki = 12 nM
   TI
   LI
   LO
   TS
CP0470684
US9181253, 108
   Show/Hide
C14H16ClN5O2
 1
1
Ki = 12.1 nM
   TI
   LI
   LO
   TS
CP0529185
US9181253, 124
   Show/Hide
C20H22ClN5O3
 1
1
Ki = 15.2 nM
   TI
   LI
   LO
   TS
CP0479875
US9181253, 126
   Show/Hide
C18H16ClF2N5O2
 1
1
Ki = 16.5 nM
   TI
   LI
   LO
   TS
CP0441098
US9181253, 116
   Show/Hide
C13H15ClFN5O2
 1
1
Ki = 32.4 nM
   TI
   LI
   LO
   TS
CP0529184
US9181253, 128
   Show/Hide
C19H18ClF2N5O3
 1
1
Ki = 40.4 nM
   TI
   LI
   LO
   TS
CP0545706
US9181253, 122
   Show/Hide
C18H17ClFN5O2
 1
1
Ki = 41.5 nM
   TI
   LI
   LO
   TS
CP0479874
US9181253, 118
   Show/Hide
C16H22ClN5O2
 1
1
Ki = 52 nM
   TI
   LI
   LO
   TS
CP0545708
US9181253, 127
   Show/Hide
C19H18ClF2N5O3
 1
1
Ki = 83.2 nM
   TI
   LI
   LO
   TS
CP0441097
US9181253, 120c
   Show/Hide
C16H20ClN5O2
 1
1
Ki = 110 nM
   TI
   LI
   LO
   TS
CP0528985
US9181253, 125
   Show/Hide
C20H21ClFN5O3
 1
1
Ki = 114 nM
   TI
   LI
   LO
   TS
CP0545707
US9181253, 107
   Show/Hide
C11H12ClN5O2
 1
1
Ki = 160 nM
   TI
   LI
   LO
   TS
CP0413121
US9326978, 32
   Show/Hide
C22H22N4O
 1
1
Ki = 410 nM
   TI
   LI
   LO
   TS
CP0536816
US9181253, 121
   Show/Hide
C18H22ClN5O2
 1
1
Ki = 470 nM
   TI
   LI
   LO
   TS
CP0436166
US9181253, 110
   Show/Hide
C17H22ClN5O2
 1
1
Ki = 500 nM
   TI
   LI
   LO
   TS
CP0423749
US9181253, 111
   Show/Hide
C18H24ClN5O2
 1
1
Ki = 560 nM
   TI
   LI
   LO
   TS
CP0445229
US9326978, 30
   Show/Hide
C21H20N4
 1
1
Ki = 786 nM
   TI
   LI
   LO
   TS
CP0507288
US9326978, 31
   Show/Hide
C22H22N4
 1
1
Ki = 1190 nM
   TI
   LI
   LO
   TS
CP0504111
US9181253, 112
   Show/Hide
C19H26ClN5O2
 1
1
Ki = 1530 nM
   TI
   LI
   LO
   TS
CP0414495
US9326978, 34
   Show/Hide
C21H19ClN4
 1
1
Ki = 1610 nM
   TI
   LI
   LO
   TS