| Compound ID |
Compound Name |
Compound Formula |
|
CP0264788
|
US9340555, 19
Show/Hide
|
C31H32FN5O7S
|
1
|
| 1 |
IC50 = 0.3 nM
|
|
|
|
CP0325013
|
US9340555, 18
Show/Hide
|
C28H28FN5O5S
|
1
|
| 1 |
IC50 = 0.8 nM
|
|
|
|
CP0050819
|
7-[(1E)-1-(methoxyimino)ethyl]-19-methyl-3-propyl-3,13,19,20-tetraazahexacyclo[14.7.0.0^{2,10}.0^{4,9}.0^{11,15}.0^{17,21}]tricosa-1(16),2(10),4,6,8,11(15),17,20-octaen-14-one
Show/Hide
|
C26H27N5O2
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0158668
|
US9266869, 26
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|
C29H30N4O5S
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0240888
|
US9266869, 33
Show/Hide
|
C27H28N4O6S
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0322718
|
US9266869, 39
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|
C24H23N3O5S
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0340235
|
US9266869, 32
Show/Hide
|
C27H28N4O6S
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0341149
|
US9266869, 23
Show/Hide
|
C27H28N4O6S
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0341150
|
US9266869, 30
Show/Hide
|
C29H30N4O6S
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0478030
|
US9266869, 27
Show/Hide
|
C29H26F4N4O5S
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0478031
|
US9266869, 1
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|
C22H20N4O4S
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0557212
|
US9266869, 36
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|
C29H33N5O6S
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0242334
|
US9340555, 37
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|
C30H31F2N5O5S
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0264792
|
US9340555, 57
Show/Hide
|
C28H26F2N4O5S
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0276145
|
19-methyl-7-[(1E)-1-[(2-methylpropoxy)imino]ethyl]-3-(propan-2-yl)-3,13,19,20-tetraazahexacyclo[14.7.0.0^{2,10}.0^{4,9}.0^{11,15}.0^{17,21}]tricosa-1(16),2(10),4,6,8,11(15),17,20-octaen-14-one
Show/Hide
|
C29H33N5O2
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
|
CP0240889
|
US9266869, 34
Show/Hide
|
C29H30N4O5S
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
|
CP0250176
|
US9266869, 40
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|
C24H24N4O5S
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
|
CP0526552
|
US9266869, 4
Show/Hide
|
C24H22N4O4S
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
|
CP0118063
|
US9340555, F1
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|
C23H18FN3O4S
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
|
CP0132769
|
US9340555, 65
Show/Hide
|
C26H23FN4O5S
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
|
CP0312653
|
US9340555, 39
Show/Hide
|
C31H31F2N5O6S
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
|
CP0326075
|
US9340555, 67
Show/Hide
|
C30H33FN6O3S
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
|
CP0091271
|
3-ethyl-19-methyl-7-[(1E)-1-[(2-methylpropoxy)imino]ethyl]-3,13,19,20-tetraazahexacyclo[14.7.0.0^{2,10}.0^{4,9}.0^{11,15}.0^{17,21}]tricosa-1(16),2(10),4,6,8,11(15),17,20-octaen-14-one
Show/Hide
|
C28H31N5O2
|
1
|
| 1 |
IC50 = 3 nM
|
|
|
|
CP0272815
|
US9266869, 3
Show/Hide
|
C24H21N3O4S
|
1
|
| 1 |
IC50 = 3 nM
|
|
|
|
CP0342877
|
US9266869, 12
Show/Hide
|
C27H27N5O6S
|
1
|
| 1 |
IC50 = 3 nM
|
|
|
|
CP0050822
|
7-[(1E)-1-(methoxyimino)ethyl]-19-methyl-3-(2-methylpropyl)-3,13,19,20-tetraazahexacyclo[14.7.0.0^{2,10}.0^{4,9}.0^{11,15}.0^{17,21}]tricosa-1(16),2(10),4,6,8,11(15),17,20-octaen-14-one
Show/Hide
|
C27H29N5O2
|
1
|
| 1 |
IC50 = 4 nM
|
|
|
|
CP0050825
|
7-[(1E)-1-(ethoxyimino)ethyl]-19-methyl-3-(propan-2-yl)-3,13,19,20-tetraazahexacyclo[14.7.0.0^{2,10}.0^{4,9}.0^{11,15}.0^{17,21}]tricosa-1(16),2(10),4,6,8,11(15),17,20-octaen-14-one
Show/Hide
|
C27H29N5O2
|
1
|
| 1 |
IC50 = 4 nM
|
|
|
|
CP0063471
|
19-methyl-7-[(1E)-1-[(2-methylpropoxy)imino]ethyl]-3,13,19,20-tetraazahexacyclo[14.7.0.0^{2,10}.0^{4,9}.0^{11,15}.0^{17,21}]tricosa-1(16),2(10),4,6,8,11(15),17,20-octaen-14-one
Show/Hide
|
C26H27N5O2
|
1
|
| 1 |
IC50 = 4 nM
|
|
|
|
CP0169060
|
7-[(1E)-1-(ethoxyimino)ethyl]-19-methyl-3-(2-methylpropyl)-3,13,19,20-tetraazahexacyclo[14.7.0.0^{2,10}.0^{4,9}.0^{11,15}.0^{17,21}]tricosa-1(16),2(10),4,6,8,11(15),17,20-octaen-14-one
Show/Hide
|
C28H31N5O2
|
1
|
| 1 |
IC50 = 4 nM
|
|
|
|
CP0169061
|
19-methyl-7-[(1E)-1-[(propan-2-yloxy)imino]ethyl]-3,13,19,20-tetraazahexacyclo[14.7.0.0^{2,10}.0^{4,9}.0^{11,15}.0^{17,21}]tricosa-1(16),2(10),4,6,8,11(15),17,20-octaen-14-one
Show/Hide
|
C25H25N5O2
|
1
|
| 1 |
IC50 = 4 nM
|
|
|
|
CP0202645
|
19-methyl-3-(2-methylpropyl)-7-[(1E)-1-[(propan-2-yloxy)imino]ethyl]-3,13,19,20-tetraazahexacyclo[14.7.0.0^{2,10}.0^{4,9}.0^{11,15}.0^{17,21}]tricosa-1(16),2(10),4,6,8,11(15),17,20-octaen-14-one
Show/Hide
|
C29H33N5O2
|
1
|
| 1 |
IC50 = 4 nM
|
|
|
|
CP0276304
|
7-[(1E)-1-(ethoxyimino)ethyl]-19-methyl-3,13,19,20-tetraazahexacyclo[14.7.0.0^{2,10}.0^{4,9}.0^{11,15}.0^{17,21}]tricosa-1(16),2(10),4,6,8,11(15),17,20-octaen-14-one
Show/Hide
|
C24H23N5O2
|
1
|
| 1 |
IC50 = 4 nM
|
|
|
|
CP0276305
|
19-methyl-3-(propan-2-yl)-7-[(1E)-1-[(propan-2-yloxy)imino]ethyl]-3,13,19,20-tetraazahexacyclo[14.7.0.0^{2,10}.0^{4,9}.0^{11,15}.0^{17,21}]tricosa-1(16),2(10),4,6,8,11(15),17,20-octaen-14-one
Show/Hide
|
C28H31N5O2
|
1
|
| 1 |
IC50 = 4 nM
|
|
|
|
CP0119401
|
US9266869, 31
Show/Hide
|
C30H32N4O7S
|
1
|
| 1 |
IC50 = 4 nM
|
|
|
|
CP0313959
|
US9266869, 28
Show/Hide
|
C29H27F3N4O5S
|
1
|
| 1 |
IC50 = 4 nM
|
|
|
|
CP0242327
|
US9340555, 54
Show/Hide
|
C29H26F2N4O7S
|
1
|
| 1 |
IC50 = 4 nM
|
|
|
|
CP0419919
|
US9340555, 42
Show/Hide
|
C31H31F2N5O5S
|
1
|
| 1 |
IC50 = 4 nM
|
|
|
|
CP0850397
|
N-(4-chloro-3-(((2S)-1-methyl-2-pyrrolidinyl)methoxy)phenyl)-5-(1H-pyrrolo[2,3-b]pyridin-4-yloxy)-1,3-benzoxazol-2-amine
Show/Hide
|
C26H24ClN5O3
|
1
|
| 1 |
IC50 = 5 nM
|
|
|
|
CP0219424
|
US9266869, 6
Show/Hide
|
C24H21FN4O3S
|
1
|
| 1 |
IC50 = 5 nM
|
|
|
|
CP0145220
|
5-[(1-ethylpiperidin-4-yl)amino]-3-[(3-fluorophenyl)-(5-methyl-1H-imidazol-2-yl)methylidene]-1H-indol-2-one
Show/Hide
|
C26H28FN5O
|
1
|
| 1 |
IC50 = 6 nM
|
|
|
|
CP0250177
|
US9266869, 2
Show/Hide
|
C22H19N3O4S
|
1
|
| 1 |
IC50 = 6 nM
|
|
|
|
CP0361436
|
US9266869, 29
Show/Hide
|
C29H26ClF3N4O5S
|
1
|
| 1 |
IC50 = 6 nM
|
|
|
|
CP0547700
|
US9340555, 43
Show/Hide
|
C29H29F2N5O3S
|
1
|
| 1 |
IC50 = 6 nM
|
|
|
|
CP0529723
|
2-aminobenzoxazole, 29
Show/Hide
|
C30H29ClN4O5
|
1
|
| 1 |
IC50 = 7 nM
|
|
|
|
CP0068404
|
3-[(3,5-difluorophenyl)-(5-methyl-1H-imidazol-2-yl)methylidene]-5-[(1-ethylpiperidin-4-yl)amino]-1H-indol-2-one
Show/Hide
|
C26H27F2N5O
|
1
|
| 1 |
IC50 = 7 nM
|
|
|
|
CP0118045
|
US9340555, 55
Show/Hide
|
C29H29F2N5O4S
|
1
|
| 1 |
IC50 = 7 nM
|
|
|
|
CP0164712
|
US9266869, 5
Show/Hide
|
C23H19ClN4O3S
|
1
|
| 1 |
IC50 = 9 nM
|
|
|
|
CP0274646
|
US9340555, 70
Show/Hide
|
C29H32FN5O3S
|
1
|
| 1 |
IC50 = 9 nM
|
|
|
|
CP0342770
|
US9340555, 87
Show/Hide
|
C28H27FN4O5S
|
1
|
| 1 |
IC50 = 9 nM
|
|
|
|
CP0450031
|
US9340555, 23
Show/Hide
|
C31H32F2N6O5S
|
1
|
| 1 |
IC50 = 9 nM
|
|
|
|
CP0060919
|
3-[benzimidazol-2-ylidene-(4-methylphenyl)methyl]-5-[(1-ethylpiperidin-4-yl)amino]-1H-indol-2-ol
Show/Hide
|
C30H31N5O
|
1
|
| 1 |
IC50 < 10 nM
|
|
|
|
CP0155784
|
3-[benzimidazol-2-ylidene-(3,5-difluorophenyl)methyl]-5-[(1-ethylpiperidin-4-yl)amino]-1H-indol-2-ol
Show/Hide
|
C29H27F2N5O
|
1
|
| 1 |
IC50 < 10 nM
|
|
|
|
CP0156220
|
3-[benzimidazol-2-ylidene(phenyl)methyl]-5-[(1-ethylpiperidin-4-yl)amino]-1H-indol-2-ol
Show/Hide
|
C29H29N5O
|
1
|
| 1 |
IC50 < 10 nM
|
|
|
|
CP0247375
|
3-[benzimidazol-2-ylidene-(3-fluorophenyl)methyl]-5-[(1-ethylpiperidin-4-yl)amino]-1H-indol-2-ol
Show/Hide
|
C29H28FN5O
|
1
|
| 1 |
IC50 < 10 nM
|
|
|
|
CP0240597
|
US9266869, 8
Show/Hide
|
C24H21FN4O3S
|
1
|
| 1 |
IC50 = 10 nM
|
|
|
|
CP0340226
|
US9266869, 13
Show/Hide
|
C32H39N5O6S
|
1
|
| 1 |
IC50 = 10 nM
|
|
|
|
CP0414207
|
US9340555, 45
Show/Hide
|
C25H23F2N5O3S
|
1
|
| 1 |
IC50 = 10 nM
|
|
|
|
CP0118093
|
3-[(4-chlorophenyl)-(1H-imidazol-2-yl)methylidene]-5-[(1-ethylpiperidin-4-yl)amino]-1H-indol-2-one
Show/Hide
|
C25H26ClN5O
|
1
|
| 1 |
IC50 = 11 nM
|
|
|
|
CP0158667
|
US9266869, 10
Show/Hide
|
C24H22N4O3S
|
1
|
| 1 |
IC50 = 11 nM
|
|
|
|
CP0132770
|
US9340555, 69
Show/Hide
|
C28H30FN5O3S
|
1
|
| 1 |
IC50 = 11 nM
|
|
|
|
CP0228170
|
US9353093, 2
Show/Hide
|
C25H22N4O4
|
1
|
| 1 |
IC50 = 11 nM
|
|
|
|
CP0145223
|
3-[benzimidazol-2-ylidene-(4-methoxyphenyl)methyl]-5-[(1-ethylpiperidin-4-yl)amino]-1H-indol-2-ol
Show/Hide
|
C30H31N5O2
|
1
|
| 1 |
IC50 = 13 nM
|
|
|
|
CP0132326
|
US9353093, 1
Show/Hide
|
C24H22N4O2
|
1
|
| 1 |
IC50 = 13 nM
|
|
|
|
CP0242328
|
US9340555, 38
Show/Hide
|
C30H31F2N5O4S
|
1
|
| 1 |
IC50 = 14 nM
|
|
|
|
CP0340984
|
US9340555, 24
Show/Hide
|
C32H34F2N6O5S
|
1
|
| 1 |
IC50 = 14 nM
|
|
|
|
CP0250157
|
US9266869, 11
Show/Hide
|
C24H22N4O3S
|
1
|
| 1 |
IC50 = 15 nM
|
|
|
|
CP0063611
|
US9353093, 4
Show/Hide
|
C25H24N4O2
|
1
|
| 1 |
IC50 = 15 nM
|
|
|
|
CP0160502
|
5-[(1-ethylpiperidin-4-yl)amino]-3-[(2-fluorophenyl)-(5-methyl-1H-imidazol-2-yl)methylidene]-1H-indol-2-one
Show/Hide
|
C26H28FN5O
|
1
|
| 1 |
IC50 = 16 nM
|
|
|
|
CP0563330
|
US9233968, 31
Show/Hide
|
C23H18FN5O
|
1
|
| 1 |
IC50 = 16 nM
|
|
|
|
CP0121178
|
US9340555, 85
Show/Hide
|
C24H20FN3O3S
|
1
|
| 1 |
IC50 = 16 nM
|
|
|
|
CP0243637
|
US9340555, 66
Show/Hide
|
C30H32FN5O3S
|
1
|
| 1 |
IC50 = 16 nM
|
|
|
|
CP0326076
|
US9340555, 75
Show/Hide
|
C20H15N3O5S
|
1
|
| 1 |
IC50 = 16 nM
|
|
|
|
CP0495828
|
US9340555, 44
Show/Hide
|
C30H31F2N5O5S
|
1
|
| 1 |
IC50 = 16 nM
|
|
|
|
CP0541800
|
2-aminobenzimidazole, 14
Show/Hide
|
C30H31ClN6O3
|
1
|
| 1 |
IC50 = 16.6 nM
|
|
|
|
CP0068403
|
3-[benzimidazol-2-ylidene(phenyl)methyl]-5-[[1-(2-methoxyethyl)piperidin-4-yl]amino]-1H-indol-2-ol
Show/Hide
|
C30H31N5O2
|
1
|
| 1 |
IC50 = 17 nM
|
|
|
|
CP0063609
|
US9353093, 3
Show/Hide
|
C23H20N4O2
|
1
|
| 1 |
IC50 = 17 nM
|
|
|
|
CP0384915
|
2-aminobenzoxazole, 27
Show/Hide
|
C25H24ClN5O4
|
1
|
| 1 |
IC50 = 18 nM
|
|
|
|
CP0056299
|
5-[(1-ethylpiperidin-4-yl)amino]-3-[(3-fluorophenyl)-(1H-imidazol-2-yl)methylidene]-1H-indol-2-one
Show/Hide
|
C25H26FN5O
|
1
|
| 1 |
IC50 = 20 nM
|
|
|
|
CP0361140
|
US9233968, 32
Show/Hide
|
C22H17N5O
|
1
|
| 1 |
IC50 = 20 nM
|
|
|
|
CP0331508
|
US9340555, 68
Show/Hide
|
C29H30FN5O3S
|
1
|
| 1 |
IC50 = 20 nM
|
|
|
|
CP0250342
|
US9238644, 18
Show/Hide
|
C25H30ClN7O
|
1
|
| 1 |
IC50 = 21 nM
|
|
|
|
CP0484285
|
2-aminobenzoxazole, 31
Show/Hide
|
C28H26ClN5O2
|
1
|
| 1 |
IC50 = 26 nM
|
|
|
|
CP0160496
|
5-[(1-ethylpiperidin-4-yl)amino]-3-[(5-methoxybenzimidazol-2-ylidene)-phenylmethyl]-1H-indol-2-ol
Show/Hide
|
C30H31N5O2
|
1
|
| 1 |
IC50 = 27 nM
|
|
|
|
CP0228357
|
US9340555, F2
Show/Hide
|
C22H16FN3O4S
|
1
|
| 1 |
IC50 = 29 nM
|
|
|
|
CP0002211
|
N-[2-(diethylamino)ethyl]-5-[(Z)-(5-fluoro-2-oxo-1H-indol-3-ylidene)methyl]-2,4-dimethyl-1H-pyrrole-3-carboxamide
Show/Hide
|
C22H27FN4O2
|
1
|
| 1 |
IC50 = 30 nM
|
|
|
|
CP0091889
|
3-(3-fluoro-4-{[2-(1-methyl-1H-imidazol-4-yl)thieno[3,2-b]pyridin-7-yl]oxy}phenyl)-1-(2-phenylacetyl)thiourea
Show/Hide
|
C26H20FN5O2S2
|
1
|
| 1 |
IC50 = 30 nM
|
|
|
|
CP0443151
|
2-aminobenzimidazole, 19
Show/Hide
|
C27H30ClN7O2
|
1
|
| 1 |
IC50 = 31 nM
|
|
|
|
CP0541798
|
2-aminobenzoxazole, 36
Show/Hide
|
C26H25ClFN5O4
|
1
|
| 1 |
IC50 = 31 nM
|
|
|
|
CP0500977
|
2-aminobenzimidazole, 12
Show/Hide
|
C29H26F3N5O2
|
1
|
| 1 |
IC50 = 32.4 nM
|
|
|
|
CP0529298
|
2-aminobenzoxazole, 24
Show/Hide
|
C26H28ClN5O4
|
1
|
| 1 |
IC50 = 34 nM
|
|
|
|
CP0173796
|
US9340555, 14
Show/Hide
|
C33H37FN6O5S
|
1
|
| 1 |
IC50 = 34 nM
|
|
|
|
CP0484284
|
2-aminobenzoxazole, 37
Show/Hide
|
C26H26Cl2N6O3
|
1
|
| 1 |
IC50 = 35 nM
|
|
|
|
CP0312652
|
US9340555, F3
Show/Hide
|
C23H18FN3O4S
|
1
|
| 1 |
IC50 = 35 nM
|
|
|
|
CP0384916
|
2-aminobenzoxazole, 20
Show/Hide
|
C26H27ClN6O3
|
1
|
| 1 |
IC50 = 36 nM
|
|
|
|
CP0251838
|
US9340555, 15
Show/Hide
|
C31H34FN5O4S
|
1
|
| 1 |
IC50 = 39 nM
|
|
|
|
CP0439706
|
2-aminobenzimidazole, 13
Show/Hide
|
C28H27ClN6O
|
1
|
| 1 |
IC50 = 40 nM
|
|
|
|
CP0578985
|
(3E)-6-bromo-3-(4,5,6,7-tetrahydro-1H-indol-2-ylmethylidene)-1H-indol-2-one
Show/Hide
|
C17H15BrN2O
|
1
|
| 1 |
IC50 = 40 nM
|
|
|
|
CP0419647
|
US9353093, 7
Show/Hide
|
C23H19FN4O2
|
1
|
| 1 |
IC50 = 41 nM
|
|
|
|
CP0228168
|
US9353093, 8
Show/Hide
|
C23H20N4O3
|
1
|
| 1 |
IC50 = 45 nM
|
|
|
|
CP0164714
|
US9238644, 16
Show/Hide
|
C27H31ClN6O
|
1
|
| 1 |
IC50 = 46 nM
|
|
|
|
CP0250175
|
US9266869, 24
Show/Hide
|
C26H26N4O6S
|
1
|
| 1 |
IC50 = 46 nM
|
|
|
|
CP0577856
|
US9266869, 9
Show/Hide
|
C23H19FN4O3S
|
1
|
| 1 |
IC50 = 48 nM
|
|
|
|
CP0529300
|
2-aminobenzimidazole, 5
Show/Hide
|
C23H18ClN5O3
|
1
|
| 1 |
IC50 = 49 nM
|
|
|
|
CP0243759
|
US9233968, 1
Show/Hide
|
C22H18N6O
|
1
|
| 1 |
IC50 = 51 nM
|
|
|
|
CP0518765
|
US9266869, 7
Show/Hide
|
C21H20N6O3S
|
1
|
| 1 |
IC50 = 51 nM
|
|
|
|
CP0439705
|
2-aminobenzoxazole, 35
Show/Hide
|
C26H25ClN6O2
|
1
|
| 1 |
IC50 = 52 nM
|
|
|
|
CP0510400
|
2-aminobenzoxazole, 38
Show/Hide
|
C28H25Cl2N5O2
|
1
|
| 1 |
IC50 = 52 nM
|
|
|
|
CP0125950
|
N-{3-fluoro-4-[(7-methoxyquinolin-4-yl)oxy]phenyl}-1,5-dimethyl-3-oxo-2-phenyl-2,3-dihydro-1H-pyrazole-4-carboxamide
Show/Hide
|
C28H23FN4O4
|
1
|
| 1 |
IC50 = 52 nM
|
|
|
|
CP0063319
|
US9353093, 6
Show/Hide
|
C23H17F3N4O2
|
1
|
| 1 |
IC50 = 58 nM
|
|
|
|
CP0361141
|
US9340555, 86
Show/Hide
|
C26H24FN3O3S
|
1
|
| 1 |
IC50 = 64 nM
|
|
|
|
CP0528442
|
2-aminobenzimidazole, 8
Show/Hide
|
C25H25F3N6O3
|
1
|
| 1 |
IC50 = 65 nM
|
|
|
|
CP0314616
|
US9238644, 21
Show/Hide
|
C24H28ClN7O
|
1
|
| 1 |
IC50 = 73 nM
|
|
|
|
CP0243634
|
US9340555, 50
Show/Hide
|
C30H29F2N5O5S
|
1
|
| 1 |
IC50 = 80 nM
|
|
|
|
CP0511120
|
2-aminobenzimidazole, 9
Show/Hide
|
C27H27F3N6O3
|
1
|
| 1 |
IC50 = 84 nM
|
|
|
|
CP0064500
|
N-{3-fluoro-4-[(7-methoxyquinolin-4-yl)oxy]phenyl}-5-methyl-3-oxo-1-(2-oxopropyl)-2-phenyl-2,3-dihydro-1H-pyrazole-4-carboxamide
Show/Hide
|
C30H25FN4O5
|
1
|
| 1 |
IC50 = 86 nM
|
|
|
|
CP0320907
|
US9340555, 84
Show/Hide
|
C22H15FN2O4S
|
1
|
| 1 |
IC50 = 87 nM
|
|
|
|
CP0443150
|
2-aminobenzoxazole, 23
Show/Hide
|
C24H24ClN5O4
|
1
|
| 1 |
IC50 = 88 nM
|
|
|
|
CP0529693
|
2-aminobenzimidazole, 10
Show/Hide
|
C28H27F5N6O3
|
1
|
| 1 |
IC50 = 93 nM
|
|
|
|
CP0541799
|
2-aminobenzoxazole, 26
Show/Hide
|
C26H26ClN5O4
|
1
|
| 1 |
IC50 = 94 nM
|
|
|
|
CP0098371
|
US9340555, 13
Show/Hide
|
C25H21FN8O3S
|
1
|
| 1 |
IC50 = 97 nM
|
|
|
|
CP0063615
|
US9353093, 5
Show/Hide
|
C22H16ClFN4O2
|
1
|
| 1 |
IC50 = 97 nM
|
|
|
|
CP0454226
|
2-aminobenzoxazole, 25
Show/Hide
|
C25H24ClN5O4
|
1
|
| 1 |
IC50 = 117 nM
|
|
|
|
CP0173795
|
US9340555, 12
Show/Hide
|
C26H23FN8O3S
|
1
|
| 1 |
IC50 = 126 nM
|
|
|
|
CP0160493
|
CHEMBL2086397
Show/Hide
|
C26H22N4O3
|
1
|
| 1 |
IC50 = 128 nM
|
|
|
|
CP0098354
|
US9233968, 3
Show/Hide
|
C22H17N5O
|
1
|
| 1 |
IC50 = 132 nM
|
|
|
|
CP0559808
|
US9238644, 44
Show/Hide
|
C24H30ClN7O
|
1
|
| 1 |
IC50 = 138 nM
|
|
|
|
CP0252564
|
US9353093, 9
Show/Hide
|
C23H16F4N4O2
|
1
|
| 1 |
IC50 = 139 nM
|
|
|
|
CP0443153
|
2-aminobenzimidazole, 16
Show/Hide
|
C26H26ClN7O
|
1
|
| 1 |
IC50 = 143 nM
|
|
|
|
CP0065767
|
N-{3-fluoro-4-[(7-methoxyquinolin-4-yl)oxy]phenyl}-5-methyl-3-oxo-2-phenyl-1-propyl-2,3-dihydro-1H-pyrazole-4-carboxamide
Show/Hide
|
C30H27FN4O4
|
1
|
| 1 |
IC50 = 143 nM
|
|
|
|
CP0290864
|
3-[benzimidazol-2-ylidene(phenyl)methyl]-N-butyl-2-hydroxy-1H-indole-5-carboxamide
Show/Hide
|
C27H24N4O2
|
1
|
| 1 |
IC50 = 145 nM
|
|
|
|
CP0541801
|
2-aminobenzimidazole, 7
Show/Hide
|
C26H28ClN7O2
|
1
|
| 1 |
IC50 = 146 nM
|
|
|
|
CP0070047
|
US9353093, 10
Show/Hide
|
C22H18N4O2
|
1
|
| 1 |
IC50 = 150 nM
|
|
|
|
CP0098353
|
US9233968, 33
Show/Hide
|
C23H18FN5O
|
1
|
| 1 |
IC50 = 162 nM
|
|
|
|
CP0536833
|
US9340555, 72
Show/Hide
|
C20H14N2O5S
|
1
|
| 1 |
IC50 = 162 nM
|
|
|
|
CP0150856
|
N-{3-fluoro-4-[(7-methoxyquinolin-4-yl)oxy]phenyl}-1-[(2S)-2-hydroxypropyl]-5-methyl-3-oxo-2-phenyl-2,3-dihydro-1H-pyrazole-4-carboxamide
Show/Hide
|
C30H27FN4O5
|
1
|
| 1 |
IC50 = 208 nM
|
|
|
|
CP0272871
|
US9238644, 24A
Show/Hide
|
C24H26ClN5O
|
1
|
| 1 |
IC50 = 209 nM
|
|
|
|
CP0145221
|
5-(1-ethylpiperidin-4-yl)oxy-3-[(5-methoxybenzimidazol-2-ylidene)-phenylmethyl]-1H-indol-2-ol
Show/Hide
|
C30H30N4O3
|
1
|
| 1 |
IC50 = 213 nM
|
|
|
|
CP0062594
|
5-[(1-ethylpiperidin-4-yl)amino]-3-[1H-imidazol-2-yl(phenyl)methylidene]-1H-indol-2-one
Show/Hide
|
C25H27N5O
|
1
|
| 1 |
IC50 = 235 nM
|
|
|
|
CP0155425
|
N-{3-fluoro-4-[(7-methoxyquinolin-4-yl)oxy]phenyl}-1-[(2R)-2-hydroxypropyl]-5-methyl-3-oxo-2-phenyl-2,3-dihydro-1H-pyrazole-4-carboxamide
Show/Hide
|
C30H27FN4O5
|
1
|
| 1 |
IC50 = 236 nM
|
|
|
|
CP0244017
|
US9238644, 19
Show/Hide
|
C19H19ClN6O
|
1
|
| 1 |
IC50 = 248 nM
|
|
|
|
CP0419578
|
US9238644, 13
Show/Hide
|
C20H21ClN6O
|
1
|
| 1 |
IC50 = 257 nM
|
|
|
|
CP0024012
|
4-(Benzothiazol-6-ylamino)-6-(benzyl-isopropyl-amino)-[1,3,5]triazin-2-ol
Show/Hide
|
C20H20N6OS
|
1
|
| 1 |
IC50 = 280 nM
|
|
|
|
CP0342880
|
US9238644, 2
Show/Hide
|
C28H30F3N5O
|
1
|
| 1 |
IC50 = 283 nM
|
|
|
|
CP0529722
|
2-aminobenzoxazole, 33
Show/Hide
|
C24H26ClN7O2
|
1
|
| 1 |
IC50 = 289 nM
|
|
|
|
CP0384914
|
2-aminobenzoxazole, 32
Show/Hide
|
C24H26ClN7O2
|
1
|
| 1 |
IC50 = 303 nM
|
|
|
|
CP0321881
|
US9340555, 46
Show/Hide
|
C29H27F2N5O6S
|
1
|
| 1 |
IC50 = 328 nM
|
|
|
|
CP0256097
|
N-{3-fluoro-4-[(7-methoxyquinolin-4-yl)oxy]phenyl}-5-methyl-1-(2-methylpropyl)-3-oxo-2-phenyl-2,3-dihydro-1H-pyrazole-4-carboxamide
Show/Hide
|
C31H29FN4O4
|
1
|
| 1 |
IC50 = 329 nM
|
|
|
|
CP0438249
|
US9238644, 14
Show/Hide
|
C22H24ClN7O
|
1
|
| 1 |
IC50 = 357 nM
|
|
|
|
CP0438251
|
US9238644, 45
Show/Hide
|
C20H23ClN6O
|
1
|
| 1 |
IC50 = 370 nM
|
|
|
|
CP0516732
|
US9238644, 57-2A
Show/Hide
|
C25H30F3N7O
|
1
|
| 1 |
IC50 = 382 nM
|
|
|
|
CP0314615
|
US9238644, 17
Show/Hide
|
C24H28ClN7O
|
1
|
| 1 |
IC50 = 393 nM
|
|
|
|
CP0483298
|
US9238644, 57
Show/Hide
|
C25H30F3N7O
|
1
|
| 1 |
IC50 = 394 nM
|
|
|
|
CP0024603
|
4-(Benzothiazol-6-ylamino)-6-(1-methyl-1-phenyl-ethylamino)-[1,3,5]triazin-2-ol
Show/Hide
|
C19H18N6OS
|
1
|
| 1 |
IC50 = 400 nM
|
|
|
|
CP0243760
|
US9233968, 4
Show/Hide
|
C22H14F4N6O
|
1
|
| 1 |
IC50 = 423 nM
|
|
|
|
CP0160501
|
5-[(1-ethylpiperidin-3-yl)amino]-3-[(5-methoxybenzimidazol-2-ylidene)-phenylmethyl]-1H-indol-2-ol
Show/Hide
|
C30H31N5O2
|
1
|
| 1 |
IC50 = 496 nM
|
|
|
|
CP0384091
|
US9353093, 26
Show/Hide
|
C21H18N4O2S
|
1
|
| 1 |
IC50 = 508 nM
|
|
|
|
CP0438250
|
US9238644, 57-1A
Show/Hide
|
C25H30F3N7O
|
1
|
| 1 |
IC50 = 518 nM
|
|
|
|
CP0028661
|
4-(Benzothiazol-6-ylamino)-6-(benzyl-ethyl-amino)-[1,3,5]triazin-2-ol
Show/Hide
|
C19H18N6OS
|
1
|
| 1 |
IC50 = 600 nM
|
|
|
|
CP0515208
|
US9238644, 7
Show/Hide
|
C27H30ClN5O
|
1
|
| 1 |
IC50 = 629 nM
|
|
|
|
CP0484287
|
2-aminobenzimidazole, 15
Show/Hide
|
C25H25ClN8O
|
1
|
| 1 |
IC50 = 645 nM
|
|
|
|
CP0026720
|
1-(2-hydroxy-2-methylpropyl)-N-{5-[(7-methoxyquinolin-4-yl)oxy]pyridin-2-yl}-5-methyl-3-oxo-2-phenyl-2,3-dihydro-1H-pyrazole-4-carboxamide
Show/Hide
|
C30H29N5O5
|
1
|
| 1 |
IC50 = 690 nM
|
|
|
|
CP0559491
|
1-(9-methoxy-3,4,5,6-tetrahydro-1H-azepino[4,3-b]indol-2-yl)-2-pyridin-2-ylethanone
Show/Hide
|
C20H21N3O2
|
1
|
| 1 |
IC50 = 700 nM
|
|
|
|
CP0290605
|
2-aminobenzoxazole, 21
Show/Hide
|
C20H15ClN4O3
|
1
|
| 1 |
IC50 = 766 nM
|
|
|
|
CP0423869
|
5-bromo-4-N-(5-methyl-1H-pyrazol-3-yl)-2-N-prop-2-enylpyrimidine-2,4-diamine
Show/Hide
|
C11H13BrN6
|
1
|
| 1 |
IC50 = 794.33 nM
|
|
|
|
CP0015779
|
N-[4-(1,3-benzothiazol-6-ylamino)-6-(2-phenylpropan-2-ylamino)-1,3,5-triazin-2-yl]hydroxylamine
Show/Hide
|
C19H19N7OS
|
1
|
| 1 |
IC50 = 840 nM
|
|
|
|
CP0331514
|
US9233968, 23
Show/Hide
|
C22H16N4O
|
1
|
| 1 |
IC50 = 862 nM
|
|
|
|
CP0266397
|
US9238644, 8
Show/Hide
|
C28H32ClN5O
|
1
|
| 1 |
IC50 = 897 nM
|
|
|
|
CP0040687
|
N-{3-fluoro-4-[(7-methoxyquinolin-4-yl)oxy]phenyl}-1-(2-hydroxy-2-methylpropyl)-5-methyl-3-oxo-2-phenyl-2,3-dihydro-1H-pyrazole-4-carboxamide
Show/Hide
|
C31H29FN4O5
|
1
|
| 1 |
IC50 = 921 nM
|
|
|
|
CP0263705
|
US9233968, 2
Show/Hide
|
C22H14F3N5O
|
1
|
| 1 |
IC50 = 962 nM
|
|
|
|
CP0454227
|
2-aminobenzimidazole, 17
Show/Hide
|
C24H27ClN8O
|
1
|
| 1 |
IC50 = 1028 nM
|
|
|
|
CP0113134
|
4-N-(1,3-benzothiazol-6-yl)-6-chloro-2-N-(2-phenylpropan-2-yl)-1,3,5-triazine-2,4-diamine
Show/Hide
|
C19H17ClN6S
|
1
|
| 1 |
IC50 = 1080 nM
|
|
|
|
CP0132656
|
US9233968, 21
Show/Hide
|
C22H16FN5O
|
1
|
| 1 |
IC50 = 1121 nM
|
|
|
|
CP0092384
|
US9353093, 27
Show/Hide
|
C21H15F3N4O2S
|
1
|
| 1 |
IC50 = 1209 nM
|
|
|
|
CP0241515
|
US9233968, 22
Show/Hide
|
C22H13F3N4O
|
1
|
| 1 |
IC50 = 1280 nM
|
|
|
|
CP0187571
|
US9233968, 24
Show/Hide
|
C21H12ClFN4O
|
1
|
| 1 |
IC50 = 1459 nM
|
|
|
|
CP0153243
|
4-N-[5-[2-(3,5-dimethoxyphenyl)ethyl]-1H-pyrazol-3-yl]-2-N-[(3-methyl-1,2-oxazol-5-yl)methyl]pyrimidine-2,4-diamine
Show/Hide
|
C22H25N7O3
|
1
|
| 1 |
IC50 = 1584.89 nM
|
|
|
|
CP0383439
|
5-bromo-2-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-4-N-[5-(2-phenylethyl)-1H-pyrazol-3-yl]pyrimidine-2,4-diamine
Show/Hide
|
C20H20BrN7O
|
1
|
| 1 |
IC50 = 1584.89 nM
|
|
|
|
CP0272870
|
US9238644, 20
Show/Hide
|
C23H26ClN7O
|
1
|
| 1 |
IC50 = 1755 nM
|
|
|
|
CP0559883
|
US9238644, 3
Show/Hide
|
C29H32F3N5O
|
1
|
| 1 |
IC50 = 1789 nM
|
|
|
|
CP0068405
|
[3-[benzimidazol-2-ylidene(phenyl)methyl]-2-hydroxy-1H-indol-5-yl]-(4-methylpiperazin-1-yl)methanone
Show/Hide
|
C28H25N5O2
|
1
|
| 1 |
IC50 = 1804 nM
|
|
|
|
CP0318933
|
US9238644, 15
Show/Hide
|
C26H29ClN6O
|
1
|
| 1 |
IC50 = 1996 nM
|
|
|
|
CP0490075
|
US9238644, 4
Show/Hide
|
C26H26F3N5O
|
1
|
| 1 |
IC50 = 2036 nM
|
|
|
|
CP0132716
|
US9233968, 7
Show/Hide
|
C22H13ClF3N5O
|
1
|
| 1 |
IC50 = 2046 nM
|
|
|
|
CP0158674
|
US9238644, 56
Show/Hide
|
C24H28F3N7O
|
1
|
| 1 |
IC50 = 2224 nM
|
|
|
|
CP0454228
|
2-aminobenzimidazole, 6
Show/Hide
|
C21H13ClF3N5O
|
1
|
| 1 |
IC50 = 2270 nM
|
|
|
|
CP0291719
|
4-(Benzothiazol-5-ylamino)-6-(benzyl-methyl-amino)-[1,3,5]triazin-2-ol
Show/Hide
|
C18H16N6OS
|
1
|
| 1 |
IC50 = 2400 nM
|
|
|
|
CP0313513
|
US9233968, 26
Show/Hide
|
C22H15FN4O
|
1
|
| 1 |
IC50 = 3038 nM
|
|
|
|
CP0807372
|
US9238644, 35
Show/Hide
|
C18H19ClN6O
|
1
|
| 1 |
IC50 = 3786 nM
|
|
|
|
CP0529725
|
2-aminobenzimidazole, 4
Show/Hide
|
C19H12ClF3N4O
|
1
|
| 1 |
IC50 = 3896 nM
|
|
|
|
CP0000999
|
(Z)-3-[2,4-dimethyl-5-(2-oxo-1,2-dihydro-indol-3-ylidenemethyl)-1H-pyrrol-3-yl]-propionic acid
Show/Hide
|
C18H18N2O3
|
1
|
| 1 |
IC50 = 3900 nM
|
|
|
|
CP0331532
|
US9233968, 20
Show/Hide
|
C22H16FN5O
|
1
|
| 1 |
IC50 = 4404 nM
|
|
|
|
CP0129192
|
US9233968, 8
Show/Hide
|
C21H15N5O
|
1
|
| 1 |
IC50 = 5428 nM
|
|
|
|
CP0578024
|
1-(9-methoxy-3,4,5,6-tetrahydro-1H-azepino[4,3-b]indol-2-yl)ethanone
Show/Hide
|
C15H18N2O2
|
1
|
| 1 |
IC50 = 6000 nM
|
|
|
|
CP0383438
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5-bromo-2-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-4-N-(5-propyl-1H-pyrazol-3-yl)pyrimidine-2,4-diamine
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C15H18BrN7O
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1
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| 1 |
IC50 = 6309.57 nM
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CP0423870
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5-bromo-2-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-4-N-(5-methyl-1H-pyrazol-3-yl)pyrimidine-2,4-diamine
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C13H14BrN7O
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1
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| 1 |
IC50 = 6309.57 nM
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CP0313365
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US9238644, 6
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C21H20ClN5O
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1
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| 1 |
IC50 = 6608 nM
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CP0063603
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US9353093, 31
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C21H14ClF3N4O2S
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1
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| 1 |
IC50 = 7350 nM
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CP0543458
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1-(9-methoxy-3,4,5,6-tetrahydro-1H-azepino[4,3-b]indol-2-yl)-3-morpholin-4-ylpropan-1-one
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C20H27N3O3
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1
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| 1 |
IC50 = 8000 nM
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CP0576747
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9-methoxy-3,4,5,6-tetrahydro-2H-azepino[4,3-b]indol-1-one
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C13H14N2O2
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1
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| 1 |
IC50 = 8000 nM
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CP0559807
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US9238644, 36
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C19H21ClN6O
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1
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| 1 |
IC50 = 8171 nM
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CP0361138
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US9233968, 9
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C22H13F4N5O
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1
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| 1 |
IC50 = 8416 nM
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CP0113141
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4-(Benzothiazol-6-yl-methyl-amino)-6-(1-methyl-1-phenyl-ethylamino)-[1,3,5]triazin-2-ol
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C20H20N6OS
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1
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| 1 |
IC50 = 9900 nM
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CP0383497
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5-bromo-4-N-(5-methyl-1H-pyrazol-3-yl)-2-N-(2-pyridin-3-ylethyl)pyrimidine-2,4-diamine
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C15H16BrN7
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1
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| 1 |
IC50 > 10000 nM
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CP0383498
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5-bromo-2-N-[(3-tert-butyl-1,2-oxazol-5-yl)methyl]-4-N-(5-methyl-1H-pyrazol-3-yl)pyrimidine-2,4-diamine
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C16H20BrN7O
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1
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| 1 |
IC50 > 10000 nM
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CP0383500
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5-bromo-4-N-[5-(3-methoxypropyl)-1H-pyrazol-3-yl]-2-N-[(3-methyl-1,2-oxazol-5-yl)methyl]pyrimidine-2,4-diamine
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C16H20BrN7O2
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1
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| 1 |
IC50 > 10000 nM
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CP0129193
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US9233968, 14
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C21H14ClFN6O
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1
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| 1 |
IC50 > 10000 nM
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CP0132657
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US9233968, 28
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C22H16N4O
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1
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| 1 |
IC50 > 10000 nM
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CP0132717
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US9233968, 25
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C23H14N4O2
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1
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| 1 |
IC50 > 10000 nM
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CP0173674
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US9233968, 12
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C26H22N6O2
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1
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| 1 |
IC50 > 10000 nM
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CP0227554
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US9233968, 13
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C22H17N5O
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1
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| 1 |
IC50 > 10000 nM
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CP0274117
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US9233968, 10
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C30H17F8N7O2
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1
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| 1 |
IC50 > 10000 nM
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CP0313546
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US9233968, 27
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C21H14N4O
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1
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| 1 |
IC50 > 10000 nM
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CP0323840
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US9233968, 19
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C21H15N5O
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1
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| 1 |
IC50 > 10000 nM
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CP0419890
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US9233968, 11
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C24H20N6O2
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1
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| 1 |
IC50 > 10000 nM
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CP0419891
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US9233968, 15
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C28H17Cl2F2N7O2
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1
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| 1 |
IC50 > 10000 nM
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CP0132099
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US9238644, 12
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C20H19ClN6O
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1
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| 1 |
IC50 > 10000 nM
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CP0314614
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BDBM202403
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C22H19ClF3N5O
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1
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| 1 |
IC50 > 10000 nM
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CP0435116
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US9238644, 1
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C28H32F3N5O
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1
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| 1 |
IC50 > 10000 nM
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CP0083279
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US9353093, 11
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C23H20N4O2
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1
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| 1 |
IC50 > 10000 nM
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CP0950856
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methyl (1S,15R,17S,18S)-17-ethyl-7-methoxy-3,13-diazapentacyclo[13.3.1.02,10.04,9.013,18]nonadeca-2(10),4(9),5,7-tetraene-1-carboxylate
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C22H28N2O3
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1
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| 1 |
IC50 = 10000 nM
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CP0282955
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4-(3H-Benzoimidazol-5-ylamino)-6-(1-methyl-1-phenyl-ethylamino)-[1,3,5]triazin-2-ol
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C19H19N7O
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1
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| 1 |
IC50 > 20000 nM
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CP0494935
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1-(9-methoxy-3,4,5,6-tetrahydro-1H-azepino[4,3-b]indol-2-yl)-3-methylbutan-1-one
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C18H24N2O2
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1
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| 1 |
IC50 > 20000 nM
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CP0562036
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1-(9-methoxy-3,4,5,6-tetrahydro-1H-azepino[4,3-b]indol-2-yl)-2-phenylethanone
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C21H22N2O2
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1
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| 1 |
IC50 > 20000 nM
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CP0575299
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9-methoxy-1,2,3,4,5,6-hexahydroazepino[4,3-b]indole
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C13H16N2O
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1
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| 1 |
IC50 > 20000 nM
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CP0575350
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1-(9-methoxy-3,4,5,6-tetrahydro-1H-azepino[4,3-b]indol-2-yl)-2-morpholin-4-ylethanone
Show/Hide
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C19H25N3O3
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1
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| 1 |
IC50 > 20000 nM
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CP0577950
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1-(9-methoxy-3,4,5,6-tetrahydro-1H-azepino[4,3-b]indol-2-yl)-2-pyridin-4-ylethanone
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C20H21N3O2
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1
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| 1 |
IC50 > 20000 nM
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CP0250770
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4-(Benzothiazol-6-ylamino)-6-benzylamino-[1,3,5]triazin-2-ol
Show/Hide
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C17H14N6OS
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1
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| 1 |
IC50 > 30000 nM
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CP0282954
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4-N-(1,3-benzothiazol-6-yl)-6-methoxy-2-N-(2-phenylpropan-2-yl)-1,3,5-triazine-2,4-diamine
Show/Hide
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C20H20N6OS
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1
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| 1 |
IC50 > 30000 nM
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CP0060918
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3-[benzimidazol-2-ylidene(phenyl)methyl]-2-hydroxy-N-(2-methoxyethyl)-1H-indole-5-sulfonamide
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C25H22N4O4S
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1
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| 1 |
IC50 = 30000 nM
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CP0145219
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3-[benzimidazol-2-ylidene(phenyl)methyl]-5-(4-methylpiperazin-1-yl)sulfonyl-1H-indol-2-ol
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C27H25N5O3S
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1
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| 1 |
IC50 = 30000 nM
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CP0098367
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US9340555, F5
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C22H16FN3O3S
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1
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| 1 |
IC50 = 100000 nM
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CP0121175
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US9340555, F4
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C23H18FN3O3S
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1
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| 1 |
IC50 = 100000 nM
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CP0310229
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2-aminobenzimidazole, 3
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C21H15ClF3N5O2
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1
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| 1 |
IC50 >= 1140 nM
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